Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.750.0050.8635 Hydroxytryptamine release stimulant

0.853 0.003 CHEMBL3278702

0.654 0.01 CHEMBL3544672

0.767 0.004 CHEMBL3278706

0.863 0.002 CHEMBL3544671

0.502 0.027 CHEMBL1105

0.71 0.006 CHEMBL3544690

0.685 0.008 CHEMBL3544691

0.538 0.022 CHEMBL3544673

0.734 0.005 CHEMBL3544692

CHEMBL3544671
0.7410.0190.804Caspase 9 stimulant

0.644 0.031 CHEMBL3278702

0.804 0.011 CHEMBL3544672

0.702 0.024 CHEMBL3278706

0.571 0.041 CHEMBL3544671

0.743 0.019 CHEMBL1105

0.592 0.037 CHEMBL3544690

0.776 0.014 CHEMBL3544691

0.69 0.025 CHEMBL3544673

0.532 0.049 CHEMBL3544692

CHEMBL3544672
0.6120.0150.612Vasodilator, peripheral

0.552 0.021 CHEMBL3278702

0.473 0.034 CHEMBL3544672

0.603 0.016 CHEMBL3278706

0.515 0.025 CHEMBL3544671

0.434 0.045 CHEMBL1105

0.397 0.056 CHEMBL3544690

0.448 0.041 CHEMBL3544691

0.403 0.054 CHEMBL3544673

0.367 0.067 CHEMBL3544692

0.5090.030.6555 Hydroxytryptamine release inhibitor

0.637 0.007 CHEMBL3278702

0.503 0.031 CHEMBL3544672

0.543 0.021 CHEMBL3278706

0.655 0.005 CHEMBL3544671

0.582 0.014 CHEMBL1105

0.577 0.014 CHEMBL3544690

0.521 0.026 CHEMBL3544691

0.599 0.011 CHEMBL3544673

0.595 0.012 CHEMBL3544692

CHEMBL3544671
0.5160.0420.594Transcription factor NF kappa B inhibitor

0.369 0.071 CHEMBL3278702

0.382 0.068 CHEMBL3544672

0.594 0.032 CHEMBL3278706

0.424 0.058 CHEMBL3544671

0.452 0.052 CHEMBL1105

0.301 0.093 CHEMBL3544690

0.436 0.056 CHEMBL3544691

0.503 0.044 CHEMBL3544673

0.354 0.075 CHEMBL3544692

CHEMBL3278706
0.4930.0340.783Aldehyde oxidase inhibitor

0.716 0.007 CHEMBL3278702

0.662 0.012 CHEMBL3544672

0.64 0.014 CHEMBL3278706

0.783 0.005 CHEMBL3544671

0.648 0.013 CHEMBL1105

0.706 0.008 CHEMBL3544690

0.725 0.007 CHEMBL3544691

0.711 0.007 CHEMBL3544673

0.772 0.005 CHEMBL3544692

CHEMBL3544671
0.4450.0090.526Non-steroidal antiinflammatory agent

0.387 0.015 CHEMBL3278702

0.231 0.052 CHEMBL3544672

0.425 0.011 CHEMBL3278706

0.35 0.02 CHEMBL3544671

0.526 0.005 CHEMBL1105

0.204 0.067 CHEMBL3544690

0.208 0.065 CHEMBL3544691

0.485 0.007 CHEMBL3544673

0.184 0.084 CHEMBL3544692

CHEMBL1105
0.4730.040.508Immunosuppressant

0.395 0.065 CHEMBL3278702

0.426 0.054 CHEMBL3544672

0.508 0.031 CHEMBL3278706

0.428 0.054 CHEMBL3544671

0.295 0.118 CHEMBL1105

0.208 0.188 CHEMBL3544690

0.457 0.045 CHEMBL3544691

0.33 0.097 CHEMBL3544673

0.232 0.164 CHEMBL3544692

CHEMBL3278706
0.4210.010.498Melanin inhibitor

0.432 0.01 CHEMBL3278702

0.362 0.015 CHEMBL3544672

0.498 0.007 CHEMBL3278706

0.47 0.008 CHEMBL3544671

0.323 0.019 CHEMBL1105

0.308 0.021 CHEMBL3544690

0.393 0.012 CHEMBL3544691

0.352 0.016 CHEMBL3544673

0.338 0.017 CHEMBL3544692

CHEMBL3278706
0.4970.0890.615Antiinflammatory

0.35 0.172 CHEMBL3278702

0.615 0.049 CHEMBL3278706

0.454 0.108 CHEMBL3544671

0.455 0.108 CHEMBL1105

0.409 0.134 CHEMBL3544690

0.329 0.19 CHEMBL3544691

0.57 0.062 CHEMBL3544673

0.514 0.082 CHEMBL3544692

CHEMBL3278706
0.4260.0220.534Superoxide dismutase inhibitor

0.404 0.026 CHEMBL3278702

0.364 0.033 CHEMBL3544672

0.465 0.017 CHEMBL3278706

0.415 0.024 CHEMBL3544671

0.521 0.011 CHEMBL1105

0.359 0.034 CHEMBL3544690

0.375 0.031 CHEMBL3544691

0.534 0.01 CHEMBL3544673

0.37 0.032 CHEMBL3544692

CHEMBL3544673
0.4140.0260.531Free radical scavenger

0.255 0.066 CHEMBL3278702

0.259 0.065 CHEMBL3544672

0.531 0.013 CHEMBL3278706

0.362 0.036 CHEMBL3544671

0.289 0.055 CHEMBL1105

0.202 0.096 CHEMBL3544690

0.363 0.036 CHEMBL3544691

0.406 0.028 CHEMBL3544673

0.305 0.05 CHEMBL3544692

CHEMBL3278706
0.4160.0340.483Lipoxygenase inhibitor

0.277 0.083 CHEMBL3278702

0.231 0.113 CHEMBL3544672

0.483 0.021 CHEMBL3278706

0.302 0.07 CHEMBL3544671

0.429 0.031 CHEMBL1105

0.192 0.149 CHEMBL3544690

0.254 0.098 CHEMBL3544691

0.457 0.025 CHEMBL3544673

0.211 0.13 CHEMBL3544692

CHEMBL3278706
0.3990.0160.484Anesthetic general

0.382 0.019 CHEMBL3278702

0.301 0.033 CHEMBL3544672

0.454 0.011 CHEMBL3278706

0.408 0.015 CHEMBL3544671

0.458 0.011 CHEMBL1105

0.257 0.047 CHEMBL3544690

0.331 0.027 CHEMBL3544691

0.484 0.009 CHEMBL3544673

0.279 0.039 CHEMBL3544692

CHEMBL3544673
0.3820.0040.465TRPA1 agonist

0.19 0.013 CHEMBL3278702

0.233 0.006 CHEMBL3544672

0.465 0.003 CHEMBL3278706

0.22 0.008 CHEMBL3544671

0.204 0.01 CHEMBL1105

0.187 0.014 CHEMBL3544690

0.293 0.005 CHEMBL3544691

0.241 0.006 CHEMBL3544673

0.216 0.008 CHEMBL3544692

CHEMBL3278706
0.3820.0180.4815 Hydroxytryptamine uptake stimulant

0.352 0.025 CHEMBL3278702

0.315 0.038 CHEMBL3544672

0.412 0.012 CHEMBL3278706

0.386 0.017 CHEMBL3544671

0.451 0.007 CHEMBL1105

0.347 0.026 CHEMBL3544690

0.347 0.026 CHEMBL3544691

0.481 0.005 CHEMBL3544673

0.381 0.018 CHEMBL3544692

CHEMBL3544673
0.4510.0910.482Apoptosis agonist

0.365 0.131 CHEMBL3278702

0.448 0.092 CHEMBL3544672

0.482 0.08 CHEMBL3278706

0.387 0.12 CHEMBL3544671

0.315 0.162 CHEMBL1105

0.328 0.153 CHEMBL3544690

0.472 0.083 CHEMBL3544691

0.334 0.149 CHEMBL3544673

0.345 0.142 CHEMBL3544692

CHEMBL3278706
0.360.0080.525Neurotrophic factor enhancer

0.35 0.009 CHEMBL3278702

0.319 0.014 CHEMBL3544672

0.525 0.004 CHEMBL3278706

0.488 0.004 CHEMBL3544671

0.315 0.014 CHEMBL1105

0.297 0.019 CHEMBL3544690

0.436 0.005 CHEMBL3544691

0.429 0.005 CHEMBL3544673

0.394 0.006 CHEMBL3544692

CHEMBL3278706
0.3630.0130.551Monophenol monooxygenase inhibitor

0.346 0.014 CHEMBL3278702

0.234 0.026 CHEMBL3544672

0.551 0.006 CHEMBL3278706

0.476 0.008 CHEMBL3544671

0.243 0.025 CHEMBL1105

0.193 0.035 CHEMBL3544690

0.313 0.016 CHEMBL3544691

0.323 0.016 CHEMBL3544673

0.264 0.022 CHEMBL3544692

CHEMBL3278706
0.3780.0310.393Tumour necrosis factor alpha release inhibitor

0.393 0.028 CHEMBL3278702

0.201 0.108 CHEMBL3544672

0.313 0.049 CHEMBL3278706

0.352 0.037 CHEMBL3544671

0.247 0.076 CHEMBL1105

0.218 0.094 CHEMBL3544690

0.17 0.134 CHEMBL3544673

CHEMBL3278702
0.3590.0180.375Platelet adhesion inhibitor

0.375 0.015 CHEMBL3278706

0.247 0.05 CHEMBL1105

0.269 0.043 CHEMBL3544673

CHEMBL3278706
0.3630.0230.464Cyclic AMP phosphodiesterase inhibitor

0.464 0.009 CHEMBL3278702

0.333 0.03 CHEMBL3544672

0.363 0.023 CHEMBL3278706

0.461 0.009 CHEMBL3544671

0.374 0.021 CHEMBL1105

0.313 0.037 CHEMBL3544690

0.329 0.031 CHEMBL3544691

0.37 0.021 CHEMBL3544673

0.31 0.038 CHEMBL3544692

CHEMBL3278702
0.4020.0750.689Histamine release inhibitor

0.632 0.008 CHEMBL3278702

0.421 0.065 CHEMBL3544672

0.473 0.039 CHEMBL3278706

0.689 0.005 CHEMBL3544671

0.584 0.012 CHEMBL1105

0.493 0.031 CHEMBL3544690

0.467 0.042 CHEMBL3544691

0.646 0.007 CHEMBL3544673

0.536 0.019 CHEMBL3544692

CHEMBL3544671
0.3650.0420.502Antioxidant

0.289 0.066 CHEMBL3278702

0.277 0.071 CHEMBL3544672

0.502 0.02 CHEMBL3278706

0.387 0.037 CHEMBL3544671

0.284 0.068 CHEMBL1105

0.309 0.058 CHEMBL3544690

0.37 0.041 CHEMBL3544691

0.397 0.035 CHEMBL3544673

0.419 0.032 CHEMBL3544692

CHEMBL3278706
0.4020.080.489Calcium channel L-type activator

0.422 0.067 CHEMBL3278702

0.358 0.111 CHEMBL3544672

0.484 0.034 CHEMBL3278706

0.48 0.036 CHEMBL3544671

0.424 0.066 CHEMBL1105

0.37 0.103 CHEMBL3544690

0.433 0.06 CHEMBL3544691

0.489 0.032 CHEMBL3544673

0.444 0.054 CHEMBL3544692

CHEMBL3544673
0.3660.0540.75Caspase 3 stimulant

0.259 0.104 CHEMBL3278702

0.737 0.005 CHEMBL3544672

0.349 0.059 CHEMBL3278706

0.237 0.125 CHEMBL3544671

0.336 0.064 CHEMBL1105

0.297 0.08 CHEMBL3544690

0.75 0.005 CHEMBL3544691

0.312 0.073 CHEMBL3544673

0.276 0.093 CHEMBL3544692

CHEMBL3544691
0.3240.0230.577Tyrosine 3 hydroxylase inhibitor

0.302 0.032 CHEMBL3278702

0.248 0.07 CHEMBL3544672

0.46 0.005 CHEMBL3278706

0.407 0.007 CHEMBL3544671

0.409 0.007 CHEMBL1105

0.264 0.056 CHEMBL3544690

0.335 0.02 CHEMBL3544691

0.577 0.003 CHEMBL3544673

0.356 0.015 CHEMBL3544692

CHEMBL3544673
0.3060.010.352Succinate dehydrogenase inhibitor

0.241 0.026 CHEMBL3278702

0.291 0.012 CHEMBL3544672

0.352 0.005 CHEMBL3278706

0.249 0.023 CHEMBL3544671

0.329 0.007 CHEMBL1105

0.232 0.029 CHEMBL3544690

0.301 0.01 CHEMBL3544691

0.341 0.006 CHEMBL3544673

0.24 0.026 CHEMBL3544692

CHEMBL3278706
0.3520.0630.6Cholesterol antagonist

0.565 0.023 CHEMBL3278702

0.416 0.046 CHEMBL3544672

0.443 0.042 CHEMBL3278706

0.6 0.019 CHEMBL3544671

0.52 0.029 CHEMBL1105

0.491 0.034 CHEMBL3544690

0.47 0.037 CHEMBL3544691

0.56 0.024 CHEMBL3544673

0.534 0.027 CHEMBL3544692

CHEMBL3544671
0.3420.0550.417Calcium channel activator

0.373 0.036 CHEMBL3278702

0.281 0.112 CHEMBL3544672

0.29 0.102 CHEMBL3278706

0.327 0.067 CHEMBL3544671

0.417 0.019 CHEMBL1105

0.344 0.054 CHEMBL3544690

0.227 0.176 CHEMBL3544691

0.372 0.037 CHEMBL3544673

0.298 0.094 CHEMBL3544692

CHEMBL1105
0.3390.0560.392Spasmolytic

0.366 0.048 CHEMBL3278702

0.241 0.095 CHEMBL3544672

0.379 0.045 CHEMBL3278706

0.392 0.042 CHEMBL3544671

0.268 0.083 CHEMBL1105

0.261 0.087 CHEMBL3544690

0.265 0.085 CHEMBL3544691

0.29 0.074 CHEMBL3544673

0.283 0.077 CHEMBL3544692

CHEMBL3544671
0.3240.0420.369Pyruvate kinase inhibitor

0.187 0.089 CHEMBL3278702

0.158 0.108 CHEMBL3544672

0.369 0.028 CHEMBL3278706

0.217 0.072 CHEMBL3544671

0.202 0.08 CHEMBL1105

0.186 0.089 CHEMBL3544691

0.238 0.065 CHEMBL3544673

0.148 0.117 CHEMBL3544692

CHEMBL3278706
0.2880.0150.328Phospholipase A2 inhibitor

0.227 0.03 CHEMBL3278702

0.194 0.046 CHEMBL3544672

0.328 0.01 CHEMBL3278706

0.241 0.026 CHEMBL3544671

0.303 0.013 CHEMBL1105

0.159 0.066 CHEMBL3544690

0.207 0.039 CHEMBL3544691

0.32 0.011 CHEMBL3544673

0.174 0.057 CHEMBL3544692

CHEMBL3278706
0.330.0670.384Apoptosis antagonist

0.282 0.099 CHEMBL3278702

0.3 0.085 CHEMBL3544672

0.384 0.043 CHEMBL3278706

0.319 0.073 CHEMBL3544671

0.3 0.085 CHEMBL1105

0.232 0.145 CHEMBL3544690

0.335 0.064 CHEMBL3544691

0.341 0.06 CHEMBL3544673

0.269 0.11 CHEMBL3544692

CHEMBL3278706
0.3080.0540.39Insulysin inhibitor

0.265 0.083 CHEMBL3278702

0.276 0.075 CHEMBL3544672

0.362 0.03 CHEMBL3278706

0.324 0.045 CHEMBL3544671

0.347 0.035 CHEMBL1105

0.226 0.122 CHEMBL3544690

0.332 0.041 CHEMBL3544691

0.39 0.024 CHEMBL3544673

0.291 0.064 CHEMBL3544692

CHEMBL3544673
0.3260.0740.496Antithrombotic

0.403 0.048 CHEMBL3278702

0.34 0.068 CHEMBL3544672

0.39 0.052 CHEMBL3278706

0.442 0.04 CHEMBL3544671

0.46 0.036 CHEMBL1105

0.31 0.082 CHEMBL3544690

0.377 0.056 CHEMBL3544691

0.496 0.029 CHEMBL3544673

0.343 0.067 CHEMBL3544692

CHEMBL3544673
0.2790.0440.334Nitric oxide antagonist

0.229 0.058 CHEMBL3278702

0.194 0.069 CHEMBL3544672

0.334 0.034 CHEMBL3278706

0.266 0.047 CHEMBL3544671

0.186 0.073 CHEMBL1105

0.169 0.082 CHEMBL3544690

0.229 0.058 CHEMBL3544691

0.226 0.059 CHEMBL3544673

0.199 0.068 CHEMBL3544692

CHEMBL3278706
0.2550.0220.255Cytokine production inhibitor

0.113 0.096 CHEMBL3544672

0.175 0.046 CHEMBL3278706

0.128 0.082 CHEMBL1105

0.106 0.105 CHEMBL3544690

0.2860.0530.345Vasodilator

0.319 0.042 CHEMBL3278702

0.221 0.089 CHEMBL3544672

0.315 0.043 CHEMBL3278706

0.345 0.034 CHEMBL3544671

0.186 0.116 CHEMBL1105

0.198 0.106 CHEMBL3544690

0.236 0.078 CHEMBL3544691

0.203 0.102 CHEMBL3544673

0.214 0.094 CHEMBL3544692

CHEMBL3544671
0.2750.0440.275Sigma receptor agonist

0.176 0.071 CHEMBL3278702

0.23 0.053 CHEMBL3278706

0.159 0.079 CHEMBL3544671

0.173 0.072 CHEMBL1105

0.157 0.081 CHEMBL3544673

0.2440.0190.372Aldehyde dehydrogenase inhibitor

0.253 0.018 CHEMBL3278702

0.258 0.017 CHEMBL3544672

0.372 0.006 CHEMBL3278706

0.354 0.007 CHEMBL3544671

0.239 0.02 CHEMBL1105

0.209 0.026 CHEMBL3544690

0.36 0.007 CHEMBL3544691

0.339 0.008 CHEMBL3544673

0.307 0.011 CHEMBL3544692

CHEMBL3278706
0.230.0070.284HIV-1 integrase (Overall Integration) inhibitor

0.151 0.025 CHEMBL3278702

0.128 0.035 CHEMBL3544672

0.279 0.004 CHEMBL3278706

0.185 0.015 CHEMBL3544671

0.252 0.005 CHEMBL1105

0.11 0.046 CHEMBL3544690

0.162 0.021 CHEMBL3544691

0.284 0.004 CHEMBL3544673

0.141 0.029 CHEMBL3544692

CHEMBL3544673
0.2670.0450.357Platelet aggregation inhibitor

0.193 0.086 CHEMBL3278702

0.152 0.127 CHEMBL3278706

0.357 0.024 CHEMBL1105

0.235 0.059 CHEMBL3544673

CHEMBL1105
0.2980.0810.37212-Lipoxygenase inhibitor

0.219 0.131 CHEMBL3278702

0.235 0.118 CHEMBL3544672

0.372 0.048 CHEMBL3278706

0.265 0.1 CHEMBL3544671

0.3 0.08 CHEMBL1105

0.211 0.139 CHEMBL3544690

0.283 0.09 CHEMBL3544691

0.345 0.059 CHEMBL3544673

0.253 0.107 CHEMBL3544692

CHEMBL3278706
0.2440.0280.352Lipid peroxidase inhibitor

0.224 0.033 CHEMBL3278702

0.132 0.082 CHEMBL3544672

0.352 0.013 CHEMBL3278706

0.311 0.017 CHEMBL3544671

0.139 0.076 CHEMBL1105

0.196 0.043 CHEMBL3544691

0.214 0.036 CHEMBL3544673

0.172 0.054 CHEMBL3544692

CHEMBL3278706
0.2460.0320.246Tumour necrosis factor antagonist

0.167 0.08 CHEMBL3278702

0.13 0.126 CHEMBL3544672

0.144 0.108 CHEMBL3278706

0.229 0.038 CHEMBL1105

0.152 0.098 CHEMBL3544690

0.139 0.114 CHEMBL3544673

0.2130.0050.415DOPA decarboxylase inhibitor

0.158 0.018 CHEMBL3278702

0.171 0.013 CHEMBL3544672

0.329 0.002 CHEMBL3278706

0.233 0.004 CHEMBL3544671

0.3 0.003 CHEMBL1105

0.14 0.027 CHEMBL3544690

0.251 0.004 CHEMBL3544691

0.415 0.001 CHEMBL3544673

0.207 0.005 CHEMBL3544692

CHEMBL3544673
0.2020.0080.239Electron transport complex I inhibitor

0.174 0.012 CHEMBL3278702

0.239 0.006 CHEMBL3544672

0.155 0.018 CHEMBL3278706

0.141 0.026 CHEMBL3544671

0.126 0.039 CHEMBL1105

0.19 0.009 CHEMBL3544690

0.184 0.01 CHEMBL3544691

0.152 0.019 CHEMBL3544692

CHEMBL3544672
0.2890.0970.435Vasodilator, coronary

0.424 0.029 CHEMBL3278702

0.357 0.052 CHEMBL3544672

0.258 0.127 CHEMBL3278706

0.383 0.041 CHEMBL3544671

0.337 0.062 CHEMBL1105

0.435 0.026 CHEMBL3544690

0.319 0.073 CHEMBL3544691

0.302 0.086 CHEMBL3544673

0.393 0.038 CHEMBL3544692

CHEMBL3544690
0.1990.0070.444Vanilloid agonist

0.082 0.063 CHEMBL3278702

0.388 0.004 CHEMBL3544672

0.246 0.005 CHEMBL3278706

0.09 0.047 CHEMBL3544671

0.106 0.027 CHEMBL1105

0.081 0.069 CHEMBL3544690

0.444 0.004 CHEMBL3544691

0.121 0.018 CHEMBL3544673

0.088 0.051 CHEMBL3544692

CHEMBL3544691
0.3140.1220.39415-Lipoxygenase inhibitor

0.394 0.077 CHEMBL3278706

0.322 0.116 CHEMBL1105

0.381 0.083 CHEMBL3544673

CHEMBL3278706
0.2840.0940.444Sodium/bile acid cotransporter inhibitor

0.347 0.042 CHEMBL3278702

0.31 0.07 CHEMBL3544672

0.348 0.041 CHEMBL3278706

0.376 0.026 CHEMBL3544671

0.42 0.012 CHEMBL1105

0.323 0.06 CHEMBL3544690

0.346 0.043 CHEMBL3544691

0.444 0.008 CHEMBL3544673

0.357 0.035 CHEMBL3544692

CHEMBL3544673
0.2120.0220.256Arachidonic acid antagonist

0.206 0.028 CHEMBL3278702

0.209 0.025 CHEMBL3544672

0.228 0.013 CHEMBL3278706

0.216 0.019 CHEMBL3544671

0.248 0.006 CHEMBL1105

0.2 0.033 CHEMBL3544690

0.219 0.018 CHEMBL3544691

0.256 0.005 CHEMBL3544673

0.211 0.023 CHEMBL3544692

CHEMBL3544673
0.2010.0130.218Calcium antagonist

0.218 0.011 CHEMBL3278702

0.161 0.02 CHEMBL3544672

0.078 0.065 CHEMBL3278706

0.103 0.046 CHEMBL3544671

0.124 0.033 CHEMBL1105

0.171 0.018 CHEMBL3544690

0.076 0.067 CHEMBL3544692

CHEMBL3278702
0.1970.0090.197Sphingosine 1-phosphate receptor 4 antagonist

0.178 0.015 CHEMBL3278702

0.167 0.021 CHEMBL3544672

0.194 0.01 CHEMBL3278706

0.171 0.019 CHEMBL3544671

0.197 0.009 CHEMBL1105

0.147 0.036 CHEMBL3544690

0.16 0.025 CHEMBL3544691

0.189 0.011 CHEMBL3544673

0.14 0.043 CHEMBL3544692

0.2670.0860.315Hypoxia-inducible factor 1 alpha inhibitor

0.198 0.154 CHEMBL3278702

0.189 0.165 CHEMBL3544672

0.28 0.077 CHEMBL3278706

0.198 0.154 CHEMBL3544671

0.315 0.059 CHEMBL1105

0.181 0.178 CHEMBL3544690

0.189 0.166 CHEMBL3544691

0.315 0.059 CHEMBL3544673

0.18 0.178 CHEMBL3544692

CHEMBL3544673
0.2310.0520.333Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.235 0.05 CHEMBL3278702

0.218 0.059 CHEMBL3544672

0.273 0.033 CHEMBL3278706

0.261 0.038 CHEMBL3544671

0.312 0.02 CHEMBL1105

0.224 0.055 CHEMBL3544690

0.245 0.045 CHEMBL3544691

0.333 0.015 CHEMBL3544673

0.251 0.042 CHEMBL3544692

CHEMBL3544673
0.1990.0250.469Cystathionine beta-synthase inhibitor

0.207 0.023 CHEMBL3278702

0.156 0.038 CHEMBL3544672

0.297 0.01 CHEMBL3278706

0.271 0.012 CHEMBL3544671

0.361 0.006 CHEMBL1105

0.171 0.032 CHEMBL3544690

0.215 0.021 CHEMBL3544691

0.469 0.004 CHEMBL3544673

0.232 0.018 CHEMBL3544692

CHEMBL3544673
0.1890.0150.198Vanilloid 1 agonist

0.161 0.029 CHEMBL3278702

0.189 0.015 CHEMBL3544672

0.192 0.014 CHEMBL3278706

0.158 0.031 CHEMBL3544671

0.198 0.012 CHEMBL1105

0.156 0.033 CHEMBL3544690

0.185 0.017 CHEMBL3544691

0.194 0.014 CHEMBL3544673

0.153 0.035 CHEMBL3544692

CHEMBL1105
0.20.0290.215MAO A inhibitor

0.215 0.026 CHEMBL3278706

CHEMBL3278706
0.2480.0770.2485 Hydroxytryptamine 1E antagonist

0.23 0.097 CHEMBL3278706

0.232 0.095 CHEMBL1105

0.235 0.092 CHEMBL3544673

0.169 0.167 CHEMBL3544692

0.1850.0150.213Phosphodiesterase IV inhibitor

0.108 0.04 CHEMBL3278702

0.213 0.011 CHEMBL1105

0.088 0.054 CHEMBL3544673

CHEMBL1105
0.1890.020.24Carbonic anhydrase XV inhibitor

0.142 0.034 CHEMBL3278702

0.134 0.038 CHEMBL3544672

0.237 0.013 CHEMBL3278706

0.164 0.026 CHEMBL3544671

0.206 0.018 CHEMBL1105

0.129 0.04 CHEMBL3544690

0.154 0.029 CHEMBL3544691

0.24 0.013 CHEMBL3544673

0.148 0.031 CHEMBL3544692

CHEMBL3544673
0.2490.080.321Gastrin inhibitor

0.219 0.12 CHEMBL3278702

0.207 0.138 CHEMBL3544672

0.251 0.078 CHEMBL3278706

0.218 0.122 CHEMBL3544671

0.321 0.021 CHEMBL1105

0.193 0.16 CHEMBL3544690

0.206 0.14 CHEMBL3544691

0.32 0.021 CHEMBL3544673

0.192 0.162 CHEMBL3544692

CHEMBL1105
0.1830.0170.251Photosensitizer

0.145 0.034 CHEMBL3278702

0.127 0.049 CHEMBL3544672

0.201 0.013 CHEMBL3278706

0.154 0.029 CHEMBL3544671

0.237 0.007 CHEMBL1105

0.117 0.061 CHEMBL3544690

0.135 0.042 CHEMBL3544691

0.251 0.006 CHEMBL3544673

0.124 0.053 CHEMBL3544692

CHEMBL3544673
0.1910.0280.276Toll-Like receptor 2 antagonist

0.25 0.009 CHEMBL3278702

0.204 0.022 CHEMBL3544672

0.224 0.015 CHEMBL3278706

0.276 0.006 CHEMBL3544671

0.245 0.01 CHEMBL1105

0.231 0.013 CHEMBL3544690

0.225 0.014 CHEMBL3544691

0.27 0.007 CHEMBL3544673

0.253 0.009 CHEMBL3544692

CHEMBL3544671
0.1830.0210.209Bronchodilator

0.208 0.017 CHEMBL3278702

0.112 0.051 CHEMBL3544672

0.18 0.022 CHEMBL3278706

0.209 0.017 CHEMBL3544671

0.157 0.029 CHEMBL1105

0.105 0.059 CHEMBL3544690

0.106 0.057 CHEMBL3544691

0.151 0.031 CHEMBL3544673

0.097 0.068 CHEMBL3544692

CHEMBL3544671
0.2240.0660.304Amyloid beta aggregation inhibitor

0.149 0.109 CHEMBL3278702

0.14 0.116 CHEMBL3544672

0.304 0.044 CHEMBL3278706

0.186 0.085 CHEMBL3544671

0.19 0.083 CHEMBL1105

0.174 0.092 CHEMBL3544691

0.24 0.061 CHEMBL3544673

0.146 0.111 CHEMBL3544692

CHEMBL3278706
0.1920.0390.204Tubulin antagonist

0.125 0.075 CHEMBL3278702

0.119 0.08 CHEMBL3544672

0.204 0.036 CHEMBL1105

0.12 0.08 CHEMBL3544690

CHEMBL1105
0.2660.1130.387Thyroid hormone antagonist

0.228 0.139 CHEMBL3278706

0.387 0.06 CHEMBL1105

0.355 0.072 CHEMBL3544673

CHEMBL1105
0.2610.1120.347Thyroid hormone beta antagonist

0.21 0.146 CHEMBL3278706

0.347 0.07 CHEMBL1105

0.303 0.086 CHEMBL3544673

CHEMBL1105
0.1830.0360.202Neurotrophic factor

0.145 0.064 CHEMBL3278702

0.151 0.058 CHEMBL3544672

0.202 0.027 CHEMBL3278706

0.16 0.051 CHEMBL3544671

0.166 0.046 CHEMBL3544691

0.114 0.106 CHEMBL3544673

0.118 0.098 CHEMBL3544692

CHEMBL3278706
0.1510.0050.182Granulocyte macrophage colony stimulating factor agonist

0.128 0.011 CHEMBL3278702

0.124 0.013 CHEMBL3544672

0.123 0.014 CHEMBL3278706

0.104 0.03 CHEMBL3544671

0.182 0.004 CHEMBL1105

0.132 0.01 CHEMBL3544690

0.101 0.034 CHEMBL3544691

0.149 0.005 CHEMBL3544673

0.107 0.027 CHEMBL3544692

CHEMBL1105
0.2270.0870.227Calpain inhibitor

0.226 0.088 CHEMBL3278706

0.18 0.134 CHEMBL1105

0.192 0.122 CHEMBL3544673

0.1570.0190.498Porphobilinogen synthase inhibitor

0.498 0.003 CHEMBL3278706

0.147 0.021 CHEMBL3544671

0.128 0.026 CHEMBL1105

0.191 0.013 CHEMBL3544691

0.34 0.005 CHEMBL3544673

0.104 0.034 CHEMBL3544692

CHEMBL3278706
0.1760.040.209CF transmembrane conductance regulator agonist

0.194 0.025 CHEMBL3278702

0.141 0.094 CHEMBL3544672

0.194 0.025 CHEMBL3278706

0.209 0.017 CHEMBL3544671

0.176 0.04 CHEMBL1105

0.173 0.043 CHEMBL3544690

0.154 0.069 CHEMBL3544691

0.191 0.027 CHEMBL3544673

0.187 0.03 CHEMBL3544692

CHEMBL3544671
0.1830.0460.183MAO inhibitor

0.183 0.046 CHEMBL3278706

0.097 0.094 CHEMBL3544673

0.1650.030.165Falcipain 3 inhibitor

0.126 0.05 CHEMBL3278702

0.103 0.067 CHEMBL3544672

0.145 0.039 CHEMBL3278706

0.111 0.06 CHEMBL3544671

0.117 0.056 CHEMBL1105

0.089 0.082 CHEMBL3544690

0.09 0.081 CHEMBL3544691

0.103 0.068 CHEMBL3544673

0.150.0160.15Acetylcholine release stimulant

0.127 0.038 CHEMBL3278702

0.105 0.077 CHEMBL3544672

0.113 0.061 CHEMBL3278706

0.101 0.086 CHEMBL3544671

0.127 0.038 CHEMBL1105

0.114 0.059 CHEMBL3544690

0.101 0.086 CHEMBL3544673

0.1690.0350.232Farnesoid X receptor antagonist

0.232 0.014 CHEMBL3278706

0.139 0.067 CHEMBL3544671

0.155 0.047 CHEMBL1105

0.134 0.075 CHEMBL3544691

0.205 0.02 CHEMBL3544673

0.121 0.102 CHEMBL3544692

CHEMBL3278706
0.2670.1370.267Calpain 2 inhibitor

0.24 0.157 CHEMBL3278706

0.1670.0370.328Cholesterol synthesis inhibitor

0.309 0.01 CHEMBL3278702

0.233 0.02 CHEMBL3544672

0.204 0.026 CHEMBL3278706

0.328 0.009 CHEMBL3544671

0.309 0.01 CHEMBL1105

0.261 0.016 CHEMBL3544690

0.258 0.017 CHEMBL3544691

0.328 0.009 CHEMBL3544673

0.284 0.013 CHEMBL3544692

CHEMBL3544673
0.1660.0380.218Sphingosine 1-phosphate receptor 5 antagonist

0.17 0.034 CHEMBL3278702

0.132 0.096 CHEMBL3544672

0.183 0.021 CHEMBL3278706

0.179 0.024 CHEMBL3544671

0.208 0.008 CHEMBL1105

0.143 0.073 CHEMBL3544690

0.143 0.073 CHEMBL3544691

0.218 0.006 CHEMBL3544673

0.154 0.055 CHEMBL3544692

CHEMBL3544673
0.1730.0450.173Interleukin 1 antagonist

0.137 0.068 CHEMBL3278702

0.139 0.066 CHEMBL3278706

0.117 0.093 CHEMBL3544671

0.162 0.05 CHEMBL1105

0.136 0.069 CHEMBL3544673

0.1460.020.194NAD(P)H dehydrogenase (quinone) inhibitor

0.095 0.04 CHEMBL3278702

0.119 0.029 CHEMBL3544672

0.194 0.01 CHEMBL3278706

0.123 0.028 CHEMBL3544671

0.146 0.02 CHEMBL1105

0.09 0.043 CHEMBL3544690

0.147 0.02 CHEMBL3544691

0.174 0.013 CHEMBL3544673

0.117 0.03 CHEMBL3544692

CHEMBL3278706
0.1410.0180.246Macrophage migration inhibitory factor inhibitor

0.106 0.032 CHEMBL3278702

0.106 0.032 CHEMBL3544672

0.2 0.008 CHEMBL3278706

0.134 0.02 CHEMBL3544671

0.195 0.008 CHEMBL1105

0.09 0.041 CHEMBL3544690

0.134 0.02 CHEMBL3544691

0.246 0.005 CHEMBL3544673

0.116 0.027 CHEMBL3544692

CHEMBL3544673
0.1680.0450.168Acetylcholinesterase inhibitor

0.12 0.078 CHEMBL3278706

0.1340.0120.149TRPA1 antagonist

0.149 0.009 CHEMBL3278706

0.062 0.041 CHEMBL3544691

CHEMBL3278706
0.190.0710.35P-glycoprotein inhibitor

0.35 0.021 CHEMBL3278702

0.22 0.053 CHEMBL3544672

0.154 0.111 CHEMBL3278706

0.299 0.029 CHEMBL3544671

0.215 0.055 CHEMBL1105

0.223 0.051 CHEMBL3544690

0.182 0.078 CHEMBL3544691

0.171 0.088 CHEMBL3544673

0.183 0.077 CHEMBL3544692

CHEMBL3278702
0.1910.0710.263Hepatoprotectant

0.231 0.05 CHEMBL3278702

0.204 0.063 CHEMBL3544672

0.225 0.052 CHEMBL3278706

0.263 0.04 CHEMBL3544671

0.193 0.07 CHEMBL1105

0.181 0.079 CHEMBL3544690

0.227 0.051 CHEMBL3544691

0.218 0.055 CHEMBL3544673

0.201 0.065 CHEMBL3544692

CHEMBL3544671
0.1960.0770.374Insulin sensitizer

0.367 0.008 CHEMBL3278702

0.263 0.028 CHEMBL3544672

0.208 0.065 CHEMBL3278706

0.363 0.008 CHEMBL3544671

0.374 0.008 CHEMBL1105

0.323 0.012 CHEMBL3544690

0.262 0.028 CHEMBL3544691

0.37 0.008 CHEMBL3544673

0.32 0.012 CHEMBL3544692

CHEMBL1105
0.1310.0130.215Bile acid receptor antagonist

0.111 0.03 CHEMBL3278702

0.106 0.038 CHEMBL3544672

0.156 0.007 CHEMBL3278706

0.121 0.019 CHEMBL3544671

0.176 0.005 CHEMBL1105

0.102 0.045 CHEMBL3544690

0.115 0.024 CHEMBL3544691

0.215 0.004 CHEMBL3544673

0.111 0.029 CHEMBL3544692

CHEMBL3544673
0.2020.0850.293Nitric-oxide synthase stimulant

0.258 0.027 CHEMBL3278702

0.235 0.044 CHEMBL3544672

0.22 0.06 CHEMBL3278706

0.276 0.019 CHEMBL3544671

0.244 0.037 CHEMBL1105

0.274 0.019 CHEMBL3544690

0.252 0.031 CHEMBL3544691

0.261 0.025 CHEMBL3544673

0.293 0.013 CHEMBL3544692

CHEMBL3544692
0.1970.0810.299DNA methylase inhibitor

0.193 0.084 CHEMBL3278702

0.191 0.085 CHEMBL3544672

0.198 0.08 CHEMBL3278706

0.179 0.094 CHEMBL3544671

0.299 0.028 CHEMBL1105

0.151 0.116 CHEMBL3544690

0.177 0.095 CHEMBL3544691

0.286 0.032 CHEMBL3544673

0.138 0.129 CHEMBL3544692

CHEMBL1105
0.1320.0160.166Aromatase inhibitor

0.166 0.011 CHEMBL3278706

0.064 0.039 CHEMBL3544671

0.064 0.039 CHEMBL1105

0.081 0.027 CHEMBL3544673

CHEMBL3278706
0.1530.0370.265-Lipoxygenase inhibitor

0.226 0.02 CHEMBL3278706

0.111 0.056 CHEMBL3544671

0.202 0.024 CHEMBL1105

0.104 0.06 CHEMBL3544691

0.26 0.014 CHEMBL3544673

0.091 0.071 CHEMBL3544692

CHEMBL3544673
0.1580.0420.309Cyclooxygenase 3 inhibitor

0.185 0.025 CHEMBL3278702

0.157 0.043 CHEMBL3544672

0.156 0.043 CHEMBL3278706

0.181 0.027 CHEMBL3544671

0.309 0.005 CHEMBL1105

0.215 0.014 CHEMBL3544690

0.153 0.046 CHEMBL3544691

0.299 0.006 CHEMBL3544673

0.21 0.015 CHEMBL3544692

CHEMBL1105
0.1430.0290.251UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.23 0.012 CHEMBL3278702

0.179 0.019 CHEMBL3544672

0.168 0.022 CHEMBL3278706

0.233 0.011 CHEMBL3544671

0.248 0.01 CHEMBL1105

0.197 0.016 CHEMBL3544690

0.182 0.019 CHEMBL3544691

0.251 0.01 CHEMBL3544673

0.201 0.016 CHEMBL3544692

CHEMBL3544673
0.1520.0390.177Interleukin 1b antagonist

0.177 0.025 CHEMBL3278702

0.138 0.049 CHEMBL3544672

0.132 0.053 CHEMBL3544671

0.177 0.026 CHEMBL1105

0.108 0.072 CHEMBL3544690

0.122 0.061 CHEMBL3544673

CHEMBL1105
0.1350.0230.151Thioredoxin inhibitor

0.151 0.017 CHEMBL3278706

0.083 0.076 CHEMBL3544673

CHEMBL3278706
0.1380.0250.17Anabolic

0.117 0.042 CHEMBL3278702

0.119 0.04 CHEMBL3544672

0.17 0.01 CHEMBL3278706

0.149 0.018 CHEMBL3544671

0.122 0.038 CHEMBL1105

0.107 0.053 CHEMBL3544690

0.151 0.017 CHEMBL3544691

0.153 0.016 CHEMBL3544673

0.141 0.023 CHEMBL3544692

CHEMBL3278706
0.1660.0570.183Thiol protease inhibitor

0.183 0.047 CHEMBL3278706

0.127 0.102 CHEMBL3544671

0.132 0.092 CHEMBL3544691

0.132 0.092 CHEMBL3544673

CHEMBL3278706
0.1380.030.196Sphingomyelinase inhibitor

0.196 0.01 CHEMBL3278702

0.154 0.023 CHEMBL3544672

0.095 0.065 CHEMBL3278706

0.138 0.03 CHEMBL3544671

0.138 0.03 CHEMBL1105

0.172 0.017 CHEMBL3544690

0.101 0.058 CHEMBL3544691

0.09 0.073 CHEMBL3544673

0.116 0.044 CHEMBL3544692

CHEMBL3278702
0.1270.0190.236Keratolytic

0.117 0.022 CHEMBL3278702

0.12 0.021 CHEMBL3544672

0.207 0.008 CHEMBL3278706

0.162 0.013 CHEMBL3544671

0.18 0.01 CHEMBL1105

0.111 0.025 CHEMBL3544690

0.166 0.012 CHEMBL3544691

0.236 0.006 CHEMBL3544673

0.152 0.014 CHEMBL3544692

CHEMBL3544673
0.1760.0690.1763C-like protease (Human coronavirus) inhibitor

0.155 0.093 CHEMBL3278702

0.15 0.102 CHEMBL3544672

0.137 0.125 CHEMBL3278706

0.167 0.078 CHEMBL1105

0.16 0.085 CHEMBL3544690

0.142 0.115 CHEMBL3544673

0.137 0.125 CHEMBL3544692

0.1650.0590.26Protein kinase stimulant

0.22 0.035 CHEMBL3278702

0.165 0.058 CHEMBL3544672

0.201 0.041 CHEMBL3278706

0.241 0.029 CHEMBL3544671

0.24 0.029 CHEMBL1105

0.176 0.052 CHEMBL3544690

0.182 0.049 CHEMBL3544691

0.26 0.024 CHEMBL3544673

0.194 0.044 CHEMBL3544692

CHEMBL3544673
0.1170.0150.117T cell inhibitor

0.114 0.016 CHEMBL3278706

0.08 0.065 CHEMBL1105

0.078 0.072 CHEMBL3544673

0.1250.0250.127CYP2A6 inhibitor

0.066 0.065 CHEMBL3544672

0.127 0.024 CHEMBL3278706

0.078 0.05 CHEMBL3544671

0.082 0.047 CHEMBL3544691

0.068 0.061 CHEMBL3544673

0.069 0.06 CHEMBL3544692

CHEMBL3278706
0.1480.0480.178Cathepsin H inhibitor

0.165 0.037 CHEMBL3278702

0.161 0.039 CHEMBL3544672

0.147 0.049 CHEMBL3278706

0.17 0.034 CHEMBL3544671

0.131 0.062 CHEMBL1105

0.173 0.033 CHEMBL3544690

0.166 0.036 CHEMBL3544691

0.136 0.057 CHEMBL3544673

0.178 0.03 CHEMBL3544692

CHEMBL3544692
0.1990.10.268Antiamyloidogenic

0.204 0.097 CHEMBL3278702

0.209 0.094 CHEMBL3278706

0.2 0.099 CHEMBL3544671

0.268 0.063 CHEMBL1105

0.264 0.065 CHEMBL3544673

CHEMBL1105
0.1260.0280.218Carbonic anhydrase XIII inhibitor

0.194 0.015 CHEMBL3278702

0.11 0.033 CHEMBL3544672

0.162 0.019 CHEMBL3278706

0.218 0.012 CHEMBL3544671

0.18 0.017 CHEMBL1105

0.108 0.034 CHEMBL3544690

0.128 0.027 CHEMBL3544691

0.205 0.013 CHEMBL3544673

0.126 0.028 CHEMBL3544692

CHEMBL3544671
0.1010.0030.119Melatonin receptor 1A agonist

0.059 0.005 CHEMBL3278702

0.04 0.014 CHEMBL3544672

0.035 0.02 CHEMBL3278706

0.119 0.003 CHEMBL1105

0.044 0.01 CHEMBL3544690

0.044 0.01 CHEMBL3544673

CHEMBL1105
0.1040.0090.133Glutamate (mGluR7) antagonist

0.098 0.011 CHEMBL3278702

0.083 0.024 CHEMBL3544672

0.086 0.021 CHEMBL3278706

0.081 0.026 CHEMBL3544671

0.133 0.004 CHEMBL1105

0.089 0.019 CHEMBL3544690

0.066 0.05 CHEMBL3544691

0.115 0.005 CHEMBL3544673

0.072 0.04 CHEMBL3544692

CHEMBL1105
0.1070.0130.182Peroxisome proliferator-activated receptor gamma antagonist

0.144 0.006 CHEMBL3278702

0.099 0.016 CHEMBL3544672

0.101 0.015 CHEMBL3278706

0.12 0.01 CHEMBL3544671

0.182 0.004 CHEMBL1105

0.108 0.012 CHEMBL3544690

0.088 0.025 CHEMBL3544691

0.148 0.006 CHEMBL3544673

0.095 0.019 CHEMBL3544692

CHEMBL1105
0.1090.0160.154Estrogen-related receptor beta agonist

0.107 0.018 CHEMBL3278702

0.099 0.026 CHEMBL3544672

0.137 0.005 CHEMBL3278706

0.125 0.008 CHEMBL3544671

0.129 0.007 CHEMBL1105

0.104 0.02 CHEMBL3544690

0.116 0.012 CHEMBL3544691

0.154 0.004 CHEMBL3544673

0.122 0.009 CHEMBL3544692

CHEMBL3544673
0.1750.0830.289DNA methyltransferase I inhibitor

0.151 0.103 CHEMBL3278702

0.181 0.079 CHEMBL3544672

0.179 0.081 CHEMBL3278706

0.142 0.113 CHEMBL3544671

0.289 0.03 CHEMBL1105

0.168 0.088 CHEMBL3544691

0.28 0.034 CHEMBL3544673

CHEMBL1105
0.1060.0140.106Alpha tubulin antagonist

0.049 0.042 CHEMBL3278702

0.049 0.042 CHEMBL3544672

0.086 0.018 CHEMBL3278706

0.08 0.02 CHEMBL1105

0.065 0.027 CHEMBL3544673

0.2470.1570.465GABA C receptor rho-3 antagonist

0.43 0.049 CHEMBL3278706

0.315 0.106 CHEMBL3544671

0.27 0.138 CHEMBL1105

0.272 0.136 CHEMBL3544691

0.465 0.036 CHEMBL3544673

0.305 0.112 CHEMBL3544692

CHEMBL3544673
0.0990.0090.099Oleamide hydrolase inhibitor

0.077 0.014 CHEMBL3278702

0.076 0.014 CHEMBL3278706

0.071 0.015 CHEMBL3544671

0.062 0.019 CHEMBL1105

0.057 0.022 CHEMBL3544673

0.1230.0330.164Interleukin 1 beta converting enzyme inhibitor

0.139 0.023 CHEMBL3278706

0.084 0.083 CHEMBL3544671

0.157 0.015 CHEMBL1105

0.084 0.083 CHEMBL3544691

0.164 0.013 CHEMBL3544673

CHEMBL3544673
0.1230.0330.435Alcohol dehydrogenase inhibitor

0.234 0.009 CHEMBL3278702

0.117 0.037 CHEMBL3544672

0.29 0.005 CHEMBL3278706

0.435 0.004 CHEMBL3544671

0.17 0.016 CHEMBL1105

0.128 0.03 CHEMBL3544690

0.243 0.008 CHEMBL3544691

0.357 0.004 CHEMBL3544673

0.268 0.006 CHEMBL3544692

CHEMBL3544671
0.1070.0190.202Leukotriene antagonist

0.166 0.008 CHEMBL3278702

0.1 0.022 CHEMBL3544672

0.115 0.016 CHEMBL3278706

0.161 0.009 CHEMBL3544671

0.202 0.005 CHEMBL1105

0.106 0.019 CHEMBL3544690

0.096 0.023 CHEMBL3544691

0.195 0.006 CHEMBL3544673

0.103 0.021 CHEMBL3544692

CHEMBL1105
0.1540.0670.294Cyclooxygenase inhibitor

0.157 0.064 CHEMBL3278706

0.278 0.021 CHEMBL1105

0.294 0.018 CHEMBL3544673

CHEMBL3544673
0.0940.0070.166Calcium channel P-type blocker

0.164 0.003 CHEMBL3278702

0.12 0.004 CHEMBL3544672

0.06 0.057 CHEMBL3278706

0.092 0.008 CHEMBL3544671

0.104 0.005 CHEMBL1105

0.166 0.003 CHEMBL3544690

0.072 0.024 CHEMBL3544691

0.065 0.039 CHEMBL3544673

0.092 0.008 CHEMBL3544692

CHEMBL3544690
0.1540.0680.204GABA C receptor rho-2 antagonist

0.171 0.05 CHEMBL3278706

0.139 0.09 CHEMBL3544671

0.182 0.041 CHEMBL1105

0.123 0.12 CHEMBL3544690

0.129 0.107 CHEMBL3544691

0.204 0.027 CHEMBL3544673

0.14 0.088 CHEMBL3544692

CHEMBL3544673
0.1150.0290.164Phosphodiesterase 6D inhibitor

0.149 0.01 CHEMBL3278702

0.096 0.061 CHEMBL3544672

0.126 0.02 CHEMBL3278706

0.164 0.007 CHEMBL3544671

0.106 0.042 CHEMBL3544690

0.104 0.044 CHEMBL3544691

0.092 0.071 CHEMBL3544673

0.115 0.03 CHEMBL3544692

CHEMBL3544671
0.0990.0160.104Protease 3C (Human rhinovirus) inhibitor

0.061 0.05 CHEMBL3278702

0.061 0.05 CHEMBL3544672

0.104 0.014 CHEMBL3278706

0.071 0.035 CHEMBL3544671

0.064 0.045 CHEMBL1105

0.071 0.035 CHEMBL3544691

0.075 0.032 CHEMBL3544673

0.065 0.044 CHEMBL3544692

CHEMBL3278706
0.1590.0750.224Thrombolytic

0.145 0.086 CHEMBL3544672

0.21 0.047 CHEMBL3278706

0.125 0.105 CHEMBL3544671

0.183 0.061 CHEMBL1105

0.124 0.106 CHEMBL3544690

0.178 0.063 CHEMBL3544691

0.224 0.041 CHEMBL3544673

0.158 0.076 CHEMBL3544692

CHEMBL3544673
0.1390.0560.139Antibacterial (Helicobacter pylori)

0.115 0.089 CHEMBL3278702

0.135 0.061 CHEMBL3278706

0.114 0.09 CHEMBL3544671

0.128 0.069 CHEMBL1105

0.128 0.07 CHEMBL3544673

0.1810.0980.181Histone acetyltransferase inhibitor

0.173 0.11 CHEMBL3278706

0.147 0.144 CHEMBL1105

0.1250.0420.164Beta glucuronidase inhibitor

0.164 0.019 CHEMBL3278706

0.095 0.079 CHEMBL1105

0.093 0.081 CHEMBL3544691

0.119 0.047 CHEMBL3544673

CHEMBL3278706
0.1110.030.143Glutamate release inhibitor

0.128 0.017 CHEMBL3278702

0.115 0.025 CHEMBL3544672

0.09 0.061 CHEMBL3278706

0.105 0.035 CHEMBL3544671

0.143 0.012 CHEMBL1105

0.128 0.018 CHEMBL3544690

0.096 0.049 CHEMBL3544691

0.116 0.024 CHEMBL3544673

0.105 0.036 CHEMBL3544692

CHEMBL1105
0.1660.0850.219Lipocortins synthesis antagonist

0.171 0.079 CHEMBL3544672

0.193 0.061 CHEMBL3278706

0.139 0.123 CHEMBL3544671

0.202 0.055 CHEMBL1105

0.182 0.069 CHEMBL3544691

0.219 0.045 CHEMBL3544673

0.136 0.128 CHEMBL3544692

CHEMBL3544673
0.1780.0980.419Interleukin antagonist

0.311 0.045 CHEMBL3278702

0.157 0.113 CHEMBL3544672

0.282 0.052 CHEMBL3278706

0.411 0.029 CHEMBL3544671

0.307 0.046 CHEMBL1105

0.205 0.081 CHEMBL3544690

0.24 0.065 CHEMBL3544691

0.419 0.028 CHEMBL3544673

0.301 0.048 CHEMBL3544692

CHEMBL3544673
0.1240.0440.124Butyrylcholinesterase inhibitor

0.083 0.078 CHEMBL3278706

0.1470.0680.218Adenylate cyclase stimulant

0.171 0.034 CHEMBL3278702

0.154 0.057 CHEMBL3544672

0.187 0.021 CHEMBL3278706

0.205 0.011 CHEMBL3544671

0.182 0.024 CHEMBL1105

0.163 0.043 CHEMBL3544690

0.186 0.022 CHEMBL3544691

0.218 0.008 CHEMBL3544673

0.196 0.015 CHEMBL3544692

CHEMBL3544673
0.0910.0120.174Leukotriene B4 antagonist

0.143 0.005 CHEMBL3278702

0.077 0.016 CHEMBL3544672

0.102 0.01 CHEMBL3278706

0.139 0.005 CHEMBL3544671

0.174 0.004 CHEMBL1105

0.075 0.017 CHEMBL3544690

0.075 0.017 CHEMBL3544691

0.171 0.004 CHEMBL3544673

0.073 0.018 CHEMBL3544692

CHEMBL1105
0.1150.0360.141Lanosterol 14 alpha demethylase inhibitor

0.108 0.044 CHEMBL3278702

0.108 0.045 CHEMBL3544672

0.141 0.015 CHEMBL3278706

0.132 0.02 CHEMBL3544671

0.111 0.04 CHEMBL1105

0.092 0.068 CHEMBL3544690

0.132 0.02 CHEMBL3544691

0.136 0.018 CHEMBL3544673

0.118 0.032 CHEMBL3544692

CHEMBL3278706
0.1590.0810.254Neurotensin receptor agonist

0.153 0.095 CHEMBL3278702

0.183 0.047 CHEMBL3278706

0.171 0.061 CHEMBL3544671

0.224 0.026 CHEMBL1105

0.147 0.11 CHEMBL3544690

0.151 0.099 CHEMBL3544691

0.254 0.02 CHEMBL3544673

0.165 0.071 CHEMBL3544692

CHEMBL3544673
0.1990.1210.231Neuropeptide Y2 antagonist

0.191 0.136 CHEMBL3278702

0.231 0.075 CHEMBL3278706

0.226 0.081 CHEMBL3544671

0.18 0.159 CHEMBL3544690

0.197 0.125 CHEMBL3544691

0.189 0.14 CHEMBL3544673

0.215 0.096 CHEMBL3544692

CHEMBL3278706
0.1290.0510.294Interleukin 8 antagonist

0.188 0.016 CHEMBL3278706

0.124 0.056 CHEMBL3544671

0.215 0.01 CHEMBL1105

0.113 0.072 CHEMBL3544691

0.294 0.004 CHEMBL3544673

0.112 0.073 CHEMBL3544692

CHEMBL3544673
0.1320.0570.158Proteasome inhibitor

0.146 0.049 CHEMBL3278702

0.117 0.068 CHEMBL3544672

0.145 0.049 CHEMBL3278706

0.158 0.042 CHEMBL3544671

0.114 0.071 CHEMBL1105

0.143 0.051 CHEMBL3544690

0.132 0.057 CHEMBL3544691

0.129 0.059 CHEMBL3544673

0.156 0.043 CHEMBL3544692

CHEMBL3544671
0.1080.0360.138Ornithine decarboxylase inhibitor

0.112 0.032 CHEMBL3278702

0.106 0.038 CHEMBL3544672

0.133 0.018 CHEMBL3278706

0.129 0.02 CHEMBL3544671

0.12 0.026 CHEMBL1105

0.095 0.05 CHEMBL3544690

0.123 0.024 CHEMBL3544691

0.138 0.015 CHEMBL3544673

0.112 0.032 CHEMBL3544692

CHEMBL3544673
0.1350.0650.169Sphingosine 1-phosphate receptor 2 antagonist

0.14 0.055 CHEMBL3278702

0.149 0.042 CHEMBL3278706

0.149 0.042 CHEMBL3544671

0.16 0.029 CHEMBL1105

0.114 0.111 CHEMBL3544690

0.114 0.112 CHEMBL3544691

0.169 0.022 CHEMBL3544673

0.124 0.088 CHEMBL3544692

CHEMBL3544673
0.1180.0490.15Mediator release inhibitor

0.094 0.077 CHEMBL3278702

0.092 0.079 CHEMBL3544672

0.15 0.029 CHEMBL3278706

0.115 0.052 CHEMBL3544671

0.123 0.045 CHEMBL1105

0.114 0.054 CHEMBL3544691

0.15 0.028 CHEMBL3544673

0.104 0.065 CHEMBL3544692

CHEMBL3544673
0.0730.0040.103Cyclophilin A inhibitor

0.103 0.004 CHEMBL3278706

CHEMBL3278706
0.0960.030.256Peroxisome proliferator-activated receptor gamma agonist

0.156 0.011 CHEMBL3278702

0.171 0.009 CHEMBL3544672

0.09 0.034 CHEMBL3278706

0.149 0.013 CHEMBL3544671

0.256 0.005 CHEMBL1105

0.199 0.007 CHEMBL3544690

0.164 0.01 CHEMBL3544691

0.251 0.005 CHEMBL3544673

0.192 0.007 CHEMBL3544692

CHEMBL1105
0.1470.0820.298Interferon gamma antagonist

0.26 0.026 CHEMBL3278702

0.163 0.063 CHEMBL3544672

0.175 0.053 CHEMBL3278706

0.298 0.02 CHEMBL3544671

0.249 0.029 CHEMBL1105

0.191 0.044 CHEMBL3544690

0.184 0.048 CHEMBL3544691

0.288 0.022 CHEMBL3544673

0.225 0.034 CHEMBL3544692

CHEMBL3544671
0.0840.020.091Exportin-1 inhibitor

0.091 0.014 CHEMBL3278702

0.082 0.022 CHEMBL3544672

0.069 0.047 CHEMBL3278706

0.083 0.021 CHEMBL3544671

0.082 0.022 CHEMBL1105

0.091 0.014 CHEMBL3544690

0.075 0.033 CHEMBL3544691

0.075 0.033 CHEMBL3544673

0.083 0.021 CHEMBL3544692

CHEMBL3544690
0.1770.1130.1775 Hydroxytryptamine 3E antagonist

0.169 0.14 CHEMBL3278706

0.163 0.16 CHEMBL1105

0.172 0.128 CHEMBL3544673

0.0960.0330.096Caspase 7 inhibitor

0.075 0.073 CHEMBL3278706

0.094 0.035 CHEMBL1105

0.078 0.065 CHEMBL3544673

0.070.0060.07Dihydrofolate reductase inhibitor

0.041 0.036 CHEMBL3278702

0.048 0.022 CHEMBL3278706

0.058 0.011 CHEMBL1105

0.042 0.034 CHEMBL3544673

0.0720.0090.108Immunoglobulin Fc receptor antagonist

0.1 0.004 CHEMBL3278702

0.072 0.01 CHEMBL3544672

0.076 0.007 CHEMBL3278706

0.108 0.004 CHEMBL3544671

0.067 0.014 CHEMBL1105

0.087 0.005 CHEMBL3544690

0.075 0.008 CHEMBL3544691

0.07 0.011 CHEMBL3544673

0.092 0.004 CHEMBL3544692

CHEMBL3544671
0.1270.0650.175Papain-like protease (SARS coronavirus) inhibitor

0.141 0.043 CHEMBL3278702

0.137 0.049 CHEMBL3544672

0.162 0.024 CHEMBL3278706

0.174 0.018 CHEMBL3544671

0.123 0.074 CHEMBL1105

0.141 0.044 CHEMBL3544690

0.168 0.021 CHEMBL3544691

0.159 0.027 CHEMBL3544673

0.175 0.018 CHEMBL3544692

CHEMBL3544692
0.0960.0330.481Histidine decarboxylase inhibitor

0.094 0.034 CHEMBL3278702

0.192 0.014 CHEMBL3544672

0.243 0.009 CHEMBL3278706

0.196 0.013 CHEMBL3544671

0.363 0.004 CHEMBL1105

0.101 0.031 CHEMBL3544690

0.336 0.005 CHEMBL3544691

0.481 0.003 CHEMBL3544673

0.211 0.012 CHEMBL3544692

CHEMBL3544673
0.1120.050.261Carbonic anhydrase III inhibitor

0.113 0.05 CHEMBL3278702

0.091 0.073 CHEMBL3544672

0.186 0.019 CHEMBL3278706

0.166 0.023 CHEMBL3544671

0.183 0.019 CHEMBL1105

0.103 0.059 CHEMBL3544690

0.133 0.036 CHEMBL3544691

0.261 0.008 CHEMBL3544673

0.151 0.028 CHEMBL3544692

CHEMBL3544673
0.1180.0560.246Mucolytic

0.164 0.025 CHEMBL3278702

0.166 0.024 CHEMBL3544672

0.122 0.052 CHEMBL3278706

0.154 0.03 CHEMBL3544671

0.246 0.007 CHEMBL1105

0.168 0.023 CHEMBL3544690

0.156 0.029 CHEMBL3544691

0.232 0.008 CHEMBL3544673

0.158 0.028 CHEMBL3544692

CHEMBL1105
0.1910.1290.415Interleukin agonist

0.304 0.046 CHEMBL3278702

0.2 0.121 CHEMBL3544672

0.238 0.088 CHEMBL3278706

0.338 0.032 CHEMBL3544671

0.375 0.023 CHEMBL1105

0.27 0.065 CHEMBL3544690

0.236 0.089 CHEMBL3544691

0.415 0.017 CHEMBL3544673

0.303 0.047 CHEMBL3544692

CHEMBL3544673
0.080.020.08Phosphodiesterase 4A inhibitor
0.1440.0860.216Hexokinase inhibitor

0.171 0.057 CHEMBL3278702

0.172 0.056 CHEMBL3544672

0.185 0.045 CHEMBL3278706

0.196 0.037 CHEMBL3544671

0.189 0.042 CHEMBL1105

0.172 0.056 CHEMBL3544690

0.197 0.037 CHEMBL3544691

0.216 0.027 CHEMBL3544673

0.198 0.036 CHEMBL3544692

CHEMBL3544673
0.0980.0390.131Glutathione S-transferase inhibitor

0.076 0.067 CHEMBL3278702

0.112 0.027 CHEMBL3278706

0.085 0.054 CHEMBL3544671

0.118 0.024 CHEMBL1105

0.131 0.018 CHEMBL3544673

CHEMBL3544673
0.1380.080.166Ca2+-transporting ATPase inhibitor

0.141 0.07 CHEMBL3278702

0.135 0.095 CHEMBL3544672

0.154 0.034 CHEMBL3278706

0.153 0.036 CHEMBL3544671

0.153 0.036 CHEMBL1105

0.139 0.078 CHEMBL3544690

0.146 0.052 CHEMBL3544691

0.166 0.017 CHEMBL3544673

0.151 0.041 CHEMBL3544692

CHEMBL3544673
0.1410.0830.595Peroxidase inhibitor

0.335 0.031 CHEMBL3278702

0.289 0.039 CHEMBL3544672

0.428 0.017 CHEMBL3278706

0.54 0.007 CHEMBL3544671

0.407 0.019 CHEMBL1105

0.341 0.03 CHEMBL3544690

0.505 0.009 CHEMBL3544691

0.595 0.005 CHEMBL3544673

0.544 0.006 CHEMBL3544692

CHEMBL3544673
0.060.0030.061Calcium-independent phospholipase A2 inhibitor

0.036 0.017 CHEMBL3278702

0.04 0.01 CHEMBL3544672

0.061 0.003 CHEMBL3278706

0.036 0.017 CHEMBL3544671

0.033 0.026 CHEMBL1105

0.04 0.01 CHEMBL3544691

0.033 0.027 CHEMBL3544673

CHEMBL3278706
0.0880.0330.145Leukotriene synthesis inhibitor

0.115 0.019 CHEMBL3278702

0.071 0.043 CHEMBL3544672

0.102 0.025 CHEMBL3278706

0.122 0.016 CHEMBL3544671

0.133 0.013 CHEMBL1105

0.069 0.045 CHEMBL3544690

0.076 0.04 CHEMBL3544691

0.145 0.01 CHEMBL3544673

0.074 0.041 CHEMBL3544692

CHEMBL3544673
0.1730.1180.173Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.169 0.122 CHEMBL3278706

0.163 0.127 CHEMBL1105

0.156 0.135 CHEMBL3544673

0.0840.0290.168HIV-1 integrase (Strand Transfer) inhibitor

0.168 0.011 CHEMBL3278706

0.053 0.047 CHEMBL1105

0.084 0.029 CHEMBL3544691

0.104 0.021 CHEMBL3544673

0.053 0.047 CHEMBL3544692

CHEMBL3278706
0.0870.0330.088Calcium channel L-type blocker

0.088 0.032 CHEMBL3278702

0.069 0.054 CHEMBL1105

CHEMBL3278702
0.0860.0330.113Amidase inhibitor

0.071 0.048 CHEMBL3278702

0.079 0.038 CHEMBL3278706

0.071 0.048 CHEMBL3544671

0.113 0.018 CHEMBL1105

0.113 0.018 CHEMBL3544673

CHEMBL3544673
0.0690.0160.071Nicotinic receptor alpha3 subunit antagonist

0.071 0.015 CHEMBL3278706

CHEMBL3278706
0.0950.0430.095Acetylcholine nicotinic antagonist

0.088 0.047 CHEMBL3278706

0.0930.0410.239Catalase inhibitor

0.135 0.03 CHEMBL3278702

0.165 0.023 CHEMBL3544672

0.151 0.026 CHEMBL3278706

0.159 0.024 CHEMBL3544671

0.22 0.012 CHEMBL1105

0.121 0.033 CHEMBL3544690

0.185 0.018 CHEMBL3544691

0.239 0.01 CHEMBL3544673

0.148 0.027 CHEMBL3544692

CHEMBL3544673
0.1030.0520.198Prolactin inhibitor

0.109 0.047 CHEMBL3278702

0.171 0.015 CHEMBL3278706

0.172 0.015 CHEMBL3544671

0.132 0.031 CHEMBL1105

0.09 0.067 CHEMBL3544690

0.128 0.033 CHEMBL3544691

0.198 0.009 CHEMBL3544673

0.148 0.023 CHEMBL3544692

CHEMBL3544673
0.0690.0190.095Ryanodine receptor antagonist

0.07 0.017 CHEMBL3278702

0.065 0.025 CHEMBL3544672

0.056 0.052 CHEMBL3278706

0.056 0.052 CHEMBL3544671

0.095 0.005 CHEMBL1105

0.07 0.017 CHEMBL3544690

0.072 0.015 CHEMBL3544673

0.056 0.052 CHEMBL3544692

CHEMBL1105
0.0580.0070.061Heme oxygenase inhibitor

0.058 0.007 CHEMBL3278702

0.051 0.012 CHEMBL3544672

0.058 0.007 CHEMBL3278706

0.061 0.005 CHEMBL3544671

0.045 0.022 CHEMBL1105

0.049 0.015 CHEMBL3544690

0.053 0.01 CHEMBL3544691

0.047 0.018 CHEMBL3544673

0.051 0.012 CHEMBL3544692

CHEMBL3544671
0.0950.0440.099Transcription factor NF kappa B stimulant

0.078 0.074 CHEMBL3278702

0.078 0.073 CHEMBL3544672

0.099 0.039 CHEMBL3278706

0.079 0.072 CHEMBL3544671

0.079 0.071 CHEMBL3544691

0.078 0.075 CHEMBL3544692

CHEMBL3278706
0.0840.0340.179GABA B receptor agonist

0.096 0.02 CHEMBL3278702

0.089 0.026 CHEMBL3544672

0.102 0.015 CHEMBL3278706

0.108 0.012 CHEMBL3544671

0.152 0.004 CHEMBL1105

0.086 0.03 CHEMBL3544690

0.1 0.016 CHEMBL3544691

0.179 0.004 CHEMBL3544673

0.097 0.019 CHEMBL3544692

CHEMBL3544673
0.1250.0750.209Cyclooxygenase 2 inhibitor

0.12 0.08 CHEMBL3278706

0.201 0.03 CHEMBL1105

0.209 0.028 CHEMBL3544673

CHEMBL3544673
0.0830.0340.162Phosphodiesterase 4B inhibitor

0.162 0.011 CHEMBL1105

0.065 0.05 CHEMBL3544673

CHEMBL1105
0.0910.0420.102Chymotrypsin inhibitor

0.074 0.063 CHEMBL3544672

0.102 0.035 CHEMBL3278706

0.084 0.05 CHEMBL3544691

0.077 0.058 CHEMBL3544673

CHEMBL3278706
0.0560.0080.056Melatonin agonist

0.037 0.018 CHEMBL3278702

0.041 0.014 CHEMBL1105

0.0870.0390.154Estrogen receptor alpha antagonist

0.081 0.047 CHEMBL3278702

0.07 0.069 CHEMBL3544672

0.154 0.011 CHEMBL3278706

0.121 0.018 CHEMBL3544671

0.092 0.033 CHEMBL1105

0.071 0.066 CHEMBL3544690

0.099 0.027 CHEMBL3544691

0.142 0.013 CHEMBL3544673

0.101 0.026 CHEMBL3544692

CHEMBL3278706
0.1020.0540.126Breast cancer-resistant protein inhibitor

0.094 0.061 CHEMBL3278702

0.126 0.035 CHEMBL1105

0.085 0.073 CHEMBL3544690

0.083 0.075 CHEMBL3544673

CHEMBL1105
0.0560.0090.056Melatonin 2 agonist

0.042 0.014 CHEMBL3278702

0.042 0.014 CHEMBL1105

0.034 0.022 CHEMBL3544690

0.0730.0260.073Transcription factor RelA inhibitor

0.063 0.046 CHEMBL3278702

0.066 0.039 CHEMBL3278706

0.071 0.028 CHEMBL1105

0.063 0.047 CHEMBL3544690

0.066 0.037 CHEMBL3544673

0.0650.0190.07Prolyl endopeptidase inhibitor

0.07 0.015 CHEMBL3278706

CHEMBL3278706
0.0690.0230.137Sphingosine kinase 2 inhibitor

0.106 0.006 CHEMBL3278702

0.088 0.012 CHEMBL3544672

0.098 0.008 CHEMBL3278706

0.137 0.004 CHEMBL3544671

0.053 0.042 CHEMBL1105

0.103 0.007 CHEMBL3544690

0.113 0.005 CHEMBL3544691

0.072 0.02 CHEMBL3544673

0.132 0.004 CHEMBL3544692

CHEMBL3544671
0.1570.110.252Psychostimulant

0.218 0.071 CHEMBL3278702

0.167 0.102 CHEMBL3278706

0.231 0.066 CHEMBL3544671

0.239 0.063 CHEMBL1105

0.158 0.11 CHEMBL3544690

0.252 0.058 CHEMBL3544673

0.167 0.102 CHEMBL3544692

CHEMBL3544673
0.0840.0390.114Lipase inhibitor

0.114 0.021 CHEMBL3278706

0.086 0.037 CHEMBL3544671

0.08 0.043 CHEMBL3544673

CHEMBL3278706
0.1360.0910.175Heat shock protein 70 antagonist

0.142 0.069 CHEMBL3278702

0.147 0.054 CHEMBL3278706

0.15 0.045 CHEMBL3544671

0.164 0.023 CHEMBL1105

0.137 0.088 CHEMBL3544690

0.133 0.103 CHEMBL3544691

0.175 0.015 CHEMBL3544673

0.145 0.059 CHEMBL3544692

CHEMBL3544673
0.1160.0720.187DNA polymerase I inhibitor

0.14 0.055 CHEMBL3278702

0.099 0.087 CHEMBL3544672

0.181 0.035 CHEMBL3278706

0.187 0.033 CHEMBL3544671

0.12 0.068 CHEMBL1105

0.094 0.093 CHEMBL3544690

0.145 0.052 CHEMBL3544691

0.174 0.037 CHEMBL3544673

0.143 0.053 CHEMBL3544692

CHEMBL3544671
0.1340.0910.134Cholinergic
0.0820.0380.105Phosphodiesterase VI inhibitor

0.105 0.017 CHEMBL3278702

0.069 0.065 CHEMBL3278706

0.089 0.029 CHEMBL3544671

0.069 0.063 CHEMBL3544690

CHEMBL3278702
0.0520.0080.107Free fatty acid receptor 1 antagonist

0.051 0.008 CHEMBL3278702

0.032 0.025 CHEMBL3544672

0.042 0.014 CHEMBL3278706

0.037 0.019 CHEMBL3544671

0.107 0.003 CHEMBL1105

0.038 0.018 CHEMBL3544690

0.079 0.004 CHEMBL3544673

CHEMBL1105
0.0870.0430.209Phosphodiesterase 4D inhibitor

0.209 0.01 CHEMBL1105

0.137 0.022 CHEMBL3544673

CHEMBL1105
0.0480.0050.048Adenosine uptake inhibitor

0.041 0.01 CHEMBL3278706

0.0630.020.107Lysophosphatidic acid 3 receptor antagonist

0.086 0.007 CHEMBL3278702

0.072 0.013 CHEMBL3544672

0.056 0.027 CHEMBL3278706

0.073 0.012 CHEMBL3544671

0.107 0.004 CHEMBL1105

0.078 0.01 CHEMBL3544690

0.061 0.022 CHEMBL3544691

0.091 0.006 CHEMBL3544673

0.066 0.017 CHEMBL3544692

CHEMBL1105
0.0790.0370.079Neuronal nicotinic receptor antagonist

0.073 0.042 CHEMBL3278706

0.1010.060.286UDP-glucose 4-epimerase inhibitor

0.098 0.063 CHEMBL3278702

0.159 0.026 CHEMBL3544672

0.19 0.019 CHEMBL3278706

0.164 0.025 CHEMBL3544671

0.102 0.059 CHEMBL1105

0.11 0.051 CHEMBL3544690

0.286 0.011 CHEMBL3544691

0.17 0.023 CHEMBL3544673

0.185 0.02 CHEMBL3544692

CHEMBL3544691
0.050.0090.05Melatonin 1 agonist

0.038 0.017 CHEMBL3278702

0.043 0.013 CHEMBL1105

0.031 0.027 CHEMBL3544690

0.0610.020.061Potassium channel Kv1.3 blocker

0.043 0.038 CHEMBL3278706

0.049 0.03 CHEMBL1105

0.0780.0380.217Sphingosine 1-phosphate receptor 4 agonist

0.126 0.015 CHEMBL3278702

0.101 0.025 CHEMBL3278706

0.137 0.011 CHEMBL3544671

0.202 0.004 CHEMBL1105

0.09 0.03 CHEMBL3544690

0.06 0.055 CHEMBL3544691

0.217 0.004 CHEMBL3544673

0.103 0.023 CHEMBL3544692

CHEMBL3544673
0.1120.0730.163Anesthetic local

0.163 0.043 CHEMBL3278702

0.1 0.083 CHEMBL3278706

0.153 0.047 CHEMBL3544671

0.094 0.088 CHEMBL3544690

CHEMBL3278702
0.0520.0130.052Diamine oxidase inhibitor

0.034 0.031 CHEMBL3278706

0.035 0.03 CHEMBL1105

0.1020.0640.102Gastric antisecretory

0.095 0.072 CHEMBL3278702

0.0630.0260.0635 Hydroxytryptamine 7 agonist

0.052 0.048 CHEMBL1105

0.0620.0250.097Leukotriene C antagonist

0.063 0.023 CHEMBL3278702

0.061 0.026 CHEMBL3544672

0.07 0.014 CHEMBL3278706

0.069 0.015 CHEMBL3544671

0.086 0.006 CHEMBL1105

0.059 0.031 CHEMBL3544690

0.067 0.018 CHEMBL3544691

0.097 0.004 CHEMBL3544673

0.064 0.021 CHEMBL3544692

CHEMBL3544673
0.060.0240.06Glucose-6-phosphate translocase inhibitor

0.048 0.042 CHEMBL3544672

0.057 0.027 CHEMBL3278706

0.051 0.037 CHEMBL1105

0.047 0.045 CHEMBL3544673

0.0620.0280.062Elastase inhibitor

0.054 0.036 CHEMBL3278706

0.0940.0590.211Uric acid excretion stimulant

0.162 0.02 CHEMBL3278706

0.138 0.028 CHEMBL1105

0.086 0.071 CHEMBL3544691

0.211 0.012 CHEMBL3544673

0.084 0.074 CHEMBL3544692

CHEMBL3544673
0.0980.0640.098Nitric-oxide synthase inhibitor

0.094 0.07 CHEMBL3278706

0.0510.0170.076Plasmepsin II inhibitor

0.076 0.007 CHEMBL3278702

0.055 0.015 CHEMBL3544672

0.053 0.015 CHEMBL3544671

0.061 0.011 CHEMBL1105

0.059 0.012 CHEMBL3544690

0.038 0.035 CHEMBL3544691

0.042 0.027 CHEMBL3544673

0.041 0.029 CHEMBL3544692

CHEMBL3278702
0.1340.1020.284Growth hormone agonist

0.216 0.053 CHEMBL3278702

0.201 0.058 CHEMBL3278706

0.284 0.035 CHEMBL3544671

0.187 0.064 CHEMBL1105

0.152 0.086 CHEMBL3544690

0.157 0.082 CHEMBL3544691

0.262 0.04 CHEMBL3544673

0.209 0.055 CHEMBL3544692

CHEMBL3544671
0.0530.020.053Histone deacetylase 8 inhibitor

0.052 0.02 CHEMBL3278706

0.0360.0040.036Melatonin receptor 1A antagonist
0.0460.0160.075Squalene synthetase inhibitor

0.034 0.021 CHEMBL3278702

0.068 0.01 CHEMBL3544672

0.053 0.014 CHEMBL3278706

0.037 0.019 CHEMBL3544671

0.034 0.021 CHEMBL1105

0.075 0.009 CHEMBL3544691

0.038 0.019 CHEMBL3544673

CHEMBL3544691
0.1130.0860.383Amylase inhibitor

0.332 0.015 CHEMBL3278702

0.205 0.043 CHEMBL3544672

0.186 0.049 CHEMBL3278706

0.383 0.01 CHEMBL3544671

0.301 0.018 CHEMBL1105

0.25 0.028 CHEMBL3544690

0.243 0.03 CHEMBL3544691

0.352 0.013 CHEMBL3544673

0.29 0.02 CHEMBL3544692

CHEMBL3544671
0.0520.0250.052Cytokine production stimulant

0.047 0.037 CHEMBL3278702

0.052 0.025 CHEMBL3278706

0.049 0.032 CHEMBL3544671

0.0530.0260.053Cholesterol esterase inhibitor

0.049 0.031 CHEMBL3278702

0.049 0.031 CHEMBL3278706

0.049 0.032 CHEMBL3544671

0.045 0.037 CHEMBL1105

0.045 0.038 CHEMBL3544673

0.0350.0080.035CYP24 inhibitor

0.032 0.009 CHEMBL3278702

0.033 0.009 CHEMBL3278706

0.032 0.009 CHEMBL3544671

0.0340.0070.042Hedgehog signaling activator

0.042 0.004 CHEMBL3278702

0.033 0.008 CHEMBL3544672

0.03 0.012 CHEMBL3278706

0.036 0.006 CHEMBL3544671

0.033 0.009 CHEMBL1105

0.037 0.005 CHEMBL3544690

0.029 0.015 CHEMBL3544691

0.028 0.016 CHEMBL3544673

0.032 0.01 CHEMBL3544692

CHEMBL3278702
0.0560.030.103Heparanase inhibitor

0.056 0.03 CHEMBL3278702

0.055 0.034 CHEMBL3544672

0.053 0.037 CHEMBL3278706

0.051 0.044 CHEMBL3544671

0.103 0.004 CHEMBL1105

0.054 0.035 CHEMBL3544690

0.049 0.048 CHEMBL3544691

0.092 0.004 CHEMBL3544673

CHEMBL1105
0.090.0650.256ABCA1 expression enhancer

0.095 0.057 CHEMBL3278702

0.099 0.051 CHEMBL3544672

0.098 0.053 CHEMBL3278706

0.097 0.054 CHEMBL3544671

0.228 0.007 CHEMBL1105

0.1 0.05 CHEMBL3544690

0.102 0.048 CHEMBL3544691

0.256 0.006 CHEMBL3544673

0.103 0.047 CHEMBL3544692

CHEMBL3544673
0.0570.0330.1853(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.094 0.012 CHEMBL3278702

0.068 0.023 CHEMBL3544672

0.125 0.007 CHEMBL3278706

0.185 0.004 CHEMBL3544671

0.069 0.022 CHEMBL1105

0.09 0.013 CHEMBL3544690

0.129 0.006 CHEMBL3544691

0.132 0.006 CHEMBL3544673

0.177 0.004 CHEMBL3544692

CHEMBL3544671
0.0440.0210.049Histone deacetylase 7 inhibitor

0.049 0.019 CHEMBL3278706

CHEMBL3278706
0.0420.0190.119Nicotinic acid receptor agonist

0.119 0.004 CHEMBL3278706

0.051 0.014 CHEMBL3544671

0.039 0.022 CHEMBL1105

0.038 0.023 CHEMBL3544691

0.093 0.005 CHEMBL3544673

CHEMBL3278706
0.0390.0170.0621-Alkyl-2-acetylglycerophosphocholine esterase inhibitor

0.038 0.019 CHEMBL3278702

0.044 0.013 CHEMBL3278706

0.04 0.016 CHEMBL3544671

0.059 0.006 CHEMBL1105

0.062 0.005 CHEMBL3544673

CHEMBL3544673
0.0520.030.099Topoisomerase II beta inhibitor

0.051 0.031 CHEMBL3544672

0.099 0.009 CHEMBL3278706

0.048 0.037 CHEMBL3544671

0.054 0.027 CHEMBL1105

0.089 0.011 CHEMBL3544691

0.097 0.01 CHEMBL3544673

0.069 0.017 CHEMBL3544692

CHEMBL3278706
0.0540.0320.073Vanilloid 2 antagonist

0.07 0.014 CHEMBL3278702

0.057 0.027 CHEMBL3278706

0.073 0.012 CHEMBL3544671

0.049 0.044 CHEMBL1105

0.049 0.043 CHEMBL3544673

CHEMBL3544671
0.0450.0240.205Liver X receptor alpha agonist

0.056 0.015 CHEMBL3278702

0.058 0.014 CHEMBL3278706

0.063 0.011 CHEMBL3544671

0.164 0.004 CHEMBL1105

0.041 0.029 CHEMBL3544690

0.037 0.035 CHEMBL3544691

0.205 0.004 CHEMBL3544673

0.048 0.021 CHEMBL3544692

CHEMBL3544673
0.060.0390.145Sphingosine kinase inhibitor

0.101 0.007 CHEMBL3278702

0.077 0.018 CHEMBL3544672

0.091 0.01 CHEMBL3278706

0.145 0.004 CHEMBL3544671

0.094 0.009 CHEMBL3544690

0.106 0.006 CHEMBL3544691

0.069 0.026 CHEMBL3544673

0.134 0.004 CHEMBL3544692

CHEMBL3544671
0.0810.060.081Inducible nitric-oxide synthase inhibitor

0.077 0.068 CHEMBL3278706

0.0420.020.196Estrogen receptor alpha agonist

0.196 0.005 CHEMBL3278706

0.104 0.008 CHEMBL3544671

0.09 0.01 CHEMBL3544691

0.097 0.009 CHEMBL3544673

0.094 0.009 CHEMBL3544692

CHEMBL3278706
0.0650.0440.093CDC25B inhibitor

0.093 0.019 CHEMBL3278706

0.061 0.05 CHEMBL1105

0.085 0.024 CHEMBL3544673

CHEMBL3278706
0.0720.0510.15Aminopeptidase I inhibitor

0.095 0.03 CHEMBL3278702

0.087 0.036 CHEMBL3544672

0.13 0.017 CHEMBL3278706

0.15 0.013 CHEMBL3544671

0.094 0.031 CHEMBL1105

0.078 0.044 CHEMBL3544690

0.138 0.015 CHEMBL3544691

0.148 0.013 CHEMBL3544673

0.126 0.018 CHEMBL3544692

CHEMBL3544671
0.0790.0580.213Carbonic anhydrase VI inhibitor

0.132 0.025 CHEMBL3278706

0.099 0.04 CHEMBL3544671

0.137 0.024 CHEMBL1105

0.09 0.046 CHEMBL3544691

0.213 0.012 CHEMBL3544673

0.094 0.044 CHEMBL3544692

CHEMBL3544673
0.1070.0860.132Cholinergic antagonist

0.132 0.064 CHEMBL3278706

CHEMBL3278706
0.0880.0680.088MAO B inhibitor

0.088 0.068 CHEMBL3278706

0.0340.0130.034Melatonin antagonist
0.0410.020.05Vanilloid 3 antagonist

0.043 0.015 CHEMBL3278702

0.036 0.035 CHEMBL3544672

0.05 0.008 CHEMBL1105

0.039 0.024 CHEMBL3544690

0.039 0.023 CHEMBL3544673

CHEMBL1105
0.0410.0220.051Nicotinic receptor beta4 subunit antagonist

0.051 0.015 CHEMBL3278706

CHEMBL3278706
0.060.040.08Beta tubulin antagonist

0.08 0.029 CHEMBL1105

CHEMBL1105
0.0860.0660.086Phosphodiesterase I inhibitor
0.0670.0470.067Acetylcholine M5 receptor agonist
0.0480.0290.064Carbonic anhydrase VII inhibitor

0.047 0.032 CHEMBL3544672

0.064 0.017 CHEMBL3278706

0.06 0.019 CHEMBL3544691

0.043 0.036 CHEMBL3544673

0.048 0.029 CHEMBL3544692

CHEMBL3278706
0.0660.0470.066Phosphodiesterase III inhibitor

0.057 0.055 CHEMBL3278702

0.0570.0390.068Pregnane X receptor antagonist

0.054 0.049 CHEMBL3278702

0.056 0.041 CHEMBL3278706

0.068 0.017 CHEMBL1105

0.054 0.049 CHEMBL3544690

0.066 0.02 CHEMBL3544673

CHEMBL1105
0.0450.0270.059Guanylate cyclase inhibitor

0.038 0.037 CHEMBL3278702

0.055 0.016 CHEMBL3544672

0.043 0.029 CHEMBL3278706

0.059 0.013 CHEMBL1105

0.042 0.031 CHEMBL3544690

0.048 0.023 CHEMBL3544691

0.053 0.018 CHEMBL3544673

CHEMBL1105
0.1120.0940.261Bone formation stimulant

0.204 0.035 CHEMBL3278702

0.129 0.077 CHEMBL3544672

0.159 0.052 CHEMBL3278706

0.261 0.023 CHEMBL3544671

0.177 0.043 CHEMBL1105

0.146 0.062 CHEMBL3544690

0.156 0.055 CHEMBL3544691

0.239 0.027 CHEMBL3544673

0.178 0.043 CHEMBL3544692

CHEMBL3544671
0.0640.0470.064Histone deacetylase inhibitor

0.064 0.048 CHEMBL3278706

0.0690.0510.105Secretase beta inhibitor

0.105 0.016 CHEMBL3278702

0.072 0.046 CHEMBL3544672

0.098 0.019 CHEMBL3544671

0.091 0.024 CHEMBL3544690

0.067 0.055 CHEMBL3544691

0.086 0.029 CHEMBL3544692

CHEMBL3278702
0.0940.0780.241Adenylate kinase inhibitor

0.096 0.075 CHEMBL3278702

0.127 0.038 CHEMBL3544672

0.137 0.032 CHEMBL3278706

0.125 0.04 CHEMBL3544671

0.171 0.02 CHEMBL1105

0.096 0.074 CHEMBL3544690

0.173 0.02 CHEMBL3544691

0.241 0.011 CHEMBL3544673

0.126 0.039 CHEMBL3544692

CHEMBL3544673
0.0950.0790.133Toll-Like receptor 4 antagonist

0.123 0.041 CHEMBL3278702

0.112 0.052 CHEMBL3544672

0.107 0.059 CHEMBL3278706

0.129 0.035 CHEMBL3544671

0.126 0.038 CHEMBL1105

0.113 0.051 CHEMBL3544690

0.117 0.046 CHEMBL3544691

0.133 0.032 CHEMBL3544673

0.118 0.045 CHEMBL3544692

CHEMBL3544673
0.1030.0870.128Caspase 3 inhibitor

0.12 0.06 CHEMBL3278702

0.114 0.07 CHEMBL3278706

0.124 0.055 CHEMBL3544671

0.124 0.054 CHEMBL1105

0.128 0.049 CHEMBL3544673

CHEMBL3544673
0.020.0040.028Calcium-dependent phospholipase A2 inhibitor

0.028 0.004 CHEMBL3278706

CHEMBL3278706
0.0930.0770.244Expectorant

0.219 0.017 CHEMBL3278702

0.148 0.036 CHEMBL3544672

0.096 0.073 CHEMBL3278706

0.201 0.02 CHEMBL3544671

0.244 0.013 CHEMBL1105

0.175 0.027 CHEMBL3544690

0.134 0.043 CHEMBL3544691

0.225 0.016 CHEMBL3544673

0.16 0.032 CHEMBL3544692

CHEMBL1105
0.0530.0380.053Nicotinic receptor alpha7 subunit antagonist
0.050.0350.213Estrogen agonist

0.213 0.007 CHEMBL3278706

0.125 0.013 CHEMBL3544671

0.104 0.016 CHEMBL3544691

0.157 0.011 CHEMBL3544673

0.104 0.016 CHEMBL3544692

CHEMBL3278706
0.0670.0520.094Elastase 1 inhibitor

0.069 0.049 CHEMBL3278706

0.064 0.055 CHEMBL3544671

0.086 0.03 CHEMBL1105

0.094 0.024 CHEMBL3544673

CHEMBL3544673
0.0480.0330.198Peroxisome proliferator-activated receptor alpha agonist

0.146 0.006 CHEMBL3278702

0.075 0.02 CHEMBL3544672

0.102 0.012 CHEMBL3544671

0.198 0.004 CHEMBL1105

0.109 0.01 CHEMBL3544690

0.044 0.037 CHEMBL3544691

0.142 0.007 CHEMBL3544673

0.074 0.02 CHEMBL3544692

CHEMBL1105
0.1510.1360.514Hypolipemic

0.476 0.014 CHEMBL3278702

0.261 0.063 CHEMBL3544672

0.191 0.101 CHEMBL3278706

0.514 0.011 CHEMBL3544671

0.359 0.033 CHEMBL1105

0.31 0.046 CHEMBL3544690

0.287 0.053 CHEMBL3544691

0.396 0.026 CHEMBL3544673

0.342 0.037 CHEMBL3544692

CHEMBL3544671
0.0550.040.126Beta 1 adrenoreceptor antagonist

0.119 0.007 CHEMBL3278702

0.086 0.014 CHEMBL3544672

0.069 0.027 CHEMBL3278706

0.126 0.006 CHEMBL3544671

0.071 0.025 CHEMBL1105

0.091 0.013 CHEMBL3544690

0.091 0.013 CHEMBL3544691

0.075 0.022 CHEMBL3544673

0.095 0.011 CHEMBL3544692

CHEMBL3544671
0.0190.0040.019Melatonin 2 antagonist
0.0890.0750.122Protease inhibitor

0.11 0.056 CHEMBL3278702

0.118 0.049 CHEMBL3544672

0.095 0.07 CHEMBL3278706

0.113 0.053 CHEMBL3544671

0.109 0.057 CHEMBL3544690

0.122 0.046 CHEMBL3544691

0.112 0.055 CHEMBL3544692

CHEMBL3544691
0.0390.0250.069Leukotriene C4 antagonist

0.04 0.025 CHEMBL3278702

0.046 0.014 CHEMBL3278706

0.044 0.016 CHEMBL3544671

0.059 0.006 CHEMBL1105

0.039 0.026 CHEMBL3544691

0.069 0.004 CHEMBL3544673

0.038 0.031 CHEMBL3544692

CHEMBL3544673
0.0920.0790.221Estrogen receptor beta antagonist

0.089 0.085 CHEMBL3278702

0.205 0.009 CHEMBL3278706

0.156 0.014 CHEMBL3544671

0.104 0.056 CHEMBL1105

0.139 0.019 CHEMBL3544691

0.221 0.008 CHEMBL3544673

0.144 0.017 CHEMBL3544692

CHEMBL3544673
0.1010.0880.123Beta amyloid protein antagonist

0.123 0.064 CHEMBL1105

CHEMBL1105
0.1020.0890.124Acetylcholine antagonist

0.124 0.067 CHEMBL3278706

CHEMBL3278706
0.0210.0090.113G-protein-coupled receptor 120 agonist

0.037 0.004 CHEMBL3278702

0.016 0.013 CHEMBL3544672

0.015 0.014 CHEMBL3278706

0.022 0.008 CHEMBL3544671

0.113 0.003 CHEMBL1105

0.023 0.007 CHEMBL3544690

0.045 0.004 CHEMBL3544673

CHEMBL1105
0.0630.050.143Beta adrenoreceptor antagonist

0.133 0.008 CHEMBL3278702

0.094 0.019 CHEMBL3544672

0.076 0.03 CHEMBL3278706

0.143 0.006 CHEMBL3544671

0.083 0.025 CHEMBL1105

0.106 0.014 CHEMBL3544690

0.103 0.015 CHEMBL3544691

0.092 0.02 CHEMBL3544673

0.116 0.011 CHEMBL3544692

CHEMBL3544671
0.0390.0270.044Histone deacetylase 9 inhibitor

0.044 0.02 CHEMBL3278706

CHEMBL3278706
0.0210.0090.023Antibiotic Anthracycline-like

0.022 0.008 CHEMBL3278702

0.02 0.012 CHEMBL3544672

0.023 0.007 CHEMBL3278706

0.023 0.007 CHEMBL3544671

0.022 0.008 CHEMBL1105

0.019 0.013 CHEMBL3544690

0.02 0.011 CHEMBL3544691

0.022 0.007 CHEMBL3544673

0.02 0.012 CHEMBL3544692

CHEMBL3544671
0.0620.050.14Beta 3 adrenoreceptor antagonist

0.124 0.009 CHEMBL3278702

0.08 0.023 CHEMBL3544672

0.075 0.027 CHEMBL3278706

0.14 0.007 CHEMBL3544671

0.075 0.027 CHEMBL1105

0.106 0.013 CHEMBL3544690

0.095 0.016 CHEMBL3544691

0.087 0.019 CHEMBL3544673

0.123 0.009 CHEMBL3544692

CHEMBL3544671
0.0380.0260.085-Alpha-reductase inhibitor

0.058 0.016 CHEMBL3278706

0.055 0.017 CHEMBL1105

0.08 0.012 CHEMBL3544673

CHEMBL3544673
0.080.0680.133D-Ala-D-Ala ligase inhibitor

0.081 0.066 CHEMBL3278702

0.08 0.067 CHEMBL3544672

0.101 0.028 CHEMBL3278706

0.095 0.036 CHEMBL3544671

0.112 0.018 CHEMBL1105

0.085 0.055 CHEMBL3544690

0.094 0.037 CHEMBL3544691

0.133 0.009 CHEMBL3544673

0.099 0.03 CHEMBL3544692

CHEMBL3544673
0.0340.0220.169Peroxisome proliferator-activated receptor delta agonist

0.098 0.006 CHEMBL3278702

0.043 0.015 CHEMBL3544672

0.053 0.012 CHEMBL3544671

0.169 0.004 CHEMBL1105

0.076 0.008 CHEMBL3544690

0.107 0.005 CHEMBL3544673

0.041 0.017 CHEMBL3544692

CHEMBL1105
0.0790.0680.09Myeloperoxidase inhibitor

0.09 0.048 CHEMBL3278706

0.08 0.068 CHEMBL3544671

0.082 0.064 CHEMBL3544673

CHEMBL3278706
0.0790.0680.111CC chemokine 5 receptor agonist

0.111 0.013 CHEMBL3278706

0.102 0.02 CHEMBL3544671

0.08 0.063 CHEMBL3544691

0.097 0.025 CHEMBL3544673

0.091 0.034 CHEMBL3544692

CHEMBL3278706
0.0490.0380.054Factor III inhibitor

0.054 0.026 CHEMBL3278706

0.049 0.038 CHEMBL1105

0.049 0.038 CHEMBL3544691

0.052 0.03 CHEMBL3544673

CHEMBL3278706
0.0670.0570.179Cathepsin G inhibitor

0.076 0.047 CHEMBL3278702

0.082 0.042 CHEMBL3278706

0.093 0.036 CHEMBL3544671

0.149 0.021 CHEMBL1105

0.068 0.056 CHEMBL3544691

0.179 0.018 CHEMBL3544673

0.074 0.049 CHEMBL3544692

CHEMBL3544673
0.0210.0110.021Melatonin 1 antagonist
0.0550.0460.089Sphingosine 1-phosphate receptor 3 antagonist

0.071 0.025 CHEMBL3278702

0.074 0.022 CHEMBL3278706

0.089 0.012 CHEMBL3544671

0.067 0.029 CHEMBL1105

0.053 0.051 CHEMBL3544690

0.054 0.048 CHEMBL3544691

0.084 0.014 CHEMBL3544673

0.069 0.027 CHEMBL3544692

CHEMBL3544671
0.0310.0210.161Prostaglandin agonist

0.141 0.004 CHEMBL3278702

0.044 0.012 CHEMBL3544672

0.041 0.013 CHEMBL3278706

0.161 0.004 CHEMBL3544671

0.1 0.005 CHEMBL1105

0.054 0.009 CHEMBL3544690

0.052 0.009 CHEMBL3544691

0.12 0.005 CHEMBL3544673

0.07 0.008 CHEMBL3544692

CHEMBL3544671
0.1080.0990.193Nav1.2 sodium channel blocker

0.193 0.037 CHEMBL3278702

0.179 0.043 CHEMBL3544671

0.108 0.099 CHEMBL1105

0.13 0.073 CHEMBL3544690

0.12 0.083 CHEMBL3544692

CHEMBL3278702
0.0810.0720.083Falcipain inhibitor

0.083 0.07 CHEMBL3278706

CHEMBL3278706
0.0390.030.122Dopamine D5 agonist

0.112 0.004 CHEMBL3278706

0.086 0.005 CHEMBL3544671

0.049 0.018 CHEMBL1105

0.068 0.009 CHEMBL3544691

0.122 0.003 CHEMBL3544673

0.084 0.005 CHEMBL3544692

CHEMBL3544673
0.0910.0820.11Glutamate (mGluR7) agonist

0.11 0.042 CHEMBL1105

CHEMBL1105
0.0260.0180.082Sodium/glucose cotransporter 2 inhibitor

0.054 0.005 CHEMBL3278702

0.038 0.009 CHEMBL3544672

0.03 0.013 CHEMBL3278706

0.057 0.005 CHEMBL3544671

0.028 0.015 CHEMBL1105

0.08 0.004 CHEMBL3544690

0.04 0.009 CHEMBL3544691

0.029 0.014 CHEMBL3544673

0.082 0.004 CHEMBL3544692

CHEMBL3544692
0.0850.0770.2Aminopeptidase B inhibitor

0.111 0.058 CHEMBL3278702

0.108 0.059 CHEMBL3544672

0.168 0.031 CHEMBL3278706

0.176 0.028 CHEMBL3544671

0.139 0.043 CHEMBL1105

0.092 0.071 CHEMBL3544690

0.174 0.029 CHEMBL3544691

0.2 0.021 CHEMBL3544673

0.159 0.034 CHEMBL3544692

CHEMBL3544673
0.0420.0350.047Dihydroorotase inhibitor

0.047 0.028 CHEMBL3278706

0.047 0.027 CHEMBL1105

0.047 0.028 CHEMBL3544673

CHEMBL3544673
0.0460.0390.048Cannabinoid CB2 receptor antagonist

0.048 0.038 CHEMBL3278706

CHEMBL3278706
0.0230.0160.058Prostaglandin F2 alpha agonist

0.045 0.005 CHEMBL3278702

0.023 0.016 CHEMBL3544672

0.032 0.008 CHEMBL3278706

0.058 0.004 CHEMBL3544671

0.03 0.009 CHEMBL1105

0.026 0.012 CHEMBL3544690

0.028 0.01 CHEMBL3544691

0.04 0.005 CHEMBL3544673

0.033 0.008 CHEMBL3544692

CHEMBL3544671
0.0250.0180.075Sodium/glucose cotransporter inhibitor

0.049 0.005 CHEMBL3278702

0.031 0.01 CHEMBL3544672

0.029 0.012 CHEMBL3278706

0.054 0.005 CHEMBL3544671

0.026 0.017 CHEMBL1105

0.069 0.004 CHEMBL3544690

0.034 0.009 CHEMBL3544691

0.027 0.014 CHEMBL3544673

0.075 0.004 CHEMBL3544692

CHEMBL3544692
0.0780.0720.08Falcipain 2 inhibitor

0.08 0.07 CHEMBL3278706

CHEMBL3278706
0.1380.1330.287Phospholipase C inhibitor

0.167 0.077 CHEMBL3278702

0.144 0.12 CHEMBL3544672

0.195 0.048 CHEMBL3278706

0.223 0.032 CHEMBL3544671

0.192 0.05 CHEMBL1105

0.146 0.115 CHEMBL3544690

0.187 0.054 CHEMBL3544691

0.287 0.019 CHEMBL3544673

0.19 0.051 CHEMBL3544692

CHEMBL3544673
0.0250.020.025Acid ceramidase inhibitor
0.0540.0490.087Acetylcholine M3 receptor antagonist

0.087 0.023 CHEMBL3278706

CHEMBL3278706
0.0360.0310.036Histone deacetylase class I inhibitor
0.0280.0240.032Thiazolidinedione

0.031 0.017 CHEMBL3544672

0.029 0.022 CHEMBL1105

0.032 0.015 CHEMBL3544690

CHEMBL3544690
0.0980.0940.136Microtubule formation inhibitor

0.133 0.048 CHEMBL3278702

0.132 0.049 CHEMBL3544672

0.121 0.059 CHEMBL3544671

0.134 0.048 CHEMBL1105

0.136 0.046 CHEMBL3544690

0.12 0.06 CHEMBL3544691

0.122 0.058 CHEMBL3544673

0.123 0.057 CHEMBL3544692

CHEMBL3544690
0.0250.0210.06Leukotriene B4 receptor 1 antagonist

0.04 0.012 CHEMBL3278702

0.035 0.015 CHEMBL3278706

0.044 0.009 CHEMBL3544671

0.052 0.006 CHEMBL1105

0.06 0.005 CHEMBL3544673

CHEMBL3544673
0.0290.0260.052Estradiol 17 beta-dehydrogenase 3 inhibitor

0.052 0.01 CHEMBL3278706

0.033 0.021 CHEMBL3544671

0.032 0.023 CHEMBL3544691

0.039 0.016 CHEMBL3544673

0.03 0.025 CHEMBL3544692

CHEMBL3278706
0.030.0260.117ATP citrate lysase inhibitor

0.046 0.009 CHEMBL3278702

0.035 0.017 CHEMBL3544672

0.062 0.005 CHEMBL3278706

0.094 0.004 CHEMBL3544671

0.054 0.007 CHEMBL1105

0.034 0.018 CHEMBL3544690

0.066 0.005 CHEMBL3544691

0.117 0.003 CHEMBL3544673

0.063 0.005 CHEMBL3544692

CHEMBL3544673
0.0630.060.122HIV-1 integrase inhibitor

0.122 0.015 CHEMBL3278706

0.071 0.046 CHEMBL1105

0.083 0.036 CHEMBL3544691

0.12 0.015 CHEMBL3544673

CHEMBL3278706
0.0310.0280.092Fumarate hydratase inhibitor

0.037 0.021 CHEMBL3278702

0.071 0.008 CHEMBL3544672

0.047 0.015 CHEMBL3278706

0.046 0.015 CHEMBL3544671

0.05 0.013 CHEMBL1105

0.045 0.016 CHEMBL3544690

0.092 0.006 CHEMBL3544691

0.063 0.009 CHEMBL3544673

0.056 0.011 CHEMBL3544692

CHEMBL3544691
0.1160.1140.151Acetylcholine M1 receptor antagonist

0.151 0.073 CHEMBL3278706

CHEMBL3278706
0.0880.0860.257Ferrochelatase inhibitor

0.087 0.086 CHEMBL3278702

0.167 0.031 CHEMBL3278706

0.144 0.04 CHEMBL3544671

0.166 0.032 CHEMBL1105

0.092 0.08 CHEMBL3544691

0.257 0.012 CHEMBL3544673

0.101 0.07 CHEMBL3544692

CHEMBL3544673
0.0290.0270.034Sirtuin 2 inhibitor

0.033 0.023 CHEMBL3278706

0.034 0.022 CHEMBL3544673

CHEMBL3544673
0.0510.0490.051Cathepsin L inhibitor
0.0380.0360.1Sphingosine kinase 1 inhibitor

0.067 0.007 CHEMBL3278702

0.04 0.03 CHEMBL3544672

0.055 0.012 CHEMBL3278706

0.1 0.004 CHEMBL3544671

0.05 0.016 CHEMBL3544690

0.053 0.014 CHEMBL3544691

0.039 0.033 CHEMBL3544673

0.066 0.007 CHEMBL3544692

CHEMBL3544671
0.160.1580.248DNA damaging

0.201 0.115 CHEMBL3278702

0.179 0.135 CHEMBL3544672

0.164 0.153 CHEMBL3278706

0.207 0.11 CHEMBL3544671

0.241 0.085 CHEMBL1105

0.184 0.13 CHEMBL3544691

0.248 0.082 CHEMBL3544673

CHEMBL3544673
0.0330.0330.06Tryptophan 5 hydroxylase inhibitor

0.035 0.029 CHEMBL3544672

0.06 0.004 CHEMBL1105

0.056 0.004 CHEMBL3544673

CHEMBL1105
0.0650.0640.065Acetylcholine M4 receptor antagonist
0.050.050.06Epithelial sodium channel blocker

0.055 0.036 CHEMBL3278702

0.051 0.047 CHEMBL3278706

0.06 0.029 CHEMBL3544671

0.05 0.048 CHEMBL1105

0.054 0.039 CHEMBL3544673

CHEMBL3544671
0.0480.0480.049Phosphodiesterase 4C inhibitor

0.049 0.047 CHEMBL1105

CHEMBL1105
0.0270.0280.052Prostaglandin D2 agonist

0.048 0.008 CHEMBL3278702

0.032 0.02 CHEMBL3278706

0.052 0.007 CHEMBL3544671

0.041 0.012 CHEMBL1105

0.045 0.01 CHEMBL3544673

CHEMBL3544671
0.2640.2650.284Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.267 0.261 CHEMBL1105

0.284 0.235 CHEMBL3544673

CHEMBL3544673
0.1060.1080.13DNA repair enzyme inhibitor

0.13 0.055 CHEMBL1105

0.126 0.061 CHEMBL3544673

CHEMBL1105
0.0990.1010.247Estrogen antagonist

0.102 0.093 CHEMBL3278702

0.207 0.012 CHEMBL3278706

0.174 0.017 CHEMBL3544671

0.12 0.055 CHEMBL1105

0.148 0.024 CHEMBL3544691

0.247 0.009 CHEMBL3544673

0.16 0.02 CHEMBL3544692

CHEMBL3544673
0.0450.0470.064Squalene epoxidase inhibitor

0.054 0.027 CHEMBL3278702

0.05 0.035 CHEMBL3278706

0.064 0.017 CHEMBL3544671

0.051 0.032 CHEMBL3544673

0.049 0.036 CHEMBL3544692

CHEMBL3544671
0.1330.1350.246ATPase inhibitor

0.174 0.065 CHEMBL3278702

0.166 0.076 CHEMBL3544672

0.145 0.11 CHEMBL3278706

0.183 0.054 CHEMBL3544671

0.235 0.018 CHEMBL1105

0.175 0.063 CHEMBL3544690

0.175 0.064 CHEMBL3544691

0.246 0.014 CHEMBL3544673

0.184 0.053 CHEMBL3544692

CHEMBL3544673
0.0450.0480.05Human rhinovirus A protease inhibitor

0.05 0.043 CHEMBL3278706

0.048 0.045 CHEMBL3544691

CHEMBL3278706
0.0480.0510.066Matrix metalloproteinase (membrane-type) inhibitor

0.06 0.032 CHEMBL3278702

0.05 0.046 CHEMBL3544671

0.066 0.027 CHEMBL1105

0.054 0.039 CHEMBL3544673

CHEMBL1105
0.0290.0330.137Retinoid X alpha receptor agonist

0.033 0.027 CHEMBL3278702

0.042 0.018 CHEMBL3278706

0.039 0.021 CHEMBL3544671

0.127 0.004 CHEMBL1105

0.137 0.003 CHEMBL3544673

0.031 0.029 CHEMBL3544692

CHEMBL3544673
0.0610.0650.098Glutamate (mGluR6) antagonist

0.063 0.057 CHEMBL3278702

0.07 0.039 CHEMBL3278706

0.067 0.045 CHEMBL3544671

0.091 0.015 CHEMBL1105

0.098 0.011 CHEMBL3544673

0.062 0.061 CHEMBL3544692

CHEMBL3544673
0.0450.0490.218CD45 antagonist

0.054 0.027 CHEMBL3278702

0.049 0.037 CHEMBL3544672

0.057 0.024 CHEMBL3278706

0.069 0.015 CHEMBL3544671

0.129 0.007 CHEMBL1105

0.059 0.022 CHEMBL3544690

0.06 0.021 CHEMBL3544691

0.218 0.004 CHEMBL3544673

0.08 0.012 CHEMBL3544692

CHEMBL3544673
0.0940.0980.121Acetylcholine muscarinic antagonist

0.121 0.066 CHEMBL3278706

CHEMBL3278706
0.0310.0360.077Glutamate (mGluR3) antagonist

0.043 0.017 CHEMBL3278702

0.037 0.025 CHEMBL3278706

0.044 0.017 CHEMBL3544671

0.075 0.005 CHEMBL1105

0.077 0.005 CHEMBL3544673

CHEMBL3544673
0.0180.0230.055Lysophosphatidic acid 1 receptor antagonist

0.03 0.007 CHEMBL3278702

0.02 0.016 CHEMBL3544672

0.055 0.004 CHEMBL1105

0.026 0.009 CHEMBL3544690

0.031 0.006 CHEMBL3544673

CHEMBL1105
0.0410.0460.087Carbonic anhydrase XIV inhibitor

0.07 0.02 CHEMBL3278702

0.05 0.033 CHEMBL3278706

0.084 0.015 CHEMBL3544671

0.073 0.019 CHEMBL1105

0.045 0.038 CHEMBL3544690

0.087 0.015 CHEMBL3544673

0.053 0.03 CHEMBL3544692

CHEMBL3544673
0.0780.0830.105ATPase (Vacuolar H+) inhibitor

0.105 0.033 CHEMBL3278702

0.105 0.033 CHEMBL3544672

0.095 0.047 CHEMBL3544671

0.091 0.054 CHEMBL1105

0.105 0.033 CHEMBL3544690

0.096 0.046 CHEMBL3544691

0.095 0.047 CHEMBL3544692

CHEMBL3544690
0.0220.0280.032Vanilloid 2 agonist

0.032 0.007 CHEMBL3278706

0.03 0.009 CHEMBL3544671

0.031 0.009 CHEMBL3544673

0.025 0.018 CHEMBL3544692

CHEMBL3278706
0.0610.0670.383Glutamate decarboxylase inhibitor

0.079 0.045 CHEMBL3278702

0.087 0.038 CHEMBL3544672

0.151 0.013 CHEMBL3278706

0.162 0.011 CHEMBL3544671

0.182 0.009 CHEMBL1105

0.074 0.05 CHEMBL3544690

0.178 0.009 CHEMBL3544691

0.383 0.003 CHEMBL3544673

0.153 0.012 CHEMBL3544692

CHEMBL3544673
0.0210.0270.035Lysophosphatidic acid receptor 1 agonist

0.034 0.008 CHEMBL3278702

0.023 0.021 CHEMBL3544672

0.033 0.009 CHEMBL3544671

0.035 0.007 CHEMBL1105

0.028 0.013 CHEMBL3544690

0.034 0.008 CHEMBL3544673

0.027 0.015 CHEMBL3544692

CHEMBL1105
0.0580.0640.159Carbonic anhydrase VA inhibitor

0.066 0.051 CHEMBL3278702

0.075 0.041 CHEMBL3278706

0.085 0.033 CHEMBL3544671

0.133 0.015 CHEMBL1105

0.159 0.009 CHEMBL3544673

0.062 0.057 CHEMBL3544692

CHEMBL3544673
0.0290.0350.216Peroxisome proliferator-activated receptor delta antagonist

0.041 0.014 CHEMBL3278702

0.038 0.017 CHEMBL3544672

0.04 0.014 CHEMBL3544671

0.205 0.004 CHEMBL1105

0.054 0.009 CHEMBL3544690

0.037 0.018 CHEMBL3544691

0.216 0.004 CHEMBL3544673

0.054 0.009 CHEMBL3544692

CHEMBL3544673
0.0690.0760.098Sphingosine 1-phosphate receptor antagonist

0.071 0.067 CHEMBL3278702

0.085 0.036 CHEMBL3278706

0.085 0.036 CHEMBL3544671

0.081 0.044 CHEMBL1105

0.098 0.023 CHEMBL3544673

CHEMBL3544673
0.0510.0580.055Acetylcholine M5 receptor antagonist

0.055 0.05 CHEMBL3278706

CHEMBL3278706
0.0440.0510.117Aconitate hydratase inhibitor

0.058 0.028 CHEMBL3278702

0.064 0.023 CHEMBL3544672

0.063 0.023 CHEMBL3278706

0.071 0.018 CHEMBL3544671

0.093 0.01 CHEMBL1105

0.054 0.032 CHEMBL3544690

0.079 0.014 CHEMBL3544691

0.117 0.006 CHEMBL3544673

0.067 0.02 CHEMBL3544692

CHEMBL3544673
0.0360.0440.077Kainate receptor agonist

0.038 0.037 CHEMBL3278702

0.042 0.028 CHEMBL3278706

0.04 0.032 CHEMBL3544671

0.073 0.004 CHEMBL1105

0.077 0.004 CHEMBL3544673

0.038 0.036 CHEMBL3544692

CHEMBL3544673
0.1210.1280.137Pregnane X receptor agonist

0.133 0.092 CHEMBL3278706

0.123 0.12 CHEMBL3544671

0.124 0.118 CHEMBL1105

0.137 0.082 CHEMBL3544673

CHEMBL3544673
0.1150.1230.163Heat shock protein 90 antagonist

0.163 0.061 CHEMBL3278706

CHEMBL3278706
0.0390.0470.053Metalloproteinase-3 inhibitor

0.046 0.038 CHEMBL3278702

0.053 0.03 CHEMBL1105

CHEMBL1105
0.0210.0310.038Nicotinic acid receptor 2 antagonist

0.033 0.01 CHEMBL3278706

0.027 0.018 CHEMBL3544671

0.029 0.014 CHEMBL1105

0.038 0.005 CHEMBL3544673

CHEMBL3544673
0.0380.0480.059Adenylate cyclase 1 inhibitor

0.05 0.026 CHEMBL3278702

0.043 0.037 CHEMBL3278706

0.056 0.02 CHEMBL3544671

0.05 0.026 CHEMBL1105

0.053 0.024 CHEMBL3544690

0.056 0.02 CHEMBL3544673

0.059 0.018 CHEMBL3544692

CHEMBL3544692
0.0630.0730.092Metalloproteinase-9 inhibitor

0.092 0.036 CHEMBL3278702

0.079 0.045 CHEMBL3544671

0.09 0.037 CHEMBL1105

0.068 0.06 CHEMBL3544690

0.077 0.046 CHEMBL3544673

CHEMBL3278702
0.0750.0860.203Triose-phosphate isomerase inhibitor

0.1 0.048 CHEMBL3278702

0.113 0.037 CHEMBL3544672

0.122 0.031 CHEMBL3278706

0.145 0.021 CHEMBL3544671

0.134 0.025 CHEMBL1105

0.098 0.049 CHEMBL3544690

0.166 0.016 CHEMBL3544691

0.203 0.01 CHEMBL3544673

0.143 0.022 CHEMBL3544692

CHEMBL3544673
0.090.1010.152Alkylator

0.134 0.056 CHEMBL3278702

0.111 0.076 CHEMBL3278706

0.152 0.046 CHEMBL3544671

0.126 0.063 CHEMBL1105

0.11 0.078 CHEMBL3544690

0.142 0.051 CHEMBL3544673

0.125 0.063 CHEMBL3544692

CHEMBL3544671
0.0160.0280.12Prostaglandin E2 agonist

0.095 0.004 CHEMBL3278702

0.025 0.015 CHEMBL3544672

0.023 0.016 CHEMBL3278706

0.12 0.004 CHEMBL3544671

0.066 0.005 CHEMBL1105

0.035 0.009 CHEMBL3544690

0.029 0.011 CHEMBL3544691

0.088 0.004 CHEMBL3544673

0.043 0.007 CHEMBL3544692

CHEMBL3544671
0.0120.0230.016Endothelin B receptor antagonist

0.016 0.015 CHEMBL1105

CHEMBL1105
0.0470.0590.133DNA helicase inhibitor

0.052 0.044 CHEMBL3278702

0.053 0.042 CHEMBL3544672

0.053 0.041 CHEMBL3278706

0.051 0.046 CHEMBL3544671

0.125 0.004 CHEMBL1105

0.055 0.036 CHEMBL3544690

0.052 0.043 CHEMBL3544691

0.133 0.003 CHEMBL3544673

0.055 0.037 CHEMBL3544692

CHEMBL3544673
0.020.0330.13Liver X receptor beta antagonist

0.039 0.013 CHEMBL3278706

0.029 0.019 CHEMBL3544671

0.086 0.004 CHEMBL1105

0.13 0.003 CHEMBL3544673

CHEMBL3544673
0.050.0630.114Purinergic P2X1 antagonist

0.061 0.042 CHEMBL3278702

0.083 0.024 CHEMBL3278706

0.091 0.02 CHEMBL3544671

0.077 0.027 CHEMBL1105

0.068 0.034 CHEMBL3544691

0.114 0.013 CHEMBL3544673

0.077 0.027 CHEMBL3544692

CHEMBL3544673
0.0790.0910.117Urease inhibitor

0.102 0.065 CHEMBL3278706

0.086 0.083 CHEMBL3544671

0.103 0.064 CHEMBL1105

0.117 0.048 CHEMBL3544673

CHEMBL3544673
0.030.0430.083Estradiol 17 beta-dehydrogenase inhibitor

0.073 0.015 CHEMBL3278706

0.052 0.023 CHEMBL3544671

0.044 0.028 CHEMBL1105

0.059 0.02 CHEMBL3544691

0.083 0.013 CHEMBL3544673

0.061 0.019 CHEMBL3544692

CHEMBL3544673
0.0240.0370.064Cholesterol ester transfer protein antagonist

0.059 0.005 CHEMBL3278702

0.044 0.01 CHEMBL3544672

0.043 0.01 CHEMBL3544671

0.045 0.01 CHEMBL1105

0.064 0.004 CHEMBL3544690

0.029 0.025 CHEMBL3544691

0.03 0.024 CHEMBL3544673

0.048 0.008 CHEMBL3544692

CHEMBL3544690
0.0350.0490.0573-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.05 0.015 CHEMBL3278706

0.044 0.024 CHEMBL3544671

0.044 0.023 CHEMBL1105

0.057 0.009 CHEMBL3544673

0.04 0.033 CHEMBL3544692

CHEMBL3544673
0.0240.0370.116Retinoid X receptor agonist

0.042 0.021 CHEMBL3278702

0.04 0.022 CHEMBL3278706

0.052 0.017 CHEMBL3544671

0.108 0.004 CHEMBL1105

0.046 0.019 CHEMBL3544690

0.035 0.025 CHEMBL3544691

0.116 0.004 CHEMBL3544673

0.056 0.015 CHEMBL3544692

CHEMBL3544673
0.0350.0490.058Geranyltranstransferase inhibitor

0.048 0.025 CHEMBL3278702

0.051 0.022 CHEMBL3278706

0.058 0.015 CHEMBL3544671

0.045 0.029 CHEMBL1105

0.056 0.017 CHEMBL3544673

0.047 0.027 CHEMBL3544692

CHEMBL3544671
0.010.0240.126Peroxisome proliferator-activated receptor alpha antagonist

0.042 0.009 CHEMBL3278702

0.027 0.013 CHEMBL3544671

0.126 0.004 CHEMBL1105

0.039 0.009 CHEMBL3544690

0.1 0.004 CHEMBL3544673

0.026 0.013 CHEMBL3544692

CHEMBL1105
0.0510.0650.058Lipocortins synthesis agonist

0.058 0.04 CHEMBL3278706

0.056 0.045 CHEMBL3544691

0.057 0.042 CHEMBL3544673

CHEMBL3278706
0.0250.0390.124Liver X receptor beta agonist

0.034 0.021 CHEMBL3278702

0.032 0.025 CHEMBL3278706

0.04 0.015 CHEMBL3544671

0.102 0.005 CHEMBL1105

0.124 0.004 CHEMBL3544673

CHEMBL3544673
0.0330.0470.087Sphingosine 1-phosphate receptor 1 agonist

0.087 0.005 CHEMBL3278702

0.045 0.026 CHEMBL3544672

0.085 0.005 CHEMBL3544671

0.073 0.008 CHEMBL1105

0.068 0.009 CHEMBL3544690

0.044 0.027 CHEMBL3544691

0.072 0.008 CHEMBL3544673

0.067 0.009 CHEMBL3544692

CHEMBL3278702
0.0480.0620.0585 Hydroxytryptamine 2A agonist

0.058 0.049 CHEMBL1105

CHEMBL1105
0.0850.10.191Chelator

0.191 0.026 CHEMBL3278706

0.093 0.088 CHEMBL3544671

0.099 0.078 CHEMBL3544691

0.152 0.035 CHEMBL3544673

CHEMBL3278706
0.0410.0550.111Carbonic anhydrase VB inhibitor

0.057 0.037 CHEMBL3278702

0.075 0.025 CHEMBL3278706

0.094 0.018 CHEMBL3544671

0.066 0.03 CHEMBL1105

0.052 0.043 CHEMBL3544691

0.111 0.014 CHEMBL3544673

0.061 0.034 CHEMBL3544692

CHEMBL3544673
0.020.0360.109Thyroid hormone agonist

0.037 0.008 CHEMBL3278706

0.034 0.009 CHEMBL3544671

0.061 0.004 CHEMBL1105

0.024 0.022 CHEMBL3544691

0.109 0.002 CHEMBL3544673

0.027 0.016 CHEMBL3544692

CHEMBL3544673
0.0140.030.026Estrogen-related receptor gamma agonist

0.026 0.005 CHEMBL3278706

0.021 0.009 CHEMBL3544671

0.017 0.016 CHEMBL3544691

0.026 0.005 CHEMBL3544673

0.019 0.012 CHEMBL3544692

CHEMBL3544673
0.0420.0590.106Argininosuccinate synthase inhibitor

0.087 0.023 CHEMBL3278706

0.061 0.036 CHEMBL1105

0.07 0.03 CHEMBL3544691

0.106 0.018 CHEMBL3544673

CHEMBL3544673
0.0090.0260.031Calcium-sensing receptor antagonist

0.029 0.006 CHEMBL3278702

0.017 0.009 CHEMBL3544672

0.031 0.006 CHEMBL3544671

0.014 0.011 CHEMBL1105

0.027 0.007 CHEMBL3544690

0.017 0.009 CHEMBL3544691

0.014 0.011 CHEMBL3544673

0.03 0.006 CHEMBL3544692

CHEMBL3544671
0.050.0680.174Carbonic anhydrase V inhibitor

0.058 0.056 CHEMBL3278702

0.071 0.042 CHEMBL3278706

0.079 0.036 CHEMBL3544671

0.142 0.016 CHEMBL1105

0.174 0.01 CHEMBL3544673

CHEMBL3544673
0.0320.050.038Leukocyte elastase inhibitor

0.038 0.036 CHEMBL1105

CHEMBL1105
0.0160.0350.036Leukotriene D4 antagonist

0.031 0.015 CHEMBL1105

0.036 0.013 CHEMBL3544673

CHEMBL3544673
0.0930.1120.406Alpha-N-acetylglucosaminidase inhibitor

0.181 0.04 CHEMBL3278702

0.192 0.037 CHEMBL3544672

0.186 0.038 CHEMBL3278706

0.296 0.017 CHEMBL3544671

0.258 0.022 CHEMBL1105

0.206 0.032 CHEMBL3544690

0.312 0.015 CHEMBL3544691

0.406 0.009 CHEMBL3544673

0.333 0.013 CHEMBL3544692

CHEMBL3544673
0.0160.0360.026Retinoid X beta receptor antagonist

0.024 0.008 CHEMBL1105

0.026 0.006 CHEMBL3544673

CHEMBL3544673
0.0620.0820.072S-adenosyl-L-methionine decarboxylase inhibitor

0.068 0.065 CHEMBL1105

0.072 0.054 CHEMBL3544673

CHEMBL3544673
0.0090.0290.085Free fatty acid receptor 1 agonist

0.02 0.01 CHEMBL3278702

0.016 0.014 CHEMBL3544671

0.085 0.004 CHEMBL1105

0.074 0.004 CHEMBL3544673

CHEMBL1105
0.0150.0350.046Leukotriene B4 receptor 2 antagonist

0.027 0.01 CHEMBL3278702

0.034 0.007 CHEMBL3544671

0.036 0.006 CHEMBL1105

0.046 0.005 CHEMBL3544673

CHEMBL3544673
0.0370.0570.102Beta 2 adrenoreceptor antagonist

0.079 0.012 CHEMBL3278702

0.062 0.022 CHEMBL3544672

0.059 0.025 CHEMBL3278706

0.102 0.008 CHEMBL3544671

0.06 0.024 CHEMBL1105

0.073 0.015 CHEMBL3544690

0.077 0.013 CHEMBL3544691

0.075 0.014 CHEMBL3544673

0.09 0.009 CHEMBL3544692

CHEMBL3544671
0.0750.0950.311Creatine kinase inhibitor

0.22 0.008 CHEMBL3278706

0.202 0.01 CHEMBL3544671

0.137 0.03 CHEMBL1105

0.181 0.014 CHEMBL3544691

0.311 0.004 CHEMBL3544673

0.201 0.01 CHEMBL3544692

CHEMBL3544673
0.0640.0850.105Interferon agonist

0.098 0.03 CHEMBL3278702

0.075 0.061 CHEMBL3278706

0.105 0.025 CHEMBL3544671

0.095 0.033 CHEMBL1105

0.078 0.056 CHEMBL3544690

0.102 0.027 CHEMBL3544673

0.084 0.046 CHEMBL3544692

CHEMBL3544671
0.0380.0590.078Glucose-6-phosphate isomerase inhibitor

0.049 0.031 CHEMBL3278702

0.052 0.026 CHEMBL3544672

0.054 0.024 CHEMBL3278706

0.063 0.016 CHEMBL3544671

0.061 0.018 CHEMBL1105

0.048 0.034 CHEMBL3544690

0.067 0.014 CHEMBL3544691

0.078 0.009 CHEMBL3544673

0.061 0.018 CHEMBL3544692

CHEMBL3544673
0.0330.0540.097Sphingosine 1-phosphate receptor agonist

0.097 0.006 CHEMBL3278702

0.042 0.033 CHEMBL3544672

0.089 0.007 CHEMBL3544671

0.092 0.006 CHEMBL1105

0.071 0.011 CHEMBL3544690

0.085 0.008 CHEMBL3544673

0.065 0.013 CHEMBL3544692

CHEMBL3278702
0.0710.0940.08Thioredoxin reductase inhibitor

0.08 0.062 CHEMBL3278702

0.079 0.065 CHEMBL3544671

CHEMBL3278702
0.0460.0690.079Sphingosine 1-phosphate receptor 1 antagonist

0.055 0.039 CHEMBL3278702

0.059 0.031 CHEMBL3278706

0.068 0.02 CHEMBL3544671

0.061 0.028 CHEMBL1105

0.079 0.014 CHEMBL3544673

0.054 0.042 CHEMBL3544692

CHEMBL3544673
0.090.1130.333Cyclooxygenase 1 inhibitor

0.113 0.087 CHEMBL3278706

0.289 0.015 CHEMBL1105

0.138 0.065 CHEMBL3544690

0.333 0.011 CHEMBL3544673

0.156 0.053 CHEMBL3544692

CHEMBL3544673
0.0070.030.012Lysophosphatidic acid receptor 3 agonist

0.012 0.011 CHEMBL3278702

CHEMBL3278702
0.1650.1880.226Transcription factor STAT3 inhibitor

0.216 0.115 CHEMBL3278702

0.175 0.172 CHEMBL3278706

0.226 0.105 CHEMBL3544671

0.187 0.153 CHEMBL1105

0.195 0.14 CHEMBL3544690

0.195 0.141 CHEMBL3544673

0.204 0.129 CHEMBL3544692

CHEMBL3544671
0.0550.0780.088Beta 2 adrenoreceptor agonist

0.071 0.018 CHEMBL3278702

0.07 0.02 CHEMBL3278706

0.088 0.005 CHEMBL3544671

0.062 0.04 CHEMBL1105

0.063 0.038 CHEMBL3544690

0.07 0.019 CHEMBL3544691

0.075 0.012 CHEMBL3544673

0.076 0.012 CHEMBL3544692

CHEMBL3544671
0.050.0740.419Phenylalanine 4-hydroxylase inhibitor

0.147 0.012 CHEMBL3278702

0.084 0.034 CHEMBL3544672

0.194 0.007 CHEMBL3278706

0.419 0.003 CHEMBL3544671

0.139 0.014 CHEMBL1105

0.126 0.016 CHEMBL3544690

0.26 0.005 CHEMBL3544691

0.401 0.003 CHEMBL3544673

0.371 0.003 CHEMBL3544692

CHEMBL3544671
0.0140.0380.019Retinoic acid beta receptor agonist

0.019 0.015 CHEMBL3544673

CHEMBL3544673
0.0570.0810.136Glutamate dehydrogenase inhibitor

0.083 0.042 CHEMBL3544672

0.106 0.028 CHEMBL3278706

0.099 0.031 CHEMBL3544671

0.083 0.042 CHEMBL1105

0.136 0.018 CHEMBL3544691

0.136 0.018 CHEMBL3544673

0.093 0.035 CHEMBL3544692

CHEMBL3544673
0.0650.0890.109Histamine N-methyltransferase inhibitor

0.105 0.041 CHEMBL3278706

0.088 0.058 CHEMBL3544671

0.109 0.038 CHEMBL3544673

CHEMBL3544673
0.0340.0580.052GABA B receptor antagonist

0.04 0.035 CHEMBL3278706

0.043 0.029 CHEMBL1105

0.052 0.018 CHEMBL3544673

CHEMBL3544673
0.0050.030.012Thromboxane agonist

0.012 0.006 CHEMBL3544671

0.01 0.009 CHEMBL3544673

CHEMBL3544671
0.0210.0460.055Lysophosphatidic acid 2 receptor antagonist

0.032 0.019 CHEMBL3278702

0.029 0.023 CHEMBL3544671

0.055 0.008 CHEMBL1105

0.049 0.009 CHEMBL3544673

CHEMBL1105
0.0990.1250.139Nav1.6 sodium channel blocker

0.139 0.068 CHEMBL3278702

0.126 0.086 CHEMBL3544671

0.116 0.102 CHEMBL1105

0.126 0.088 CHEMBL3544690

0.112 0.109 CHEMBL3544692

CHEMBL3278702
0.0590.0850.096Glycine receptor agonist

0.07 0.055 CHEMBL3278706

0.068 0.059 CHEMBL3544671

0.086 0.032 CHEMBL1105

0.096 0.023 CHEMBL3544673

CHEMBL3544673
0.0430.070.133-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.08 0.025 CHEMBL3278702

0.079 0.025 CHEMBL3278706

0.13 0.01 CHEMBL3544671

0.076 0.027 CHEMBL1105

0.065 0.034 CHEMBL3544690

0.071 0.03 CHEMBL3544691

0.125 0.011 CHEMBL3544673

0.109 0.014 CHEMBL3544692

CHEMBL3544671
0.010.0370.035Nicotinic acid receptor 1 antagonist

0.032 0.004 CHEMBL3278706

0.027 0.005 CHEMBL3544671

0.017 0.012 CHEMBL3544691

0.035 0.004 CHEMBL3544673

0.02 0.009 CHEMBL3544692

CHEMBL3544673
0.0080.0350.02Ileal bile acid transport inhibitor

0.018 0.011 CHEMBL3278702

0.02 0.009 CHEMBL3544671

0.017 0.012 CHEMBL1105

0.019 0.01 CHEMBL3544673

CHEMBL3544671
0.0240.0510.087Carnitine palmitoyltransferase inhibitor

0.087 0.004 CHEMBL1105

0.05 0.008 CHEMBL3544673

CHEMBL1105
0.0280.0550.054GABA uptake inhibitor

0.036 0.032 CHEMBL3278706

0.039 0.027 CHEMBL3544671

0.048 0.017 CHEMBL1105

0.054 0.013 CHEMBL3544673

CHEMBL3544673
0.0760.1040.223Xanthine oxidase inhibitor

0.131 0.042 CHEMBL3278702

0.092 0.068 CHEMBL3544672

0.113 0.051 CHEMBL3278706

0.181 0.024 CHEMBL3544671

0.17 0.027 CHEMBL1105

0.121 0.047 CHEMBL3544690

0.135 0.041 CHEMBL3544691

0.223 0.015 CHEMBL3544673

0.171 0.027 CHEMBL3544692

CHEMBL3544673
0.0450.0730.077Matrix metalloproteinase inhibitor

0.075 0.041 CHEMBL3278702

0.06 0.054 CHEMBL3544671

0.077 0.039 CHEMBL1105

0.062 0.051 CHEMBL3544673

CHEMBL1105
0.0280.0560.066Retinoid X receptor antagonist

0.035 0.033 CHEMBL3278706

0.062 0.005 CHEMBL1105

0.066 0.004 CHEMBL3544673

CHEMBL3544673
0.0770.1060.192GABA C receptor rho-1 antagonist

0.096 0.067 CHEMBL3278702

0.106 0.055 CHEMBL3278706

0.124 0.037 CHEMBL3544671

0.152 0.02 CHEMBL1105

0.096 0.068 CHEMBL3544690

0.11 0.05 CHEMBL3544691

0.192 0.009 CHEMBL3544673

0.123 0.037 CHEMBL3544692

CHEMBL3544673
0.0320.0610.052Fructose-1,6-bisphosphatase inhibitor

0.052 0.023 CHEMBL1105

0.049 0.026 CHEMBL3544673

CHEMBL1105
0.0080.0370.015KiSS-1 receptor antagonist

0.015 0.014 CHEMBL3278706

0.015 0.014 CHEMBL3544691

CHEMBL3544691
0.0180.0470.04Calcium-sensing receptor agonist

0.04 0.007 CHEMBL1105

0.026 0.019 CHEMBL3544673

CHEMBL1105
0.0960.1260.296Interleukin 4 antagonist

0.127 0.076 CHEMBL3278702

0.164 0.039 CHEMBL3278706

0.174 0.033 CHEMBL3544671

0.201 0.022 CHEMBL1105

0.146 0.053 CHEMBL3544691

0.296 0.009 CHEMBL3544673

0.148 0.051 CHEMBL3544692

CHEMBL3544673
0.0130.0430.019Caspase 8 inhibitor

0.019 0.016 CHEMBL3544673

CHEMBL3544673
0.0120.0410.046Prostaglandin H2 antagonist

0.024 0.019 CHEMBL3278702

0.026 0.017 CHEMBL3544671

0.045 0.004 CHEMBL1105

0.046 0.004 CHEMBL3544673

CHEMBL3544673
0.0250.0560.055Retinoid X alpha receptor antagonist

0.052 0.005 CHEMBL1105

0.055 0.005 CHEMBL3544673

CHEMBL3544673
0.0190.0510.09Liver X receptor alpha antagonist

0.027 0.025 CHEMBL3278706

0.06 0.005 CHEMBL1105

0.09 0.004 CHEMBL3544673

CHEMBL3544673
0.0230.0550.085Carnitine palmitoyltransferase 1 inhibitor

0.085 0.004 CHEMBL1105

0.048 0.009 CHEMBL3544673

CHEMBL1105
0.0210.0530.046Catechol O-methyltransferase inhibitor

0.046 0.01 CHEMBL3278706

0.041 0.013 CHEMBL3544673

CHEMBL3278706
0.0110.0430.04Estradiol 17 beta-dehydrogenase 1 inhibitor

0.032 0.011 CHEMBL3278706

0.022 0.016 CHEMBL3544671

0.04 0.009 CHEMBL3544673

0.021 0.017 CHEMBL3544692

CHEMBL3544673
0.0430.0760.121Sphingosine 1-phosphate receptor 5 agonist

0.068 0.018 CHEMBL3278702

0.071 0.016 CHEMBL3544671

0.111 0.007 CHEMBL1105

0.055 0.034 CHEMBL3544690

0.121 0.006 CHEMBL3544673

0.056 0.032 CHEMBL3544692

CHEMBL3544673
0.0930.1260.25NADPH oxidase inhibitor

0.234 0.024 CHEMBL1105

0.25 0.021 CHEMBL3544673

CHEMBL3544673
0.0250.0590.039Dihydropteroate synthase inhibitor

0.037 0.031 CHEMBL1105

0.039 0.028 CHEMBL3544673

CHEMBL3544673
0.0210.0540.052Phosphoglycerate kinase inhibitor

0.05 0.014 CHEMBL3278702

0.031 0.03 CHEMBL3544672

0.052 0.013 CHEMBL3544671

0.036 0.023 CHEMBL3544690

0.032 0.028 CHEMBL3544691

0.031 0.03 CHEMBL3544673

0.037 0.022 CHEMBL3544692

CHEMBL3544671
0.0040.0370.063Thyroid hormone beta agonist

0.02 0.004 CHEMBL1105

0.063 0.002 CHEMBL3544673

CHEMBL3544673
0.0110.0450.158Estrogen receptor beta agonist

0.158 0.007 CHEMBL3278706

0.093 0.013 CHEMBL3544671

0.089 0.013 CHEMBL3544691

0.118 0.009 CHEMBL3544673

0.099 0.012 CHEMBL3544692

CHEMBL3278706
0.0690.1030.162NADH dehydrogenase inhibitor

0.101 0.043 CHEMBL3278702

0.098 0.046 CHEMBL3544672

0.094 0.051 CHEMBL3278706

0.126 0.026 CHEMBL3544671

0.129 0.024 CHEMBL1105

0.107 0.037 CHEMBL3544690

0.122 0.028 CHEMBL3544691

0.162 0.015 CHEMBL3544673

0.134 0.022 CHEMBL3544692

CHEMBL3544673
0.0050.0390.093Prostaglandin EP4 agonist

0.059 0.005 CHEMBL3278702

0.013 0.012 CHEMBL3544672

0.08 0.004 CHEMBL3544671

0.073 0.004 CHEMBL1105

0.032 0.007 CHEMBL3544690

0.019 0.009 CHEMBL3544691

0.093 0.004 CHEMBL3544673

0.045 0.005 CHEMBL3544692

CHEMBL3544673
0.0140.0490.043Beta 1 adrenoreceptor agonist

0.029 0.008 CHEMBL3278702

0.021 0.019 CHEMBL3544672

0.022 0.017 CHEMBL3278706

0.043 0.004 CHEMBL3544671

0.023 0.015 CHEMBL1105

0.028 0.009 CHEMBL3544690

0.029 0.009 CHEMBL3544691

0.032 0.007 CHEMBL3544673

0.04 0.005 CHEMBL3544692

CHEMBL3544671
0.0140.0490.02511-Beta-hydroxysteroid dehydrogenase 2 inhibitor

0.025 0.022 CHEMBL3278706

0.025 0.021 CHEMBL3544673

CHEMBL3544673
0.0240.0590.051Estrogen-related receptor beta antagonist

0.048 0.006 CHEMBL3278706

0.046 0.007 CHEMBL3544671

0.041 0.01 CHEMBL3544691

0.051 0.005 CHEMBL3544673

0.046 0.007 CHEMBL3544692

CHEMBL3544673
0.0420.0780.081Neutrophil collagenase inhibitor

0.081 0.031 CHEMBL1105

0.077 0.034 CHEMBL3544673

CHEMBL1105
0.010.0460.083Prostaglandin EP2 agonist

0.066 0.004 CHEMBL3278702

0.02 0.017 CHEMBL3544672

0.083 0.004 CHEMBL3544671

0.044 0.007 CHEMBL1105

0.039 0.009 CHEMBL3544690

0.032 0.012 CHEMBL3544691

0.054 0.005 CHEMBL3544673

0.048 0.006 CHEMBL3544692

CHEMBL3544671
0.0250.0610.084Macrophage elastase inhibitor

0.082 0.012 CHEMBL3278702

0.084 0.011 CHEMBL3544671

0.061 0.018 CHEMBL1105

0.061 0.018 CHEMBL3544673

CHEMBL3544671
0.0260.0630.07Glycine transporter 2 inhibitor

0.041 0.037 CHEMBL3544671

0.049 0.031 CHEMBL1105

0.07 0.021 CHEMBL3544673

CHEMBL3544673
0.0560.0930.163GABA aminotransferase inhibitor

0.092 0.034 CHEMBL3278706

0.097 0.029 CHEMBL3544671

0.114 0.019 CHEMBL1105

0.085 0.04 CHEMBL3544691

0.163 0.006 CHEMBL3544673

0.093 0.032 CHEMBL3544692

CHEMBL3544673
0.010.0480.019Vitamin D receptor agonist

0.015 0.014 CHEMBL3278702

0.019 0.008 CHEMBL3544671

0.017 0.01 CHEMBL3544673

CHEMBL3544671
0.0140.0530.029Endothelin receptor antagonist

0.029 0.018 CHEMBL1105

CHEMBL1105
0.0360.0750.064Dopamine beta hydroxylase inhibitor

0.053 0.025 CHEMBL3278706

0.054 0.023 CHEMBL3544671

0.047 0.037 CHEMBL1105

0.064 0.011 CHEMBL3544673

0.046 0.04 CHEMBL3544692

CHEMBL3544673
0.0350.0740.445Alcohol oxidase inhibitor

0.075 0.026 CHEMBL3278702

0.071 0.028 CHEMBL3544672

0.123 0.014 CHEMBL3278706

0.226 0.005 CHEMBL3544671

0.124 0.013 CHEMBL1105

0.079 0.024 CHEMBL3544690

0.213 0.006 CHEMBL3544691

0.445 0.004 CHEMBL3544673

0.24 0.005 CHEMBL3544692

CHEMBL3544673
0.0440.0830.066Cathepsin E inhibitor

0.066 0.033 CHEMBL3278702

0.056 0.047 CHEMBL3544672

0.063 0.036 CHEMBL3544671

0.062 0.037 CHEMBL3544690

0.059 0.041 CHEMBL3544692

CHEMBL3278702
0.060.10.092Glycine receptor antagonist

0.082 0.053 CHEMBL3278706

0.074 0.067 CHEMBL3544671

0.092 0.04 CHEMBL3544673

CHEMBL3544673
0.0160.0570.022Vitamin D receptor antagonist

0.021 0.018 CHEMBL3278702

0.022 0.015 CHEMBL3544671

CHEMBL3544671
0.0410.0820.088Collagenase 3 inhibitor

0.071 0.031 CHEMBL3278702

0.088 0.02 CHEMBL1105

0.053 0.052 CHEMBL3544673

CHEMBL1105
0.0140.0550.032Neuraminidase (Influenza B) inhibitor

0.026 0.007 CHEMBL3278702

0.032 0.004 CHEMBL3544671

0.024 0.009 CHEMBL3544692

CHEMBL3544671
0.0370.0790.085Beta adrenoreceptor agonist

0.058 0.009 CHEMBL3278702

0.043 0.041 CHEMBL3544672

0.049 0.02 CHEMBL3278706

0.085 0.004 CHEMBL3544671

0.047 0.025 CHEMBL1105

0.048 0.021 CHEMBL3544690

0.053 0.013 CHEMBL3544691

0.06 0.008 CHEMBL3544673

0.063 0.007 CHEMBL3544692

CHEMBL3544671
0.0410.0840.177Phosphofructokinase-1 inhibitor

0.07 0.047 CHEMBL3278702

0.078 0.043 CHEMBL3544672

0.1 0.032 CHEMBL3278706

0.13 0.022 CHEMBL3544671

0.107 0.029 CHEMBL1105

0.065 0.051 CHEMBL3544690

0.14 0.02 CHEMBL3544691

0.177 0.014 CHEMBL3544673

0.123 0.024 CHEMBL3544692

CHEMBL3544673
0.0570.10.084MDM2 inhibitor

0.066 0.051 CHEMBL3278702

0.068 0.043 CHEMBL3544671

0.081 0.019 CHEMBL1105

0.084 0.015 CHEMBL3544673

CHEMBL3544673
0.0210.0650.073HMG CoA reductase inhibitor

0.064 0.004 CHEMBL3278702

0.035 0.022 CHEMBL3544672

0.073 0.004 CHEMBL3544671

0.036 0.02 CHEMBL3544690

0.039 0.015 CHEMBL3544691

0.034 0.025 CHEMBL3544673

0.041 0.014 CHEMBL3544692

CHEMBL3544671
0.0270.0710.056Glutamate (mGluR8) agonist

0.05 0.012 CHEMBL1105

0.056 0.008 CHEMBL3544673

CHEMBL3544673
0.0140.0590.079Prostacyclin antagonist

0.034 0.022 CHEMBL3278702

0.079 0.005 CHEMBL1105

0.038 0.019 CHEMBL3544690

0.072 0.007 CHEMBL3544673

CHEMBL1105
0.0150.0590.023Retinoic acid gamma receptor agonist

0.021 0.02 CHEMBL3544691

0.023 0.015 CHEMBL3544673

CHEMBL3544673
0.010.0560.062Retinoid X beta receptor agonist

0.053 0.005 CHEMBL1105

0.062 0.004 CHEMBL3544673

CHEMBL3544673
0.0230.0680.045Glutamate (mGluR group II) antagonist

0.045 0.02 CHEMBL1105

0.038 0.027 CHEMBL3544673

CHEMBL1105
0.0140.060.067Prostaglandin EP4 antagonist

0.055 0.008 CHEMBL3278702

0.024 0.02 CHEMBL3544672

0.05 0.008 CHEMBL3544671

0.067 0.006 CHEMBL1105

0.034 0.013 CHEMBL3544690

0.023 0.022 CHEMBL3544691

0.062 0.007 CHEMBL3544673

0.031 0.015 CHEMBL3544692

CHEMBL1105
0.0920.1380.151Sphingosine 1-phosphate receptor 2 agonist

0.142 0.031 CHEMBL3278702

0.151 0.025 CHEMBL3544671

0.108 0.079 CHEMBL1105

0.126 0.046 CHEMBL3544690

0.113 0.067 CHEMBL3544673

0.133 0.038 CHEMBL3544692

CHEMBL3544671
0.1510.1980.234RNA-directed DNA polymerase inhibitor

0.201 0.099 CHEMBL3278702

0.193 0.11 CHEMBL3278706

0.234 0.061 CHEMBL3544671

0.197 0.104 CHEMBL1105

0.195 0.107 CHEMBL3544690

0.186 0.122 CHEMBL3544691

0.23 0.064 CHEMBL3544673

0.228 0.066 CHEMBL3544692

CHEMBL3544671
0.0310.0790.041VCAM antagonist

0.041 0.022 CHEMBL1105

0.041 0.021 CHEMBL3544673

CHEMBL3544673
0.0530.1020.097Metalloproteinase-2 inhibitor

0.076 0.057 CHEMBL3278702

0.073 0.06 CHEMBL3544671

0.097 0.04 CHEMBL1105

0.093 0.042 CHEMBL3544673

CHEMBL1105
0.0140.0630.02Thymidine kinase (Herpes simplex virus 2) inhibitor

0.02 0.017 CHEMBL3544671

CHEMBL3544671
0.0060.0560.022Prostacyclin agonist

0.019 0.009 CHEMBL3278702

0.022 0.008 CHEMBL3544671

CHEMBL3544671
0.0290.0790.063AICAR transformylase inhibitor

0.045 0.029 CHEMBL3278706

0.042 0.034 CHEMBL3544671

0.045 0.029 CHEMBL1105

0.063 0.013 CHEMBL3544673

CHEMBL3544673
0.0110.0620.052Kynurenine 3 monooxygenase inhibitor

0.052 0.006 CHEMBL1105

0.033 0.013 CHEMBL3544673

CHEMBL1105
0.0310.0820.041VCAM-1 antagonist

0.041 0.022 CHEMBL1105

0.041 0.021 CHEMBL3544673

CHEMBL3544673
0.0240.0760.087Adenosine deaminase inhibitor

0.076 0.01 CHEMBL3278702

0.045 0.035 CHEMBL3278706

0.087 0.008 CHEMBL3544671

0.047 0.033 CHEMBL1105

0.056 0.025 CHEMBL3544690

0.05 0.03 CHEMBL3544691

0.061 0.02 CHEMBL3544673

0.067 0.015 CHEMBL3544692

CHEMBL3544671
0.0070.0590.046Integrin beta7 antagonist

0.046 0.007 CHEMBL1105

0.032 0.009 CHEMBL3544673

CHEMBL1105
0.0090.0620.041Thyroid hormone alpha agonist

0.029 0.004 CHEMBL1105

0.041 0.003 CHEMBL3544673

CHEMBL3544673
0.1140.1670.198Aryl hydrocarbon receptor agonist

0.198 0.103 CHEMBL1105

0.17 0.121 CHEMBL3544673

CHEMBL1105
0.0190.0720.03Estrogen-related receptor gamma antagonist

0.029 0.018 CHEMBL3278706

0.028 0.021 CHEMBL3544671

0.03 0.017 CHEMBL3544673

CHEMBL3544673
0.0130.0660.028Urotensin II agonist

0.028 0.017 CHEMBL3544673

CHEMBL3544673
0.0760.1310.124Multidrug resistance-associated protein 1 inhibitor

0.124 0.044 CHEMBL1105

0.112 0.059 CHEMBL3544673

CHEMBL1105
0.0680.1230.0783C-Like protease (SARS coronavirus) inhibitor

0.078 0.075 CHEMBL3544691

CHEMBL3544691
0.0210.0760.029Elastase 2B inhibitor

0.029 0.025 CHEMBL1105

CHEMBL1105
0.0210.0760.029Elastase 3B inhibitor

0.029 0.025 CHEMBL1105

CHEMBL1105
0.0210.0760.029Elastase 3A inhibitor

0.029 0.025 CHEMBL1105

CHEMBL1105
0.0670.1230.493GABA C receptor agonist

0.143 0.037 CHEMBL3278706

0.116 0.052 CHEMBL3544671

0.303 0.009 CHEMBL1105

0.103 0.063 CHEMBL3544691

0.493 0.004 CHEMBL3544673

0.112 0.056 CHEMBL3544692

CHEMBL3544673
0.0450.1040.058Caspase 9 inhibitor

0.058 0.053 CHEMBL3544673

CHEMBL3544673
0.0040.0630.013Glutamate (mGluR6) agonist

0.013 0.007 CHEMBL3544673

CHEMBL3544673
0.0040.0640.025Beta 3 adrenoreceptor agonist

0.011 0.009 CHEMBL3278702

0.025 0.004 CHEMBL3544671

0.015 0.006 CHEMBL3544673

0.015 0.005 CHEMBL3544692

CHEMBL3544671
0.0850.1450.155Alkaline phosphatase inhibitor

0.15 0.06 CHEMBL1105

0.155 0.056 CHEMBL3544673

CHEMBL3544673
0.0930.1540.144Anticoagulant

0.121 0.111 CHEMBL1105

0.144 0.086 CHEMBL3544673

CHEMBL3544673
0.0340.0940.111Carbamoyl phosphate synthetase inhibitor

0.054 0.049 CHEMBL3544672

0.066 0.038 CHEMBL3278706

0.079 0.029 CHEMBL3544671

0.073 0.032 CHEMBL1105

0.085 0.026 CHEMBL3544691

0.111 0.018 CHEMBL3544673

0.073 0.032 CHEMBL3544692

CHEMBL3544673
0.1240.1850.283Catenin beta inhibitor

0.152 0.101 CHEMBL3278702

0.18 0.051 CHEMBL3544672

0.156 0.092 CHEMBL3278706

0.173 0.061 CHEMBL3544671

0.242 0.013 CHEMBL1105

0.2 0.032 CHEMBL3544690

0.203 0.03 CHEMBL3544691

0.283 0.007 CHEMBL3544673

0.226 0.017 CHEMBL3544692

CHEMBL3544673
0.0760.1390.122Folate antagonist

0.092 0.081 CHEMBL3278702

0.122 0.037 CHEMBL1105

0.115 0.044 CHEMBL3544673

CHEMBL1105
0.010.0720.059Sphingosine 1-phosphate receptor 3 agonist

0.051 0.015 CHEMBL3278702

0.059 0.012 CHEMBL3544671

0.038 0.023 CHEMBL3544673

0.038 0.022 CHEMBL3544692

CHEMBL3544671
0.0290.0910.073Acyl-CoA dehydrogenase inhibitor

0.051 0.042 CHEMBL3278706

0.066 0.029 CHEMBL3544671

0.07 0.027 CHEMBL3544691

0.073 0.025 CHEMBL3544673

0.063 0.031 CHEMBL3544692

CHEMBL3544673
0.0140.0770.035Plasmepsin I inhibitor

0.035 0.016 CHEMBL3278702

0.034 0.017 CHEMBL3544671

0.029 0.023 CHEMBL3544690

0.027 0.024 CHEMBL3544692

CHEMBL3278702
0.0260.090.098Xanthine dehydrogenase inhibitor

0.051 0.045 CHEMBL3278706

0.068 0.033 CHEMBL3544671

0.075 0.028 CHEMBL1105

0.051 0.045 CHEMBL3544690

0.049 0.047 CHEMBL3544691

0.098 0.016 CHEMBL3544673

0.075 0.027 CHEMBL3544692

CHEMBL3544673
0.0080.0720.017Retinoic acid receptor antagonist

0.017 0.015 CHEMBL3544673

CHEMBL3544673
0.0140.0780.093Liver X receptor antagonist

0.061 0.008 CHEMBL1105

0.093 0.005 CHEMBL3544673

CHEMBL3544673
0.0280.0930.11Plasminogen activator inhibitor antagonist

0.049 0.034 CHEMBL3544672

0.096 0.011 CHEMBL1105

0.054 0.028 CHEMBL3544690

0.052 0.03 CHEMBL3544691

0.11 0.009 CHEMBL3544673

0.059 0.025 CHEMBL3544692

CHEMBL3544673
0.0720.1370.216GABA C receptor antagonist

0.128 0.045 CHEMBL3278706

0.143 0.034 CHEMBL3544671

0.142 0.035 CHEMBL1105

0.121 0.051 CHEMBL3544691

0.216 0.01 CHEMBL3544673

0.139 0.037 CHEMBL3544692

CHEMBL3544673
0.0380.1030.171Antineoplastic antibiotic

0.082 0.056 CHEMBL3278702

0.076 0.06 CHEMBL3544672

0.102 0.045 CHEMBL3544671

0.136 0.034 CHEMBL3544690

0.093 0.049 CHEMBL3544691

0.171 0.026 CHEMBL3544692

CHEMBL3544692
0.0070.0730.153Thyroid hormone alpha antagonist

0.083 0.004 CHEMBL1105

0.153 0.003 CHEMBL3544673

CHEMBL3544673
0.0920.1580.194Diuretic

0.137 0.088 CHEMBL3278706

0.147 0.08 CHEMBL1105

0.143 0.083 CHEMBL3544691

0.194 0.046 CHEMBL3544673

0.133 0.091 CHEMBL3544692

CHEMBL3544673
0.030.0980.066Glutamate (mGluR group III) antagonist

0.066 0.011 CHEMBL1105

0.062 0.012 CHEMBL3544673

CHEMBL1105
0.120.1880.363Immunostimulant

0.274 0.087 CHEMBL3278702

0.218 0.11 CHEMBL3278706

0.363 0.061 CHEMBL3544671

0.198 0.121 CHEMBL1105

0.234 0.103 CHEMBL3544690

0.232 0.104 CHEMBL3544691

0.289 0.082 CHEMBL3544673

0.329 0.07 CHEMBL3544692

CHEMBL3544671
0.0080.0760.021Complement factor D inhibitor

0.021 0.008 CHEMBL1105

0.018 0.013 CHEMBL3544673

CHEMBL1105
0.0080.0770.021Retinoic acid alpha receptor antagonist

0.018 0.017 CHEMBL1105

0.021 0.013 CHEMBL3544673

CHEMBL3544673
0.0050.0740.021Aminopeptidase A inhibitor

0.021 0.01 CHEMBL3544673

CHEMBL3544673
0.0320.1020.122Biliverdin reductase inhibitor

0.055 0.046 CHEMBL3278702

0.063 0.037 CHEMBL3278706

0.094 0.02 CHEMBL3544671

0.072 0.03 CHEMBL1105

0.068 0.034 CHEMBL3544691

0.122 0.013 CHEMBL3544673

0.074 0.029 CHEMBL3544692

CHEMBL3544673
0.0840.1540.137Calcium channel blocker

0.137 0.071 CHEMBL3278702

CHEMBL3278702
0.0210.0920.064Ribonucleoside-diphosphate reductase inhibitor

0.064 0.032 CHEMBL3278706

0.064 0.032 CHEMBL3544671

0.047 0.043 CHEMBL3544691

0.054 0.038 CHEMBL3544673

0.048 0.042 CHEMBL3544692

CHEMBL3544671
0.0610.1320.107MAP kinase kinase 7 inhibitor

0.092 0.021 CHEMBL3278706

0.096 0.017 CHEMBL3544671

0.078 0.052 CHEMBL1105

0.089 0.025 CHEMBL3544691

0.107 0.008 CHEMBL3544673

0.099 0.013 CHEMBL3544692

CHEMBL3544673
0.0420.1130.061Enoyl-[acyl-carrier-protein] reductase inhibitor

0.061 0.041 CHEMBL3278706

0.056 0.054 CHEMBL3544673

CHEMBL3278706
0.0940.1650.168Mannose-6-phosphate isomerase inhibitor

0.125 0.092 CHEMBL3278702

0.122 0.097 CHEMBL3544672

0.126 0.091 CHEMBL3544671

0.167 0.051 CHEMBL1105

0.137 0.077 CHEMBL3544690

0.123 0.096 CHEMBL3544691

0.168 0.05 CHEMBL3544673

0.139 0.075 CHEMBL3544692

CHEMBL3544673
0.0330.1050.059Bombesin 2 receptor antagonist

0.047 0.039 CHEMBL3544671

0.052 0.031 CHEMBL1105

0.059 0.024 CHEMBL3544673

CHEMBL3544673
0.0330.1060.069Androgen agonist

0.062 0.038 CHEMBL3278706

0.069 0.031 CHEMBL3544673

CHEMBL3544673
0.0550.1290.102Topoisomerase I inhibitor

0.102 0.068 CHEMBL3278706

0.1 0.07 CHEMBL3544673

0.09 0.079 CHEMBL3544692

CHEMBL3278706
0.040.1130.088Na+ K+ transporting ATPase inhibitor

0.068 0.062 CHEMBL3278706

0.081 0.049 CHEMBL3544671

0.082 0.048 CHEMBL3544691

0.085 0.046 CHEMBL3544673

0.088 0.043 CHEMBL3544692

CHEMBL3544692
0.020.0940.051Angiotensin AT1 receptor antagonist

0.042 0.029 CHEMBL1105

0.051 0.017 CHEMBL3544673

CHEMBL3544673
0.020.0940.033Ceramide glucosyltransferase inhibitor

0.033 0.031 CHEMBL3544673

CHEMBL3544673
0.0180.0930.04Angiotensin II receptor antagonist

0.031 0.029 CHEMBL1105

0.04 0.015 CHEMBL3544673

CHEMBL3544673
0.0350.110.087Thromboxane synthase inhibitor

0.052 0.043 CHEMBL3544671

0.075 0.014 CHEMBL1105

0.087 0.009 CHEMBL3544673

CHEMBL3544673
0.0440.1190.077Interferon inducer

0.068 0.038 CHEMBL3278702

0.077 0.026 CHEMBL3544671

0.065 0.044 CHEMBL1105

0.074 0.03 CHEMBL3544673

0.062 0.05 CHEMBL3544692

CHEMBL3544671
0.040.1150.059Heat shock protein 90 beta antagonist

0.055 0.048 CHEMBL3278706

0.059 0.041 CHEMBL3544671

0.056 0.047 CHEMBL3544692

CHEMBL3544671
0.0630.1380.122Topoisomerase II inhibitor

0.122 0.065 CHEMBL3278706

0.12 0.067 CHEMBL3544671

0.096 0.09 CHEMBL3544691

0.119 0.067 CHEMBL3544673

CHEMBL3278706
0.1430.2190.31DNA synthesis inhibitor

0.199 0.125 CHEMBL3278702

0.21 0.109 CHEMBL3544672

0.207 0.112 CHEMBL3278706

0.238 0.075 CHEMBL3544671

0.217 0.099 CHEMBL1105

0.252 0.065 CHEMBL3544690

0.252 0.065 CHEMBL3544691

0.262 0.059 CHEMBL3544673

0.31 0.04 CHEMBL3544692

CHEMBL3544692
0.020.0950.066Ribonucleotide reductase inhibitor

0.065 0.034 CHEMBL3278706

0.066 0.033 CHEMBL3544671

0.046 0.045 CHEMBL3544691

0.055 0.039 CHEMBL3544673

0.048 0.044 CHEMBL3544692

CHEMBL3544671
0.0360.1120.117HIV-1 integrase (3'-Processing) inhibitor

0.075 0.036 CHEMBL3278706

0.059 0.048 CHEMBL1105

0.085 0.032 CHEMBL3544691

0.117 0.02 CHEMBL3544673

0.067 0.041 CHEMBL3544692

CHEMBL3544673
0.0250.1020.257Prostaglandin EP2 antagonist

0.237 0.005 CHEMBL3278702

0.179 0.008 CHEMBL3544672

0.257 0.005 CHEMBL3544671

0.189 0.007 CHEMBL1105

0.221 0.005 CHEMBL3544690

0.192 0.007 CHEMBL3544691

0.205 0.006 CHEMBL3544673

0.238 0.005 CHEMBL3544692

CHEMBL3544671
0.0090.0860.054Retinoid X gamma receptor agonist

0.044 0.006 CHEMBL1105

0.054 0.005 CHEMBL3544673

CHEMBL3544673
0.0090.0870.056Prostaglandin EP3 antagonist

0.053 0.009 CHEMBL3278702

0.034 0.018 CHEMBL3544672

0.056 0.009 CHEMBL3544671

0.041 0.013 CHEMBL1105

0.043 0.013 CHEMBL3544690

0.034 0.018 CHEMBL3544691

0.042 0.013 CHEMBL3544673

0.044 0.012 CHEMBL3544692

CHEMBL3544671
0.0060.0840.015Thromboxane A2 agonist

0.015 0.011 CHEMBL3544673

CHEMBL3544673
0.0480.1270.223Adrenaline agonist

0.153 0.014 CHEMBL3278702

0.094 0.041 CHEMBL3278706

0.223 0.005 CHEMBL3544671

0.09 0.045 CHEMBL1105

0.103 0.035 CHEMBL3544690

0.115 0.028 CHEMBL3544691

0.143 0.016 CHEMBL3544673

0.159 0.013 CHEMBL3544692

CHEMBL3544671
0.0090.0880.0335-Alpha-reductase 2 inhibitor

0.021 0.012 CHEMBL1105

0.033 0.009 CHEMBL3544673

CHEMBL3544673
0.0040.0840.015Integrin alpha4beta1 antagonist

0.015 0.011 CHEMBL1105

CHEMBL1105
0.0130.0940.03NMDA 2D receptor antagonist

0.025 0.022 CHEMBL1105

0.03 0.015 CHEMBL3544673

CHEMBL3544673
0.0630.1440.095 Hydroxytryptamine 3A agonist

0.09 0.088 CHEMBL3544673

CHEMBL3544673
0.0150.0960.047Farnesoid X receptor agonist

0.037 0.027 CHEMBL3278702

0.047 0.016 CHEMBL1105

0.041 0.023 CHEMBL3544673

CHEMBL1105
0.020.1020.042Glutamate (mGluR3) agonist

0.035 0.017 CHEMBL1105

0.042 0.008 CHEMBL3544673

CHEMBL3544673
0.0050.0870.064VLA-4 antagonist

0.061 0.011 CHEMBL1105

0.064 0.01 CHEMBL3544673

CHEMBL3544673
0.0090.0920.041Glucagon receptor antagonist

0.026 0.025 CHEMBL3544671

0.031 0.019 CHEMBL1105

0.041 0.013 CHEMBL3544673

CHEMBL3544673
0.0220.1050.082Liver X receptor agonist

0.068 0.014 CHEMBL1105

0.082 0.01 CHEMBL3544673

CHEMBL3544673
0.0180.1030.138NMDA 2A receptor antagonist

0.071 0.024 CHEMBL3278706

0.077 0.021 CHEMBL3544671

0.053 0.035 CHEMBL1105

0.138 0.008 CHEMBL3544673

0.052 0.035 CHEMBL3544692

CHEMBL3544673
0.0390.1240.051Kallikrein 1 inhibitor

0.051 0.049 CHEMBL3544692

CHEMBL3544692
0.0350.1210.059Dihydroorotate oxidase inhibitor

0.055 0.038 CHEMBL3278706

0.059 0.03 CHEMBL3544673

CHEMBL3544673
0.0390.1240.06I kappa B kinase 2 inhibitor

0.06 0.047 CHEMBL3278706

CHEMBL3278706
0.0050.090.042Integrin alpha4beta7 antagonist

0.042 0.006 CHEMBL1105

0.033 0.008 CHEMBL3544673

CHEMBL1105
0.0320.120.065Carbonic anhydrase stimulant

0.056 0.045 CHEMBL1105

0.065 0.036 CHEMBL3544673

CHEMBL3544673
0.0110.1020.059Estradiol 17 beta-dehydrogenase 2 inhibitor

0.048 0.017 CHEMBL3278706

0.041 0.02 CHEMBL3544671

0.044 0.019 CHEMBL3544691

0.059 0.011 CHEMBL3544673

0.052 0.015 CHEMBL3544692

CHEMBL3544673
0.0140.1050.029Retinoid X gamma receptor antagonist

0.027 0.018 CHEMBL1105

0.029 0.015 CHEMBL3544673

CHEMBL3544673
0.0190.1140.103Thromboxane A2 antagonist

0.049 0.037 CHEMBL3278702

0.067 0.023 CHEMBL3544671

0.088 0.011 CHEMBL1105

0.103 0.007 CHEMBL3544673

CHEMBL3544673
0.0130.1110.039Nicotinic acid receptor 2 agonist

0.039 0.021 CHEMBL3544673

CHEMBL3544673
0.0130.1120.113Urate transporter 1 inhibitor

0.081 0.008 CHEMBL1105

0.113 0.005 CHEMBL3544673

CHEMBL3544673
0.0220.1210.043Nerve growth factor antagonist

0.043 0.029 CHEMBL3544673

CHEMBL3544673
0.010.110.017Tryptophan hydroxylase 1 inhibitor

0.017 0.014 CHEMBL1105

0.017 0.013 CHEMBL3544673

CHEMBL3544673
0.0260.1270.064Aminopeptidase microsomal inhibitor

0.064 0.036 CHEMBL3544673

CHEMBL3544673
0.0210.1220.115Thromboxane antagonist

0.052 0.04 CHEMBL3278702

0.072 0.025 CHEMBL3544671

0.097 0.012 CHEMBL1105

0.115 0.007 CHEMBL3544673

CHEMBL3544673
0.0140.1150.241NMDA receptor subunit 3A antagonist

0.044 0.023 CHEMBL3278706

0.086 0.01 CHEMBL1105

0.241 0.004 CHEMBL3544673

CHEMBL3544673
0.020.1220.28NMDA receptor subunit 3B antagonist

0.048 0.026 CHEMBL3278706

0.043 0.031 CHEMBL3544671

0.116 0.009 CHEMBL1105

0.28 0.004 CHEMBL3544673

CHEMBL3544673
0.0380.140.096Topoisomerase II alpha inhibitor

0.067 0.065 CHEMBL3278706

0.096 0.042 CHEMBL3544673

CHEMBL3544673
0.0010.1030.009Mannitol 2-dehydrogenase inhibitor

0.009 0.005 CHEMBL3544691

CHEMBL3544691
0.0050.1080.0175-Alpha-reductase 1 inhibitor

0.017 0.012 CHEMBL3544673

CHEMBL3544673
0.0280.1310.06Cathepsin D inhibitor

0.06 0.034 CHEMBL3278702

0.048 0.044 CHEMBL3544672

0.06 0.034 CHEMBL3544671

0.051 0.04 CHEMBL3544690

0.047 0.046 CHEMBL3544691

0.05 0.041 CHEMBL3544692

CHEMBL3544671
0.0810.1850.125Transcription factor STAT6 inhibitor

0.113 0.073 CHEMBL3278706

0.125 0.051 CHEMBL3544673

CHEMBL3544673
0.050.1540.219Protein-tyrosine phosphatase 1B inhibitor

0.116 0.066 CHEMBL3278702

0.114 0.067 CHEMBL3544672

0.091 0.088 CHEMBL3278706

0.151 0.045 CHEMBL3544671

0.169 0.039 CHEMBL1105

0.128 0.057 CHEMBL3544690

0.147 0.047 CHEMBL3544691

0.219 0.024 CHEMBL3544673

0.169 0.038 CHEMBL3544692

CHEMBL3544673
0.0260.1290.162NMDA 2 receptor antagonist

0.107 0.028 CHEMBL3278706

0.066 0.056 CHEMBL3544671

0.162 0.014 CHEMBL3544673

0.063 0.059 CHEMBL3544692

CHEMBL3544673
0.1190.2240.324Cardiotonic

0.324 0.047 CHEMBL3278702

0.307 0.053 CHEMBL3544671

0.165 0.158 CHEMBL1105

CHEMBL3278702
0.1450.250.297Transcription factor STAT inhibitor

0.253 0.084 CHEMBL3278702

0.297 0.057 CHEMBL3544671

0.191 0.151 CHEMBL3544673

0.19 0.153 CHEMBL3544692

CHEMBL3544671
0.0180.1230.044Aminopeptidase N inhibitor

0.044 0.037 CHEMBL3544673

CHEMBL3544673
0.0430.1480.286NMDA receptor antagonist

0.079 0.067 CHEMBL3278702

0.127 0.032 CHEMBL3278706

0.201 0.014 CHEMBL3544671

0.114 0.038 CHEMBL1105

0.076 0.071 CHEMBL3544691

0.286 0.007 CHEMBL3544673

0.082 0.063 CHEMBL3544692

CHEMBL3544673
0.0620.1690.205AMP-activated protein kinase stimulant

0.125 0.044 CHEMBL3278702

0.153 0.027 CHEMBL3544671

0.169 0.018 CHEMBL1105

0.115 0.054 CHEMBL3544690

0.109 0.06 CHEMBL3544691

0.205 0.01 CHEMBL3544673

0.144 0.032 CHEMBL3544692

CHEMBL3544673
0.0250.1330.123Carnitine palmitoyltransferase 1B inhibitor

0.123 0.004 CHEMBL1105

0.097 0.005 CHEMBL3544673

CHEMBL1105
0.0150.1250.038Oxytocin agonist

0.038 0.033 CHEMBL3278706

0.038 0.034 CHEMBL3544673

CHEMBL3544673
0.0790.190.154Mcl-1 antagonist

0.138 0.103 CHEMBL3278706

0.154 0.086 CHEMBL3544673

CHEMBL3544673
0.0060.120.039NMDA receptor glycine site antagonist

0.039 0.008 CHEMBL3544673

CHEMBL3544673
0.0030.1180.012Thrombopoietin agonist

0.012 0.008 CHEMBL3544673

CHEMBL3544673
0.0130.1280.035Calcitonin receptor agonist

0.035 0.023 CHEMBL3544671

0.031 0.026 CHEMBL3544673

0.034 0.024 CHEMBL3544692

CHEMBL3544671
0.0230.1380.111Neuraminidase inhibitor

0.065 0.038 CHEMBL3278702

0.054 0.051 CHEMBL3278706

0.094 0.018 CHEMBL3544671

0.079 0.026 CHEMBL3544690

0.065 0.037 CHEMBL3544691

0.111 0.012 CHEMBL3544692

CHEMBL3544692
0.0430.1580.06Heme oxygenase stimulant

0.06 0.045 CHEMBL3544673

CHEMBL3544673
0.1620.2790.398Antibacterial

0.234 0.192 CHEMBL3278702

0.281 0.15 CHEMBL3544672

0.275 0.155 CHEMBL3278706

0.324 0.118 CHEMBL3544671

0.308 0.129 CHEMBL3544690

0.371 0.091 CHEMBL3544691

0.286 0.146 CHEMBL3544673

0.398 0.078 CHEMBL3544692

CHEMBL3544692
0.0180.1350.053Mannosidase inhibitor

0.045 0.032 CHEMBL3278702

0.053 0.022 CHEMBL3544671

0.04 0.039 CHEMBL1105

0.041 0.038 CHEMBL3544690

0.048 0.027 CHEMBL3544673

0.049 0.026 CHEMBL3544692

CHEMBL3544671
0.0380.1560.121Androgen antagonist

0.079 0.067 CHEMBL3278702

0.074 0.073 CHEMBL3278706

0.121 0.033 CHEMBL3544671

0.083 0.061 CHEMBL3544692

CHEMBL3544671
0.0240.1470.061Alpha-mannosidase inhibitor

0.054 0.036 CHEMBL3278702

0.061 0.026 CHEMBL3544671

0.052 0.039 CHEMBL1105

0.054 0.036 CHEMBL3544690

0.059 0.028 CHEMBL3544673

0.06 0.026 CHEMBL3544692

CHEMBL3544671
0.0250.1470.042Purinergic P2X4 antagonist

0.042 0.041 CHEMBL3544673

CHEMBL3544673
0.0180.1430.044Retinoic acid alpha receptor agonist

0.038 0.028 CHEMBL1105

0.044 0.02 CHEMBL3544673

CHEMBL3544673
0.070.1950.251Cell adhesion inhibitor

0.251 0.015 CHEMBL1105

0.239 0.016 CHEMBL3544673

CHEMBL1105
0.0120.1370.027ICAM 1 antagonist

0.022 0.018 CHEMBL1105

0.027 0.01 CHEMBL3544673

CHEMBL3544673
0.0050.1310.055Arginase inhibitor

0.055 0.012 CHEMBL3544673

CHEMBL3544673
0.010.1360.094Kainate receptor antagonist

0.053 0.019 CHEMBL1105

0.094 0.008 CHEMBL3544673

CHEMBL3544673
0.0090.1350.061Kainate receptor 2 antagonist

0.043 0.02 CHEMBL1105

0.061 0.011 CHEMBL3544673

CHEMBL3544673
0.1160.2430.84Hypoglycemic

0.419 0.025 CHEMBL3278702

0.364 0.034 CHEMBL3544672

0.467 0.019 CHEMBL3544671

0.398 0.028 CHEMBL1105

0.791 0.004 CHEMBL3544690

0.406 0.027 CHEMBL3544691

0.454 0.02 CHEMBL3544673

0.84 0.004 CHEMBL3544692

CHEMBL3544692
0.0320.1590.051Angiotensin-converting enzyme inhibitor

0.05 0.048 CHEMBL3544671

0.051 0.045 CHEMBL3544673

CHEMBL3544673
0.0080.1360.045HCV NS5B polymerase inhibitor

0.032 0.021 CHEMBL1105

0.045 0.012 CHEMBL3544673

CHEMBL3544673
0.0280.1570.089Adrenaline uptake inhibitor

0.084 0.025 CHEMBL3544672

0.089 0.022 CHEMBL3544691

CHEMBL3544691
0.0140.1440.055HIV-1 protease inhibitor

0.045 0.027 CHEMBL3278702

0.043 0.031 CHEMBL3544672

0.055 0.016 CHEMBL3544671

0.045 0.027 CHEMBL3544690

0.052 0.019 CHEMBL3544691

0.055 0.016 CHEMBL3544692

CHEMBL3544692
0.0190.150.086Opioid delta receptor antagonist

0.077 0.037 CHEMBL3278706

0.056 0.049 CHEMBL3544671

0.086 0.034 CHEMBL3544673

CHEMBL3544673
0.0560.1880.114Protein kinase C gamma inhibitor

0.114 0.058 CHEMBL3544671

0.097 0.083 CHEMBL3544673

CHEMBL3544671
0.0840.2170.124Heat shock protein 90 alpha antagonist

0.124 0.121 CHEMBL3278706

CHEMBL3278706
0.0070.1410.027Glutamate (mGluR1a) agonist

0.027 0.01 CHEMBL3544673

CHEMBL3544673
0.0160.1520.044Growth hormone release inhibitor

0.044 0.026 CHEMBL3544671

0.042 0.029 CHEMBL3544692

CHEMBL3544671
0.0440.180.089Opioid kappa receptor antagonist

0.086 0.05 CHEMBL3278706

0.089 0.046 CHEMBL3544673

CHEMBL3544673
0.0090.1450.038Complement C3a chemotactic receptor antagonist

0.038 0.034 CHEMBL3544673

CHEMBL3544673
0.0160.1530.157NMDA 2C receptor antagonist

0.055 0.052 CHEMBL3278706

0.056 0.052 CHEMBL3544671

0.083 0.023 CHEMBL1105

0.157 0.006 CHEMBL3544673

CHEMBL3544673
0.0060.1420.054Renin inhibitor

0.053 0.016 CHEMBL3544690

0.054 0.015 CHEMBL3544692

CHEMBL3544692
0.0540.1910.186Adenylate cyclase inhibitor

0.098 0.086 CHEMBL3278702

0.099 0.085 CHEMBL3278706

0.157 0.041 CHEMBL3544671

0.129 0.06 CHEMBL1105

0.13 0.059 CHEMBL3544690

0.15 0.045 CHEMBL3544691

0.185 0.029 CHEMBL3544673

0.186 0.028 CHEMBL3544692

CHEMBL3544692
0.0840.2220.437Insulin secretagoues

0.384 0.007 CHEMBL3278702

0.14 0.085 CHEMBL3544672

0.437 0.005 CHEMBL3544671

0.292 0.013 CHEMBL1105

0.195 0.039 CHEMBL3544690

0.146 0.079 CHEMBL3544691

0.322 0.01 CHEMBL3544673

0.206 0.033 CHEMBL3544692

CHEMBL3544671
0.0040.1440.049Integrin alpha4 antagonist

0.048 0.012 CHEMBL1105

0.049 0.011 CHEMBL3544673

CHEMBL3544673
0.0130.1540.045Opioid mu receptor agonist

0.041 0.039 CHEMBL3278706

0.045 0.033 CHEMBL3544673

CHEMBL3544673
0.040.1830.104Opioid antagonist

0.101 0.047 CHEMBL3278706

0.085 0.062 CHEMBL3544671

0.104 0.045 CHEMBL3544673

0.085 0.063 CHEMBL3544692

CHEMBL3544673
0.0150.1580.05RNA-directed RNA polymerase inhibitor

0.033 0.026 CHEMBL1105

0.05 0.013 CHEMBL3544673

CHEMBL3544673
0.0230.1660.083Prostaglandin-E synthase inhibitor

0.063 0.059 CHEMBL1105

0.083 0.037 CHEMBL3544673

CHEMBL3544673
0.0030.1480.014Egl nine homolog 3 inhibitor

0.014 0.006 CHEMBL3544673

CHEMBL3544673
0.0310.1770.077Phospholipase D inhibitor

0.077 0.039 CHEMBL3544673

CHEMBL3544673
0.0690.2150.276Protein-tyrosine phosphatase inhibitor

0.143 0.086 CHEMBL3278702

0.139 0.091 CHEMBL3544672

0.122 0.111 CHEMBL3278706

0.18 0.056 CHEMBL3544671

0.216 0.041 CHEMBL1105

0.15 0.078 CHEMBL3544690

0.173 0.06 CHEMBL3544691

0.276 0.024 CHEMBL3544673

0.191 0.05 CHEMBL3544692

CHEMBL3544673
0.0440.1910.081Antineoplastic alkaloid

0.081 0.064 CHEMBL3544673

CHEMBL3544673
0.0470.1950.071Vanilloid 4 agonist

0.071 0.061 CHEMBL3544671

CHEMBL3544671
0.0330.1830.075Analgesic, opioid

0.075 0.054 CHEMBL3278706

0.075 0.054 CHEMBL3544673

CHEMBL3544673
0.0510.2020.091Protein kinase C zeta inhibitor

0.091 0.063 CHEMBL3544673

CHEMBL3544673
0.0230.1740.058Glutamate (mGluR4) antagonist

0.047 0.025 CHEMBL1105

0.058 0.015 CHEMBL3544673

CHEMBL3544673
0.0030.1550.041Egl nine homolog 1 inhibitor

0.021 0.005 CHEMBL1105

0.041 0.004 CHEMBL3544673

CHEMBL3544673
0.1330.2850.217Alpha-glucosidase inhibitor

0.217 0.208 CHEMBL3544671

CHEMBL3544671
0.0820.2340.278Antimitotic

0.163 0.11 CHEMBL3278702

0.278 0.05 CHEMBL3544690

0.175 0.1 CHEMBL3544692

CHEMBL3544690
0.1530.3060.261Analgesic

0.261 0.173 CHEMBL3278706

CHEMBL3278706
0.0070.1610.03Lysine carboxypeptidase inhibitor

0.03 0.016 CHEMBL3544673

CHEMBL3544673
0.080.2330.225NOS3 expression enhancer

0.165 0.06 CHEMBL3278706

0.195 0.043 CHEMBL3544671

0.132 0.094 CHEMBL3544691

0.225 0.032 CHEMBL3544673

0.163 0.061 CHEMBL3544692

CHEMBL3544673
0.0160.1720.044Integrin alpha2 antagonist

0.044 0.016 CHEMBL1105

0.041 0.019 CHEMBL3544673

CHEMBL1105
0.0520.2090.12Interleukin 5 antagonist

0.101 0.04 CHEMBL1105

0.12 0.024 CHEMBL3544673

CHEMBL3544673
0.0550.2120.166Nav1.1 sodium channel blocker

0.144 0.035 CHEMBL3278702

0.166 0.027 CHEMBL3544671

0.112 0.054 CHEMBL3544690

0.129 0.042 CHEMBL3544692

CHEMBL3544671
0.0340.1930.113CDC25A inhibitor

0.083 0.04 CHEMBL1105

0.113 0.022 CHEMBL3544673

CHEMBL3544673
0.1080.2670.193Growth factor agonist

0.178 0.09 CHEMBL3544690

0.193 0.07 CHEMBL3544692

CHEMBL3544692
0.0220.1810.064Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.057 0.038 CHEMBL3544671

0.057 0.038 CHEMBL3544691

0.064 0.031 CHEMBL3544673

0.064 0.03 CHEMBL3544692

CHEMBL3544692
0.0020.1610.008Integrin alpha5beta6 antagonist

0.008 0.004 CHEMBL3544673

CHEMBL3544673
0.020.180.043Glutamate (mGluR8) antagonist

0.039 0.018 CHEMBL1105

0.043 0.013 CHEMBL3544673

CHEMBL3544673
0.0270.1870.058Fatty acid synthase inhibitor

0.058 0.039 CHEMBL3544673

CHEMBL3544673
0.0120.1730.057Ornithine carbamoyltransferase inhibitor

0.057 0.033 CHEMBL3544673

CHEMBL3544673
0.0220.1850.065Farnesyltransferase inhibitor

0.056 0.023 CHEMBL3544672

0.065 0.017 CHEMBL3544691

CHEMBL3544691
0.0870.2510.427Platelet antagonist

0.169 0.127 CHEMBL3278702

0.175 0.121 CHEMBL3544671

0.396 0.028 CHEMBL1105

0.427 0.023 CHEMBL3544673

CHEMBL3544673
0.0320.1990.28Potassium channel (Ca-activated) activator

0.213 0.012 CHEMBL1105

0.28 0.006 CHEMBL3544673

CHEMBL3544673
0.0180.1890.093NMDA receptor glycine site agonist

0.081 0.028 CHEMBL1105

0.093 0.02 CHEMBL3544673

CHEMBL3544673
0.0170.1880.086Opioid mu receptor antagonist

0.071 0.045 CHEMBL3278706

0.06 0.053 CHEMBL3544671

0.086 0.037 CHEMBL3544673

0.059 0.054 CHEMBL3544692

CHEMBL3544673
0.0260.1980.071Botulinum neurotoxin type A inhibitor

0.056 0.043 CHEMBL3544671

0.071 0.024 CHEMBL3544673

CHEMBL3544673
0.0140.1880.254Aldose reductase inhibitor

0.178 0.008 CHEMBL1105

0.254 0.005 CHEMBL3544673

CHEMBL3544673
0.0070.1810.044Carnitine palmitoyltransferase 1A inhibitor

0.044 0.009 CHEMBL1105

0.032 0.016 CHEMBL3544673

CHEMBL1105
0.0110.1850.029Integrin alpha2beta1 antagonist

0.028 0.015 CHEMBL1105

0.029 0.013 CHEMBL3544673

CHEMBL3544673
0.0330.2180.064Adenine nucleotide translocase inhibitor

0.052 0.049 CHEMBL1105

0.064 0.022 CHEMBL3544673

CHEMBL3544673
0.0280.2140.051Glucosylceramidase inhibitor

0.051 0.047 CHEMBL3544671

0.05 0.048 CHEMBL3544692

CHEMBL3544671
0.0580.2460.26Angiogenesis stimulant

0.192 0.099 CHEMBL3278702

0.247 0.071 CHEMBL3544671

0.199 0.095 CHEMBL1105

0.26 0.065 CHEMBL3544673

0.137 0.131 CHEMBL3544692

CHEMBL3544673
0.0420.230.164Cell adhesion molecule inhibitor

0.164 0.013 CHEMBL1105

0.144 0.016 CHEMBL3544673

CHEMBL1105
0.0260.2160.132NMDA receptor agonist

0.092 0.022 CHEMBL1105

0.132 0.011 CHEMBL3544673

CHEMBL3544673
0.0460.2360.109Nav1.3 sodium channel blocker

0.109 0.086 CHEMBL3278702

CHEMBL3278702
0.0480.2390.138Electrolyte absorption antagonist

0.087 0.081 CHEMBL3544671

0.107 0.048 CHEMBL1105

0.096 0.063 CHEMBL3544691

0.138 0.025 CHEMBL3544673

0.109 0.047 CHEMBL3544692

CHEMBL3544673
0.0320.2280.113Somatostatin 1 agonist

0.069 0.066 CHEMBL3278702

0.074 0.058 CHEMBL3278706

0.113 0.027 CHEMBL3544671

0.089 0.042 CHEMBL3544691

0.082 0.049 CHEMBL3544673

0.112 0.027 CHEMBL3544692

CHEMBL3544671
0.0080.2060.039Protocollagen prolyl hydroxylase inhibitor

0.027 0.02 CHEMBL1105

0.039 0.008 CHEMBL3544673

CHEMBL3544673
0.0150.2150.059Plasminogen activator inhibitor

0.059 0.04 CHEMBL3544673

CHEMBL3544673
0.0160.2180.087Maillard reaction inhibitor

0.087 0.022 CHEMBL3544673

CHEMBL3544673
0.0190.2250.048NMDA 2B receptor antagonist

0.048 0.047 CHEMBL3278706

CHEMBL3278706
0.0170.2230.069Glucagon-like peptide 1 agonist

0.054 0.052 CHEMBL3278702

0.069 0.042 CHEMBL3544671

0.064 0.045 CHEMBL3544673

0.062 0.047 CHEMBL3544692

CHEMBL3544671
0.0140.2220.056p53 inhibitor

0.054 0.012 CHEMBL1105

0.056 0.011 CHEMBL3544673

CHEMBL3544673
0.0030.2130.036Kainate receptor 1 antagonist

0.036 0.008 CHEMBL3544673

CHEMBL3544673
0.0170.2280.096Neuropeptide agonist

0.06 0.038 CHEMBL3278702

0.096 0.028 CHEMBL3544671

0.057 0.039 CHEMBL3544690

0.094 0.028 CHEMBL3544692

CHEMBL3544671
0.0620.2730.143MAP3K9 inhibitor

0.14 0.075 CHEMBL3278702

0.142 0.073 CHEMBL3544671

0.141 0.074 CHEMBL3544690

0.143 0.072 CHEMBL3544692

CHEMBL3544692
0.0270.2390.119Adrenaline antagonist

0.119 0.044 CHEMBL3278702

0.103 0.052 CHEMBL3544671

CHEMBL3278702
0.0280.2410.122Antiadrenergic

0.122 0.044 CHEMBL3278702

0.106 0.052 CHEMBL3544671

CHEMBL3278702
0.0710.2910.237Interleukin 6 antagonist

0.149 0.09 CHEMBL3278702

0.135 0.115 CHEMBL3544672

0.164 0.071 CHEMBL3544671

0.207 0.037 CHEMBL1105

0.158 0.078 CHEMBL3544690

0.147 0.093 CHEMBL3544691

0.237 0.026 CHEMBL3544673

0.174 0.06 CHEMBL3544692

CHEMBL3544673
0.0710.2910.174Hemostatic

0.12 0.114 CHEMBL3544671

0.147 0.071 CHEMBL1105

0.174 0.046 CHEMBL3544673

CHEMBL3544673
0.0040.2250.434Prostaglandin D2 antagonist

0.409 0.003 CHEMBL1105

0.434 0.003 CHEMBL3544673

CHEMBL3544673
0.0190.2430.058Nitric oxide donor

0.058 0.053 CHEMBL3278702

CHEMBL3278702
0.0030.2320.014Integrin alphaVbeta6 antagonist

0.014 0.01 CHEMBL3544673

CHEMBL3544673
0.0160.2460.254Selectin antagonist

0.066 0.045 CHEMBL3544671

0.077 0.038 CHEMBL1105

0.19 0.012 CHEMBL3544690

0.117 0.023 CHEMBL3544673

0.254 0.008 CHEMBL3544692

CHEMBL3544692
0.010.240.065Prostaglandin E2 antagonist

0.065 0.026 CHEMBL3278702

0.063 0.027 CHEMBL3544671

0.047 0.038 CHEMBL1105

0.045 0.04 CHEMBL3544690

0.045 0.041 CHEMBL3544673

CHEMBL3278702
0.0870.3190.153MAP kinase kinase 4 inhibitor

0.135 0.099 CHEMBL3278706

0.153 0.056 CHEMBL3544671

0.139 0.088 CHEMBL3544691

0.143 0.078 CHEMBL3544673

0.153 0.055 CHEMBL3544692

CHEMBL3544692
0.0080.240.066Phosphorylase inhibitor

0.066 0.022 CHEMBL3544673

CHEMBL3544673
0.010.2440.066Thymidylate synthase inhibitor

0.041 0.04 CHEMBL1105

0.066 0.014 CHEMBL3544673

CHEMBL3544673
0.0150.2540.075Diacylglycerol O-acyltransferase inhibitor

0.072 0.018 CHEMBL1105

0.075 0.016 CHEMBL3544673

CHEMBL3544673
0.1390.3830.853Cyclophilin D inhibitor

0.478 0.057 CHEMBL3278702

0.333 0.135 CHEMBL3544672

0.233 0.232 CHEMBL3278706

0.548 0.038 CHEMBL3544671

0.562 0.035 CHEMBL1105

0.809 0.006 CHEMBL3544690

0.39 0.096 CHEMBL3544691

0.634 0.022 CHEMBL3544673

0.853 0.005 CHEMBL3544692

CHEMBL3544692
0.0130.2620.105AMPA 4 receptor antagonist

0.038 0.031 CHEMBL1105

0.105 0.005 CHEMBL3544673

CHEMBL3544673
0.0180.2680.132Neuraminidase (influenza) inhibitor

0.064 0.045 CHEMBL3278702

0.091 0.019 CHEMBL3544671

0.084 0.023 CHEMBL3544690

0.069 0.036 CHEMBL3544691

0.132 0.009 CHEMBL3544692

CHEMBL3544692
0.0490.3050.237Dual specificity phosphatase 3 inhibitor

0.142 0.104 CHEMBL3544671

0.2 0.061 CHEMBL1105

0.237 0.044 CHEMBL3544673

CHEMBL3544673
0.010.2660.531Prostaglandin antagonist

0.057 0.034 CHEMBL3278702

0.051 0.039 CHEMBL3544671

0.495 0.004 CHEMBL1105

0.531 0.004 CHEMBL3544673

CHEMBL3544673
0.0060.2630.02Integrin beta5 antagonist

0.02 0.015 CHEMBL1105

0.02 0.016 CHEMBL3544673

CHEMBL3544673
0.0220.280.176Prostaglandin F2 alpha antagonist

0.142 0.005 CHEMBL3278702

0.176 0.004 CHEMBL3544671

0.069 0.034 CHEMBL1105

0.057 0.052 CHEMBL3544690

0.057 0.051 CHEMBL3544691

0.087 0.017 CHEMBL3544673

0.073 0.029 CHEMBL3544692

CHEMBL3544671
0.0240.2850.139M18 aspartyl aminopeptidase inhibitor

0.139 0.058 CHEMBL3544673

CHEMBL3544673
0.0210.2840.037Integrin alpha1beta1 antagonist

0.037 0.032 CHEMBL1105

CHEMBL1105
0.0090.2810.028Glutamate (mGluR1) agonist

0.028 0.011 CHEMBL3544673

CHEMBL3544673
0.0290.3020.141M17 leucyl aminopeptidase inhibitor

0.141 0.062 CHEMBL1105

0.14 0.062 CHEMBL3544673

CHEMBL1105
0.0050.2820.102Integrin antagonist

0.077 0.02 CHEMBL1105

0.102 0.016 CHEMBL3544673

CHEMBL3544673
0.0280.310.186Potassium channel large-conductance Ca-activated activator

0.126 0.015 CHEMBL1105

0.186 0.007 CHEMBL3544673

CHEMBL3544673
0.0120.30.045Erythropoietin receptor agonist

0.045 0.025 CHEMBL3544673

CHEMBL3544673
0.0590.3530.149Antipruritic

0.138 0.109 CHEMBL3544671

0.149 0.095 CHEMBL3544673

CHEMBL3544673
0.0450.3430.16Cell wall synthesis inhibitor

0.113 0.11 CHEMBL3544671

0.16 0.056 CHEMBL3544673

CHEMBL3544673
0.0130.3120.054Neuraminidase (Influenza A) inhibitor

0.045 0.032 CHEMBL3278702

0.054 0.019 CHEMBL3544671

0.044 0.035 CHEMBL3544692

CHEMBL3544671
0.0440.3460.215Dual specificity phosphatase inhibitor

0.133 0.116 CHEMBL3544671

0.177 0.069 CHEMBL1105

0.215 0.048 CHEMBL3544673

CHEMBL3544673
0.0790.3840.243Angiogenesis inhibitor

0.243 0.129 CHEMBL3544690

0.198 0.172 CHEMBL3544692

CHEMBL3544690
0.0490.3550.143Amyloid beta precursor protein antagonist

0.137 0.116 CHEMBL1105

0.143 0.109 CHEMBL3544673

CHEMBL3544673
0.0050.3130.053AMPA 3 receptor antagonist

0.053 0.008 CHEMBL3544673

CHEMBL3544673
0.0120.3290.031Purinergic P2Y2 antagonist

0.031 0.028 CHEMBL3544673

CHEMBL3544673
0.0040.3230.056GP IIb/IIIa receptor antagonist

0.046 0.036 CHEMBL1105

0.056 0.029 CHEMBL3544673

CHEMBL3544673
0.0190.3480.056CXC chemokine 1 receptor antagonist

0.056 0.027 CHEMBL3544673

CHEMBL3544673
0.0460.3810.126Interleukin 12 antagonist

0.104 0.047 CHEMBL3278702

0.126 0.024 CHEMBL3544671

0.104 0.048 CHEMBL3544673

CHEMBL3544671
0.0040.3510.024Vitronectin receptor antagonist

0.024 0.013 CHEMBL3544673

CHEMBL3544673
0.0020.3610.046AMPA 1 receptor antagonist

0.046 0.012 CHEMBL3544673

CHEMBL3544673
0.0080.3740.039Integrin alpha5beta1 antagonist

0.037 0.035 CHEMBL1105

0.039 0.031 CHEMBL3544673

CHEMBL3544673
0.1020.4690.449Interleukin 2 agonist

0.203 0.184 CHEMBL3278702

0.228 0.145 CHEMBL3278706

0.285 0.085 CHEMBL3544671

0.376 0.035 CHEMBL1105

0.269 0.099 CHEMBL3544691

0.449 0.016 CHEMBL3544673

0.279 0.09 CHEMBL3544692

CHEMBL3544673
0.0040.3750.073AMPA receptor antagonist

0.073 0.019 CHEMBL3544673

CHEMBL3544673
0.010.3890.105Protein kinase (CK2) alpha inhibitor

0.105 0.073 CHEMBL3544673

CHEMBL3544673
0.0050.4090.018Integrin alphaVbeta1 antagonist

0.018 0.015 CHEMBL3544673

CHEMBL3544673
0.0590.4930.306Antiobesity

0.261 0.146 CHEMBL1105

0.306 0.112 CHEMBL3544673

CHEMBL3544673
0.0050.5120.016Integrin beta6 antagonist

0.016 0.006 CHEMBL3544673

CHEMBL3544673
0.0110.5380.083Protein kinase C delta inhibitor

0.083 0.072 CHEMBL3544692

CHEMBL3544692
0.0040.540.074Diacylglycerol O-acyltransferase 1 inhibitor

0.062 0.007 CHEMBL1105

0.074 0.005 CHEMBL3544673

CHEMBL3544673
0.0450.5880.511Toll-Like receptor agonist

0.205 0.195 CHEMBL3278702

0.213 0.186 CHEMBL3544671

0.473 0.037 CHEMBL1105

0.511 0.03 CHEMBL3544673

CHEMBL3544673
0.0460.5880.515Toll-Like receptor 7 agonist

0.205 0.194 CHEMBL3544671

0.476 0.037 CHEMBL1105

0.515 0.029 CHEMBL3544673

CHEMBL3544673
0.0220.5940.143Nav1.4 sodium channel blocker

0.099 0.078 CHEMBL1105

0.143 0.037 CHEMBL3544673

CHEMBL3544673
0.0730.6780.214Peptidyltransferase inhibitor

0.214 0.083 CHEMBL3544671

0.172 0.142 CHEMBL3544691

0.201 0.097 CHEMBL3544673

0.205 0.092 CHEMBL3544692

CHEMBL3544671
0.0070.6350.119Glutamate receptor antagonist

0.119 0.075 CHEMBL3544673

CHEMBL3544673
0.0290.7210.226Immunomodulator

0.212 0.149 CHEMBL3544671

0.226 0.136 CHEMBL3544692

CHEMBL3544692
0.0040.7590.041AMPA 2 receptor antagonist

0.041 0.014 CHEMBL3544673

CHEMBL3544673
0.0130.8430.331Aurora-C kinase inhibitor

0.311 0.004 CHEMBL3544690

0.331 0.004 CHEMBL3544692

CHEMBL3544692
0.0110.860.098CDK3/cyclin E inhibitor

0.098 0.091 CHEMBL3544692

CHEMBL3544692
Ext Pa Pi Pmax Activity Other Results ID Pa_max