| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.663 | 0.005 | 0.774 | Anticonvulsant | 0.264 0.052 CHEMBL4525756 0.774 0.004 CHEMBL315985 0.774 0.004 CHEMBL313120 0.584 0.008 CHEMBL3526499 0.584 0.008 CHEMBL4525805 | CHEMBL313120 | |
| 0.451 | 0.041 | 0.451 | GABA C receptor rho-3 antagonist | 0.205 0.201 CHEMBL4525756 0.319 0.104 CHEMBL315985 0.319 0.104 CHEMBL313120 0.44 0.045 CHEMBL3526499 0.44 0.045 CHEMBL4525805 | ||
| 0.444 | 0.037 | 0.444 | 5 Hydroxytryptamine release stimulant | 0.289 0.073 CHEMBL4525757 0.403 0.045 CHEMBL315985 0.403 0.045 CHEMBL313120 0.439 0.038 CHEMBL3526872 0.407 0.044 CHEMBL3526499 0.407 0.044 CHEMBL4525805 0.439 0.038 CHEMBL3526693 | ||
| 0.409 | 0.005 | 0.409 | Interleukin 1 antagonist | 0.123 0.085 CHEMBL4525756 0.243 0.02 CHEMBL4525757 0.256 0.018 CHEMBL315985 0.256 0.018 CHEMBL313120 0.159 0.052 CHEMBL3526872 0.321 0.009 CHEMBL3526499 0.321 0.009 CHEMBL4525805 0.159 0.052 CHEMBL3526693 | ||
| 0.457 | 0.057 | 0.474 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.417 0.086 CHEMBL315985 0.417 0.086 CHEMBL313120 0.474 0.046 CHEMBL3526499 0.474 0.046 CHEMBL4525805 | CHEMBL4525805 | |
| 0.452 | 0.065 | 0.604 | Analgesic | 0.604 0.026 CHEMBL315985 0.604 0.026 CHEMBL313120 0.225 0.208 CHEMBL3526872 0.523 0.043 CHEMBL3526499 0.523 0.043 CHEMBL4525805 0.225 0.208 CHEMBL3526693 | CHEMBL313120 | |
| 0.396 | 0.017 | 0.528 | Anesthetic general | 0.455 0.011 CHEMBL4525757 0.485 0.009 CHEMBL315985 0.485 0.009 CHEMBL313120 0.511 0.007 CHEMBL3526872 0.528 0.006 CHEMBL3526499 0.528 0.006 CHEMBL4525805 0.511 0.007 CHEMBL3526693 | CHEMBL4525805 | |
| 0.41 | 0.074 | 0.41 | Calcium channel L-type activator | 0.257 0.197 CHEMBL4525757 0.257 0.197 CHEMBL3526499 0.257 0.197 CHEMBL4525805 | ||
| 0.35 | 0.019 | 0.578 | Non-steroidal antiinflammatory agent | 0.149 0.116 CHEMBL4525756 0.578 0.005 CHEMBL4525757 0.198 0.073 CHEMBL315985 0.198 0.073 CHEMBL313120 0.394 0.014 CHEMBL3526872 0.216 0.059 CHEMBL3526499 0.216 0.059 CHEMBL4525805 0.394 0.014 CHEMBL3526693 | CHEMBL4525757 | |
| 0.4 | 0.076 | 0.506 | Histamine release inhibitor | 0.287 0.131 CHEMBL4525756 0.506 0.027 CHEMBL4525757 0.216 0.185 CHEMBL315985 0.216 0.185 CHEMBL313120 0.486 0.034 CHEMBL3526872 0.25 0.155 CHEMBL3526499 0.25 0.155 CHEMBL4525805 0.486 0.034 CHEMBL3526693 | CHEMBL4525757 | |
| 0.427 | 0.123 | 0.812 | Antiinflammatory | 0.508 0.084 CHEMBL4525756 0.787 0.017 CHEMBL4525757 0.66 0.039 CHEMBL315985 0.66 0.039 CHEMBL313120 0.812 0.014 CHEMBL3526872 0.624 0.047 CHEMBL3526499 0.624 0.047 CHEMBL4525805 0.812 0.014 CHEMBL3526693 | CHEMBL3526693 | |
| 0.315 | 0.038 | 0.315 | 5 Hydroxytryptamine uptake stimulant | 0.256 0.075 CHEMBL315985 0.256 0.075 CHEMBL313120 0.295 0.048 CHEMBL3526499 0.295 0.048 CHEMBL4525805 | ||
| 0.295 | 0.036 | 0.295 | Tyrosine 3 hydroxylase inhibitor | 0.255 0.063 CHEMBL315985 0.255 0.063 CHEMBL313120 0.284 0.042 CHEMBL3526499 0.284 0.042 CHEMBL4525805 | ||
| 0.305 | 0.047 | 0.376 | Interleukin antagonist | 0.232 0.069 CHEMBL4525757 0.233 0.068 CHEMBL315985 0.233 0.068 CHEMBL313120 0.376 0.034 CHEMBL3526499 0.376 0.034 CHEMBL4525805 | CHEMBL4525805 | |
| 0.292 | 0.046 | 0.498 | DNA synthesis inhibitor | 0.199 0.125 CHEMBL4525756 0.498 0.014 CHEMBL4525757 0.291 0.047 CHEMBL315985 0.291 0.047 CHEMBL313120 0.489 0.014 CHEMBL3526872 0.336 0.033 CHEMBL3526499 0.336 0.033 CHEMBL4525805 0.489 0.014 CHEMBL3526693 | CHEMBL4525757 | |
| 0.321 | 0.083 | 0.684 | Angiogenesis inhibitor | 0.684 0.01 CHEMBL4525756 0.49 0.031 CHEMBL4525757 0.295 0.095 CHEMBL315985 0.295 0.095 CHEMBL313120 0.359 0.067 CHEMBL3526872 0.341 0.075 CHEMBL3526499 0.341 0.075 CHEMBL4525805 0.359 0.067 CHEMBL3526693 | CHEMBL4525756 | |
| 0.223 | 0.034 | 0.223 | 5 Hydroxytryptamine 3E antagonist | 0.171 0.131 CHEMBL3526499 0.171 0.131 CHEMBL4525805 | ||
| 0.238 | 0.05 | 0.389 | Peroxidase inhibitor | 0.254 0.046 CHEMBL4525756 0.216 0.055 CHEMBL315985 0.216 0.055 CHEMBL313120 0.389 0.022 CHEMBL3526499 0.389 0.022 CHEMBL4525805 | CHEMBL4525805 | |
| 0.253 | 0.076 | 0.279 | Gastrin inhibitor | 0.207 0.138 CHEMBL315985 0.207 0.138 CHEMBL313120 0.279 0.05 CHEMBL3526499 0.279 0.05 CHEMBL4525805 | CHEMBL4525805 | |
| 0.217 | 0.04 | 0.217 | Heat shock protein 90 alpha antagonist | |||
| 0.248 | 0.077 | 0.248 | 5 Hydroxytryptamine 1E antagonist | |||
| 0.191 | 0.023 | 0.191 | Butyrylcholinesterase inhibitor | 0.098 0.064 CHEMBL315985 0.098 0.064 CHEMBL313120 0.086 0.075 CHEMBL3526499 0.086 0.075 CHEMBL4525805 | ||
| 0.261 | 0.093 | 0.284 | Lipoxygenase inhibitor | 0.236 0.11 CHEMBL315985 0.236 0.11 CHEMBL313120 0.284 0.079 CHEMBL3526499 0.284 0.079 CHEMBL4525805 | CHEMBL4525805 | |
| 0.314 | 0.149 | 0.473 | 5 Hydroxytryptamine release inhibitor | 0.473 0.042 CHEMBL4525757 0.282 0.186 CHEMBL3526872 0.292 0.175 CHEMBL3526499 0.292 0.175 CHEMBL4525805 0.282 0.186 CHEMBL3526693 | CHEMBL4525757 | |
| 0.205 | 0.04 | 0.266 | Lipid peroxidase inhibitor | 0.266 0.024 CHEMBL4525757 0.111 0.104 CHEMBL315985 0.111 0.104 CHEMBL313120 0.232 0.031 CHEMBL3526872 0.135 0.079 CHEMBL3526499 0.135 0.079 CHEMBL4525805 0.232 0.031 CHEMBL3526693 | CHEMBL4525757 | |
| 0.17 | 0.017 | 0.17 | Creatine kinase inhibitor | 0.128 0.035 CHEMBL4525756 0.16 0.02 CHEMBL315985 0.16 0.02 CHEMBL313120 0.169 0.017 CHEMBL3526499 0.169 0.017 CHEMBL4525805 | ||
| 0.19 | 0.038 | 0.256 | Nav1.2 sodium channel blocker | 0.256 0.021 CHEMBL4525756 0.155 0.054 CHEMBL315985 0.155 0.054 CHEMBL313120 0.18 0.042 CHEMBL3526499 0.18 0.042 CHEMBL4525805 | CHEMBL4525756 | |
| 0.234 | 0.086 | 0.476 | Superoxide dismutase inhibitor | 0.476 0.015 CHEMBL4525756 0.225 0.093 CHEMBL315985 0.225 0.093 CHEMBL313120 0.297 0.051 CHEMBL3526499 0.297 0.051 CHEMBL4525805 | CHEMBL4525756 | |
| 0.244 | 0.098 | 0.572 | Immunostimulant | 0.347 0.065 CHEMBL4525756 0.549 0.023 CHEMBL4525757 0.328 0.071 CHEMBL315985 0.328 0.071 CHEMBL313120 0.572 0.02 CHEMBL3526872 0.316 0.074 CHEMBL3526499 0.316 0.074 CHEMBL4525805 0.572 0.02 CHEMBL3526693 | CHEMBL3526693 | |
| 0.318 | 0.175 | 0.347 | Caspase 9 stimulant | 0.347 0.148 CHEMBL4525757 0.263 0.238 CHEMBL315985 0.263 0.238 CHEMBL313120 0.319 0.174 CHEMBL3526872 0.297 0.197 CHEMBL3526499 0.297 0.197 CHEMBL4525805 0.319 0.174 CHEMBL3526693 | CHEMBL4525757 | |
| 0.215 | 0.084 | 0.215 | MAP kinase kinase 3 inhibitor | 0.192 0.146 CHEMBL315985 0.192 0.146 CHEMBL313120 0.213 0.088 CHEMBL3526499 0.213 0.088 CHEMBL4525805 | ||
| 0.206 | 0.077 | 0.251 | Platelet aggregation inhibitor | 0.251 0.051 CHEMBL4525757 0.155 0.123 CHEMBL315985 0.155 0.123 CHEMBL313120 0.182 0.095 CHEMBL3526499 0.182 0.095 CHEMBL4525805 | CHEMBL4525757 | |
| 0.164 | 0.035 | 0.164 | 5 Hydroxytryptamine 2B antagonist | |||
| 0.177 | 0.05 | 0.177 | Heat shock protein 90 antagonist | |||
| 0.175 | 0.05 | 0.175 | MAO inhibitor | |||
| 0.155 | 0.032 | 0.188 | GABA C receptor agonist | 0.156 0.032 CHEMBL315985 0.156 0.032 CHEMBL313120 0.188 0.023 CHEMBL3526499 0.188 0.023 CHEMBL4525805 | CHEMBL4525805 | |
| 0.259 | 0.137 | 0.28 | Calcium channel activator | 0.28 0.113 CHEMBL315985 0.28 0.113 CHEMBL313120 0.268 0.126 CHEMBL3526499 0.268 0.126 CHEMBL4525805 | CHEMBL313120 | |
| 0.17 | 0.051 | 0.17 | GABA C receptor rho-2 antagonist | 0.124 0.118 CHEMBL315985 0.124 0.118 CHEMBL313120 0.158 0.064 CHEMBL3526499 0.158 0.064 CHEMBL4525805 | ||
| 0.207 | 0.09 | 0.282 | RNA-directed DNA polymerase inhibitor | 0.282 0.036 CHEMBL4525756 0.192 0.112 CHEMBL4525757 0.21 0.085 CHEMBL315985 0.21 0.085 CHEMBL313120 0.2 0.099 CHEMBL3526872 0.248 0.05 CHEMBL3526499 0.248 0.05 CHEMBL4525805 0.2 0.099 CHEMBL3526693 | CHEMBL4525756 | |
| 0.161 | 0.047 | 0.161 | Sodium channel (voltage-gated) blocker | 0.122 0.082 CHEMBL4525756 0.109 0.098 CHEMBL3526499 0.109 0.098 CHEMBL4525805 | ||
| 0.129 | 0.018 | 0.129 | Glutamate decarboxylase inhibitor | 0.069 0.056 CHEMBL315985 0.069 0.056 CHEMBL313120 0.093 0.034 CHEMBL3526499 0.093 0.034 CHEMBL4525805 | ||
| 0.161 | 0.05 | 0.161 | Sodium channel blocker | 0.131 0.073 CHEMBL4525756 0.106 0.103 CHEMBL3526499 0.106 0.103 CHEMBL4525805 | ||
| 0.159 | 0.049 | 0.181 | NADPH oxidase inhibitor | 0.171 0.044 CHEMBL4525757 0.162 0.048 CHEMBL315985 0.162 0.048 CHEMBL313120 0.181 0.04 CHEMBL3526872 0.139 0.062 CHEMBL3526499 0.139 0.062 CHEMBL4525805 0.181 0.04 CHEMBL3526693 | CHEMBL3526693 | |
| 0.146 | 0.038 | 0.146 | GABA receptor agonist | |||
| 0.2 | 0.094 | 0.334 | Cyclic AMP phosphodiesterase inhibitor | 0.334 0.03 CHEMBL4525757 0.224 0.078 CHEMBL3526872 0.224 0.078 CHEMBL3526693 | CHEMBL4525757 | |
| 0.135 | 0.029 | 0.135 | GABA C receptor rho-1 antagonist | 0.11 0.05 CHEMBL315985 0.11 0.05 CHEMBL313120 0.131 0.031 CHEMBL3526499 0.131 0.031 CHEMBL4525805 | ||
| 0.144 | 0.039 | 0.144 | 5 Hydroxytryptamine 3A agonist | 0.093 0.085 CHEMBL3526499 0.093 0.085 CHEMBL4525805 | ||
| 0.113 | 0.014 | 0.113 | Acetylcholine M5 receptor agonist | |||
| 0.139 | 0.044 | 0.139 | MAO A inhibitor | |||
| 0.135 | 0.043 | 0.135 | MAO B inhibitor | |||
| 0.174 | 0.085 | 0.184 | P-glycoprotein inhibitor | 0.175 0.085 CHEMBL4525757 0.184 0.076 CHEMBL315985 0.184 0.076 CHEMBL313120 0.183 0.077 CHEMBL3526872 0.174 0.086 CHEMBL3526499 0.174 0.086 CHEMBL4525805 0.183 0.077 CHEMBL3526693 | CHEMBL313120 | |
| 0.098 | 0.016 | 0.478 | NMDA 2B receptor antagonist | 0.478 0.003 CHEMBL4525756 0.3 0.004 CHEMBL315985 0.3 0.004 CHEMBL313120 0.284 0.004 CHEMBL3526499 0.284 0.004 CHEMBL4525805 | CHEMBL4525756 | |
| 0.191 | 0.109 | 0.38 | Aldehyde oxidase inhibitor | 0.218 0.096 CHEMBL315985 0.218 0.096 CHEMBL313120 0.38 0.05 CHEMBL3526499 0.38 0.05 CHEMBL4525805 | CHEMBL4525805 | |
| 0.127 | 0.046 | 0.141 | GABA C receptor antagonist | 0.118 0.055 CHEMBL4525756 0.118 0.055 CHEMBL315985 0.118 0.055 CHEMBL313120 0.141 0.035 CHEMBL3526499 0.141 0.035 CHEMBL4525805 | CHEMBL4525805 | |
| 0.09 | 0.017 | 0.09 | Glutamate (mGluR7) antagonist | 0.068 0.045 CHEMBL315985 0.068 0.045 CHEMBL313120 0.088 0.019 CHEMBL3526499 0.088 0.019 CHEMBL4525805 | ||
| 0.112 | 0.04 | 0.114 | Glutamate (mGluR7) agonist | 0.114 0.037 CHEMBL315985 0.114 0.037 CHEMBL313120 0.112 0.04 CHEMBL3526499 0.112 0.04 CHEMBL4525805 | CHEMBL313120 | |
| 0.162 | 0.092 | 0.177 | Succinate dehydrogenase inhibitor | 0.149 0.115 CHEMBL315985 0.149 0.115 CHEMBL313120 0.177 0.071 CHEMBL3526499 0.177 0.071 CHEMBL4525805 | CHEMBL4525805 | |
| 0.091 | 0.02 | 0.091 | Aminopeptidase microsomal inhibitor | |||
| 0.109 | 0.041 | 0.109 | NMDA receptor antagonist | 0.095 0.05 CHEMBL4525756 0.078 0.068 CHEMBL315985 0.078 0.068 CHEMBL313120 | ||
| 0.078 | 0.01 | 0.093 | Ryanodine receptor antagonist | 0.076 0.011 CHEMBL315985 0.076 0.011 CHEMBL313120 0.093 0.005 CHEMBL3526499 0.093 0.005 CHEMBL4525805 | CHEMBL4525805 | |
| 0.108 | 0.041 | 0.108 | 5 Hydroxytryptamine 2C antagonist | |||
| 0.122 | 0.055 | 0.149 | Photosensitizer | 0.149 0.032 CHEMBL4525757 0.116 0.062 CHEMBL3526872 0.109 0.073 CHEMBL3526499 0.109 0.073 CHEMBL4525805 0.116 0.062 CHEMBL3526693 | CHEMBL4525757 | |
| 0.1 | 0.035 | 0.1 | Granulocyte macrophage colony stimulating factor agonist | 0.084 0.065 CHEMBL3526499 0.084 0.065 CHEMBL4525805 | ||
| 0.085 | 0.022 | 0.085 | 5 Hydroxytryptamine 3 antagonist | 0.075 0.026 CHEMBL315985 0.075 0.026 CHEMBL313120 0.055 0.042 CHEMBL3526499 0.055 0.042 CHEMBL4525805 | ||
| 0.084 | 0.023 | 0.234 | Alcohol oxidase inhibitor | 0.15 0.01 CHEMBL315985 0.15 0.01 CHEMBL313120 0.234 0.005 CHEMBL3526499 0.234 0.005 CHEMBL4525805 | CHEMBL4525805 | |
| 0.119 | 0.059 | 0.217 | Cystathionine beta-synthase inhibitor | 0.217 0.021 CHEMBL4525757 0.122 0.056 CHEMBL315985 0.122 0.056 CHEMBL313120 0.096 0.081 CHEMBL3526872 0.184 0.029 CHEMBL3526499 0.184 0.029 CHEMBL4525805 0.096 0.081 CHEMBL3526693 | CHEMBL4525757 | |
| 0.081 | 0.024 | 0.155 | Purinergic P2X1 antagonist | 0.068 0.034 CHEMBL4525756 0.071 0.031 CHEMBL4525757 0.117 0.012 CHEMBL315985 0.117 0.012 CHEMBL313120 0.055 0.051 CHEMBL3526872 0.155 0.006 CHEMBL3526499 0.155 0.006 CHEMBL4525805 0.055 0.051 CHEMBL3526693 | CHEMBL4525805 | |
| 0.139 | 0.083 | 0.169 | Adenylate cyclase stimulant | 0.137 0.086 CHEMBL4525756 0.164 0.043 CHEMBL315985 0.164 0.043 CHEMBL313120 0.169 0.036 CHEMBL3526499 0.169 0.036 CHEMBL4525805 | CHEMBL4525805 | |
| 0.205 | 0.15 | 0.205 | Insulysin inhibitor | |||
| 0.153 | 0.101 | 0.195 | Phospholipase C inhibitor | 0.195 0.047 CHEMBL4525756 0.146 0.115 CHEMBL4525757 0.165 0.079 CHEMBL315985 0.165 0.079 CHEMBL313120 0.193 0.049 CHEMBL3526499 0.193 0.049 CHEMBL4525805 | CHEMBL4525756 | |
| 0.123 | 0.071 | 0.127 | Cathepsin H inhibitor | 0.104 0.1 CHEMBL315985 0.104 0.1 CHEMBL313120 0.127 0.067 CHEMBL3526499 0.127 0.067 CHEMBL4525805 | CHEMBL4525805 | |
| 0.106 | 0.055 | 0.115 | Anabolic | 0.113 0.047 CHEMBL4525756 0.115 0.044 CHEMBL315985 0.115 0.044 CHEMBL313120 0.11 0.05 CHEMBL3526499 0.11 0.05 CHEMBL4525805 | CHEMBL313120 | |
| 0.182 | 0.132 | 0.295 | DNA damaging | 0.295 0.059 CHEMBL4525757 0.264 0.073 CHEMBL3526872 0.264 0.073 CHEMBL3526499 0.264 0.073 CHEMBL4525805 0.264 0.073 CHEMBL3526693 | CHEMBL4525757 | |
| 0.107 | 0.057 | 0.231 | Adenylate kinase inhibitor | 0.097 0.072 CHEMBL4525756 0.112 0.052 CHEMBL4525757 0.157 0.024 CHEMBL315985 0.157 0.024 CHEMBL313120 0.096 0.074 CHEMBL3526872 0.231 0.011 CHEMBL3526499 0.231 0.011 CHEMBL4525805 0.096 0.074 CHEMBL3526693 | CHEMBL4525805 | |
| 0.118 | 0.07 | 0.349 | Alkylator | 0.169 0.038 CHEMBL4525756 0.309 0.012 CHEMBL4525757 0.164 0.04 CHEMBL315985 0.164 0.04 CHEMBL313120 0.349 0.01 CHEMBL3526872 0.187 0.03 CHEMBL3526499 0.187 0.03 CHEMBL4525805 0.349 0.01 CHEMBL3526693 | CHEMBL3526693 | |
| 0.136 | 0.089 | 0.16 | Ca2+-transporting ATPase inhibitor | 0.138 0.083 CHEMBL4525757 0.152 0.038 CHEMBL315985 0.152 0.038 CHEMBL313120 0.158 0.026 CHEMBL3526872 0.16 0.024 CHEMBL3526499 0.16 0.024 CHEMBL4525805 0.158 0.026 CHEMBL3526693 | CHEMBL4525805 | |
| 0.068 | 0.021 | 0.068 | Aminopeptidase N inhibitor | |||
| 0.07 | 0.024 | 0.07 | NMDA 2A receptor antagonist | 0.049 0.039 CHEMBL4525756 | ||
| 0.163 | 0.119 | 0.221 | Neurotrophic factor enhancer | 0.221 0.058 CHEMBL4525757 0.192 0.084 CHEMBL315985 0.192 0.084 CHEMBL313120 0.172 0.108 CHEMBL3526872 0.188 0.089 CHEMBL3526499 0.188 0.089 CHEMBL4525805 0.172 0.108 CHEMBL3526693 | CHEMBL4525757 | |
| 0.087 | 0.043 | 0.102 | Porphobilinogen synthase inhibitor | 0.067 0.059 CHEMBL4525756 0.102 0.035 CHEMBL3526499 0.102 0.035 CHEMBL4525805 | CHEMBL4525805 | |
| 0.1 | 0.057 | 0.148 | MAP kinase kinase 1 inhibitor | 0.13 0.027 CHEMBL315985 0.13 0.027 CHEMBL313120 0.148 0.017 CHEMBL3526499 0.148 0.017 CHEMBL4525805 | CHEMBL4525805 | |
| 0.108 | 0.066 | 0.108 | 5 Hydroxytryptamine 2 antagonist | |||
| 0.134 | 0.092 | 0.134 | Sphingosine 1-phosphate receptor 5 antagonist | 0.131 0.098 CHEMBL3526499 0.131 0.098 CHEMBL4525805 | ||
| 0.098 | 0.057 | 0.123 | HIV-1 integrase (Overall Integration) inhibitor | 0.087 0.069 CHEMBL315985 0.087 0.069 CHEMBL313120 0.123 0.038 CHEMBL3526499 0.123 0.038 CHEMBL4525805 | CHEMBL4525805 | |
| 0.076 | 0.036 | 0.087 | Protein kinase C beta inhibitor | 0.084 0.025 CHEMBL315985 0.084 0.025 CHEMBL313120 0.087 0.022 CHEMBL3526499 0.087 0.022 CHEMBL4525805 | CHEMBL4525805 | |
| 0.178 | 0.139 | 0.307 | Spasmolytic | 0.279 0.079 CHEMBL4525757 0.273 0.081 CHEMBL315985 0.273 0.081 CHEMBL313120 0.307 0.067 CHEMBL3526872 0.201 0.118 CHEMBL3526499 0.201 0.118 CHEMBL4525805 0.307 0.067 CHEMBL3526693 | CHEMBL3526693 | |
| 0.069 | 0.03 | 0.073 | Cyclin D1 inhibitor | 0.073 0.024 CHEMBL3526499 0.073 0.024 CHEMBL4525805 | CHEMBL4525805 | |
| 0.105 | 0.066 | 0.105 | DOPA decarboxylase inhibitor | 0.103 0.07 CHEMBL3526499 0.103 0.07 CHEMBL4525805 | ||
| 0.114 | 0.077 | 0.177 | Aldehyde dehydrogenase inhibitor | 0.177 0.034 CHEMBL4525757 0.119 0.072 CHEMBL3526499 0.119 0.072 CHEMBL4525805 | CHEMBL4525757 | |
| 0.061 | 0.025 | 0.076 | Aconitate hydratase inhibitor | 0.061 0.025 CHEMBL315985 0.061 0.025 CHEMBL313120 0.076 0.015 CHEMBL3526499 0.076 0.015 CHEMBL4525805 | CHEMBL4525805 | |
| 0.076 | 0.04 | 0.103 | Phospholipase D inhibitor | 0.103 0.013 CHEMBL4525756 0.08 0.034 CHEMBL315985 0.08 0.034 CHEMBL313120 0.092 0.02 CHEMBL3526499 0.092 0.02 CHEMBL4525805 | CHEMBL4525756 | |
| 0.098 | 0.063 | 0.276 | UDP-glucose 4-epimerase inhibitor | 0.276 0.012 CHEMBL4525757 0.142 0.032 CHEMBL315985 0.142 0.032 CHEMBL313120 0.245 0.014 CHEMBL3526872 0.198 0.018 CHEMBL3526499 0.198 0.018 CHEMBL4525805 0.245 0.014 CHEMBL3526693 | CHEMBL4525757 | |
| 0.125 | 0.092 | 0.125 | Cyclooxygenase inhibitor | |||
| 0.102 | 0.069 | 0.167 | Ferrochelatase inhibitor | 0.098 0.073 CHEMBL315985 0.098 0.073 CHEMBL313120 0.167 0.031 CHEMBL3526499 0.167 0.031 CHEMBL4525805 | CHEMBL4525805 | |
| 0.077 | 0.044 | 0.121 | Histidine decarboxylase inhibitor | 0.105 0.03 CHEMBL315985 0.105 0.03 CHEMBL313120 0.121 0.025 CHEMBL3526499 0.121 0.025 CHEMBL4525805 | CHEMBL4525805 | |
| 0.136 | 0.104 | 0.154 | CF transmembrane conductance regulator agonist | 0.154 0.069 CHEMBL3526499 0.154 0.069 CHEMBL4525805 | CHEMBL4525805 | |
| 0.103 | 0.072 | 0.184 | Nav1.4 sodium channel blocker | 0.184 0.023 CHEMBL4525756 0.108 0.064 CHEMBL315985 0.108 0.064 CHEMBL313120 0.127 0.046 CHEMBL3526499 0.127 0.046 CHEMBL4525805 | CHEMBL4525756 | |
| 0.144 | 0.112 | 0.144 | 3C-like protease (Human coronavirus) inhibitor | |||
| 0.063 | 0.035 | 0.123 | Argininosuccinate synthase inhibitor | 0.089 0.022 CHEMBL315985 0.089 0.022 CHEMBL313120 0.123 0.015 CHEMBL3526499 0.123 0.015 CHEMBL4525805 | CHEMBL4525805 | |
| 0.031 | 0.004 | 0.031 | Complement factor D inhibitor | 0.023 0.005 CHEMBL315985 0.023 0.005 CHEMBL313120 0.027 0.005 CHEMBL3526499 0.027 0.005 CHEMBL4525805 | ||
| 0.063 | 0.036 | 0.063 | Heat shock protein 90 beta antagonist | |||
| 0.132 | 0.106 | 0.201 | Interferon gamma antagonist | 0.201 0.04 CHEMBL4525757 0.134 0.103 CHEMBL315985 0.134 0.103 CHEMBL313120 0.201 0.04 CHEMBL3526872 0.132 0.108 CHEMBL3526499 0.132 0.108 CHEMBL4525805 0.201 0.04 CHEMBL3526693 | CHEMBL3526693 | |
| 0.074 | 0.049 | 0.088 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.075 0.049 CHEMBL315985 0.075 0.049 CHEMBL313120 0.088 0.024 CHEMBL3526499 0.088 0.024 CHEMBL4525805 | CHEMBL4525805 | |
| 0.05 | 0.025 | 0.051 | Purinergic P2X4 antagonist | 0.051 0.023 CHEMBL3526499 0.051 0.023 CHEMBL4525805 | CHEMBL4525805 | |
| 0.093 | 0.068 | 0.093 | Platelet activating factor beta antagonist | |||
| 0.104 | 0.081 | 0.142 | TRPA1 agonist | 0.142 0.037 CHEMBL4525756 | CHEMBL4525756 | |
| 0.087 | 0.064 | 0.232 | Triose-phosphate isomerase inhibitor | 0.232 0.008 CHEMBL4525756 0.178 0.014 CHEMBL4525757 0.11 0.039 CHEMBL315985 0.11 0.039 CHEMBL313120 0.158 0.018 CHEMBL3526872 0.154 0.019 CHEMBL3526499 0.154 0.019 CHEMBL4525805 0.158 0.018 CHEMBL3526693 | CHEMBL4525756 | |
| 0.043 | 0.021 | 0.043 | Vascular adhesion protein 1 inhibitor | 0.038 0.028 CHEMBL315985 0.038 0.028 CHEMBL313120 0.041 0.025 CHEMBL3526499 0.041 0.025 CHEMBL4525805 | ||
| 0.089 | 0.068 | 0.11 | Prolactin inhibitor | 0.091 0.066 CHEMBL315985 0.091 0.066 CHEMBL313120 0.11 0.046 CHEMBL3526499 0.11 0.046 CHEMBL4525805 | CHEMBL4525805 | |
| 0.062 | 0.041 | 0.145 | Carbamoyl phosphate synthetase inhibitor | 0.113 0.017 CHEMBL315985 0.113 0.017 CHEMBL313120 0.145 0.012 CHEMBL3526499 0.145 0.012 CHEMBL4525805 | CHEMBL4525805 | |
| 0.04 | 0.022 | 0.062 | Kinesin-like protein 1 inhibitor | 0.062 0.014 CHEMBL4525756 | CHEMBL4525756 | |
| 0.04 | 0.022 | 0.062 | Kinesin antagonist | 0.062 0.014 CHEMBL4525756 | CHEMBL4525756 | |
| 0.087 | 0.069 | 0.179 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.148 0.027 CHEMBL4525757 0.127 0.035 CHEMBL315985 0.127 0.035 CHEMBL313120 0.139 0.03 CHEMBL3526872 0.179 0.019 CHEMBL3526499 0.179 0.019 CHEMBL4525805 0.139 0.03 CHEMBL3526693 | CHEMBL4525805 | |
| 0.079 | 0.064 | 0.079 | Caspase 7 inhibitor | |||
| 0.083 | 0.068 | 0.207 | NADH dehydrogenase inhibitor | 0.207 0.01 CHEMBL4525757 0.118 0.03 CHEMBL315985 0.118 0.03 CHEMBL313120 0.171 0.014 CHEMBL3526872 0.164 0.015 CHEMBL3526499 0.164 0.015 CHEMBL4525805 0.171 0.014 CHEMBL3526693 | CHEMBL4525757 | |
| 0.053 | 0.04 | 0.053 | GABA receptor antagonist | |||
| 0.188 | 0.176 | 0.602 | Cholesterol antagonist | 0.307 0.087 CHEMBL4525756 0.446 0.041 CHEMBL4525757 0.299 0.092 CHEMBL315985 0.299 0.092 CHEMBL313120 0.602 0.018 CHEMBL3526872 0.274 0.109 CHEMBL3526499 0.274 0.109 CHEMBL4525805 0.602 0.018 CHEMBL3526693 | CHEMBL3526693 | |
| 0.125 | 0.113 | 0.169 | Growth hormone agonist | 0.169 0.074 CHEMBL315985 0.169 0.074 CHEMBL313120 0.146 0.09 CHEMBL3526499 0.146 0.09 CHEMBL4525805 | CHEMBL313120 | |
| 0.096 | 0.085 | 0.105 | Protein kinase C gamma inhibitor | 0.105 0.069 CHEMBL315985 0.105 0.069 CHEMBL313120 0.102 0.074 CHEMBL3526499 0.102 0.074 CHEMBL4525805 | CHEMBL313120 | |
| 0.061 | 0.051 | 0.061 | Protease 3C (Human rhinovirus) inhibitor | 0.061 0.051 CHEMBL4525756 | ||
| 0.064 | 0.054 | 0.083 | Glutamate (mGluR6) antagonist | 0.074 0.032 CHEMBL315985 0.074 0.032 CHEMBL313120 0.083 0.021 CHEMBL3526499 0.083 0.021 CHEMBL4525805 | CHEMBL4525805 | |
| 0.043 | 0.034 | 0.043 | Poly(ADP-ribose) polymerase inhibitor | |||
| 0.102 | 0.094 | 0.102 | Glutamate receptor antagonist | |||
| 0.074 | 0.066 | 0.143 | Glycine receptor antagonist | 0.143 0.009 CHEMBL4525756 0.135 0.011 CHEMBL4525757 0.118 0.019 CHEMBL315985 0.118 0.019 CHEMBL313120 0.132 0.013 CHEMBL3526872 0.105 0.028 CHEMBL3526499 0.105 0.028 CHEMBL4525805 0.132 0.013 CHEMBL3526693 | CHEMBL4525756 | |
| 0.043 | 0.036 | 0.043 | Farnesyltransferase inhibitor | |||
| 0.061 | 0.054 | 0.063 | Calcium channel P-type blocker | 0.06 0.056 CHEMBL315985 0.06 0.056 CHEMBL313120 0.063 0.048 CHEMBL3526499 0.063 0.048 CHEMBL4525805 | CHEMBL4525805 | |
| 0.03 | 0.024 | 0.03 | Estradiol 17 beta-dehydrogenase 3 inhibitor | |||
| 0.076 | 0.07 | 0.093 | Inducible nitric-oxide synthase inhibitor | 0.093 0.044 CHEMBL315985 0.093 0.044 CHEMBL313120 | CHEMBL313120 | |
| 0.098 | 0.093 | 0.121 | Acetylcholine release stimulant | 0.121 0.047 CHEMBL4525756 0.113 0.06 CHEMBL3526872 0.113 0.06 CHEMBL3526693 | CHEMBL4525756 | |
| 0.115 | 0.11 | 0.12 | Sphingosine 1-phosphate receptor 2 antagonist | 0.12 0.096 CHEMBL3526499 0.12 0.096 CHEMBL4525805 | CHEMBL4525805 | |
| 0.048 | 0.043 | 0.048 | GABA A receptor antagonist | |||
| 0.066 | 0.062 | 0.125 | Glycine receptor agonist | 0.125 0.011 CHEMBL315985 0.125 0.011 CHEMBL313120 0.115 0.014 CHEMBL3526872 0.105 0.018 CHEMBL3526499 0.105 0.018 CHEMBL4525805 0.115 0.014 CHEMBL3526693 | CHEMBL313120 | |
| 0.085 | 0.081 | 0.264 | Xanthine oxidase inhibitor | 0.264 0.011 CHEMBL4525757 0.137 0.04 CHEMBL3526872 0.091 0.07 CHEMBL3526499 0.091 0.07 CHEMBL4525805 0.137 0.04 CHEMBL3526693 | CHEMBL4525757 | |
| 0.091 | 0.087 | 0.091 | Platelet activating factor antagonist | |||
| 0.041 | 0.041 | 0.057 | Adenylate cyclase 1 inhibitor | 0.055 0.022 CHEMBL315985 0.055 0.022 CHEMBL313120 0.057 0.02 CHEMBL3526499 0.057 0.02 CHEMBL4525805 | CHEMBL4525805 | |
| 0.051 | 0.055 | 0.086 | Androgen agonist | 0.086 0.021 CHEMBL315985 0.086 0.021 CHEMBL313120 0.068 0.032 CHEMBL3526499 0.068 0.032 CHEMBL4525805 | CHEMBL313120 | |
| 0.076 | 0.082 | 0.091 | D-Ala-D-Ala ligase inhibitor | 0.091 0.044 CHEMBL3526499 0.091 0.044 CHEMBL4525805 | CHEMBL4525805 | |
| 0.047 | 0.054 | 0.135 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.092 0.016 CHEMBL4525757 0.088 0.017 CHEMBL315985 0.088 0.017 CHEMBL313120 0.072 0.025 CHEMBL3526872 0.135 0.01 CHEMBL3526499 0.135 0.01 CHEMBL4525805 0.072 0.025 CHEMBL3526693 | CHEMBL4525805 | |
| 0.071 | 0.078 | 0.088 | MAP kinase kinase 7 inhibitor | 0.079 0.048 CHEMBL315985 0.079 0.048 CHEMBL313120 0.088 0.028 CHEMBL3526499 0.088 0.028 CHEMBL4525805 | CHEMBL4525805 | |
| 0.098 | 0.105 | 0.305 | Alpha-N-acetylglucosaminidase inhibitor | 0.241 0.024 CHEMBL4525757 0.222 0.028 CHEMBL315985 0.222 0.028 CHEMBL313120 0.254 0.022 CHEMBL3526872 0.305 0.016 CHEMBL3526499 0.305 0.016 CHEMBL4525805 0.254 0.022 CHEMBL3526693 | CHEMBL4525805 | |
| 0.033 | 0.04 | 0.036 | Dopamine D5 agonist | 0.036 0.034 CHEMBL3526499 0.036 0.034 CHEMBL4525805 | CHEMBL4525805 | |
| 0.031 | 0.039 | 0.036 | Adenosine uptake inhibitor | 0.036 0.019 CHEMBL4525756 | CHEMBL4525756 | |
| 0.062 | 0.071 | 0.123 | Glutamate dehydrogenase inhibitor | 0.09 0.036 CHEMBL315985 0.09 0.036 CHEMBL313120 0.123 0.022 CHEMBL3526499 0.123 0.022 CHEMBL4525805 | CHEMBL4525805 | |
| 0.13 | 0.14 | 0.185 | Lipocortins synthesis antagonist | 0.14 0.121 CHEMBL4525757 0.176 0.074 CHEMBL315985 0.176 0.074 CHEMBL313120 0.185 0.067 CHEMBL3526499 0.185 0.067 CHEMBL4525805 | CHEMBL4525805 | |
| 0.082 | 0.092 | 0.092 | Nitric-oxide synthase inhibitor | 0.092 0.075 CHEMBL315985 0.092 0.075 CHEMBL313120 | CHEMBL313120 | |
| 0.117 | 0.131 | 0.169 | Arachidonic acid antagonist | 0.148 0.091 CHEMBL315985 0.148 0.091 CHEMBL313120 0.169 0.066 CHEMBL3526499 0.169 0.066 CHEMBL4525805 | CHEMBL4525805 | |
| 0.061 | 0.077 | 0.077 | Analgesic, opioid | 0.077 0.052 CHEMBL315985 0.077 0.052 CHEMBL313120 | CHEMBL313120 | |
| 0.051 | 0.067 | 0.187 | Phosphofructokinase-1 inhibitor | 0.157 0.017 CHEMBL4525757 0.101 0.031 CHEMBL315985 0.101 0.031 CHEMBL313120 0.187 0.012 CHEMBL3526872 0.135 0.021 CHEMBL3526499 0.135 0.021 CHEMBL4525805 0.187 0.012 CHEMBL3526693 | CHEMBL3526693 | |
| 0.031 | 0.048 | 0.037 | Glutamate (mGluR8) agonist | 0.037 0.027 CHEMBL3526499 0.037 0.027 CHEMBL4525805 | CHEMBL4525805 | |
| 0.113 | 0.13 | 0.283 | Hexokinase inhibitor | 0.283 0.012 CHEMBL4525757 0.184 0.046 CHEMBL3526872 0.148 0.081 CHEMBL3526499 0.148 0.081 CHEMBL4525805 0.184 0.046 CHEMBL3526693 | CHEMBL4525757 | |
| 0.034 | 0.053 | 0.049 | Kainate receptor agonist | 0.042 0.026 CHEMBL315985 0.042 0.026 CHEMBL313120 0.049 0.015 CHEMBL3526499 0.049 0.015 CHEMBL4525805 | CHEMBL4525805 | |
| 0.045 | 0.063 | 0.136 | Biliverdin reductase inhibitor | 0.085 0.024 CHEMBL315985 0.085 0.024 CHEMBL313120 0.136 0.011 CHEMBL3526499 0.136 0.011 CHEMBL4525805 | CHEMBL4525805 | |
| 0.053 | 0.072 | 0.162 | NMDA 2 receptor antagonist | 0.162 0.014 CHEMBL4525756 0.1 0.032 CHEMBL315985 0.1 0.032 CHEMBL313120 0.069 0.052 CHEMBL3526499 0.069 0.052 CHEMBL4525805 | CHEMBL4525756 | |
| 0.107 | 0.127 | 0.169 | Mannose-6-phosphate isomerase inhibitor | 0.169 0.049 CHEMBL4525757 0.156 0.06 CHEMBL3526499 0.156 0.06 CHEMBL4525805 | CHEMBL4525757 | |
| 0.061 | 0.081 | 0.073 | GABA aminotransferase inhibitor | 0.073 0.057 CHEMBL3526499 0.073 0.057 CHEMBL4525805 | CHEMBL4525805 | |
| 0.056 | 0.077 | 0.087 | Aminopeptidase I inhibitor | 0.07 0.053 CHEMBL315985 0.07 0.053 CHEMBL313120 0.087 0.036 CHEMBL3526499 0.087 0.036 CHEMBL4525805 | CHEMBL4525805 | |
| 0.031 | 0.053 | 0.04 | Guanylate cyclase inhibitor | 0.04 0.033 CHEMBL4525757 | CHEMBL4525757 | |
| 0.021 | 0.049 | 0.026 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.026 0.022 CHEMBL3526499 0.026 0.022 CHEMBL4525805 | CHEMBL4525805 | |
| 0.142 | 0.17 | 0.233 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.174 0.102 CHEMBL315985 0.174 0.102 CHEMBL313120 0.233 0.051 CHEMBL3526499 0.233 0.051 CHEMBL4525805 | CHEMBL4525805 | |
| 0.051 | 0.084 | 0.079 | Interferon inducer | 0.079 0.025 CHEMBL4525757 0.061 0.052 CHEMBL315985 0.061 0.052 CHEMBL313120 0.069 0.036 CHEMBL3526872 0.067 0.04 CHEMBL3526499 0.067 0.04 CHEMBL4525805 0.069 0.036 CHEMBL3526693 | CHEMBL4525757 | |
| 0.061 | 0.097 | 0.083 | Histamine N-methyltransferase inhibitor | 0.083 0.063 CHEMBL3526499 0.083 0.063 CHEMBL4525805 | CHEMBL4525805 | |
| 0.075 | 0.111 | 0.085 | Electrolyte absorption antagonist | 0.085 0.084 CHEMBL3526499 0.085 0.084 CHEMBL4525805 | CHEMBL4525805 | |
| 0.01 | 0.047 | 0.02 | Telomerase stimulant | 0.016 0.013 CHEMBL4525757 0.02 0.008 CHEMBL3526872 0.02 0.008 CHEMBL3526693 | CHEMBL3526693 | |
| 0.065 | 0.102 | 0.154 | Aminopeptidase B inhibitor | 0.154 0.036 CHEMBL4525756 0.105 0.062 CHEMBL3526499 0.105 0.062 CHEMBL4525805 | CHEMBL4525756 | |
| 0.053 | 0.093 | 0.059 | Prolactin release inhibitor | 0.059 0.056 CHEMBL315985 0.059 0.056 CHEMBL313120 | CHEMBL313120 | |
| 0.045 | 0.086 | 0.107 | Phenylalanine 4-hydroxylase inhibitor | 0.065 0.052 CHEMBL315985 0.065 0.052 CHEMBL313120 0.107 0.023 CHEMBL3526499 0.107 0.023 CHEMBL4525805 | CHEMBL4525805 | |
| 0.019 | 0.059 | 0.05 | Fumarate hydratase inhibitor | 0.034 0.024 CHEMBL315985 0.034 0.024 CHEMBL313120 0.05 0.013 CHEMBL3526499 0.05 0.013 CHEMBL4525805 | CHEMBL4525805 | |
| 0.058 | 0.1 | 0.1 | Interferon agonist | 0.1 0.028 CHEMBL4525757 0.071 0.068 CHEMBL315985 0.071 0.068 CHEMBL313120 0.083 0.047 CHEMBL3526872 0.079 0.053 CHEMBL3526499 0.079 0.053 CHEMBL4525805 0.083 0.047 CHEMBL3526693 | CHEMBL4525757 | |
| 0.113 | 0.155 | 0.164 | Psychostimulant | 0.154 0.113 CHEMBL4525757 0.151 0.115 CHEMBL315985 0.151 0.115 CHEMBL313120 0.164 0.104 CHEMBL3526872 0.164 0.104 CHEMBL3526693 | CHEMBL3526693 | |
| 0.012 | 0.054 | 0.032 | Glutamate (mGluR1a) agonist | 0.032 0.008 CHEMBL4525756 | CHEMBL4525756 | |
| 0.071 | 0.114 | 0.166 | Protein kinase C zeta inhibitor | 0.166 0.016 CHEMBL4525756 | CHEMBL4525756 | |
| 0.093 | 0.137 | 0.352 | Protein kinase stimulant | 0.193 0.044 CHEMBL4525757 0.189 0.046 CHEMBL315985 0.189 0.046 CHEMBL313120 0.352 0.012 CHEMBL3526872 0.154 0.066 CHEMBL3526499 0.154 0.066 CHEMBL4525805 0.352 0.012 CHEMBL3526693 | CHEMBL3526693 | |
| 0.066 | 0.111 | 0.139 | Mediator release inhibitor | 0.139 0.034 CHEMBL4525757 0.107 0.062 CHEMBL3526872 0.107 0.062 CHEMBL3526693 | CHEMBL4525757 | |
| 0.103 | 0.152 | 0.174 | Cyclin-dependent kinase 8 inhibitor | 0.14 0.089 CHEMBL315985 0.14 0.089 CHEMBL313120 0.174 0.057 CHEMBL3526499 0.174 0.057 CHEMBL4525805 | CHEMBL4525805 | |
| 0.033 | 0.083 | 0.059 | Glucose-6-phosphate isomerase inhibitor | 0.058 0.02 CHEMBL4525757 0.048 0.032 CHEMBL315985 0.048 0.032 CHEMBL313120 0.055 0.023 CHEMBL3526872 0.059 0.019 CHEMBL3526499 0.059 0.019 CHEMBL4525805 0.055 0.023 CHEMBL3526693 | CHEMBL4525805 | |
| 0.036 | 0.087 | 0.051 | Cytokine production stimulant | 0.051 0.027 CHEMBL4525757 0.051 0.027 CHEMBL3526872 0.051 0.027 CHEMBL3526693 | CHEMBL3526693 | |
| 0.013 | 0.064 | 0.042 | Acetylcholine M4 receptor agonist | 0.042 0.014 CHEMBL315985 0.042 0.014 CHEMBL313120 | CHEMBL313120 | |
| 0.079 | 0.133 | 0.115 | Microtubule formation inhibitor | 0.106 0.079 CHEMBL4525757 0.112 0.071 CHEMBL3526872 0.115 0.067 CHEMBL3526499 0.115 0.067 CHEMBL4525805 0.112 0.071 CHEMBL3526693 | CHEMBL4525805 | |
| 0.189 | 0.243 | 0.619 | Antibacterial | 0.418 0.069 CHEMBL4525756 0.617 0.017 CHEMBL4525757 0.225 0.201 CHEMBL315985 0.225 0.201 CHEMBL313120 0.619 0.016 CHEMBL3526872 0.274 0.155 CHEMBL3526499 0.274 0.155 CHEMBL4525805 0.619 0.016 CHEMBL3526693 | CHEMBL3526693 | |
| 0.077 | 0.131 | 0.136 | MAP kinase kinase inhibitor | 0.107 0.087 CHEMBL315985 0.107 0.087 CHEMBL313120 0.136 0.06 CHEMBL3526499 0.136 0.06 CHEMBL4525805 | CHEMBL4525805 | |
| 0.13 | 0.184 | 0.389 | Interleukin agonist | 0.313 0.042 CHEMBL4525757 0.241 0.086 CHEMBL315985 0.241 0.086 CHEMBL313120 0.389 0.02 CHEMBL3526872 0.241 0.086 CHEMBL3526499 0.241 0.086 CHEMBL4525805 0.389 0.02 CHEMBL3526693 | CHEMBL3526693 | |
| 0.03 | 0.085 | 0.09 | Acyl-CoA dehydrogenase inhibitor | 0.057 0.035 CHEMBL315985 0.057 0.035 CHEMBL313120 0.09 0.019 CHEMBL3526499 0.09 0.019 CHEMBL4525805 | CHEMBL4525805 | |
| 0.027 | 0.082 | 0.039 | Thymidine kinase inhibitor | 0.039 0.031 CHEMBL3526499 0.039 0.031 CHEMBL4525805 | CHEMBL4525805 | |
| 0.024 | 0.079 | 0.087 | Antibiotic Aminoglycoside-like | 0.08 0.004 CHEMBL4525757 0.037 0.024 CHEMBL315985 0.037 0.024 CHEMBL313120 0.087 0.004 CHEMBL3526872 0.04 0.021 CHEMBL3526499 0.04 0.021 CHEMBL4525805 0.087 0.004 CHEMBL3526693 | CHEMBL3526693 | |
| 0.011 | 0.067 | 0.03 | Antibiotic Anthracycline-like | 0.022 0.008 CHEMBL4525757 0.03 0.004 CHEMBL3526872 0.03 0.004 CHEMBL3526693 | CHEMBL3526693 | |
| 0.025 | 0.085 | 0.065 | Ornithine carbamoyltransferase inhibitor | 0.046 0.044 CHEMBL315985 0.046 0.044 CHEMBL313120 0.065 0.028 CHEMBL3526499 0.065 0.028 CHEMBL4525805 | CHEMBL4525805 | |
| 0.017 | 0.077 | 0.036 | Purinergic P2Y15 antagonist | 0.03 0.017 CHEMBL315985 0.03 0.017 CHEMBL313120 0.036 0.01 CHEMBL3526499 0.036 0.01 CHEMBL4525805 | CHEMBL4525805 | |
| 0.131 | 0.191 | 0.557 | Antioxidant | 0.262 0.078 CHEMBL4525756 0.557 0.014 CHEMBL4525757 0.17 0.142 CHEMBL315985 0.17 0.142 CHEMBL313120 0.479 0.023 CHEMBL3526872 0.479 0.023 CHEMBL3526693 | CHEMBL4525757 | |
| 0.041 | 0.103 | 0.057 | NMDA receptor agonist | 0.057 0.052 CHEMBL4525756 | CHEMBL4525756 | |
| 0.042 | 0.105 | 0.104 | Na+ K+ transporting ATPase inhibitor | 0.098 0.033 CHEMBL4525757 0.073 0.057 CHEMBL315985 0.073 0.057 CHEMBL313120 0.104 0.028 CHEMBL3526872 0.076 0.054 CHEMBL3526499 0.076 0.054 CHEMBL4525805 0.104 0.028 CHEMBL3526693 | CHEMBL3526693 | |
| 0.015 | 0.079 | 0.032 | Vanilloid 2 agonist | 0.032 0.008 CHEMBL4525757 0.028 0.013 CHEMBL3526872 0.028 0.013 CHEMBL3526693 | CHEMBL4525757 | |
| 0.149 | 0.215 | 0.21 | Nitric-oxide synthase stimulant | 0.204 0.082 CHEMBL4525757 0.17 0.153 CHEMBL315985 0.17 0.153 CHEMBL313120 0.168 0.157 CHEMBL3526872 0.21 0.074 CHEMBL3526499 0.21 0.074 CHEMBL4525805 0.168 0.157 CHEMBL3526693 | CHEMBL4525805 | |
| 0.052 | 0.123 | 0.069 | Keratolytic | 0.069 0.067 CHEMBL3526499 0.069 0.067 CHEMBL4525805 | CHEMBL4525805 | |
| 0.014 | 0.09 | 0.078 | Vasopressin 2 antagonist | 0.078 0.008 CHEMBL315985 0.078 0.008 CHEMBL313120 0.046 0.015 CHEMBL3526499 0.046 0.015 CHEMBL4525805 | CHEMBL313120 | |
| 0.057 | 0.134 | 0.118 | Alcohol dehydrogenase inhibitor | 0.118 0.036 CHEMBL4525757 0.085 0.072 CHEMBL3526499 0.085 0.072 CHEMBL4525805 | CHEMBL4525757 | |
| 0.086 | 0.163 | 0.103 | Transcription factor STAT6 inhibitor | 0.103 0.099 CHEMBL3526499 0.103 0.099 CHEMBL4525805 | CHEMBL4525805 | |
| 0.009 | 0.088 | 0.028 | Uridine phosphorylase inhibitor | 0.028 0.019 CHEMBL3526499 0.028 0.019 CHEMBL4525805 | CHEMBL4525805 | |
| 0.017 | 0.096 | 0.039 | Purinergic P2Y antagonist | 0.039 0.038 CHEMBL3526499 0.039 0.038 CHEMBL4525805 | CHEMBL4525805 | |
| 0.012 | 0.091 | 0.066 | Protein 30S ribosomal subunit inhibitor | 0.057 0.007 CHEMBL4525757 0.066 0.005 CHEMBL3526872 0.066 0.005 CHEMBL3526693 | CHEMBL3526693 | |
| 0.064 | 0.144 | 0.106 | Adenylate cyclase inhibitor | 0.106 0.079 CHEMBL3526499 0.106 0.079 CHEMBL4525805 | CHEMBL4525805 | |
| 0.075 | 0.156 | 0.303 | Cyclooxygenase 3 inhibitor | 0.243 0.009 CHEMBL4525757 0.11 0.09 CHEMBL315985 0.11 0.09 CHEMBL313120 0.303 0.006 CHEMBL3526872 0.103 0.098 CHEMBL3526499 0.103 0.098 CHEMBL4525805 0.303 0.006 CHEMBL3526693 | CHEMBL3526693 | |
| 0.036 | 0.118 | 0.093 | Catalase inhibitor | 0.093 0.041 CHEMBL4525756 | CHEMBL4525756 | |
| 0.067 | 0.151 | 0.277 | Beta glucuronidase inhibitor | 0.277 0.007 CHEMBL4525757 0.121 0.045 CHEMBL3526872 0.121 0.045 CHEMBL3526693 | CHEMBL4525757 | |
| 0.103 | 0.187 | 0.43 | Hepatoprotectant | 0.175 0.084 CHEMBL4525756 0.43 0.011 CHEMBL4525757 0.191 0.071 CHEMBL315985 0.191 0.071 CHEMBL313120 0.421 0.012 CHEMBL3526872 0.173 0.086 CHEMBL3526499 0.173 0.086 CHEMBL4525805 0.421 0.012 CHEMBL3526693 | CHEMBL4525757 | |
| 0.118 | 0.202 | 0.145 | Heat shock protein 70 antagonist | 0.145 0.058 CHEMBL4525757 0.139 0.08 CHEMBL3526499 0.139 0.08 CHEMBL4525805 | CHEMBL4525757 | |
| 0.053 | 0.137 | 0.096 | Falcipain 2 inhibitor | 0.096 0.055 CHEMBL4525757 | CHEMBL4525757 | |
| 0.055 | 0.14 | 0.071 | GABA B receptor agonist | 0.071 0.065 CHEMBL3526499 0.071 0.065 CHEMBL4525805 | CHEMBL4525805 | |
| 0.067 | 0.152 | 0.113 | Mucolytic | 0.113 0.061 CHEMBL3526872 0.096 0.084 CHEMBL3526499 0.096 0.084 CHEMBL4525805 0.113 0.061 CHEMBL3526693 | CHEMBL3526693 | |
| 0.055 | 0.141 | 0.098 | Falcipain inhibitor | 0.098 0.056 CHEMBL4525757 | CHEMBL4525757 | |
| 0.039 | 0.127 | 0.11 | Cathepsin G inhibitor | 0.11 0.03 CHEMBL4525756 | CHEMBL4525756 | |
| 0.021 | 0.11 | 0.126 | Leukocyte elastase inhibitor | 0.126 0.007 CHEMBL4525756 | CHEMBL4525756 | |
| 0.007 | 0.1 | 0.046 | Arginase inhibitor | 0.044 0.019 CHEMBL4525757 0.046 0.017 CHEMBL3526872 0.046 0.017 CHEMBL3526693 | CHEMBL3526693 | |
| 0.098 | 0.192 | 0.198 | Melanin inhibitor | 0.198 0.042 CHEMBL4525757 0.164 0.065 CHEMBL3526872 0.164 0.065 CHEMBL3526693 | CHEMBL4525757 | |
| 0.03 | 0.127 | 0.276 | Antineoplastic antibiotic | 0.174 0.026 CHEMBL4525757 0.276 0.011 CHEMBL3526872 0.276 0.011 CHEMBL3526693 | CHEMBL3526693 | |
| 0.031 | 0.131 | 0.053 | Sphingosine kinase 2 inhibitor | 0.053 0.041 CHEMBL3526499 0.053 0.041 CHEMBL4525805 | CHEMBL4525805 | |
| 0.088 | 0.19 | 0.189 | DNA repair enzyme inhibitor | 0.179 0.014 CHEMBL4525757 0.189 0.011 CHEMBL3526872 0.107 0.105 CHEMBL3526499 0.107 0.105 CHEMBL4525805 0.189 0.011 CHEMBL3526693 | CHEMBL3526693 | |
| 0.017 | 0.12 | 0.076 | Phosphorylase inhibitor | 0.076 0.018 CHEMBL4525757 0.054 0.028 CHEMBL315985 0.054 0.028 CHEMBL313120 0.069 0.021 CHEMBL3526872 0.043 0.034 CHEMBL3526499 0.043 0.034 CHEMBL4525805 0.069 0.021 CHEMBL3526693 | CHEMBL4525757 | |
| 0.119 | 0.225 | 0.292 | Cardiotonic | 0.292 0.06 CHEMBL315985 0.292 0.06 CHEMBL313120 0.166 0.156 CHEMBL3526872 0.166 0.156 CHEMBL3526693 | CHEMBL313120 | |
| 0.018 | 0.128 | 0.057 | Adenosine deaminase inhibitor | 0.057 0.023 CHEMBL3526499 0.057 0.023 CHEMBL4525805 | CHEMBL4525805 | |
| 0.041 | 0.156 | 0.226 | Monophenol monooxygenase inhibitor | 0.226 0.027 CHEMBL4525757 0.132 0.054 CHEMBL3526872 0.132 0.054 CHEMBL3526693 | CHEMBL4525757 | |
| 0.028 | 0.143 | 0.063 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.063 0.037 CHEMBL4525757 | CHEMBL4525757 | |
| 0.017 | 0.135 | 0.026 | Hedgehog signaling activator | 0.026 0.025 CHEMBL315985 0.026 0.025 CHEMBL313120 | CHEMBL313120 | |
| 0.06 | 0.179 | 0.078 | Estrogen-related receptor beta agonist | 0.078 0.073 CHEMBL3526499 0.078 0.073 CHEMBL4525805 | CHEMBL4525805 | |
| 0.091 | 0.212 | 0.171 | MAP kinase kinase 2 inhibitor | 0.171 0.103 CHEMBL315985 0.171 0.103 CHEMBL313120 0.171 0.103 CHEMBL3526499 0.171 0.103 CHEMBL4525805 | CHEMBL4525805 | |
| 0.156 | 0.282 | 0.449 | Interleukin 2 agonist | 0.415 0.023 CHEMBL4525757 0.345 0.048 CHEMBL315985 0.345 0.048 CHEMBL313120 0.449 0.016 CHEMBL3526872 0.279 0.09 CHEMBL3526499 0.279 0.09 CHEMBL4525805 0.449 0.016 CHEMBL3526693 | CHEMBL3526693 | |
| 0.023 | 0.152 | 0.035 | Glucose-6-phosphate dehydrogenase inhibitor | 0.035 0.034 CHEMBL315985 0.035 0.034 CHEMBL313120 | CHEMBL313120 | |
| 0.086 | 0.216 | 0.338 | Nitric oxide antagonist | 0.338 0.034 CHEMBL4525757 0.134 0.112 CHEMBL315985 0.134 0.112 CHEMBL313120 0.32 0.037 CHEMBL3526872 0.32 0.037 CHEMBL3526693 | CHEMBL4525757 | |
| 0.047 | 0.18 | 0.229 | Expectorant | 0.21 0.018 CHEMBL4525757 0.229 0.015 CHEMBL3526872 0.229 0.015 CHEMBL3526693 | CHEMBL3526693 | |
| 0.076 | 0.213 | 0.277 | Cell wall synthesis inhibitor | 0.221 0.023 CHEMBL4525756 0.277 0.012 CHEMBL4525757 0.223 0.022 CHEMBL3526872 0.134 0.081 CHEMBL3526499 0.134 0.081 CHEMBL4525805 0.223 0.022 CHEMBL3526693 | CHEMBL4525757 | |
| 0.004 | 0.147 | 0.049 | Estrone sulfatase inhibitor | 0.049 0.007 CHEMBL4525756 | CHEMBL4525756 | |
| 0.024 | 0.168 | 0.049 | Leukotriene B4 antagonist | 0.049 0.046 CHEMBL4525757 | CHEMBL4525757 | |
| 0.013 | 0.158 | 0.061 | Carbonic anhydrase VB inhibitor | 0.061 0.034 CHEMBL4525756 | CHEMBL4525756 | |
| 0.038 | 0.185 | 0.225 | Topoisomerase I inhibitor | 0.225 0.021 CHEMBL4525757 0.221 0.022 CHEMBL3526872 0.221 0.022 CHEMBL3526693 | CHEMBL4525757 | |
| 0.005 | 0.155 | 0.349 | Cholecystokinin B antagonist | 0.349 0.003 CHEMBL4525756 | CHEMBL4525756 | |
| 0.01 | 0.16 | 0.133 | Factor Xa inhibitor | 0.133 0.009 CHEMBL4525756 | CHEMBL4525756 | |
| 0.021 | 0.172 | 0.073 | Alpha-mannosidase inhibitor | 0.071 0.016 CHEMBL4525757 0.073 0.015 CHEMBL3526872 0.059 0.028 CHEMBL3526499 0.059 0.028 CHEMBL4525805 0.073 0.015 CHEMBL3526693 | CHEMBL3526693 | |
| 0.015 | 0.171 | 0.068 | Mannosidase inhibitor | 0.067 0.013 CHEMBL4525757 0.068 0.013 CHEMBL3526872 0.049 0.027 CHEMBL3526499 0.049 0.027 CHEMBL4525805 0.068 0.013 CHEMBL3526693 | CHEMBL3526693 | |
| 0.007 | 0.174 | 0.053 | Antidiuretic hormone antagonist | 0.053 0.022 CHEMBL315985 0.053 0.022 CHEMBL313120 | CHEMBL313120 | |
| 0.006 | 0.178 | 0.369 | Cholecystokinin antagonist | 0.369 0.004 CHEMBL4525756 | CHEMBL4525756 | |
| 0.12 | 0.3 | 0.246 | Vasodilator, peripheral | 0.219 0.155 CHEMBL315985 0.219 0.155 CHEMBL313120 0.218 0.156 CHEMBL3526872 0.246 0.13 CHEMBL3526499 0.246 0.13 CHEMBL4525805 0.218 0.156 CHEMBL3526693 | CHEMBL4525805 | |
| 0.121 | 0.302 | 0.351 | Vasodilator, coronary | 0.351 0.055 CHEMBL4525757 0.335 0.063 CHEMBL3526872 0.335 0.063 CHEMBL3526693 | CHEMBL4525757 | |
| 0.077 | 0.258 | 0.276 | DNA methylase inhibitor | 0.276 0.036 CHEMBL4525757 0.235 0.057 CHEMBL3526872 0.235 0.057 CHEMBL3526693 | CHEMBL4525757 | |
| 0.079 | 0.263 | 0.225 | Interleukin 6 antagonist | 0.225 0.029 CHEMBL4525757 0.135 0.115 CHEMBL315985 0.135 0.115 CHEMBL313120 0.177 0.057 CHEMBL3526872 0.177 0.057 CHEMBL3526693 | CHEMBL4525757 | |
| 0.022 | 0.207 | 0.09 | Carbonic anhydrase VA inhibitor | 0.09 0.03 CHEMBL4525756 | CHEMBL4525756 | |
| 0.047 | 0.233 | 0.313 | Amylase inhibitor | 0.313 0.017 CHEMBL4525757 0.274 0.022 CHEMBL3526872 0.106 0.092 CHEMBL3526499 0.106 0.092 CHEMBL4525805 0.274 0.022 CHEMBL3526693 | CHEMBL4525757 | |
| 0.071 | 0.262 | 0.249 | DNA methyltransferase I inhibitor | 0.249 0.047 CHEMBL4525757 0.135 0.123 CHEMBL3526872 0.135 0.123 CHEMBL3526693 | CHEMBL4525757 | |
| 0.004 | 0.197 | 0.027 | RNA-directed RNA polymerase stimulant | 0.027 0.023 CHEMBL315985 0.027 0.023 CHEMBL313120 | CHEMBL313120 | |
| 0.018 | 0.217 | 0.13 | Carbonic anhydrase V inhibitor | 0.13 0.019 CHEMBL4525756 | CHEMBL4525756 | |
| 0.024 | 0.224 | 0.124 | Carbonic anhydrase XIII inhibitor | 0.124 0.028 CHEMBL4525756 | CHEMBL4525756 | |
| 0.016 | 0.218 | 0.054 | Neuraminidase (Influenza A) inhibitor | 0.054 0.019 CHEMBL4525757 0.046 0.031 CHEMBL3526872 0.046 0.031 CHEMBL3526693 | CHEMBL4525757 | |
| 0.062 | 0.266 | 0.237 | Diuretic | 0.237 0.033 CHEMBL4525756 0.133 0.092 CHEMBL4525757 0.228 0.035 CHEMBL3526872 0.228 0.035 CHEMBL3526693 | CHEMBL4525756 | |
| 0.117 | 0.324 | 0.409 | Peptidyltransferase inhibitor | 0.383 0.008 CHEMBL4525757 0.219 0.078 CHEMBL315985 0.219 0.078 CHEMBL313120 0.409 0.006 CHEMBL3526872 0.242 0.056 CHEMBL3526499 0.242 0.056 CHEMBL4525805 0.409 0.006 CHEMBL3526693 | CHEMBL3526693 | |
| 0.053 | 0.262 | 0.098 | Phosphodiesterase 6D inhibitor | 0.098 0.057 CHEMBL4525757 | CHEMBL4525757 | |
| 0.068 | 0.295 | 0.292 | NOS3 expression enhancer | 0.292 0.019 CHEMBL4525757 0.138 0.086 CHEMBL315985 0.138 0.086 CHEMBL313120 0.259 0.025 CHEMBL3526872 0.259 0.025 CHEMBL3526693 | CHEMBL4525757 | |
| 0.04 | 0.268 | 0.234 | AMP-activated protein kinase stimulant | 0.208 0.01 CHEMBL4525757 0.234 0.008 CHEMBL3526872 0.234 0.008 CHEMBL3526693 | CHEMBL3526693 | |
| 0.027 | 0.257 | 0.101 | Histone deacetylase stimulant | 0.101 0.027 CHEMBL4525757 0.073 0.052 CHEMBL3526872 0.073 0.052 CHEMBL3526693 | CHEMBL4525757 | |
| 0.027 | 0.257 | 0.101 | Histone deacetylase SIRT1 stimulant | 0.101 0.027 CHEMBL4525757 0.073 0.052 CHEMBL3526872 0.073 0.052 CHEMBL3526693 | CHEMBL4525757 | |
| 0.033 | 0.264 | 0.358 | Topoisomerase II inhibitor | 0.24 0.026 CHEMBL4525757 0.358 0.013 CHEMBL3526872 0.358 0.013 CHEMBL3526693 | CHEMBL3526693 | |
| 0.006 | 0.237 | 0.022 | Dopamine D1 agonist | 0.022 0.018 CHEMBL4525756 | CHEMBL4525756 | |
| 0.036 | 0.268 | 0.13 | Uric acid excretion stimulant | 0.13 0.032 CHEMBL4525757 0.094 0.06 CHEMBL3526872 0.094 0.06 CHEMBL3526693 | CHEMBL4525757 | |
| 0.001 | 0.237 | 0.013 | Antibiotic Macrolide-like | 0.013 0.011 CHEMBL3526872 0.013 0.011 CHEMBL3526693 | CHEMBL3526693 | |
| 0.004 | 0.244 | 0.779 | Cholecystokinin agonist | 0.779 0.002 CHEMBL4525756 | CHEMBL4525756 | |
| 0.044 | 0.286 | 0.116 | Protein kinase C nu inhibitor | 0.116 0.098 CHEMBL315985 0.116 0.098 CHEMBL313120 | CHEMBL313120 | |
| 0.005 | 0.247 | 0.764 | Cholecystokinin A agonist | 0.764 0.001 CHEMBL4525756 | CHEMBL4525756 | |
| 0.039 | 0.282 | 0.302 | Thrombolytic | 0.146 0.085 CHEMBL4525756 0.272 0.029 CHEMBL4525757 0.302 0.024 CHEMBL3526872 0.302 0.024 CHEMBL3526693 | CHEMBL3526693 | |
| 0.007 | 0.253 | 0.123 | Estrogen agonist | 0.123 0.014 CHEMBL4525756 | CHEMBL4525756 | |
| 0.005 | 0.253 | 0.05 | Sodium/glucose cotransporter 2 inhibitor | 0.05 0.006 CHEMBL4525757 0.024 0.023 CHEMBL3526872 0.024 0.023 CHEMBL3526693 | CHEMBL4525757 | |
| 0.087 | 0.335 | 0.472 | Transcription factor NF kappa B inhibitor | 0.472 0.049 CHEMBL4525757 0.453 0.052 CHEMBL3526872 0.453 0.052 CHEMBL3526693 | CHEMBL4525757 | |
| 0.042 | 0.291 | 0.089 | Lanosterol 14 alpha demethylase inhibitor | 0.089 0.074 CHEMBL3526499 0.089 0.074 CHEMBL4525805 | CHEMBL4525805 | |
| 0.05 | 0.299 | 0.534 | Anticoagulant | 0.534 0.008 CHEMBL4525756 0.229 0.044 CHEMBL4525757 0.248 0.039 CHEMBL3526872 0.248 0.039 CHEMBL3526693 | CHEMBL4525756 | |
| 0.091 | 0.342 | 0.387 | Alpha-glucosidase inhibitor | 0.387 0.121 CHEMBL4525757 0.26 0.181 CHEMBL3526872 0.26 0.181 CHEMBL3526693 | CHEMBL4525757 | |
| 0.004 | 0.256 | 0.05 | Estrogen receptor beta agonist | 0.05 0.019 CHEMBL4525756 | CHEMBL4525756 | |
| 0.004 | 0.256 | 0.421 | Cholecystokinin A antagonist | 0.421 0.003 CHEMBL4525756 | CHEMBL4525756 | |
| 0.021 | 0.276 | 0.087 | Heparanase inhibitor | 0.052 0.04 CHEMBL4525756 0.087 0.005 CHEMBL4525757 0.078 0.007 CHEMBL3526872 0.078 0.007 CHEMBL3526693 | CHEMBL4525757 | |
| 0.096 | 0.356 | 0.567 | Antithrombotic | 0.275 0.107 CHEMBL4525756 0.567 0.02 CHEMBL4525757 0.565 0.02 CHEMBL3526872 0.565 0.02 CHEMBL3526693 | CHEMBL4525757 | |
| 0.076 | 0.347 | 0.24 | ATPase inhibitor | 0.24 0.016 CHEMBL4525757 0.187 0.05 CHEMBL3526872 0.187 0.05 CHEMBL3526693 | CHEMBL4525757 | |
| 0.064 | 0.337 | 0.329 | Hemostatic | 0.314 0.014 CHEMBL4525756 0.248 0.022 CHEMBL4525757 0.329 0.013 CHEMBL3526872 0.329 0.013 CHEMBL3526693 | CHEMBL3526693 | |
| 0.006 | 0.282 | 0.053 | Sodium/glucose cotransporter inhibitor | 0.053 0.005 CHEMBL4525757 0.027 0.015 CHEMBL3526872 0.027 0.015 CHEMBL3526693 | CHEMBL4525757 | |
| 0.027 | 0.314 | 0.257 | DNA intercalator | 0.093 0.082 CHEMBL4525756 0.136 0.049 CHEMBL4525757 0.257 0.015 CHEMBL3526872 0.257 0.015 CHEMBL3526693 | CHEMBL3526693 | |
| 0.013 | 0.305 | 0.708 | Cholecystokinin B agonist | 0.708 0.001 CHEMBL4525756 | CHEMBL4525756 | |
| 0.009 | 0.302 | 0.045 | Aldose reductase inhibitor | 0.045 0.044 CHEMBL4525757 | CHEMBL4525757 | |
| 0.024 | 0.321 | 0.051 | Factor III inhibitor | 0.051 0.031 CHEMBL4525757 | CHEMBL4525757 | |
| 0.081 | 0.381 | 0.181 | Hypoxia-inducible factor 1 alpha inhibitor | 0.181 0.177 CHEMBL3526872 0.181 0.177 CHEMBL3526693 | CHEMBL3526693 | |
| 0.032 | 0.334 | 0.062 | Lipocortins synthesis agonist | 0.062 0.032 CHEMBL4525757 0.06 0.035 CHEMBL3526872 0.06 0.035 CHEMBL3526693 | CHEMBL4525757 | |
| 0.052 | 0.368 | 0.496 | Free radical scavenger | 0.496 0.017 CHEMBL4525757 0.415 0.026 CHEMBL3526872 0.415 0.026 CHEMBL3526693 | CHEMBL4525757 | |
| 0.012 | 0.344 | 0.088 | Elastase inhibitor | 0.088 0.013 CHEMBL4525756 | CHEMBL4525756 | |
| 0.017 | 0.36 | 0.086 | Thrombin inhibitor | 0.086 0.036 CHEMBL4525756 | CHEMBL4525756 | |
| 0.018 | 0.362 | 0.269 | Topoisomerase II alpha inhibitor | 0.143 0.024 CHEMBL4525757 0.269 0.009 CHEMBL3526872 0.269 0.009 CHEMBL3526693 | CHEMBL3526693 | |
| 0.012 | 0.362 | 0.034 | Toll-Like receptor 4 agonist | 0.034 0.008 CHEMBL4525756 0.032 0.009 CHEMBL4525757 0.032 0.01 CHEMBL3526872 0.032 0.01 CHEMBL3526693 | CHEMBL4525756 | |
| 0.014 | 0.369 | 0.125 | CDC25A inhibitor | 0.125 0.018 CHEMBL4525756 | CHEMBL4525756 | |
| 0.011 | 0.372 | 0.038 | Purinergic P2Y2 antagonist | 0.038 0.017 CHEMBL4525756 | CHEMBL4525756 | |
| 0.103 | 0.469 | 0.756 | Cyclophilin D inhibitor | 0.727 0.012 CHEMBL4525757 0.363 0.113 CHEMBL315985 0.363 0.113 CHEMBL313120 0.756 0.009 CHEMBL3526872 0.345 0.125 CHEMBL3526499 0.345 0.125 CHEMBL4525805 0.756 0.009 CHEMBL3526693 | CHEMBL3526693 | |
| 0.097 | 0.482 | 0.487 | Apoptosis agonist | 0.486 0.079 CHEMBL4525757 0.487 0.078 CHEMBL3526872 0.487 0.078 CHEMBL3526693 | CHEMBL3526693 | |
| 0.033 | 0.42 | 0.335 | Dual specificity phosphatase inhibitor | 0.335 0.023 CHEMBL4525756 | CHEMBL4525756 | |
| 0.041 | 0.433 | 0.116 | Interleukin 4 antagonist | 0.116 0.091 CHEMBL4525757 0.11 0.101 CHEMBL3526872 0.11 0.101 CHEMBL3526693 | CHEMBL4525757 | |
| 0.021 | 0.418 | 0.087 | Gastric antisecretory | 0.087 0.083 CHEMBL3526499 0.087 0.083 CHEMBL4525805 | CHEMBL4525805 | |
| 0.016 | 0.424 | 0.064 | HIV-1 integrase inhibitor | 0.064 0.058 CHEMBL4525756 | CHEMBL4525756 | |
| 0.007 | 0.426 | 0.151 | HIV-1 integrase (Strand Transfer) inhibitor | 0.151 0.013 CHEMBL4525756 0.073 0.034 CHEMBL3526499 0.073 0.034 CHEMBL4525805 | CHEMBL4525756 | |
| 0.024 | 0.444 | 0.213 | Multidrug resistance-associated protein 1 inhibitor | 0.213 0.008 CHEMBL4525756 0.104 0.072 CHEMBL3526872 0.104 0.072 CHEMBL3526693 | CHEMBL4525756 | |
| 0.004 | 0.434 | 0.032 | Factor XI inhibitor | 0.032 0.027 CHEMBL4525756 | CHEMBL4525756 | |
| 0.019 | 0.455 | 0.115 | Cell adhesion molecule inhibitor | 0.115 0.026 CHEMBL4525757 0.099 0.035 CHEMBL3526872 0.099 0.035 CHEMBL3526693 | CHEMBL4525757 | |
| 0.037 | 0.476 | 0.338 | Platelet adhesion inhibitor | 0.188 0.078 CHEMBL4525756 0.328 0.025 CHEMBL4525757 0.338 0.023 CHEMBL3526872 0.338 0.023 CHEMBL3526693 | CHEMBL3526693 | |
| 0.029 | 0.471 | 0.135 | DNA polymerase I inhibitor | 0.117 0.071 CHEMBL4525757 0.102 0.084 CHEMBL315985 0.102 0.084 CHEMBL313120 0.135 0.058 CHEMBL3526872 0.135 0.058 CHEMBL3526693 | CHEMBL3526693 | |
| 0.04 | 0.482 | 0.094 | Interleukin 12 antagonist | 0.094 0.065 CHEMBL4525757 | CHEMBL4525757 | |
| 0.007 | 0.467 | 0.06 | Neuraminidase inhibitor | 0.06 0.044 CHEMBL4525757 | CHEMBL4525757 | |
| 0.079 | 0.548 | 0.14 | CC chemokine 6 receptor antagonist | 0.137 0.047 CHEMBL4525757 0.14 0.04 CHEMBL3526872 0.14 0.04 CHEMBL3526693 | CHEMBL3526693 | |
| 0.009 | 0.483 | 0.071 | Neuraminidase (influenza) inhibitor | 0.071 0.034 CHEMBL4525757 0.064 0.044 CHEMBL3526872 0.064 0.044 CHEMBL3526693 | CHEMBL4525757 | |
| 0.012 | 0.496 | 0.065 | Nitric oxide donor | 0.065 0.04 CHEMBL3526872 0.065 0.04 CHEMBL3526693 | CHEMBL3526693 | |
| 0.022 | 0.516 | 0.098 | Thioredoxin inhibitor | 0.098 0.05 CHEMBL4525757 | CHEMBL4525757 | |
| 0.006 | 0.505 | 0.134 | HIV-1 integrase (3'-Processing) inhibitor | 0.134 0.016 CHEMBL4525756 | CHEMBL4525756 | |
| 0.054 | 0.556 | 0.524 | Immunomodulator | 0.335 0.065 CHEMBL4525757 0.191 0.174 CHEMBL315985 0.191 0.174 CHEMBL313120 0.524 0.02 CHEMBL3526872 0.524 0.02 CHEMBL3526693 | CHEMBL3526693 | |
| 0.032 | 0.537 | 0.138 | Transcription factor NF kappa B stimulant | 0.118 0.026 CHEMBL4525757 0.138 0.019 CHEMBL3526872 0.138 0.019 CHEMBL3526693 | CHEMBL3526693 | |
| 0.022 | 0.532 | 0.642 | Angiogenesis stimulant | 0.39 0.023 CHEMBL4525756 0.642 0.005 CHEMBL4525757 0.598 0.007 CHEMBL3526872 0.598 0.007 CHEMBL3526693 | CHEMBL4525757 | |
| 0.02 | 0.537 | 0.311 | Dual specificity phosphatase 3 inhibitor | 0.311 0.027 CHEMBL4525756 | CHEMBL4525756 | |
| 0.021 | 0.54 | 0.074 | Adenine nucleotide translocase inhibitor | 0.074 0.012 CHEMBL4525756 0.063 0.024 CHEMBL4525757 0.059 0.031 CHEMBL3526872 0.059 0.031 CHEMBL3526693 | CHEMBL4525756 | |
| 0.024 | 0.546 | 0.207 | Cell adhesion inhibitor | 0.207 0.023 CHEMBL4525757 0.199 0.025 CHEMBL3526872 0.199 0.025 CHEMBL3526693 | CHEMBL4525757 | |
| 0.025 | 0.554 | 0.151 | Toll-Like receptor 4 antagonist | 0.151 0.02 CHEMBL4525757 0.146 0.023 CHEMBL3526872 0.146 0.023 CHEMBL3526693 | CHEMBL4525757 | |
| 0.005 | 0.552 | 0.082 | NMDA 2D receptor antagonist | 0.082 0.004 CHEMBL4525756 | CHEMBL4525756 | |
| 0.05 | 0.602 | 0.113 | Sphingosine 1-phosphate receptor 2 agonist | 0.113 0.067 CHEMBL315985 0.113 0.067 CHEMBL313120 | CHEMBL313120 | |
| 0.012 | 0.581 | 0.072 | Glucose-6-phosphate translocase inhibitor | 0.072 0.015 CHEMBL4525757 0.06 0.024 CHEMBL3526872 0.06 0.024 CHEMBL3526693 | CHEMBL4525757 | |
| 0.011 | 0.583 | 0.275 | Protein-tyrosine phosphatase inhibitor | 0.275 0.024 CHEMBL4525756 | CHEMBL4525756 | |
| 0.009 | 0.594 | 0.109 | Protein 50S ribosomal subunit inhibitor | 0.094 0.015 CHEMBL4525757 0.109 0.011 CHEMBL3526872 0.109 0.011 CHEMBL3526693 | CHEMBL3526693 | |
| 0.004 | 0.604 | 0.023 | Motilin receptor agonist | 0.023 0.015 CHEMBL3526872 0.023 0.015 CHEMBL3526693 | CHEMBL3526693 | |
| 0.005 | 0.623 | 0.115 | Protein-tyrosine phosphatase 1B inhibitor | 0.115 0.066 CHEMBL4525756 | CHEMBL4525756 | |
| 0.003 | 0.625 | 0.036 | 1,3-Beta-glucan synthase inhibitor | 0.036 0.005 CHEMBL4525756 | CHEMBL4525756 | |
| 0.013 | 0.65 | 0.115 | ATPase (Vacuolar H+) inhibitor | 0.115 0.023 CHEMBL4525757 0.097 0.044 CHEMBL3526872 0.097 0.044 CHEMBL3526693 | CHEMBL4525757 | |
| 0.027 | 0.67 | 0.392 | Immunosuppressant | 0.382 0.071 CHEMBL4525757 0.392 0.066 CHEMBL3526872 0.392 0.066 CHEMBL3526693 | CHEMBL3526693 | |
| 0.041 | 0.719 | 0.409 | Apoptosis antagonist | 0.366 0.049 CHEMBL4525757 0.222 0.155 CHEMBL315985 0.222 0.155 CHEMBL313120 0.409 0.036 CHEMBL3526872 0.409 0.036 CHEMBL3526693 | CHEMBL3526693 | |
| 0.015 | 0.701 | 0.279 | Vasodilator | 0.211 0.096 CHEMBL4525757 0.279 0.056 CHEMBL3526872 0.279 0.056 CHEMBL3526693 | CHEMBL3526693 | |
| 0.01 | 0.704 | 0.259 | Platelet antagonist | 0.221 0.087 CHEMBL4525757 0.259 0.068 CHEMBL3526872 0.259 0.068 CHEMBL3526693 | CHEMBL3526693 | |
| 0.039 | 0.744 | 0.252 | Caspase 3 stimulant | 0.194 0.178 CHEMBL4525757 0.252 0.111 CHEMBL3526872 0.252 0.111 CHEMBL3526693 | CHEMBL3526693 | |
| 0.011 | 0.789 | 0.216 | Insulin secretagoues | 0.193 0.04 CHEMBL4525757 0.216 0.029 CHEMBL3526872 0.216 0.029 CHEMBL3526693 | CHEMBL3526693 | |
| 0.011 | 0.801 | 0.098 | Factor IXa inhibitor | 0.098 0.01 CHEMBL4525756 0.087 0.014 CHEMBL4525757 0.072 0.019 CHEMBL3526872 0.072 0.019 CHEMBL3526693 | CHEMBL4525756 | |
| 0.017 | 0.82 | 0.541 | Hypoglycemic | 0.541 0.012 CHEMBL4525757 0.508 0.014 CHEMBL3526872 0.508 0.014 CHEMBL3526693 | CHEMBL4525757 | |
| 0.004 | 0.818 | 0.338 | Selectin antagonist | 0.141 0.019 CHEMBL4525756 0.338 0.004 CHEMBL4525757 0.335 0.004 CHEMBL3526872 0.335 0.004 CHEMBL3526693 | CHEMBL4525757 | |
| 0.007 | 0.853 | 0.274 | Tumour necrosis factor alpha release inhibitor | 0.274 0.064 CHEMBL4525757 0.17 0.134 CHEMBL3526872 0.17 0.134 CHEMBL3526693 | CHEMBL4525757 | |
| 0.005 | 0.917 | 0.168 | Hypolipemic | 0.168 0.12 CHEMBL3526872 0.168 0.12 CHEMBL3526693 | CHEMBL3526693 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |