Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9020.0050.904Antiinflammatory

0.7 0.031 CHEMBL3544786

0.868 0.008 CHEMBL1228

0.881 0.006 CHEMBL3544829

0.857 0.009 CHEMBL3544828

0.904 0.005 CHEMBL3544827

0.475 0.098 CHEMBL3544842

CHEMBL3544827
0.7790.0070.779Analgesic

0.702 0.013 CHEMBL1228

0.584 0.03 CHEMBL3544829

0.541 0.039 CHEMBL3544828

0.361 0.103 CHEMBL3544827

0.5760.0140.6615 Hydroxytryptamine release inhibitor

0.582 0.013 CHEMBL3544786

0.6 0.011 CHEMBL1228

0.524 0.025 CHEMBL3544829

0.533 0.023 CHEMBL3544828

0.661 0.005 CHEMBL3544827

0.356 0.11 CHEMBL3544842

CHEMBL3544827
0.5460.0210.7455 Hydroxytryptamine release stimulant

0.262 0.083 CHEMBL3544786

0.559 0.019 CHEMBL1228

0.735 0.005 CHEMBL3544829

0.745 0.005 CHEMBL3544828

0.396 0.047 CHEMBL3544827

0.522 0.024 CHEMBL3544842

CHEMBL3544828
0.5460.0230.882Antithrombotic

0.732 0.006 CHEMBL3544786

0.563 0.02 CHEMBL1228

0.568 0.02 CHEMBL3544829

0.562 0.02 CHEMBL3544828

0.882 0.003 CHEMBL3544827

0.44 0.04 CHEMBL3544842

CHEMBL3544827
0.5140.0220.543GABA C receptor rho-3 antagonist

0.543 0.016 CHEMBL1228

0.263 0.143 CHEMBL3544829

0.312 0.108 CHEMBL3544828

CHEMBL1228
0.4790.0040.479Uric acid excretion stimulant

0.14 0.027 CHEMBL3544786

0.434 0.004 CHEMBL1228

0.381 0.004 CHEMBL3544829

0.363 0.004 CHEMBL3544828

0.366 0.004 CHEMBL3544827

0.4470.0140.447Platelet aggregation inhibitor

0.313 0.033 CHEMBL1228

0.314 0.033 CHEMBL3544829

0.238 0.057 CHEMBL3544828

0.235 0.059 CHEMBL3544827

0.440.010.744Non-steroidal antiinflammatory agent

0.336 0.022 CHEMBL3544786

0.461 0.009 CHEMBL1228

0.494 0.007 CHEMBL3544829

0.498 0.007 CHEMBL3544828

0.744 0.003 CHEMBL3544827

CHEMBL3544827
0.4290.0030.509UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.333 0.005 CHEMBL3544786

0.382 0.004 CHEMBL1228

0.509 0.002 CHEMBL3544829

0.445 0.003 CHEMBL3544828

0.467 0.003 CHEMBL3544827

0.235 0.011 CHEMBL3544842

CHEMBL3544829
0.4610.0450.614Histamine release inhibitor

0.583 0.012 CHEMBL3544786

0.508 0.026 CHEMBL1228

0.508 0.026 CHEMBL3544829

0.535 0.019 CHEMBL3544828

0.614 0.009 CHEMBL3544827

0.29 0.129 CHEMBL3544842

CHEMBL3544827
0.4570.0450.553Immunosuppressant

0.493 0.035 CHEMBL3544786

0.439 0.05 CHEMBL1228

0.462 0.043 CHEMBL3544829

0.439 0.05 CHEMBL3544828

0.553 0.02 CHEMBL3544827

0.384 0.07 CHEMBL3544842

CHEMBL3544827
0.3910.0030.391Electrolyte absorption antagonist

0.303 0.004 CHEMBL1228

0.29 0.004 CHEMBL3544829

0.208 0.007 CHEMBL3544828

0.103 0.054 CHEMBL3544827

0.430.0640.716Antibacterial

0.668 0.011 CHEMBL3544786

0.478 0.047 CHEMBL1228

0.451 0.056 CHEMBL3544829

0.475 0.048 CHEMBL3544828

0.716 0.008 CHEMBL3544827

0.552 0.028 CHEMBL3544842

CHEMBL3544827
0.3880.0420.562Spasmolytic

0.316 0.064 CHEMBL3544786

0.437 0.033 CHEMBL1228

0.463 0.029 CHEMBL3544829

0.489 0.024 CHEMBL3544828

0.562 0.017 CHEMBL3544827

CHEMBL3544827
0.3660.0340.44Platelet antagonist

0.362 0.035 CHEMBL3544786

0.316 0.048 CHEMBL1228

0.316 0.048 CHEMBL3544829

0.268 0.065 CHEMBL3544828

0.44 0.02 CHEMBL3544827

CHEMBL3544827
0.3490.0260.3495 Hydroxytryptamine uptake stimulant

0.342 0.028 CHEMBL1228

0.228 0.107 CHEMBL3544829

0.226 0.109 CHEMBL3544828

0.3150.0120.315Cyclooxygenase 1 inhibitor

0.31 0.013 CHEMBL1228

0.209 0.031 CHEMBL3544829

0.222 0.027 CHEMBL3544828

0.202 0.033 CHEMBL3544827

0.101 0.099 CHEMBL3544842

0.3990.1020.399Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.277 0.246 CHEMBL1228

0.309 0.2 CHEMBL3544829

0.3570.0610.68Cholesterol antagonist

0.632 0.015 CHEMBL3544786

0.448 0.041 CHEMBL1228

0.34 0.068 CHEMBL3544829

0.37 0.057 CHEMBL3544828

0.68 0.009 CHEMBL3544827

0.345 0.066 CHEMBL3544842

CHEMBL3544827
0.2950.0080.295Ferrochelatase inhibitor

0.17 0.03 CHEMBL1228

0.233 0.016 CHEMBL3544829

0.104 0.066 CHEMBL3544828

0.3120.0270.42P-glycoprotein inhibitor

0.282 0.033 CHEMBL1228

0.42 0.014 CHEMBL3544829

0.388 0.018 CHEMBL3544828

0.249 0.042 CHEMBL3544827

CHEMBL3544829
0.3050.030.305Gastrin inhibitor

0.194 0.157 CHEMBL3544786

0.261 0.067 CHEMBL1228

0.247 0.083 CHEMBL3544829

0.189 0.166 CHEMBL3544828

0.222 0.116 CHEMBL3544827

0.290.0190.29Cyclooxygenase inhibitor

0.27 0.022 CHEMBL1228

0.213 0.037 CHEMBL3544829

0.212 0.037 CHEMBL3544828

0.188 0.047 CHEMBL3544827

0.2780.0170.321Phospholipase A2 inhibitor

0.18 0.054 CHEMBL3544786

0.321 0.011 CHEMBL1228

0.211 0.037 CHEMBL3544829

0.226 0.031 CHEMBL3544828

0.281 0.017 CHEMBL3544827

CHEMBL1228
0.2940.0360.364Tyrosine 3 hydroxylase inhibitor

0.364 0.013 CHEMBL1228

0.237 0.081 CHEMBL3544829

0.283 0.043 CHEMBL3544828

CHEMBL1228
0.380.1230.47Caspase 9 stimulant

0.47 0.073 CHEMBL3544786

0.449 0.083 CHEMBL1228

0.289 0.207 CHEMBL3544829

0.338 0.156 CHEMBL3544828

0.424 0.097 CHEMBL3544827

0.324 0.169 CHEMBL3544842

CHEMBL3544786
0.2730.0410.308Anesthetic general

0.308 0.031 CHEMBL3544786

0.299 0.033 CHEMBL1228

0.253 0.049 CHEMBL3544829

0.256 0.048 CHEMBL3544828

0.277 0.039 CHEMBL3544827

0.175 0.09 CHEMBL3544842

CHEMBL3544786
0.3020.0770.356Sodium/bile acid cotransporter inhibitor

0.248 0.13 CHEMBL3544786

0.356 0.036 CHEMBL1228

0.274 0.103 CHEMBL3544829

0.322 0.06 CHEMBL3544828

0.296 0.083 CHEMBL3544827

CHEMBL1228
0.2710.0530.2715 Hydroxytryptamine 1E antagonist

0.263 0.061 CHEMBL1228

0.2920.0790.45Interleukin 2 agonist

0.45 0.015 CHEMBL3544786

0.318 0.062 CHEMBL1228

0.261 0.107 CHEMBL3544829

0.273 0.095 CHEMBL3544828

0.444 0.017 CHEMBL3544827

0.395 0.029 CHEMBL3544842

CHEMBL3544786
0.3090.0970.309Thioredoxin glutathione reductase inhibitor

0.288 0.11 CHEMBL1228

0.2420.0320.437Diuretic

0.216 0.039 CHEMBL3544786

0.207 0.041 CHEMBL1228

0.186 0.05 CHEMBL3544829

0.157 0.071 CHEMBL3544828

0.437 0.011 CHEMBL3544827

CHEMBL3544827
0.3020.0960.38Vasodilator, peripheral

0.223 0.151 CHEMBL3544786

0.308 0.093 CHEMBL1228

0.38 0.062 CHEMBL3544829

0.367 0.067 CHEMBL3544828

0.287 0.104 CHEMBL3544827

CHEMBL3544829
0.2780.0730.296Insulysin inhibitor

0.296 0.061 CHEMBL1228

0.223 0.125 CHEMBL3544829

0.233 0.113 CHEMBL3544828

CHEMBL1228
0.2060.0120.206GABA C receptor antagonist

0.196 0.014 CHEMBL1228

0.158 0.026 CHEMBL3544829

0.139 0.037 CHEMBL3544828

0.2340.0420.322Anticoagulant

0.193 0.056 CHEMBL3544786

0.174 0.064 CHEMBL1228

0.156 0.075 CHEMBL3544829

0.127 0.103 CHEMBL3544828

0.322 0.025 CHEMBL3544827

CHEMBL3544827
0.2930.1050.335Prostaglandin dehydrogenase inhibitor

0.335 0.088 CHEMBL1228

CHEMBL1228
0.2220.0340.454Protein kinase stimulant

0.315 0.015 CHEMBL3544786

0.274 0.021 CHEMBL1228

0.146 0.071 CHEMBL3544829

0.171 0.055 CHEMBL3544828

0.454 0.005 CHEMBL3544827

0.171 0.055 CHEMBL3544842

CHEMBL3544827
0.1990.0120.199Sphingosine 1-phosphate receptor 5 antagonist

0.194 0.014 CHEMBL1228

0.134 0.091 CHEMBL3544829

0.2160.0370.228Succinate dehydrogenase inhibitor

0.228 0.031 CHEMBL1228

0.201 0.048 CHEMBL3544829

0.192 0.055 CHEMBL3544828

CHEMBL1228
0.2040.0270.204GABA C receptor rho-2 antagonist

0.2 0.029 CHEMBL1228

0.124 0.117 CHEMBL3544829

0.123 0.118 CHEMBL3544828

0.2530.0760.418Interleukin agonist

0.418 0.016 CHEMBL3544786

0.242 0.085 CHEMBL1228

0.231 0.093 CHEMBL3544829

0.209 0.113 CHEMBL3544828

0.374 0.023 CHEMBL3544827

0.288 0.054 CHEMBL3544842

CHEMBL3544786
0.1880.0120.188Sphingosine 1-phosphate receptor 4 antagonist

0.172 0.018 CHEMBL1228

0.124 0.065 CHEMBL3544829

0.107 0.1 CHEMBL3544828

0.1810.0060.181Acetylcholine release stimulant

0.155 0.014 CHEMBL3544786

0.145 0.02 CHEMBL1228

0.109 0.068 CHEMBL3544829

0.153 0.015 CHEMBL3544827

0.2030.030.21Arachidonic acid antagonist

0.175 0.059 CHEMBL3544786

0.21 0.024 CHEMBL1228

0.186 0.048 CHEMBL3544829

0.186 0.047 CHEMBL3544828

0.147 0.092 CHEMBL3544827

CHEMBL1228
0.2340.0650.234Psychostimulant

0.166 0.103 CHEMBL3544786

0.219 0.07 CHEMBL1228

0.227 0.067 CHEMBL3544827

0.180.0180.267Photosensitizer

0.174 0.02 CHEMBL3544786

0.182 0.017 CHEMBL1228

0.099 0.09 CHEMBL3544829

0.097 0.095 CHEMBL3544828

0.267 0.005 CHEMBL3544827

CHEMBL3544827
0.1880.0260.188Cathepsin H inhibitor

0.158 0.041 CHEMBL1228

0.174 0.032 CHEMBL3544829

0.15 0.046 CHEMBL3544828

0.1690.0160.206Prolactin inhibitor

0.206 0.008 CHEMBL1228

0.089 0.068 CHEMBL3544829

0.112 0.044 CHEMBL3544828

CHEMBL1228
0.2050.0530.205Lipocortins synthesis antagonist

0.201 0.055 CHEMBL3544786

0.192 0.061 CHEMBL1228

0.17 0.08 CHEMBL3544829

0.153 0.1 CHEMBL3544828

0.173 0.078 CHEMBL3544827

0.2150.0630.273Neurotrophic factor enhancer

0.234 0.048 CHEMBL3544786

0.268 0.029 CHEMBL1228

0.165 0.117 CHEMBL3544829

0.206 0.07 CHEMBL3544828

0.273 0.027 CHEMBL3544827

0.151 0.137 CHEMBL3544842

CHEMBL3544827
0.1690.020.189TRPA1 agonist

0.189 0.013 CHEMBL1228

0.101 0.085 CHEMBL3544829

0.119 0.06 CHEMBL3544828

0.119 0.059 CHEMBL3544827

CHEMBL1228
0.170.0210.17Sphingosine 1-phosphate receptor 2 antagonist

0.166 0.024 CHEMBL1228

0.1830.0360.183Cyclooxygenase 2 inhibitor

0.167 0.043 CHEMBL1228

0.122 0.077 CHEMBL3544829

0.123 0.076 CHEMBL3544828

0.126 0.074 CHEMBL3544827

0.1620.0210.172Ca2+-transporting ATPase inhibitor

0.172 0.012 CHEMBL3544786

0.159 0.024 CHEMBL1228

0.145 0.057 CHEMBL3544829

0.138 0.079 CHEMBL3544828

0.155 0.033 CHEMBL3544827

0.132 0.111 CHEMBL3544842

CHEMBL3544786
0.180.040.379Cell wall synthesis inhibitor

0.262 0.014 CHEMBL3544786

0.187 0.036 CHEMBL1228

0.172 0.045 CHEMBL3544829

0.167 0.05 CHEMBL3544828

0.379 0.007 CHEMBL3544827

0.146 0.069 CHEMBL3544842

CHEMBL3544827
0.1570.0210.253Creatine kinase inhibitor

0.253 0.005 CHEMBL1228

0.107 0.052 CHEMBL3544829

0.157 0.021 CHEMBL3544828

CHEMBL1228
0.1440.0080.166Androgen agonist

0.166 0.006 CHEMBL1228

0.107 0.013 CHEMBL3544829

0.114 0.011 CHEMBL3544828

0.054 0.05 CHEMBL3544827

CHEMBL1228
0.1830.0470.212Neurotensin receptor agonist

0.212 0.03 CHEMBL1228

0.151 0.099 CHEMBL3544828

CHEMBL1228
0.160.030.16GABA C receptor agonist

0.134 0.041 CHEMBL1228

0.145 0.036 CHEMBL3544829

0.101 0.066 CHEMBL3544828

0.2210.0940.221Calpain inhibitor

0.19 0.124 CHEMBL1228

0.1760.0530.383Interferon gamma antagonist

0.304 0.019 CHEMBL3544786

0.218 0.035 CHEMBL1228

0.196 0.042 CHEMBL3544829

0.228 0.033 CHEMBL3544828

0.383 0.012 CHEMBL3544827

0.2 0.041 CHEMBL3544842

CHEMBL3544827
0.1320.0130.161Glycine receptor antagonist

0.161 0.005 CHEMBL3544786

0.111 0.024 CHEMBL1228

0.078 0.06 CHEMBL3544829

0.16 0.005 CHEMBL3544827

0.074 0.067 CHEMBL3544842

CHEMBL3544786
0.1620.0430.271DNA polymerase I inhibitor

0.271 0.014 CHEMBL3544786

0.188 0.032 CHEMBL1228

0.102 0.084 CHEMBL3544828

0.193 0.03 CHEMBL3544827

0.173 0.038 CHEMBL3544842

CHEMBL3544786
0.2070.0890.215RNA-directed DNA polymerase inhibitor

0.189 0.117 CHEMBL3544786

0.215 0.08 CHEMBL1228

0.205 0.092 CHEMBL3544829

0.202 0.097 CHEMBL3544828

0.179 0.134 CHEMBL3544827

CHEMBL1228
0.260.1430.26Calpain 2 inhibitor

0.203 0.185 CHEMBL1228

0.1220.0040.122Glutamate (mGluR7) antagonist

0.117 0.005 CHEMBL1228

0.079 0.028 CHEMBL3544829

0.075 0.034 CHEMBL3544828

0.250.1350.427Vasodilator, coronary

0.374 0.045 CHEMBL3544786

0.257 0.128 CHEMBL1228

0.242 0.142 CHEMBL3544829

0.244 0.141 CHEMBL3544828

0.427 0.028 CHEMBL3544827

0.192 0.19 CHEMBL3544842

CHEMBL3544827
0.1780.0630.214Phospholipase C inhibitor

0.173 0.069 CHEMBL3544786

0.214 0.036 CHEMBL1228

0.144 0.119 CHEMBL3544829

0.158 0.091 CHEMBL3544828

0.18 0.061 CHEMBL3544827

CHEMBL1228
0.1780.0660.391Peroxidase inhibitor

0.391 0.022 CHEMBL1228

0.203 0.058 CHEMBL3544829

0.36 0.027 CHEMBL3544828

CHEMBL1228
0.1390.0270.139GABA C receptor rho-1 antagonist

0.125 0.036 CHEMBL1228

0.113 0.046 CHEMBL3544829

0.096 0.068 CHEMBL3544828

0.1530.0430.223Cholesterol synthesis inhibitor

0.112 0.073 CHEMBL3544786

0.192 0.029 CHEMBL1228

0.195 0.028 CHEMBL3544829

0.223 0.022 CHEMBL3544828

0.14 0.05 CHEMBL3544827

CHEMBL3544828
0.1450.0370.329Xanthine oxidase inhibitor

0.14 0.038 CHEMBL3544786

0.227 0.015 CHEMBL1228

0.167 0.028 CHEMBL3544829

0.227 0.015 CHEMBL3544828

0.329 0.006 CHEMBL3544827

CHEMBL3544827
0.1370.0290.137Electron transport complex I inhibitor

0.129 0.036 CHEMBL1228

0.2240.1190.346Lipoxygenase inhibitor

0.346 0.052 CHEMBL1228

CHEMBL1228
0.160.0590.188CF transmembrane conductance regulator agonist

0.188 0.03 CHEMBL1228

0.142 0.091 CHEMBL3544828

0.136 0.104 CHEMBL3544827

CHEMBL1228
0.1160.0180.116Sphingosine 1-phosphate receptor 4 agonist

0.106 0.022 CHEMBL1228

0.06 0.054 CHEMBL3544829

0.1870.0890.187Histone acetyltransferase inhibitor

0.181 0.098 CHEMBL1228

0.1210.0230.126Interleukin 5 antagonist

0.09 0.054 CHEMBL3544786

0.126 0.02 CHEMBL1228

0.082 0.069 CHEMBL3544829

0.091 0.054 CHEMBL3544828

0.114 0.028 CHEMBL3544827

CHEMBL1228
0.1280.0320.142Anabolic

0.142 0.022 CHEMBL1228

0.105 0.056 CHEMBL3544829

0.114 0.046 CHEMBL3544828

CHEMBL1228
0.130.0340.13Sphingomyelinase inhibitor

0.084 0.081 CHEMBL3544786

0.112 0.047 CHEMBL1228

0.096 0.064 CHEMBL3544829

0.102 0.057 CHEMBL3544827

0.2460.1520.246Calcium channel activator

0.231 0.17 CHEMBL1228

0.222 0.183 CHEMBL3544829

0.213 0.194 CHEMBL3544828

0.1050.0140.105Vanilloid 4 agonist

0.082 0.036 CHEMBL1228

0.082 0.037 CHEMBL3544829

0.1910.10.336Cyclic AMP phosphodiesterase inhibitor

0.302 0.041 CHEMBL3544786

0.194 0.098 CHEMBL1228

0.282 0.049 CHEMBL3544829

0.282 0.049 CHEMBL3544828

0.336 0.029 CHEMBL3544827

0.156 0.142 CHEMBL3544842

CHEMBL3544827
0.1340.0450.134Falcipain 3 inhibitor

0.117 0.056 CHEMBL1228

0.1950.1070.55Aldehyde oxidase inhibitor

0.411 0.045 CHEMBL1228

0.381 0.05 CHEMBL3544829

0.55 0.026 CHEMBL3544828

CHEMBL3544828
0.1040.0180.115CC chemokine 5 receptor agonist

0.115 0.01 CHEMBL1228

0.077 0.076 CHEMBL3544829

0.085 0.048 CHEMBL3544828

CHEMBL1228
0.1490.0640.166Adenylate cyclase stimulant

0.129 0.103 CHEMBL3544786

0.166 0.04 CHEMBL1228

0.138 0.084 CHEMBL3544829

0.148 0.066 CHEMBL3544828

CHEMBL1228
0.1110.030.124Bile acid receptor antagonist

0.124 0.016 CHEMBL1228

0.095 0.06 CHEMBL3544829

0.104 0.042 CHEMBL3544828

0.089 0.075 CHEMBL3544827

CHEMBL1228
0.1010.020.103Glycine receptor agonist

0.103 0.019 CHEMBL3544786

0.098 0.022 CHEMBL1228

0.067 0.06 CHEMBL3544829

0.086 0.032 CHEMBL3544827

CHEMBL3544786
0.1380.0590.403Cyclooxygenase 3 inhibitor

0.256 0.008 CHEMBL3544786

0.158 0.042 CHEMBL1228

0.127 0.07 CHEMBL3544829

0.145 0.053 CHEMBL3544828

0.403 0.004 CHEMBL3544827

0.127 0.07 CHEMBL3544842

CHEMBL3544827
0.1620.0830.291ATPase inhibitor

0.228 0.02 CHEMBL3544786

0.167 0.074 CHEMBL1228

0.164 0.079 CHEMBL3544829

0.166 0.076 CHEMBL3544828

0.291 0.007 CHEMBL3544827

0.151 0.1 CHEMBL3544842

CHEMBL3544827
0.0840.0060.084Cholesterol esterase inhibitor

0.072 0.009 CHEMBL1228

0.053 0.025 CHEMBL3544829

0.048 0.033 CHEMBL3544828

0.1990.1210.199Neuropeptide Y2 antagonist

0.198 0.122 CHEMBL1228

0.185 0.149 CHEMBL3544829

0.188 0.143 CHEMBL3544828

0.0970.0220.097Acetylcholine M5 receptor agonist
0.1370.0620.19Toll-Like receptor 2 antagonist

0.19 0.028 CHEMBL1228

0.133 0.065 CHEMBL3544829

0.173 0.038 CHEMBL3544828

CHEMBL1228
0.090.0160.194Prostaglandin F2 alpha antagonist

0.086 0.018 CHEMBL1228

0.194 0.004 CHEMBL3544829

0.16 0.004 CHEMBL3544828

0.066 0.037 CHEMBL3544827

0.073 0.029 CHEMBL3544842

CHEMBL3544829
0.1330.060.149Vanilloid 1 agonist

0.123 0.081 CHEMBL3544786

0.149 0.039 CHEMBL1228

0.136 0.056 CHEMBL3544827

CHEMBL1228
0.1360.0640.307Alpha-N-acetylglucosaminidase inhibitor

0.307 0.015 CHEMBL3544786

0.105 0.094 CHEMBL1228

0.246 0.024 CHEMBL3544829

0.158 0.05 CHEMBL3544828

0.187 0.038 CHEMBL3544827

0.225 0.028 CHEMBL3544842

CHEMBL3544786
0.1390.0680.139Nav1.6 sodium channel blocker
0.1530.0850.185Growth hormone agonist

0.185 0.065 CHEMBL1228

0.129 0.109 CHEMBL3544829

0.149 0.088 CHEMBL3544828

CHEMBL1228
0.0980.030.115Interferon agonist

0.106 0.024 CHEMBL3544786

0.085 0.044 CHEMBL1228

0.076 0.058 CHEMBL3544829

0.115 0.019 CHEMBL3544827

CHEMBL3544827
0.1510.0840.168Sigma receptor agonist

0.168 0.074 CHEMBL1228

CHEMBL1228
0.1910.1260.519Immunostimulant

0.479 0.032 CHEMBL3544786

0.23 0.105 CHEMBL1228

0.266 0.09 CHEMBL3544829

0.283 0.084 CHEMBL3544828

0.519 0.027 CHEMBL3544827

0.354 0.063 CHEMBL3544842

CHEMBL3544827
0.1140.0490.125Adenylate kinase inhibitor

0.103 0.063 CHEMBL3544786

0.099 0.069 CHEMBL1228

0.125 0.039 CHEMBL3544829

0.098 0.071 CHEMBL3544828

CHEMBL3544829
0.0780.0130.078Oleamide hydrolase inhibitor

0.059 0.021 CHEMBL1228

0.0730.0080.094Nicotinic acid receptor agonist

0.094 0.005 CHEMBL1228

CHEMBL1228
0.0780.0180.078Corticotropin releasing factor 2 receptor antagonist
0.0810.0230.093Interferon inducer

0.088 0.018 CHEMBL3544786

0.07 0.035 CHEMBL1228

0.063 0.047 CHEMBL3544829

0.093 0.015 CHEMBL3544827

CHEMBL3544827
0.1860.1280.219DNA damaging

0.178 0.136 CHEMBL3544786

0.194 0.121 CHEMBL1228

0.219 0.101 CHEMBL3544827

CHEMBL3544827
0.0850.0280.085Phospholipase D inhibitor

0.066 0.063 CHEMBL1228

0.1330.0770.133Neurotrophic factor

0.129 0.082 CHEMBL1228

0.121 0.093 CHEMBL3544827

0.1810.1260.233Nitric-oxide synthase stimulant

0.185 0.118 CHEMBL3544786

0.193 0.101 CHEMBL1228

0.223 0.057 CHEMBL3544829

0.233 0.045 CHEMBL3544828

0.189 0.109 CHEMBL3544827

0.223 0.056 CHEMBL3544842

CHEMBL3544828
0.1750.1210.1755 Hydroxytryptamine 3E antagonist
0.1010.0470.259Triose-phosphate isomerase inhibitor

0.259 0.006 CHEMBL3544786

0.092 0.057 CHEMBL1228

0.134 0.025 CHEMBL3544829

0.106 0.042 CHEMBL3544828

0.172 0.015 CHEMBL3544827

0.162 0.017 CHEMBL3544842

CHEMBL3544786
0.1030.0510.103Lanosterol 14 alpha demethylase inhibitor

0.096 0.061 CHEMBL1228

0.0720.0220.079Sphingosine kinase inhibitor

0.079 0.017 CHEMBL1228

0.062 0.036 CHEMBL3544829

0.062 0.036 CHEMBL3544828

CHEMBL1228
0.0770.0280.077Glutamate (mGluR6) antagonist

0.067 0.047 CHEMBL1228

0.062 0.061 CHEMBL3544829

0.1020.0530.102Antihistaminic
0.0750.0270.075Cathepsin L inhibitor

0.06 0.039 CHEMBL1228

0.1080.060.129Aminopeptidase B inhibitor

0.106 0.061 CHEMBL1228

0.129 0.048 CHEMBL3544829

0.11 0.058 CHEMBL3544828

CHEMBL3544829
0.0720.0260.075Acyl-CoA dehydrogenase inhibitor

0.048 0.045 CHEMBL1228

0.075 0.024 CHEMBL3544829

CHEMBL3544829
0.0610.0140.061Histamine H2 receptor agonist
0.0710.0250.086Fatty acid synthase inhibitor

0.086 0.016 CHEMBL1228

CHEMBL1228
0.0590.0140.079Cytokine production stimulant

0.079 0.005 CHEMBL3544786

0.047 0.037 CHEMBL1228

0.045 0.043 CHEMBL3544829

0.062 0.011 CHEMBL3544827

CHEMBL3544786
0.0520.0070.067Prostaglandin D2 agonist

0.047 0.009 CHEMBL1228

0.067 0.004 CHEMBL3544829

0.059 0.005 CHEMBL3544828

0.036 0.016 CHEMBL3544827

CHEMBL3544829
0.1620.1170.215Insulin sensitizer

0.184 0.091 CHEMBL1228

0.209 0.065 CHEMBL3544829

0.215 0.059 CHEMBL3544828

0.177 0.098 CHEMBL3544827

CHEMBL3544828
0.110.0660.2Cystathionine beta-synthase inhibitor

0.097 0.08 CHEMBL3544786

0.2 0.024 CHEMBL1228

0.128 0.052 CHEMBL3544828

0.154 0.039 CHEMBL3544827

CHEMBL1228
0.0540.010.054Glutamate (mGluR3) antagonist

0.05 0.013 CHEMBL1228

0.039 0.022 CHEMBL3544829

0.0630.0190.064Immunoglobulin Fc receptor antagonist

0.058 0.03 CHEMBL1228

0.064 0.017 CHEMBL3544829

0.059 0.027 CHEMBL3544828

CHEMBL3544829
0.0520.010.052Delayed rectifier potassium channel blocker

0.044 0.017 CHEMBL1228

0.0460.0040.046Nicotinic acid receptor 2 antagonist

0.04 0.005 CHEMBL1228

0.1120.0730.112Anesthetic local

0.095 0.088 CHEMBL1228

0.103 0.08 CHEMBL3544829

0.0530.0140.053Angiotensin AT1 receptor antagonist

0.039 0.035 CHEMBL1228

0.0430.0040.043Acid ceramidase inhibitor

0.029 0.011 CHEMBL1228

0.0690.0310.069Argininosuccinate synthase inhibitor

0.057 0.039 CHEMBL3544786

0.056 0.04 CHEMBL1228

0.0920.0530.092Histamine antagonist
0.1790.1420.22Superoxide dismutase inhibitor

0.22 0.098 CHEMBL1228

0.172 0.152 CHEMBL3544828

CHEMBL1228
0.110.0740.117Sphingosine 1-phosphate receptor 2 agonist

0.107 0.082 CHEMBL1228

0.117 0.06 CHEMBL3544829

0.113 0.067 CHEMBL3544828

CHEMBL3544829
0.0510.0150.051Membrane dipeptidase inhibitor

0.038 0.03 CHEMBL1228

0.045 0.02 CHEMBL3544829

0.0790.0440.089Lipase inhibitor

0.089 0.034 CHEMBL1228

0.067 0.058 CHEMBL3544827

CHEMBL1228
0.0710.0360.086MDM2 inhibitor

0.086 0.014 CHEMBL3544829

0.071 0.037 CHEMBL3544828

CHEMBL3544829
0.0790.0440.079Adenosine A3 receptor antagonist

0.07 0.058 CHEMBL1228

0.1930.1590.30612-Lipoxygenase inhibitor

0.306 0.076 CHEMBL1228

CHEMBL1228
0.0580.0240.058Lysophosphatidic acid 3 receptor antagonist

0.049 0.038 CHEMBL1228

0.053 0.031 CHEMBL3544829

0.0640.0320.064Sphingosine 1-phosphate receptor 3 antagonist

0.064 0.033 CHEMBL1228

0.060.0290.064Leukotriene C antagonist

0.064 0.022 CHEMBL1228

CHEMBL1228
0.060.030.06Pregnane X receptor antagonist

0.057 0.037 CHEMBL1228

0.2210.190.34615-Lipoxygenase inhibitor

0.346 0.102 CHEMBL1228

CHEMBL1228
0.0480.0180.048Sphingosine kinase 1 inhibitor

0.048 0.018 CHEMBL1228

0.042 0.028 CHEMBL3544829

0.038 0.037 CHEMBL3544828

0.0650.0360.065Histone deacetylase SIRT3 inhibitor

0.059 0.054 CHEMBL1228

0.0470.0180.047Kainate receptor agonist

0.043 0.024 CHEMBL1228

0.04 0.032 CHEMBL3544829

0.0630.0340.063Phosphodiesterase 1A inhibitor
0.2460.2170.754Cyclophilin D inhibitor

0.634 0.022 CHEMBL3544786

0.291 0.17 CHEMBL1228

0.482 0.056 CHEMBL3544829

0.455 0.065 CHEMBL3544828

0.754 0.009 CHEMBL3544827

0.41 0.085 CHEMBL3544842

CHEMBL3544827
0.1070.0780.107Proteasome inhibitor

0.103 0.084 CHEMBL1228

0.0330.0070.053Vanilloid 2 agonist

0.043 0.004 CHEMBL3544786

0.032 0.008 CHEMBL1228

0.053 0.003 CHEMBL3544827

CHEMBL3544827
0.0760.050.092GABA B receptor agonist

0.092 0.024 CHEMBL1228

0.075 0.054 CHEMBL3544829

0.083 0.036 CHEMBL3544828

CHEMBL1228
0.040.0140.04Angiotensin II receptor antagonist
0.0520.0260.057Aldosterone antagonist

0.057 0.022 CHEMBL3544829

CHEMBL3544829
0.030.0040.045Nicotinic acid receptor 1 antagonist

0.045 0.003 CHEMBL1228

0.021 0.008 CHEMBL3544828

CHEMBL1228
0.0380.0130.038Calcium-independent phospholipase A2 inhibitor

0.036 0.019 CHEMBL1228

0.0590.0330.065Sphingosine kinase 2 inhibitor

0.065 0.026 CHEMBL1228

CHEMBL1228
0.0390.0130.039Adenosine uptake inhibitor
0.0720.0460.072Amidase inhibitor

0.069 0.05 CHEMBL1228

0.0930.0680.141Phosphodiesterase 6D inhibitor

0.119 0.026 CHEMBL3544786

0.098 0.057 CHEMBL1228

0.12 0.025 CHEMBL3544829

0.125 0.021 CHEMBL3544828

0.141 0.013 CHEMBL3544827

0.133 0.016 CHEMBL3544842

CHEMBL3544827
0.0830.0580.108Estrogen-related receptor beta agonist

0.108 0.017 CHEMBL1228

0.09 0.041 CHEMBL3544828

CHEMBL1228
0.1330.1090.317Melanin inhibitor

0.23 0.032 CHEMBL3544786

0.179 0.052 CHEMBL1228

0.14 0.097 CHEMBL3544829

0.175 0.055 CHEMBL3544828

0.317 0.02 CHEMBL3544827

0.181 0.051 CHEMBL3544842

CHEMBL3544827
0.0690.0450.071Exportin-1 inhibitor

0.071 0.041 CHEMBL3544829

CHEMBL3544829
0.0550.0330.055Nicotinic alpha3beta2 receptor antagonist
0.0320.010.032Hedgehog signaling activator

0.03 0.013 CHEMBL1228

0.0540.0320.086Aconitate hydratase inhibitor

0.086 0.012 CHEMBL3544829

0.056 0.03 CHEMBL3544828

CHEMBL3544829
0.0750.0550.112Na+ K+ transporting ATPase inhibitor

0.112 0.021 CHEMBL3544786

0.081 0.05 CHEMBL1228

0.112 0.022 CHEMBL3544827

0.096 0.035 CHEMBL3544842

CHEMBL3544827
0.0290.0090.044Prostaglandin F2 alpha agonist

0.034 0.007 CHEMBL1228

0.043 0.005 CHEMBL3544829

0.044 0.005 CHEMBL3544828

CHEMBL3544828
0.0370.0170.037Melatonin receptor 1A agonist
0.0840.0650.084Granulocyte macrophage colony stimulating factor agonist

0.082 0.069 CHEMBL1228

0.0640.0450.064Protease 3C (Human rhinovirus) inhibitor
0.030.0110.03Lysophosphatidic acid receptor 1 agonist

0.028 0.013 CHEMBL3544829

0.0980.0790.0985 Hydroxytryptamine 3A agonist
0.1270.1090.127Pregnane X receptor agonist
0.0350.0170.035Peptide deformylase inhibitor
0.0520.0350.0525 Hydroxytryptamine 4 antagonist
0.0370.0210.037Glutamate (mGluR8) antagonist

0.036 0.024 CHEMBL1228

0.034 0.03 CHEMBL3544827

0.0340.0180.094Prostaglandin agonist

0.035 0.017 CHEMBL1228

0.094 0.005 CHEMBL3544829

0.082 0.006 CHEMBL3544828

CHEMBL3544829
0.0270.0130.053Prostaglandin EP2 agonist

0.027 0.014 CHEMBL1228

0.053 0.005 CHEMBL3544829

0.046 0.007 CHEMBL3544828

CHEMBL3544829
0.0790.0650.079Ca(v)3.1 blocker

0.076 0.073 CHEMBL1228

0.1040.0910.149Aldehyde dehydrogenase inhibitor

0.149 0.048 CHEMBL1228

0.104 0.09 CHEMBL3544829

0.135 0.057 CHEMBL3544828

0.12 0.071 CHEMBL3544827

CHEMBL1228
0.0470.0340.084Glucose-6-phosphate isomerase inhibitor

0.084 0.008 CHEMBL3544786

0.044 0.042 CHEMBL1228

0.057 0.021 CHEMBL3544829

0.047 0.034 CHEMBL3544828

0.064 0.016 CHEMBL3544827

0.077 0.009 CHEMBL3544842

CHEMBL3544786
0.0880.0760.269UDP-glucose 4-epimerase inhibitor

0.269 0.012 CHEMBL3544786

0.091 0.072 CHEMBL1228

0.124 0.041 CHEMBL3544829

0.115 0.047 CHEMBL3544828

0.196 0.019 CHEMBL3544827

0.199 0.018 CHEMBL3544842

CHEMBL3544786
0.0920.0790.092Glutamate (mGluR7) agonist
0.070.0580.07Acetylcholine M4 receptor antagonist
0.0430.0320.043Histamine H1 receptor agonist
0.0390.0270.041Leukotriene C4 antagonist

0.041 0.022 CHEMBL1228

CHEMBL1228
0.0340.0230.034Free fatty acid receptor 1 antagonist
0.0680.0560.068Cathepsin G inhibitor

0.068 0.057 CHEMBL1228

0.0290.0180.029Purinergic P2Y15 antagonist
0.0280.0170.028Glucosylceramidase stimulant
0.0680.0570.088Porphobilinogen synthase inhibitor

0.088 0.042 CHEMBL1228

CHEMBL1228
0.0430.0320.043Glutamate (mGluR group III) antagonist
0.0580.0480.075Enoyl-[acyl-carrier-protein] reductase inhibitor

0.075 0.023 CHEMBL1228

CHEMBL1228
0.0480.0380.048Cannabinoid CB2 receptor antagonist
0.080.070.0863C-Like protease (SARS coronavirus) inhibitor

0.086 0.054 CHEMBL3544829

0.082 0.062 CHEMBL3544828

CHEMBL3544829
0.0670.0580.099Aminopeptidase I inhibitor

0.099 0.028 CHEMBL3544829

0.083 0.039 CHEMBL3544828

CHEMBL3544829
0.0170.0080.017Thromboxane A2 agonist

0.015 0.011 CHEMBL3544829

0.0310.0230.044ATP citrate lysase inhibitor

0.044 0.01 CHEMBL1228

0.029 0.028 CHEMBL3544829

0.034 0.018 CHEMBL3544828

CHEMBL1228
0.0670.0580.102Catalase inhibitor

0.102 0.038 CHEMBL3544829

0.07 0.054 CHEMBL3544828

CHEMBL3544829
0.0220.0140.022Angiotensin AT1A receptor antagonist
0.1890.1810.606Transcription factor NF kappa B inhibitor

0.482 0.047 CHEMBL3544786

0.281 0.106 CHEMBL1228

0.242 0.133 CHEMBL3544828

0.606 0.03 CHEMBL3544827

CHEMBL3544827
0.0210.0140.029Neuraminidase (Influenza B) inhibitor

0.02 0.016 CHEMBL1228

0.029 0.005 CHEMBL3544829

0.025 0.008 CHEMBL3544828

CHEMBL3544829
0.0390.0320.053Oxytocin agonist

0.053 0.022 CHEMBL1228

CHEMBL1228
0.1230.1160.127Neuropeptide Y1 antagonist

0.127 0.106 CHEMBL1228

CHEMBL1228
0.0350.0290.035Melanocortin 1 antagonist
0.0610.0550.202Phosphofructokinase-1 inhibitor

0.202 0.011 CHEMBL3544786

0.06 0.056 CHEMBL1228

0.09 0.036 CHEMBL3544829

0.073 0.046 CHEMBL3544828

0.138 0.02 CHEMBL3544827

0.142 0.02 CHEMBL3544842

CHEMBL3544786
0.0330.0270.033Kainate receptor 2 antagonist
0.050.0440.0853(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.085 0.014 CHEMBL1228

0.056 0.034 CHEMBL3544829

0.083 0.015 CHEMBL3544828

CHEMBL1228
0.0290.0230.029Acetylcholine M4 receptor agonist
0.0470.0420.047Prolyl endopeptidase inhibitor
0.1170.1120.117Acetylcholine M1 receptor antagonist

0.116 0.115 CHEMBL1228

0.0610.0560.068Calcium channel P-type blocker

0.068 0.032 CHEMBL3544829

CHEMBL3544829
0.0510.0470.051Glucosylceramidase inhibitor
0.0570.0540.087Dopamine D1 antagonist

0.087 0.03 CHEMBL1228

CHEMBL1228
0.0110.0070.013Thromboxane agonist

0.013 0.006 CHEMBL3544829

CHEMBL3544829
0.0330.0290.039Nicotinic acid receptor 2 agonist

0.039 0.021 CHEMBL1228

CHEMBL1228
0.0530.050.053Cannabinoid CB1 receptor agonist
0.0370.0330.037AMPA 4 receptor antagonist
0.1060.1030.142NADPH oxidase inhibitor

0.142 0.06 CHEMBL1228

CHEMBL1228
0.0810.0780.133Alcohol dehydrogenase inhibitor

0.112 0.041 CHEMBL1228

0.11 0.042 CHEMBL3544829

0.133 0.027 CHEMBL3544828

0.086 0.07 CHEMBL3544827

CHEMBL3544828
0.0210.0190.057Prostaglandin E2 agonist

0.022 0.017 CHEMBL1228

0.057 0.005 CHEMBL3544829

0.047 0.006 CHEMBL3544828

CHEMBL3544829
0.0120.0110.012Lysophosphatidic acid receptor 3 agonist
0.0690.0670.069Potassium channel (Tandem pore domain) blocker
0.0520.0510.052Carbonic anhydrase stimulant
0.0250.0230.037Toll-Like receptor 4 agonist

0.037 0.006 CHEMBL3544786

0.036 0.006 CHEMBL3544827

0.028 0.015 CHEMBL3544842

CHEMBL3544786
0.1160.1140.158Farnesoid X receptor antagonist

0.158 0.044 CHEMBL1228

0.122 0.098 CHEMBL3544828

CHEMBL1228
0.0180.0170.018Angiotensin AT2 receptor antagonist
0.050.0490.05Thromboxane synthase inhibitor
0.0240.0230.024Complement factor 1s inhibitor
0.040.040.063Adenosine deaminase inhibitor

0.046 0.034 CHEMBL3544786

0.063 0.018 CHEMBL3544829

0.054 0.026 CHEMBL3544828

CHEMBL3544829
0.1190.1180.119Death-associated protein kinase 1 inhibitor
0.0510.0520.083Biliverdin reductase inhibitor

0.083 0.025 CHEMBL3544829

CHEMBL3544829
0.1690.170.336DNA synthesis inhibitor

0.336 0.033 CHEMBL3544786

0.181 0.152 CHEMBL1228

0.189 0.14 CHEMBL3544829

0.181 0.151 CHEMBL3544828

0.319 0.038 CHEMBL3544827

0.222 0.092 CHEMBL3544842

CHEMBL3544786
0.0730.0750.078Ornithine decarboxylase inhibitor

0.078 0.069 CHEMBL1228

CHEMBL1228
0.0660.070.082GABA aminotransferase inhibitor

0.069 0.063 CHEMBL3544786

0.082 0.044 CHEMBL1228

0.07 0.061 CHEMBL3544827

CHEMBL1228
0.0460.050.105Alcohol oxidase inhibitor

0.083 0.023 CHEMBL1228

0.074 0.027 CHEMBL3544829

0.105 0.017 CHEMBL3544828

CHEMBL3544828
0.0470.0510.099Alpha-mannosidase inhibitor

0.099 0.006 CHEMBL3544786

0.056 0.032 CHEMBL3544829

0.096 0.007 CHEMBL3544827

0.085 0.009 CHEMBL3544842

CHEMBL3544786
0.0720.0760.099Androgen antagonist

0.093 0.052 CHEMBL1228

0.085 0.06 CHEMBL3544829

0.099 0.047 CHEMBL3544828

CHEMBL3544828
0.0670.0720.137Macrophage migration inhibitory factor inhibitor

0.137 0.019 CHEMBL1228

0.069 0.068 CHEMBL3544828

CHEMBL1228
0.050.0550.084Carbamoyl phosphate synthetase inhibitor

0.084 0.026 CHEMBL3544829

0.059 0.044 CHEMBL3544828

CHEMBL3544829
0.0630.070.08CDC25A inhibitor

0.08 0.044 CHEMBL1228

CHEMBL1228
0.0670.0750.108Estrogen receptor alpha antagonist

0.108 0.023 CHEMBL1228

CHEMBL1228
0.0540.0610.057Ryanodine receptor antagonist

0.057 0.046 CHEMBL1228

CHEMBL1228
0.1480.1560.18Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.18 0.093 CHEMBL1228

CHEMBL1228
0.0720.0810.084Myeloperoxidase inhibitor

0.084 0.06 CHEMBL1228

CHEMBL1228
0.0080.0190.035Prostaglandin EP4 agonist

0.035 0.006 CHEMBL3544829

0.017 0.009 CHEMBL3544828

CHEMBL3544829
0.1270.1390.14Heat shock protein 70 antagonist

0.129 0.128 CHEMBL3544786

0.137 0.089 CHEMBL1228

0.14 0.074 CHEMBL3544827

CHEMBL3544827
0.0210.0340.099Sodium/glucose cotransporter inhibitor

0.073 0.004 CHEMBL3544786

0.024 0.022 CHEMBL1228

0.024 0.022 CHEMBL3544828

0.099 0.003 CHEMBL3544827

0.04 0.007 CHEMBL3544842

CHEMBL3544827
0.0150.0280.018Methylmalonyl-CoA mutase inhibitor

0.018 0.014 CHEMBL3544829

CHEMBL3544829
0.0310.0450.054Dopamine D5 agonist

0.054 0.015 CHEMBL1228

CHEMBL1228
0.0240.0380.054Arginase inhibitor

0.036 0.025 CHEMBL3544786

0.054 0.013 CHEMBL3544827

CHEMBL3544827
0.020.0350.03Thyroid hormone agonist

0.03 0.013 CHEMBL1228

CHEMBL1228
0.0240.040.045Fumarate hydratase inhibitor

0.045 0.016 CHEMBL3544829

CHEMBL3544829
0.1070.1230.134Papain-like protease (SARS coronavirus) inhibitor

0.134 0.053 CHEMBL1228

0.111 0.107 CHEMBL3544829

0.133 0.055 CHEMBL3544828

CHEMBL1228
0.010.0260.043Ileal bile acid transport inhibitor

0.028 0.005 CHEMBL3544786

0.043 0.004 CHEMBL3544827

CHEMBL3544827
0.0590.0760.091Glutamate dehydrogenase inhibitor

0.091 0.036 CHEMBL3544829

0.072 0.053 CHEMBL3544828

CHEMBL3544829
0.0180.0350.025Prostaglandin EP4 antagonist

0.025 0.019 CHEMBL3544829

CHEMBL3544829
0.1460.1630.337Vasodilator

0.29 0.052 CHEMBL3544786

0.186 0.116 CHEMBL1228

0.24 0.075 CHEMBL3544829

0.254 0.067 CHEMBL3544828

0.337 0.037 CHEMBL3544827

0.27 0.059 CHEMBL3544842

CHEMBL3544827
0.0340.0520.1Mannosidase inhibitor

0.1 0.006 CHEMBL3544786

0.042 0.036 CHEMBL3544829

0.097 0.006 CHEMBL3544827

0.072 0.011 CHEMBL3544842

CHEMBL3544786
0.0090.0270.025Prostacyclin agonist

0.025 0.007 CHEMBL3544829

0.019 0.009 CHEMBL3544828

CHEMBL3544829
0.0230.0430.04Estradiol 17 beta-dehydrogenase 3 inhibitor

0.04 0.016 CHEMBL1228

CHEMBL1228
0.0160.0380.02Thymidine kinase (Herpes simplex virus 2) inhibitor

0.02 0.017 CHEMBL3544829

CHEMBL3544829
0.0240.0470.036Farnesoid X receptor agonist

0.036 0.028 CHEMBL3544829

CHEMBL3544829
0.0720.0960.155NADH dehydrogenase inhibitor

0.155 0.016 CHEMBL3544786

0.096 0.049 CHEMBL3544829

0.086 0.063 CHEMBL3544828

0.119 0.029 CHEMBL3544827

0.124 0.027 CHEMBL3544842

CHEMBL3544786
0.0410.0660.07Leukotriene B4 antagonist

0.051 0.043 CHEMBL3544786

0.051 0.043 CHEMBL1228

0.07 0.02 CHEMBL3544827

CHEMBL3544827
0.1310.160.151Death-associated protein kinase 2 inhibitor

0.151 0.105 CHEMBL1228

CHEMBL1228
0.0410.0710.07Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.058 0.037 CHEMBL3544786

0.062 0.032 CHEMBL3544829

0.07 0.026 CHEMBL3544842

CHEMBL3544842
0.0430.0740.057NMDA 2C receptor antagonist

0.057 0.05 CHEMBL1228

CHEMBL1228
0.0860.1180.116Microtubule formation inhibitor

0.116 0.066 CHEMBL3544786

0.105 0.082 CHEMBL3544829

0.097 0.096 CHEMBL3544828

0.116 0.066 CHEMBL3544827

CHEMBL3544827
0.0110.0420.02Telomerase stimulant

0.02 0.008 CHEMBL3544786

0.016 0.015 CHEMBL3544842

CHEMBL3544786
0.0460.0780.057Leukotriene antagonist

0.057 0.056 CHEMBL1228

CHEMBL1228
0.0840.1160.117DOPA decarboxylase inhibitor

0.117 0.049 CHEMBL1228

0.095 0.086 CHEMBL3544828

CHEMBL1228
0.0520.0860.094Glutamate decarboxylase inhibitor

0.075 0.049 CHEMBL1228

0.079 0.045 CHEMBL3544829

0.094 0.033 CHEMBL3544828

CHEMBL3544828
0.0520.0880.067Beta 3 adrenoreceptor antagonist

0.067 0.04 CHEMBL1228

0.066 0.04 CHEMBL3544828

CHEMBL1228
0.0160.0540.021Vitamin D receptor antagonist

0.021 0.017 CHEMBL3544829

0.021 0.018 CHEMBL3544828

CHEMBL3544828
0.0350.0750.17Prostaglandin EP2 antagonist

0.17 0.008 CHEMBL3544829

0.14 0.011 CHEMBL3544828

0.06 0.041 CHEMBL3544827

0.059 0.042 CHEMBL3544842

CHEMBL3544829
0.0220.0630.071HMG CoA reductase inhibitor

0.071 0.004 CHEMBL3544829

0.061 0.005 CHEMBL3544828

0.045 0.01 CHEMBL3544842

CHEMBL3544829
0.0890.1320.303Lipid peroxidase inhibitor

0.248 0.027 CHEMBL3544786

0.195 0.044 CHEMBL1228

0.159 0.062 CHEMBL3544829

0.22 0.034 CHEMBL3544828

0.303 0.018 CHEMBL3544827

0.174 0.053 CHEMBL3544842

CHEMBL3544827
0.0690.1130.086Vanilloid agonist

0.086 0.055 CHEMBL1228

CHEMBL1228
0.10.1460.13Mannose-6-phosphate isomerase inhibitor

0.13 0.086 CHEMBL3544786

0.121 0.1 CHEMBL3544829

0.115 0.109 CHEMBL3544842

CHEMBL3544786
0.0560.1030.067Peroxisome proliferator-activated receptor gamma antagonist

0.067 0.06 CHEMBL3544829

CHEMBL3544829
0.0180.0650.0311,3-Beta-glucan synthase inhibitor

0.03 0.015 CHEMBL3544786

0.031 0.014 CHEMBL3544827

CHEMBL3544827
0.0530.1020.084Somatostatin 1 agonist

0.077 0.055 CHEMBL1228

0.084 0.047 CHEMBL3544828

CHEMBL3544828
0.0680.1190.123Thioredoxin inhibitor

0.108 0.04 CHEMBL3544786

0.085 0.071 CHEMBL1228

0.123 0.029 CHEMBL3544827

CHEMBL3544827
0.0280.0790.077Prostaglandin antagonist

0.077 0.024 CHEMBL3544829

0.046 0.043 CHEMBL3544828

CHEMBL3544829
0.0250.0770.039NMDA receptor subunit 3B antagonist

0.039 0.037 CHEMBL1228

CHEMBL1228
0.0510.1060.062Beta 2 adrenoreceptor agonist

0.062 0.04 CHEMBL1228

0.061 0.047 CHEMBL3544828

CHEMBL1228
0.0320.0880.064Beta 1 adrenoreceptor antagonist

0.049 0.048 CHEMBL1228

0.051 0.045 CHEMBL3544829

0.064 0.032 CHEMBL3544828

CHEMBL3544828
0.0880.1440.159Interleukin 4 antagonist

0.159 0.042 CHEMBL3544786

0.159 0.042 CHEMBL1228

0.149 0.051 CHEMBL3544827

CHEMBL1228
0.0680.1240.106Carbonic anhydrase III inhibitor

0.106 0.056 CHEMBL1228

CHEMBL1228
0.2060.2640.378Calcium channel L-type activator

0.378 0.097 CHEMBL1228

0.266 0.188 CHEMBL3544829

0.37 0.103 CHEMBL3544828

CHEMBL1228
0.0540.1130.076Keratolytic

0.076 0.055 CHEMBL1228

CHEMBL1228
0.0360.0970.0573-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.053 0.049 CHEMBL3544786

0.057 0.043 CHEMBL1228

0.055 0.046 CHEMBL3544827

CHEMBL1228
0.040.1020.134Phenylalanine 4-hydroxylase inhibitor

0.066 0.05 CHEMBL1228

0.102 0.025 CHEMBL3544829

0.134 0.015 CHEMBL3544828

CHEMBL3544828
0.0370.10.048Vanilloid 2 antagonist

0.048 0.047 CHEMBL1228

CHEMBL1228
0.0390.1020.06Leukotriene synthesis inhibitor

0.06 0.055 CHEMBL1228

CHEMBL1228
0.0280.0920.046Beta 2 adrenoreceptor antagonist

0.046 0.042 CHEMBL1228

CHEMBL1228
0.0350.0990.109Heparanase inhibitor

0.091 0.004 CHEMBL3544786

0.109 0.004 CHEMBL3544827

CHEMBL3544827
0.1010.1660.371Hemostatic

0.185 0.039 CHEMBL3544786

0.371 0.01 CHEMBL3544827

CHEMBL3544827
0.0260.0940.151Neuraminidase (Influenza A) inhibitor

0.055 0.018 CHEMBL3544786

0.049 0.026 CHEMBL3544829

0.046 0.03 CHEMBL3544828

0.057 0.015 CHEMBL3544827

0.151 0.003 CHEMBL3544842

CHEMBL3544842
0.2010.2720.553Apoptosis agonist

0.553 0.06 CHEMBL3544786

0.322 0.157 CHEMBL1228

0.293 0.177 CHEMBL3544828

0.546 0.061 CHEMBL3544827

0.432 0.099 CHEMBL3544842

CHEMBL3544786
0.050.1210.122Adrenaline agonist

0.087 0.049 CHEMBL1228

0.084 0.052 CHEMBL3544829

0.122 0.025 CHEMBL3544828

CHEMBL3544828
0.0690.1440.382Amylase inhibitor

0.3 0.018 CHEMBL3544786

0.134 0.073 CHEMBL1228

0.224 0.036 CHEMBL3544829

0.283 0.021 CHEMBL3544828

0.376 0.011 CHEMBL3544827

0.382 0.01 CHEMBL3544842

CHEMBL3544842
0.0080.0840.048Squalene synthetase inhibitor

0.048 0.015 CHEMBL3544786

0.038 0.019 CHEMBL3544827

CHEMBL3544786
0.0020.080.019Antibiotic Macrolide-like

0.019 0.007 CHEMBL3544786

0.017 0.008 CHEMBL3544842

CHEMBL3544786
0.1410.220.383Peptidyltransferase inhibitor

0.383 0.008 CHEMBL3544786

0.194 0.108 CHEMBL1228

0.228 0.068 CHEMBL3544829

0.236 0.061 CHEMBL3544828

0.378 0.009 CHEMBL3544827

0.344 0.013 CHEMBL3544842

CHEMBL3544786
0.0250.1060.163Protein 50S ribosomal subunit inhibitor

0.163 0.006 CHEMBL3544786

0.101 0.013 CHEMBL3544827

0.148 0.007 CHEMBL3544842

CHEMBL3544786
0.110.1910.366Hypolipemic

0.233 0.075 CHEMBL3544786

0.366 0.032 CHEMBL3544829

0.339 0.038 CHEMBL3544828

0.302 0.048 CHEMBL3544827

0.193 0.1 CHEMBL3544842

CHEMBL3544829
0.0630.1460.079D-Ala-D-Ala ligase inhibitor

0.079 0.07 CHEMBL1228

CHEMBL1228
0.0430.1260.077Lipocortins synthesis agonist

0.077 0.015 CHEMBL3544786

0.067 0.025 CHEMBL3544827

0.061 0.034 CHEMBL3544842

CHEMBL3544786
0.0580.1460.076MAP kinase kinase 7 inhibitor

0.076 0.058 CHEMBL1228

0.073 0.071 CHEMBL3544828

CHEMBL1228
0.0150.1040.036Estradiol 17 beta-dehydrogenase inhibitor

0.036 0.034 CHEMBL1228

CHEMBL1228
0.0670.1560.094Nav1.4 sodium channel blocker

0.094 0.085 CHEMBL1228

CHEMBL1228
0.0650.1590.094Mucolytic

0.093 0.088 CHEMBL3544786

0.094 0.087 CHEMBL3544828

CHEMBL3544828
0.0090.1050.071Sodium/glucose cotransporter 2 inhibitor

0.05 0.006 CHEMBL3544786

0.071 0.004 CHEMBL3544827

0.027 0.017 CHEMBL3544842

CHEMBL3544827
0.0070.1070.033Prostaglandin EP3 antagonist

0.033 0.019 CHEMBL3544829

CHEMBL3544829
0.0940.1940.208DNA methyltransferase I inhibitor

0.208 0.065 CHEMBL3544827

CHEMBL3544827
0.0090.1120.022Antibiotic Anthracycline-like

0.022 0.007 CHEMBL3544786

0.019 0.014 CHEMBL3544827

0.019 0.014 CHEMBL3544842

CHEMBL3544786
0.0350.1390.067Beta adrenoreceptor antagonist

0.067 0.043 CHEMBL3544828

CHEMBL3544828
0.0490.1550.158Mediator release inhibitor

0.11 0.059 CHEMBL3544786

0.158 0.025 CHEMBL3544827

CHEMBL3544827
0.080.1860.66Angiogenesis stimulant

0.628 0.005 CHEMBL3544786

0.176 0.107 CHEMBL1228

0.151 0.122 CHEMBL3544828

0.66 0.005 CHEMBL3544827

0.388 0.024 CHEMBL3544842

CHEMBL3544827
0.0410.1540.25Monophenol monooxygenase inhibitor

0.185 0.037 CHEMBL3544786

0.108 0.07 CHEMBL1228

0.118 0.063 CHEMBL3544828

0.25 0.024 CHEMBL3544827

CHEMBL3544827
0.060.1750.184Alkylator

0.184 0.031 CHEMBL3544786

0.147 0.048 CHEMBL3544827

0.119 0.069 CHEMBL3544842

CHEMBL3544786
0.1030.220.52Free radical scavenger

0.41 0.027 CHEMBL3544786

0.275 0.059 CHEMBL1228

0.26 0.064 CHEMBL3544828

0.52 0.014 CHEMBL3544827

0.238 0.074 CHEMBL3544842

CHEMBL3544827
0.0870.2080.382Platelet adhesion inhibitor

0.333 0.024 CHEMBL3544786

0.382 0.014 CHEMBL3544827

CHEMBL3544827
0.0440.1710.1035-Lipoxygenase inhibitor

0.103 0.062 CHEMBL1228

CHEMBL1228
0.0280.1560.045Beta adrenoreceptor agonist

0.045 0.033 CHEMBL3544828

CHEMBL3544828
0.0370.1690.075NMDA receptor antagonist

0.075 0.071 CHEMBL3544828

CHEMBL3544828
0.1410.2740.496Alpha-glucosidase inhibitor

0.244 0.191 CHEMBL1228

0.264 0.179 CHEMBL3544828

0.496 0.082 CHEMBL3544827

CHEMBL3544827
0.0550.1950.214AMP-activated protein kinase stimulant

0.17 0.018 CHEMBL3544786

0.214 0.009 CHEMBL3544827

CHEMBL3544827
0.0590.20.164Toll-Like receptor 4 antagonist

0.162 0.015 CHEMBL3544786

0.095 0.079 CHEMBL1228

0.164 0.014 CHEMBL3544827

0.143 0.025 CHEMBL3544842

CHEMBL3544827
0.0440.1890.201Expectorant

0.182 0.025 CHEMBL3544786

0.1 0.069 CHEMBL3544829

0.111 0.057 CHEMBL3544828

0.201 0.02 CHEMBL3544827

0.111 0.058 CHEMBL3544842

CHEMBL3544827
0.0630.2110.155Estrogen antagonist

0.155 0.021 CHEMBL1228

0.118 0.059 CHEMBL3544828

CHEMBL1228
0.0780.2260.2Hexokinase inhibitor

0.2 0.035 CHEMBL3544786

0.2 0.035 CHEMBL3544827

0.13 0.104 CHEMBL3544842

CHEMBL3544827
0.0830.2370.21DNA methylase inhibitor

0.21 0.073 CHEMBL3544827

CHEMBL3544827
0.0040.170.039Estrogen receptor alpha agonist

0.039 0.021 CHEMBL1228

CHEMBL1228
0.0490.2180.17Beta glucuronidase inhibitor

0.117 0.049 CHEMBL3544786

0.17 0.018 CHEMBL3544827

CHEMBL3544827
0.0750.2630.396Hepatoprotectant

0.375 0.016 CHEMBL3544786

0.186 0.075 CHEMBL3544829

0.204 0.063 CHEMBL3544828

0.396 0.014 CHEMBL3544827

0.306 0.028 CHEMBL3544842

CHEMBL3544827
0.130.3250.409Apoptosis antagonist

0.36 0.051 CHEMBL3544786

0.208 0.169 CHEMBL1228

0.213 0.163 CHEMBL3544828

0.409 0.036 CHEMBL3544827

0.278 0.102 CHEMBL3544842

CHEMBL3544827
0.020.2160.062Nitric oxide donor

0.062 0.044 CHEMBL3544827

CHEMBL3544827
0.0090.2070.048Protein 30S ribosomal subunit inhibitor

0.046 0.009 CHEMBL3544786

0.048 0.008 CHEMBL3544827

0.039 0.01 CHEMBL3544842

CHEMBL3544827
0.0040.2060.029Estrogen receptor beta agonist

0.029 0.024 CHEMBL1228

CHEMBL1228
0.0460.2530.308Thrombolytic

0.308 0.023 CHEMBL3544786

0.293 0.025 CHEMBL3544827

CHEMBL3544786
0.0170.2340.072Antibiotic Aminoglycoside-like

0.072 0.005 CHEMBL3544786

0.07 0.006 CHEMBL3544827

0.071 0.006 CHEMBL3544842

CHEMBL3544786
0.0410.2610.132Estrogen receptor beta antagonist

0.132 0.022 CHEMBL1228

0.102 0.06 CHEMBL3544828

CHEMBL1228
0.0670.2920.348Nitric oxide antagonist

0.307 0.039 CHEMBL3544786

0.13 0.119 CHEMBL1228

0.132 0.115 CHEMBL3544829

0.169 0.082 CHEMBL3544828

0.348 0.032 CHEMBL3544827

0.262 0.048 CHEMBL3544842

CHEMBL3544827
0.0070.2350.054Estrogen agonist

0.054 0.033 CHEMBL1228

CHEMBL1228
0.0780.310.552Antioxidant

0.481 0.022 CHEMBL3544786

0.24 0.089 CHEMBL1228

0.245 0.087 CHEMBL3544828

0.552 0.015 CHEMBL3544827

0.378 0.039 CHEMBL3544842

CHEMBL3544827
0.0120.2510.264Antineoplastic antibiotic

0.213 0.019 CHEMBL3544786

0.068 0.067 CHEMBL3544828

0.164 0.028 CHEMBL3544827

0.264 0.013 CHEMBL3544842

CHEMBL3544842
0.0660.3260.139DNA repair enzyme inhibitor

0.137 0.045 CHEMBL3544786

0.139 0.043 CHEMBL3544827

CHEMBL3544827
0.0110.2820.203Neuraminidase inhibitor

0.063 0.04 CHEMBL3544786

0.057 0.047 CHEMBL3544828

0.072 0.032 CHEMBL3544827

0.203 0.004 CHEMBL3544842

CHEMBL3544842
0.0160.2950.214Neuraminidase (influenza) inhibitor

0.071 0.033 CHEMBL3544786

0.063 0.046 CHEMBL3544828

0.078 0.027 CHEMBL3544827

0.214 0.004 CHEMBL3544842

CHEMBL3544842
0.0390.320.127Bone formation stimulant

0.127 0.079 CHEMBL3544786

0.108 0.098 CHEMBL3544828

CHEMBL3544786
0.0120.2980.334Selectin antagonist

0.316 0.005 CHEMBL3544786

0.334 0.004 CHEMBL3544827

0.259 0.008 CHEMBL3544842

CHEMBL3544827
0.0090.2990.041Macrophage elastase inhibitor

0.041 0.033 CHEMBL3544829

CHEMBL3544829
0.060.3550.244Insulin secretagoues

0.19 0.042 CHEMBL3544786

0.244 0.02 CHEMBL3544829

0.225 0.025 CHEMBL3544828

0.229 0.024 CHEMBL3544827

0.184 0.045 CHEMBL3544842

CHEMBL3544829
0.090.3920.213Antiobesity

0.213 0.194 CHEMBL3544827

CHEMBL3544827
0.0150.3340.094Protein-tyrosine phosphatase 1B inhibitor

0.094 0.084 CHEMBL3544827

CHEMBL3544827
0.040.3720.129Transcription factor NF kappa B stimulant

0.129 0.022 CHEMBL3544786

0.125 0.023 CHEMBL3544827

0.116 0.027 CHEMBL3544842

CHEMBL3544786
0.0180.3520.078Glucose-6-phosphate translocase inhibitor

0.072 0.015 CHEMBL3544786

0.078 0.012 CHEMBL3544827

CHEMBL3544827
0.0820.4270.808Immunomodulator

0.808 0.004 CHEMBL3544786

0.382 0.049 CHEMBL3544827

0.718 0.005 CHEMBL3544842

CHEMBL3544786
0.0230.3810.113ATPase (Vacuolar H+) inhibitor

0.097 0.044 CHEMBL3544786

0.113 0.025 CHEMBL3544827

0.103 0.036 CHEMBL3544842

CHEMBL3544827
0.0260.3840.063Adenine nucleotide translocase inhibitor

0.063 0.024 CHEMBL3544786

0.061 0.027 CHEMBL3544827

CHEMBL3544786
0.0520.4230.25NOS3 expression enhancer

0.211 0.037 CHEMBL3544786

0.25 0.026 CHEMBL3544827

0.151 0.071 CHEMBL3544842

CHEMBL3544827
0.0460.430.236Interleukin 6 antagonist

0.236 0.026 CHEMBL3544786

0.182 0.053 CHEMBL3544827

0.186 0.05 CHEMBL3544842

CHEMBL3544786
0.010.4140.031Estrogen-related receptor beta antagonist

0.031 0.026 CHEMBL1228

CHEMBL1228
0.0570.4890.576Hypoglycemic

0.486 0.016 CHEMBL3544786

0.2 0.112 CHEMBL3544829

0.245 0.08 CHEMBL3544828

0.576 0.009 CHEMBL3544827

0.333 0.042 CHEMBL3544842

CHEMBL3544827
0.0150.4620.179Topoisomerase I inhibitor

0.179 0.032 CHEMBL3544786

0.17 0.034 CHEMBL3544827

0.085 0.084 CHEMBL3544842

CHEMBL3544786
0.0170.4840.097Cell adhesion molecule inhibitor

0.095 0.038 CHEMBL3544786

0.097 0.037 CHEMBL3544827

CHEMBL3544827
0.0630.5850.23Caspase 3 stimulant

0.193 0.18 CHEMBL3544786

0.23 0.131 CHEMBL3544827

CHEMBL3544827
0.0220.5760.187Cell adhesion inhibitor

0.179 0.031 CHEMBL3544786

0.187 0.028 CHEMBL3544827

CHEMBL3544827
0.020.5890.201Interleukin antagonist

0.134 0.132 CHEMBL3544829

0.201 0.084 CHEMBL3544828

CHEMBL3544828
0.0140.6030.072Factor IXa inhibitor

0.072 0.019 CHEMBL3544786

0.068 0.021 CHEMBL3544827

CHEMBL3544786
0.0320.630.093Interleukin 12 antagonist

0.089 0.074 CHEMBL3544828

0.093 0.066 CHEMBL3544827

CHEMBL3544827
0.0230.6460.31Tumour necrosis factor alpha release inhibitor

0.203 0.107 CHEMBL3544786

0.31 0.05 CHEMBL3544827

0.155 0.152 CHEMBL3544842

CHEMBL3544827
0.0040.6480.31S-adenosyl-L-homocysteine hydrolase inhibitor

0.31 0.002 CHEMBL3544842

CHEMBL3544842
0.010.6580.094Topoisomerase II alpha inhibitor

0.09 0.046 CHEMBL3544786

0.094 0.043 CHEMBL3544827

CHEMBL3544827
0.0670.7270.141CC chemokine 6 receptor antagonist

0.141 0.038 CHEMBL3544786

0.135 0.055 CHEMBL3544827

CHEMBL3544786
0.0060.7790.143Topoisomerase II inhibitor

0.123 0.065 CHEMBL3544786

0.143 0.053 CHEMBL3544827

CHEMBL3544827
Ext Pa Pi Pmax Activity Other Results ID Pa_max