| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.887 | 0.001 | 0.887 | Endothelin A receptor antagonist | 0.146 0.004 CHEMBL3706457 0.645 0.001 CHEMBL3706458 0.833 0.001 CHEMBL3706459 0.824 0.001 CHEMBL3706460 0.869 0.001 CHEMBL3706461 0.595 0.001 CHEMBL3706463 0.724 0.001 CHEMBL3706464 0.623 0.001 CHEMBL3706462 | ||
| 0.884 | 0.001 | 0.884 | Endothelin receptor antagonist | 0.145 0.004 CHEMBL3706457 0.64 0.002 CHEMBL3706458 0.819 0.001 CHEMBL3706459 0.802 0.001 CHEMBL3706460 0.864 0.001 CHEMBL3706461 0.591 0.002 CHEMBL3706463 0.723 0.001 CHEMBL3706464 0.614 0.002 CHEMBL3706462 | ||
| 0.847 | 0.004 | 0.847 | Cardiotonic | 0.624 0.007 CHEMBL3706458 0.812 0.004 CHEMBL3706459 0.701 0.005 CHEMBL3706460 0.841 0.004 CHEMBL3706461 0.596 0.008 CHEMBL3706463 0.659 0.005 CHEMBL3706464 0.619 0.007 CHEMBL3706462 | ||
| 0.832 | 0.001 | 0.832 | Endothelin B receptor antagonist | 0.129 0.004 CHEMBL3706457 0.557 0.002 CHEMBL3706458 0.757 0.001 CHEMBL3706459 0.803 0.001 CHEMBL3706460 0.801 0.001 CHEMBL3706461 0.484 0.002 CHEMBL3706463 0.732 0.001 CHEMBL3706464 0.525 0.002 CHEMBL3706462 | ||
| 0.676 | 0.01 | 0.764 | Toll-Like receptor 7 agonist | 0.223 0.174 CHEMBL3706457 0.335 0.09 CHEMBL3706458 0.671 0.011 CHEMBL3706459 0.764 0.005 CHEMBL3706460 0.719 0.008 CHEMBL3706461 0.365 0.075 CHEMBL3706463 0.749 0.006 CHEMBL3706464 0.396 0.061 CHEMBL3706462 | CHEMBL3706460 | |
| 0.673 | 0.01 | 0.759 | Toll-Like receptor agonist | 0.221 0.178 CHEMBL3706457 0.353 0.08 CHEMBL3706458 0.67 0.011 CHEMBL3706459 0.759 0.005 CHEMBL3706460 0.716 0.008 CHEMBL3706461 0.385 0.067 CHEMBL3706463 0.746 0.006 CHEMBL3706464 0.414 0.055 CHEMBL3706462 | CHEMBL3706460 | |
| 0.444 | 0.054 | 0.608 | Calcium channel L-type activator | 0.472 0.04 CHEMBL3706457 0.253 0.202 CHEMBL3706458 0.608 0.005 CHEMBL3706459 0.352 0.116 CHEMBL3706460 0.6 0.005 CHEMBL3706461 0.525 0.019 CHEMBL3706463 0.594 0.006 CHEMBL3706464 0.506 0.025 CHEMBL3706462 | CHEMBL3706459 | |
| 0.391 | 0.058 | 0.552 | Vasodilator, peripheral | 0.369 0.066 CHEMBL3706457 0.372 0.065 CHEMBL3706458 0.514 0.025 CHEMBL3706459 0.35 0.074 CHEMBL3706460 0.552 0.021 CHEMBL3706461 0.496 0.028 CHEMBL3706463 0.478 0.033 CHEMBL3706464 0.527 0.023 CHEMBL3706462 | CHEMBL3706461 | |
| 0.309 | 0.038 | 0.483 | Cyclic AMP phosphodiesterase inhibitor | 0.413 0.015 CHEMBL3706457 0.37 0.021 CHEMBL3706458 0.416 0.014 CHEMBL3706459 0.377 0.02 CHEMBL3706460 0.354 0.025 CHEMBL3706461 0.477 0.008 CHEMBL3706463 0.483 0.008 CHEMBL3706464 0.422 0.014 CHEMBL3706462 | CHEMBL3706464 | |
| 0.337 | 0.07 | 0.598 | Cholesterol antagonist | 0.326 0.076 CHEMBL3706457 0.553 0.025 CHEMBL3706458 0.373 0.056 CHEMBL3706459 0.411 0.047 CHEMBL3706460 0.38 0.054 CHEMBL3706461 0.592 0.02 CHEMBL3706463 0.469 0.037 CHEMBL3706464 0.598 0.019 CHEMBL3706462 | CHEMBL3706462 | |
| 0.305 | 0.087 | 0.328 | Calcium channel activator | 0.328 0.066 CHEMBL3706457 0.318 0.075 CHEMBL3706459 0.308 0.084 CHEMBL3706460 0.306 0.086 CHEMBL3706461 0.32 0.072 CHEMBL3706464 | CHEMBL3706457 | |
| 0.182 | 0.006 | 0.297 | Leukotriene synthesis inhibitor | 0.091 0.031 CHEMBL3706458 0.251 0.005 CHEMBL3706459 0.297 0.004 CHEMBL3706461 0.128 0.014 CHEMBL3706463 0.112 0.02 CHEMBL3706464 0.14 0.011 CHEMBL3706462 | CHEMBL3706461 | |
| 0.319 | 0.145 | 0.45 | 5 Hydroxytryptamine release inhibitor | 0.45 0.051 CHEMBL3706457 0.269 0.203 CHEMBL3706458 0.333 0.131 CHEMBL3706460 | CHEMBL3706457 | |
| 0.155 | 0.012 | 0.165 | Peroxisome proliferator-activated receptor gamma agonist | 0.137 0.016 CHEMBL3706459 0.165 0.01 CHEMBL3706460 0.152 0.012 CHEMBL3706461 0.146 0.014 CHEMBL3706464 | CHEMBL3706460 | |
| 0.178 | 0.042 | 0.384 | Alpha-N-acetylglucosaminidase inhibitor | 0.384 0.01 CHEMBL3706457 0.209 0.031 CHEMBL3706458 0.171 0.044 CHEMBL3706459 0.26 0.021 CHEMBL3706460 0.245 0.024 CHEMBL3706461 0.202 0.034 CHEMBL3706463 0.251 0.023 CHEMBL3706464 0.286 0.018 CHEMBL3706462 | CHEMBL3706457 | |
| 0.167 | 0.037 | 0.504 | Interleukin 4 antagonist | 0.504 0.004 CHEMBL3706457 0.189 0.026 CHEMBL3706458 0.145 0.054 CHEMBL3706459 0.157 0.044 CHEMBL3706460 0.158 0.043 CHEMBL3706461 0.169 0.035 CHEMBL3706463 0.135 0.066 CHEMBL3706464 0.181 0.029 CHEMBL3706462 | CHEMBL3706457 | |
| 0.143 | 0.015 | 0.144 | Interleukin 12 antagonist | 0.142 0.015 CHEMBL3706457 0.126 0.024 CHEMBL3706458 0.128 0.023 CHEMBL3706459 0.144 0.014 CHEMBL3706460 0.136 0.018 CHEMBL3706461 0.116 0.033 CHEMBL3706463 0.128 0.023 CHEMBL3706464 0.122 0.028 CHEMBL3706462 | CHEMBL3706460 | |
| 0.129 | 0.004 | 0.531 | Heme oxygenase stimulant | 0.531 0 CHEMBL3706457 0.1 0.007 CHEMBL3706458 0.114 0.005 CHEMBL3706459 0.135 0.003 CHEMBL3706460 0.121 0.004 CHEMBL3706461 0.091 0.009 CHEMBL3706463 0.118 0.005 CHEMBL3706464 0.095 0.009 CHEMBL3706462 | CHEMBL3706457 | |
| 0.172 | 0.048 | 0.292 | Mannose-6-phosphate isomerase inhibitor | 0.292 0.006 CHEMBL3706457 0.147 0.067 CHEMBL3706458 0.133 0.082 CHEMBL3706459 0.18 0.042 CHEMBL3706460 0.134 0.08 CHEMBL3706461 0.115 0.109 CHEMBL3706463 0.141 0.073 CHEMBL3706464 0.116 0.107 CHEMBL3706462 | CHEMBL3706457 | |
| 0.155 | 0.036 | 0.208 | 5-Lipoxygenase inhibitor | 0.18 0.029 CHEMBL3706459 0.208 0.023 CHEMBL3706461 | CHEMBL3706461 | |
| 0.166 | 0.058 | 0.199 | Protein kinase stimulant | 0.146 0.071 CHEMBL3706457 0.156 0.064 CHEMBL3706458 0.161 0.061 CHEMBL3706459 0.199 0.042 CHEMBL3706460 0.171 0.055 CHEMBL3706461 0.151 0.067 CHEMBL3706463 0.193 0.044 CHEMBL3706464 0.161 0.061 CHEMBL3706462 | CHEMBL3706460 | |
| 0.109 | 0.007 | 0.128 | Aconitate hydratase inhibitor | 0.094 0.01 CHEMBL3706457 0.066 0.021 CHEMBL3706459 0.128 0.005 CHEMBL3706460 0.101 0.008 CHEMBL3706461 0.076 0.016 CHEMBL3706464 | CHEMBL3706460 | |
| 0.167 | 0.069 | 0.206 | Arachidonic acid antagonist | 0.206 0.028 CHEMBL3706457 0.142 0.098 CHEMBL3706459 0.173 0.061 CHEMBL3706460 0.148 0.091 CHEMBL3706461 0.151 0.087 CHEMBL3706464 | CHEMBL3706457 | |
| 0.124 | 0.03 | 0.175 | Triose-phosphate isomerase inhibitor | 0.165 0.016 CHEMBL3706457 0.132 0.026 CHEMBL3706458 0.118 0.033 CHEMBL3706459 0.175 0.014 CHEMBL3706460 0.16 0.017 CHEMBL3706461 0.126 0.029 CHEMBL3706463 0.166 0.016 CHEMBL3706464 0.171 0.015 CHEMBL3706462 | CHEMBL3706460 | |
| 0.235 | 0.149 | 0.383 | Vasodilator, coronary | 0.272 0.113 CHEMBL3706457 0.322 0.071 CHEMBL3706458 0.294 0.092 CHEMBL3706459 0.193 0.188 CHEMBL3706460 0.292 0.094 CHEMBL3706461 0.383 0.041 CHEMBL3706463 0.264 0.12 CHEMBL3706464 0.381 0.042 CHEMBL3706462 | CHEMBL3706463 | |
| 0.131 | 0.045 | 0.15 | Mucolytic | 0.102 0.074 CHEMBL3706457 0.116 0.058 CHEMBL3706459 0.15 0.033 CHEMBL3706460 0.141 0.038 CHEMBL3706461 0.134 0.043 CHEMBL3706464 | CHEMBL3706460 | |
| 0.111 | 0.028 | 0.162 | Phosphofructokinase-1 inhibitor | 0.157 0.017 CHEMBL3706457 0.131 0.022 CHEMBL3706458 0.106 0.029 CHEMBL3706459 0.157 0.017 CHEMBL3706460 0.141 0.02 CHEMBL3706461 0.126 0.024 CHEMBL3706463 0.152 0.018 CHEMBL3706464 0.162 0.016 CHEMBL3706462 | CHEMBL3706462 | |
| 0.123 | 0.041 | 0.233 | Adenylate kinase inhibitor | 0.233 0.011 CHEMBL3706457 0.102 0.065 CHEMBL3706459 0.144 0.029 CHEMBL3706460 0.118 0.045 CHEMBL3706461 0.117 0.046 CHEMBL3706464 | CHEMBL3706457 | |
| 0.2 | 0.12 | 0.535 | Immunostimulant | 0.283 0.084 CHEMBL3706457 0.498 0.029 CHEMBL3706458 0.209 0.115 CHEMBL3706459 0.209 0.115 CHEMBL3706460 0.246 0.098 CHEMBL3706461 0.508 0.028 CHEMBL3706463 0.22 0.109 CHEMBL3706464 0.535 0.025 CHEMBL3706462 | CHEMBL3706462 | |
| 0.176 | 0.1 | 0.179 | Insulin sensitizer | 0.156 0.125 CHEMBL3706459 0.179 0.096 CHEMBL3706460 0.177 0.099 CHEMBL3706461 0.16 0.12 CHEMBL3706464 | CHEMBL3706460 | |
| 0.187 | 0.112 | 0.477 | Aldehyde oxidase inhibitor | 0.477 0.036 CHEMBL3706457 0.213 0.098 CHEMBL3706460 | CHEMBL3706457 | |
| 0.163 | 0.09 | 0.23 | Succinate dehydrogenase inhibitor | 0.23 0.03 CHEMBL3706457 0.179 0.069 CHEMBL3706460 0.15 0.112 CHEMBL3706461 | CHEMBL3706457 | |
| 0.158 | 0.088 | 0.194 | ATPase inhibitor | 0.184 0.053 CHEMBL3706457 0.194 0.042 CHEMBL3706458 0.168 0.073 CHEMBL3706460 | CHEMBL3706458 | |
| 0.147 | 0.082 | 0.237 | Interferon gamma antagonist | 0.188 0.046 CHEMBL3706457 0.237 0.031 CHEMBL3706458 0.133 0.104 CHEMBL3706459 0.138 0.095 CHEMBL3706460 0.136 0.1 CHEMBL3706461 0.204 0.039 CHEMBL3706463 0.125 0.121 CHEMBL3706464 0.209 0.038 CHEMBL3706462 | CHEMBL3706458 | |
| 0.102 | 0.039 | 0.19 | Interleukin 5 antagonist | 0.19 0.006 CHEMBL3706457 0.084 0.065 CHEMBL3706458 0.09 0.054 CHEMBL3706459 0.097 0.044 CHEMBL3706460 0.09 0.054 CHEMBL3706461 0.086 0.061 CHEMBL3706464 | CHEMBL3706457 | |
| 0.124 | 0.062 | 0.153 | Cholesterol synthesis inhibitor | 0.11 0.075 CHEMBL3706457 0.153 0.043 CHEMBL3706460 0.112 0.073 CHEMBL3706464 | CHEMBL3706460 | |
| 0.094 | 0.034 | 0.133 | Glutamate dehydrogenase inhibitor | 0.13 0.02 CHEMBL3706457 0.07 0.056 CHEMBL3706459 0.133 0.019 CHEMBL3706460 0.088 0.038 CHEMBL3706461 0.097 0.032 CHEMBL3706464 | CHEMBL3706460 | |
| 0.106 | 0.049 | 0.164 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.164 0.023 CHEMBL3706457 0.089 0.066 CHEMBL3706459 0.149 0.027 CHEMBL3706460 0.123 0.037 CHEMBL3706461 0.123 0.038 CHEMBL3706464 0.087 0.07 CHEMBL3706462 | CHEMBL3706457 | |
| 0.138 | 0.081 | 0.171 | Ca2+-transporting ATPase inhibitor | 0.171 0.012 CHEMBL3706457 0.144 0.061 CHEMBL3706458 0.147 0.05 CHEMBL3706460 0.132 0.107 CHEMBL3706461 0.131 0.113 CHEMBL3706463 0.135 0.096 CHEMBL3706464 0.138 0.082 CHEMBL3706462 | CHEMBL3706457 | |
| 0.113 | 0.058 | 0.337 | Ferrochelatase inhibitor | 0.337 0.005 CHEMBL3706457 0.187 0.025 CHEMBL3706460 | CHEMBL3706457 | |
| 0.081 | 0.028 | 0.133 | Carbamoyl phosphate synthetase inhibitor | 0.133 0.013 CHEMBL3706457 0.063 0.04 CHEMBL3706459 0.115 0.017 CHEMBL3706460 0.097 0.022 CHEMBL3706461 0.091 0.024 CHEMBL3706464 | CHEMBL3706457 | |
| 0.091 | 0.038 | 0.122 | Interferon agonist | 0.122 0.016 CHEMBL3706457 0.111 0.021 CHEMBL3706458 0.083 0.047 CHEMBL3706459 0.087 0.042 CHEMBL3706460 0.083 0.047 CHEMBL3706461 0.102 0.027 CHEMBL3706463 0.08 0.053 CHEMBL3706464 0.102 0.027 CHEMBL3706462 | CHEMBL3706457 | |
| 0.057 | 0.011 | 0.059 | Fumarate hydratase inhibitor | 0.05 0.014 CHEMBL3706457 0.039 0.019 CHEMBL3706459 0.056 0.011 CHEMBL3706460 0.059 0.01 CHEMBL3706461 0.038 0.02 CHEMBL3706464 | CHEMBL3706461 | |
| 0.075 | 0.029 | 0.103 | Interferon inducer | 0.103 0.011 CHEMBL3706457 0.093 0.015 CHEMBL3706458 0.069 0.036 CHEMBL3706459 0.071 0.033 CHEMBL3706460 0.069 0.037 CHEMBL3706461 0.086 0.019 CHEMBL3706463 0.066 0.042 CHEMBL3706464 0.086 0.02 CHEMBL3706462 | CHEMBL3706457 | |
| 0.15 | 0.105 | 0.162 | Lipocortins synthesis antagonist | 0.162 0.089 CHEMBL3706460 | CHEMBL3706460 | |
| 0.106 | 0.063 | 0.217 | Expectorant | 0.198 0.021 CHEMBL3706458 0.092 0.078 CHEMBL3706459 0.121 0.05 CHEMBL3706460 0.117 0.053 CHEMBL3706461 0.173 0.027 CHEMBL3706463 0.105 0.063 CHEMBL3706464 0.217 0.017 CHEMBL3706462 | CHEMBL3706462 | |
| 0.081 | 0.042 | 0.136 | Histidine decarboxylase inhibitor | 0.136 0.022 CHEMBL3706457 0.072 0.049 CHEMBL3706459 0.077 0.045 CHEMBL3706460 0.103 0.031 CHEMBL3706461 0.068 0.053 CHEMBL3706464 | CHEMBL3706457 | |
| 0.067 | 0.03 | 0.207 | Alcohol oxidase inhibitor | 0.207 0.006 CHEMBL3706457 0.081 0.024 CHEMBL3706460 0.055 0.04 CHEMBL3706461 | CHEMBL3706457 | |
| 0.057 | 0.021 | 0.076 | Glucose-6-phosphate isomerase inhibitor | 0.076 0.01 CHEMBL3706457 0.055 0.023 CHEMBL3706458 0.056 0.022 CHEMBL3706459 0.071 0.012 CHEMBL3706460 0.073 0.011 CHEMBL3706461 0.055 0.023 CHEMBL3706463 0.07 0.012 CHEMBL3706464 0.07 0.012 CHEMBL3706462 | CHEMBL3706457 | |
| 0.091 | 0.055 | 0.22 | NADH dehydrogenase inhibitor | 0.197 0.011 CHEMBL3706457 0.168 0.014 CHEMBL3706458 0.088 0.059 CHEMBL3706459 0.111 0.034 CHEMBL3706460 0.114 0.032 CHEMBL3706461 0.163 0.015 CHEMBL3706463 0.108 0.037 CHEMBL3706464 0.22 0.009 CHEMBL3706462 | CHEMBL3706462 | |
| 0.076 | 0.041 | 0.164 | Phenylalanine 4-hydroxylase inhibitor | 0.164 0.01 CHEMBL3706457 0.12 0.018 CHEMBL3706460 0.065 0.051 CHEMBL3706464 | CHEMBL3706457 | |
| 0.128 | 0.093 | 0.437 | Peroxidase inhibitor | 0.437 0.016 CHEMBL3706457 0.191 0.062 CHEMBL3706460 | CHEMBL3706457 | |
| 0.193 | 0.159 | 0.267 | Gastrin inhibitor | 0.267 0.06 CHEMBL3706457 0.209 0.135 CHEMBL3706460 0.191 0.163 CHEMBL3706464 | CHEMBL3706457 | |
| 0.209 | 0.176 | 0.209 | Sodium/bile acid cotransporter inhibitor | 0.203 0.184 CHEMBL3706460 | ||
| 0.185 | 0.157 | 0.262 | Lipoxygenase inhibitor | 0.262 0.092 CHEMBL3706457 0.18 0.164 CHEMBL3706459 0.192 0.149 CHEMBL3706461 | CHEMBL3706457 | |
| 0.187 | 0.16 | 0.306 | Tyrosine 3 hydroxylase inhibitor | 0.306 0.031 CHEMBL3706457 0.213 0.113 CHEMBL3706460 | CHEMBL3706457 | |
| 0.147 | 0.12 | 0.261 | Interleukin antagonist | 0.261 0.058 CHEMBL3706457 0.152 0.116 CHEMBL3706460 | CHEMBL3706457 | |
| 0.082 | 0.057 | 0.112 | Thioredoxin reductase inhibitor | 0.112 0.02 CHEMBL3706457 0.078 0.067 CHEMBL3706458 0.081 0.059 CHEMBL3706459 0.082 0.056 CHEMBL3706460 0.082 0.056 CHEMBL3706461 0.078 0.067 CHEMBL3706463 0.081 0.058 CHEMBL3706464 0.079 0.065 CHEMBL3706462 | CHEMBL3706457 | |
| 0.061 | 0.04 | 0.158 | Biliverdin reductase inhibitor | 0.158 0.009 CHEMBL3706457 0.095 0.02 CHEMBL3706460 0.054 0.047 CHEMBL3706461 0.062 0.039 CHEMBL3706464 | CHEMBL3706457 | |
| 0.072 | 0.053 | 0.116 | Glutamate decarboxylase inhibitor | 0.116 0.022 CHEMBL3706457 0.097 0.031 CHEMBL3706460 | CHEMBL3706457 | |
| 0.07 | 0.056 | 0.396 | Porphobilinogen synthase inhibitor | 0.396 0.004 CHEMBL3706457 0.127 0.026 CHEMBL3706460 0.094 0.039 CHEMBL3706464 | CHEMBL3706457 | |
| 0.095 | 0.083 | 0.2 | Cystathionine beta-synthase inhibitor | 0.2 0.025 CHEMBL3706457 | CHEMBL3706457 | |
| 0.067 | 0.057 | 0.069 | Catalase inhibitor | 0.066 0.059 CHEMBL3706460 0.069 0.056 CHEMBL3706461 | CHEMBL3706461 | |
| 0.036 | 0.03 | 0.065 | Glutamate (mGluR8) agonist | 0.065 0.006 CHEMBL3706457 0.04 0.022 CHEMBL3706460 | CHEMBL3706457 | |
| 0.032 | 0.027 | 0.048 | Free fatty acid receptor 1 antagonist | 0.048 0.01 CHEMBL3706457 0.032 0.026 CHEMBL3706459 0.041 0.015 CHEMBL3706460 0.042 0.014 CHEMBL3706464 | CHEMBL3706457 | |
| 0.069 | 0.067 | 0.105 | Keratolytic | 0.105 0.028 CHEMBL3706457 | CHEMBL3706457 | |
| 0.061 | 0.062 | 0.082 | Glutamate (mGluR6) antagonist | 0.082 0.022 CHEMBL3706457 0.066 0.048 CHEMBL3706460 | CHEMBL3706457 | |
| 0.028 | 0.03 | 0.031 | Peroxisome proliferator-activated receptor delta agonist | 0.031 0.027 CHEMBL3706460 | CHEMBL3706460 | |
| 0.03 | 0.032 | 0.032 | Peroxisome proliferator-activated receptor delta antagonist | 0.032 0.025 CHEMBL3706460 | CHEMBL3706460 | |
| 0.053 | 0.057 | 0.188 | Purinergic P2X1 antagonist | 0.188 0.004 CHEMBL3706457 0.068 0.034 CHEMBL3706460 | CHEMBL3706457 | |
| 0.159 | 0.164 | 0.388 | Hypoglycemic | 0.355 0.037 CHEMBL3706458 0.19 0.122 CHEMBL3706459 0.202 0.11 CHEMBL3706461 0.365 0.034 CHEMBL3706463 0.193 0.119 CHEMBL3706464 0.388 0.03 CHEMBL3706462 | CHEMBL3706462 | |
| 0.042 | 0.048 | 0.057 | Prostaglandin antagonist | 0.057 0.034 CHEMBL3706460 | CHEMBL3706460 | |
| 0.046 | 0.057 | 0.13 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.13 0.01 CHEMBL3706457 0.064 0.031 CHEMBL3706460 0.064 0.03 CHEMBL3706461 0.066 0.029 CHEMBL3706464 0.061 0.033 CHEMBL3706462 | CHEMBL3706457 | |
| 0.158 | 0.174 | 0.335 | Peptidyltransferase inhibitor | 0.174 0.139 CHEMBL3706457 0.335 0.015 CHEMBL3706458 0.174 0.139 CHEMBL3706460 0.312 0.021 CHEMBL3706463 0.321 0.018 CHEMBL3706462 | CHEMBL3706458 | |
| 0.159 | 0.178 | 0.287 | RNA-directed DNA polymerase inhibitor | 0.287 0.034 CHEMBL3706457 | CHEMBL3706457 | |
| 0.124 | 0.144 | 0.37 | Hepatoprotectant | 0.342 0.02 CHEMBL3706458 0.167 0.092 CHEMBL3706459 0.14 0.121 CHEMBL3706460 0.172 0.088 CHEMBL3706461 0.351 0.019 CHEMBL3706463 0.182 0.078 CHEMBL3706464 0.37 0.016 CHEMBL3706462 | CHEMBL3706462 | |
| 0.222 | 0.245 | 0.509 | Cyclophilin D inhibitor | 0.441 0.07 CHEMBL3706458 0.285 0.176 CHEMBL3706459 0.268 0.192 CHEMBL3706460 0.336 0.133 CHEMBL3706461 0.463 0.062 CHEMBL3706463 0.329 0.139 CHEMBL3706464 0.509 0.048 CHEMBL3706462 | CHEMBL3706462 | |
| 0.13 | 0.16 | 0.161 | Hypolipemic | 0.145 0.142 CHEMBL3706458 0.152 0.134 CHEMBL3706461 0.15 0.137 CHEMBL3706463 0.15 0.136 CHEMBL3706464 0.161 0.126 CHEMBL3706462 | CHEMBL3706462 | |
| 0.084 | 0.114 | 0.145 | DOPA decarboxylase inhibitor | 0.145 0.024 CHEMBL3706457 | CHEMBL3706457 | |
| 0.04 | 0.071 | 0.072 | Alpha-mannosidase inhibitor | 0.053 0.037 CHEMBL3706457 0.054 0.036 CHEMBL3706458 0.056 0.032 CHEMBL3706461 0.055 0.035 CHEMBL3706463 0.072 0.015 CHEMBL3706462 | CHEMBL3706462 | |
| 0.112 | 0.145 | 0.165 | Adenylate cyclase stimulant | 0.165 0.041 CHEMBL3706457 0.124 0.115 CHEMBL3706460 | CHEMBL3706457 | |
| 0.037 | 0.071 | 0.102 | Argininosuccinate synthase inhibitor | 0.102 0.019 CHEMBL3706457 0.057 0.04 CHEMBL3706460 | CHEMBL3706457 | |
| 0.075 | 0.11 | 0.121 | Electrolyte absorption antagonist | 0.121 0.035 CHEMBL3706457 | CHEMBL3706457 | |
| 0.085 | 0.12 | 0.142 | Microtubule formation inhibitor | 0.109 0.076 CHEMBL3706457 0.142 0.042 CHEMBL3706458 0.112 0.071 CHEMBL3706463 0.125 0.055 CHEMBL3706462 | CHEMBL3706458 | |
| 0.116 | 0.154 | 0.199 | CF transmembrane conductance regulator agonist | 0.199 0.022 CHEMBL3706457 | CHEMBL3706457 | |
| 0.184 | 0.223 | 0.398 | Histamine release inhibitor | 0.398 0.077 CHEMBL3706457 0.24 0.163 CHEMBL3706458 0.226 0.175 CHEMBL3706460 0.216 0.185 CHEMBL3706463 0.204 0.198 CHEMBL3706464 0.224 0.176 CHEMBL3706462 | CHEMBL3706457 | |
| 0.045 | 0.085 | 0.08 | Adenine nucleotide translocase inhibitor | 0.078 0.01 CHEMBL3706458 0.076 0.011 CHEMBL3706463 0.08 0.009 CHEMBL3706462 | CHEMBL3706462 | |
| 0.041 | 0.082 | 0.06 | Botulinum neurotoxin type A inhibitor | 0.058 0.04 CHEMBL3706457 0.06 0.037 CHEMBL3706460 | CHEMBL3706460 | |
| 0.026 | 0.068 | 0.056 | Angiotensin AT1 receptor antagonist | 0.056 0.01 CHEMBL3706457 | CHEMBL3706457 | |
| 0.05 | 0.092 | 0.086 | Aminopeptidase I inhibitor | 0.086 0.037 CHEMBL3706457 0.069 0.055 CHEMBL3706460 | CHEMBL3706457 | |
| 0.071 | 0.113 | 0.309 | GABA C receptor agonist | 0.309 0.009 CHEMBL3706457 0.104 0.062 CHEMBL3706460 | CHEMBL3706457 | |
| 0.055 | 0.098 | 0.087 | Glycine receptor agonist | 0.087 0.031 CHEMBL3706457 | CHEMBL3706457 | |
| 0.013 | 0.056 | 0.062 | Uridine phosphorylase inhibitor | 0.062 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.008 | 0.052 | 0.015 | Thromboxane A2 agonist | 0.015 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.074 | 0.048 | Kainate receptor agonist | 0.048 0.016 CHEMBL3706457 | CHEMBL3706457 | |
| 0.068 | 0.116 | 0.276 | UDP-glucose 4-epimerase inhibitor | 0.228 0.015 CHEMBL3706457 0.19 0.019 CHEMBL3706458 0.097 0.064 CHEMBL3706460 0.094 0.068 CHEMBL3706461 0.192 0.019 CHEMBL3706463 0.098 0.063 CHEMBL3706464 0.276 0.012 CHEMBL3706462 | CHEMBL3706462 | |
| 0.032 | 0.079 | 0.104 | Acyl-CoA dehydrogenase inhibitor | 0.104 0.015 CHEMBL3706457 0.048 0.045 CHEMBL3706460 | CHEMBL3706457 | |
| 0.016 | 0.065 | 0.028 | Glutamate (mGluR1) agonist | 0.028 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.025 | 0.074 | 0.053 | Guanylate cyclase inhibitor | 0.053 0.018 CHEMBL3706457 | CHEMBL3706457 | |
| 0.102 | 0.151 | 0.167 | Sphingosine 1-phosphate receptor 2 antagonist | 0.167 0.024 CHEMBL3706457 0.118 0.103 CHEMBL3706460 | CHEMBL3706457 | |
| 0.072 | 0.121 | 0.153 | GABA C receptor rho-1 antagonist | 0.153 0.02 CHEMBL3706457 | CHEMBL3706457 | |
| 0.02 | 0.071 | 0.032 | Hedgehog signaling activator | 0.032 0.009 CHEMBL3706457 | CHEMBL3706457 | |
| 0.06 | 0.111 | 0.09 | GABA B receptor agonist | 0.09 0.025 CHEMBL3706457 | CHEMBL3706457 | |
| 0.026 | 0.078 | 0.065 | Mannosidase inhibitor | 0.041 0.038 CHEMBL3706457 0.043 0.034 CHEMBL3706458 0.043 0.034 CHEMBL3706461 0.045 0.032 CHEMBL3706463 0.065 0.014 CHEMBL3706462 | CHEMBL3706462 | |
| 0.053 | 0.105 | 0.077 | GABA aminotransferase inhibitor | 0.077 0.051 CHEMBL3706457 | CHEMBL3706457 | |
| 0.012 | 0.067 | 0.018 | Methylmalonyl-CoA mutase inhibitor | 0.018 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.034 | 0.089 | 0.068 | Topoisomerase II beta inhibitor | 0.068 0.017 CHEMBL3706457 | CHEMBL3706457 | |
| 0.02 | 0.075 | 0.043 | Angiotensin II receptor antagonist | 0.043 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.043 | 0.099 | 0.072 | Pregnane X receptor antagonist | 0.072 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.065 | 0.019 | Telomerase stimulant | 0.019 0.009 CHEMBL3706457 | CHEMBL3706457 | |
| 0.109 | 0.166 | 0.21 | Anesthetic general | 0.21 0.069 CHEMBL3706457 | CHEMBL3706457 | |
| 0.067 | 0.125 | 0.106 | Granulocyte macrophage colony stimulating factor agonist | 0.106 0.028 CHEMBL3706457 0.08 0.075 CHEMBL3706461 | CHEMBL3706457 | |
| 0.068 | 0.127 | 0.129 | Anabolic | 0.129 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.08 | 0.141 | 0.118 | Photosensitizer | 0.118 0.059 CHEMBL3706457 | CHEMBL3706457 | |
| 0.064 | 0.127 | 0.087 | ATPase (Vacuolar H+) inhibitor | 0.087 0.062 CHEMBL3706458 0.084 0.069 CHEMBL3706462 | CHEMBL3706458 | |
| 0.074 | 0.138 | 0.115 | Glutamate (mGluR7) agonist | 0.115 0.036 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.074 | 0.047 | Glutamate (mGluR1a) agonist | 0.047 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.021 | 0.086 | 0.042 | Erythropoietin receptor agonist | 0.042 0.027 CHEMBL3706457 | CHEMBL3706457 | |
| 0.088 | 0.153 | 0.364 | Cytidine deaminase inhibitor | 0.364 0.012 CHEMBL3706457 0.115 0.107 CHEMBL3706460 | CHEMBL3706457 | |
| 0.013 | 0.082 | 0.037 | Nicotinic acid receptor 2 antagonist | 0.037 0.006 CHEMBL3706457 | CHEMBL3706457 | |
| 0.054 | 0.124 | 0.128 | Aminopeptidase B inhibitor | 0.128 0.048 CHEMBL3706457 0.083 0.078 CHEMBL3706460 | CHEMBL3706457 | |
| 0.166 | 0.236 | 0.281 | 5 Hydroxytryptamine uptake stimulant | 0.281 0.056 CHEMBL3706457 | CHEMBL3706457 | |
| 0.022 | 0.092 | 0.037 | Membrane dipeptidase inhibitor | 0.037 0.03 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.101 | 0.321 | Selectin antagonist | 0.302 0.005 CHEMBL3706458 0.06 0.049 CHEMBL3706461 0.301 0.005 CHEMBL3706463 0.321 0.005 CHEMBL3706462 | CHEMBL3706462 | |
| 0.145 | 0.215 | 0.257 | DNA synthesis inhibitor | 0.257 0.062 CHEMBL3706457 0.237 0.076 CHEMBL3706458 0.189 0.14 CHEMBL3706460 0.23 0.083 CHEMBL3706463 0.18 0.153 CHEMBL3706464 0.253 0.064 CHEMBL3706462 | CHEMBL3706457 | |
| 0.022 | 0.094 | 0.063 | Ornithine carbamoyltransferase inhibitor | 0.063 0.03 CHEMBL3706457 | CHEMBL3706457 | |
| 0.066 | 0.138 | 0.094 | Estrogen-related receptor beta agonist | 0.094 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.036 | 0.111 | 0.064 | HIV-1 integrase (3'-Processing) inhibitor | 0.064 0.044 CHEMBL3706457 | CHEMBL3706457 | |
| 0.029 | 0.105 | 0.055 | HIV-1 integrase (Strand Transfer) inhibitor | 0.055 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.147 | 0.223 | 0.236 | Nitric-oxide synthase stimulant | 0.236 0.044 CHEMBL3706457 | CHEMBL3706457 | |
| 0.071 | 0.148 | 0.158 | Toll-Like receptor 4 antagonist | 0.155 0.019 CHEMBL3706458 0.149 0.021 CHEMBL3706463 0.158 0.017 CHEMBL3706462 | CHEMBL3706462 | |
| 0.022 | 0.101 | 0.041 | Tryptophan 5 hydroxylase inhibitor | 0.041 0.013 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.089 | 0.02 | Antibiotic Anthracycline-like | 0.02 0.01 CHEMBL3706458 0.02 0.012 CHEMBL3706462 | CHEMBL3706462 | |
| 0.101 | 0.183 | 0.133 | Melanin inhibitor | 0.133 0.108 CHEMBL3706457 0.127 0.12 CHEMBL3706458 0.131 0.113 CHEMBL3706462 | CHEMBL3706457 | |
| 0.012 | 0.094 | 0.02 | Toll-Like receptor 8 agonist | 0.02 0.015 CHEMBL3706457 | CHEMBL3706457 | |
| 0.045 | 0.129 | 0.075 | Ornithine decarboxylase inhibitor | 0.075 0.073 CHEMBL3706457 | CHEMBL3706457 | |
| 0.098 | 0.183 | 0.215 | GABA C receptor rho-2 antagonist | 0.215 0.022 CHEMBL3706457 | CHEMBL3706457 | |
| 0.129 | 0.214 | 0.238 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.238 0.048 CHEMBL3706457 | CHEMBL3706457 | |
| 0.066 | 0.154 | 0.177 | GABA C receptor antagonist | 0.177 0.019 CHEMBL3706457 | CHEMBL3706457 | |
| 0.043 | 0.132 | 0.059 | Lipocortins synthesis agonist | 0.059 0.037 CHEMBL3706458 0.056 0.044 CHEMBL3706463 0.058 0.041 CHEMBL3706462 | CHEMBL3706458 | |
| 0.042 | 0.135 | 0.076 | Glutamate (mGluR7) antagonist | 0.076 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.062 | 0.156 | 0.184 | Xanthine oxidase inhibitor | 0.184 0.023 CHEMBL3706457 | CHEMBL3706457 | |
| 0.036 | 0.131 | 0.087 | Na+ K+ transporting ATPase inhibitor | 0.087 0.044 CHEMBL3706457 0.068 0.062 CHEMBL3706458 0.071 0.059 CHEMBL3706462 | CHEMBL3706457 | |
| 0.139 | 0.235 | 0.299 | Beta lactamase inhibitor | 0.299 0.135 CHEMBL3706457 | CHEMBL3706457 | |
| 0.113 | 0.209 | 0.161 | Phospholipase C inhibitor | 0.161 0.086 CHEMBL3706457 | CHEMBL3706457 | |
| 0.014 | 0.111 | 0.025 | Integrin alpha2beta1 antagonist | 0.025 0.02 CHEMBL3706457 | CHEMBL3706457 | |
| 0.071 | 0.169 | 0.177 | Cyclooxygenase 3 inhibitor | 0.111 0.087 CHEMBL3706457 0.175 0.03 CHEMBL3706458 0.169 0.034 CHEMBL3706463 0.177 0.029 CHEMBL3706462 | CHEMBL3706462 | |
| 0.034 | 0.135 | 0.088 | Carbonic anhydrase XIII inhibitor | 0.088 0.044 CHEMBL3706457 | CHEMBL3706457 | |
| 0.208 | 0.309 | 0.358 | Caspase 9 stimulant | 0.358 0.139 CHEMBL3706457 0.332 0.161 CHEMBL3706458 0.284 0.211 CHEMBL3706463 0.336 0.157 CHEMBL3706462 | CHEMBL3706457 | |
| 0.025 | 0.126 | 0.064 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.064 0.006 CHEMBL3706457 | CHEMBL3706457 | |
| 0.042 | 0.145 | 0.058 | Ryanodine receptor antagonist | 0.058 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.071 | 0.177 | 0.107 | Toll-Like receptor 2 antagonist | 0.107 0.093 CHEMBL3706457 | CHEMBL3706457 | |
| 0.089 | 0.195 | 0.115 | Vanilloid 1 agonist | 0.115 0.099 CHEMBL3706457 | CHEMBL3706457 | |
| 0.116 | 0.222 | 0.152 | Heat shock protein 70 antagonist | 0.152 0.042 CHEMBL3706457 | CHEMBL3706457 | |
| 0.149 | 0.256 | 0.262 | Insulysin inhibitor | 0.262 0.086 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.127 | 0.03 | Glutamate (mGluR3) agonist | 0.03 0.028 CHEMBL3706457 | CHEMBL3706457 | |
| 0.03 | 0.138 | 0.069 | Heparanase inhibitor | 0.064 0.018 CHEMBL3706458 0.058 0.026 CHEMBL3706463 0.069 0.012 CHEMBL3706462 | CHEMBL3706462 | |
| 0.147 | 0.256 | 0.421 | Antithrombotic | 0.34 0.068 CHEMBL3706458 0.2 0.178 CHEMBL3706461 0.372 0.057 CHEMBL3706463 0.421 0.044 CHEMBL3706462 | CHEMBL3706462 | |
| 0.019 | 0.129 | 0.034 | Integrin alpha2 antagonist | 0.034 0.031 CHEMBL3706457 | CHEMBL3706457 | |
| 0.06 | 0.171 | 0.202 | Amylase inhibitor | 0.134 0.073 CHEMBL3706457 0.177 0.052 CHEMBL3706458 0.164 0.058 CHEMBL3706463 0.202 0.043 CHEMBL3706462 | CHEMBL3706462 | |
| 0.022 | 0.134 | 0.087 | Protein 50S ribosomal subunit inhibitor | 0.087 0.017 CHEMBL3706458 0.079 0.02 CHEMBL3706463 0.084 0.018 CHEMBL3706462 | CHEMBL3706458 | |
| 0.057 | 0.17 | 0.148 | Transcription factor NF kappa B stimulant | 0.136 0.019 CHEMBL3706458 0.136 0.019 CHEMBL3706463 0.148 0.016 CHEMBL3706462 | CHEMBL3706462 | |
| 0.017 | 0.131 | 0.045 | Adenosine deaminase inhibitor | 0.045 0.035 CHEMBL3706457 | CHEMBL3706457 | |
| 0.023 | 0.138 | 0.068 | Adenylate cyclase 1 inhibitor | 0.068 0.013 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.125 | 0.015 | Purinergic P2Y1 agonist | 0.015 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.089 | 0.208 | 0.322 | Nitric oxide antagonist | 0.313 0.038 CHEMBL3706458 0.297 0.041 CHEMBL3706463 0.322 0.036 CHEMBL3706462 | CHEMBL3706462 | |
| 0.078 | 0.203 | 0.177 | Cell wall synthesis inhibitor | 0.114 0.108 CHEMBL3706457 0.166 0.051 CHEMBL3706458 0.153 0.063 CHEMBL3706463 0.177 0.042 CHEMBL3706462 | CHEMBL3706462 | |
| 0.066 | 0.194 | 0.106 | Aldehyde dehydrogenase inhibitor | 0.106 0.088 CHEMBL3706457 | CHEMBL3706457 | |
| 0.022 | 0.151 | 0.067 | Microtubule stabilization | 0.067 0.008 CHEMBL3706458 0.064 0.01 CHEMBL3706463 0.066 0.009 CHEMBL3706462 | CHEMBL3706458 | |
| 0.096 | 0.226 | 0.15 | Non-steroidal antiinflammatory agent | 0.147 0.119 CHEMBL3706458 0.15 0.114 CHEMBL3706463 | CHEMBL3706463 | |
| 0.027 | 0.157 | 0.06 | Carbonic anhydrase stimulant | 0.06 0.04 CHEMBL3706457 | CHEMBL3706457 | |
| 0.057 | 0.188 | 0.097 | D-Ala-D-Ala ligase inhibitor | 0.097 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.15 | 0.061 | Dihydroorotase inhibitor | 0.061 0.016 CHEMBL3706457 | CHEMBL3706457 | |
| 0.047 | 0.178 | 0.18 | HIV-1 integrase (Overall Integration) inhibitor | 0.18 0.016 CHEMBL3706457 | CHEMBL3706457 | |
| 0.015 | 0.148 | 0.05 | Glutamate (mGluR3) antagonist | 0.05 0.013 CHEMBL3706457 | CHEMBL3706457 | |
| 0.027 | 0.16 | 0.09 | Sphingosine 1-phosphate receptor 4 agonist | 0.09 0.031 CHEMBL3706457 | CHEMBL3706457 | |
| 0.043 | 0.178 | 0.077 | Transcription factor RelA inhibitor | 0.077 0.02 CHEMBL3706457 | CHEMBL3706457 | |
| 0.003 | 0.14 | 0.018 | Egl nine homolog 3 inhibitor | 0.018 0.004 CHEMBL3706457 | CHEMBL3706457 | |
| 0.054 | 0.191 | 0.139 | DNA polymerase I inhibitor | 0.122 0.067 CHEMBL3706458 0.123 0.066 CHEMBL3706463 0.139 0.055 CHEMBL3706462 | CHEMBL3706462 | |
| 0.004 | 0.143 | 0.026 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.026 0.021 CHEMBL3706457 | CHEMBL3706457 | |
| 0.065 | 0.204 | 0.114 | TRPA1 agonist | 0.114 0.066 CHEMBL3706457 | CHEMBL3706457 | |
| 0.017 | 0.156 | 0.081 | Dihydroorotate dehydrogenase inhibitor | 0.081 0.017 CHEMBL3706457 | CHEMBL3706457 | |
| 0.025 | 0.165 | 0.07 | Cytokine production stimulant | 0.07 0.007 CHEMBL3706457 0.046 0.041 CHEMBL3706463 0.046 0.039 CHEMBL3706462 | CHEMBL3706457 | |
| 0.026 | 0.168 | 0.143 | Toll-Like receptor 7 antagonist | 0.143 0.007 CHEMBL3706457 | CHEMBL3706457 | |
| 0.083 | 0.226 | 0.141 | Insulin secretagoues | 0.141 0.084 CHEMBL3706458 | CHEMBL3706458 | |
| 0.115 | 0.258 | 0.27 | Superoxide dismutase inhibitor | 0.27 0.063 CHEMBL3706457 | CHEMBL3706457 | |
| 0.016 | 0.16 | 0.094 | Xanthine dehydrogenase inhibitor | 0.094 0.018 CHEMBL3706457 | CHEMBL3706457 | |
| 0.123 | 0.269 | 0.186 | Hypoxia-inducible factor 1 alpha inhibitor | 0.186 0.169 CHEMBL3706457 | CHEMBL3706457 | |
| 0.036 | 0.181 | 0.103 | Monophenol monooxygenase inhibitor | 0.103 0.073 CHEMBL3706458 0.094 0.08 CHEMBL3706462 | CHEMBL3706458 | |
| 0.016 | 0.164 | 0.031 | Toll-Like receptor 4 agonist | 0.029 0.012 CHEMBL3706458 0.029 0.013 CHEMBL3706463 0.031 0.011 CHEMBL3706462 | CHEMBL3706462 | |
| 0.061 | 0.209 | 0.088 | Glutamate release inhibitor | 0.088 0.067 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.159 | 0.04 | Nicotinic acid receptor agonist | 0.04 0.021 CHEMBL3706457 | CHEMBL3706457 | |
| 0.088 | 0.237 | 0.24 | Tumour necrosis factor antagonist | 0.24 0.034 CHEMBL3706457 | CHEMBL3706457 | |
| 0.008 | 0.159 | 0.026 | Corticotropin releasing factor 1 receptor antagonist | 0.026 0.013 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.165 | 0.027 | Vanilloid 2 agonist | 0.027 0.014 CHEMBL3706457 | CHEMBL3706457 | |
| 0.011 | 0.169 | 0.042 | Glutamate (mGluR group II) antagonist | 0.042 0.022 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.165 | 0.044 | Sodium/glucose cotransporter 2 inhibitor | 0.027 0.016 CHEMBL3706458 0.035 0.01 CHEMBL3706463 0.044 0.008 CHEMBL3706462 | CHEMBL3706462 | |
| 0.016 | 0.175 | 0.031 | Glutamate (mGluR4) agonist | 0.031 0.029 CHEMBL3706457 | CHEMBL3706457 | |
| 0.119 | 0.277 | 0.186 | Transcription factor STAT3 inhibitor | 0.186 0.154 CHEMBL3706457 | CHEMBL3706457 | |
| 0.056 | 0.216 | 0.188 | Thrombolytic | 0.162 0.073 CHEMBL3706458 0.171 0.067 CHEMBL3706463 0.188 0.058 CHEMBL3706462 | CHEMBL3706462 | |
| 0.081 | 0.246 | 0.221 | Interleukin agonist | 0.221 0.102 CHEMBL3706457 0.22 0.103 CHEMBL3706458 0.195 0.125 CHEMBL3706463 0.209 0.112 CHEMBL3706462 | CHEMBL3706457 | |
| 0.019 | 0.185 | 0.137 | Antineoplastic antibiotic | 0.137 0.034 CHEMBL3706458 0.119 0.039 CHEMBL3706463 0.133 0.035 CHEMBL3706462 | CHEMBL3706458 | |
| 0.029 | 0.196 | 0.071 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.071 0.06 CHEMBL3706457 | CHEMBL3706457 | |
| 0.015 | 0.183 | 0.034 | Glucosylceramidase stimulant | 0.034 0.008 CHEMBL3706457 | CHEMBL3706457 | |
| 0.074 | 0.242 | 0.157 | Hexokinase inhibitor | 0.157 0.071 CHEMBL3706457 | CHEMBL3706457 | |
| 0.093 | 0.262 | 0.324 | Vasodilator | 0.275 0.057 CHEMBL3706458 0.155 0.149 CHEMBL3706459 0.314 0.044 CHEMBL3706463 0.324 0.041 CHEMBL3706462 | CHEMBL3706462 | |
| 0.047 | 0.218 | 0.09 | Interleukin 1 beta converting enzyme inhibitor | 0.09 0.071 CHEMBL3706457 | CHEMBL3706457 | |
| 0.006 | 0.179 | 0.031 | Glutamate (mGluR2) antagonist | 0.031 0.019 CHEMBL3706457 | CHEMBL3706457 | |
| 0.001 | 0.175 | 0.017 | DNA topoisomerase III inhibitor | 0.017 0.002 CHEMBL3706457 | CHEMBL3706457 | |
| 0.085 | 0.259 | 0.198 | Spasmolytic | 0.169 0.146 CHEMBL3706460 0.165 0.15 CHEMBL3706463 0.184 0.134 CHEMBL3706464 0.198 0.121 CHEMBL3706462 | CHEMBL3706462 | |
| 0.049 | 0.223 | 0.103 | Carbonic anhydrase III inhibitor | 0.103 0.059 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.187 | 0.048 | Antimetabolite | 0.048 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.027 | 0.206 | 0.06 | Beta adrenoreceptor antagonist | 0.06 0.055 CHEMBL3706457 | CHEMBL3706457 | |
| 0.008 | 0.192 | 0.037 | Sodium/glucose cotransporter inhibitor | 0.026 0.017 CHEMBL3706458 0.03 0.011 CHEMBL3706463 0.037 0.008 CHEMBL3706462 | CHEMBL3706462 | |
| 0.015 | 0.2 | 0.027 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.027 0.016 CHEMBL3706457 | CHEMBL3706457 | |
| 0.017 | 0.203 | 0.037 | Acid-sensing ion channel blocker | 0.037 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.204 | 0.045 | Thymidine kinase inhibitor | 0.045 0.023 CHEMBL3706457 | CHEMBL3706457 | |
| 0.135 | 0.321 | 0.556 | GABA C receptor rho-3 antagonist | 0.556 0.013 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.205 | 0.063 | Antibiotic Aminoglycoside-like | 0.059 0.009 CHEMBL3706458 0.059 0.009 CHEMBL3706463 0.063 0.008 CHEMBL3706462 | CHEMBL3706462 | |
| 0.018 | 0.208 | 0.039 | Glutamate (mGluR group III) agonist | 0.039 0.035 CHEMBL3706457 | CHEMBL3706457 | |
| 0.024 | 0.214 | 0.055 | Glucose-6-phosphate translocase inhibitor | 0.053 0.033 CHEMBL3706458 0.049 0.042 CHEMBL3706463 0.055 0.03 CHEMBL3706462 | CHEMBL3706462 | |
| 0.004 | 0.198 | 0.022 | Nicotinic acid receptor 1 antagonist | 0.022 0.007 CHEMBL3706457 | CHEMBL3706457 | |
| 0.138 | 0.333 | 0.424 | Interleukin 2 agonist | 0.404 0.026 CHEMBL3706458 0.2 0.19 CHEMBL3706461 0.406 0.026 CHEMBL3706463 0.208 0.176 CHEMBL3706464 0.424 0.021 CHEMBL3706462 | CHEMBL3706462 | |
| 0.009 | 0.204 | 0.036 | Dihydropteroate synthase inhibitor | 0.036 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.227 | 0.07 | Macrophage migration inhibitory factor inhibitor | 0.07 0.067 CHEMBL3706457 | CHEMBL3706457 | |
| 0.037 | 0.235 | 0.168 | Creatine kinase inhibitor | 0.168 0.018 CHEMBL3706457 | CHEMBL3706457 | |
| 0.003 | 0.203 | 0.013 | Egl nine homolog 1 inhibitor | 0.013 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.086 | 0.288 | 0.191 | Neurotrophic factor enhancer | 0.191 0.086 CHEMBL3706457 | CHEMBL3706457 | |
| 0.074 | 0.276 | 0.147 | Hemostatic | 0.147 0.072 CHEMBL3706458 0.131 0.094 CHEMBL3706463 0.13 0.096 CHEMBL3706462 | CHEMBL3706458 | |
| 0.029 | 0.232 | 0.197 | M18 aspartyl aminopeptidase inhibitor | 0.197 0.034 CHEMBL3706457 | CHEMBL3706457 | |
| 0.035 | 0.241 | 0.057 | Immunoglobulin Fc receptor antagonist | 0.057 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.03 | 0.237 | 0.092 | Glycine receptor antagonist | 0.092 0.04 CHEMBL3706457 | CHEMBL3706457 | |
| 0.011 | 0.221 | 0.061 | Thymidylate synthase inhibitor | 0.061 0.017 CHEMBL3706457 | CHEMBL3706457 | |
| 0.028 | 0.239 | 0.121 | Potassium channel (Ca-activated) activator | 0.121 0.041 CHEMBL3706457 | CHEMBL3706457 | |
| 0.004 | 0.216 | 0.034 | Orexin receptor 2 antagonist | 0.034 0.027 CHEMBL3706457 | CHEMBL3706457 | |
| 0.066 | 0.283 | 0.17 | Neuropeptide Y1 antagonist | 0.17 0.039 CHEMBL3706457 | CHEMBL3706457 | |
| 0.03 | 0.248 | 0.059 | Beta 3 adrenoreceptor antagonist | 0.059 0.058 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.226 | 0.06 | Carbonic anhydrase VB inhibitor | 0.06 0.035 CHEMBL3706457 | CHEMBL3706457 | |
| 0.036 | 0.255 | 0.111 | Prolactin inhibitor | 0.111 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.005 | 0.224 | 0.13 | Purinergic P2Y12 antagonist | 0.13 0.004 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.238 | 0.057 | Androgen agonist | 0.057 0.046 CHEMBL3706457 | CHEMBL3706457 | |
| 0.025 | 0.245 | 0.073 | Dihydroorotate oxidase inhibitor | 0.073 0.015 CHEMBL3706457 | CHEMBL3706457 | |
| 0.04 | 0.259 | 0.146 | Alkylator | 0.127 0.062 CHEMBL3706458 0.13 0.059 CHEMBL3706463 0.146 0.048 CHEMBL3706462 | CHEMBL3706462 | |
| 0.027 | 0.248 | 0.164 | Glucosylceramidase inhibitor | 0.164 0.004 CHEMBL3706457 | CHEMBL3706457 | |
| 0.063 | 0.287 | 0.121 | Sphingosine 1-phosphate receptor 4 antagonist | 0.121 0.071 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.231 | 0.054 | Potassium channel small-conductance Ca-activated activator | 0.054 0.01 CHEMBL3706457 | CHEMBL3706457 | |
| 0.079 | 0.308 | 0.439 | Antioxidant | 0.437 0.029 CHEMBL3706458 0.408 0.034 CHEMBL3706463 0.439 0.029 CHEMBL3706462 | CHEMBL3706462 | |
| 0.013 | 0.242 | 0.043 | Nerve growth factor antagonist | 0.043 0.029 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.245 | 0.061 | Adenosine A2a receptor antagonist | 0.061 0.044 CHEMBL3706457 | CHEMBL3706457 | |
| 0.08 | 0.319 | 0.165 | Sphingosine 1-phosphate receptor 5 antagonist | 0.165 0.04 CHEMBL3706457 | CHEMBL3706457 | |
| 0.032 | 0.27 | 0.097 | Caspase 7 inhibitor | 0.097 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.039 | 0.279 | 0.086 | Bile acid receptor antagonist | 0.086 0.085 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.253 | 0.021 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.021 0.015 CHEMBL3706457 | CHEMBL3706457 | |
| 0.091 | 0.338 | 0.162 | Neurotensin receptor agonist | 0.162 0.075 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.26 | 0.295 | Phosphodiesterase 2A inhibitor | 0.295 0.003 CHEMBL3706457 | CHEMBL3706457 | |
| 0.048 | 0.301 | 0.164 | Cell adhesion inhibitor | 0.164 0.038 CHEMBL3706458 0.127 0.06 CHEMBL3706463 0.15 0.047 CHEMBL3706462 | CHEMBL3706458 | |
| 0.008 | 0.263 | 0.035 | Purinergic P2Y15 antagonist | 0.035 0.01 CHEMBL3706457 | CHEMBL3706457 | |
| 0.044 | 0.302 | 0.104 | Cathepsin H inhibitor | 0.104 0.099 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.27 | 0.052 | Thymidine phosphorylase inhibitor | 0.052 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.036 | 0.296 | 0.081 | Estrogen receptor alpha antagonist | 0.081 0.047 CHEMBL3706457 | CHEMBL3706457 | |
| 0.015 | 0.276 | 0.068 | Carbonic anhydrase V inhibitor | 0.068 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.093 | 0.355 | 0.29 | 5 Hydroxytryptamine release stimulant | 0.29 0.073 CHEMBL3706457 | CHEMBL3706457 | |
| 0.008 | 0.271 | 0.306 | Phosphodiesterase II inhibitor | 0.306 0.003 CHEMBL3706457 | CHEMBL3706457 | |
| 0.174 | 0.438 | 0.451 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.451 0.061 CHEMBL3706457 | CHEMBL3706457 | |
| 0.069 | 0.338 | 0.136 | Pregnane X receptor agonist | 0.136 0.083 CHEMBL3706457 | CHEMBL3706457 | |
| 0.065 | 0.334 | 0.159 | DNA repair enzyme inhibitor | 0.129 0.057 CHEMBL3706457 0.133 0.051 CHEMBL3706458 0.146 0.035 CHEMBL3706463 0.159 0.024 CHEMBL3706462 | CHEMBL3706462 | |
| 0.005 | 0.277 | 0.049 | Geranyltranstransferase inhibitor | 0.049 0.024 CHEMBL3706457 | CHEMBL3706457 | |
| 0.043 | 0.316 | 0.133 | Pyruvate kinase inhibitor | 0.133 0.132 CHEMBL3706457 | CHEMBL3706457 | |
| 0.025 | 0.298 | 0.078 | Corticotropin releasing factor 2 receptor antagonist | 0.078 0.019 CHEMBL3706457 | CHEMBL3706457 | |
| 0.028 | 0.304 | 0.093 | Adenosine A3 receptor antagonist | 0.093 0.03 CHEMBL3706457 | CHEMBL3706457 | |
| 0.017 | 0.293 | 0.067 | Carbonic anhydrase VA inhibitor | 0.067 0.05 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.286 | 0.059 | Adenosine A1 receptor antagonist | 0.059 0.04 CHEMBL3706457 | CHEMBL3706457 | |
| 0.016 | 0.294 | 0.056 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.056 0.034 CHEMBL3706457 | CHEMBL3706457 | |
| 0.079 | 0.357 | 0.455 | Transcription factor NF kappa B inhibitor | 0.455 0.052 CHEMBL3706458 0.442 0.055 CHEMBL3706463 0.455 0.052 CHEMBL3706462 | CHEMBL3706462 | |
| 0.092 | 0.374 | 0.225 | Neuropeptide Y2 antagonist | 0.225 0.083 CHEMBL3706457 | CHEMBL3706457 | |
| 0.043 | 0.326 | 0.099 | Carbonic anhydrase XV inhibitor | 0.099 0.069 CHEMBL3706457 | CHEMBL3706457 | |
| 0.032 | 0.317 | 0.076 | Cell adhesion molecule inhibitor | 0.076 0.059 CHEMBL3706458 | CHEMBL3706458 | |
| 0.007 | 0.293 | 0.058 | Purinergic P2Y antagonist | 0.058 0.021 CHEMBL3706457 | CHEMBL3706457 | |
| 0.012 | 0.299 | 0.043 | Glutamate (mGluR1a) antagonist | 0.043 0.026 CHEMBL3706457 | CHEMBL3706457 | |
| 0.004 | 0.295 | 0.038 | Nicotinic alpha4beta2 receptor agonist | 0.038 0.009 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.319 | 0.04 | CF transmembrane conductance regulator antagonist | 0.04 0.027 CHEMBL3706457 | CHEMBL3706457 | |
| 0.026 | 0.326 | 0.081 | Orexin receptor 1 antagonist | 0.081 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.01 | 0.31 | 0.027 | Estrogen-related receptor gamma antagonist | 0.027 0.022 CHEMBL3706457 | CHEMBL3706457 | |
| 0.044 | 0.347 | 0.082 | Ca(v)3.1 blocker | 0.082 0.054 CHEMBL3706457 | CHEMBL3706457 | |
| 0.023 | 0.328 | 0.105 | M17 leucyl aminopeptidase inhibitor | 0.105 0.095 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.339 | 0.14 | Alkaline phosphatase inhibitor | 0.14 0.067 CHEMBL3706457 | CHEMBL3706457 | |
| 0.021 | 0.329 | 0.082 | Alcohol dehydrogenase inhibitor | 0.082 0.076 CHEMBL3706457 | CHEMBL3706457 | |
| 0.02 | 0.33 | 0.07 | Orexin receptor antagonist | 0.07 0.041 CHEMBL3706457 | CHEMBL3706457 | |
| 0.037 | 0.347 | 0.092 | mTOR complex 2 inhibitor | 0.092 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.04 | 0.35 | 0.53 | Angiogenesis stimulant | 0.505 0.011 CHEMBL3706458 0.474 0.013 CHEMBL3706463 0.53 0.01 CHEMBL3706462 | CHEMBL3706462 | |
| 0.065 | 0.376 | 0.151 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.151 0.143 CHEMBL3706460 | CHEMBL3706460 | |
| 0.007 | 0.321 | 0.048 | Dopamine D5 agonist | 0.048 0.019 CHEMBL3706457 | CHEMBL3706457 | |
| 0.034 | 0.348 | 0.073 | Vanilloid 4 agonist | 0.073 0.057 CHEMBL3706457 | CHEMBL3706457 | |
| 0.012 | 0.33 | 0.041 | DNA polymerase III inhibitor | 0.041 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.089 | 0.409 | 0.134 | CC chemokine 6 receptor antagonist | 0.128 0.078 CHEMBL3706457 0.134 0.057 CHEMBL3706458 0.128 0.077 CHEMBL3706463 0.127 0.083 CHEMBL3706462 | CHEMBL3706458 | |
| 0.048 | 0.368 | 0.482 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.482 0.022 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.339 | 0.101 | Inducible nitric-oxide synthase inhibitor | 0.101 0.036 CHEMBL3706457 | CHEMBL3706457 | |
| 0.037 | 0.358 | 0.095 | Lanosterol 14 alpha demethylase inhibitor | 0.095 0.063 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.34 | 0.089 | Phospholipase D inhibitor | 0.089 0.023 CHEMBL3706457 | CHEMBL3706457 | |
| 0.051 | 0.374 | 0.276 | Platelet adhesion inhibitor | 0.276 0.041 CHEMBL3706458 0.267 0.044 CHEMBL3706463 0.276 0.041 CHEMBL3706462 | CHEMBL3706462 | |
| 0.041 | 0.367 | 0.089 | Phosphodiesterase 6D inhibitor | 0.089 0.078 CHEMBL3706457 | CHEMBL3706457 | |
| 0.02 | 0.349 | 0.063 | Factor IXa inhibitor | 0.055 0.032 CHEMBL3706458 0.059 0.028 CHEMBL3706463 0.063 0.024 CHEMBL3706462 | CHEMBL3706462 | |
| 0.048 | 0.378 | 0.156 | Platelet antagonist | 0.156 0.138 CHEMBL3706462 | CHEMBL3706462 | |
| 0.018 | 0.352 | 0.083 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.083 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.027 | 0.368 | 0.129 | Uric acid excretion stimulant | 0.129 0.033 CHEMBL3706457 | CHEMBL3706457 | |
| 0.029 | 0.372 | 0.119 | MAP kinase kinase 1 inhibitor | 0.119 0.036 CHEMBL3706457 | CHEMBL3706457 | |
| 0.033 | 0.376 | 0.086 | MAP kinase kinase 7 inhibitor | 0.086 0.031 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.376 | 0.214 | Aryl hydrocarbon receptor agonist | 0.214 0.095 CHEMBL3706457 | CHEMBL3706457 | |
| 0.035 | 0.381 | 0.115 | Antibacterial (Helicobacter pylori) | 0.115 0.088 CHEMBL3706457 | CHEMBL3706457 | |
| 0.014 | 0.361 | 0.071 | Protein kinase C beta inhibitor | 0.071 0.046 CHEMBL3706457 | CHEMBL3706457 | |
| 0.033 | 0.382 | 0.081 | Bromodomain-containing protein 2 inhibitor | 0.081 0.074 CHEMBL3706457 | CHEMBL3706457 | |
| 0.033 | 0.382 | 0.143 | Beta amyloid protein antagonist | 0.143 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.034 | 0.384 | 0.139 | Toll-Like receptor antagonist | 0.139 0.064 CHEMBL3706457 | CHEMBL3706457 | |
| 0.015 | 0.369 | 0.076 | CYP2A6 inhibitor | 0.076 0.052 CHEMBL3706457 | CHEMBL3706457 | |
| 0.02 | 0.377 | 0.107 | Histamine N-methyltransferase inhibitor | 0.107 0.04 CHEMBL3706457 | CHEMBL3706457 | |
| 0.092 | 0.455 | 0.343 | Apoptosis antagonist | 0.326 0.069 CHEMBL3706458 0.327 0.068 CHEMBL3706463 0.343 0.059 CHEMBL3706462 | CHEMBL3706462 | |
| 0.015 | 0.38 | 0.049 | Dopamine beta hydroxylase inhibitor | 0.049 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.004 | 0.376 | 0.053 | Glutamate (mGluR1) antagonist | 0.053 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.006 | 0.379 | 0.046 | Alpha 1d adrenoreceptor agonist | 0.046 0.019 CHEMBL3706457 | CHEMBL3706457 | |
| 0.045 | 0.427 | 0.172 | P-glycoprotein inhibitor | 0.165 0.096 CHEMBL3706458 0.162 0.1 CHEMBL3706463 0.172 0.087 CHEMBL3706462 | CHEMBL3706462 | |
| 0.026 | 0.41 | 0.11 | Beta glucuronidase inhibitor | 0.11 0.056 CHEMBL3706458 | CHEMBL3706458 | |
| 0.003 | 0.394 | 0.028 | Nicotinic alpha3beta4 receptor agonist | 0.028 0.024 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.411 | 0.084 | Potassium channel activator | 0.084 0.068 CHEMBL3706457 | CHEMBL3706457 | |
| 0.005 | 0.408 | 0.8 | Phosphodiesterase 3B inhibitor | 0.8 0.001 CHEMBL3706457 | CHEMBL3706457 | |
| 0.038 | 0.443 | 0.355 | Free radical scavenger | 0.35 0.039 CHEMBL3706458 0.329 0.044 CHEMBL3706463 0.355 0.038 CHEMBL3706462 | CHEMBL3706462 | |
| 0.023 | 0.437 | 0.483 | Phosphodiesterase inhibitor | 0.483 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.046 | 0.472 | 0.239 | DNA damaging | 0.239 0.087 CHEMBL3706457 | CHEMBL3706457 | |
| 0.045 | 0.472 | 0.101 | Interleukin 2 antagonist | 0.101 0.088 CHEMBL3706457 | CHEMBL3706457 | |
| 0.011 | 0.442 | 0.745 | Phosphodiesterase III inhibitor | 0.745 0.002 CHEMBL3706457 | CHEMBL3706457 | |
| 0.065 | 0.496 | 0.432 | Antibacterial | 0.239 0.187 CHEMBL3706457 0.432 0.063 CHEMBL3706458 0.402 0.076 CHEMBL3706463 0.418 0.069 CHEMBL3706462 | CHEMBL3706458 | |
| 0.032 | 0.464 | 0.179 | Activin receptor-like kinase 4 inhibitor | 0.179 0.018 CHEMBL3706457 | CHEMBL3706457 | |
| 0.022 | 0.461 | 0.168 | Lipid peroxidase inhibitor | 0.168 0.056 CHEMBL3706458 0.142 0.074 CHEMBL3706463 0.148 0.07 CHEMBL3706462 | CHEMBL3706458 | |
| 0.015 | 0.461 | 0.065 | 5 Hydroxytryptamine 3 agonist | 0.065 0.041 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.454 | 0.044 | Histamine H2 receptor agonist | 0.044 0.028 CHEMBL3706457 | CHEMBL3706457 | |
| 0.042 | 0.49 | 0.264 | 12-Lipoxygenase inhibitor | 0.264 0.101 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.477 | 0.193 | 5 Hydroxytryptamine 3A agonist | 0.193 0.017 CHEMBL3706457 | CHEMBL3706457 | |
| 0.035 | 0.494 | 0.443 | Alpha-glucosidase inhibitor | 0.443 0.098 CHEMBL3706457 | CHEMBL3706457 | |
| 0.092 | 0.552 | 0.593 | Antiinflammatory | 0.571 0.062 CHEMBL3706458 0.567 0.063 CHEMBL3706463 0.593 0.055 CHEMBL3706462 | CHEMBL3706462 | |
| 0.005 | 0.465 | 0.056 | GABA receptor antagonist | 0.056 0.036 CHEMBL3706457 | CHEMBL3706457 | |
| 0.005 | 0.466 | 0.026 | Protein 30S ribosomal subunit inhibitor | 0.024 0.017 CHEMBL3706458 0.023 0.018 CHEMBL3706463 0.026 0.015 CHEMBL3706462 | CHEMBL3706462 | |
| 0.005 | 0.471 | 0.054 | GABA A receptor antagonist | 0.054 0.036 CHEMBL3706457 | CHEMBL3706457 | |
| 0.044 | 0.511 | 0.155 | NOS3 expression enhancer | 0.155 0.068 CHEMBL3706458 0.137 0.088 CHEMBL3706463 0.146 0.076 CHEMBL3706462 | CHEMBL3706458 | |
| 0.013 | 0.494 | 0.158 | Glutamate receptor antagonist | 0.158 0.045 CHEMBL3706457 | CHEMBL3706457 | |
| 0.016 | 0.499 | 0.057 | Phosphodiesterase 1A inhibitor | 0.057 0.05 CHEMBL3706457 | CHEMBL3706457 | |
| 0.013 | 0.499 | 0.108 | MAP kinase kinase inhibitor | 0.108 0.086 CHEMBL3706457 | CHEMBL3706457 | |
| 0.031 | 0.517 | 0.494 | Thioredoxin glutathione reductase inhibitor | 0.494 0.03 CHEMBL3706457 | CHEMBL3706457 | |
| 0.014 | 0.503 | 0.096 | Nitric-oxide synthase inhibitor | 0.096 0.066 CHEMBL3706457 | CHEMBL3706457 | |
| 0.044 | 0.534 | 0.4 | Immunosuppressant | 0.4 0.063 CHEMBL3706458 0.375 0.074 CHEMBL3706463 0.393 0.066 CHEMBL3706462 | CHEMBL3706458 | |
| 0.033 | 0.523 | 0.407 | DNA polymerase beta inhibitor | 0.407 0.116 CHEMBL3706457 | CHEMBL3706457 | |
| 0.042 | 0.537 | 0.47 | 15-Lipoxygenase inhibitor | 0.47 0.048 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.514 | 0.095 | Phosphodiesterase 1C inhibitor | 0.095 0.012 CHEMBL3706457 | CHEMBL3706457 | |
| 0.028 | 0.524 | 0.179 | Amyloid beta precursor protein antagonist | 0.179 0.073 CHEMBL3706457 | CHEMBL3706457 | |
| 0.023 | 0.522 | 0.362 | Prostaglandin dehydrogenase inhibitor | 0.362 0.079 CHEMBL3706457 | CHEMBL3706457 | |
| 0.046 | 0.55 | 0.336 | Transcription factor inhibitor | 0.336 0.137 CHEMBL3706457 | CHEMBL3706457 | |
| 0.093 | 0.599 | 0.192 | 5 Hydroxytryptamine 3E antagonist | 0.192 0.076 CHEMBL3706457 | CHEMBL3706457 | |
| 0.009 | 0.517 | 0.097 | HIV-1 reverse transcriptase inhibitor | 0.097 0.032 CHEMBL3706457 | CHEMBL3706457 | |
| 0.034 | 0.55 | 0.244 | Thyroid hormone antagonist | 0.244 0.128 CHEMBL3706457 | CHEMBL3706457 | |
| 0.033 | 0.549 | 0.44 | DNA directed DNA polymerase inhibitor | 0.44 0.101 CHEMBL3706457 | CHEMBL3706457 | |
| 0.028 | 0.544 | 0.388 | Streptokinase A inhibitor | 0.388 0.05 CHEMBL3706457 | CHEMBL3706457 | |
| 0.029 | 0.548 | 0.233 | 5 Hydroxytryptamine 1E antagonist | 0.233 0.093 CHEMBL3706457 | CHEMBL3706457 | |
| 0.012 | 0.534 | 0.156 | Topoisomerase I inhibitor | 0.12 0.055 CHEMBL3706458 0.134 0.048 CHEMBL3706463 0.156 0.039 CHEMBL3706462 | CHEMBL3706462 | |
| 0.034 | 0.556 | 0.229 | Thyroid hormone beta antagonist | 0.229 0.132 CHEMBL3706457 | CHEMBL3706457 | |
| 0.022 | 0.544 | 0.097 | Phosphodiesterase I inhibitor | 0.097 0.048 CHEMBL3706457 | CHEMBL3706457 | |
| 0.037 | 0.571 | 0.086 | CC chemokine 5 receptor agonist | 0.086 0.047 CHEMBL3706457 | CHEMBL3706457 | |
| 0.016 | 0.552 | 0.077 | Phosphodiesterase 1B inhibitor | 0.077 0.025 CHEMBL3706457 | CHEMBL3706457 | |
| 0.022 | 0.565 | 0.132 | Heat shock protein 90 antagonist | 0.132 0.094 CHEMBL3706457 | CHEMBL3706457 | |
| 0.029 | 0.576 | 0.271 | Tumour necrosis factor alpha release inhibitor | 0.264 0.068 CHEMBL3706458 0.25 0.075 CHEMBL3706463 0.271 0.065 CHEMBL3706462 | CHEMBL3706462 | |
| 0.005 | 0.601 | 0.054 | Phosphodiesterase 4C inhibitor | 0.054 0.041 CHEMBL3706457 | CHEMBL3706457 | |
| 0.047 | 0.645 | 0.329 | MAP kinase 1 inhibitor | 0.329 0.151 CHEMBL3706457 | CHEMBL3706457 | |
| 0.019 | 0.637 | 0.159 | Antiamyloidogenic | 0.159 0.135 CHEMBL3706457 | CHEMBL3706457 | |
| 0.014 | 0.644 | 0.165 | Calpain inhibitor | 0.165 0.156 CHEMBL3706457 | CHEMBL3706457 | |
| 0.018 | 0.654 | 0.285 | Calpain 2 inhibitor | 0.285 0.124 CHEMBL3706457 | CHEMBL3706457 | |
| 0.029 | 0.719 | 0.353 | Immunomodulator | 0.246 0.118 CHEMBL3706458 0.318 0.073 CHEMBL3706463 0.353 0.059 CHEMBL3706462 | CHEMBL3706462 | |
| 0.006 | 0.707 | 0.295 | Phosphodiesterase 3A inhibitor | 0.295 0.005 CHEMBL3706457 | CHEMBL3706457 | |
| 0.005 | 0.747 | 0.103 | Purinergic P2 antagonist | 0.103 0.02 CHEMBL3706457 | CHEMBL3706457 | |
| 0.007 | 0.788 | 0.166 | Antimitotic | 0.166 0.107 CHEMBL3706458 | CHEMBL3706458 | |
| 0.011 | 0.874 | 0.429 | Apoptosis agonist | 0.405 0.111 CHEMBL3706458 0.401 0.113 CHEMBL3706463 0.429 0.1 CHEMBL3706462 | CHEMBL3706462 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |