| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.902 | 0.005 | 0.904 | Antiinflammatory | 0.7 0.031 CHEMBL3544786 0.868 0.008 CHEMBL1228 0.881 0.006 CHEMBL3544829 0.857 0.009 CHEMBL3544828 0.904 0.005 CHEMBL3544827 0.475 0.098 CHEMBL3544842 | CHEMBL3544827 | |
| 0.779 | 0.007 | 0.779 | Analgesic | 0.702 0.013 CHEMBL1228 0.584 0.03 CHEMBL3544829 0.541 0.039 CHEMBL3544828 0.361 0.103 CHEMBL3544827 | ||
| 0.576 | 0.014 | 0.661 | 5 Hydroxytryptamine release inhibitor | 0.582 0.013 CHEMBL3544786 0.6 0.011 CHEMBL1228 0.524 0.025 CHEMBL3544829 0.533 0.023 CHEMBL3544828 0.661 0.005 CHEMBL3544827 0.356 0.11 CHEMBL3544842 | CHEMBL3544827 | |
| 0.546 | 0.021 | 0.745 | 5 Hydroxytryptamine release stimulant | 0.262 0.083 CHEMBL3544786 0.559 0.019 CHEMBL1228 0.735 0.005 CHEMBL3544829 0.745 0.005 CHEMBL3544828 0.396 0.047 CHEMBL3544827 0.522 0.024 CHEMBL3544842 | CHEMBL3544828 | |
| 0.546 | 0.023 | 0.882 | Antithrombotic | 0.732 0.006 CHEMBL3544786 0.563 0.02 CHEMBL1228 0.568 0.02 CHEMBL3544829 0.562 0.02 CHEMBL3544828 0.882 0.003 CHEMBL3544827 0.44 0.04 CHEMBL3544842 | CHEMBL3544827 | |
| 0.514 | 0.022 | 0.543 | GABA C receptor rho-3 antagonist | 0.543 0.016 CHEMBL1228 0.263 0.143 CHEMBL3544829 0.312 0.108 CHEMBL3544828 | CHEMBL1228 | |
| 0.479 | 0.004 | 0.479 | Uric acid excretion stimulant | 0.14 0.027 CHEMBL3544786 0.434 0.004 CHEMBL1228 0.381 0.004 CHEMBL3544829 0.363 0.004 CHEMBL3544828 0.366 0.004 CHEMBL3544827 | ||
| 0.447 | 0.014 | 0.447 | Platelet aggregation inhibitor | 0.313 0.033 CHEMBL1228 0.314 0.033 CHEMBL3544829 0.238 0.057 CHEMBL3544828 0.235 0.059 CHEMBL3544827 | ||
| 0.44 | 0.01 | 0.744 | Non-steroidal antiinflammatory agent | 0.336 0.022 CHEMBL3544786 0.461 0.009 CHEMBL1228 0.494 0.007 CHEMBL3544829 0.498 0.007 CHEMBL3544828 0.744 0.003 CHEMBL3544827 | CHEMBL3544827 | |
| 0.429 | 0.003 | 0.509 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.333 0.005 CHEMBL3544786 0.382 0.004 CHEMBL1228 0.509 0.002 CHEMBL3544829 0.445 0.003 CHEMBL3544828 0.467 0.003 CHEMBL3544827 0.235 0.011 CHEMBL3544842 | CHEMBL3544829 | |
| 0.461 | 0.045 | 0.614 | Histamine release inhibitor | 0.583 0.012 CHEMBL3544786 0.508 0.026 CHEMBL1228 0.508 0.026 CHEMBL3544829 0.535 0.019 CHEMBL3544828 0.614 0.009 CHEMBL3544827 0.29 0.129 CHEMBL3544842 | CHEMBL3544827 | |
| 0.457 | 0.045 | 0.553 | Immunosuppressant | 0.493 0.035 CHEMBL3544786 0.439 0.05 CHEMBL1228 0.462 0.043 CHEMBL3544829 0.439 0.05 CHEMBL3544828 0.553 0.02 CHEMBL3544827 0.384 0.07 CHEMBL3544842 | CHEMBL3544827 | |
| 0.391 | 0.003 | 0.391 | Electrolyte absorption antagonist | 0.303 0.004 CHEMBL1228 0.29 0.004 CHEMBL3544829 0.208 0.007 CHEMBL3544828 0.103 0.054 CHEMBL3544827 | ||
| 0.43 | 0.064 | 0.716 | Antibacterial | 0.668 0.011 CHEMBL3544786 0.478 0.047 CHEMBL1228 0.451 0.056 CHEMBL3544829 0.475 0.048 CHEMBL3544828 0.716 0.008 CHEMBL3544827 0.552 0.028 CHEMBL3544842 | CHEMBL3544827 | |
| 0.388 | 0.042 | 0.562 | Spasmolytic | 0.316 0.064 CHEMBL3544786 0.437 0.033 CHEMBL1228 0.463 0.029 CHEMBL3544829 0.489 0.024 CHEMBL3544828 0.562 0.017 CHEMBL3544827 | CHEMBL3544827 | |
| 0.366 | 0.034 | 0.44 | Platelet antagonist | 0.362 0.035 CHEMBL3544786 0.316 0.048 CHEMBL1228 0.316 0.048 CHEMBL3544829 0.268 0.065 CHEMBL3544828 0.44 0.02 CHEMBL3544827 | CHEMBL3544827 | |
| 0.349 | 0.026 | 0.349 | 5 Hydroxytryptamine uptake stimulant | 0.342 0.028 CHEMBL1228 0.228 0.107 CHEMBL3544829 0.226 0.109 CHEMBL3544828 | ||
| 0.315 | 0.012 | 0.315 | Cyclooxygenase 1 inhibitor | 0.31 0.013 CHEMBL1228 0.209 0.031 CHEMBL3544829 0.222 0.027 CHEMBL3544828 0.202 0.033 CHEMBL3544827 0.101 0.099 CHEMBL3544842 | ||
| 0.399 | 0.102 | 0.399 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.277 0.246 CHEMBL1228 0.309 0.2 CHEMBL3544829 | ||
| 0.357 | 0.061 | 0.68 | Cholesterol antagonist | 0.632 0.015 CHEMBL3544786 0.448 0.041 CHEMBL1228 0.34 0.068 CHEMBL3544829 0.37 0.057 CHEMBL3544828 0.68 0.009 CHEMBL3544827 0.345 0.066 CHEMBL3544842 | CHEMBL3544827 | |
| 0.295 | 0.008 | 0.295 | Ferrochelatase inhibitor | 0.17 0.03 CHEMBL1228 0.233 0.016 CHEMBL3544829 0.104 0.066 CHEMBL3544828 | ||
| 0.312 | 0.027 | 0.42 | P-glycoprotein inhibitor | 0.282 0.033 CHEMBL1228 0.42 0.014 CHEMBL3544829 0.388 0.018 CHEMBL3544828 0.249 0.042 CHEMBL3544827 | CHEMBL3544829 | |
| 0.305 | 0.03 | 0.305 | Gastrin inhibitor | 0.194 0.157 CHEMBL3544786 0.261 0.067 CHEMBL1228 0.247 0.083 CHEMBL3544829 0.189 0.166 CHEMBL3544828 0.222 0.116 CHEMBL3544827 | ||
| 0.29 | 0.019 | 0.29 | Cyclooxygenase inhibitor | 0.27 0.022 CHEMBL1228 0.213 0.037 CHEMBL3544829 0.212 0.037 CHEMBL3544828 0.188 0.047 CHEMBL3544827 | ||
| 0.278 | 0.017 | 0.321 | Phospholipase A2 inhibitor | 0.18 0.054 CHEMBL3544786 0.321 0.011 CHEMBL1228 0.211 0.037 CHEMBL3544829 0.226 0.031 CHEMBL3544828 0.281 0.017 CHEMBL3544827 | CHEMBL1228 | |
| 0.294 | 0.036 | 0.364 | Tyrosine 3 hydroxylase inhibitor | 0.364 0.013 CHEMBL1228 0.237 0.081 CHEMBL3544829 0.283 0.043 CHEMBL3544828 | CHEMBL1228 | |
| 0.38 | 0.123 | 0.47 | Caspase 9 stimulant | 0.47 0.073 CHEMBL3544786 0.449 0.083 CHEMBL1228 0.289 0.207 CHEMBL3544829 0.338 0.156 CHEMBL3544828 0.424 0.097 CHEMBL3544827 0.324 0.169 CHEMBL3544842 | CHEMBL3544786 | |
| 0.273 | 0.041 | 0.308 | Anesthetic general | 0.308 0.031 CHEMBL3544786 0.299 0.033 CHEMBL1228 0.253 0.049 CHEMBL3544829 0.256 0.048 CHEMBL3544828 0.277 0.039 CHEMBL3544827 0.175 0.09 CHEMBL3544842 | CHEMBL3544786 | |
| 0.302 | 0.077 | 0.356 | Sodium/bile acid cotransporter inhibitor | 0.248 0.13 CHEMBL3544786 0.356 0.036 CHEMBL1228 0.274 0.103 CHEMBL3544829 0.322 0.06 CHEMBL3544828 0.296 0.083 CHEMBL3544827 | CHEMBL1228 | |
| 0.271 | 0.053 | 0.271 | 5 Hydroxytryptamine 1E antagonist | 0.263 0.061 CHEMBL1228 | ||
| 0.292 | 0.079 | 0.45 | Interleukin 2 agonist | 0.45 0.015 CHEMBL3544786 0.318 0.062 CHEMBL1228 0.261 0.107 CHEMBL3544829 0.273 0.095 CHEMBL3544828 0.444 0.017 CHEMBL3544827 0.395 0.029 CHEMBL3544842 | CHEMBL3544786 | |
| 0.309 | 0.097 | 0.309 | Thioredoxin glutathione reductase inhibitor | 0.288 0.11 CHEMBL1228 | ||
| 0.242 | 0.032 | 0.437 | Diuretic | 0.216 0.039 CHEMBL3544786 0.207 0.041 CHEMBL1228 0.186 0.05 CHEMBL3544829 0.157 0.071 CHEMBL3544828 0.437 0.011 CHEMBL3544827 | CHEMBL3544827 | |
| 0.302 | 0.096 | 0.38 | Vasodilator, peripheral | 0.223 0.151 CHEMBL3544786 0.308 0.093 CHEMBL1228 0.38 0.062 CHEMBL3544829 0.367 0.067 CHEMBL3544828 0.287 0.104 CHEMBL3544827 | CHEMBL3544829 | |
| 0.278 | 0.073 | 0.296 | Insulysin inhibitor | 0.296 0.061 CHEMBL1228 0.223 0.125 CHEMBL3544829 0.233 0.113 CHEMBL3544828 | CHEMBL1228 | |
| 0.206 | 0.012 | 0.206 | GABA C receptor antagonist | 0.196 0.014 CHEMBL1228 0.158 0.026 CHEMBL3544829 0.139 0.037 CHEMBL3544828 | ||
| 0.234 | 0.042 | 0.322 | Anticoagulant | 0.193 0.056 CHEMBL3544786 0.174 0.064 CHEMBL1228 0.156 0.075 CHEMBL3544829 0.127 0.103 CHEMBL3544828 0.322 0.025 CHEMBL3544827 | CHEMBL3544827 | |
| 0.293 | 0.105 | 0.335 | Prostaglandin dehydrogenase inhibitor | 0.335 0.088 CHEMBL1228 | CHEMBL1228 | |
| 0.222 | 0.034 | 0.454 | Protein kinase stimulant | 0.315 0.015 CHEMBL3544786 0.274 0.021 CHEMBL1228 0.146 0.071 CHEMBL3544829 0.171 0.055 CHEMBL3544828 0.454 0.005 CHEMBL3544827 0.171 0.055 CHEMBL3544842 | CHEMBL3544827 | |
| 0.199 | 0.012 | 0.199 | Sphingosine 1-phosphate receptor 5 antagonist | 0.194 0.014 CHEMBL1228 0.134 0.091 CHEMBL3544829 | ||
| 0.216 | 0.037 | 0.228 | Succinate dehydrogenase inhibitor | 0.228 0.031 CHEMBL1228 0.201 0.048 CHEMBL3544829 0.192 0.055 CHEMBL3544828 | CHEMBL1228 | |
| 0.204 | 0.027 | 0.204 | GABA C receptor rho-2 antagonist | 0.2 0.029 CHEMBL1228 0.124 0.117 CHEMBL3544829 0.123 0.118 CHEMBL3544828 | ||
| 0.253 | 0.076 | 0.418 | Interleukin agonist | 0.418 0.016 CHEMBL3544786 0.242 0.085 CHEMBL1228 0.231 0.093 CHEMBL3544829 0.209 0.113 CHEMBL3544828 0.374 0.023 CHEMBL3544827 0.288 0.054 CHEMBL3544842 | CHEMBL3544786 | |
| 0.188 | 0.012 | 0.188 | Sphingosine 1-phosphate receptor 4 antagonist | 0.172 0.018 CHEMBL1228 0.124 0.065 CHEMBL3544829 0.107 0.1 CHEMBL3544828 | ||
| 0.181 | 0.006 | 0.181 | Acetylcholine release stimulant | 0.155 0.014 CHEMBL3544786 0.145 0.02 CHEMBL1228 0.109 0.068 CHEMBL3544829 0.153 0.015 CHEMBL3544827 | ||
| 0.203 | 0.03 | 0.21 | Arachidonic acid antagonist | 0.175 0.059 CHEMBL3544786 0.21 0.024 CHEMBL1228 0.186 0.048 CHEMBL3544829 0.186 0.047 CHEMBL3544828 0.147 0.092 CHEMBL3544827 | CHEMBL1228 | |
| 0.234 | 0.065 | 0.234 | Psychostimulant | 0.166 0.103 CHEMBL3544786 0.219 0.07 CHEMBL1228 0.227 0.067 CHEMBL3544827 | ||
| 0.18 | 0.018 | 0.267 | Photosensitizer | 0.174 0.02 CHEMBL3544786 0.182 0.017 CHEMBL1228 0.099 0.09 CHEMBL3544829 0.097 0.095 CHEMBL3544828 0.267 0.005 CHEMBL3544827 | CHEMBL3544827 | |
| 0.188 | 0.026 | 0.188 | Cathepsin H inhibitor | 0.158 0.041 CHEMBL1228 0.174 0.032 CHEMBL3544829 0.15 0.046 CHEMBL3544828 | ||
| 0.169 | 0.016 | 0.206 | Prolactin inhibitor | 0.206 0.008 CHEMBL1228 0.089 0.068 CHEMBL3544829 0.112 0.044 CHEMBL3544828 | CHEMBL1228 | |
| 0.205 | 0.053 | 0.205 | Lipocortins synthesis antagonist | 0.201 0.055 CHEMBL3544786 0.192 0.061 CHEMBL1228 0.17 0.08 CHEMBL3544829 0.153 0.1 CHEMBL3544828 0.173 0.078 CHEMBL3544827 | ||
| 0.215 | 0.063 | 0.273 | Neurotrophic factor enhancer | 0.234 0.048 CHEMBL3544786 0.268 0.029 CHEMBL1228 0.165 0.117 CHEMBL3544829 0.206 0.07 CHEMBL3544828 0.273 0.027 CHEMBL3544827 0.151 0.137 CHEMBL3544842 | CHEMBL3544827 | |
| 0.169 | 0.02 | 0.189 | TRPA1 agonist | 0.189 0.013 CHEMBL1228 0.101 0.085 CHEMBL3544829 0.119 0.06 CHEMBL3544828 0.119 0.059 CHEMBL3544827 | CHEMBL1228 | |
| 0.17 | 0.021 | 0.17 | Sphingosine 1-phosphate receptor 2 antagonist | 0.166 0.024 CHEMBL1228 | ||
| 0.183 | 0.036 | 0.183 | Cyclooxygenase 2 inhibitor | 0.167 0.043 CHEMBL1228 0.122 0.077 CHEMBL3544829 0.123 0.076 CHEMBL3544828 0.126 0.074 CHEMBL3544827 | ||
| 0.162 | 0.021 | 0.172 | Ca2+-transporting ATPase inhibitor | 0.172 0.012 CHEMBL3544786 0.159 0.024 CHEMBL1228 0.145 0.057 CHEMBL3544829 0.138 0.079 CHEMBL3544828 0.155 0.033 CHEMBL3544827 0.132 0.111 CHEMBL3544842 | CHEMBL3544786 | |
| 0.18 | 0.04 | 0.379 | Cell wall synthesis inhibitor | 0.262 0.014 CHEMBL3544786 0.187 0.036 CHEMBL1228 0.172 0.045 CHEMBL3544829 0.167 0.05 CHEMBL3544828 0.379 0.007 CHEMBL3544827 0.146 0.069 CHEMBL3544842 | CHEMBL3544827 | |
| 0.157 | 0.021 | 0.253 | Creatine kinase inhibitor | 0.253 0.005 CHEMBL1228 0.107 0.052 CHEMBL3544829 0.157 0.021 CHEMBL3544828 | CHEMBL1228 | |
| 0.144 | 0.008 | 0.166 | Androgen agonist | 0.166 0.006 CHEMBL1228 0.107 0.013 CHEMBL3544829 0.114 0.011 CHEMBL3544828 0.054 0.05 CHEMBL3544827 | CHEMBL1228 | |
| 0.183 | 0.047 | 0.212 | Neurotensin receptor agonist | 0.212 0.03 CHEMBL1228 0.151 0.099 CHEMBL3544828 | CHEMBL1228 | |
| 0.16 | 0.03 | 0.16 | GABA C receptor agonist | 0.134 0.041 CHEMBL1228 0.145 0.036 CHEMBL3544829 0.101 0.066 CHEMBL3544828 | ||
| 0.221 | 0.094 | 0.221 | Calpain inhibitor | 0.19 0.124 CHEMBL1228 | ||
| 0.176 | 0.053 | 0.383 | Interferon gamma antagonist | 0.304 0.019 CHEMBL3544786 0.218 0.035 CHEMBL1228 0.196 0.042 CHEMBL3544829 0.228 0.033 CHEMBL3544828 0.383 0.012 CHEMBL3544827 0.2 0.041 CHEMBL3544842 | CHEMBL3544827 | |
| 0.132 | 0.013 | 0.161 | Glycine receptor antagonist | 0.161 0.005 CHEMBL3544786 0.111 0.024 CHEMBL1228 0.078 0.06 CHEMBL3544829 0.16 0.005 CHEMBL3544827 0.074 0.067 CHEMBL3544842 | CHEMBL3544786 | |
| 0.162 | 0.043 | 0.271 | DNA polymerase I inhibitor | 0.271 0.014 CHEMBL3544786 0.188 0.032 CHEMBL1228 0.102 0.084 CHEMBL3544828 0.193 0.03 CHEMBL3544827 0.173 0.038 CHEMBL3544842 | CHEMBL3544786 | |
| 0.207 | 0.089 | 0.215 | RNA-directed DNA polymerase inhibitor | 0.189 0.117 CHEMBL3544786 0.215 0.08 CHEMBL1228 0.205 0.092 CHEMBL3544829 0.202 0.097 CHEMBL3544828 0.179 0.134 CHEMBL3544827 | CHEMBL1228 | |
| 0.26 | 0.143 | 0.26 | Calpain 2 inhibitor | 0.203 0.185 CHEMBL1228 | ||
| 0.122 | 0.004 | 0.122 | Glutamate (mGluR7) antagonist | 0.117 0.005 CHEMBL1228 0.079 0.028 CHEMBL3544829 0.075 0.034 CHEMBL3544828 | ||
| 0.25 | 0.135 | 0.427 | Vasodilator, coronary | 0.374 0.045 CHEMBL3544786 0.257 0.128 CHEMBL1228 0.242 0.142 CHEMBL3544829 0.244 0.141 CHEMBL3544828 0.427 0.028 CHEMBL3544827 0.192 0.19 CHEMBL3544842 | CHEMBL3544827 | |
| 0.178 | 0.063 | 0.214 | Phospholipase C inhibitor | 0.173 0.069 CHEMBL3544786 0.214 0.036 CHEMBL1228 0.144 0.119 CHEMBL3544829 0.158 0.091 CHEMBL3544828 0.18 0.061 CHEMBL3544827 | CHEMBL1228 | |
| 0.178 | 0.066 | 0.391 | Peroxidase inhibitor | 0.391 0.022 CHEMBL1228 0.203 0.058 CHEMBL3544829 0.36 0.027 CHEMBL3544828 | CHEMBL1228 | |
| 0.139 | 0.027 | 0.139 | GABA C receptor rho-1 antagonist | 0.125 0.036 CHEMBL1228 0.113 0.046 CHEMBL3544829 0.096 0.068 CHEMBL3544828 | ||
| 0.153 | 0.043 | 0.223 | Cholesterol synthesis inhibitor | 0.112 0.073 CHEMBL3544786 0.192 0.029 CHEMBL1228 0.195 0.028 CHEMBL3544829 0.223 0.022 CHEMBL3544828 0.14 0.05 CHEMBL3544827 | CHEMBL3544828 | |
| 0.145 | 0.037 | 0.329 | Xanthine oxidase inhibitor | 0.14 0.038 CHEMBL3544786 0.227 0.015 CHEMBL1228 0.167 0.028 CHEMBL3544829 0.227 0.015 CHEMBL3544828 0.329 0.006 CHEMBL3544827 | CHEMBL3544827 | |
| 0.137 | 0.029 | 0.137 | Electron transport complex I inhibitor | 0.129 0.036 CHEMBL1228 | ||
| 0.224 | 0.119 | 0.346 | Lipoxygenase inhibitor | 0.346 0.052 CHEMBL1228 | CHEMBL1228 | |
| 0.16 | 0.059 | 0.188 | CF transmembrane conductance regulator agonist | 0.188 0.03 CHEMBL1228 0.142 0.091 CHEMBL3544828 0.136 0.104 CHEMBL3544827 | CHEMBL1228 | |
| 0.116 | 0.018 | 0.116 | Sphingosine 1-phosphate receptor 4 agonist | 0.106 0.022 CHEMBL1228 0.06 0.054 CHEMBL3544829 | ||
| 0.187 | 0.089 | 0.187 | Histone acetyltransferase inhibitor | 0.181 0.098 CHEMBL1228 | ||
| 0.121 | 0.023 | 0.126 | Interleukin 5 antagonist | 0.09 0.054 CHEMBL3544786 0.126 0.02 CHEMBL1228 0.082 0.069 CHEMBL3544829 0.091 0.054 CHEMBL3544828 0.114 0.028 CHEMBL3544827 | CHEMBL1228 | |
| 0.128 | 0.032 | 0.142 | Anabolic | 0.142 0.022 CHEMBL1228 0.105 0.056 CHEMBL3544829 0.114 0.046 CHEMBL3544828 | CHEMBL1228 | |
| 0.13 | 0.034 | 0.13 | Sphingomyelinase inhibitor | 0.084 0.081 CHEMBL3544786 0.112 0.047 CHEMBL1228 0.096 0.064 CHEMBL3544829 0.102 0.057 CHEMBL3544827 | ||
| 0.246 | 0.152 | 0.246 | Calcium channel activator | 0.231 0.17 CHEMBL1228 0.222 0.183 CHEMBL3544829 0.213 0.194 CHEMBL3544828 | ||
| 0.105 | 0.014 | 0.105 | Vanilloid 4 agonist | 0.082 0.036 CHEMBL1228 0.082 0.037 CHEMBL3544829 | ||
| 0.191 | 0.1 | 0.336 | Cyclic AMP phosphodiesterase inhibitor | 0.302 0.041 CHEMBL3544786 0.194 0.098 CHEMBL1228 0.282 0.049 CHEMBL3544829 0.282 0.049 CHEMBL3544828 0.336 0.029 CHEMBL3544827 0.156 0.142 CHEMBL3544842 | CHEMBL3544827 | |
| 0.134 | 0.045 | 0.134 | Falcipain 3 inhibitor | 0.117 0.056 CHEMBL1228 | ||
| 0.195 | 0.107 | 0.55 | Aldehyde oxidase inhibitor | 0.411 0.045 CHEMBL1228 0.381 0.05 CHEMBL3544829 0.55 0.026 CHEMBL3544828 | CHEMBL3544828 | |
| 0.104 | 0.018 | 0.115 | CC chemokine 5 receptor agonist | 0.115 0.01 CHEMBL1228 0.077 0.076 CHEMBL3544829 0.085 0.048 CHEMBL3544828 | CHEMBL1228 | |
| 0.149 | 0.064 | 0.166 | Adenylate cyclase stimulant | 0.129 0.103 CHEMBL3544786 0.166 0.04 CHEMBL1228 0.138 0.084 CHEMBL3544829 0.148 0.066 CHEMBL3544828 | CHEMBL1228 | |
| 0.111 | 0.03 | 0.124 | Bile acid receptor antagonist | 0.124 0.016 CHEMBL1228 0.095 0.06 CHEMBL3544829 0.104 0.042 CHEMBL3544828 0.089 0.075 CHEMBL3544827 | CHEMBL1228 | |
| 0.101 | 0.02 | 0.103 | Glycine receptor agonist | 0.103 0.019 CHEMBL3544786 0.098 0.022 CHEMBL1228 0.067 0.06 CHEMBL3544829 0.086 0.032 CHEMBL3544827 | CHEMBL3544786 | |
| 0.138 | 0.059 | 0.403 | Cyclooxygenase 3 inhibitor | 0.256 0.008 CHEMBL3544786 0.158 0.042 CHEMBL1228 0.127 0.07 CHEMBL3544829 0.145 0.053 CHEMBL3544828 0.403 0.004 CHEMBL3544827 0.127 0.07 CHEMBL3544842 | CHEMBL3544827 | |
| 0.162 | 0.083 | 0.291 | ATPase inhibitor | 0.228 0.02 CHEMBL3544786 0.167 0.074 CHEMBL1228 0.164 0.079 CHEMBL3544829 0.166 0.076 CHEMBL3544828 0.291 0.007 CHEMBL3544827 0.151 0.1 CHEMBL3544842 | CHEMBL3544827 | |
| 0.084 | 0.006 | 0.084 | Cholesterol esterase inhibitor | 0.072 0.009 CHEMBL1228 0.053 0.025 CHEMBL3544829 0.048 0.033 CHEMBL3544828 | ||
| 0.199 | 0.121 | 0.199 | Neuropeptide Y2 antagonist | 0.198 0.122 CHEMBL1228 0.185 0.149 CHEMBL3544829 0.188 0.143 CHEMBL3544828 | ||
| 0.097 | 0.022 | 0.097 | Acetylcholine M5 receptor agonist | |||
| 0.137 | 0.062 | 0.19 | Toll-Like receptor 2 antagonist | 0.19 0.028 CHEMBL1228 0.133 0.065 CHEMBL3544829 0.173 0.038 CHEMBL3544828 | CHEMBL1228 | |
| 0.09 | 0.016 | 0.194 | Prostaglandin F2 alpha antagonist | 0.086 0.018 CHEMBL1228 0.194 0.004 CHEMBL3544829 0.16 0.004 CHEMBL3544828 0.066 0.037 CHEMBL3544827 0.073 0.029 CHEMBL3544842 | CHEMBL3544829 | |
| 0.133 | 0.06 | 0.149 | Vanilloid 1 agonist | 0.123 0.081 CHEMBL3544786 0.149 0.039 CHEMBL1228 0.136 0.056 CHEMBL3544827 | CHEMBL1228 | |
| 0.136 | 0.064 | 0.307 | Alpha-N-acetylglucosaminidase inhibitor | 0.307 0.015 CHEMBL3544786 0.105 0.094 CHEMBL1228 0.246 0.024 CHEMBL3544829 0.158 0.05 CHEMBL3544828 0.187 0.038 CHEMBL3544827 0.225 0.028 CHEMBL3544842 | CHEMBL3544786 | |
| 0.139 | 0.068 | 0.139 | Nav1.6 sodium channel blocker | |||
| 0.153 | 0.085 | 0.185 | Growth hormone agonist | 0.185 0.065 CHEMBL1228 0.129 0.109 CHEMBL3544829 0.149 0.088 CHEMBL3544828 | CHEMBL1228 | |
| 0.098 | 0.03 | 0.115 | Interferon agonist | 0.106 0.024 CHEMBL3544786 0.085 0.044 CHEMBL1228 0.076 0.058 CHEMBL3544829 0.115 0.019 CHEMBL3544827 | CHEMBL3544827 | |
| 0.151 | 0.084 | 0.168 | Sigma receptor agonist | 0.168 0.074 CHEMBL1228 | CHEMBL1228 | |
| 0.191 | 0.126 | 0.519 | Immunostimulant | 0.479 0.032 CHEMBL3544786 0.23 0.105 CHEMBL1228 0.266 0.09 CHEMBL3544829 0.283 0.084 CHEMBL3544828 0.519 0.027 CHEMBL3544827 0.354 0.063 CHEMBL3544842 | CHEMBL3544827 | |
| 0.114 | 0.049 | 0.125 | Adenylate kinase inhibitor | 0.103 0.063 CHEMBL3544786 0.099 0.069 CHEMBL1228 0.125 0.039 CHEMBL3544829 0.098 0.071 CHEMBL3544828 | CHEMBL3544829 | |
| 0.078 | 0.013 | 0.078 | Oleamide hydrolase inhibitor | 0.059 0.021 CHEMBL1228 | ||
| 0.073 | 0.008 | 0.094 | Nicotinic acid receptor agonist | 0.094 0.005 CHEMBL1228 | CHEMBL1228 | |
| 0.078 | 0.018 | 0.078 | Corticotropin releasing factor 2 receptor antagonist | |||
| 0.081 | 0.023 | 0.093 | Interferon inducer | 0.088 0.018 CHEMBL3544786 0.07 0.035 CHEMBL1228 0.063 0.047 CHEMBL3544829 0.093 0.015 CHEMBL3544827 | CHEMBL3544827 | |
| 0.186 | 0.128 | 0.219 | DNA damaging | 0.178 0.136 CHEMBL3544786 0.194 0.121 CHEMBL1228 0.219 0.101 CHEMBL3544827 | CHEMBL3544827 | |
| 0.085 | 0.028 | 0.085 | Phospholipase D inhibitor | 0.066 0.063 CHEMBL1228 | ||
| 0.133 | 0.077 | 0.133 | Neurotrophic factor | 0.129 0.082 CHEMBL1228 0.121 0.093 CHEMBL3544827 | ||
| 0.181 | 0.126 | 0.233 | Nitric-oxide synthase stimulant | 0.185 0.118 CHEMBL3544786 0.193 0.101 CHEMBL1228 0.223 0.057 CHEMBL3544829 0.233 0.045 CHEMBL3544828 0.189 0.109 CHEMBL3544827 0.223 0.056 CHEMBL3544842 | CHEMBL3544828 | |
| 0.175 | 0.121 | 0.175 | 5 Hydroxytryptamine 3E antagonist | |||
| 0.101 | 0.047 | 0.259 | Triose-phosphate isomerase inhibitor | 0.259 0.006 CHEMBL3544786 0.092 0.057 CHEMBL1228 0.134 0.025 CHEMBL3544829 0.106 0.042 CHEMBL3544828 0.172 0.015 CHEMBL3544827 0.162 0.017 CHEMBL3544842 | CHEMBL3544786 | |
| 0.103 | 0.051 | 0.103 | Lanosterol 14 alpha demethylase inhibitor | 0.096 0.061 CHEMBL1228 | ||
| 0.072 | 0.022 | 0.079 | Sphingosine kinase inhibitor | 0.079 0.017 CHEMBL1228 0.062 0.036 CHEMBL3544829 0.062 0.036 CHEMBL3544828 | CHEMBL1228 | |
| 0.077 | 0.028 | 0.077 | Glutamate (mGluR6) antagonist | 0.067 0.047 CHEMBL1228 0.062 0.061 CHEMBL3544829 | ||
| 0.102 | 0.053 | 0.102 | Antihistaminic | |||
| 0.075 | 0.027 | 0.075 | Cathepsin L inhibitor | 0.06 0.039 CHEMBL1228 | ||
| 0.108 | 0.06 | 0.129 | Aminopeptidase B inhibitor | 0.106 0.061 CHEMBL1228 0.129 0.048 CHEMBL3544829 0.11 0.058 CHEMBL3544828 | CHEMBL3544829 | |
| 0.072 | 0.026 | 0.075 | Acyl-CoA dehydrogenase inhibitor | 0.048 0.045 CHEMBL1228 0.075 0.024 CHEMBL3544829 | CHEMBL3544829 | |
| 0.061 | 0.014 | 0.061 | Histamine H2 receptor agonist | |||
| 0.071 | 0.025 | 0.086 | Fatty acid synthase inhibitor | 0.086 0.016 CHEMBL1228 | CHEMBL1228 | |
| 0.059 | 0.014 | 0.079 | Cytokine production stimulant | 0.079 0.005 CHEMBL3544786 0.047 0.037 CHEMBL1228 0.045 0.043 CHEMBL3544829 0.062 0.011 CHEMBL3544827 | CHEMBL3544786 | |
| 0.052 | 0.007 | 0.067 | Prostaglandin D2 agonist | 0.047 0.009 CHEMBL1228 0.067 0.004 CHEMBL3544829 0.059 0.005 CHEMBL3544828 0.036 0.016 CHEMBL3544827 | CHEMBL3544829 | |
| 0.162 | 0.117 | 0.215 | Insulin sensitizer | 0.184 0.091 CHEMBL1228 0.209 0.065 CHEMBL3544829 0.215 0.059 CHEMBL3544828 0.177 0.098 CHEMBL3544827 | CHEMBL3544828 | |
| 0.11 | 0.066 | 0.2 | Cystathionine beta-synthase inhibitor | 0.097 0.08 CHEMBL3544786 0.2 0.024 CHEMBL1228 0.128 0.052 CHEMBL3544828 0.154 0.039 CHEMBL3544827 | CHEMBL1228 | |
| 0.054 | 0.01 | 0.054 | Glutamate (mGluR3) antagonist | 0.05 0.013 CHEMBL1228 0.039 0.022 CHEMBL3544829 | ||
| 0.063 | 0.019 | 0.064 | Immunoglobulin Fc receptor antagonist | 0.058 0.03 CHEMBL1228 0.064 0.017 CHEMBL3544829 0.059 0.027 CHEMBL3544828 | CHEMBL3544829 | |
| 0.052 | 0.01 | 0.052 | Delayed rectifier potassium channel blocker | 0.044 0.017 CHEMBL1228 | ||
| 0.046 | 0.004 | 0.046 | Nicotinic acid receptor 2 antagonist | 0.04 0.005 CHEMBL1228 | ||
| 0.112 | 0.073 | 0.112 | Anesthetic local | 0.095 0.088 CHEMBL1228 0.103 0.08 CHEMBL3544829 | ||
| 0.053 | 0.014 | 0.053 | Angiotensin AT1 receptor antagonist | 0.039 0.035 CHEMBL1228 | ||
| 0.043 | 0.004 | 0.043 | Acid ceramidase inhibitor | 0.029 0.011 CHEMBL1228 | ||
| 0.069 | 0.031 | 0.069 | Argininosuccinate synthase inhibitor | 0.057 0.039 CHEMBL3544786 0.056 0.04 CHEMBL1228 | ||
| 0.092 | 0.053 | 0.092 | Histamine antagonist | |||
| 0.179 | 0.142 | 0.22 | Superoxide dismutase inhibitor | 0.22 0.098 CHEMBL1228 0.172 0.152 CHEMBL3544828 | CHEMBL1228 | |
| 0.11 | 0.074 | 0.117 | Sphingosine 1-phosphate receptor 2 agonist | 0.107 0.082 CHEMBL1228 0.117 0.06 CHEMBL3544829 0.113 0.067 CHEMBL3544828 | CHEMBL3544829 | |
| 0.051 | 0.015 | 0.051 | Membrane dipeptidase inhibitor | 0.038 0.03 CHEMBL1228 0.045 0.02 CHEMBL3544829 | ||
| 0.079 | 0.044 | 0.089 | Lipase inhibitor | 0.089 0.034 CHEMBL1228 0.067 0.058 CHEMBL3544827 | CHEMBL1228 | |
| 0.071 | 0.036 | 0.086 | MDM2 inhibitor | 0.086 0.014 CHEMBL3544829 0.071 0.037 CHEMBL3544828 | CHEMBL3544829 | |
| 0.079 | 0.044 | 0.079 | Adenosine A3 receptor antagonist | 0.07 0.058 CHEMBL1228 | ||
| 0.193 | 0.159 | 0.306 | 12-Lipoxygenase inhibitor | 0.306 0.076 CHEMBL1228 | CHEMBL1228 | |
| 0.058 | 0.024 | 0.058 | Lysophosphatidic acid 3 receptor antagonist | 0.049 0.038 CHEMBL1228 0.053 0.031 CHEMBL3544829 | ||
| 0.064 | 0.032 | 0.064 | Sphingosine 1-phosphate receptor 3 antagonist | 0.064 0.033 CHEMBL1228 | ||
| 0.06 | 0.029 | 0.064 | Leukotriene C antagonist | 0.064 0.022 CHEMBL1228 | CHEMBL1228 | |
| 0.06 | 0.03 | 0.06 | Pregnane X receptor antagonist | 0.057 0.037 CHEMBL1228 | ||
| 0.221 | 0.19 | 0.346 | 15-Lipoxygenase inhibitor | 0.346 0.102 CHEMBL1228 | CHEMBL1228 | |
| 0.048 | 0.018 | 0.048 | Sphingosine kinase 1 inhibitor | 0.048 0.018 CHEMBL1228 0.042 0.028 CHEMBL3544829 0.038 0.037 CHEMBL3544828 | ||
| 0.065 | 0.036 | 0.065 | Histone deacetylase SIRT3 inhibitor | 0.059 0.054 CHEMBL1228 | ||
| 0.047 | 0.018 | 0.047 | Kainate receptor agonist | 0.043 0.024 CHEMBL1228 0.04 0.032 CHEMBL3544829 | ||
| 0.063 | 0.034 | 0.063 | Phosphodiesterase 1A inhibitor | |||
| 0.246 | 0.217 | 0.754 | Cyclophilin D inhibitor | 0.634 0.022 CHEMBL3544786 0.291 0.17 CHEMBL1228 0.482 0.056 CHEMBL3544829 0.455 0.065 CHEMBL3544828 0.754 0.009 CHEMBL3544827 0.41 0.085 CHEMBL3544842 | CHEMBL3544827 | |
| 0.107 | 0.078 | 0.107 | Proteasome inhibitor | 0.103 0.084 CHEMBL1228 | ||
| 0.033 | 0.007 | 0.053 | Vanilloid 2 agonist | 0.043 0.004 CHEMBL3544786 0.032 0.008 CHEMBL1228 0.053 0.003 CHEMBL3544827 | CHEMBL3544827 | |
| 0.076 | 0.05 | 0.092 | GABA B receptor agonist | 0.092 0.024 CHEMBL1228 0.075 0.054 CHEMBL3544829 0.083 0.036 CHEMBL3544828 | CHEMBL1228 | |
| 0.04 | 0.014 | 0.04 | Angiotensin II receptor antagonist | |||
| 0.052 | 0.026 | 0.057 | Aldosterone antagonist | 0.057 0.022 CHEMBL3544829 | CHEMBL3544829 | |
| 0.03 | 0.004 | 0.045 | Nicotinic acid receptor 1 antagonist | 0.045 0.003 CHEMBL1228 0.021 0.008 CHEMBL3544828 | CHEMBL1228 | |
| 0.038 | 0.013 | 0.038 | Calcium-independent phospholipase A2 inhibitor | 0.036 0.019 CHEMBL1228 | ||
| 0.059 | 0.033 | 0.065 | Sphingosine kinase 2 inhibitor | 0.065 0.026 CHEMBL1228 | CHEMBL1228 | |
| 0.039 | 0.013 | 0.039 | Adenosine uptake inhibitor | |||
| 0.072 | 0.046 | 0.072 | Amidase inhibitor | 0.069 0.05 CHEMBL1228 | ||
| 0.093 | 0.068 | 0.141 | Phosphodiesterase 6D inhibitor | 0.119 0.026 CHEMBL3544786 0.098 0.057 CHEMBL1228 0.12 0.025 CHEMBL3544829 0.125 0.021 CHEMBL3544828 0.141 0.013 CHEMBL3544827 0.133 0.016 CHEMBL3544842 | CHEMBL3544827 | |
| 0.083 | 0.058 | 0.108 | Estrogen-related receptor beta agonist | 0.108 0.017 CHEMBL1228 0.09 0.041 CHEMBL3544828 | CHEMBL1228 | |
| 0.133 | 0.109 | 0.317 | Melanin inhibitor | 0.23 0.032 CHEMBL3544786 0.179 0.052 CHEMBL1228 0.14 0.097 CHEMBL3544829 0.175 0.055 CHEMBL3544828 0.317 0.02 CHEMBL3544827 0.181 0.051 CHEMBL3544842 | CHEMBL3544827 | |
| 0.069 | 0.045 | 0.071 | Exportin-1 inhibitor | 0.071 0.041 CHEMBL3544829 | CHEMBL3544829 | |
| 0.055 | 0.033 | 0.055 | Nicotinic alpha3beta2 receptor antagonist | |||
| 0.032 | 0.01 | 0.032 | Hedgehog signaling activator | 0.03 0.013 CHEMBL1228 | ||
| 0.054 | 0.032 | 0.086 | Aconitate hydratase inhibitor | 0.086 0.012 CHEMBL3544829 0.056 0.03 CHEMBL3544828 | CHEMBL3544829 | |
| 0.075 | 0.055 | 0.112 | Na+ K+ transporting ATPase inhibitor | 0.112 0.021 CHEMBL3544786 0.081 0.05 CHEMBL1228 0.112 0.022 CHEMBL3544827 0.096 0.035 CHEMBL3544842 | CHEMBL3544827 | |
| 0.029 | 0.009 | 0.044 | Prostaglandin F2 alpha agonist | 0.034 0.007 CHEMBL1228 0.043 0.005 CHEMBL3544829 0.044 0.005 CHEMBL3544828 | CHEMBL3544828 | |
| 0.037 | 0.017 | 0.037 | Melatonin receptor 1A agonist | |||
| 0.084 | 0.065 | 0.084 | Granulocyte macrophage colony stimulating factor agonist | 0.082 0.069 CHEMBL1228 | ||
| 0.064 | 0.045 | 0.064 | Protease 3C (Human rhinovirus) inhibitor | |||
| 0.03 | 0.011 | 0.03 | Lysophosphatidic acid receptor 1 agonist | 0.028 0.013 CHEMBL3544829 | ||
| 0.098 | 0.079 | 0.098 | 5 Hydroxytryptamine 3A agonist | |||
| 0.127 | 0.109 | 0.127 | Pregnane X receptor agonist | |||
| 0.035 | 0.017 | 0.035 | Peptide deformylase inhibitor | |||
| 0.052 | 0.035 | 0.052 | 5 Hydroxytryptamine 4 antagonist | |||
| 0.037 | 0.021 | 0.037 | Glutamate (mGluR8) antagonist | 0.036 0.024 CHEMBL1228 0.034 0.03 CHEMBL3544827 | ||
| 0.034 | 0.018 | 0.094 | Prostaglandin agonist | 0.035 0.017 CHEMBL1228 0.094 0.005 CHEMBL3544829 0.082 0.006 CHEMBL3544828 | CHEMBL3544829 | |
| 0.027 | 0.013 | 0.053 | Prostaglandin EP2 agonist | 0.027 0.014 CHEMBL1228 0.053 0.005 CHEMBL3544829 0.046 0.007 CHEMBL3544828 | CHEMBL3544829 | |
| 0.079 | 0.065 | 0.079 | Ca(v)3.1 blocker | 0.076 0.073 CHEMBL1228 | ||
| 0.104 | 0.091 | 0.149 | Aldehyde dehydrogenase inhibitor | 0.149 0.048 CHEMBL1228 0.104 0.09 CHEMBL3544829 0.135 0.057 CHEMBL3544828 0.12 0.071 CHEMBL3544827 | CHEMBL1228 | |
| 0.047 | 0.034 | 0.084 | Glucose-6-phosphate isomerase inhibitor | 0.084 0.008 CHEMBL3544786 0.044 0.042 CHEMBL1228 0.057 0.021 CHEMBL3544829 0.047 0.034 CHEMBL3544828 0.064 0.016 CHEMBL3544827 0.077 0.009 CHEMBL3544842 | CHEMBL3544786 | |
| 0.088 | 0.076 | 0.269 | UDP-glucose 4-epimerase inhibitor | 0.269 0.012 CHEMBL3544786 0.091 0.072 CHEMBL1228 0.124 0.041 CHEMBL3544829 0.115 0.047 CHEMBL3544828 0.196 0.019 CHEMBL3544827 0.199 0.018 CHEMBL3544842 | CHEMBL3544786 | |
| 0.092 | 0.079 | 0.092 | Glutamate (mGluR7) agonist | |||
| 0.07 | 0.058 | 0.07 | Acetylcholine M4 receptor antagonist | |||
| 0.043 | 0.032 | 0.043 | Histamine H1 receptor agonist | |||
| 0.039 | 0.027 | 0.041 | Leukotriene C4 antagonist | 0.041 0.022 CHEMBL1228 | CHEMBL1228 | |
| 0.034 | 0.023 | 0.034 | Free fatty acid receptor 1 antagonist | |||
| 0.068 | 0.056 | 0.068 | Cathepsin G inhibitor | 0.068 0.057 CHEMBL1228 | ||
| 0.029 | 0.018 | 0.029 | Purinergic P2Y15 antagonist | |||
| 0.028 | 0.017 | 0.028 | Glucosylceramidase stimulant | |||
| 0.068 | 0.057 | 0.088 | Porphobilinogen synthase inhibitor | 0.088 0.042 CHEMBL1228 | CHEMBL1228 | |
| 0.043 | 0.032 | 0.043 | Glutamate (mGluR group III) antagonist | |||
| 0.058 | 0.048 | 0.075 | Enoyl-[acyl-carrier-protein] reductase inhibitor | 0.075 0.023 CHEMBL1228 | CHEMBL1228 | |
| 0.048 | 0.038 | 0.048 | Cannabinoid CB2 receptor antagonist | |||
| 0.08 | 0.07 | 0.086 | 3C-Like protease (SARS coronavirus) inhibitor | 0.086 0.054 CHEMBL3544829 0.082 0.062 CHEMBL3544828 | CHEMBL3544829 | |
| 0.067 | 0.058 | 0.099 | Aminopeptidase I inhibitor | 0.099 0.028 CHEMBL3544829 0.083 0.039 CHEMBL3544828 | CHEMBL3544829 | |
| 0.017 | 0.008 | 0.017 | Thromboxane A2 agonist | 0.015 0.011 CHEMBL3544829 | ||
| 0.031 | 0.023 | 0.044 | ATP citrate lysase inhibitor | 0.044 0.01 CHEMBL1228 0.029 0.028 CHEMBL3544829 0.034 0.018 CHEMBL3544828 | CHEMBL1228 | |
| 0.067 | 0.058 | 0.102 | Catalase inhibitor | 0.102 0.038 CHEMBL3544829 0.07 0.054 CHEMBL3544828 | CHEMBL3544829 | |
| 0.022 | 0.014 | 0.022 | Angiotensin AT1A receptor antagonist | |||
| 0.189 | 0.181 | 0.606 | Transcription factor NF kappa B inhibitor | 0.482 0.047 CHEMBL3544786 0.281 0.106 CHEMBL1228 0.242 0.133 CHEMBL3544828 0.606 0.03 CHEMBL3544827 | CHEMBL3544827 | |
| 0.021 | 0.014 | 0.029 | Neuraminidase (Influenza B) inhibitor | 0.02 0.016 CHEMBL1228 0.029 0.005 CHEMBL3544829 0.025 0.008 CHEMBL3544828 | CHEMBL3544829 | |
| 0.039 | 0.032 | 0.053 | Oxytocin agonist | 0.053 0.022 CHEMBL1228 | CHEMBL1228 | |
| 0.123 | 0.116 | 0.127 | Neuropeptide Y1 antagonist | 0.127 0.106 CHEMBL1228 | CHEMBL1228 | |
| 0.035 | 0.029 | 0.035 | Melanocortin 1 antagonist | |||
| 0.061 | 0.055 | 0.202 | Phosphofructokinase-1 inhibitor | 0.202 0.011 CHEMBL3544786 0.06 0.056 CHEMBL1228 0.09 0.036 CHEMBL3544829 0.073 0.046 CHEMBL3544828 0.138 0.02 CHEMBL3544827 0.142 0.02 CHEMBL3544842 | CHEMBL3544786 | |
| 0.033 | 0.027 | 0.033 | Kainate receptor 2 antagonist | |||
| 0.05 | 0.044 | 0.085 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.085 0.014 CHEMBL1228 0.056 0.034 CHEMBL3544829 0.083 0.015 CHEMBL3544828 | CHEMBL1228 | |
| 0.029 | 0.023 | 0.029 | Acetylcholine M4 receptor agonist | |||
| 0.047 | 0.042 | 0.047 | Prolyl endopeptidase inhibitor | |||
| 0.117 | 0.112 | 0.117 | Acetylcholine M1 receptor antagonist | 0.116 0.115 CHEMBL1228 | ||
| 0.061 | 0.056 | 0.068 | Calcium channel P-type blocker | 0.068 0.032 CHEMBL3544829 | CHEMBL3544829 | |
| 0.051 | 0.047 | 0.051 | Glucosylceramidase inhibitor | |||
| 0.057 | 0.054 | 0.087 | Dopamine D1 antagonist | 0.087 0.03 CHEMBL1228 | CHEMBL1228 | |
| 0.011 | 0.007 | 0.013 | Thromboxane agonist | 0.013 0.006 CHEMBL3544829 | CHEMBL3544829 | |
| 0.033 | 0.029 | 0.039 | Nicotinic acid receptor 2 agonist | 0.039 0.021 CHEMBL1228 | CHEMBL1228 | |
| 0.053 | 0.05 | 0.053 | Cannabinoid CB1 receptor agonist | |||
| 0.037 | 0.033 | 0.037 | AMPA 4 receptor antagonist | |||
| 0.106 | 0.103 | 0.142 | NADPH oxidase inhibitor | 0.142 0.06 CHEMBL1228 | CHEMBL1228 | |
| 0.081 | 0.078 | 0.133 | Alcohol dehydrogenase inhibitor | 0.112 0.041 CHEMBL1228 0.11 0.042 CHEMBL3544829 0.133 0.027 CHEMBL3544828 0.086 0.07 CHEMBL3544827 | CHEMBL3544828 | |
| 0.021 | 0.019 | 0.057 | Prostaglandin E2 agonist | 0.022 0.017 CHEMBL1228 0.057 0.005 CHEMBL3544829 0.047 0.006 CHEMBL3544828 | CHEMBL3544829 | |
| 0.012 | 0.011 | 0.012 | Lysophosphatidic acid receptor 3 agonist | |||
| 0.069 | 0.067 | 0.069 | Potassium channel (Tandem pore domain) blocker | |||
| 0.052 | 0.051 | 0.052 | Carbonic anhydrase stimulant | |||
| 0.025 | 0.023 | 0.037 | Toll-Like receptor 4 agonist | 0.037 0.006 CHEMBL3544786 0.036 0.006 CHEMBL3544827 0.028 0.015 CHEMBL3544842 | CHEMBL3544786 | |
| 0.116 | 0.114 | 0.158 | Farnesoid X receptor antagonist | 0.158 0.044 CHEMBL1228 0.122 0.098 CHEMBL3544828 | CHEMBL1228 | |
| 0.018 | 0.017 | 0.018 | Angiotensin AT2 receptor antagonist | |||
| 0.05 | 0.049 | 0.05 | Thromboxane synthase inhibitor | |||
| 0.024 | 0.023 | 0.024 | Complement factor 1s inhibitor | |||
| 0.04 | 0.04 | 0.063 | Adenosine deaminase inhibitor | 0.046 0.034 CHEMBL3544786 0.063 0.018 CHEMBL3544829 0.054 0.026 CHEMBL3544828 | CHEMBL3544829 | |
| 0.119 | 0.118 | 0.119 | Death-associated protein kinase 1 inhibitor | |||
| 0.051 | 0.052 | 0.083 | Biliverdin reductase inhibitor | 0.083 0.025 CHEMBL3544829 | CHEMBL3544829 | |
| 0.169 | 0.17 | 0.336 | DNA synthesis inhibitor | 0.336 0.033 CHEMBL3544786 0.181 0.152 CHEMBL1228 0.189 0.14 CHEMBL3544829 0.181 0.151 CHEMBL3544828 0.319 0.038 CHEMBL3544827 0.222 0.092 CHEMBL3544842 | CHEMBL3544786 | |
| 0.073 | 0.075 | 0.078 | Ornithine decarboxylase inhibitor | 0.078 0.069 CHEMBL1228 | CHEMBL1228 | |
| 0.066 | 0.07 | 0.082 | GABA aminotransferase inhibitor | 0.069 0.063 CHEMBL3544786 0.082 0.044 CHEMBL1228 0.07 0.061 CHEMBL3544827 | CHEMBL1228 | |
| 0.046 | 0.05 | 0.105 | Alcohol oxidase inhibitor | 0.083 0.023 CHEMBL1228 0.074 0.027 CHEMBL3544829 0.105 0.017 CHEMBL3544828 | CHEMBL3544828 | |
| 0.047 | 0.051 | 0.099 | Alpha-mannosidase inhibitor | 0.099 0.006 CHEMBL3544786 0.056 0.032 CHEMBL3544829 0.096 0.007 CHEMBL3544827 0.085 0.009 CHEMBL3544842 | CHEMBL3544786 | |
| 0.072 | 0.076 | 0.099 | Androgen antagonist | 0.093 0.052 CHEMBL1228 0.085 0.06 CHEMBL3544829 0.099 0.047 CHEMBL3544828 | CHEMBL3544828 | |
| 0.067 | 0.072 | 0.137 | Macrophage migration inhibitory factor inhibitor | 0.137 0.019 CHEMBL1228 0.069 0.068 CHEMBL3544828 | CHEMBL1228 | |
| 0.05 | 0.055 | 0.084 | Carbamoyl phosphate synthetase inhibitor | 0.084 0.026 CHEMBL3544829 0.059 0.044 CHEMBL3544828 | CHEMBL3544829 | |
| 0.063 | 0.07 | 0.08 | CDC25A inhibitor | 0.08 0.044 CHEMBL1228 | CHEMBL1228 | |
| 0.067 | 0.075 | 0.108 | Estrogen receptor alpha antagonist | 0.108 0.023 CHEMBL1228 | CHEMBL1228 | |
| 0.054 | 0.061 | 0.057 | Ryanodine receptor antagonist | 0.057 0.046 CHEMBL1228 | CHEMBL1228 | |
| 0.148 | 0.156 | 0.18 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.18 0.093 CHEMBL1228 | CHEMBL1228 | |
| 0.072 | 0.081 | 0.084 | Myeloperoxidase inhibitor | 0.084 0.06 CHEMBL1228 | CHEMBL1228 | |
| 0.008 | 0.019 | 0.035 | Prostaglandin EP4 agonist | 0.035 0.006 CHEMBL3544829 0.017 0.009 CHEMBL3544828 | CHEMBL3544829 | |
| 0.127 | 0.139 | 0.14 | Heat shock protein 70 antagonist | 0.129 0.128 CHEMBL3544786 0.137 0.089 CHEMBL1228 0.14 0.074 CHEMBL3544827 | CHEMBL3544827 | |
| 0.021 | 0.034 | 0.099 | Sodium/glucose cotransporter inhibitor | 0.073 0.004 CHEMBL3544786 0.024 0.022 CHEMBL1228 0.024 0.022 CHEMBL3544828 0.099 0.003 CHEMBL3544827 0.04 0.007 CHEMBL3544842 | CHEMBL3544827 | |
| 0.015 | 0.028 | 0.018 | Methylmalonyl-CoA mutase inhibitor | 0.018 0.014 CHEMBL3544829 | CHEMBL3544829 | |
| 0.031 | 0.045 | 0.054 | Dopamine D5 agonist | 0.054 0.015 CHEMBL1228 | CHEMBL1228 | |
| 0.024 | 0.038 | 0.054 | Arginase inhibitor | 0.036 0.025 CHEMBL3544786 0.054 0.013 CHEMBL3544827 | CHEMBL3544827 | |
| 0.02 | 0.035 | 0.03 | Thyroid hormone agonist | 0.03 0.013 CHEMBL1228 | CHEMBL1228 | |
| 0.024 | 0.04 | 0.045 | Fumarate hydratase inhibitor | 0.045 0.016 CHEMBL3544829 | CHEMBL3544829 | |
| 0.107 | 0.123 | 0.134 | Papain-like protease (SARS coronavirus) inhibitor | 0.134 0.053 CHEMBL1228 0.111 0.107 CHEMBL3544829 0.133 0.055 CHEMBL3544828 | CHEMBL1228 | |
| 0.01 | 0.026 | 0.043 | Ileal bile acid transport inhibitor | 0.028 0.005 CHEMBL3544786 0.043 0.004 CHEMBL3544827 | CHEMBL3544827 | |
| 0.059 | 0.076 | 0.091 | Glutamate dehydrogenase inhibitor | 0.091 0.036 CHEMBL3544829 0.072 0.053 CHEMBL3544828 | CHEMBL3544829 | |
| 0.018 | 0.035 | 0.025 | Prostaglandin EP4 antagonist | 0.025 0.019 CHEMBL3544829 | CHEMBL3544829 | |
| 0.146 | 0.163 | 0.337 | Vasodilator | 0.29 0.052 CHEMBL3544786 0.186 0.116 CHEMBL1228 0.24 0.075 CHEMBL3544829 0.254 0.067 CHEMBL3544828 0.337 0.037 CHEMBL3544827 0.27 0.059 CHEMBL3544842 | CHEMBL3544827 | |
| 0.034 | 0.052 | 0.1 | Mannosidase inhibitor | 0.1 0.006 CHEMBL3544786 0.042 0.036 CHEMBL3544829 0.097 0.006 CHEMBL3544827 0.072 0.011 CHEMBL3544842 | CHEMBL3544786 | |
| 0.009 | 0.027 | 0.025 | Prostacyclin agonist | 0.025 0.007 CHEMBL3544829 0.019 0.009 CHEMBL3544828 | CHEMBL3544829 | |
| 0.023 | 0.043 | 0.04 | Estradiol 17 beta-dehydrogenase 3 inhibitor | 0.04 0.016 CHEMBL1228 | CHEMBL1228 | |
| 0.016 | 0.038 | 0.02 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.02 0.017 CHEMBL3544829 | CHEMBL3544829 | |
| 0.024 | 0.047 | 0.036 | Farnesoid X receptor agonist | 0.036 0.028 CHEMBL3544829 | CHEMBL3544829 | |
| 0.072 | 0.096 | 0.155 | NADH dehydrogenase inhibitor | 0.155 0.016 CHEMBL3544786 0.096 0.049 CHEMBL3544829 0.086 0.063 CHEMBL3544828 0.119 0.029 CHEMBL3544827 0.124 0.027 CHEMBL3544842 | CHEMBL3544786 | |
| 0.041 | 0.066 | 0.07 | Leukotriene B4 antagonist | 0.051 0.043 CHEMBL3544786 0.051 0.043 CHEMBL1228 0.07 0.02 CHEMBL3544827 | CHEMBL3544827 | |
| 0.131 | 0.16 | 0.151 | Death-associated protein kinase 2 inhibitor | 0.151 0.105 CHEMBL1228 | CHEMBL1228 | |
| 0.041 | 0.071 | 0.07 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.058 0.037 CHEMBL3544786 0.062 0.032 CHEMBL3544829 0.07 0.026 CHEMBL3544842 | CHEMBL3544842 | |
| 0.043 | 0.074 | 0.057 | NMDA 2C receptor antagonist | 0.057 0.05 CHEMBL1228 | CHEMBL1228 | |
| 0.086 | 0.118 | 0.116 | Microtubule formation inhibitor | 0.116 0.066 CHEMBL3544786 0.105 0.082 CHEMBL3544829 0.097 0.096 CHEMBL3544828 0.116 0.066 CHEMBL3544827 | CHEMBL3544827 | |
| 0.011 | 0.042 | 0.02 | Telomerase stimulant | 0.02 0.008 CHEMBL3544786 0.016 0.015 CHEMBL3544842 | CHEMBL3544786 | |
| 0.046 | 0.078 | 0.057 | Leukotriene antagonist | 0.057 0.056 CHEMBL1228 | CHEMBL1228 | |
| 0.084 | 0.116 | 0.117 | DOPA decarboxylase inhibitor | 0.117 0.049 CHEMBL1228 0.095 0.086 CHEMBL3544828 | CHEMBL1228 | |
| 0.052 | 0.086 | 0.094 | Glutamate decarboxylase inhibitor | 0.075 0.049 CHEMBL1228 0.079 0.045 CHEMBL3544829 0.094 0.033 CHEMBL3544828 | CHEMBL3544828 | |
| 0.052 | 0.088 | 0.067 | Beta 3 adrenoreceptor antagonist | 0.067 0.04 CHEMBL1228 0.066 0.04 CHEMBL3544828 | CHEMBL1228 | |
| 0.016 | 0.054 | 0.021 | Vitamin D receptor antagonist | 0.021 0.017 CHEMBL3544829 0.021 0.018 CHEMBL3544828 | CHEMBL3544828 | |
| 0.035 | 0.075 | 0.17 | Prostaglandin EP2 antagonist | 0.17 0.008 CHEMBL3544829 0.14 0.011 CHEMBL3544828 0.06 0.041 CHEMBL3544827 0.059 0.042 CHEMBL3544842 | CHEMBL3544829 | |
| 0.022 | 0.063 | 0.071 | HMG CoA reductase inhibitor | 0.071 0.004 CHEMBL3544829 0.061 0.005 CHEMBL3544828 0.045 0.01 CHEMBL3544842 | CHEMBL3544829 | |
| 0.089 | 0.132 | 0.303 | Lipid peroxidase inhibitor | 0.248 0.027 CHEMBL3544786 0.195 0.044 CHEMBL1228 0.159 0.062 CHEMBL3544829 0.22 0.034 CHEMBL3544828 0.303 0.018 CHEMBL3544827 0.174 0.053 CHEMBL3544842 | CHEMBL3544827 | |
| 0.069 | 0.113 | 0.086 | Vanilloid agonist | 0.086 0.055 CHEMBL1228 | CHEMBL1228 | |
| 0.1 | 0.146 | 0.13 | Mannose-6-phosphate isomerase inhibitor | 0.13 0.086 CHEMBL3544786 0.121 0.1 CHEMBL3544829 0.115 0.109 CHEMBL3544842 | CHEMBL3544786 | |
| 0.056 | 0.103 | 0.067 | Peroxisome proliferator-activated receptor gamma antagonist | 0.067 0.06 CHEMBL3544829 | CHEMBL3544829 | |
| 0.018 | 0.065 | 0.031 | 1,3-Beta-glucan synthase inhibitor | 0.03 0.015 CHEMBL3544786 0.031 0.014 CHEMBL3544827 | CHEMBL3544827 | |
| 0.053 | 0.102 | 0.084 | Somatostatin 1 agonist | 0.077 0.055 CHEMBL1228 0.084 0.047 CHEMBL3544828 | CHEMBL3544828 | |
| 0.068 | 0.119 | 0.123 | Thioredoxin inhibitor | 0.108 0.04 CHEMBL3544786 0.085 0.071 CHEMBL1228 0.123 0.029 CHEMBL3544827 | CHEMBL3544827 | |
| 0.028 | 0.079 | 0.077 | Prostaglandin antagonist | 0.077 0.024 CHEMBL3544829 0.046 0.043 CHEMBL3544828 | CHEMBL3544829 | |
| 0.025 | 0.077 | 0.039 | NMDA receptor subunit 3B antagonist | 0.039 0.037 CHEMBL1228 | CHEMBL1228 | |
| 0.051 | 0.106 | 0.062 | Beta 2 adrenoreceptor agonist | 0.062 0.04 CHEMBL1228 0.061 0.047 CHEMBL3544828 | CHEMBL1228 | |
| 0.032 | 0.088 | 0.064 | Beta 1 adrenoreceptor antagonist | 0.049 0.048 CHEMBL1228 0.051 0.045 CHEMBL3544829 0.064 0.032 CHEMBL3544828 | CHEMBL3544828 | |
| 0.088 | 0.144 | 0.159 | Interleukin 4 antagonist | 0.159 0.042 CHEMBL3544786 0.159 0.042 CHEMBL1228 0.149 0.051 CHEMBL3544827 | CHEMBL1228 | |
| 0.068 | 0.124 | 0.106 | Carbonic anhydrase III inhibitor | 0.106 0.056 CHEMBL1228 | CHEMBL1228 | |
| 0.206 | 0.264 | 0.378 | Calcium channel L-type activator | 0.378 0.097 CHEMBL1228 0.266 0.188 CHEMBL3544829 0.37 0.103 CHEMBL3544828 | CHEMBL1228 | |
| 0.054 | 0.113 | 0.076 | Keratolytic | 0.076 0.055 CHEMBL1228 | CHEMBL1228 | |
| 0.036 | 0.097 | 0.057 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.053 0.049 CHEMBL3544786 0.057 0.043 CHEMBL1228 0.055 0.046 CHEMBL3544827 | CHEMBL1228 | |
| 0.04 | 0.102 | 0.134 | Phenylalanine 4-hydroxylase inhibitor | 0.066 0.05 CHEMBL1228 0.102 0.025 CHEMBL3544829 0.134 0.015 CHEMBL3544828 | CHEMBL3544828 | |
| 0.037 | 0.1 | 0.048 | Vanilloid 2 antagonist | 0.048 0.047 CHEMBL1228 | CHEMBL1228 | |
| 0.039 | 0.102 | 0.06 | Leukotriene synthesis inhibitor | 0.06 0.055 CHEMBL1228 | CHEMBL1228 | |
| 0.028 | 0.092 | 0.046 | Beta 2 adrenoreceptor antagonist | 0.046 0.042 CHEMBL1228 | CHEMBL1228 | |
| 0.035 | 0.099 | 0.109 | Heparanase inhibitor | 0.091 0.004 CHEMBL3544786 0.109 0.004 CHEMBL3544827 | CHEMBL3544827 | |
| 0.101 | 0.166 | 0.371 | Hemostatic | 0.185 0.039 CHEMBL3544786 0.371 0.01 CHEMBL3544827 | CHEMBL3544827 | |
| 0.026 | 0.094 | 0.151 | Neuraminidase (Influenza A) inhibitor | 0.055 0.018 CHEMBL3544786 0.049 0.026 CHEMBL3544829 0.046 0.03 CHEMBL3544828 0.057 0.015 CHEMBL3544827 0.151 0.003 CHEMBL3544842 | CHEMBL3544842 | |
| 0.201 | 0.272 | 0.553 | Apoptosis agonist | 0.553 0.06 CHEMBL3544786 0.322 0.157 CHEMBL1228 0.293 0.177 CHEMBL3544828 0.546 0.061 CHEMBL3544827 0.432 0.099 CHEMBL3544842 | CHEMBL3544786 | |
| 0.05 | 0.121 | 0.122 | Adrenaline agonist | 0.087 0.049 CHEMBL1228 0.084 0.052 CHEMBL3544829 0.122 0.025 CHEMBL3544828 | CHEMBL3544828 | |
| 0.069 | 0.144 | 0.382 | Amylase inhibitor | 0.3 0.018 CHEMBL3544786 0.134 0.073 CHEMBL1228 0.224 0.036 CHEMBL3544829 0.283 0.021 CHEMBL3544828 0.376 0.011 CHEMBL3544827 0.382 0.01 CHEMBL3544842 | CHEMBL3544842 | |
| 0.008 | 0.084 | 0.048 | Squalene synthetase inhibitor | 0.048 0.015 CHEMBL3544786 0.038 0.019 CHEMBL3544827 | CHEMBL3544786 | |
| 0.002 | 0.08 | 0.019 | Antibiotic Macrolide-like | 0.019 0.007 CHEMBL3544786 0.017 0.008 CHEMBL3544842 | CHEMBL3544786 | |
| 0.141 | 0.22 | 0.383 | Peptidyltransferase inhibitor | 0.383 0.008 CHEMBL3544786 0.194 0.108 CHEMBL1228 0.228 0.068 CHEMBL3544829 0.236 0.061 CHEMBL3544828 0.378 0.009 CHEMBL3544827 0.344 0.013 CHEMBL3544842 | CHEMBL3544786 | |
| 0.025 | 0.106 | 0.163 | Protein 50S ribosomal subunit inhibitor | 0.163 0.006 CHEMBL3544786 0.101 0.013 CHEMBL3544827 0.148 0.007 CHEMBL3544842 | CHEMBL3544786 | |
| 0.11 | 0.191 | 0.366 | Hypolipemic | 0.233 0.075 CHEMBL3544786 0.366 0.032 CHEMBL3544829 0.339 0.038 CHEMBL3544828 0.302 0.048 CHEMBL3544827 0.193 0.1 CHEMBL3544842 | CHEMBL3544829 | |
| 0.063 | 0.146 | 0.079 | D-Ala-D-Ala ligase inhibitor | 0.079 0.07 CHEMBL1228 | CHEMBL1228 | |
| 0.043 | 0.126 | 0.077 | Lipocortins synthesis agonist | 0.077 0.015 CHEMBL3544786 0.067 0.025 CHEMBL3544827 0.061 0.034 CHEMBL3544842 | CHEMBL3544786 | |
| 0.058 | 0.146 | 0.076 | MAP kinase kinase 7 inhibitor | 0.076 0.058 CHEMBL1228 0.073 0.071 CHEMBL3544828 | CHEMBL1228 | |
| 0.015 | 0.104 | 0.036 | Estradiol 17 beta-dehydrogenase inhibitor | 0.036 0.034 CHEMBL1228 | CHEMBL1228 | |
| 0.067 | 0.156 | 0.094 | Nav1.4 sodium channel blocker | 0.094 0.085 CHEMBL1228 | CHEMBL1228 | |
| 0.065 | 0.159 | 0.094 | Mucolytic | 0.093 0.088 CHEMBL3544786 0.094 0.087 CHEMBL3544828 | CHEMBL3544828 | |
| 0.009 | 0.105 | 0.071 | Sodium/glucose cotransporter 2 inhibitor | 0.05 0.006 CHEMBL3544786 0.071 0.004 CHEMBL3544827 0.027 0.017 CHEMBL3544842 | CHEMBL3544827 | |
| 0.007 | 0.107 | 0.033 | Prostaglandin EP3 antagonist | 0.033 0.019 CHEMBL3544829 | CHEMBL3544829 | |
| 0.094 | 0.194 | 0.208 | DNA methyltransferase I inhibitor | 0.208 0.065 CHEMBL3544827 | CHEMBL3544827 | |
| 0.009 | 0.112 | 0.022 | Antibiotic Anthracycline-like | 0.022 0.007 CHEMBL3544786 0.019 0.014 CHEMBL3544827 0.019 0.014 CHEMBL3544842 | CHEMBL3544786 | |
| 0.035 | 0.139 | 0.067 | Beta adrenoreceptor antagonist | 0.067 0.043 CHEMBL3544828 | CHEMBL3544828 | |
| 0.049 | 0.155 | 0.158 | Mediator release inhibitor | 0.11 0.059 CHEMBL3544786 0.158 0.025 CHEMBL3544827 | CHEMBL3544827 | |
| 0.08 | 0.186 | 0.66 | Angiogenesis stimulant | 0.628 0.005 CHEMBL3544786 0.176 0.107 CHEMBL1228 0.151 0.122 CHEMBL3544828 0.66 0.005 CHEMBL3544827 0.388 0.024 CHEMBL3544842 | CHEMBL3544827 | |
| 0.041 | 0.154 | 0.25 | Monophenol monooxygenase inhibitor | 0.185 0.037 CHEMBL3544786 0.108 0.07 CHEMBL1228 0.118 0.063 CHEMBL3544828 0.25 0.024 CHEMBL3544827 | CHEMBL3544827 | |
| 0.06 | 0.175 | 0.184 | Alkylator | 0.184 0.031 CHEMBL3544786 0.147 0.048 CHEMBL3544827 0.119 0.069 CHEMBL3544842 | CHEMBL3544786 | |
| 0.103 | 0.22 | 0.52 | Free radical scavenger | 0.41 0.027 CHEMBL3544786 0.275 0.059 CHEMBL1228 0.26 0.064 CHEMBL3544828 0.52 0.014 CHEMBL3544827 0.238 0.074 CHEMBL3544842 | CHEMBL3544827 | |
| 0.087 | 0.208 | 0.382 | Platelet adhesion inhibitor | 0.333 0.024 CHEMBL3544786 0.382 0.014 CHEMBL3544827 | CHEMBL3544827 | |
| 0.044 | 0.171 | 0.103 | 5-Lipoxygenase inhibitor | 0.103 0.062 CHEMBL1228 | CHEMBL1228 | |
| 0.028 | 0.156 | 0.045 | Beta adrenoreceptor agonist | 0.045 0.033 CHEMBL3544828 | CHEMBL3544828 | |
| 0.037 | 0.169 | 0.075 | NMDA receptor antagonist | 0.075 0.071 CHEMBL3544828 | CHEMBL3544828 | |
| 0.141 | 0.274 | 0.496 | Alpha-glucosidase inhibitor | 0.244 0.191 CHEMBL1228 0.264 0.179 CHEMBL3544828 0.496 0.082 CHEMBL3544827 | CHEMBL3544827 | |
| 0.055 | 0.195 | 0.214 | AMP-activated protein kinase stimulant | 0.17 0.018 CHEMBL3544786 0.214 0.009 CHEMBL3544827 | CHEMBL3544827 | |
| 0.059 | 0.2 | 0.164 | Toll-Like receptor 4 antagonist | 0.162 0.015 CHEMBL3544786 0.095 0.079 CHEMBL1228 0.164 0.014 CHEMBL3544827 0.143 0.025 CHEMBL3544842 | CHEMBL3544827 | |
| 0.044 | 0.189 | 0.201 | Expectorant | 0.182 0.025 CHEMBL3544786 0.1 0.069 CHEMBL3544829 0.111 0.057 CHEMBL3544828 0.201 0.02 CHEMBL3544827 0.111 0.058 CHEMBL3544842 | CHEMBL3544827 | |
| 0.063 | 0.211 | 0.155 | Estrogen antagonist | 0.155 0.021 CHEMBL1228 0.118 0.059 CHEMBL3544828 | CHEMBL1228 | |
| 0.078 | 0.226 | 0.2 | Hexokinase inhibitor | 0.2 0.035 CHEMBL3544786 0.2 0.035 CHEMBL3544827 0.13 0.104 CHEMBL3544842 | CHEMBL3544827 | |
| 0.083 | 0.237 | 0.21 | DNA methylase inhibitor | 0.21 0.073 CHEMBL3544827 | CHEMBL3544827 | |
| 0.004 | 0.17 | 0.039 | Estrogen receptor alpha agonist | 0.039 0.021 CHEMBL1228 | CHEMBL1228 | |
| 0.049 | 0.218 | 0.17 | Beta glucuronidase inhibitor | 0.117 0.049 CHEMBL3544786 0.17 0.018 CHEMBL3544827 | CHEMBL3544827 | |
| 0.075 | 0.263 | 0.396 | Hepatoprotectant | 0.375 0.016 CHEMBL3544786 0.186 0.075 CHEMBL3544829 0.204 0.063 CHEMBL3544828 0.396 0.014 CHEMBL3544827 0.306 0.028 CHEMBL3544842 | CHEMBL3544827 | |
| 0.13 | 0.325 | 0.409 | Apoptosis antagonist | 0.36 0.051 CHEMBL3544786 0.208 0.169 CHEMBL1228 0.213 0.163 CHEMBL3544828 0.409 0.036 CHEMBL3544827 0.278 0.102 CHEMBL3544842 | CHEMBL3544827 | |
| 0.02 | 0.216 | 0.062 | Nitric oxide donor | 0.062 0.044 CHEMBL3544827 | CHEMBL3544827 | |
| 0.009 | 0.207 | 0.048 | Protein 30S ribosomal subunit inhibitor | 0.046 0.009 CHEMBL3544786 0.048 0.008 CHEMBL3544827 0.039 0.01 CHEMBL3544842 | CHEMBL3544827 | |
| 0.004 | 0.206 | 0.029 | Estrogen receptor beta agonist | 0.029 0.024 CHEMBL1228 | CHEMBL1228 | |
| 0.046 | 0.253 | 0.308 | Thrombolytic | 0.308 0.023 CHEMBL3544786 0.293 0.025 CHEMBL3544827 | CHEMBL3544786 | |
| 0.017 | 0.234 | 0.072 | Antibiotic Aminoglycoside-like | 0.072 0.005 CHEMBL3544786 0.07 0.006 CHEMBL3544827 0.071 0.006 CHEMBL3544842 | CHEMBL3544786 | |
| 0.041 | 0.261 | 0.132 | Estrogen receptor beta antagonist | 0.132 0.022 CHEMBL1228 0.102 0.06 CHEMBL3544828 | CHEMBL1228 | |
| 0.067 | 0.292 | 0.348 | Nitric oxide antagonist | 0.307 0.039 CHEMBL3544786 0.13 0.119 CHEMBL1228 0.132 0.115 CHEMBL3544829 0.169 0.082 CHEMBL3544828 0.348 0.032 CHEMBL3544827 0.262 0.048 CHEMBL3544842 | CHEMBL3544827 | |
| 0.007 | 0.235 | 0.054 | Estrogen agonist | 0.054 0.033 CHEMBL1228 | CHEMBL1228 | |
| 0.078 | 0.31 | 0.552 | Antioxidant | 0.481 0.022 CHEMBL3544786 0.24 0.089 CHEMBL1228 0.245 0.087 CHEMBL3544828 0.552 0.015 CHEMBL3544827 0.378 0.039 CHEMBL3544842 | CHEMBL3544827 | |
| 0.012 | 0.251 | 0.264 | Antineoplastic antibiotic | 0.213 0.019 CHEMBL3544786 0.068 0.067 CHEMBL3544828 0.164 0.028 CHEMBL3544827 0.264 0.013 CHEMBL3544842 | CHEMBL3544842 | |
| 0.066 | 0.326 | 0.139 | DNA repair enzyme inhibitor | 0.137 0.045 CHEMBL3544786 0.139 0.043 CHEMBL3544827 | CHEMBL3544827 | |
| 0.011 | 0.282 | 0.203 | Neuraminidase inhibitor | 0.063 0.04 CHEMBL3544786 0.057 0.047 CHEMBL3544828 0.072 0.032 CHEMBL3544827 0.203 0.004 CHEMBL3544842 | CHEMBL3544842 | |
| 0.016 | 0.295 | 0.214 | Neuraminidase (influenza) inhibitor | 0.071 0.033 CHEMBL3544786 0.063 0.046 CHEMBL3544828 0.078 0.027 CHEMBL3544827 0.214 0.004 CHEMBL3544842 | CHEMBL3544842 | |
| 0.039 | 0.32 | 0.127 | Bone formation stimulant | 0.127 0.079 CHEMBL3544786 0.108 0.098 CHEMBL3544828 | CHEMBL3544786 | |
| 0.012 | 0.298 | 0.334 | Selectin antagonist | 0.316 0.005 CHEMBL3544786 0.334 0.004 CHEMBL3544827 0.259 0.008 CHEMBL3544842 | CHEMBL3544827 | |
| 0.009 | 0.299 | 0.041 | Macrophage elastase inhibitor | 0.041 0.033 CHEMBL3544829 | CHEMBL3544829 | |
| 0.06 | 0.355 | 0.244 | Insulin secretagoues | 0.19 0.042 CHEMBL3544786 0.244 0.02 CHEMBL3544829 0.225 0.025 CHEMBL3544828 0.229 0.024 CHEMBL3544827 0.184 0.045 CHEMBL3544842 | CHEMBL3544829 | |
| 0.09 | 0.392 | 0.213 | Antiobesity | 0.213 0.194 CHEMBL3544827 | CHEMBL3544827 | |
| 0.015 | 0.334 | 0.094 | Protein-tyrosine phosphatase 1B inhibitor | 0.094 0.084 CHEMBL3544827 | CHEMBL3544827 | |
| 0.04 | 0.372 | 0.129 | Transcription factor NF kappa B stimulant | 0.129 0.022 CHEMBL3544786 0.125 0.023 CHEMBL3544827 0.116 0.027 CHEMBL3544842 | CHEMBL3544786 | |
| 0.018 | 0.352 | 0.078 | Glucose-6-phosphate translocase inhibitor | 0.072 0.015 CHEMBL3544786 0.078 0.012 CHEMBL3544827 | CHEMBL3544827 | |
| 0.082 | 0.427 | 0.808 | Immunomodulator | 0.808 0.004 CHEMBL3544786 0.382 0.049 CHEMBL3544827 0.718 0.005 CHEMBL3544842 | CHEMBL3544786 | |
| 0.023 | 0.381 | 0.113 | ATPase (Vacuolar H+) inhibitor | 0.097 0.044 CHEMBL3544786 0.113 0.025 CHEMBL3544827 0.103 0.036 CHEMBL3544842 | CHEMBL3544827 | |
| 0.026 | 0.384 | 0.063 | Adenine nucleotide translocase inhibitor | 0.063 0.024 CHEMBL3544786 0.061 0.027 CHEMBL3544827 | CHEMBL3544786 | |
| 0.052 | 0.423 | 0.25 | NOS3 expression enhancer | 0.211 0.037 CHEMBL3544786 0.25 0.026 CHEMBL3544827 0.151 0.071 CHEMBL3544842 | CHEMBL3544827 | |
| 0.046 | 0.43 | 0.236 | Interleukin 6 antagonist | 0.236 0.026 CHEMBL3544786 0.182 0.053 CHEMBL3544827 0.186 0.05 CHEMBL3544842 | CHEMBL3544786 | |
| 0.01 | 0.414 | 0.031 | Estrogen-related receptor beta antagonist | 0.031 0.026 CHEMBL1228 | CHEMBL1228 | |
| 0.057 | 0.489 | 0.576 | Hypoglycemic | 0.486 0.016 CHEMBL3544786 0.2 0.112 CHEMBL3544829 0.245 0.08 CHEMBL3544828 0.576 0.009 CHEMBL3544827 0.333 0.042 CHEMBL3544842 | CHEMBL3544827 | |
| 0.015 | 0.462 | 0.179 | Topoisomerase I inhibitor | 0.179 0.032 CHEMBL3544786 0.17 0.034 CHEMBL3544827 0.085 0.084 CHEMBL3544842 | CHEMBL3544786 | |
| 0.017 | 0.484 | 0.097 | Cell adhesion molecule inhibitor | 0.095 0.038 CHEMBL3544786 0.097 0.037 CHEMBL3544827 | CHEMBL3544827 | |
| 0.063 | 0.585 | 0.23 | Caspase 3 stimulant | 0.193 0.18 CHEMBL3544786 0.23 0.131 CHEMBL3544827 | CHEMBL3544827 | |
| 0.022 | 0.576 | 0.187 | Cell adhesion inhibitor | 0.179 0.031 CHEMBL3544786 0.187 0.028 CHEMBL3544827 | CHEMBL3544827 | |
| 0.02 | 0.589 | 0.201 | Interleukin antagonist | 0.134 0.132 CHEMBL3544829 0.201 0.084 CHEMBL3544828 | CHEMBL3544828 | |
| 0.014 | 0.603 | 0.072 | Factor IXa inhibitor | 0.072 0.019 CHEMBL3544786 0.068 0.021 CHEMBL3544827 | CHEMBL3544786 | |
| 0.032 | 0.63 | 0.093 | Interleukin 12 antagonist | 0.089 0.074 CHEMBL3544828 0.093 0.066 CHEMBL3544827 | CHEMBL3544827 | |
| 0.023 | 0.646 | 0.31 | Tumour necrosis factor alpha release inhibitor | 0.203 0.107 CHEMBL3544786 0.31 0.05 CHEMBL3544827 0.155 0.152 CHEMBL3544842 | CHEMBL3544827 | |
| 0.004 | 0.648 | 0.31 | S-adenosyl-L-homocysteine hydrolase inhibitor | 0.31 0.002 CHEMBL3544842 | CHEMBL3544842 | |
| 0.01 | 0.658 | 0.094 | Topoisomerase II alpha inhibitor | 0.09 0.046 CHEMBL3544786 0.094 0.043 CHEMBL3544827 | CHEMBL3544827 | |
| 0.067 | 0.727 | 0.141 | CC chemokine 6 receptor antagonist | 0.141 0.038 CHEMBL3544786 0.135 0.055 CHEMBL3544827 | CHEMBL3544786 | |
| 0.006 | 0.779 | 0.143 | Topoisomerase II inhibitor | 0.123 0.065 CHEMBL3544786 0.143 0.053 CHEMBL3544827 | CHEMBL3544827 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |