| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.481 | 0.013 | 0.807 | Psychostimulant | 0.215 0.072 CHEMBL3706522 0.52 0.009 CHEMBL3706525 0.391 0.024 CHEMBL3706526 0.807 0.004 CHEMBL3706527 0.41 0.021 CHEMBL3706528 0.34 0.033 CHEMBL3706529 | CHEMBL3706527 | |
| 0.427 | 0.003 | 0.482 | HIV-1 protease inhibitor | 0.079 0.006 CHEMBL3706522 0.101 0.005 CHEMBL3706523 0.335 0.003 CHEMBL3706525 0.047 0.024 CHEMBL3706526 0.482 0.003 CHEMBL3706527 0.364 0.003 CHEMBL3706528 0.304 0.003 CHEMBL3706529 0.06 0.012 CHEMBL3706524 | CHEMBL3706527 | |
| 0.402 | 0.004 | 0.402 | Protease inhibitor | 0.124 0.045 CHEMBL3706522 0.313 0.005 CHEMBL3706523 0.328 0.005 CHEMBL3706525 0.154 0.028 CHEMBL3706526 0.329 0.005 CHEMBL3706527 0.364 0.004 CHEMBL3706528 0.341 0.005 CHEMBL3706529 0.208 0.013 CHEMBL3706524 | ||
| 0.422 | 0.028 | 0.561 | Interleukin antagonist | 0.561 0.015 CHEMBL3706523 0.263 0.057 CHEMBL3706525 0.548 0.016 CHEMBL3706526 0.409 0.029 CHEMBL3706528 0.388 0.033 CHEMBL3706529 0.542 0.016 CHEMBL3706524 | CHEMBL3706523 | |
| 0.315 | 0.004 | 0.315 | Human rhinovirus A protease inhibitor | 0.097 0.017 CHEMBL3706522 0.253 0.005 CHEMBL3706523 0.274 0.004 CHEMBL3706525 0.174 0.007 CHEMBL3706526 0.237 0.005 CHEMBL3706527 0.288 0.004 CHEMBL3706528 0.285 0.004 CHEMBL3706529 0.179 0.007 CHEMBL3706524 | ||
| 0.269 | 0.013 | 0.269 | Proteasome inhibitor | 0.17 0.036 CHEMBL3706522 0.265 0.014 CHEMBL3706523 0.239 0.017 CHEMBL3706525 0.18 0.032 CHEMBL3706526 0.208 0.023 CHEMBL3706527 0.233 0.018 CHEMBL3706528 0.221 0.02 CHEMBL3706529 0.198 0.026 CHEMBL3706524 | ||
| 0.312 | 0.069 | 0.343 | Nootropic | 0.206 0.15 CHEMBL3706522 0.197 0.162 CHEMBL3706523 0.312 0.069 CHEMBL3706525 0.273 0.09 CHEMBL3706528 0.343 0.056 CHEMBL3706529 | CHEMBL3706529 | |
| 0.258 | 0.041 | 0.34 | Growth hormone agonist | 0.2 0.059 CHEMBL3706522 0.303 0.032 CHEMBL3706523 0.282 0.036 CHEMBL3706525 0.34 0.025 CHEMBL3706526 0.24 0.046 CHEMBL3706527 0.283 0.036 CHEMBL3706528 0.25 0.043 CHEMBL3706529 0.314 0.03 CHEMBL3706524 | CHEMBL3706526 | |
| 0.271 | 0.062 | 0.349 | Antiamyloidogenic | 0.211 0.092 CHEMBL3706522 0.202 0.098 CHEMBL3706523 0.224 0.084 CHEMBL3706525 0.349 0.039 CHEMBL3706526 0.213 0.091 CHEMBL3706528 0.154 0.142 CHEMBL3706529 0.214 0.091 CHEMBL3706524 | CHEMBL3706526 | |
| 0.294 | 0.089 | 0.469 | Apoptosis antagonist | 0.24 0.137 CHEMBL3706522 0.348 0.057 CHEMBL3706523 0.409 0.036 CHEMBL3706525 0.328 0.067 CHEMBL3706526 0.234 0.144 CHEMBL3706527 0.335 0.063 CHEMBL3706528 0.266 0.112 CHEMBL3706529 0.469 0.024 CHEMBL3706524 | CHEMBL3706524 | |
| 0.227 | 0.026 | 0.233 | Nav1.2 sodium channel blocker | 0.211 0.031 CHEMBL3706522 0.147 0.059 CHEMBL3706523 0.128 0.074 CHEMBL3706525 0.159 0.052 CHEMBL3706526 0.224 0.027 CHEMBL3706527 0.148 0.058 CHEMBL3706528 0.233 0.025 CHEMBL3706529 | CHEMBL3706529 | |
| 0.257 | 0.09 | 0.402 | Ca(v)3.3 blocker | 0.402 0.005 CHEMBL3706522 0.246 0.107 CHEMBL3706525 0.273 0.069 CHEMBL3706527 0.227 0.139 CHEMBL3706528 0.203 0.185 CHEMBL3706529 | CHEMBL3706522 | |
| 0.207 | 0.049 | 0.395 | Thrombolytic | 0.245 0.035 CHEMBL3706523 0.244 0.035 CHEMBL3706525 0.395 0.012 CHEMBL3706526 0.129 0.1 CHEMBL3706527 0.212 0.046 CHEMBL3706528 0.193 0.055 CHEMBL3706529 0.302 0.024 CHEMBL3706524 | CHEMBL3706526 | |
| 0.192 | 0.039 | 0.334 | Neurotensin receptor agonist | 0.187 0.044 CHEMBL3706522 0.213 0.029 CHEMBL3706523 0.189 0.042 CHEMBL3706525 0.334 0.011 CHEMBL3706526 0.16 0.079 CHEMBL3706527 0.143 0.119 CHEMBL3706528 0.164 0.071 CHEMBL3706529 0.273 0.018 CHEMBL3706524 | CHEMBL3706526 | |
| 0.258 | 0.109 | 0.329 | Immunomodulator | 0.247 0.117 CHEMBL3706523 0.273 0.098 CHEMBL3706525 0.329 0.068 CHEMBL3706526 0.315 0.074 CHEMBL3706527 0.307 0.078 CHEMBL3706528 0.294 0.086 CHEMBL3706529 0.213 0.149 CHEMBL3706524 | CHEMBL3706526 | |
| 0.185 | 0.046 | 0.319 | Catenin beta inhibitor | 0.152 0.102 CHEMBL3706522 0.254 0.01 CHEMBL3706523 0.223 0.019 CHEMBL3706525 0.277 0.007 CHEMBL3706526 0.164 0.076 CHEMBL3706528 0.178 0.054 CHEMBL3706529 0.319 0.005 CHEMBL3706524 | CHEMBL3706524 | |
| 0.187 | 0.058 | 0.28 | Anticoagulant | 0.205 0.051 CHEMBL3706523 0.213 0.049 CHEMBL3706525 0.28 0.032 CHEMBL3706526 0.17 0.066 CHEMBL3706527 0.169 0.067 CHEMBL3706528 0.159 0.073 CHEMBL3706529 0.174 0.064 CHEMBL3706524 | CHEMBL3706526 | |
| 0.226 | 0.098 | 0.309 | Cardiotonic | 0.255 0.079 CHEMBL3706522 0.229 0.097 CHEMBL3706525 0.309 0.052 CHEMBL3706527 0.294 0.059 CHEMBL3706528 0.187 0.132 CHEMBL3706529 | CHEMBL3706527 | |
| 0.143 | 0.015 | 0.148 | Neuropeptide agonist | 0.05 0.043 CHEMBL3706522 0.148 0.014 CHEMBL3706523 0.089 0.029 CHEMBL3706525 0.134 0.018 CHEMBL3706526 0.098 0.027 CHEMBL3706527 0.132 0.019 CHEMBL3706528 0.14 0.016 CHEMBL3706529 0.147 0.014 CHEMBL3706524 | CHEMBL3706523 | |
| 0.213 | 0.088 | 0.363 | Angiogenesis stimulant | 0.292 0.052 CHEMBL3706523 0.178 0.106 CHEMBL3706525 0.363 0.029 CHEMBL3706526 0.261 0.065 CHEMBL3706528 0.223 0.083 CHEMBL3706529 0.334 0.037 CHEMBL3706524 | CHEMBL3706526 | |
| 0.248 | 0.128 | 0.393 | Antithrombotic | 0.256 0.121 CHEMBL3706523 0.367 0.059 CHEMBL3706525 0.286 0.099 CHEMBL3706526 0.393 0.051 CHEMBL3706527 0.303 0.086 CHEMBL3706528 0.192 0.187 CHEMBL3706524 | CHEMBL3706527 | |
| 0.206 | 0.092 | 0.277 | Peptidyltransferase inhibitor | 0.212 0.085 CHEMBL3706523 0.181 0.127 CHEMBL3706525 0.249 0.051 CHEMBL3706526 0.244 0.055 CHEMBL3706527 0.243 0.056 CHEMBL3706528 0.277 0.034 CHEMBL3706529 0.226 0.07 CHEMBL3706524 | CHEMBL3706529 | |
| 0.242 | 0.128 | 0.352 | Interleukin 2 agonist | 0.282 0.088 CHEMBL3706523 0.316 0.063 CHEMBL3706525 0.352 0.045 CHEMBL3706526 0.282 0.088 CHEMBL3706527 0.293 0.079 CHEMBL3706528 0.244 0.126 CHEMBL3706529 0.306 0.069 CHEMBL3706524 | CHEMBL3706526 | |
| 0.128 | 0.016 | 0.188 | 3C-Like protease (SARS coronavirus) inhibitor | 0.188 0.005 CHEMBL3706523 0.116 0.021 CHEMBL3706525 0.093 0.042 CHEMBL3706526 0.098 0.036 CHEMBL3706527 0.116 0.021 CHEMBL3706528 0.118 0.02 CHEMBL3706529 0.121 0.019 CHEMBL3706524 | CHEMBL3706523 | |
| 0.118 | 0.007 | 0.304 | Gonadotropin-releasing hormone receptor agonist | 0.304 0.003 CHEMBL3706522 0.062 0.036 CHEMBL3706523 0.098 0.011 CHEMBL3706525 0.057 0.047 CHEMBL3706526 0.119 0.006 CHEMBL3706527 0.101 0.01 CHEMBL3706528 0.118 0.007 CHEMBL3706529 0.066 0.03 CHEMBL3706524 | CHEMBL3706522 | |
| 0.138 | 0.029 | 0.185 | Opioid antagonist | 0.083 0.065 CHEMBL3706523 0.121 0.036 CHEMBL3706525 0.083 0.065 CHEMBL3706526 0.185 0.017 CHEMBL3706527 0.122 0.036 CHEMBL3706528 0.123 0.035 CHEMBL3706529 0.088 0.059 CHEMBL3706524 | CHEMBL3706527 | |
| 0.217 | 0.114 | 0.34 | Transcription factor STAT3 inhibitor | 0.34 0.036 CHEMBL3706523 0.333 0.039 CHEMBL3706526 0.198 0.137 CHEMBL3706528 0.269 0.07 CHEMBL3706524 | CHEMBL3706523 | |
| 0.167 | 0.063 | 0.276 | Diuretic | 0.17 0.061 CHEMBL3706522 0.276 0.027 CHEMBL3706525 0.167 0.064 CHEMBL3706526 0.249 0.031 CHEMBL3706527 0.151 0.077 CHEMBL3706528 0.21 0.041 CHEMBL3706529 | CHEMBL3706525 | |
| 0.116 | 0.014 | 0.147 | Cathepsin D inhibitor | 0.147 0.008 CHEMBL3706523 0.103 0.018 CHEMBL3706525 0.047 0.046 CHEMBL3706526 0.06 0.034 CHEMBL3706527 0.103 0.018 CHEMBL3706528 0.114 0.014 CHEMBL3706529 0.071 0.029 CHEMBL3706524 | CHEMBL3706523 | |
| 0.121 | 0.022 | 0.423 | Hematopoietic | 0.133 0.018 CHEMBL3706522 0.179 0.012 CHEMBL3706523 0.129 0.019 CHEMBL3706525 0.423 0.004 CHEMBL3706526 0.112 0.026 CHEMBL3706528 0.117 0.023 CHEMBL3706529 0.193 0.01 CHEMBL3706524 | CHEMBL3706526 | |
| 0.101 | 0.009 | 0.231 | Dipeptidyl peptidase inhibitor | 0.054 0.034 CHEMBL3706525 0.231 0.003 CHEMBL3706527 0.061 0.024 CHEMBL3706528 0.097 0.009 CHEMBL3706529 0.057 0.03 CHEMBL3706524 | CHEMBL3706527 | |
| 0.13 | 0.044 | 0.154 | Nav1.4 sodium channel blocker | 0.142 0.037 CHEMBL3706523 0.127 0.046 CHEMBL3706525 0.149 0.034 CHEMBL3706526 0.106 0.068 CHEMBL3706527 0.118 0.054 CHEMBL3706528 0.122 0.05 CHEMBL3706529 0.154 0.032 CHEMBL3706524 | CHEMBL3706524 | |
| 0.089 | 0.008 | 0.101 | HCV NS3/NS4A protease inhibitor | 0.058 0.023 CHEMBL3706522 0.046 0.041 CHEMBL3706523 0.101 0.004 CHEMBL3706525 0.065 0.017 CHEMBL3706526 0.085 0.009 CHEMBL3706527 0.083 0.01 CHEMBL3706528 0.063 0.018 CHEMBL3706529 | CHEMBL3706525 | |
| 0.123 | 0.043 | 0.167 | Falcipain inhibitor | 0.167 0.024 CHEMBL3706523 0.096 0.058 CHEMBL3706525 0.094 0.059 CHEMBL3706526 0.094 0.059 CHEMBL3706528 0.103 0.052 CHEMBL3706529 0.161 0.026 CHEMBL3706524 | CHEMBL3706523 | |
| 0.108 | 0.029 | 0.158 | Opioid mu receptor antagonist | 0.094 0.034 CHEMBL3706525 0.158 0.016 CHEMBL3706527 0.093 0.034 CHEMBL3706528 0.095 0.034 CHEMBL3706529 0.058 0.056 CHEMBL3706524 | CHEMBL3706527 | |
| 0.1 | 0.022 | 0.108 | Glucagon-like peptide 1 agonist | 0.096 0.024 CHEMBL3706523 0.1 0.022 CHEMBL3706525 0.108 0.018 CHEMBL3706526 0.089 0.029 CHEMBL3706527 0.093 0.026 CHEMBL3706528 0.098 0.023 CHEMBL3706529 0.095 0.025 CHEMBL3706524 | CHEMBL3706526 | |
| 0.083 | 0.005 | 0.101 | Plasmepsin II inhibitor | 0.054 0.015 CHEMBL3706522 0.101 0.004 CHEMBL3706523 0.064 0.01 CHEMBL3706525 0.044 0.023 CHEMBL3706526 0.043 0.026 CHEMBL3706527 0.064 0.01 CHEMBL3706528 0.063 0.01 CHEMBL3706529 0.067 0.009 CHEMBL3706524 | CHEMBL3706523 | |
| 0.096 | 0.021 | 0.125 | Secretase beta inhibitor | 0.089 0.026 CHEMBL3706522 0.125 0.009 CHEMBL3706523 0.064 0.061 CHEMBL3706525 0.084 0.031 CHEMBL3706526 0.071 0.047 CHEMBL3706528 0.095 0.021 CHEMBL3706529 0.09 0.025 CHEMBL3706524 | CHEMBL3706523 | |
| 0.205 | 0.131 | 0.362 | Transcription factor STAT inhibitor | 0.346 0.036 CHEMBL3706523 0.362 0.03 CHEMBL3706526 0.185 0.16 CHEMBL3706528 0.357 0.032 CHEMBL3706524 | CHEMBL3706526 | |
| 0.116 | 0.043 | 0.2 | Factor V inhibitor | 0.2 0.005 CHEMBL3706523 0.117 0.042 CHEMBL3706525 0.106 0.057 CHEMBL3706526 0.107 0.055 CHEMBL3706527 0.111 0.049 CHEMBL3706528 0.112 0.048 CHEMBL3706529 0.129 0.031 CHEMBL3706524 | CHEMBL3706523 | |
| 0.099 | 0.03 | 0.157 | Opioid delta receptor antagonist | 0.055 0.05 CHEMBL3706523 0.089 0.033 CHEMBL3706525 0.055 0.05 CHEMBL3706526 0.157 0.018 CHEMBL3706527 0.082 0.036 CHEMBL3706528 0.083 0.035 CHEMBL3706529 0.066 0.043 CHEMBL3706524 | CHEMBL3706527 | |
| 0.087 | 0.019 | 0.114 | Cathepsin E inhibitor | 0.114 0.01 CHEMBL3706523 0.073 0.027 CHEMBL3706525 0.076 0.025 CHEMBL3706526 0.056 0.048 CHEMBL3706527 0.077 0.024 CHEMBL3706528 0.081 0.022 CHEMBL3706529 0.087 0.018 CHEMBL3706524 | CHEMBL3706523 | |
| 0.085 | 0.018 | 0.095 | Protease activated receptor 1 antagonist | 0.073 0.021 CHEMBL3706523 0.063 0.026 CHEMBL3706525 0.051 0.032 CHEMBL3706526 0.073 0.021 CHEMBL3706528 0.07 0.023 CHEMBL3706529 0.095 0.015 CHEMBL3706524 | CHEMBL3706524 | |
| 0.141 | 0.079 | 0.219 | Hemostatic | 0.133 0.091 CHEMBL3706522 0.219 0.027 CHEMBL3706526 0.136 0.087 CHEMBL3706527 0.133 0.091 CHEMBL3706528 0.119 0.115 CHEMBL3706529 0.19 0.037 CHEMBL3706524 | CHEMBL3706526 | |
| 0.081 | 0.025 | 0.108 | Bombesin 1 receptor agonist | 0.054 0.049 CHEMBL3706522 0.092 0.02 CHEMBL3706523 0.053 0.051 CHEMBL3706525 0.074 0.029 CHEMBL3706526 0.068 0.033 CHEMBL3706528 0.077 0.027 CHEMBL3706529 0.108 0.015 CHEMBL3706524 | CHEMBL3706524 | |
| 0.12 | 0.065 | 0.347 | Cell adhesion inhibitor | 0.105 0.081 CHEMBL3706523 0.187 0.028 CHEMBL3706525 0.347 0.007 CHEMBL3706526 0.099 0.09 CHEMBL3706527 0.124 0.062 CHEMBL3706528 0.102 0.086 CHEMBL3706529 0.173 0.034 CHEMBL3706524 | CHEMBL3706526 | |
| 0.187 | 0.133 | 0.466 | Interleukin agonist | 0.278 0.06 CHEMBL3706522 0.266 0.067 CHEMBL3706523 0.239 0.087 CHEMBL3706525 0.466 0.011 CHEMBL3706526 0.231 0.093 CHEMBL3706527 0.278 0.06 CHEMBL3706528 0.28 0.059 CHEMBL3706529 0.318 0.04 CHEMBL3706524 | CHEMBL3706526 | |
| 0.111 | 0.06 | 0.187 | Falcipain 3 inhibitor | 0.187 0.022 CHEMBL3706523 0.109 0.062 CHEMBL3706525 0.102 0.068 CHEMBL3706526 0.131 0.047 CHEMBL3706527 0.089 0.082 CHEMBL3706529 0.093 0.078 CHEMBL3706524 | CHEMBL3706523 | |
| 0.129 | 0.082 | 0.156 | Neurotrophic factor | 0.117 0.1 CHEMBL3706523 0.121 0.094 CHEMBL3706525 0.147 0.062 CHEMBL3706527 0.156 0.054 CHEMBL3706528 0.121 0.094 CHEMBL3706529 | CHEMBL3706528 | |
| 0.171 | 0.125 | 0.332 | Platelet antagonist | 0.153 0.141 CHEMBL3706523 0.314 0.048 CHEMBL3706525 0.332 0.043 CHEMBL3706526 0.196 0.104 CHEMBL3706528 0.194 0.105 CHEMBL3706524 | CHEMBL3706526 | |
| 0.051 | 0.007 | 0.076 | Plasmepsin I inhibitor | 0.027 0.025 CHEMBL3706522 0.076 0.004 CHEMBL3706523 0.047 0.009 CHEMBL3706525 0.042 0.011 CHEMBL3706526 0.046 0.009 CHEMBL3706528 0.047 0.009 CHEMBL3706529 0.05 0.008 CHEMBL3706524 | CHEMBL3706523 | |
| 0.07 | 0.032 | 0.132 | Caspase 9 inhibitor | 0.132 0.008 CHEMBL3706523 0.099 0.014 CHEMBL3706525 0.111 0.011 CHEMBL3706526 0.069 0.033 CHEMBL3706528 0.066 0.037 CHEMBL3706529 0.095 0.016 CHEMBL3706524 | CHEMBL3706523 | |
| 0.085 | 0.048 | 0.128 | Chymotrypsin inhibitor | 0.128 0.023 CHEMBL3706523 0.093 0.041 CHEMBL3706525 0.08 0.054 CHEMBL3706526 0.073 0.065 CHEMBL3706527 0.075 0.061 CHEMBL3706528 0.081 0.053 CHEMBL3706529 0.107 0.032 CHEMBL3706524 | CHEMBL3706523 | |
| 0.231 | 0.201 | 0.467 | Analgesic | 0.221 0.213 CHEMBL3706525 0.467 0.059 CHEMBL3706527 0.222 0.211 CHEMBL3706528 0.233 0.199 CHEMBL3706529 | CHEMBL3706527 | |
| 0.169 | 0.14 | 0.385 | Immunostimulant | 0.355 0.063 CHEMBL3706523 0.163 0.144 CHEMBL3706525 0.385 0.054 CHEMBL3706526 0.246 0.098 CHEMBL3706527 0.267 0.09 CHEMBL3706528 0.195 0.123 CHEMBL3706529 0.285 0.083 CHEMBL3706524 | CHEMBL3706526 | |
| 0.061 | 0.032 | 0.107 | Bombesin 3 receptor antagonist | 0.107 0.01 CHEMBL3706522 0.065 0.028 CHEMBL3706527 0.054 0.041 CHEMBL3706528 | CHEMBL3706522 | |
| 0.048 | 0.02 | 0.052 | Melanocortin 1 antagonist | 0.052 0.019 CHEMBL3706527 0.034 0.031 CHEMBL3706524 | CHEMBL3706527 | |
| 0.04 | 0.013 | 0.052 | Dipeptidyl peptidase I inhibitor | 0.032 0.019 CHEMBL3706523 0.032 0.019 CHEMBL3706525 0.052 0.008 CHEMBL3706527 0.034 0.017 CHEMBL3706528 0.034 0.017 CHEMBL3706529 0.033 0.018 CHEMBL3706524 | CHEMBL3706527 | |
| 0.077 | 0.051 | 0.123 | Analgesic, opioid | 0.069 0.063 CHEMBL3706525 0.123 0.021 CHEMBL3706527 0.072 0.059 CHEMBL3706528 0.074 0.056 CHEMBL3706529 | CHEMBL3706527 | |
| 0.046 | 0.02 | 0.056 | Renin inhibitor | 0.056 0.014 CHEMBL3706523 0.041 0.023 CHEMBL3706525 0.036 0.026 CHEMBL3706527 0.036 0.026 CHEMBL3706528 0.043 0.021 CHEMBL3706529 | CHEMBL3706523 | |
| 0.052 | 0.026 | 0.055 | Bombesin antagonist | 0.053 0.025 CHEMBL3706523 0.047 0.033 CHEMBL3706526 0.043 0.042 CHEMBL3706527 0.049 0.031 CHEMBL3706528 0.048 0.032 CHEMBL3706529 0.055 0.023 CHEMBL3706524 | CHEMBL3706524 | |
| 0.115 | 0.09 | 0.191 | Bone formation stimulant | 0.137 0.07 CHEMBL3706523 0.13 0.076 CHEMBL3706525 0.191 0.038 CHEMBL3706526 0.119 0.087 CHEMBL3706528 0.113 0.092 CHEMBL3706529 0.162 0.051 CHEMBL3706524 | CHEMBL3706526 | |
| 0.193 | 0.168 | 0.388 | Insulysin inhibitor | 0.196 0.163 CHEMBL3706522 0.344 0.036 CHEMBL3706523 0.388 0.024 CHEMBL3706526 0.202 0.154 CHEMBL3706527 0.35 0.034 CHEMBL3706524 | CHEMBL3706526 | |
| 0.06 | 0.035 | 0.13 | Cathepsin B inhibitor | 0.13 0.009 CHEMBL3706523 0.058 0.037 CHEMBL3706525 0.053 0.044 CHEMBL3706528 0.055 0.041 CHEMBL3706529 0.077 0.025 CHEMBL3706524 | CHEMBL3706523 | |
| 0.07 | 0.047 | 0.105 | Elastase 1 inhibitor | 0.105 0.017 CHEMBL3706523 0.085 0.03 CHEMBL3706525 0.081 0.035 CHEMBL3706526 0.066 0.053 CHEMBL3706529 0.083 0.033 CHEMBL3706524 | CHEMBL3706523 | |
| 0.047 | 0.025 | 0.171 | Dipeptidyl peptidase IV inhibitor | 0.171 0.003 CHEMBL3706527 0.046 0.027 CHEMBL3706529 | CHEMBL3706527 | |
| 0.048 | 0.026 | 0.052 | Baculoviral IAP repeat-containing protein inhibitor | 0.048 0.027 CHEMBL3706525 0.052 0.015 CHEMBL3706527 0.045 0.035 CHEMBL3706528 0.046 0.032 CHEMBL3706529 | CHEMBL3706527 | |
| 0.077 | 0.055 | 0.101 | Somatostatin 1 agonist | 0.101 0.034 CHEMBL3706523 0.074 0.058 CHEMBL3706526 0.084 0.047 CHEMBL3706527 0.069 0.067 CHEMBL3706528 0.07 0.064 CHEMBL3706529 0.097 0.036 CHEMBL3706524 | CHEMBL3706523 | |
| 0.08 | 0.058 | 0.125 | Opioid kappa receptor antagonist | 0.073 0.07 CHEMBL3706525 0.125 0.022 CHEMBL3706527 0.072 0.071 CHEMBL3706528 | CHEMBL3706527 | |
| 0.056 | 0.035 | 0.066 | Angiotensin-converting enzyme inhibitor | 0.061 0.029 CHEMBL3706525 0.066 0.023 CHEMBL3706526 0.06 0.03 CHEMBL3706527 0.052 0.043 CHEMBL3706528 0.053 0.041 CHEMBL3706529 0.051 0.045 CHEMBL3706524 | CHEMBL3706526 | |
| 0.052 | 0.031 | 0.069 | Bombesin 2 receptor antagonist | 0.062 0.023 CHEMBL3706523 0.069 0.02 CHEMBL3706526 0.05 0.033 CHEMBL3706527 0.047 0.039 CHEMBL3706529 0.057 0.026 CHEMBL3706524 | CHEMBL3706526 | |
| 0.062 | 0.044 | 0.065 | Protease activated receptor antagonist | 0.065 0.041 CHEMBL3706524 | CHEMBL3706524 | |
| 0.029 | 0.01 | 0.101 | Aminopeptidase P inhibitor | 0.026 0.013 CHEMBL3706523 0.025 0.014 CHEMBL3706525 0.022 0.017 CHEMBL3706526 0.101 0.002 CHEMBL3706527 0.025 0.014 CHEMBL3706528 0.026 0.013 CHEMBL3706529 0.023 0.017 CHEMBL3706524 | CHEMBL3706527 | |
| 0.082 | 0.063 | 0.121 | Factor XII inhibitor | 0.115 0.026 CHEMBL3706523 0.121 0.023 CHEMBL3706526 0.078 0.071 CHEMBL3706529 0.105 0.033 CHEMBL3706524 | CHEMBL3706526 | |
| 0.032 | 0.013 | 0.032 | Vasopressin 1A agonist | 0.029 0.018 CHEMBL3706523 0.027 0.025 CHEMBL3706525 0.028 0.02 CHEMBL3706527 0.03 0.016 CHEMBL3706528 0.031 0.015 CHEMBL3706529 0.028 0.02 CHEMBL3706524 | ||
| 0.037 | 0.019 | 0.044 | Growth factor receptor-bound protein 2 antagonist | 0.041 0.013 CHEMBL3706523 0.044 0.008 CHEMBL3706526 0.035 0.025 CHEMBL3706528 0.036 0.022 CHEMBL3706529 0.043 0.009 CHEMBL3706524 | CHEMBL3706526 | |
| 0.071 | 0.054 | 0.079 | Thrombin inhibitor | 0.076 0.046 CHEMBL3706523 0.079 0.043 CHEMBL3706527 | CHEMBL3706527 | |
| 0.053 | 0.037 | 0.073 | Opioid agonist | 0.073 0.022 CHEMBL3706527 0.048 0.042 CHEMBL3706528 | CHEMBL3706527 | |
| 0.047 | 0.033 | 0.047 | Melanocortin antagonist | 0.045 0.035 CHEMBL3706527 | ||
| 0.042 | 0.028 | 0.07 | Cholecystokinin antagonist | 0.044 0.028 CHEMBL3706522 0.07 0.014 CHEMBL3706525 0.051 0.024 CHEMBL3706526 0.056 0.022 CHEMBL3706524 | CHEMBL3706525 | |
| 0.032 | 0.019 | 0.06 | AMPA 2 receptor antagonist | 0.032 0.019 CHEMBL3706525 0.034 0.018 CHEMBL3706526 0.06 0.009 CHEMBL3706527 | CHEMBL3706527 | |
| 0.041 | 0.029 | 0.046 | Neurokinin 2 agonist | 0.042 0.027 CHEMBL3706523 0.042 0.028 CHEMBL3706525 0.04 0.03 CHEMBL3706529 0.046 0.023 CHEMBL3706524 | CHEMBL3706524 | |
| 0.041 | 0.03 | 0.041 | Melanocortin 4 antagonist | 0.039 0.033 CHEMBL3706527 | ||
| 0.039 | 0.029 | 0.061 | Cathepsin L2 inhibitor | 0.056 0.02 CHEMBL3706523 0.055 0.02 CHEMBL3706526 0.035 0.032 CHEMBL3706528 0.061 0.017 CHEMBL3706524 | CHEMBL3706524 | |
| 0.165 | 0.155 | 0.332 | Calpain inhibitor | 0.228 0.087 CHEMBL3706522 0.332 0.02 CHEMBL3706523 0.272 0.046 CHEMBL3706526 0.329 0.021 CHEMBL3706524 | CHEMBL3706523 | |
| 0.044 | 0.035 | 0.102 | Endothelin-converting enzyme inhibitor | 0.078 0.018 CHEMBL3706523 0.043 0.035 CHEMBL3706525 0.102 0.014 CHEMBL3706526 0.069 0.021 CHEMBL3706524 | CHEMBL3706526 | |
| 0.031 | 0.022 | 0.069 | Caspase 2 inhibitor | 0.06 0.009 CHEMBL3706523 0.055 0.01 CHEMBL3706525 0.069 0.007 CHEMBL3706526 0.028 0.025 CHEMBL3706528 0.029 0.024 CHEMBL3706529 0.058 0.009 CHEMBL3706524 | CHEMBL3706526 | |
| 0.022 | 0.014 | 0.034 | Human T-cell leukemia virus type I protease inhibitor | 0.034 0.006 CHEMBL3706523 0.019 0.017 CHEMBL3706529 0.021 0.015 CHEMBL3706524 | CHEMBL3706523 | |
| 0.042 | 0.034 | 0.085 | Neurotensin receptor antagonist | 0.085 0.017 CHEMBL3706526 0.045 0.032 CHEMBL3706524 | CHEMBL3706526 | |
| 0.043 | 0.036 | 0.06 | Opioid mu receptor agonist | 0.06 0.023 CHEMBL3706527 | CHEMBL3706527 | |
| 0.032 | 0.025 | 0.032 | Growth hormone releasing factor agonist | 0.032 0.024 CHEMBL3706527 0.029 0.027 CHEMBL3706529 | ||
| 0.022 | 0.016 | 0.123 | Follicle-stimulating hormone agonist | 0.123 0.004 CHEMBL3706522 0.024 0.013 CHEMBL3706527 0.031 0.01 CHEMBL3706529 | CHEMBL3706522 | |
| 0.035 | 0.03 | 0.054 | Cholecystokinin B agonist | 0.04 0.023 CHEMBL3706523 0.041 0.022 CHEMBL3706525 0.054 0.014 CHEMBL3706526 0.034 0.032 CHEMBL3706529 0.046 0.018 CHEMBL3706524 | CHEMBL3706526 | |
| 0.201 | 0.196 | 0.488 | Immunosuppressant | 0.234 0.162 CHEMBL3706525 0.316 0.105 CHEMBL3706527 0.279 0.128 CHEMBL3706528 0.342 0.091 CHEMBL3706529 0.488 0.036 CHEMBL3706524 | CHEMBL3706524 | |
| 0.04 | 0.035 | 0.047 | Cathepsin F inhibitor | 0.043 0.024 CHEMBL3706523 0.047 0.017 CHEMBL3706524 | CHEMBL3706524 | |
| 0.033 | 0.029 | 0.064 | Cholecystokinin A antagonist | 0.046 0.021 CHEMBL3706522 0.064 0.016 CHEMBL3706525 0.042 0.023 CHEMBL3706526 0.039 0.025 CHEMBL3706524 | CHEMBL3706525 | |
| 0.034 | 0.03 | 0.037 | Bombesin 1 receptor antagonist | 0.034 0.029 CHEMBL3706523 0.037 0.025 CHEMBL3706524 | CHEMBL3706524 | |
| 0.026 | 0.023 | 0.04 | Bradykinin B2 receptor agonist | 0.04 0.012 CHEMBL3706526 0.025 0.024 CHEMBL3706528 0.027 0.022 CHEMBL3706529 0.025 0.024 CHEMBL3706524 | CHEMBL3706526 | |
| 0.02 | 0.019 | 0.02 | Vasopressin 1 agonist | |||
| 0.033 | 0.032 | 0.033 | Antidiuretic hormone antagonist | |||
| 0.037 | 0.036 | 0.041 | Growth hormone release inhibitor | 0.041 0.03 CHEMBL3706523 0.037 0.036 CHEMBL3706527 0.04 0.032 CHEMBL3706524 | CHEMBL3706523 | |
| 0.02 | 0.019 | 0.02 | Melanocortin 4 agonist | |||
| 0.028 | 0.029 | 0.057 | Calcitonin receptor agonist | 0.047 0.018 CHEMBL3706523 0.057 0.015 CHEMBL3706526 0.03 0.027 CHEMBL3706529 0.035 0.023 CHEMBL3706524 | CHEMBL3706526 | |
| 0.063 | 0.064 | 0.193 | Aminopeptidase I inhibitor | 0.064 0.062 CHEMBL3706522 0.123 0.019 CHEMBL3706523 0.088 0.035 CHEMBL3706525 0.193 0.007 CHEMBL3706526 0.154 0.012 CHEMBL3706527 0.112 0.022 CHEMBL3706524 | CHEMBL3706526 | |
| 0.025 | 0.027 | 0.04 | Cholecystokinin B antagonist | 0.04 0.014 CHEMBL3706525 | CHEMBL3706525 | |
| 0.04 | 0.044 | 0.16 | Chemokine receptor agonist | 0.16 0.004 CHEMBL3706522 0.062 0.026 CHEMBL3706527 | CHEMBL3706522 | |
| 0.03 | 0.034 | 0.063 | Calpain 1 inhibitor | 0.063 0.004 CHEMBL3706523 0.039 0.012 CHEMBL3706524 | CHEMBL3706523 | |
| 0.03 | 0.035 | 0.034 | Opioid delta receptor agonist | 0.034 0.027 CHEMBL3706527 | CHEMBL3706527 | |
| 0.017 | 0.022 | 0.021 | Growth hormone releasing factor antagonist | 0.02 0.019 CHEMBL3706523 0.021 0.019 CHEMBL3706524 | CHEMBL3706524 | |
| 0.024 | 0.03 | 0.029 | Baculoviral IAP repeat-containing protein 4 inhibitor | 0.029 0.015 CHEMBL3706526 0.027 0.019 CHEMBL3706527 0.026 0.023 CHEMBL3706524 | CHEMBL3706526 | |
| 0.049 | 0.056 | 0.064 | Kallikrein 1 inhibitor | 0.064 0.029 CHEMBL3706523 0.059 0.035 CHEMBL3706524 | CHEMBL3706523 | |
| 0.021 | 0.029 | 0.033 | Bradykinin B2 receptor antagonist | 0.033 0.021 CHEMBL3706526 | CHEMBL3706526 | |
| 0.084 | 0.092 | 0.148 | Nav1.1 sodium channel blocker | 0.148 0.034 CHEMBL3706527 | CHEMBL3706527 | |
| 0.072 | 0.081 | 0.156 | Falcipain 2 inhibitor | 0.142 0.032 CHEMBL3706523 0.091 0.059 CHEMBL3706526 0.156 0.026 CHEMBL3706524 | CHEMBL3706524 | |
| 0.011 | 0.024 | 0.016 | Dipeptidyl peptidase IX inhibitor | 0.016 0.011 CHEMBL3706527 | CHEMBL3706527 | |
| 0.054 | 0.068 | 0.062 | Trypsin inhibitor | 0.062 0.044 CHEMBL3706523 0.062 0.044 CHEMBL3706526 | CHEMBL3706526 | |
| 0.011 | 0.025 | 0.02 | KiSS-1 receptor antagonist | 0.02 0.009 CHEMBL3706523 0.02 0.009 CHEMBL3706524 | CHEMBL3706524 | |
| 0.02 | 0.035 | 0.095 | CXC chemokine receptor agonist | 0.095 0.003 CHEMBL3706522 0.037 0.02 CHEMBL3706527 | CHEMBL3706522 | |
| 0.034 | 0.049 | 0.052 | Plasmin inhibitor | 0.052 0.031 CHEMBL3706523 | CHEMBL3706523 | |
| 0.022 | 0.038 | 0.072 | Thrombin receptor antagonist | 0.049 0.009 CHEMBL3706523 0.044 0.01 CHEMBL3706526 0.072 0.005 CHEMBL3706524 | CHEMBL3706524 | |
| 0.131 | 0.148 | 0.18 | P-glycoprotein inhibitor | 0.147 0.122 CHEMBL3706525 0.18 0.08 CHEMBL3706527 0.153 0.112 CHEMBL3706528 | CHEMBL3706527 | |
| 0.114 | 0.132 | 0.411 | Thiol protease inhibitor | 0.146 0.072 CHEMBL3706522 0.411 0.013 CHEMBL3706523 0.305 0.019 CHEMBL3706526 0.326 0.017 CHEMBL3706524 | CHEMBL3706523 | |
| 0.026 | 0.043 | 0.048 | GHS receptor antagonist | 0.048 0.008 CHEMBL3706522 | CHEMBL3706522 | |
| 0.012 | 0.029 | 0.018 | Neurokinin 1 agonist | 0.018 0.016 CHEMBL3706524 | CHEMBL3706524 | |
| 0.027 | 0.045 | 0.037 | Nicotinic receptor beta4 subunit antagonist | 0.035 0.029 CHEMBL3706522 0.037 0.026 CHEMBL3706527 | CHEMBL3706527 | |
| 0.145 | 0.164 | 0.219 | Vasodilator | 0.177 0.124 CHEMBL3706525 0.219 0.09 CHEMBL3706527 0.17 0.131 CHEMBL3706528 | CHEMBL3706527 | |
| 0.008 | 0.029 | 0.015 | Protease activated receptor agonist | 0.015 0.014 CHEMBL3706524 | CHEMBL3706524 | |
| 0.019 | 0.041 | 0.025 | Cathepsin K inhibitor | 0.025 0.021 CHEMBL3706523 | CHEMBL3706523 | |
| 0.009 | 0.032 | 0.015 | Calcium-sensing receptor antagonist | 0.015 0.011 CHEMBL3706527 | CHEMBL3706527 | |
| 0.051 | 0.075 | 0.155 | Protease 3C (Human rhinovirus) inhibitor | 0.155 0.006 CHEMBL3706523 0.094 0.018 CHEMBL3706526 0.12 0.01 CHEMBL3706524 | CHEMBL3706523 | |
| 0.024 | 0.049 | 0.033 | Bradykinin antagonist | 0.033 0.031 CHEMBL3706522 | CHEMBL3706522 | |
| 0.029 | 0.055 | 0.067 | Integrin alpha5beta1 antagonist | 0.038 0.033 CHEMBL3706523 0.067 0.009 CHEMBL3706526 0.042 0.026 CHEMBL3706524 | CHEMBL3706526 | |
| 0.026 | 0.055 | 0.054 | Erythropoietin receptor agonist | 0.036 0.033 CHEMBL3706523 0.054 0.019 CHEMBL3706526 0.043 0.026 CHEMBL3706524 | CHEMBL3706526 | |
| 0.04 | 0.069 | 0.063 | Carbonic anhydrase II stimulant | 0.063 0.02 CHEMBL3706526 0.048 0.045 CHEMBL3706524 | CHEMBL3706526 | |
| 0.007 | 0.039 | 0.012 | 3 Beta-hydroxy-delta 5-steroid dehydrogenase inhibitor | 0.012 0.01 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.042 | 0.041 | Integrin beta7 antagonist | 0.041 0.007 CHEMBL3706526 | CHEMBL3706526 | |
| 0.038 | 0.071 | 0.174 | Cannabinoid CB1 receptor agonist | 0.174 0.008 CHEMBL3706522 0.067 0.037 CHEMBL3706526 0.069 0.036 CHEMBL3706529 | CHEMBL3706522 | |
| 0.014 | 0.049 | 0.024 | Follicle-stimulating hormone antagonist | 0.024 0.006 CHEMBL3706522 0.02 0.013 CHEMBL3706526 | CHEMBL3706522 | |
| 0.006 | 0.042 | 0.017 | 3C-Like protease (MERS coronavirus) inhibitor | 0.017 0.004 CHEMBL3706523 | CHEMBL3706523 | |
| 0.03 | 0.066 | 0.061 | Kallikrein inhibitor | 0.061 0.023 CHEMBL3706523 0.055 0.026 CHEMBL3706524 | CHEMBL3706523 | |
| 0.013 | 0.049 | 0.032 | Elastase 2A inhibitor | 0.02 0.018 CHEMBL3706523 0.032 0.009 CHEMBL3706524 | CHEMBL3706524 | |
| 0.013 | 0.049 | 0.032 | Elastase 2 inhibitor | 0.02 0.018 CHEMBL3706523 0.032 0.009 CHEMBL3706524 | CHEMBL3706524 | |
| 0.094 | 0.132 | 0.268 | Histone deacetylase SIRT1 inhibitor | 0.166 0.049 CHEMBL3706523 0.19 0.034 CHEMBL3706526 0.268 0.013 CHEMBL3706524 | CHEMBL3706524 | |
| 0.068 | 0.106 | 0.086 | Transcription factor NF kappa B stimulant | 0.081 0.067 CHEMBL3706523 0.086 0.058 CHEMBL3706526 0.084 0.061 CHEMBL3706524 | CHEMBL3706526 | |
| 0.01 | 0.049 | 0.061 | Integrin alpha4 antagonist | 0.022 0.019 CHEMBL3706525 0.061 0.01 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.048 | 0.019 | Cholecystokinin agonist | 0.019 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.084 | 0.125 | 0.151 | Calcium channel N-type blocker | 0.151 0.037 CHEMBL3706522 0.102 0.092 CHEMBL3706525 0.119 0.065 CHEMBL3706527 | CHEMBL3706522 | |
| 0.113 | 0.154 | 0.23 | Platelet adhesion inhibitor | 0.16 0.096 CHEMBL3706525 0.23 0.057 CHEMBL3706526 0.144 0.113 CHEMBL3706528 | CHEMBL3706526 | |
| 0.031 | 0.074 | 0.053 | Plasminogen activator inhibitor | 0.053 0.045 CHEMBL3706523 | CHEMBL3706523 | |
| 0.026 | 0.071 | 0.043 | Glutamate (mGluR8) antagonist | 0.043 0.013 CHEMBL3706526 0.038 0.02 CHEMBL3706527 | CHEMBL3706526 | |
| 0.007 | 0.052 | 0.038 | Integrin alpha4beta7 antagonist | 0.038 0.007 CHEMBL3706526 | CHEMBL3706526 | |
| 0.018 | 0.064 | 0.11 | Complement C3a chemotactic receptor antagonist | 0.042 0.031 CHEMBL3706523 0.11 0.006 CHEMBL3706526 0.047 0.028 CHEMBL3706524 | CHEMBL3706526 | |
| 0.013 | 0.06 | 0.078 | AMPA 3 receptor antagonist | 0.078 0.004 CHEMBL3706526 | CHEMBL3706526 | |
| 0.014 | 0.064 | 0.021 | Baculoviral IAP repeat-containing protein 3 inhibitor | 0.021 0.014 CHEMBL3706527 | CHEMBL3706527 | |
| 0.015 | 0.065 | 0.031 | Trypsin I inhibitor | 0.031 0.025 CHEMBL3706526 | CHEMBL3706526 | |
| 0.029 | 0.08 | 0.041 | Glucagon-like peptide 1 receptor antagonist | 0.041 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.101 | 0.152 | 0.156 | Insulin secretagoues | 0.156 0.068 CHEMBL3706525 0.126 0.102 CHEMBL3706526 0.144 0.08 CHEMBL3706527 | CHEMBL3706525 | |
| 0.047 | 0.099 | 0.166 | Cathepsin G inhibitor | 0.166 0.019 CHEMBL3706523 0.064 0.062 CHEMBL3706525 0.122 0.027 CHEMBL3706526 0.088 0.038 CHEMBL3706524 | CHEMBL3706523 | |
| 0.045 | 0.097 | 0.126 | Sirtuin 1 inhibitor | 0.068 0.047 CHEMBL3706523 0.087 0.03 CHEMBL3706526 0.126 0.012 CHEMBL3706524 | CHEMBL3706524 | |
| 0.058 | 0.11 | 0.205 | Cell adhesion molecule inhibitor | 0.098 0.036 CHEMBL3706525 0.205 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.019 | 0.074 | 0.043 | Carbonic anhydrase I stimulant | 0.043 0.021 CHEMBL3706526 | CHEMBL3706526 | |
| 0.034 | 0.089 | 0.09 | Selectin antagonist | 0.071 0.042 CHEMBL3706523 0.09 0.032 CHEMBL3706526 0.078 0.038 CHEMBL3706524 | CHEMBL3706526 | |
| 0.032 | 0.087 | 0.066 | Aminopeptidase microsomal inhibitor | 0.056 0.042 CHEMBL3706523 0.061 0.039 CHEMBL3706526 0.066 0.034 CHEMBL3706527 0.061 0.039 CHEMBL3706524 | CHEMBL3706527 | |
| 0.016 | 0.073 | 0.163 | Integrin antagonist | 0.035 0.034 CHEMBL3706525 0.163 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.112 | 0.17 | 0.198 | Antipruritic | 0.198 0.05 CHEMBL3706527 | CHEMBL3706527 | |
| 0.029 | 0.091 | 0.068 | Cathepsin L inhibitor | 0.068 0.031 CHEMBL3706523 0.055 0.045 CHEMBL3706524 | CHEMBL3706523 | |
| 0.022 | 0.084 | 0.048 | Aminopeptidase N inhibitor | 0.043 0.038 CHEMBL3706526 0.048 0.034 CHEMBL3706527 0.043 0.038 CHEMBL3706524 | CHEMBL3706527 | |
| 0.006 | 0.069 | 0.133 | AMPA 1 receptor antagonist | 0.133 0.004 CHEMBL3706526 0.031 0.019 CHEMBL3706524 | CHEMBL3706526 | |
| 0.007 | 0.07 | 0.016 | Cholecystokinin A agonist | 0.016 0.012 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.072 | 0.06 | VLA-4 antagonist | 0.06 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.073 | 0.143 | 0.133 | Calcium channel (voltage-sensitive) blocker | 0.111 0.069 CHEMBL3706522 0.098 0.088 CHEMBL3706525 0.133 0.044 CHEMBL3706527 | CHEMBL3706527 | |
| 0.029 | 0.099 | 0.046 | VCAM-1 antagonist | 0.046 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.073 | 0.009 | Phosphoribosylglycinamide formyltransferase inhibitor | 0.009 0.004 CHEMBL3706526 | CHEMBL3706526 | |
| 0.029 | 0.099 | 0.045 | VCAM antagonist | 0.045 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.011 | 0.082 | 0.038 | Plasma kallikrein inhibitor | 0.038 0.02 CHEMBL3706524 | CHEMBL3706524 | |
| 0.019 | 0.092 | 0.053 | Macrophage elastase inhibitor | 0.053 0.022 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.09 | 0.038 | Cathepsin L1 inhibitor | 0.038 0.028 CHEMBL3706523 | CHEMBL3706523 | |
| 0.019 | 0.096 | 0.104 | NMDA 2A receptor antagonist | 0.104 0.012 CHEMBL3706526 | CHEMBL3706526 | |
| 0.079 | 0.161 | 0.274 | Cathepsin H inhibitor | 0.106 0.097 CHEMBL3706522 0.274 0.011 CHEMBL3706523 0.226 0.017 CHEMBL3706526 0.111 0.088 CHEMBL3706527 0.188 0.026 CHEMBL3706524 | CHEMBL3706523 | |
| 0.01 | 0.094 | 0.071 | GP IIb/IIIa receptor antagonist | 0.071 0.024 CHEMBL3706526 | CHEMBL3706526 | |
| 0.016 | 0.1 | 0.067 | Glutamate (mGluR group II) agonist | 0.067 0.011 CHEMBL3706522 0.048 0.016 CHEMBL3706526 | CHEMBL3706522 | |
| 0.117 | 0.203 | 0.385 | Spasmolytic | 0.183 0.134 CHEMBL3706522 0.385 0.043 CHEMBL3706527 | CHEMBL3706527 | |
| 0.165 | 0.253 | 0.245 | Antiobesity | 0.245 0.161 CHEMBL3706522 0.207 0.201 CHEMBL3706525 0.229 0.178 CHEMBL3706527 | CHEMBL3706522 | |
| 0.027 | 0.117 | 0.048 | Farnesyltransferase inhibitor | 0.048 0.03 CHEMBL3706526 | CHEMBL3706526 | |
| 0.01 | 0.109 | 0.019 | Tryptophan hydroxylase 1 inhibitor | 0.019 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.062 | 0.162 | 0.134 | Nav1.3 sodium channel blocker | 0.112 0.083 CHEMBL3706522 0.134 0.06 CHEMBL3706527 | CHEMBL3706527 | |
| 0.063 | 0.164 | 0.13 | Glutamate receptor antagonist | 0.13 0.066 CHEMBL3706522 0.13 0.065 CHEMBL3706526 | CHEMBL3706526 | |
| 0.016 | 0.118 | 0.125 | Ribonucleoside-diphosphate reductase inhibitor | 0.103 0.019 CHEMBL3706523 0.125 0.015 CHEMBL3706526 0.068 0.03 CHEMBL3706524 | CHEMBL3706526 | |
| 0.011 | 0.115 | 0.062 | Glutamate (mGluR2) agonist | 0.062 0.01 CHEMBL3706522 0.035 0.02 CHEMBL3706526 | CHEMBL3706522 | |
| 0.024 | 0.134 | 0.242 | Glutamate (mGluR) agonist | 0.242 0.007 CHEMBL3706522 0.119 0.019 CHEMBL3706526 | CHEMBL3706522 | |
| 0.014 | 0.125 | 0.12 | Ribonucleotide reductase inhibitor | 0.101 0.02 CHEMBL3706523 0.12 0.017 CHEMBL3706526 0.069 0.032 CHEMBL3706524 | CHEMBL3706526 | |
| 0.013 | 0.125 | 0.043 | Urokinase inhibitor | 0.043 0.037 CHEMBL3706526 | CHEMBL3706526 | |
| 0.021 | 0.134 | 0.049 | Dopamine transporter inhibitor | 0.049 0.033 CHEMBL3706527 | CHEMBL3706527 | |
| 0.008 | 0.122 | 0.034 | Integrin alphaVbeta1 antagonist | 0.034 0.005 CHEMBL3706526 | CHEMBL3706526 | |
| 0.042 | 0.16 | 0.119 | Antiadrenergic | 0.119 0.046 CHEMBL3706527 | CHEMBL3706527 | |
| 0.04 | 0.159 | 0.115 | Adrenaline antagonist | 0.115 0.046 CHEMBL3706527 | CHEMBL3706527 | |
| 0.183 | 0.302 | 0.376 | Cyclophilin D inhibitor | 0.261 0.201 CHEMBL3706525 0.254 0.208 CHEMBL3706526 0.376 0.105 CHEMBL3706527 0.249 0.214 CHEMBL3706528 0.241 0.224 CHEMBL3706529 | CHEMBL3706527 | |
| 0.022 | 0.143 | 0.192 | Cannabinoid receptor agonist | 0.192 0.008 CHEMBL3706522 | CHEMBL3706522 | |
| 0.028 | 0.148 | 0.066 | Matrix metalloproteinase inhibitor | 0.066 0.047 CHEMBL3706526 | CHEMBL3706526 | |
| 0.068 | 0.191 | 0.245 | Folate antagonist | 0.105 0.056 CHEMBL3706523 0.091 0.084 CHEMBL3706525 0.245 0.005 CHEMBL3706526 0.116 0.043 CHEMBL3706524 | CHEMBL3706526 | |
| 0.076 | 0.199 | 0.212 | Amyloid beta aggregation inhibitor | 0.212 0.072 CHEMBL3706526 0.172 0.094 CHEMBL3706524 | CHEMBL3706526 | |
| 0.121 | 0.244 | 0.701 | Superoxide dismutase inhibitor | 0.306 0.048 CHEMBL3706522 0.507 0.012 CHEMBL3706523 0.701 0.004 CHEMBL3706526 0.361 0.034 CHEMBL3706524 | CHEMBL3706526 | |
| 0.007 | 0.138 | 0.035 | Purinergic P2Y12 antagonist | 0.027 0.013 CHEMBL3706522 0.035 0.01 CHEMBL3706526 | CHEMBL3706526 | |
| 0.136 | 0.267 | 0.4 | Vasodilator, peripheral | 0.207 0.168 CHEMBL3706522 0.286 0.104 CHEMBL3706525 0.4 0.055 CHEMBL3706527 | CHEMBL3706527 | |
| 0.003 | 0.157 | 0.018 | Aminopeptidase A inhibitor | 0.018 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.017 | 0.173 | 0.065 | AMPA 4 receptor antagonist | 0.065 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.014 | 0.172 | 0.043 | Factor XIIIa inhibitor | 0.043 0.021 CHEMBL3706526 | CHEMBL3706526 | |
| 0.024 | 0.184 | 0.145 | Carbonic anhydrase stimulant | 0.145 0.011 CHEMBL3706526 0.066 0.034 CHEMBL3706524 | CHEMBL3706526 | |
| 0.153 | 0.314 | 0.27 | MAP kinase kinase 3 inhibitor | 0.27 0.017 CHEMBL3706522 0.185 0.173 CHEMBL3706523 0.229 0.058 CHEMBL3706526 0.197 0.131 CHEMBL3706524 | CHEMBL3706522 | |
| 0.017 | 0.192 | 0.048 | Prolyl endopeptidase inhibitor | 0.048 0.039 CHEMBL3706527 | CHEMBL3706527 | |
| 0.025 | 0.202 | 0.05 | Factor IXa inhibitor | 0.05 0.037 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.186 | 0.03 | Integrin alphaVbeta3 antagonist | 0.03 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.192 | 0.029 | Vitronectin receptor antagonist | 0.029 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.055 | 0.257 | 0.141 | Calcium channel blocker | 0.109 0.101 CHEMBL3706522 0.141 0.067 CHEMBL3706527 | CHEMBL3706527 | |
| 0.044 | 0.246 | 0.153 | Nav1.6 sodium channel blocker | 0.153 0.051 CHEMBL3706522 0.115 0.104 CHEMBL3706527 | CHEMBL3706522 | |
| 0.017 | 0.22 | 0.059 | Transforming growth factor beta 2 antagonist | 0.059 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.113 | 0.318 | 0.237 | Neuropeptide Y2 antagonist | 0.23 0.076 CHEMBL3706523 0.237 0.07 CHEMBL3706526 0.225 0.082 CHEMBL3706524 | CHEMBL3706526 | |
| 0.046 | 0.257 | 0.151 | Adenylate cyclase inhibitor | 0.151 0.044 CHEMBL3706526 | CHEMBL3706526 | |
| 0.022 | 0.237 | 0.046 | Integrin alpha1beta1 antagonist | 0.046 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.011 | 0.227 | 0.077 | Toll-Like receptor 2 agonist | 0.077 0.017 CHEMBL3706526 | CHEMBL3706526 | |
| 0.012 | 0.232 | 0.045 | Dipeptidyl peptidase II inhibitor | 0.045 0.011 CHEMBL3706527 | CHEMBL3706527 | |
| 0.004 | 0.227 | 0.014 | Integrin alphaLbeta2 antagonist | 0.014 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.041 | 0.268 | 0.184 | Histone deacetylase class III inhibitor | 0.096 0.094 CHEMBL3706523 0.125 0.065 CHEMBL3706526 0.184 0.025 CHEMBL3706524 | CHEMBL3706524 | |
| 0.038 | 0.267 | 0.143 | Chelator | 0.143 0.038 CHEMBL3706526 | CHEMBL3706526 | |
| 0.037 | 0.267 | 0.096 | Aminoacyl-tRNA synthetase inhibitor | 0.096 0.05 CHEMBL3706526 | CHEMBL3706526 | |
| 0.021 | 0.265 | 0.254 | Anesthetic local | 0.254 0.019 CHEMBL3706527 | CHEMBL3706527 | |
| 0.094 | 0.343 | 0.291 | Gastrin inhibitor | 0.214 0.128 CHEMBL3706522 0.291 0.039 CHEMBL3706526 0.244 0.086 CHEMBL3706524 | CHEMBL3706526 | |
| 0.006 | 0.257 | 0.047 | Prostacyclin antagonist | 0.047 0.014 CHEMBL3706526 | CHEMBL3706526 | |
| 0.054 | 0.305 | 0.148 | CDK3/cyclin E inhibitor | 0.148 0.028 CHEMBL3706522 | CHEMBL3706522 | |
| 0.021 | 0.273 | 0.132 | Phospholipase D inhibitor | 0.132 0.004 CHEMBL3706522 0.124 0.005 CHEMBL3706526 | CHEMBL3706522 | |
| 0.039 | 0.292 | 0.175 | Acetylcholine antagonist | 0.175 0.038 CHEMBL3706527 | CHEMBL3706527 | |
| 0.147 | 0.402 | 0.297 | Calcium channel L-type activator | 0.297 0.16 CHEMBL3706522 0.275 0.18 CHEMBL3706526 | CHEMBL3706522 | |
| 0.01 | 0.265 | 0.082 | Neutrophil collagenase inhibitor | 0.067 0.042 CHEMBL3706523 0.082 0.031 CHEMBL3706526 0.062 0.048 CHEMBL3706524 | CHEMBL3706526 | |
| 0.039 | 0.298 | 0.178 | Cholinergic antagonist | 0.178 0.039 CHEMBL3706527 | CHEMBL3706527 | |
| 0.014 | 0.275 | 0.052 | Matrix metalloproteinase (membrane-type) inhibitor | 0.052 0.042 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.264 | 0.033 | Kainate receptor 1 antagonist | 0.033 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.019 | 0.282 | 0.076 | NMDA receptor antagonist | 0.076 0.071 CHEMBL3706527 | CHEMBL3706527 | |
| 0.026 | 0.291 | 0.099 | Ca(v)3.2 blocker | 0.099 0.009 CHEMBL3706522 | CHEMBL3706522 | |
| 0.081 | 0.347 | 0.199 | Hypoglycemic | 0.199 0.113 CHEMBL3706523 | CHEMBL3706523 | |
| 0.018 | 0.284 | 0.08 | Sphingosine kinase inhibitor | 0.08 0.016 CHEMBL3706527 | CHEMBL3706527 | |
| 0.004 | 0.274 | 0.041 | Leukotriene A4 hydrolase inhibitor | 0.041 0.024 CHEMBL3706527 | CHEMBL3706527 | |
| 0.012 | 0.284 | 0.048 | Sphingosine kinase 1 inhibitor | 0.048 0.018 CHEMBL3706527 | CHEMBL3706527 | |
| 0.022 | 0.295 | 0.136 | Glutamate (mGluR) antagonist | 0.136 0.021 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.282 | 0.026 | Caspase 8 inhibitor | 0.019 0.015 CHEMBL3706523 0.026 0.007 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.282 | 0.084 | Glutamate (mGluR1) antagonist | 0.084 0.021 CHEMBL3706522 0.072 0.029 CHEMBL3706526 | CHEMBL3706522 | |
| 0.046 | 0.324 | 0.111 | Ca(v)3.1 blocker | 0.111 0.015 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.285 | 0.076 | NMDA 2 receptor antagonist | 0.076 0.046 CHEMBL3706526 | CHEMBL3706526 | |
| 0.024 | 0.311 | 0.122 | CD45 antagonist | 0.122 0.007 CHEMBL3706526 0.048 0.041 CHEMBL3706524 | CHEMBL3706526 | |
| 0.031 | 0.327 | 0.069 | Immunoglobulin Fc receptor antagonist | 0.056 0.033 CHEMBL3706522 0.069 0.012 CHEMBL3706523 0.057 0.032 CHEMBL3706526 0.067 0.014 CHEMBL3706524 | CHEMBL3706523 | |
| 0.029 | 0.326 | 0.067 | Histone deacetylase SIRT3 inhibitor | 0.063 0.041 CHEMBL3706526 0.067 0.032 CHEMBL3706524 | CHEMBL3706524 | |
| 0.014 | 0.312 | 0.31 | Catalase inhibitor | 0.065 0.059 CHEMBL3706522 0.282 0.007 CHEMBL3706523 0.31 0.005 CHEMBL3706526 0.183 0.018 CHEMBL3706524 | CHEMBL3706526 | |
| 0.026 | 0.333 | 0.187 | Aminopeptidase B inhibitor | 0.158 0.034 CHEMBL3706523 0.187 0.024 CHEMBL3706526 0.124 0.05 CHEMBL3706527 0.1 0.065 CHEMBL3706524 | CHEMBL3706526 | |
| 0.018 | 0.325 | 0.051 | Glutamate (mGluR group III) antagonist | 0.051 0.019 CHEMBL3706526 0.048 0.024 CHEMBL3706527 | CHEMBL3706526 | |
| 0.002 | 0.312 | 0.041 | Arginase inhibitor | 0.041 0.021 CHEMBL3706527 | CHEMBL3706527 | |
| 0.094 | 0.405 | 0.215 | Toll-Like receptor agonist | 0.215 0.184 CHEMBL3706527 | CHEMBL3706527 | |
| 0.084 | 0.408 | 0.588 | 5 Hydroxytryptamine release stimulant | 0.237 0.096 CHEMBL3706522 0.588 0.016 CHEMBL3706527 | CHEMBL3706527 | |
| 0.022 | 0.35 | 0.125 | Histone deacetylase stimulant | 0.125 0.015 CHEMBL3706522 0.094 0.032 CHEMBL3706526 0.064 0.063 CHEMBL3706524 | CHEMBL3706522 | |
| 0.022 | 0.35 | 0.125 | Histone deacetylase SIRT1 stimulant | 0.125 0.015 CHEMBL3706522 0.094 0.032 CHEMBL3706526 0.064 0.063 CHEMBL3706524 | CHEMBL3706522 | |
| 0.016 | 0.346 | 0.068 | Metalloproteinase-9 inhibitor | 0.068 0.06 CHEMBL3706526 | CHEMBL3706526 | |
| 0.017 | 0.349 | 0.078 | Metalloproteinase-2 inhibitor | 0.078 0.055 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.339 | 0.032 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.032 0.018 CHEMBL3706522 | CHEMBL3706522 | |
| 0.016 | 0.354 | 0.099 | Nav1.8 sodium channel blocker | 0.099 0.029 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.352 | 0.048 | Metalloproteinase-3 inhibitor | 0.048 0.035 CHEMBL3706526 | CHEMBL3706526 | |
| 0.086 | 0.435 | 0.296 | Vasodilator, coronary | 0.227 0.157 CHEMBL3706522 0.296 0.091 CHEMBL3706527 | CHEMBL3706527 | |
| 0.085 | 0.435 | 0.202 | Toll-Like receptor 7 agonist | 0.202 0.198 CHEMBL3706527 | CHEMBL3706527 | |
| 0.009 | 0.361 | 0.03 | Carboxypeptidase B inhibitor | 0.03 0.029 CHEMBL3706526 | CHEMBL3706526 | |
| 0.027 | 0.397 | 0.108 | Microtubule formation inhibitor | 0.108 0.076 CHEMBL3706522 | CHEMBL3706522 | |
| 0.082 | 0.453 | 0.259 | Sodium/bile acid cotransporter inhibitor | 0.259 0.119 CHEMBL3706528 | CHEMBL3706528 | |
| 0.017 | 0.394 | 0.08 | Glutamate (mGluR group I) antagonist | 0.08 0.038 CHEMBL3706522 | CHEMBL3706522 | |
| 0.051 | 0.428 | 0.15 | Adenylate cyclase stimulant | 0.14 0.081 CHEMBL3706522 0.15 0.063 CHEMBL3706527 | CHEMBL3706527 | |
| 0.004 | 0.382 | 0.039 | Glutamate (mGluR group II) antagonist | 0.035 0.031 CHEMBL3706522 0.039 0.025 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.387 | 0.13 | Phosphorylase inhibitor | 0.114 0.011 CHEMBL3706523 0.13 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.045 | 0.434 | 0.123 | Transcription factor STAT6 inhibitor | 0.122 0.056 CHEMBL3706526 0.123 0.054 CHEMBL3706524 | CHEMBL3706524 | |
| 0.004 | 0.394 | 0.059 | Kainate receptor antagonist | 0.059 0.016 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.416 | 0.064 | Epithelial sodium channel blocker | 0.063 0.024 CHEMBL3706522 0.064 0.024 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.41 | 0.024 | Protease (Human cytomegalovirus) inhibitor | 0.024 0.013 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.423 | 0.044 | Purinergic P2Y15 antagonist | 0.044 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.426 | 0.05 | NMDA receptor subunit 3B antagonist | 0.05 0.025 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.427 | 0.036 | Protocollagen prolyl hydroxylase inhibitor | 0.036 0.009 CHEMBL3706522 0.026 0.021 CHEMBL3706526 | CHEMBL3706522 | |
| 0.018 | 0.443 | 0.091 | Transforming growth factor antagonist | 0.091 0.026 CHEMBL3706522 | CHEMBL3706522 | |
| 0.064 | 0.49 | 0.163 | Growth factor agonist | 0.163 0.115 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.431 | 0.088 | AMPA receptor antagonist | 0.088 0.015 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.432 | 0.038 | NMDA receptor subunit 3A antagonist | 0.038 0.027 CHEMBL3706526 | CHEMBL3706526 | |
| 0.03 | 0.46 | 0.105 | Interleukin 1b antagonist | 0.105 0.075 CHEMBL3706522 | CHEMBL3706522 | |
| 0.02 | 0.451 | 0.142 | Acetylcholine muscarinic antagonist | 0.142 0.049 CHEMBL3706527 | CHEMBL3706527 | |
| 0.008 | 0.447 | 0.064 | Dopamine uptake inhibitor | 0.064 0.035 CHEMBL3706527 | CHEMBL3706527 | |
| 0.046 | 0.487 | 0.21 | NOS3 expression enhancer | 0.21 0.037 CHEMBL3706522 | CHEMBL3706522 | |
| 0.028 | 0.471 | 0.172 | Potassium channel blocker | 0.172 0.113 CHEMBL3706522 | CHEMBL3706522 | |
| 0.029 | 0.472 | 0.178 | Insulin sensitizer | 0.178 0.097 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.451 | 0.051 | Glycine transporter 2 inhibitor | 0.051 0.03 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.462 | 0.065 | HIV-1 integrase inhibitor | 0.063 0.061 CHEMBL3706522 0.065 0.056 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.463 | 0.119 | Alcohol dehydrogenase inhibitor | 0.099 0.054 CHEMBL3706522 0.119 0.035 CHEMBL3706526 | CHEMBL3706526 | |
| 0.019 | 0.471 | 0.168 | Interleukin 1 beta converting enzyme inhibitor | 0.141 0.022 CHEMBL3706523 0.168 0.012 CHEMBL3706526 0.125 0.031 CHEMBL3706524 | CHEMBL3706526 | |
| 0.005 | 0.458 | 0.074 | NMDA 2C receptor antagonist | 0.074 0.03 CHEMBL3706526 | CHEMBL3706526 | |
| 0.014 | 0.468 | 0.044 | Glutamate (mGluR4) antagonist | 0.044 0.029 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.464 | 0.101 | Nicotinic alpha4beta2 receptor antagonist | 0.101 0.03 CHEMBL3706522 | CHEMBL3706522 | |
| 0.041 | 0.497 | 0.077 | Transforming growth factor beta 3 antagonist | 0.077 0.075 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.468 | 0.161 | Glutamate decarboxylase inhibitor | 0.093 0.034 CHEMBL3706523 0.161 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.463 | 0.165 | Cannabinoid CB2 receptor agonist | 0.165 0.009 CHEMBL3706522 | CHEMBL3706522 | |
| 0.039 | 0.501 | 0.099 | Interleukin 12 antagonist | 0.099 0.055 CHEMBL3706526 | CHEMBL3706526 | |
| 0.042 | 0.504 | 0.233 | 3C-like protease (Human coronavirus) inhibitor | 0.233 0.035 CHEMBL3706522 0.224 0.039 CHEMBL3706523 0.145 0.11 CHEMBL3706526 0.138 0.123 CHEMBL3706524 | CHEMBL3706522 | |
| 0.018 | 0.485 | 0.072 | Corticotropin releasing factor 2 receptor antagonist | 0.072 0.026 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.482 | 0.05 | Glutamate (mGluR3) antagonist | 0.05 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.495 | 0.191 | Glutamate receptor agonist | 0.175 0.013 CHEMBL3706522 0.191 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.038 | 0.53 | 0.365 | Calpain 2 inhibitor | 0.274 0.132 CHEMBL3706522 0.365 0.079 CHEMBL3706523 0.205 0.183 CHEMBL3706526 0.351 0.086 CHEMBL3706524 | CHEMBL3706523 | |
| 0.004 | 0.498 | 0.039 | LFA antagonist | 0.039 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.01 | 0.508 | 0.096 | Sphingosine 1-phosphate receptor 3 antagonist | 0.096 0.009 CHEMBL3706522 0.059 0.04 CHEMBL3706526 | CHEMBL3706522 | |
| 0.016 | 0.518 | 0.113 | Phosphodiesterase 11A inhibitor | 0.113 0.023 CHEMBL3706522 | CHEMBL3706522 | |
| 0.016 | 0.518 | 0.113 | Phosphodiesterase XI inhibitor | 0.113 0.023 CHEMBL3706522 | CHEMBL3706522 | |
| 0.012 | 0.515 | 0.093 | Botulinum neurotoxin type A inhibitor | 0.057 0.042 CHEMBL3706522 0.056 0.045 CHEMBL3706523 0.093 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.029 | 0.538 | 0.121 | Activin receptor-like kinase 4 inhibitor | 0.121 0.051 CHEMBL3706522 | CHEMBL3706522 | |
| 0.014 | 0.527 | 0.185 | Sodium channel blocker | 0.185 0.038 CHEMBL3706522 | CHEMBL3706522 | |
| 0.074 | 0.589 | 0.332 | Tyrosine 3 hydroxylase inhibitor | 0.302 0.032 CHEMBL3706522 0.332 0.021 CHEMBL3706526 0.251 0.067 CHEMBL3706527 0.185 0.164 CHEMBL3706524 | CHEMBL3706526 | |
| 0.004 | 0.524 | 0.021 | Geranylgeranyltransferase inhibitor | 0.021 0.017 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.531 | 0.05 | Thromboxane synthase inhibitor | 0.05 0.049 CHEMBL3706522 | CHEMBL3706522 | |
| 0.006 | 0.539 | 0.059 | Calcium channel T-type blocker | 0.059 0.038 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.536 | 0.02 | Integrin alphaVbeta6 antagonist | 0.02 0.006 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.546 | 0.077 | Adrenaline agonist | 0.077 0.062 CHEMBL3706527 | CHEMBL3706527 | |
| 0.01 | 0.551 | 0.109 | Platelet growth factor antagonist | 0.109 0.035 CHEMBL3706522 | CHEMBL3706522 | |
| 0.019 | 0.564 | 0.164 | Toll-Like receptor 2 antagonist | 0.164 0.043 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.552 | 0.051 | Membrane dipeptidase inhibitor | 0.051 0.015 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.552 | 0.063 | Collagenase 3 inhibitor | 0.053 0.052 CHEMBL3706522 0.063 0.038 CHEMBL3706526 | CHEMBL3706526 | |
| 0.018 | 0.568 | 0.104 | Glutamate (mGluR6) antagonist | 0.077 0.028 CHEMBL3706522 0.104 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.558 | 0.15 | Phenylalanine 4-hydroxylase inhibitor | 0.076 0.041 CHEMBL3706522 0.15 0.012 CHEMBL3706526 | CHEMBL3706526 | |
| 0.016 | 0.566 | 0.085 | Prolactin inhibitor | 0.085 0.074 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.565 | 0.052 | Tryptophan 5 hydroxylase inhibitor | 0.052 0.005 CHEMBL3706526 | CHEMBL3706526 | |
| 0.036 | 0.594 | 0.137 | Vanilloid 1 agonist | 0.137 0.055 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.565 | 0.022 | Toll-Like receptor 8 agonist | 0.022 0.01 CHEMBL3706522 | CHEMBL3706522 | |
| 0.019 | 0.579 | 0.173 | Acetylcholine M1 receptor antagonist | 0.173 0.056 CHEMBL3706527 | CHEMBL3706527 | |
| 0.021 | 0.583 | 0.075 | Vanilloid 4 agonist | 0.075 0.051 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.573 | 0.19 | Sodium channel (voltage-gated) blocker | 0.19 0.033 CHEMBL3706522 | CHEMBL3706522 | |
| 0.02 | 0.586 | 0.174 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.174 0.02 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.575 | 0.131 | Pim-1 kinase inhibitor | 0.131 0.036 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.579 | 0.034 | Benzodiazepine receptor peripheral-type antagonist | 0.034 0.024 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.577 | 0.057 | Glucagon receptor antagonist | 0.057 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.586 | 0.078 | Protein kinase C beta inhibitor | 0.078 0.032 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.586 | 0.119 | Ornithine carbamoyltransferase inhibitor | 0.119 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.594 | 0.087 | Expectorant | 0.087 0.086 CHEMBL3706527 | CHEMBL3706527 | |
| 0.002 | 0.594 | 0.105 | Antimetabolite | 0.041 0.039 CHEMBL3706523 0.105 0.015 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.609 | 0.139 | Alkylator | 0.109 0.078 CHEMBL3706523 0.139 0.053 CHEMBL3706526 | CHEMBL3706526 | |
| 0.012 | 0.616 | 0.14 | Caspase 3 inhibitor | 0.121 0.059 CHEMBL3706523 0.14 0.036 CHEMBL3706526 0.103 0.087 CHEMBL3706524 | CHEMBL3706526 | |
| 0.01 | 0.616 | 0.097 | Mucolytic | 0.097 0.082 CHEMBL3706527 | CHEMBL3706527 | |
| 0 | 0.608 | 0.005 | Reverse transcriptase (HBV) inhibitor | 0.005 0.003 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.613 | 0.034 | Lysine carboxypeptidase inhibitor | 0.034 0.013 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.618 | 0.112 | AICAR transformylase inhibitor | 0.042 0.035 CHEMBL3706522 0.054 0.018 CHEMBL3706523 0.112 0.004 CHEMBL3706526 0.04 0.037 CHEMBL3706524 | CHEMBL3706526 | |
| 0.006 | 0.622 | 0.057 | Lysophosphatidic acid 3 receptor antagonist | 0.057 0.026 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.62 | 0.095 | Nav1.7 sodium channel blocker | 0.095 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.622 | 0.19 | Cannabinoid receptor antagonist | 0.19 0.009 CHEMBL3706522 | CHEMBL3706522 | |
| 0.016 | 0.633 | 0.123 | Interleukin 8 antagonist | 0.123 0.057 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.628 | 0.18 | Phospholipase A2 inhibitor | 0.18 0.054 CHEMBL3706526 0.129 0.102 CHEMBL3706524 | CHEMBL3706526 | |
| 0.004 | 0.625 | 0.043 | Glutamate (mGluR5) antagonist | 0.043 0.038 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.627 | 0.038 | Kainate receptor 2 antagonist | 0.038 0.023 CHEMBL3706526 | CHEMBL3706526 | |
| 0.02 | 0.645 | 0.258 | Transcription factor NF kappa B inhibitor | 0.258 0.121 CHEMBL3706526 | CHEMBL3706526 | |
| 0.015 | 0.641 | 0.106 | Sphingomyelinase inhibitor | 0.106 0.053 CHEMBL3706522 | CHEMBL3706522 | |
| 0.014 | 0.644 | 0.214 | Glutamate dehydrogenase inhibitor | 0.214 0.009 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.634 | 0.137 | Glutamate (mGluR group I) agonist | 0.137 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.644 | 0.058 | Sphingosine 1-phosphate receptor 1 antagonist | 0.058 0.033 CHEMBL3706522 | CHEMBL3706522 | |
| 0.008 | 0.657 | 0.098 | MAP kinase 9 inhibitor | 0.098 0.064 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.656 | 0.178 | Cannabinoid CB1 receptor antagonist | 0.178 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.663 | 0.02 | Integrin beta2 antagonist | 0.02 0.005 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.667 | 0.04 | Vascular adhesion protein 1 inhibitor | 0.04 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.674 | 0.102 | Aconitate hydratase inhibitor | 0.072 0.017 CHEMBL3706522 0.102 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.009 | 0.679 | 0.09 | Mediator release inhibitor | 0.09 0.081 CHEMBL3706526 | CHEMBL3706526 | |
| 0.015 | 0.687 | 0.246 | DNA synthesis inhibitor | 0.246 0.069 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.676 | 0.077 | Cannabinoid CB2 receptor antagonist | 0.077 0.021 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.682 | 0.095 | Diacylglycerol O-acyltransferase inhibitor | 0.095 0.009 CHEMBL3706522 0.087 0.011 CHEMBL3706526 | CHEMBL3706522 | |
| 0.003 | 0.695 | 0.118 | Glutamate (mGluR5) agonist | 0.118 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.705 | 0.04 | Angiotensin AT1 receptor antagonist | 0.04 0.034 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.708 | 0.087 | Histidine decarboxylase inhibitor | 0.087 0.038 CHEMBL3706526 | CHEMBL3706526 | |
| 0.011 | 0.716 | 0.069 | Keratolytic | 0.069 0.068 CHEMBL3706522 | CHEMBL3706522 | |
| 0.013 | 0.727 | 0.103 | Acetylcholine release stimulant | 0.103 0.08 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.715 | 0.009 | Integrin alphaVbeta5 antagonist | 0.009 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.01 | 0.729 | 0.174 | Alpha-N-acetylglucosaminidase inhibitor | 0.167 0.046 CHEMBL3706522 0.128 0.07 CHEMBL3706523 0.174 0.043 CHEMBL3706526 | CHEMBL3706526 | |
| 0.02 | 0.739 | 0.158 | Phospholipase C inhibitor | 0.158 0.092 CHEMBL3706526 | CHEMBL3706526 | |
| 0.019 | 0.741 | 0.198 | Neurotrophic factor enhancer | 0.198 0.079 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.725 | 0.05 | Histamine agonist | 0.05 0.041 CHEMBL3706522 | CHEMBL3706522 | |
| 0.016 | 0.748 | 0.29 | Antibacterial | 0.29 0.143 CHEMBL3706526 | CHEMBL3706526 | |
| 0.001 | 0.734 | 0.035 | Fumarate hydratase inhibitor | 0.035 0.023 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.743 | 0.06 | Biliverdin reductase inhibitor | 0.06 0.04 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.751 | 0.081 | TRPA1 antagonist | 0.081 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.01 | 0.762 | 0.052 | Nicotinic alpha3beta2 receptor antagonist | 0.052 0.04 CHEMBL3706522 | CHEMBL3706522 | |
| 0.006 | 0.758 | 0.043 | Kainate receptor agonist | 0.043 0.025 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.76 | 0.102 | Glycine receptor antagonist | 0.102 0.03 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.763 | 0.049 | Cytokine production stimulant | 0.049 0.032 CHEMBL3706522 | CHEMBL3706522 | |
| 0.053 | 0.812 | 0.216 | 5 Hydroxytryptamine uptake stimulant | 0.216 0.123 CHEMBL3706522 0.206 0.14 CHEMBL3706526 0.214 0.126 CHEMBL3706527 | CHEMBL3706522 | |
| 0.005 | 0.765 | 0.094 | Sphingosine 1-phosphate receptor antagonist | 0.094 0.026 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.768 | 0.06 | Histone deacetylase inhibitor | 0.06 0.055 CHEMBL3706522 | CHEMBL3706522 | |
| 0.025 | 0.791 | 0.464 | Histamine release inhibitor | 0.464 0.043 CHEMBL3706522 0.403 0.074 CHEMBL3706526 | CHEMBL3706522 | |
| 0.002 | 0.772 | 0.037 | Epoxide hydrolase 1 inhibitor | 0.037 0.014 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.773 | 0.107 | Carbamoyl phosphate synthetase inhibitor | 0.107 0.019 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.777 | 0.09 | Sphingosine 1-phosphate receptor 4 agonist | 0.083 0.034 CHEMBL3706522 0.09 0.03 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.777 | 0.211 | Porphobilinogen synthase inhibitor | 0.143 0.022 CHEMBL3706522 0.211 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.788 | 0.189 | GABA C receptor rho-1 antagonist | 0.189 0.01 CHEMBL3706522 0.167 0.015 CHEMBL3706526 | CHEMBL3706522 | |
| 0.006 | 0.788 | 0.084 | Potassium channel (Tandem pore domain) blocker | 0.084 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.027 | 0.81 | 0.098 | Glutamate release inhibitor | 0.098 0.045 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.789 | 0.049 | Glutamate (mGluR8) agonist | 0.049 0.012 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.788 | 0.037 | ICAM 1 antagonist | 0.037 0.005 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.791 | 0.072 | Pim-2 kinase inhibitor | 0.072 0.023 CHEMBL3706522 | CHEMBL3706522 | |
| 0.016 | 0.806 | 0.129 | Glutamate (mGluR7) agonist | 0.129 0.023 CHEMBL3706522 0.117 0.034 CHEMBL3706526 | CHEMBL3706522 | |
| 0.003 | 0.798 | 0.105 | Glutamate (mGluR1a) antagonist | 0.105 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.799 | 0.025 | Glutamate (mGluR1) agonist | 0.025 0.016 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.809 | 0.107 | Cyclooxygenase 3 inhibitor | 0.107 0.093 CHEMBL3706526 | CHEMBL3706526 | |
| 0.012 | 0.811 | 0.167 | Cytokine production inhibitor | 0.167 0.051 CHEMBL3706522 | CHEMBL3706522 | |
| 0.013 | 0.814 | 0.301 | Peroxidase inhibitor | 0.19 0.062 CHEMBL3706522 0.301 0.037 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.804 | 0.12 | Thymidylate synthase inhibitor | 0.042 0.039 CHEMBL3706522 0.049 0.029 CHEMBL3706523 0.12 0.004 CHEMBL3706526 | CHEMBL3706526 | |
| 0.006 | 0.808 | 0.256 | Ferrochelatase inhibitor | 0.184 0.026 CHEMBL3706522 0.256 0.012 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.808 | 0.134 | Beta amyloid protein antagonist | 0.134 0.053 CHEMBL3706522 0.103 0.086 CHEMBL3706526 | CHEMBL3706522 | |
| 0.002 | 0.807 | 0.061 | Alcohol oxidase inhibitor | 0.061 0.035 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.81 | 0.07 | Glutamate (mGluR7) antagonist | 0.07 0.043 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.813 | 0.091 | Interleukin-1 receptor-associated protein kinase 4 inhibitor | 0.091 0.056 CHEMBL3706522 | CHEMBL3706522 | |
| 0.014 | 0.829 | 0.139 | Photosensitizer | 0.139 0.039 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.821 | 0.078 | GABA B receptor agonist | 0.078 0.047 CHEMBL3706526 | CHEMBL3706526 | |
| 0.008 | 0.827 | 0.093 | Glutathione S-transferase inhibitor | 0.093 0.045 CHEMBL3706526 | CHEMBL3706526 | |
| 0.009 | 0.834 | 0.135 | Granulocyte macrophage colony stimulating factor agonist | 0.135 0.009 CHEMBL3706522 0.119 0.016 CHEMBL3706526 | CHEMBL3706522 | |
| 0.002 | 0.828 | 0.113 | Argininosuccinate synthase inhibitor | 0.113 0.016 CHEMBL3706526 | CHEMBL3706526 | |
| 0.001 | 0.828 | 0.04 | Protein kinase (CK1) epsilon inhibitor | 0.04 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.832 | 0.102 | Heat shock protein 90 beta antagonist | 0.102 0.01 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.831 | 0.093 | Androgen antagonist | 0.093 0.052 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.834 | 0.121 | Creatine kinase inhibitor | 0.121 0.04 CHEMBL3706522 0.114 0.046 CHEMBL3706526 | CHEMBL3706522 | |
| 0.006 | 0.835 | 0.049 | Aldosterone antagonist | 0.049 0.031 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.836 | 0.197 | Pregnane X receptor agonist | 0.197 0.012 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.84 | 0.132 | Sphingosine 1-phosphate receptor 5 antagonist | 0.132 0.096 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.835 | 0.045 | Histamine H2 receptor agonist | 0.045 0.027 CHEMBL3706522 | CHEMBL3706522 | |
| 0.007 | 0.841 | 0.108 | DOPA decarboxylase inhibitor | 0.099 0.077 CHEMBL3706522 0.108 0.062 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.845 | 0.089 | Adenosine A3 receptor antagonist | 0.089 0.033 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.845 | 0.044 | Histamine H1 receptor agonist | 0.044 0.031 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.847 | 0.116 | Glutamate (mGluR group III) agonist | 0.054 0.021 CHEMBL3706522 0.116 0.008 CHEMBL3706526 | CHEMBL3706526 | |
| 0.009 | 0.853 | 0.122 | Sphingosine 1-phosphate receptor 4 antagonist | 0.122 0.069 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.854 | 0.084 | Triose-phosphate isomerase inhibitor | 0.084 0.068 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.85 | 0.106 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.106 0.01 CHEMBL3706522 0.085 0.028 CHEMBL3706526 | CHEMBL3706522 | |
| 0.005 | 0.855 | 0.165 | GABA C receptor antagonist | 0.165 0.023 CHEMBL3706522 0.144 0.033 CHEMBL3706526 | CHEMBL3706522 | |
| 0.006 | 0.858 | 0.203 | Succinate dehydrogenase inhibitor | 0.159 0.096 CHEMBL3706522 0.203 0.047 CHEMBL3706526 | CHEMBL3706526 | |
| 0.009 | 0.863 | 0.214 | DNA methylase inhibitor | 0.214 0.07 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.86 | 0.128 | NMDA receptor agonist | 0.128 0.011 CHEMBL3706526 | CHEMBL3706526 | |
| 0.017 | 0.875 | 0.43 | 5 Hydroxytryptamine release inhibitor | 0.43 0.061 CHEMBL3706522 0.387 0.086 CHEMBL3706526 | CHEMBL3706522 | |
| 0.001 | 0.861 | 0.042 | Carbonic anhydrase IV inhibitor | 0.042 0.03 CHEMBL3706526 | CHEMBL3706526 | |
| 0.007 | 0.869 | 0.16 | DNA methyltransferase I inhibitor | 0.16 0.094 CHEMBL3706526 | CHEMBL3706526 | |
| 0.01 | 0.873 | 0.194 | ATPase inhibitor | 0.194 0.042 CHEMBL3706522 | CHEMBL3706522 | |
| 0.011 | 0.878 | 0.088 | Lanosterol 14 alpha demethylase inhibitor | 0.088 0.075 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.878 | 0.063 | Phosphodiesterase 1C inhibitor | 0.063 0.042 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.876 | 0.04 | Diamine oxidase inhibitor | 0.04 0.023 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.877 | 0.053 | Glutamate (mGluR4) agonist | 0.034 0.022 CHEMBL3706522 0.053 0.01 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.893 | 0.103 | Adenylate kinase inhibitor | 0.103 0.063 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.882 | 0.044 | Purinergic P2Y antagonist | 0.044 0.032 CHEMBL3706522 0.041 0.036 CHEMBL3706526 | CHEMBL3706522 | |
| 0.005 | 0.886 | 0.199 | Heat shock protein 90 antagonist | 0.199 0.038 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.89 | 0.171 | GABA C receptor agonist | 0.086 0.085 CHEMBL3706522 0.171 0.027 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.893 | 0.231 | DNA damaging | 0.231 0.092 CHEMBL3706526 | CHEMBL3706526 | |
| 0.002 | 0.894 | 0.106 | TRKA antagonist | 0.106 0.081 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.893 | 0.061 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.061 0.033 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.894 | 0.062 | Benzodiazepine antagonist | 0.062 0.012 CHEMBL3706522 | CHEMBL3706522 | |
| 0.006 | 0.899 | 0.145 | Aldehyde oxidase inhibitor | 0.145 0.144 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.895 | 0.112 | Tyrosine-protein kinase receptor antagonist | 0.112 0.095 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.895 | 0.048 | Dihydrofolate reductase inhibitor | 0.048 0.022 CHEMBL3706526 | CHEMBL3706526 | |
| 0.005 | 0.899 | 0.086 | Phosphodiesterase I inhibitor | 0.086 0.066 CHEMBL3706522 | CHEMBL3706522 | |
| 0 | 0.896 | 0.018 | Egl nine homolog 1 inhibitor | 0.018 0.007 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.905 | 0.098 | D-Ala-D-Ala ligase inhibitor | 0.098 0.032 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.899 | 0.036 | Glucosylceramidase stimulant | 0.036 0.005 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.901 | 0.02 | Glutamate (mGluR1a) agonist | 0.02 0.019 CHEMBL3706526 | CHEMBL3706526 | |
| 0.027 | 0.931 | 0.41 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.41 0.092 CHEMBL3706522 | CHEMBL3706522 | |
| 0.031 | 0.935 | 0.214 | Nitric-oxide synthase stimulant | 0.214 0.067 CHEMBL3706522 | CHEMBL3706522 | |
| 0.006 | 0.911 | 0.303 | GABA C receptor rho-2 antagonist | 0.303 0.005 CHEMBL3706522 0.158 0.064 CHEMBL3706526 | CHEMBL3706522 | |
| 0.003 | 0.909 | 0.163 | Cyclin-dependent kinase 8 inhibitor | 0.163 0.067 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.911 | 0.168 | Pyruvate kinase inhibitor | 0.168 0.102 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.911 | 0.044 | MAP3K5 inhibitor | 0.044 0.019 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.911 | 0.083 | Pim-3 kinase inhibitor | 0.083 0.07 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.914 | 0.14 | Non-steroidal antiinflammatory agent | 0.14 0.13 CHEMBL3706526 | CHEMBL3706526 | |
| 0.003 | 0.914 | 0.093 | 5 Hydroxytryptamine 3A agonist | 0.093 0.085 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.92 | 0.167 | Cell wall synthesis inhibitor | 0.167 0.05 CHEMBL3706526 | CHEMBL3706526 | |
| 0.013 | 0.929 | 0.133 | Ca2+-transporting ATPase inhibitor | 0.133 0.105 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.919 | 0.131 | Arachidonic acid antagonist | 0.131 0.112 CHEMBL3706522 | CHEMBL3706522 | |
| 0.008 | 0.926 | 0.163 | MAP kinase 3 inhibitor | 0.163 0.05 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.919 | 0.093 | Aryl hydrocarbon receptor antagonist | 0.093 0.017 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.923 | 0.262 | MAP kinase 1 inhibitor | 0.262 0.219 CHEMBL3706522 | CHEMBL3706522 | |
| 0.028 | 0.946 | 0.18 | 5 Hydroxytryptamine 3E antagonist | 0.18 0.106 CHEMBL3706522 | CHEMBL3706522 | |
| 0.009 | 0.928 | 0.192 | CF transmembrane conductance regulator agonist | 0.192 0.027 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.922 | 0.064 | Benzodiazepine agonist | 0.064 0.061 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.925 | 0.059 | Phosphodiesterase 1A inhibitor | 0.059 0.044 CHEMBL3706522 | CHEMBL3706522 | |
| 0.01 | 0.931 | 0.576 | GABA C receptor rho-3 antagonist | 0.576 0.01 CHEMBL3706522 0.316 0.106 CHEMBL3706526 | CHEMBL3706522 | |
| 0.002 | 0.929 | 0.04 | Potassium channel Kv1.1 blocker | 0.04 0.023 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.93 | 0.106 | Cystathionine beta-synthase inhibitor | 0.106 0.07 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.934 | 0.23 | Transcription factor inhibitor | 0.23 0.201 CHEMBL3706522 | CHEMBL3706522 | |
| 0.003 | 0.936 | 0.237 | Heat shock protein 90 alpha antagonist | 0.237 0.031 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.935 | 0.193 | MAP kinase kinase 2 inhibitor | 0.193 0.086 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.936 | 0.044 | Inosine monophosphate dehydrogenase inhibitor | 0.044 0.019 CHEMBL3706522 | CHEMBL3706522 | |
| 0.005 | 0.947 | 0.067 | Transcription factor RelA inhibitor | 0.067 0.036 CHEMBL3706522 | CHEMBL3706522 | |
| 0.014 | 0.956 | 0.271 | Calcium channel activator | 0.271 0.123 CHEMBL3706522 | CHEMBL3706522 | |
| 0.006 | 0.953 | 0.166 | Histone acetyltransferase inhibitor | 0.166 0.118 CHEMBL3706522 | CHEMBL3706522 | |
| 0.004 | 0.953 | 0.124 | DNA repair enzyme inhibitor | 0.124 0.065 CHEMBL3706526 | CHEMBL3706526 | |
| 0.004 | 0.955 | 0.25 | Hypoxia-inducible factor 1 alpha inhibitor | 0.25 0.1 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.956 | 0.079 | Potassium channel activator | 0.079 0.077 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.956 | 0.053 | Potassium channel (ATP-sensitive) activator | 0.053 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.957 | 0.056 | Potassium channel (Inward rectifier) activator | 0.056 0.025 CHEMBL3706522 | CHEMBL3706522 | |
| 0.002 | 0.959 | 0.152 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.152 0.144 CHEMBL3706522 | CHEMBL3706522 | |
| 0.001 | 0.968 | 0.156 | Aryl hydrocarbon receptor agonist | 0.156 0.131 CHEMBL3706522 | CHEMBL3706522 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |