| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.848 | 0.002 | 0.878 | Protease inhibitor | 0.719 0.003 CHEMBL3526717 0.878 0.002 CHEMBL3526718 0.267 0.007 CHEMBL3526892 0.606 0.003 CHEMBL3988903 0.807 0.003 CHEMBL3526789 0.807 0.003 CHEMBL3526788 0.556 0.003 CHEMBL3526896 0.124 0.044 CHEMBL3988901 0.808 0.003 CHEMBL3526787 0.868 0.002 CHEMBL3526719 0.107 0.059 CHEMBL3988902 | CHEMBL3526718 | |
| 0.645 | 0.002 | 0.645 | HIV-1 protease inhibitor | 0.405 0.003 CHEMBL3526717 0.537 0.003 CHEMBL3526718 0.065 0.009 CHEMBL3526892 0.262 0.003 CHEMBL3988903 0.61 0.002 CHEMBL3526789 0.61 0.002 CHEMBL3526788 0.284 0.003 CHEMBL3526896 0.567 0.003 CHEMBL3526787 0.52 0.003 CHEMBL3526719 | ||
| 0.224 | 0.019 | 0.319 | Proteasome inhibitor | 0.294 0.01 CHEMBL3526717 0.197 0.026 CHEMBL3526718 0.181 0.032 CHEMBL3526892 0.319 0.008 CHEMBL3988903 0.199 0.025 CHEMBL3526789 0.199 0.025 CHEMBL3526788 0.206 0.023 CHEMBL3526896 0.149 0.047 CHEMBL3988901 0.209 0.022 CHEMBL3526787 0.19 0.029 CHEMBL3526719 0.096 0.093 CHEMBL3542352 0.148 0.048 CHEMBL3988902 | CHEMBL3988903 | |
| 0.201 | 0.022 | 0.32 | Cathepsin H inhibitor | 0.286 0.011 CHEMBL3526717 0.145 0.05 CHEMBL3542349 0.152 0.045 CHEMBL3526718 0.215 0.019 CHEMBL3526892 0.309 0.009 CHEMBL3988903 0.207 0.021 CHEMBL3526789 0.207 0.021 CHEMBL3526788 0.32 0.009 CHEMBL3526896 0.199 0.023 CHEMBL3542351 0.166 0.036 CHEMBL3526787 0.166 0.036 CHEMBL3526719 0.129 0.065 CHEMBL3542352 0.13 0.064 CHEMBL3988902 | CHEMBL3526896 | |
| 0.269 | 0.093 | 0.269 | Nootropic | 0.21 0.145 CHEMBL3526718 0.215 0.139 CHEMBL3526789 0.215 0.139 CHEMBL3526788 0.225 0.129 CHEMBL3542350 0.248 0.11 CHEMBL3526787 0.234 0.122 CHEMBL3526719 | ||
| 0.181 | 0.005 | 0.273 | Cathepsin D inhibitor | 0.256 0.004 CHEMBL3526717 0.157 0.007 CHEMBL3526718 0.177 0.005 CHEMBL3988903 0.165 0.006 CHEMBL3526789 0.165 0.006 CHEMBL3526788 0.273 0.004 CHEMBL3526896 0.163 0.006 CHEMBL3526787 0.158 0.007 CHEMBL3526719 | CHEMBL3526896 | |
| 0.184 | 0.046 | 0.353 | Thiol protease inhibitor | 0.211 0.036 CHEMBL3526717 0.12 0.118 CHEMBL3542349 0.147 0.072 CHEMBL3526718 0.157 0.063 CHEMBL3526892 0.271 0.023 CHEMBL3988903 0.161 0.06 CHEMBL3526789 0.161 0.06 CHEMBL3526788 0.171 0.053 CHEMBL3526896 0.149 0.069 CHEMBL3542351 0.353 0.015 CHEMBL3988901 0.168 0.055 CHEMBL3526787 0.168 0.055 CHEMBL3526719 0.141 0.079 CHEMBL3542352 0.257 0.025 CHEMBL3988902 | CHEMBL3988901 | |
| 0.139 | 0.01 | 0.296 | Human rhinovirus A protease inhibitor | 0.247 0.005 CHEMBL3526717 0.113 0.013 CHEMBL3526718 0.103 0.015 CHEMBL3526892 0.296 0.004 CHEMBL3988903 0.13 0.011 CHEMBL3526789 0.13 0.011 CHEMBL3526788 0.231 0.005 CHEMBL3526896 0.119 0.012 CHEMBL3526787 0.091 0.019 CHEMBL3526719 0.049 0.044 CHEMBL3988902 | CHEMBL3988903 | |
| 0.131 | 0.007 | 0.131 | Cathepsin E inhibitor | 0.113 0.01 CHEMBL3526717 0.116 0.009 CHEMBL3526718 0.105 0.012 CHEMBL3988903 0.123 0.008 CHEMBL3526789 0.123 0.008 CHEMBL3526788 0.098 0.014 CHEMBL3526896 0.12 0.009 CHEMBL3526787 0.12 0.009 CHEMBL3526719 | ||
| 0.212 | 0.108 | 0.225 | Cardiotonic | 0.187 0.132 CHEMBL3526718 0.171 0.151 CHEMBL3526789 0.171 0.151 CHEMBL3526788 0.225 0.099 CHEMBL3526787 0.187 0.131 CHEMBL3526719 | CHEMBL3526787 | |
| 0.105 | 0.004 | 0.12 | Plasmepsin II inhibitor | 0.083 0.005 CHEMBL3526717 0.074 0.007 CHEMBL3526718 0.056 0.014 CHEMBL3988903 0.08 0.006 CHEMBL3526789 0.08 0.006 CHEMBL3526788 0.12 0.004 CHEMBL3526896 0.084 0.005 CHEMBL3526787 0.084 0.005 CHEMBL3526719 | CHEMBL3526896 | |
| 0.204 | 0.11 | 0.391 | Calpain inhibitor | 0.296 0.032 CHEMBL3526717 0.249 0.065 CHEMBL3542349 0.325 0.022 CHEMBL3526892 0.391 0.01 CHEMBL3988903 0.324 0.022 CHEMBL3526896 0.233 0.081 CHEMBL3542350 0.162 0.16 CHEMBL3542351 0.273 0.046 CHEMBL3988901 0.194 0.119 CHEMBL3542352 0.269 0.049 CHEMBL3988902 | CHEMBL3988903 | |
| 0.096 | 0.007 | 0.096 | Glucose-6-phosphate translocase inhibitor | 0.095 0.007 CHEMBL3542349 0.086 0.009 CHEMBL3526718 0.09 0.008 CHEMBL3526789 0.09 0.008 CHEMBL3526788 0.052 0.035 CHEMBL3542350 0.053 0.034 CHEMBL3542351 0.088 0.009 CHEMBL3526787 0.088 0.009 CHEMBL3526719 | ||
| 0.123 | 0.036 | 0.22 | Factor V inhibitor | 0.143 0.022 CHEMBL3526717 0.117 0.042 CHEMBL3526718 0.111 0.05 CHEMBL3526892 0.22 0.004 CHEMBL3988903 0.127 0.033 CHEMBL3526789 0.127 0.033 CHEMBL3526788 0.14 0.023 CHEMBL3526896 0.149 0.019 CHEMBL3988901 0.118 0.041 CHEMBL3526787 0.118 0.041 CHEMBL3526719 0.107 0.055 CHEMBL3988902 | CHEMBL3988903 | |
| 0.101 | 0.016 | 0.229 | Cathepsin B inhibitor | 0.16 0.006 CHEMBL3526717 0.087 0.021 CHEMBL3526718 0.089 0.02 CHEMBL3526892 0.229 0.004 CHEMBL3988903 0.091 0.02 CHEMBL3526789 0.091 0.02 CHEMBL3526788 0.145 0.007 CHEMBL3526896 0.067 0.03 CHEMBL3988901 0.091 0.019 CHEMBL3526787 0.083 0.023 CHEMBL3526719 | CHEMBL3988903 | |
| 0.081 | 0.004 | 0.081 | Plasmepsin I inhibitor | 0.075 0.004 CHEMBL3526717 0.073 0.004 CHEMBL3526718 0.056 0.005 CHEMBL3988903 0.075 0.004 CHEMBL3526789 0.075 0.004 CHEMBL3526788 0.063 0.005 CHEMBL3526896 0.075 0.004 CHEMBL3526787 0.075 0.004 CHEMBL3526719 | ||
| 0.105 | 0.028 | 0.105 | HIV-1 reverse transcriptase inhibitor | 0.08 0.042 CHEMBL3526718 0.083 0.04 CHEMBL3526789 0.083 0.04 CHEMBL3526788 0.089 0.036 CHEMBL3526787 0.081 0.041 CHEMBL3526719 | ||
| 0.114 | 0.041 | 0.211 | Interleukin 1 beta converting enzyme inhibitor | 0.135 0.025 CHEMBL3526717 0.088 0.076 CHEMBL3542349 0.131 0.027 CHEMBL3526892 0.201 0.005 CHEMBL3988903 0.09 0.072 CHEMBL3526896 0.111 0.044 CHEMBL3542351 0.173 0.01 CHEMBL3988901 0.09 0.072 CHEMBL3526787 0.164 0.013 CHEMBL3542352 0.211 0.005 CHEMBL3988902 | CHEMBL3988902 | |
| 0.224 | 0.153 | 0.496 | Apoptosis antagonist | 0.261 0.117 CHEMBL3526717 0.274 0.105 CHEMBL3542349 0.193 0.189 CHEMBL3526718 0.341 0.06 CHEMBL3988903 0.207 0.17 CHEMBL3526789 0.207 0.17 CHEMBL3526788 0.229 0.148 CHEMBL3542351 0.458 0.026 CHEMBL3988901 0.209 0.168 CHEMBL3526787 0.209 0.168 CHEMBL3526719 0.261 0.117 CHEMBL3542352 0.496 0.021 CHEMBL3988902 | CHEMBL3988902 | |
| 0.096 | 0.039 | 0.219 | Chymotrypsin inhibitor | 0.141 0.019 CHEMBL3526717 0.086 0.047 CHEMBL3526718 0.089 0.044 CHEMBL3526892 0.219 0.007 CHEMBL3988903 0.094 0.04 CHEMBL3526789 0.094 0.04 CHEMBL3526788 0.148 0.017 CHEMBL3526896 0.073 0.065 CHEMBL3988901 0.09 0.044 CHEMBL3526787 0.084 0.05 CHEMBL3526719 | CHEMBL3988903 | |
| 0.089 | 0.043 | 0.354 | Catalase inhibitor | 0.226 0.011 CHEMBL3526717 0.077 0.049 CHEMBL3526718 0.354 0.004 CHEMBL3988903 0.1 0.039 CHEMBL3526789 0.1 0.039 CHEMBL3526788 0.167 0.022 CHEMBL3526896 0.178 0.02 CHEMBL3542351 0.162 0.023 CHEMBL3988901 0.098 0.039 CHEMBL3526787 0.098 0.039 CHEMBL3526719 0.109 0.036 CHEMBL3542352 0.134 0.03 CHEMBL3988902 | CHEMBL3988903 | |
| 0.059 | 0.013 | 0.149 | Renin inhibitor | 0.133 0.005 CHEMBL3526717 0.053 0.016 CHEMBL3526718 0.149 0.005 CHEMBL3988903 0.056 0.015 CHEMBL3526789 0.056 0.015 CHEMBL3526788 0.102 0.006 CHEMBL3526896 0.055 0.015 CHEMBL3526787 0.055 0.015 CHEMBL3526719 | CHEMBL3988903 | |
| 0.099 | 0.055 | 0.153 | Falcipain inhibitor | 0.153 0.029 CHEMBL3526717 0.136 0.037 CHEMBL3542349 0.079 0.075 CHEMBL3526718 0.129 0.04 CHEMBL3526892 0.15 0.031 CHEMBL3988903 0.086 0.066 CHEMBL3526789 0.086 0.066 CHEMBL3526788 0.102 0.054 CHEMBL3526896 0.085 0.068 CHEMBL3526787 0.085 0.068 CHEMBL3526719 | CHEMBL3526717 | |
| 0.088 | 0.051 | 0.187 | 3C-Like protease (SARS coronavirus) inhibitor | 0.102 0.031 CHEMBL3526717 0.083 0.06 CHEMBL3526718 0.187 0.005 CHEMBL3988903 0.082 0.062 CHEMBL3526789 0.082 0.062 CHEMBL3526788 0.099 0.034 CHEMBL3526896 0.079 0.072 CHEMBL3542351 0.085 0.055 CHEMBL3526787 0.085 0.055 CHEMBL3526719 | CHEMBL3988903 | |
| 0.071 | 0.035 | 0.233 | Protease 3C (Human rhinovirus) inhibitor | 0.195 0.004 CHEMBL3526717 0.072 0.034 CHEMBL3542349 0.088 0.022 CHEMBL3526718 0.09 0.02 CHEMBL3526892 0.233 0.003 CHEMBL3988903 0.069 0.038 CHEMBL3526789 0.069 0.038 CHEMBL3526788 0.12 0.01 CHEMBL3526896 0.082 0.025 CHEMBL3988901 0.08 0.027 CHEMBL3526787 0.081 0.026 CHEMBL3526719 0.073 0.034 CHEMBL3988902 | CHEMBL3988903 | |
| 0.068 | 0.034 | 0.161 | Caspase 9 inhibitor | 0.088 0.018 CHEMBL3526717 0.063 0.042 CHEMBL3526718 0.072 0.03 CHEMBL3526892 0.161 0.005 CHEMBL3988903 0.064 0.04 CHEMBL3526789 0.064 0.04 CHEMBL3526788 0.085 0.02 CHEMBL3526896 0.06 0.048 CHEMBL3988901 0.064 0.039 CHEMBL3526787 0.064 0.04 CHEMBL3542352 0.06 0.047 CHEMBL3988902 | CHEMBL3988903 | |
| 0.039 | 0.005 | 0.06 | HCV NS5A inhibitor | 0.048 0.004 CHEMBL3526717 0.036 0.008 CHEMBL3526718 0.06 0.004 CHEMBL3526892 0.055 0.004 CHEMBL3988903 0.036 0.008 CHEMBL3526789 0.036 0.008 CHEMBL3526788 0.046 0.004 CHEMBL3526896 0.037 0.007 CHEMBL3526787 0.036 0.008 CHEMBL3526719 | CHEMBL3526892 | |
| 0.05 | 0.023 | 0.121 | Cathepsin L2 inhibitor | 0.092 0.009 CHEMBL3526717 0.035 0.032 CHEMBL3526718 0.037 0.031 CHEMBL3526892 0.121 0.006 CHEMBL3988903 0.037 0.031 CHEMBL3526789 0.037 0.031 CHEMBL3526788 0.083 0.01 CHEMBL3526896 0.039 0.029 CHEMBL3526787 | CHEMBL3988903 | |
| 0.036 | 0.01 | 0.038 | Neutral endopeptidase inhibitor | 0.034 0.01 CHEMBL3526718 0.028 0.012 CHEMBL3526789 0.028 0.012 CHEMBL3526788 0.023 0.014 CHEMBL3988901 0.038 0.01 CHEMBL3526787 0.036 0.01 CHEMBL3526719 0.024 0.014 CHEMBL3988902 | CHEMBL3526787 | |
| 0.057 | 0.032 | 0.084 | Immunoglobulin Fc receptor antagonist | 0.07 0.011 CHEMBL3526717 0.056 0.036 CHEMBL3542349 0.084 0.005 CHEMBL3988903 0.053 0.047 CHEMBL3526789 0.053 0.047 CHEMBL3526788 0.065 0.016 CHEMBL3526896 0.064 0.017 CHEMBL3542350 0.064 0.017 CHEMBL3542351 0.054 0.044 CHEMBL3988901 0.073 0.009 CHEMBL3988902 | CHEMBL3988903 | |
| 0.086 | 0.063 | 0.136 | Falcipain 2 inhibitor | 0.136 0.035 CHEMBL3526717 0.134 0.036 CHEMBL3542349 0.127 0.039 CHEMBL3526892 0.119 0.043 CHEMBL3988903 0.085 0.064 CHEMBL3526896 | CHEMBL3526717 | |
| 0.037 | 0.017 | 0.049 | HCV polyprotein inhibitor | 0.044 0.008 CHEMBL3526717 0.034 0.023 CHEMBL3526718 0.04 0.012 CHEMBL3526892 0.049 0.005 CHEMBL3988903 0.035 0.021 CHEMBL3526789 0.035 0.021 CHEMBL3526788 0.043 0.009 CHEMBL3526896 0.035 0.021 CHEMBL3526787 | CHEMBL3988903 | |
| 0.024 | 0.011 | 0.062 | Human T-cell leukemia virus type I protease inhibitor | 0.048 0.004 CHEMBL3526717 0.02 0.015 CHEMBL3526718 0.062 0.004 CHEMBL3988903 0.023 0.013 CHEMBL3526789 0.023 0.013 CHEMBL3526788 0.045 0.004 CHEMBL3526896 0.021 0.014 CHEMBL3526787 | CHEMBL3988903 | |
| 0.044 | 0.034 | 0.081 | Endothelin-converting enzyme inhibitor | 0.072 0.02 CHEMBL3526717 0.049 0.031 CHEMBL3526892 0.081 0.017 CHEMBL3988903 0.04 0.038 CHEMBL3526789 0.04 0.038 CHEMBL3526788 0.063 0.023 CHEMBL3526896 0.054 0.028 CHEMBL3988901 0.046 0.033 CHEMBL3988902 | CHEMBL3988903 | |
| 0.124 | 0.115 | 0.299 | Growth hormone agonist | 0.191 0.062 CHEMBL3526717 0.203 0.058 CHEMBL3988903 0.149 0.088 CHEMBL3526789 0.149 0.088 CHEMBL3526788 0.18 0.068 CHEMBL3526896 0.299 0.032 CHEMBL3988901 0.123 0.116 CHEMBL3526787 0.123 0.116 CHEMBL3526719 0.163 0.077 CHEMBL3988902 | CHEMBL3988901 | |
| 0.026 | 0.019 | 0.063 | Cathepsin K inhibitor | 0.059 0.007 CHEMBL3526717 0.049 0.008 CHEMBL3526892 0.063 0.007 CHEMBL3988903 0.025 0.021 CHEMBL3526896 | CHEMBL3988903 | |
| 0.044 | 0.038 | 0.047 | Baculoviral IAP repeat-containing protein inhibitor | 0.047 0.028 CHEMBL3526717 0.045 0.036 CHEMBL3526892 0.047 0.03 CHEMBL3988903 0.044 0.04 CHEMBL3526789 0.044 0.04 CHEMBL3526788 | CHEMBL3988903 | |
| 0.031 | 0.029 | 0.123 | Calpain 1 inhibitor | 0.037 0.015 CHEMBL3526717 0.034 0.021 CHEMBL3526892 0.123 0.004 CHEMBL3988903 0.036 0.017 CHEMBL3526896 | CHEMBL3988903 | |
| 0.02 | 0.018 | 0.053 | Elastase 2 inhibitor | 0.031 0.009 CHEMBL3526717 0.032 0.009 CHEMBL3526892 0.053 0.005 CHEMBL3988903 0.028 0.01 CHEMBL3526896 | CHEMBL3988903 | |
| 0.02 | 0.018 | 0.053 | Elastase 2A inhibitor | 0.031 0.009 CHEMBL3526717 0.032 0.009 CHEMBL3526892 0.053 0.005 CHEMBL3988903 0.028 0.01 CHEMBL3526896 | CHEMBL3988903 | |
| 0.111 | 0.112 | 0.158 | Neurotrophic factor | 0.158 0.052 CHEMBL3542349 0.119 0.097 CHEMBL3542351 0.141 0.068 CHEMBL3988902 | CHEMBL3542349 | |
| 0.032 | 0.033 | 0.038 | Bombesin 1 receptor antagonist | 0.034 0.029 CHEMBL3526717 0.038 0.025 CHEMBL3988903 0.033 0.031 CHEMBL3526896 | CHEMBL3988903 | |
| 0.05 | 0.053 | 0.061 | Kallikrein 1 inhibitor | 0.061 0.033 CHEMBL3988903 0.053 0.046 CHEMBL3526789 0.053 0.046 CHEMBL3526788 0.054 0.044 CHEMBL3526896 | CHEMBL3988903 | |
| 0.037 | 0.043 | 0.074 | Neurotensin receptor antagonist | 0.074 0.019 CHEMBL3526717 0.055 0.026 CHEMBL3988903 0.047 0.03 CHEMBL3526896 0.043 0.033 CHEMBL3988901 | CHEMBL3526717 | |
| 0.135 | 0.141 | 0.138 | P-glycoprotein inhibitor | 0.138 0.136 CHEMBL3526787 | CHEMBL3526787 | |
| 0.065 | 0.074 | 0.086 | Somatostatin 1 agonist | 0.072 0.061 CHEMBL3526717 0.077 0.055 CHEMBL3988903 0.076 0.055 CHEMBL3526789 0.076 0.055 CHEMBL3526788 0.069 0.066 CHEMBL3526896 0.086 0.045 CHEMBL3988901 | CHEMBL3988901 | |
| 0.049 | 0.058 | 0.084 | Bombesin 1 receptor agonist | 0.084 0.023 CHEMBL3988901 | CHEMBL3988901 | |
| 0.045 | 0.057 | 0.14 | Cathepsin L inhibitor | 0.113 0.018 CHEMBL3526717 0.069 0.03 CHEMBL3526892 0.14 0.015 CHEMBL3988903 0.065 0.034 CHEMBL3526896 0.065 0.034 CHEMBL3988901 | CHEMBL3988903 | |
| 0.039 | 0.054 | 0.046 | Bombesin antagonist | 0.044 0.04 CHEMBL3988903 0.046 0.035 CHEMBL3988901 | CHEMBL3988901 | |
| 0.055 | 0.071 | 0.108 | Elastase 1 inhibitor | 0.072 0.044 CHEMBL3526717 0.061 0.06 CHEMBL3526892 0.108 0.016 CHEMBL3988903 0.068 0.05 CHEMBL3526896 | CHEMBL3988903 | |
| 0.132 | 0.152 | 0.234 | Neurotensin receptor agonist | 0.167 0.066 CHEMBL3526717 0.151 0.099 CHEMBL3542349 0.148 0.107 CHEMBL3526892 0.182 0.048 CHEMBL3988903 0.139 0.132 CHEMBL3526789 0.139 0.132 CHEMBL3526788 0.157 0.086 CHEMBL3526896 0.151 0.098 CHEMBL3542350 0.2 0.035 CHEMBL3542351 0.234 0.024 CHEMBL3988901 0.198 0.036 CHEMBL3542352 0.215 0.029 CHEMBL3988902 | CHEMBL3988901 | |
| 0.044 | 0.063 | 0.049 | Bombesin 3 receptor antagonist | 0.049 0.048 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.03 | 0.018 | KiSS-1 receptor antagonist | 0.018 0.011 CHEMBL3526717 | CHEMBL3526717 | |
| 0.032 | 0.055 | 0.074 | Plasmin inhibitor | 0.074 0.023 CHEMBL3988903 | CHEMBL3988903 | |
| 0.071 | 0.095 | 0.106 | Transcription factor NF kappa B stimulant | 0.091 0.049 CHEMBL3526717 0.091 0.049 CHEMBL3988903 0.088 0.054 CHEMBL3526896 0.106 0.033 CHEMBL3988901 0.078 0.074 CHEMBL3988902 | CHEMBL3988901 | |
| 0.025 | 0.05 | 0.034 | Factor XI inhibitor | 0.034 0.024 CHEMBL3526892 0.032 0.027 CHEMBL3988903 0.032 0.028 CHEMBL3542351 | CHEMBL3526892 | |
| 0.007 | 0.032 | 0.02 | 3C-Like protease (MERS coronavirus) inhibitor | 0.02 0.004 CHEMBL3988903 | CHEMBL3988903 | |
| 0.218 | 0.245 | 0.449 | Calcium channel L-type activator | 0.305 0.153 CHEMBL3526717 0.244 0.212 CHEMBL3526892 0.339 0.126 CHEMBL3988903 0.288 0.168 CHEMBL3526896 0.449 0.051 CHEMBL3542351 0.335 0.129 CHEMBL3542352 | CHEMBL3542351 | |
| 0.032 | 0.061 | 0.051 | Neuropeptide agonist | 0.051 0.042 CHEMBL3988901 | CHEMBL3988901 | |
| 0.032 | 0.062 | 0.057 | Kallikrein inhibitor | 0.057 0.025 CHEMBL3988903 | CHEMBL3988903 | |
| 0.017 | 0.053 | 0.05 | Cholecystokinin A antagonist | 0.05 0.019 CHEMBL3526717 0.037 0.027 CHEMBL3988901 | CHEMBL3526717 | |
| 0.035 | 0.072 | 0.048 | Collagenase inhibitor | 0.046 0.041 CHEMBL3988903 0.048 0.037 CHEMBL3988901 0.047 0.04 CHEMBL3988902 | CHEMBL3988901 | |
| 0.048 | 0.088 | 0.086 | Sirtuin 1 inhibitor | 0.065 0.051 CHEMBL3526717 0.073 0.042 CHEMBL3988903 0.061 0.057 CHEMBL3526896 0.086 0.031 CHEMBL3988901 0.077 0.038 CHEMBL3988902 | CHEMBL3988901 | |
| 0.046 | 0.089 | 0.056 | Gonadotropin-releasing hormone receptor agonist | 0.054 0.053 CHEMBL3988901 0.056 0.048 CHEMBL3542352 | CHEMBL3542352 | |
| 0.025 | 0.068 | 0.04 | Growth hormone release inhibitor | 0.04 0.032 CHEMBL3988901 | CHEMBL3988901 | |
| 0.05 | 0.095 | 0.06 | Trypsin inhibitor | 0.06 0.047 CHEMBL3988903 0.059 0.05 CHEMBL3988901 | CHEMBL3988903 | |
| 0.031 | 0.078 | 0.05 | Cathepsin F inhibitor | 0.05 0.012 CHEMBL3988901 | CHEMBL3988901 | |
| 0.015 | 0.063 | 0.044 | Cholecystokinin antagonist | 0.044 0.027 CHEMBL3526717 0.042 0.029 CHEMBL3988901 | CHEMBL3526717 | |
| 0.067 | 0.116 | 0.231 | Falcipain 3 inhibitor | 0.207 0.016 CHEMBL3526717 0.231 0.01 CHEMBL3988903 0.16 0.032 CHEMBL3526896 0.091 0.08 CHEMBL3542351 0.094 0.077 CHEMBL3542352 | CHEMBL3988903 | |
| 0.01 | 0.061 | 0.027 | Cholecystokinin B antagonist | 0.027 0.025 CHEMBL3988901 | CHEMBL3988901 | |
| 0.008 | 0.06 | 0.019 | Cathepsin S inhibitor | 0.019 0.014 CHEMBL3988903 | CHEMBL3988903 | |
| 0.022 | 0.077 | 0.046 | Cholecystokinin B agonist | 0.046 0.018 CHEMBL3988901 | CHEMBL3988901 | |
| 0.029 | 0.083 | 0.049 | Microtubule stabilization | 0.049 0.029 CHEMBL3988903 | CHEMBL3988903 | |
| 0.05 | 0.106 | 0.085 | Secretase beta inhibitor | 0.085 0.031 CHEMBL3526717 0.067 0.054 CHEMBL3526896 | CHEMBL3526717 | |
| 0.035 | 0.096 | 0.061 | Carbonic anhydrase II stimulant | 0.061 0.022 CHEMBL3988901 | CHEMBL3988901 | |
| 0.016 | 0.077 | 0.064 | Cathepsin L1 inhibitor | 0.058 0.016 CHEMBL3526717 0.041 0.026 CHEMBL3526892 0.064 0.015 CHEMBL3988903 | CHEMBL3988903 | |
| 0.022 | 0.085 | 0.049 | Factor XIa inhibitor | 0.049 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.089 | 0.087 | Beta tubulin antagonist | 0.049 0.047 CHEMBL3526892 0.087 0.027 CHEMBL3988903 | CHEMBL3988903 | |
| 0.067 | 0.131 | 0.275 | Hematopoietic | 0.103 0.033 CHEMBL3542351 0.275 0.005 CHEMBL3988901 0.119 0.022 CHEMBL3542352 0.116 0.024 CHEMBL3988902 | CHEMBL3988901 | |
| 0.072 | 0.138 | 0.107 | Nav1.4 sodium channel blocker | 0.107 0.065 CHEMBL3988901 | CHEMBL3988901 | |
| 0.025 | 0.092 | 0.042 | Neurokinin 2 agonist | 0.042 0.027 CHEMBL3988901 | CHEMBL3988901 | |
| 0.038 | 0.107 | 0.093 | Angiotensin-converting enzyme inhibitor | 0.085 0.012 CHEMBL3988901 0.093 0.01 CHEMBL3988902 | CHEMBL3988902 | |
| 0.032 | 0.102 | 0.086 | HCV NS3/NS4A protease inhibitor | 0.058 0.022 CHEMBL3526717 0.046 0.039 CHEMBL3526892 0.086 0.008 CHEMBL3988903 0.052 0.029 CHEMBL3526896 | CHEMBL3988903 | |
| 0.013 | 0.083 | 0.031 | Caspase 2 inhibitor | 0.031 0.022 CHEMBL3988903 0.029 0.025 CHEMBL3988902 | CHEMBL3988903 | |
| 0.074 | 0.147 | 0.206 | Bone formation stimulant | 0.129 0.077 CHEMBL3526717 0.206 0.034 CHEMBL3988903 0.114 0.091 CHEMBL3526896 0.135 0.072 CHEMBL3988901 0.117 0.088 CHEMBL3542352 | CHEMBL3988903 | |
| 0.021 | 0.094 | 0.086 | Ribonucleoside-diphosphate reductase inhibitor | 0.062 0.033 CHEMBL3526717 0.082 0.024 CHEMBL3988903 0.073 0.028 CHEMBL3526896 0.086 0.023 CHEMBL3988901 0.048 0.042 CHEMBL3542352 | CHEMBL3988901 | |
| 0.019 | 0.097 | 0.085 | Ribonucleotide reductase inhibitor | 0.064 0.034 CHEMBL3526717 0.083 0.025 CHEMBL3988903 0.074 0.029 CHEMBL3526896 0.085 0.025 CHEMBL3988901 0.049 0.043 CHEMBL3542352 | CHEMBL3988901 | |
| 0.011 | 0.091 | 0.034 | Caspase 8 inhibitor | 0.023 0.009 CHEMBL3988903 0.023 0.009 CHEMBL3988901 0.034 0.004 CHEMBL3988902 | CHEMBL3988902 | |
| 0.013 | 0.094 | 0.036 | Granulocyte colony stimulating factor receptor agonist | 0.036 0.003 CHEMBL3542349 0.018 0.014 CHEMBL3542350 0.023 0.005 CHEMBL3542351 0.018 0.017 CHEMBL3988901 0.02 0.009 CHEMBL3542352 | CHEMBL3542349 | |
| 0.086 | 0.169 | 0.254 | Anticoagulant | 0.15 0.081 CHEMBL3988903 0.254 0.038 CHEMBL3988901 0.165 0.069 CHEMBL3542352 0.136 0.093 CHEMBL3988902 | CHEMBL3988901 | |
| 0.162 | 0.246 | 0.433 | Sodium/bile acid cotransporter inhibitor | 0.312 0.069 CHEMBL3542351 0.406 0.015 CHEMBL3988901 0.433 0.01 CHEMBL3542352 0.206 0.18 CHEMBL3988902 | CHEMBL3542352 | |
| 0.08 | 0.166 | 0.195 | Histone deacetylase SIRT1 inhibitor | 0.119 0.093 CHEMBL3988903 0.195 0.032 CHEMBL3988901 0.146 0.065 CHEMBL3542352 0.166 0.049 CHEMBL3988902 | CHEMBL3988901 | |
| 0.009 | 0.094 | 0.03 | Bombesin 3 receptor agonist | 0.03 0.006 CHEMBL3526892 0.02 0.011 CHEMBL3542351 | CHEMBL3526892 | |
| 0.118 | 0.206 | 0.192 | Catenin beta inhibitor | 0.153 0.099 CHEMBL3526892 0.192 0.038 CHEMBL3542351 0.149 0.107 CHEMBL3542352 0.14 0.132 CHEMBL3988902 | CHEMBL3542351 | |
| 0.027 | 0.116 | 0.078 | Aminopeptidase microsomal inhibitor | 0.078 0.026 CHEMBL3988901 | CHEMBL3988901 | |
| 0.087 | 0.175 | 0.351 | Angiogenesis stimulant | 0.162 0.115 CHEMBL3526717 0.213 0.088 CHEMBL3988903 0.145 0.126 CHEMBL3526896 0.351 0.032 CHEMBL3988901 0.174 0.108 CHEMBL3542352 0.286 0.055 CHEMBL3988902 | CHEMBL3988901 | |
| 0.009 | 0.098 | 0.035 | Bombesin agonist | 0.035 0.006 CHEMBL3526892 0.025 0.012 CHEMBL3542351 | CHEMBL3526892 | |
| 0.018 | 0.113 | 0.056 | Aminopeptidase N inhibitor | 0.056 0.026 CHEMBL3988901 | CHEMBL3988901 | |
| 0.009 | 0.105 | 0.023 | Integrin alphaVbeta3 antagonist | 0.023 0.013 CHEMBL3542352 | CHEMBL3542352 | |
| 0.027 | 0.124 | 0.094 | Glucagon-like peptide 1 agonist | 0.094 0.026 CHEMBL3988901 | CHEMBL3988901 | |
| 0.04 | 0.137 | 0.079 | Thrombin inhibitor | 0.066 0.061 CHEMBL3988903 0.079 0.043 CHEMBL3988901 | CHEMBL3988901 | |
| 0.001 | 0.099 | 0.01 | Mannitol 2-dehydrogenase inhibitor | 0.01 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.123 | 0.062 | Elastase inhibitor | 0.062 0.028 CHEMBL3988903 | CHEMBL3988903 | |
| 0.024 | 0.125 | 0.147 | Maillard reaction inhibitor | 0.147 0.006 CHEMBL3526896 | CHEMBL3526896 | |
| 0.02 | 0.13 | 0.077 | Plasminogen activator inhibitor | 0.077 0.027 CHEMBL3988903 | CHEMBL3988903 | |
| 0.012 | 0.127 | 0.054 | Peptide deformylase inhibitor | 0.028 0.024 CHEMBL3526717 0.032 0.019 CHEMBL3988903 0.054 0.009 CHEMBL3526896 0.031 0.02 CHEMBL3988901 | CHEMBL3526896 | |
| 0.158 | 0.275 | 0.311 | Interleukin 2 agonist | 0.231 0.141 CHEMBL3526717 0.247 0.122 CHEMBL3988903 0.197 0.194 CHEMBL3526789 0.197 0.194 CHEMBL3526788 0.222 0.154 CHEMBL3526896 0.311 0.066 CHEMBL3988901 0.296 0.077 CHEMBL3988902 | CHEMBL3988901 | |
| 0.008 | 0.134 | 0.019 | Integrin alphaVbeta1 antagonist | 0.019 0.013 CHEMBL3542352 | CHEMBL3542352 | |
| 0.016 | 0.146 | 0.07 | Metalloproteinase-3 inhibitor | 0.043 0.042 CHEMBL3526717 0.068 0.02 CHEMBL3988903 0.07 0.019 CHEMBL3988901 0.058 0.025 CHEMBL3988902 | CHEMBL3988901 | |
| 0.008 | 0.139 | 0.047 | Prostacyclin antagonist | 0.032 0.024 CHEMBL3542352 0.047 0.014 CHEMBL3988902 | CHEMBL3988902 | |
| 0.023 | 0.155 | 0.068 | Matrix metalloproteinase (membrane-type) inhibitor | 0.058 0.035 CHEMBL3526717 0.067 0.026 CHEMBL3988903 0.065 0.028 CHEMBL3526896 0.068 0.026 CHEMBL3988901 0.057 0.036 CHEMBL3988902 | CHEMBL3988901 | |
| 0.015 | 0.149 | 0.047 | Factor XIIIa inhibitor | 0.047 0.018 CHEMBL3526896 | CHEMBL3526896 | |
| 0.067 | 0.201 | 0.155 | Folate antagonist | 0.094 0.076 CHEMBL3542351 0.131 0.031 CHEMBL3988901 0.155 0.02 CHEMBL3542352 0.107 0.053 CHEMBL3988902 | CHEMBL3542352 | |
| 0.004 | 0.14 | 0.021 | Integrin alpha4 antagonist | 0.021 0.02 CHEMBL3988902 | CHEMBL3988902 | |
| 0.008 | 0.151 | 0.056 | Complement C3a chemotactic receptor antagonist | 0.056 0.024 CHEMBL3988901 0.04 0.032 CHEMBL3988902 | CHEMBL3988901 | |
| 0.009 | 0.152 | 0.197 | Methionyl aminopeptidase 1 inhibitor | 0.149 0.003 CHEMBL3542349 0.03 0.025 CHEMBL3526892 0.033 0.02 CHEMBL3542350 0.1 0.004 CHEMBL3542351 0.16 0.003 CHEMBL3988901 0.044 0.009 CHEMBL3542352 0.197 0.003 CHEMBL3988902 | CHEMBL3988902 | |
| 0.059 | 0.202 | 0.256 | Microtubule formation inhibitor | 0.17 0.029 CHEMBL3526717 0.256 0.007 CHEMBL3988903 0.152 0.037 CHEMBL3526896 0.104 0.083 CHEMBL3542351 | CHEMBL3988903 | |
| 0.056 | 0.204 | 0.257 | Caspase 3 inhibitor | 0.114 0.07 CHEMBL3526717 0.165 0.019 CHEMBL3988903 0.119 0.062 CHEMBL3542351 0.211 0.008 CHEMBL3988901 0.126 0.051 CHEMBL3542352 0.257 0.005 CHEMBL3988902 | CHEMBL3988902 | |
| 0.005 | 0.154 | 0.055 | GP IIb/IIIa receptor antagonist | 0.055 0.03 CHEMBL3988901 0.044 0.038 CHEMBL3542352 | CHEMBL3988901 | |
| 0.016 | 0.167 | 0.135 | Neutrophil collagenase inhibitor | 0.08 0.032 CHEMBL3988903 0.062 0.048 CHEMBL3526896 0.135 0.014 CHEMBL3988901 0.071 0.038 CHEMBL3988902 | CHEMBL3988901 | |
| 0.021 | 0.177 | 0.092 | Selectin antagonist | 0.092 0.031 CHEMBL3988901 | CHEMBL3988901 | |
| 0.012 | 0.178 | 0.053 | Carbonic anhydrase I stimulant | 0.053 0.015 CHEMBL3988901 | CHEMBL3988901 | |
| 0.15 | 0.316 | 0.22 | Ca(v)3.3 blocker | 0.22 0.152 CHEMBL3526892 0.212 0.166 CHEMBL3542352 | CHEMBL3526892 | |
| 0.009 | 0.175 | 0.039 | Integrin antagonist | 0.039 0.032 CHEMBL3542352 | CHEMBL3542352 | |
| 0.009 | 0.179 | 0.019 | Tryptophan hydroxylase 1 inhibitor | 0.019 0.008 CHEMBL3542352 | CHEMBL3542352 | |
| 0.012 | 0.185 | 0.183 | Toll-Like receptor 2 agonist | 0.183 0.008 CHEMBL3988901 0.035 0.034 CHEMBL3542352 0.072 0.018 CHEMBL3988902 | CHEMBL3988901 | |
| 0.017 | 0.192 | 0.077 | Lysophosphatidic acid 3 receptor antagonist | 0.061 0.022 CHEMBL3988903 0.073 0.013 CHEMBL3542351 0.073 0.013 CHEMBL3988901 0.077 0.011 CHEMBL3988902 | CHEMBL3988902 | |
| 0.041 | 0.217 | 0.091 | ATPase (Vacuolar H+) inhibitor | 0.091 0.054 CHEMBL3542350 | CHEMBL3542350 | |
| 0.021 | 0.204 | 0.117 | Matrix metalloproteinase inhibitor | 0.058 0.057 CHEMBL3526717 0.096 0.028 CHEMBL3988903 0.067 0.047 CHEMBL3526896 0.117 0.02 CHEMBL3988901 0.079 0.037 CHEMBL3988902 | CHEMBL3988901 | |
| 0.069 | 0.253 | 0.152 | Amyloid beta precursor protein antagonist | 0.142 0.111 CHEMBL3988903 0.152 0.099 CHEMBL3526896 0.135 0.119 CHEMBL3542351 | CHEMBL3526896 | |
| 0.027 | 0.211 | 0.094 | Prostaglandin F2 alpha antagonist | 0.094 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.027 | 0.212 | 0.198 | Aminopeptidase I inhibitor | 0.066 0.059 CHEMBL3526717 0.08 0.042 CHEMBL3542349 0.075 0.047 CHEMBL3988903 0.173 0.009 CHEMBL3542351 0.198 0.007 CHEMBL3988901 0.15 0.012 CHEMBL3542352 0.124 0.018 CHEMBL3988902 | CHEMBL3988901 | |
| 0.043 | 0.233 | 0.111 | Factor XII inhibitor | 0.111 0.029 CHEMBL3988901 0.084 0.059 CHEMBL3988902 | CHEMBL3988901 | |
| 0.007 | 0.202 | 0.037 | Lysophosphatidic acid 1 receptor antagonist | 0.037 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.206 | 0.027 | Lysophosphatidic acid receptor 1 agonist | 0.027 0.015 CHEMBL3988903 | CHEMBL3988903 | |
| 0.014 | 0.212 | 0.06 | Neuraminidase inhibitor | 0.06 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.101 | 0.301 | 0.182 | Cyclin-dependent kinase 3 inhibitor | 0.174 0.055 CHEMBL3542349 0.137 0.132 CHEMBL3526718 0.151 0.094 CHEMBL3542350 0.182 0.046 CHEMBL3542351 0.141 0.12 CHEMBL3526787 0.141 0.12 CHEMBL3526719 0.182 0.046 CHEMBL3542352 | CHEMBL3542352 | |
| 0.009 | 0.21 | 0.071 | Matrix metalloproteinase 1 inhibitor | 0.071 0.025 CHEMBL3988903 0.062 0.03 CHEMBL3988901 | CHEMBL3988903 | |
| 0.117 | 0.32 | 0.274 | Peptidyltransferase inhibitor | 0.165 0.157 CHEMBL3526717 0.177 0.134 CHEMBL3988903 0.265 0.041 CHEMBL3988901 0.272 0.037 CHEMBL3542352 0.274 0.036 CHEMBL3988902 | CHEMBL3988902 | |
| 0.025 | 0.231 | 0.074 | Topoisomerase II alpha inhibitor | 0.068 0.064 CHEMBL3542349 0.066 0.065 CHEMBL3542351 0.074 0.058 CHEMBL3542352 | CHEMBL3542352 | |
| 0.008 | 0.214 | 0.029 | Bradykinin B2 receptor agonist | 0.029 0.019 CHEMBL3988901 | CHEMBL3988901 | |
| 0.016 | 0.223 | 0.051 | Neuraminidase (Influenza A) inhibitor | 0.051 0.022 CHEMBL3542351 | CHEMBL3542351 | |
| 0.011 | 0.219 | 0.046 | Integrin alpha5beta1 antagonist | 0.044 0.024 CHEMBL3988901 0.046 0.022 CHEMBL3542352 | CHEMBL3542352 | |
| 0.082 | 0.291 | 0.171 | Vasodilator | 0.171 0.131 CHEMBL3988902 | CHEMBL3988902 | |
| 0.055 | 0.266 | 0.157 | Cell adhesion inhibitor | 0.098 0.093 CHEMBL3542351 0.157 0.042 CHEMBL3542352 0.109 0.075 CHEMBL3988902 | CHEMBL3542352 | |
| 0.021 | 0.234 | 0.068 | Neuraminidase (influenza) inhibitor | 0.068 0.038 CHEMBL3542351 | CHEMBL3542351 | |
| 0.118 | 0.335 | 0.397 | Insulysin inhibitor | 0.249 0.097 CHEMBL3542349 0.21 0.143 CHEMBL3988903 0.234 0.112 CHEMBL3542350 0.364 0.03 CHEMBL3542351 0.397 0.022 CHEMBL3988901 0.373 0.027 CHEMBL3542352 0.322 0.046 CHEMBL3988902 | CHEMBL3988901 | |
| 0.109 | 0.327 | 0.366 | Antithrombotic | 0.193 0.186 CHEMBL3526717 0.366 0.059 CHEMBL3988903 0.262 0.117 CHEMBL3526896 0.306 0.084 CHEMBL3542351 0.277 0.105 CHEMBL3988901 0.348 0.065 CHEMBL3542352 | CHEMBL3988903 | |
| 0.127 | 0.348 | 0.352 | Caspase 3 stimulant | 0.329 0.066 CHEMBL3542349 0.201 0.168 CHEMBL3988903 0.352 0.058 CHEMBL3542350 0.232 0.129 CHEMBL3542351 | CHEMBL3542350 | |
| 0.041 | 0.265 | 0.174 | Histone deacetylase class III inhibitor | 0.174 0.029 CHEMBL3988901 0.111 0.078 CHEMBL3542352 0.155 0.04 CHEMBL3988902 | CHEMBL3988901 | |
| 0.038 | 0.265 | 0.305 | Chelator | 0.151 0.035 CHEMBL3542351 0.236 0.018 CHEMBL3988901 0.305 0.01 CHEMBL3542352 0.129 0.046 CHEMBL3988902 | CHEMBL3542352 | |
| 0.025 | 0.253 | 0.129 | Metalloproteinase-9 inhibitor | 0.072 0.052 CHEMBL3988903 0.067 0.061 CHEMBL3526896 0.129 0.022 CHEMBL3988901 0.096 0.034 CHEMBL3988902 | CHEMBL3988901 | |
| 0.024 | 0.257 | 0.13 | Metalloproteinase-2 inhibitor | 0.072 0.062 CHEMBL3526717 0.13 0.025 CHEMBL3988903 0.07 0.066 CHEMBL3526896 0.123 0.028 CHEMBL3988901 0.09 0.044 CHEMBL3988902 | CHEMBL3988903 | |
| 0.018 | 0.251 | 0.043 | VCAM-1 antagonist | 0.04 0.027 CHEMBL3988901 0.039 0.028 CHEMBL3542352 0.043 0.018 CHEMBL3988902 | CHEMBL3988902 | |
| 0.018 | 0.251 | 0.043 | VCAM antagonist | 0.039 0.027 CHEMBL3988901 0.039 0.028 CHEMBL3542352 0.043 0.018 CHEMBL3988902 | CHEMBL3988902 | |
| 0.054 | 0.289 | 0.763 | Peroxidase inhibitor | 0.483 0.011 CHEMBL3542349 0.315 0.034 CHEMBL3542350 0.657 0.004 CHEMBL3542351 0.763 0.002 CHEMBL3988901 0.681 0.003 CHEMBL3542352 0.444 0.015 CHEMBL3988902 | CHEMBL3988901 | |
| 0.021 | 0.258 | 0.038 | Glucagon-like peptide 1 receptor antagonist | 0.038 0.031 CHEMBL3542352 | CHEMBL3542352 | |
| 0.103 | 0.346 | 0.446 | Vasodilator, peripheral | 0.208 0.167 CHEMBL3526717 0.277 0.109 CHEMBL3988903 0.324 0.085 CHEMBL3526896 0.446 0.042 CHEMBL3542351 | CHEMBL3542351 | |
| 0.036 | 0.281 | 0.102 | Cell adhesion molecule inhibitor | 0.102 0.033 CHEMBL3542352 | CHEMBL3542352 | |
| 0.034 | 0.28 | 0.122 | Tubulin antagonist | 0.122 0.078 CHEMBL3542349 | CHEMBL3542349 | |
| 0.017 | 0.265 | 0.049 | Farnesyltransferase inhibitor | 0.048 0.03 CHEMBL3988901 0.049 0.028 CHEMBL3988902 | CHEMBL3988902 | |
| 0.004 | 0.255 | 0.039 | Somatostatin 5 antagonist | 0.039 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.038 | 0.289 | 0.318 | Thrombolytic | 0.134 0.095 CHEMBL3542351 0.318 0.021 CHEMBL3988901 0.199 0.053 CHEMBL3542352 0.201 0.052 CHEMBL3988902 | CHEMBL3988901 | |
| 0.008 | 0.262 | 0.086 | NMDA 2D receptor antagonist | 0.086 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.032 | 0.288 | 0.099 | Sphingomyelinase inhibitor | 0.099 0.06 CHEMBL3988903 | CHEMBL3988903 | |
| 0.06 | 0.318 | 0.499 | Immunostimulant | 0.157 0.149 CHEMBL3542349 0.287 0.082 CHEMBL3988903 0.229 0.105 CHEMBL3526896 0.499 0.029 CHEMBL3988901 0.204 0.118 CHEMBL3542352 0.352 0.064 CHEMBL3988902 | CHEMBL3988901 | |
| 0.01 | 0.269 | 0.063 | Leukocyte elastase inhibitor | 0.038 0.037 CHEMBL3526892 0.063 0.017 CHEMBL3988903 0.04 0.033 CHEMBL3542351 | CHEMBL3988903 | |
| 0.018 | 0.279 | 0.108 | Carbonic anhydrase stimulant | 0.108 0.017 CHEMBL3988901 0.078 0.026 CHEMBL3542352 0.058 0.042 CHEMBL3988902 | CHEMBL3988901 | |
| 0.046 | 0.307 | 0.317 | Toll-Like receptor 2 antagonist | 0.172 0.038 CHEMBL3542349 0.137 0.062 CHEMBL3988903 0.131 0.067 CHEMBL3542351 0.317 0.004 CHEMBL3988901 0.166 0.042 CHEMBL3542352 0.277 0.006 CHEMBL3988902 | CHEMBL3988901 | |
| 0.021 | 0.282 | 0.201 | Botulinum neurotoxin type A inhibitor | 0.201 0.004 CHEMBL3542349 0.059 0.038 CHEMBL3542350 0.088 0.013 CHEMBL3542351 0.092 0.011 CHEMBL3988901 0.106 0.008 CHEMBL3542352 0.074 0.021 CHEMBL3988902 | CHEMBL3542349 | |
| 0.033 | 0.303 | 0.145 | Aminoacyl-tRNA synthetase inhibitor | 0.088 0.061 CHEMBL3542351 0.145 0.02 CHEMBL3988901 0.089 0.061 CHEMBL3542352 0.08 0.077 CHEMBL3988902 | CHEMBL3988901 | |
| 0.005 | 0.279 | 0.033 | Diamine oxidase inhibitor | 0.033 0.032 CHEMBL3542351 | CHEMBL3542351 | |
| 0.051 | 0.327 | 0.221 | Insulin sensitizer | 0.162 0.118 CHEMBL3526717 0.157 0.123 CHEMBL3542349 0.22 0.055 CHEMBL3988903 0.221 0.054 CHEMBL3542351 0.219 0.055 CHEMBL3988901 0.211 0.063 CHEMBL3542352 0.206 0.068 CHEMBL3988902 | CHEMBL3542351 | |
| 0.012 | 0.293 | 0.088 | Erythropoietin receptor agonist | 0.051 0.021 CHEMBL3988901 0.088 0.011 CHEMBL3542352 | CHEMBL3542352 | |
| 0.01 | 0.3 | 0.033 | Benzodiazepine receptor peripheral-type antagonist | 0.033 0.028 CHEMBL3542349 | CHEMBL3542349 | |
| 0.026 | 0.318 | 0.199 | Mediator release inhibitor | 0.199 0.015 CHEMBL3542351 0.111 0.057 CHEMBL3542352 | CHEMBL3542351 | |
| 0.05 | 0.344 | 0.473 | Interleukin antagonist | 0.142 0.124 CHEMBL3542351 0.473 0.022 CHEMBL3988901 0.329 0.042 CHEMBL3988902 | CHEMBL3988901 | |
| 0.017 | 0.323 | 0.073 | Guanylate cyclase stimulant | 0.073 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.026 | 0.332 | 0.134 | Alkylator | 0.123 0.065 CHEMBL3542349 0.134 0.056 CHEMBL3988903 0.101 0.087 CHEMBL3542351 0.112 0.075 CHEMBL3988901 0.121 0.067 CHEMBL3542352 | CHEMBL3988903 | |
| 0.016 | 0.329 | 0.077 | Nitric oxide donor | 0.077 0.025 CHEMBL3988901 0.06 0.049 CHEMBL3988902 | CHEMBL3988901 | |
| 0.127 | 0.449 | 0.272 | MAP kinase kinase 3 inhibitor | 0.272 0.016 CHEMBL3542349 0.235 0.049 CHEMBL3542350 0.259 0.024 CHEMBL3542351 0.25 0.032 CHEMBL3542352 | CHEMBL3542349 | |
| 0.016 | 0.345 | 0.065 | DNA gyrase subunit A inhibitor | 0.065 0.008 CHEMBL3988902 | CHEMBL3988902 | |
| 0.076 | 0.41 | 0.313 | Growth factor agonist | 0.313 0.013 CHEMBL3542349 0.234 0.039 CHEMBL3542350 0.24 0.036 CHEMBL3542351 0.25 0.031 CHEMBL3542352 0.151 0.139 CHEMBL3988902 | CHEMBL3542349 | |
| 0.029 | 0.366 | 0.193 | Protein-tyrosine phosphatase inhibitor | 0.193 0.05 CHEMBL3542351 0.141 0.088 CHEMBL3988901 0.177 0.058 CHEMBL3988902 | CHEMBL3542351 | |
| 0.008 | 0.345 | 0.054 | Angiotensin II receptor antagonist | 0.035 0.022 CHEMBL3542349 0.054 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.371 | 0.089 | Potassium channel large-conductance Ca-activated activator | 0.089 0.029 CHEMBL3542351 | CHEMBL3542351 | |
| 0.106 | 0.456 | 0.418 | Apoptosis agonist | 0.418 0.105 CHEMBL3542349 0.242 0.223 CHEMBL3988903 0.238 0.228 CHEMBL3542351 | CHEMBL3542349 | |
| 0.024 | 0.374 | 0.359 | Aminopeptidase B inhibitor | 0.099 0.066 CHEMBL3542349 0.131 0.047 CHEMBL3988903 0.216 0.018 CHEMBL3542351 0.359 0.005 CHEMBL3988901 0.193 0.023 CHEMBL3542352 0.173 0.029 CHEMBL3988902 | CHEMBL3988901 | |
| 0.037 | 0.387 | 0.141 | Activin receptor-like kinase 4 inhibitor | 0.141 0.034 CHEMBL3542349 0.131 0.041 CHEMBL3542350 0.134 0.039 CHEMBL3542351 0.121 0.051 CHEMBL3542352 | CHEMBL3542349 | |
| 0.019 | 0.37 | 0.208 | Cathepsin G inhibitor | 0.069 0.055 CHEMBL3526717 0.208 0.015 CHEMBL3988903 0.108 0.03 CHEMBL3526896 | CHEMBL3988903 | |
| 0.005 | 0.364 | 0.061 | Angiotensin AT1 receptor antagonist | 0.047 0.021 CHEMBL3542349 0.061 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.367 | 0.347 | Leukotriene A4 hydrolase inhibitor | 0.258 0.004 CHEMBL3988901 0.347 0.004 CHEMBL3988902 | CHEMBL3988902 | |
| 0.02 | 0.389 | 0.059 | Bombesin 2 receptor antagonist | 0.059 0.025 CHEMBL3988901 0.049 0.035 CHEMBL3542352 | CHEMBL3988901 | |
| 0.005 | 0.375 | 0.322 | Protocollagen prolyl hydroxylase inhibitor | 0.041 0.007 CHEMBL3542351 0.055 0.005 CHEMBL3988901 0.322 0.002 CHEMBL3542352 | CHEMBL3542352 | |
| 0.017 | 0.389 | 0.069 | Autotaxin inhibitor | 0.069 0.023 CHEMBL3542351 | CHEMBL3542351 | |
| 0.055 | 0.428 | 0.423 | Calpain 2 inhibitor | 0.252 0.148 CHEMBL3526717 0.263 0.14 CHEMBL3542349 0.423 0.049 CHEMBL3988903 0.353 0.085 CHEMBL3542350 0.324 0.1 CHEMBL3988901 0.381 0.071 CHEMBL3988902 | CHEMBL3988903 | |
| 0.012 | 0.386 | 0.143 | Protein-tyrosine phosphatase 1B inhibitor | 0.115 0.067 CHEMBL3542351 0.143 0.049 CHEMBL3988902 | CHEMBL3988902 | |
| 0.052 | 0.427 | 0.324 | 3C-like protease (Human coronavirus) inhibitor | 0.324 0.008 CHEMBL3542349 0.179 0.066 CHEMBL3988903 0.158 0.088 CHEMBL3542350 0.283 0.015 CHEMBL3542351 0.164 0.08 CHEMBL3542352 | CHEMBL3542349 | |
| 0.012 | 0.388 | 0.472 | Phenylalanine 4-hydroxylase inhibitor | 0.144 0.013 CHEMBL3542349 0.066 0.05 CHEMBL3542350 0.472 0.003 CHEMBL3542351 0.193 0.007 CHEMBL3988901 0.283 0.004 CHEMBL3542352 0.317 0.004 CHEMBL3988902 | CHEMBL3542351 | |
| 0.002 | 0.38 | 0.015 | Integrin alphaVbeta6 antagonist | 0.015 0.009 CHEMBL3542352 | CHEMBL3542352 | |
| 0.027 | 0.407 | 0.188 | Antineoplastic alkaloid | 0.188 0.017 CHEMBL3542349 0.081 0.064 CHEMBL3542351 | CHEMBL3542349 | |
| 0.056 | 0.443 | 0.116 | Vanilloid 1 agonist | 0.115 0.101 CHEMBL3988903 0.116 0.098 CHEMBL3988901 0.115 0.1 CHEMBL3542352 | CHEMBL3988901 | |
| 0.04 | 0.433 | 0.267 | Antiamyloidogenic | 0.18 0.114 CHEMBL3542349 0.267 0.064 CHEMBL3542351 0.182 0.112 CHEMBL3988901 0.196 0.102 CHEMBL3542352 | CHEMBL3542351 | |
| 0.037 | 0.431 | 0.323 | Platelet antagonist | 0.155 0.139 CHEMBL3542351 0.323 0.045 CHEMBL3988901 0.243 0.076 CHEMBL3542352 0.236 0.079 CHEMBL3988902 | CHEMBL3988901 | |
| 0.02 | 0.415 | 0.057 | Factor III inhibitor | 0.057 0.021 CHEMBL3542351 0.052 0.03 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.4 | 0.031 | AMPA 2 receptor antagonist | 0.031 0.019 CHEMBL3542351 0.029 0.021 CHEMBL3988901 | CHEMBL3542351 | |
| 0.037 | 0.432 | 0.159 | CDC-like kinase 3 inhibitor | 0.159 0.015 CHEMBL3542349 0.133 0.029 CHEMBL3542350 0.109 0.06 CHEMBL3542351 | CHEMBL3542349 | |
| 0.028 | 0.423 | 0.143 | Protein kinase (CK1) gamma 3 inhibitor | 0.143 0.098 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.412 | 0.153 | GABA aminotransferase inhibitor | 0.068 0.066 CHEMBL3526717 0.104 0.024 CHEMBL3542349 0.153 0.007 CHEMBL3526896 0.114 0.019 CHEMBL3542351 | CHEMBL3526896 | |
| 0.084 | 0.484 | 0.155 | CC chemokine 6 receptor antagonist | 0.123 0.1 CHEMBL3542349 0.155 0.016 CHEMBL3542351 | CHEMBL3542351 | |
| 0.022 | 0.427 | 0.071 | DNA helicase inhibitor | 0.05 0.049 CHEMBL3542351 0.071 0.016 CHEMBL3542352 0.064 0.023 CHEMBL3988902 | CHEMBL3542352 | |
| 0.004 | 0.415 | 0.025 | Leukotriene B4 receptor 1 antagonist | 0.025 0.022 CHEMBL3542351 | CHEMBL3542351 | |
| 0.008 | 0.42 | 0.052 | Prolyl endopeptidase inhibitor | 0.052 0.034 CHEMBL3542349 | CHEMBL3542349 | |
| 0.019 | 0.433 | 0.151 | Protein kinase C mu inhibitor | 0.151 0.025 CHEMBL3542349 0.095 0.062 CHEMBL3542351 0.121 0.041 CHEMBL3542352 | CHEMBL3542349 | |
| 0.02 | 0.436 | 0.069 | Histone deacetylase SIRT3 inhibitor | 0.069 0.029 CHEMBL3542352 | CHEMBL3542352 | |
| 0.018 | 0.437 | 0.101 | Transforming growth factor antagonist | 0.101 0.021 CHEMBL3542349 0.071 0.046 CHEMBL3542351 0.066 0.054 CHEMBL3542352 | CHEMBL3542349 | |
| 0.006 | 0.426 | 0.034 | Histone deacetylase 7 inhibitor | 0.034 0.029 CHEMBL3542352 | CHEMBL3542352 | |
| 0.002 | 0.422 | 0.031 | Retinoic acid beta receptor antagonist | 0.031 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.054 | 0.48 | 0.376 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.376 0.019 CHEMBL3542349 | CHEMBL3542349 | |
| 0.053 | 0.479 | 0.283 | Angiogenesis inhibitor | 0.283 0.102 CHEMBL3542349 0.217 0.151 CHEMBL3526892 0.261 0.115 CHEMBL3542350 | CHEMBL3542349 | |
| 0.004 | 0.431 | 0.034 | Kainate receptor 4 antagonist | 0.034 0.012 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.434 | 0.095 | Prostaglandin EP2 antagonist | 0.095 0.02 CHEMBL3542351 0.051 0.05 CHEMBL3542352 0.057 0.044 CHEMBL3988902 | CHEMBL3542351 | |
| 0.001 | 0.431 | 0.011 | Integrin alphaVbeta5 antagonist | 0.011 0.006 CHEMBL3542352 | CHEMBL3542352 | |
| 0.017 | 0.451 | 0.151 | Topoisomerase II inhibitor | 0.112 0.074 CHEMBL3542349 0.151 0.049 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.45 | 0.12 | M18 aspartyl aminopeptidase inhibitor | 0.12 0.071 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.437 | 0.025 | Retinoic acid receptor gamma antagonist | 0.025 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.054 | 0.49 | 0.699 | Superoxide dismutase inhibitor | 0.378 0.031 CHEMBL3542349 0.247 0.077 CHEMBL3542350 0.699 0.004 CHEMBL3542351 0.386 0.029 CHEMBL3988901 0.51 0.012 CHEMBL3542352 0.318 0.045 CHEMBL3988902 | CHEMBL3542351 | |
| 0.036 | 0.474 | 0.117 | Toll-Like receptor 3 antagonist | 0.117 0.032 CHEMBL3542349 0.095 0.059 CHEMBL3542350 0.089 0.071 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.443 | 0.082 | Methionyl aminopeptidase 2 inhibitor | 0.082 0.004 CHEMBL3542351 0.035 0.011 CHEMBL3988902 | CHEMBL3542351 | |
| 0.041 | 0.481 | 0.084 | Transforming growth factor beta 3 antagonist | 0.084 0.051 CHEMBL3542349 0.08 0.066 CHEMBL3542351 | CHEMBL3542349 | |
| 0.012 | 0.454 | 0.16 | Cytokine production stimulant | 0.053 0.023 CHEMBL3542349 0.16 0.002 CHEMBL3542350 0.052 0.025 CHEMBL3542351 | CHEMBL3542350 | |
| 0.062 | 0.505 | 0.147 | Death-associated protein kinase 2 inhibitor | 0.147 0.114 CHEMBL3542352 | CHEMBL3542352 | |
| 0.01 | 0.457 | 0.354 | Histidine decarboxylase inhibitor | 0.155 0.019 CHEMBL3542349 0.079 0.043 CHEMBL3526896 0.274 0.008 CHEMBL3542351 0.354 0.005 CHEMBL3988901 0.135 0.022 CHEMBL3542352 | CHEMBL3988901 | |
| 0.032 | 0.48 | 0.164 | Free radical scavenger | 0.164 0.13 CHEMBL3988901 | CHEMBL3988901 | |
| 0.015 | 0.464 | 0.122 | Topoisomerase I inhibitor | 0.105 0.066 CHEMBL3542349 0.122 0.054 CHEMBL3542350 0.099 0.071 CHEMBL3542351 0.085 0.084 CHEMBL3542352 | CHEMBL3542350 | |
| 0.017 | 0.47 | 0.128 | Caspase 7 inhibitor | 0.087 0.047 CHEMBL3542351 0.087 0.047 CHEMBL3542352 0.128 0.012 CHEMBL3988902 | CHEMBL3988902 | |
| 0.007 | 0.46 | 0.898 | Alcohol oxidase inhibitor | 0.206 0.006 CHEMBL3542349 0.069 0.029 CHEMBL3542350 0.898 0.002 CHEMBL3542351 0.158 0.009 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.457 | 0.038 | Egl nine homolog 2 inhibitor | 0.013 0.008 CHEMBL3542351 0.038 0.004 CHEMBL3542352 | CHEMBL3542352 | |
| 0.008 | 0.467 | 0.095 | Glutamate (mGluR1a) antagonist | 0.077 0.009 CHEMBL3542349 0.095 0.005 CHEMBL3542351 0.069 0.011 CHEMBL3542352 | CHEMBL3542351 | |
| 0.036 | 0.496 | 0.188 | Antioxidant | 0.188 0.124 CHEMBL3988901 0.168 0.144 CHEMBL3988902 | CHEMBL3988901 | |
| 0.01 | 0.471 | 0.046 | Beta 2 adrenoreceptor antagonist | 0.046 0.042 CHEMBL3542352 | CHEMBL3542352 | |
| 0.009 | 0.472 | 0.036 | Protein kinase C beta I inhibitor | 0.036 0.015 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.471 | 0.034 | Protein kinase C beta II inhibitor | 0.034 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.475 | 0.1 | Protein kinase C eta inhibitor | 0.057 0.036 CHEMBL3542349 0.1 0.017 CHEMBL3542351 | CHEMBL3542351 | |
| 0.008 | 0.474 | 0.071 | Collagenase 3 inhibitor | 0.071 0.031 CHEMBL3988902 | CHEMBL3988902 | |
| 0.036 | 0.505 | 0.158 | Interleukin 4 antagonist | 0.158 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.486 | 0.053 | Benzodiazepine inverse agonist | 0.048 0.029 CHEMBL3542349 0.053 0.021 CHEMBL3542350 0.043 0.042 CHEMBL3542351 | CHEMBL3542350 | |
| 0.039 | 0.51 | 0.128 | Adenylate cyclase stimulant | 0.128 0.105 CHEMBL3988903 0.123 0.118 CHEMBL3542351 | CHEMBL3988903 | |
| 0.005 | 0.476 | 0.035 | Purinergic P2X3 antagonist | 0.035 0.023 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.476 | 0.052 | Retinoid X beta receptor agonist | 0.052 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.49 | 0.037 | Integrin alpha1beta1 antagonist | 0.037 0.032 CHEMBL3542352 0.036 0.033 CHEMBL3988902 | CHEMBL3542352 | |
| 0.022 | 0.496 | 0.074 | Adenine nucleotide translocase inhibitor | 0.074 0.012 CHEMBL3542351 0.073 0.013 CHEMBL3988901 | CHEMBL3542351 | |
| 0.028 | 0.504 | 0.146 | Interleukin 1b antagonist | 0.1 0.081 CHEMBL3542349 0.131 0.054 CHEMBL3526892 0.146 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.487 | 0.079 | CDC25B inhibitor | 0.079 0.029 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.489 | 0.084 | Platelet activating factor alpha antagonist | 0.084 0.075 CHEMBL3542350 | CHEMBL3542350 | |
| 0.013 | 0.494 | 0.153 | MAP-kinase-activated kinase 2 inhibitor | 0.153 0.01 CHEMBL3542349 0.114 0.022 CHEMBL3542350 0.105 0.026 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.485 | 0.073 | Lysine carboxypeptidase inhibitor | 0.026 0.02 CHEMBL3542351 0.045 0.009 CHEMBL3988901 0.073 0.005 CHEMBL3542352 | CHEMBL3542352 | |
| 0.015 | 0.502 | 0.166 | DNA intercalator | 0.09 0.086 CHEMBL3542349 0.166 0.036 CHEMBL3542350 0.106 0.068 CHEMBL3542351 0.096 0.078 CHEMBL3542352 | CHEMBL3542350 | |
| 0.012 | 0.5 | 0.071 | Nav1.8 sodium channel blocker | 0.071 0.054 CHEMBL3542351 | CHEMBL3542351 | |
| 0.019 | 0.509 | 0.162 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.124 0.097 CHEMBL3542349 0.162 0.069 CHEMBL3542351 | CHEMBL3542351 | |
| 0.024 | 0.516 | 0.167 | EphB2 antagonist | 0.167 0.113 CHEMBL3542351 | CHEMBL3542351 | |
| 0.013 | 0.506 | 0.111 | Protein kinase C delta inhibitor | 0.111 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.505 | 0.065 | Myc inhibitor | 0.065 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.506 | 0.097 | Leukotriene synthesis inhibitor | 0.097 0.028 CHEMBL3542351 | CHEMBL3542351 | |
| 0.008 | 0.505 | 0.104 | Plasminogen activator inhibitor antagonist | 0.104 0.009 CHEMBL3542350 0.096 0.011 CHEMBL3542351 | CHEMBL3542350 | |
| 0.109 | 0.608 | 0.212 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.2 0.166 CHEMBL3542349 0.202 0.16 CHEMBL3542351 0.212 0.134 CHEMBL3542352 | CHEMBL3542352 | |
| 0.001 | 0.501 | 0.016 | Aminopeptidase A inhibitor | 0.016 0.015 CHEMBL3988901 | CHEMBL3988901 | |
| 0.007 | 0.509 | 0.074 | Alpha tubulin antagonist | 0.074 0.022 CHEMBL3542349 | CHEMBL3542349 | |
| 0.01 | 0.515 | 0.129 | Stem cell growth factor agonist | 0.129 0.027 CHEMBL3542350 | CHEMBL3542350 | |
| 0.016 | 0.521 | 0.164 | MAP-kinase-activated kinase inhibitor | 0.164 0.011 CHEMBL3542349 0.119 0.026 CHEMBL3542350 0.114 0.029 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.51 | 0.056 | Retinoid X gamma receptor agonist | 0.056 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.51 | 0.027 | Kainate receptor 5 antagonist | 0.019 0.017 CHEMBL3542349 0.027 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.532 | 0.262 | Granulocyte macrophage colony stimulating factor agonist | 0.262 0.002 CHEMBL3542349 0.134 0.009 CHEMBL3542350 0.194 0.003 CHEMBL3542351 0.166 0.004 CHEMBL3542352 0.088 0.055 CHEMBL3988902 | CHEMBL3542349 | |
| 0.038 | 0.546 | 0.338 | Phospholipase C inhibitor | 0.188 0.053 CHEMBL3542349 0.143 0.122 CHEMBL3988903 0.203 0.042 CHEMBL3542351 0.338 0.015 CHEMBL3988901 0.188 0.053 CHEMBL3542352 0.149 0.107 CHEMBL3988902 | CHEMBL3988901 | |
| 0.02 | 0.532 | 0.216 | Death-associated protein kinase 3 inhibitor | 0.216 0.066 CHEMBL3542349 0.207 0.071 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.516 | 0.043 | Retinoic acid receptor antagonist | 0.043 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.017 | 0.531 | 0.551 | Glutathione S-transferase inhibitor | 0.083 0.056 CHEMBL3542351 0.551 0.001 CHEMBL3988901 0.105 0.033 CHEMBL3542352 0.271 0.003 CHEMBL3988902 | CHEMBL3988901 | |
| 0.006 | 0.521 | 0.034 | Carboxypeptidase B inhibitor | 0.034 0.021 CHEMBL3988901 0.033 0.022 CHEMBL3988902 | CHEMBL3988901 | |
| 0.007 | 0.523 | 0.086 | Retinoic acid alpha receptor agonist | 0.086 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.015 | 0.534 | 0.093 | Histone deacetylase SIRT1 stimulant | 0.086 0.038 CHEMBL3542349 0.093 0.033 CHEMBL3542351 | CHEMBL3542351 | |
| 0.015 | 0.534 | 0.093 | Histone deacetylase stimulant | 0.086 0.038 CHEMBL3542349 0.093 0.033 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.525 | 0.038 | Retinoic acid beta receptor agonist | 0.038 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.526 | 0.032 | Retinoic acid gamma receptor agonist | 0.032 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.039 | 0.56 | 0.26 | Hepatoprotectant | 0.26 0.041 CHEMBL3988901 0.182 0.078 CHEMBL3988902 | CHEMBL3988901 | |
| 0.005 | 0.528 | 0.121 | Catechol O-methyltransferase inhibitor | 0.121 0.004 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.529 | 0.103 | Nicotinic acid receptor 2 agonist | 0.103 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.532 | 0.216 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.196 0.007 CHEMBL3542349 0.09 0.017 CHEMBL3542350 0.216 0.006 CHEMBL3542351 0.125 0.01 CHEMBL3542352 | CHEMBL3542351 | |
| 0.014 | 0.539 | 0.117 | Protein kinase C nu inhibitor | 0.117 0.097 CHEMBL3542351 | CHEMBL3542351 | |
| 0.074 | 0.601 | 0.618 | 5 Hydroxytryptamine release inhibitor | 0.354 0.112 CHEMBL3542349 0.242 0.24 CHEMBL3542350 0.618 0.009 CHEMBL3542351 0.45 0.052 CHEMBL3542352 | CHEMBL3542351 | |
| 0.008 | 0.535 | 0.745 | Aconitate hydratase inhibitor | 0.146 0.004 CHEMBL3542349 0.08 0.014 CHEMBL3542350 0.745 0.001 CHEMBL3542351 0.2 0.003 CHEMBL3542352 | CHEMBL3542351 | |
| 0.078 | 0.608 | 0.758 | Caspase 9 stimulant | 0.758 0.017 CHEMBL3542349 0.663 0.028 CHEMBL3542350 0.481 0.068 CHEMBL3542351 0.412 0.104 CHEMBL3542352 | CHEMBL3542349 | |
| 0.03 | 0.562 | 0.113 | CDK3/cyclin E inhibitor | 0.113 0.065 CHEMBL3542352 | CHEMBL3542352 | |
| 0.037 | 0.569 | 0.238 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.238 0.007 CHEMBL3542351 0.148 0.075 CHEMBL3542352 | CHEMBL3542351 | |
| 0.016 | 0.551 | 0.402 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.402 0.01 CHEMBL3542349 0.217 0.065 CHEMBL3542350 0.231 0.055 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.539 | 0.039 | Retinoic acid alpha receptor antagonist | 0.039 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.543 | 0.138 | Cyclin-dependent kinase 5 inhibitor | 0.138 0.047 CHEMBL3542349 0.097 0.078 CHEMBL3542350 | CHEMBL3542349 | |
| 0.042 | 0.58 | 0.555 | Cholesterol antagonist | 0.192 0.172 CHEMBL3988903 0.555 0.024 CHEMBL3542351 0.284 0.102 CHEMBL3542352 | CHEMBL3542351 | |
| 0.049 | 0.587 | 0.29 | Vasodilator, coronary | 0.29 0.096 CHEMBL3542351 0.192 0.19 CHEMBL3542352 | CHEMBL3542351 | |
| 0.026 | 0.567 | 0.171 | Interleukin 1 antagonist | 0.127 0.079 CHEMBL3542349 0.112 0.102 CHEMBL3526892 0.137 0.068 CHEMBL3542350 0.171 0.046 CHEMBL3542351 0.11 0.104 CHEMBL3988902 | CHEMBL3542351 | |
| 0.005 | 0.549 | 0.122 | Monophenol monooxygenase inhibitor | 0.122 0.06 CHEMBL3542349 0.118 0.063 CHEMBL3542351 | CHEMBL3542349 | |
| 0.009 | 0.553 | 0.157 | M17 leucyl aminopeptidase inhibitor | 0.157 0.051 CHEMBL3542351 0.12 0.078 CHEMBL3988902 | CHEMBL3542351 | |
| 0.008 | 0.556 | 0.076 | Protein kinase A inhibitor | 0.076 0.064 CHEMBL3542351 | CHEMBL3542351 | |
| 0.037 | 0.587 | 0.23 | Immunosuppressant | 0.23 0.166 CHEMBL3542350 | CHEMBL3542350 | |
| 0.007 | 0.557 | 0.039 | Integrin alpha2 antagonist | 0.039 0.022 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.555 | 0.044 | Proto-oncogene tyrosine-protein kinase Met inhibitor | 0.044 0.038 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.556 | 0.138 | Proto-oncogene tyrosine-protein kinase Kit inhibitor | 0.138 0.037 CHEMBL3542350 | CHEMBL3542350 | |
| 0.003 | 0.554 | 0.107 | Glucagon receptor antagonist | 0.107 0.004 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.556 | 0.082 | Fibroblast growth factor 4 antagonist | 0.082 0.017 CHEMBL3542349 | CHEMBL3542349 | |
| 0.006 | 0.558 | 0.075 | Acetylcholine M2 receptor agonist | 0.075 0.016 CHEMBL3542350 | CHEMBL3542350 | |
| 0.005 | 0.557 | 0.077 | HIV-1 integrase (Strand Transfer) inhibitor | 0.055 0.045 CHEMBL3542349 0.077 0.032 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.569 | 0.275 | GABA C receptor rho-1 antagonist | 0.149 0.022 CHEMBL3542349 0.127 0.034 CHEMBL3542350 0.275 0.004 CHEMBL3542351 0.241 0.005 CHEMBL3542352 | CHEMBL3542351 | |
| 0.01 | 0.563 | 0.173 | Purinergic P2X2 antagonist | 0.173 0.007 CHEMBL3542349 | CHEMBL3542349 | |
| 0.004 | 0.56 | 0.035 | Retinoid X gamma receptor antagonist | 0.035 0.007 CHEMBL3542351 | CHEMBL3542351 | |
| 0.022 | 0.579 | 0.08 | Thioredoxin reductase inhibitor | 0.078 0.067 CHEMBL3542349 0.08 0.063 CHEMBL3542351 | CHEMBL3542351 | |
| 0.029 | 0.586 | 0.121 | ABCA1 expression enhancer | 0.085 0.076 CHEMBL3542350 0.121 0.03 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.569 | 0.03 | DNA topoisomerase IV inhibitor | 0.03 0.02 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.585 | 0.173 | Hemostatic | 0.166 0.052 CHEMBL3542351 0.142 0.078 CHEMBL3988901 0.173 0.047 CHEMBL3542352 | CHEMBL3542352 | |
| 0.003 | 0.564 | 0.118 | Phosphorylase inhibitor | 0.043 0.034 CHEMBL3542349 0.067 0.022 CHEMBL3542351 0.118 0.01 CHEMBL3542352 | CHEMBL3542352 | |
| 0.022 | 0.583 | 0.24 | Platelet aggregation inhibitor | 0.194 0.085 CHEMBL3542351 0.24 0.056 CHEMBL3542352 | CHEMBL3542352 | |
| 0.057 | 0.619 | 0.294 | 5 Hydroxytryptamine release stimulant | 0.267 0.082 CHEMBL3542349 0.17 0.153 CHEMBL3542350 0.294 0.072 CHEMBL3542351 0.17 0.152 CHEMBL3542352 | CHEMBL3542351 | |
| 0.025 | 0.589 | 0.183 | Insulin secretagoues | 0.183 0.046 CHEMBL3542351 0.136 0.089 CHEMBL3988901 0.163 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.569 | 0.042 | Histone deacetylase 9 inhibitor | 0.042 0.023 CHEMBL3542350 0.039 0.027 CHEMBL3542352 | CHEMBL3542350 | |
| 0.05 | 0.621 | 0.224 | Lipocortins synthesis antagonist | 0.224 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.576 | 0.068 | Cyclin B2 inhibitor | 0.068 0.024 CHEMBL3542349 | CHEMBL3542349 | |
| 0.049 | 0.621 | 0.121 | Sphingosine 1-phosphate receptor 2 agonist | 0.121 0.053 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.578 | 0.064 | Leukotriene B4 antagonist | 0.064 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.581 | 0.062 | Cyclin B inhibitor | 0.062 0.03 CHEMBL3542349 | CHEMBL3542349 | |
| 0.006 | 0.582 | 0.075 | Cyclin B1 inhibitor | 0.075 0.026 CHEMBL3542349 | CHEMBL3542349 | |
| 0.008 | 0.584 | 0.11 | DNA gyrase inhibitor | 0.11 0.015 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.583 | 0.05 | Retinoic acid receptor agonist | 0.05 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.585 | 0.034 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.028 0.021 CHEMBL3542351 0.034 0.016 CHEMBL3542352 | CHEMBL3542352 | |
| 0.022 | 0.605 | 0.274 | DNA synthesis inhibitor | 0.199 0.125 CHEMBL3542349 0.263 0.059 CHEMBL3988903 0.274 0.054 CHEMBL3542351 0.194 0.133 CHEMBL3542352 | CHEMBL3542351 | |
| 0.007 | 0.59 | 0.063 | Alpha-mannosidase inhibitor | 0.063 0.023 CHEMBL3988903 | CHEMBL3988903 | |
| 0.035 | 0.618 | 0.254 | Transcription factor STAT inhibitor | 0.176 0.174 CHEMBL3988903 0.254 0.084 CHEMBL3542351 0.214 0.119 CHEMBL3988902 | CHEMBL3542351 | |
| 0.009 | 0.593 | 0.346 | CDC-like kinase 4 inhibitor | 0.346 0.022 CHEMBL3542349 0.129 0.118 CHEMBL3542350 0.164 0.09 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.588 | 0.031 | Prostaglandin EP1 antagonist | 0.031 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.013 | 0.599 | 0.109 | GABA B receptor agonist | 0.109 0.011 CHEMBL3542351 0.079 0.043 CHEMBL3542352 | CHEMBL3542351 | |
| 0.043 | 0.628 | 0.385 | Immunomodulator | 0.267 0.102 CHEMBL3526718 0.385 0.048 CHEMBL3988901 0.278 0.095 CHEMBL3526719 0.247 0.117 CHEMBL3988902 | CHEMBL3988901 | |
| 0.037 | 0.623 | 0.344 | NOS3 expression enhancer | 0.185 0.047 CHEMBL3542349 0.344 0.012 CHEMBL3542351 0.166 0.059 CHEMBL3542352 | CHEMBL3542351 | |
| 0.031 | 0.617 | 0.147 | Transcription factor STAT6 inhibitor | 0.147 0.026 CHEMBL3542349 0.121 0.058 CHEMBL3542351 | CHEMBL3542349 | |
| 0.024 | 0.614 | 0.165 | Cyclooxygenase 3 inhibitor | 0.145 0.052 CHEMBL3542351 0.165 0.036 CHEMBL3988902 | CHEMBL3988902 | |
| 0.026 | 0.616 | 0.145 | Melanin inhibitor | 0.145 0.088 CHEMBL3542349 0.132 0.111 CHEMBL3542351 | CHEMBL3542349 | |
| 0.008 | 0.603 | 0.173 | Hepatocyte growth factor antagonist | 0.108 0.044 CHEMBL3542349 0.173 0.016 CHEMBL3542350 | CHEMBL3542350 | |
| 0.006 | 0.601 | 0.204 | Glutamate decarboxylase inhibitor | 0.172 0.01 CHEMBL3542351 0.204 0.007 CHEMBL3988901 0.098 0.031 CHEMBL3542352 | CHEMBL3988901 | |
| 0.005 | 0.6 | 0.093 | Purinergic P2Y14 antagonist | 0.093 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.602 | 0.063 | Protein kinase C alpha inhibitor | 0.063 0.055 CHEMBL3542351 | CHEMBL3542351 | |
| 0.015 | 0.614 | 0.477 | Alpha-N-acetylglucosaminidase inhibitor | 0.155 0.052 CHEMBL3542349 0.319 0.014 CHEMBL3988903 0.477 0.006 CHEMBL3542351 0.178 0.041 CHEMBL3542352 0.245 0.024 CHEMBL3988902 | CHEMBL3542351 | |
| 0.028 | 0.627 | 0.408 | DNA damaging | 0.408 0.027 CHEMBL3542349 0.221 0.099 CHEMBL3542350 0.303 0.056 CHEMBL3542351 0.309 0.054 CHEMBL3542352 | CHEMBL3542349 | |
| 0.009 | 0.609 | 0.136 | Platelet growth factor antagonist | 0.136 0.023 CHEMBL3542349 0.081 0.056 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.606 | 0.014 | Integrin beta6 antagonist | 0.014 0.01 CHEMBL3542352 | CHEMBL3542352 | |
| 0.006 | 0.608 | 0.83 | Porphobilinogen synthase inhibitor | 0.736 0.002 CHEMBL3542349 0.118 0.029 CHEMBL3542350 0.83 0.001 CHEMBL3542351 0.491 0.003 CHEMBL3542352 0.082 0.046 CHEMBL3988902 | CHEMBL3542351 | |
| 0.005 | 0.608 | 0.072 | HIV-1 integrase (3'-Processing) inhibitor | 0.072 0.038 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.616 | 0.118 | Ca2+/calmodulin-dependent kinase II delta inhibitor | 0.118 0.086 CHEMBL3542351 | CHEMBL3542351 | |
| 0.023 | 0.632 | 0.163 | Photosensitizer | 0.117 0.061 CHEMBL3542349 0.163 0.024 CHEMBL3542351 0.116 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.011 | 0.62 | 0.04 | Glutamate (mGluR8) antagonist | 0.038 0.021 CHEMBL3542351 0.04 0.017 CHEMBL3988901 | CHEMBL3988901 | |
| 0.002 | 0.611 | 0.057 | Antimetabolite | 0.057 0.027 CHEMBL3542352 | CHEMBL3542352 | |
| 0.001 | 0.611 | 0.057 | AMPA 1 receptor antagonist | 0.026 0.022 CHEMBL3542349 0.057 0.009 CHEMBL3542351 0.037 0.016 CHEMBL3988901 0.042 0.014 CHEMBL3542352 | CHEMBL3542351 | |
| 0.018 | 0.63 | 0.156 | DOPA decarboxylase inhibitor | 0.099 0.078 CHEMBL3542349 0.156 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.62 | 0.084 | Tryptophan 5 hydroxylase inhibitor | 0.052 0.005 CHEMBL3542351 0.084 0.003 CHEMBL3542352 | CHEMBL3542352 | |
| 0.01 | 0.624 | 0.344 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.344 0.009 CHEMBL3542349 0.177 0.055 CHEMBL3542350 0.159 0.067 CHEMBL3542351 | CHEMBL3542349 | |
| 0.029 | 0.644 | 0.326 | Interleukin agonist | 0.326 0.037 CHEMBL3542351 0.233 0.092 CHEMBL3988901 0.258 0.073 CHEMBL3542352 0.257 0.074 CHEMBL3988902 | CHEMBL3542351 | |
| 0.005 | 0.621 | 0.047 | Mannosidase inhibitor | 0.047 0.029 CHEMBL3988903 | CHEMBL3988903 | |
| 0.068 | 0.685 | 0.428 | MAP kinase kinase 6 inhibitor | 0.34 0.101 CHEMBL3542349 0.428 0.043 CHEMBL3542351 0.302 0.134 CHEMBL3542352 | CHEMBL3542351 | |
| 0.008 | 0.625 | 0.541 | CYP2A6 inhibitor | 0.541 0.002 CHEMBL3542349 0.138 0.02 CHEMBL3542350 0.144 0.018 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.62 | 0.062 | Geranyltranstransferase inhibitor | 0.062 0.012 CHEMBL3542351 0.041 0.036 CHEMBL3542352 | CHEMBL3542351 | |
| 0.014 | 0.632 | 0.201 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.201 0.006 CHEMBL3542349 0.106 0.033 CHEMBL3542350 0.152 0.014 CHEMBL3542351 | CHEMBL3542349 | |
| 0.03 | 0.65 | 0.257 | Neuropeptide Y2 antagonist | 0.176 0.167 CHEMBL3542351 0.257 0.05 CHEMBL3988901 0.256 0.051 CHEMBL3988902 | CHEMBL3988901 | |
| 0.005 | 0.627 | 0.054 | Glutamate (mGluR group II) agonist | 0.054 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.024 | 0.648 | 0.309 | GABA C receptor rho-2 antagonist | 0.241 0.014 CHEMBL3542349 0.236 0.015 CHEMBL3542350 0.302 0.005 CHEMBL3542351 0.309 0.005 CHEMBL3542352 | CHEMBL3542352 | |
| 0.018 | 0.643 | 0.216 | Carbonic anhydrase III inhibitor | 0.216 0.014 CHEMBL3542351 0.086 0.081 CHEMBL3988901 0.148 0.029 CHEMBL3988902 | CHEMBL3542351 | |
| 0.011 | 0.636 | 0.051 | Carnitine palmitoyltransferase 1B inhibitor | 0.051 0.028 CHEMBL3542351 | CHEMBL3542351 | |
| 0.012 | 0.645 | 0.13 | Topoisomerase II beta inhibitor | 0.093 0.01 CHEMBL3542349 0.13 0.006 CHEMBL3542351 0.089 0.011 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.634 | 0.037 | Arginase inhibitor | 0.037 0.025 CHEMBL3988901 | CHEMBL3988901 | |
| 0.009 | 0.642 | 0.268 | Mucolytic | 0.114 0.06 CHEMBL3542351 0.187 0.017 CHEMBL3988901 0.131 0.045 CHEMBL3542352 0.268 0.005 CHEMBL3988902 | CHEMBL3988902 | |
| 0.001 | 0.636 | 0.015 | Human herpes virus 5 capsid protein P40 inhibitor | 0.015 0.007 CHEMBL3542351 | CHEMBL3542351 | |
| 0.014 | 0.649 | 0.202 | Acetylcholine M3 receptor agonist | 0.202 0.004 CHEMBL3542350 | CHEMBL3542350 | |
| 0.004 | 0.639 | 0.108 | TRPA1 antagonist | 0.108 0.016 CHEMBL3542349 0.062 0.041 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.639 | 0.033 | Kinesin-like protein 1 inhibitor | 0.033 0.031 CHEMBL3988901 0.033 0.031 CHEMBL3988902 | CHEMBL3988902 | |
| 0.004 | 0.639 | 0.033 | Kinesin antagonist | 0.033 0.031 CHEMBL3988901 0.033 0.031 CHEMBL3988902 | CHEMBL3988902 | |
| 0.019 | 0.657 | 0.308 | Transcription factor NF kappa B inhibitor | 0.308 0.09 CHEMBL3542349 0.213 0.157 CHEMBL3988903 0.197 0.172 CHEMBL3526896 0.29 0.1 CHEMBL3542351 0.267 0.116 CHEMBL3988901 0.279 0.107 CHEMBL3988902 | CHEMBL3542349 | |
| 0.01 | 0.648 | 0.136 | Beta amyloid protein antagonist | 0.136 0.052 CHEMBL3542351 0.125 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.644 | 0.088 | MAO A inhibitor | 0.088 0.073 CHEMBL3542349 | CHEMBL3542349 | |
| 0.01 | 0.651 | 0.073 | Potassium channel (Ca-activated) blocker | 0.073 0.024 CHEMBL3542350 | CHEMBL3542350 | |
| 0.027 | 0.669 | 0.351 | Neurotrophic factor enhancer | 0.351 0.009 CHEMBL3542349 0.179 0.099 CHEMBL3542350 0.282 0.024 CHEMBL3542351 0.288 0.021 CHEMBL3542352 | CHEMBL3542349 | |
| 0.021 | 0.665 | 0.1 | Interleukin 5 antagonist | 0.1 0.041 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.651 | 0.086 | Peroxisome proliferator-activated receptor gamma antagonist | 0.075 0.043 CHEMBL3542349 0.086 0.026 CHEMBL3542351 0.078 0.037 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.65 | 0.053 | Membrane dipeptidase inhibitor | 0.041 0.025 CHEMBL3542351 0.046 0.019 CHEMBL3988901 0.05 0.016 CHEMBL3542352 0.053 0.014 CHEMBL3988902 | CHEMBL3988902 | |
| 0.012 | 0.657 | 0.124 | MAP kinase 12 inhibitor | 0.124 0.065 CHEMBL3542349 | CHEMBL3542349 | |
| 0.021 | 0.666 | 0.238 | Transcription factor STAT3 inhibitor | 0.238 0.094 CHEMBL3542351 0.224 0.107 CHEMBL3988902 | CHEMBL3542351 | |
| 0.007 | 0.655 | 0.367 | CDC-like kinase 2 inhibitor | 0.367 0.018 CHEMBL3542349 0.152 0.092 CHEMBL3542351 | CHEMBL3542349 | |
| 0.022 | 0.67 | 0.168 | MAP3K9 inhibitor | 0.13 0.094 CHEMBL3542351 0.168 0.037 CHEMBL3988902 | CHEMBL3988902 | |
| 0.018 | 0.667 | 0.186 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.183 0.086 CHEMBL3542349 0.186 0.084 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.66 | 0.12 | Ornithine decarboxylase inhibitor | 0.086 0.06 CHEMBL3542349 0.093 0.052 CHEMBL3542350 0.12 0.026 CHEMBL3542351 | CHEMBL3542351 | |
| 0.018 | 0.668 | 0.131 | Farnesoid X receptor antagonist | 0.131 0.08 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.656 | 0.083 | Glutamate (mGluR group I) antagonist | 0.083 0.035 CHEMBL3542349 0.065 0.055 CHEMBL3542351 | CHEMBL3542349 | |
| 0.03 | 0.681 | 0.345 | Gastrin inhibitor | 0.187 0.168 CHEMBL3542349 0.327 0.018 CHEMBL3542351 0.265 0.063 CHEMBL3988901 0.345 0.012 CHEMBL3542352 0.23 0.104 CHEMBL3988902 | CHEMBL3542352 | |
| 0.016 | 0.668 | 0.126 | Neuropeptide Y1 antagonist | 0.126 0.108 CHEMBL3988901 | CHEMBL3988901 | |
| 0.013 | 0.666 | 0.138 | CD45 antagonist | 0.055 0.026 CHEMBL3542349 0.086 0.011 CHEMBL3542351 0.063 0.019 CHEMBL3988901 0.138 0.006 CHEMBL3542352 0.051 0.033 CHEMBL3988902 | CHEMBL3542352 | |
| 0.009 | 0.663 | 0.293 | CDC-like kinase 1 inhibitor | 0.293 0.011 CHEMBL3542349 0.158 0.064 CHEMBL3542350 0.146 0.073 CHEMBL3542351 | CHEMBL3542349 | |
| 0.005 | 0.662 | 0.097 | Sphingosine 1-phosphate receptor 3 antagonist | 0.097 0.009 CHEMBL3542350 0.073 0.023 CHEMBL3542351 0.061 0.036 CHEMBL3542352 | CHEMBL3542350 | |
| 0.005 | 0.662 | 0.199 | Pim-1 kinase inhibitor | 0.199 0.014 CHEMBL3542349 0.1 0.058 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.662 | 0.02 | Neuraminidase (Influenza B) inhibitor | 0.02 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.026 | 0.686 | 0.099 | T cell inhibitor | 0.099 0.025 CHEMBL3542352 | CHEMBL3542352 | |
| 0.003 | 0.664 | 0.102 | Leukotriene antagonist | 0.102 0.021 CHEMBL3542351 0.072 0.038 CHEMBL3988902 | CHEMBL3542351 | |
| 0.005 | 0.666 | 0.072 | Protein kinase C theta inhibitor | 0.072 0.02 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.669 | 0.317 | Clk dual-specificity kinase inhibitor | 0.317 0.035 CHEMBL3542349 0.144 0.12 CHEMBL3542350 0.158 0.107 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.669 | 0.034 | Glutamate (mGluR3) agonist | 0.034 0.017 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.675 | 0.243 | GABA C receptor antagonist | 0.132 0.041 CHEMBL3542349 0.118 0.055 CHEMBL3542350 0.243 0.007 CHEMBL3542351 0.203 0.012 CHEMBL3542352 | CHEMBL3542351 | |
| 0.016 | 0.681 | 0.485 | Aldehyde dehydrogenase inhibitor | 0.485 0.004 CHEMBL3542349 0.107 0.087 CHEMBL3542350 0.343 0.008 CHEMBL3542351 0.295 0.012 CHEMBL3988901 0.247 0.018 CHEMBL3542352 0.328 0.009 CHEMBL3988902 | CHEMBL3542349 | |
| 0.016 | 0.682 | 0.135 | Interleukin 6 antagonist | 0.135 0.115 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.671 | 0.031 | Glutamate (mGluR1) agonist | 0.031 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.672 | 0.062 | Benzodiazepine antagonist | 0.062 0.012 CHEMBL3542349 0.056 0.017 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.671 | 0.127 | Glutamate (mGluR1) antagonist | 0.113 0.013 CHEMBL3542349 0.127 0.01 CHEMBL3542351 0.083 0.022 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.67 | 0.047 | Fumarate hydratase inhibitor | 0.047 0.015 CHEMBL3542351 | CHEMBL3542351 | |
| 0.016 | 0.684 | 0.196 | Thioredoxin inhibitor | 0.196 0.009 CHEMBL3542349 0.093 0.057 CHEMBL3542351 | CHEMBL3542349 | |
| 0.001 | 0.67 | 0.022 | Angiotensin AT1B receptor antagonist | 0.022 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.025 | 0.695 | 0.095 | Estrogen-related receptor beta agonist | 0.095 0.032 CHEMBL3542352 | CHEMBL3542352 | |
| 0.002 | 0.672 | 0.064 | AMPA 3 receptor antagonist | 0.03 0.02 CHEMBL3542349 0.064 0.005 CHEMBL3542351 0.041 0.013 CHEMBL3988901 0.051 0.008 CHEMBL3542352 | CHEMBL3542351 | |
| 0.011 | 0.682 | 0.222 | Dual specificity phosphatase 3 inhibitor | 0.222 0.05 CHEMBL3542351 | CHEMBL3542351 | |
| 0.021 | 0.694 | 0.173 | ATPase inhibitor | 0.163 0.081 CHEMBL3542350 0.173 0.067 CHEMBL3542351 0.151 0.099 CHEMBL3542352 | CHEMBL3542351 | |
| 0.023 | 0.699 | 0.373 | Antibacterial | 0.267 0.161 CHEMBL3542349 0.373 0.089 CHEMBL3542350 0.352 0.101 CHEMBL3542351 0.273 0.156 CHEMBL3988901 0.362 0.096 CHEMBL3988902 | CHEMBL3542350 | |
| 0.015 | 0.694 | 0.272 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.272 0.008 CHEMBL3542351 0.219 0.013 CHEMBL3988901 0.256 0.009 CHEMBL3988902 | CHEMBL3542351 | |
| 0.004 | 0.684 | 0.122 | Prostaglandin E2 antagonist | 0.122 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.017 | 0.697 | 0.233 | Carbonic anhydrase XV inhibitor | 0.233 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.013 | 0.694 | 0.209 | Dual specificity phosphatase inhibitor | 0.209 0.05 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.684 | 0.074 | Ornithine carbamoyltransferase inhibitor | 0.074 0.024 CHEMBL3542351 0.073 0.024 CHEMBL3988901 | CHEMBL3542351 | |
| 0.005 | 0.689 | 0.304 | Phospholipase A2 inhibitor | 0.184 0.052 CHEMBL3542351 0.304 0.013 CHEMBL3988901 0.123 0.111 CHEMBL3542352 0.21 0.037 CHEMBL3988902 | CHEMBL3988901 | |
| 0.058 | 0.743 | 0.328 | Nitric-oxide synthase stimulant | 0.23 0.049 CHEMBL3542349 0.206 0.079 CHEMBL3542350 0.243 0.038 CHEMBL3542351 0.328 0.006 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.693 | 0.077 | Proto-oncogene tyrosine-protein kinase c-hck inhibitor | 0.077 0.056 CHEMBL3542349 | CHEMBL3542349 | |
| 0.006 | 0.697 | 0.252 | Expectorant | 0.092 0.078 CHEMBL3542351 0.168 0.029 CHEMBL3988901 0.093 0.078 CHEMBL3542352 0.252 0.012 CHEMBL3988902 | CHEMBL3988902 | |
| 0.007 | 0.699 | 0.18 | Vascular endothelial growth factor 3 antagonist | 0.18 0.05 CHEMBL3542350 | CHEMBL3542350 | |
| 0.015 | 0.708 | 0.235 | TRPA1 agonist | 0.235 0.006 CHEMBL3542349 0.217 0.008 CHEMBL3542351 0.147 0.033 CHEMBL3542352 | CHEMBL3542349 | |
| 0.007 | 0.701 | 0.284 | Macrophage migration inhibitory factor inhibitor | 0.201 0.008 CHEMBL3542349 0.284 0.005 CHEMBL3542350 0.245 0.005 CHEMBL3542351 | CHEMBL3542350 | |
| 0.004 | 0.699 | 0.086 | Glutamate (mGluR) agonist | 0.086 0.028 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.704 | 0.162 | Cholesterol synthesis inhibitor | 0.162 0.039 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.702 | 0.018 | Methylmalonyl-CoA mutase inhibitor | 0.018 0.012 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.701 | 0.169 | TRPM8 blocker | 0.036 0.03 CHEMBL3542349 0.169 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.023 | 0.723 | 0.176 | Tumour necrosis factor antagonist | 0.158 0.091 CHEMBL3542349 0.176 0.071 CHEMBL3542350 0.172 0.074 CHEMBL3542351 | CHEMBL3542350 | |
| 0.007 | 0.706 | 0.048 | H+/K+-transporting ATPase inhibitor | 0.048 0.04 CHEMBL3542349 | CHEMBL3542349 | |
| 0.062 | 0.762 | 0.393 | 5 Hydroxytryptamine uptake stimulant | 0.233 0.1 CHEMBL3542349 0.23 0.103 CHEMBL3542350 0.393 0.015 CHEMBL3542351 0.248 0.083 CHEMBL3542352 0.207 0.139 CHEMBL3988902 | CHEMBL3542351 | |
| 0.028 | 0.728 | 0.177 | Hypoglycemic | 0.177 0.138 CHEMBL3988903 0.176 0.139 CHEMBL3542351 0.166 0.153 CHEMBL3542352 | CHEMBL3988903 | |
| 0.007 | 0.709 | 0.403 | Anesthetic general | 0.403 0.016 CHEMBL3542349 0.144 0.12 CHEMBL3542350 0.279 0.039 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.71 | 0.085 | Prostaglandin antagonist | 0.085 0.021 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.712 | 0.111 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.099 0.014 CHEMBL3542349 0.111 0.008 CHEMBL3542350 0.108 0.009 CHEMBL3542351 0.093 0.019 CHEMBL3542352 | CHEMBL3542350 | |
| 0.004 | 0.711 | 0.078 | Carbonic anhydrase V inhibitor | 0.078 0.037 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.713 | 0.082 | HIV-1 integrase inhibitor | 0.082 0.037 CHEMBL3542351 0.072 0.045 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.711 | 0.039 | Prostaglandin EP4 antagonist | 0.039 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.013 | 0.722 | 0.377 | Streptokinase A inhibitor | 0.377 0.054 CHEMBL3542350 0.256 0.099 CHEMBL3542351 | CHEMBL3542350 | |
| 0.002 | 0.715 | 0.139 | Oleamide hydrolase inhibitor | 0.109 0.008 CHEMBL3542349 0.139 0.005 CHEMBL3542350 0.093 0.01 CHEMBL3542351 0.044 0.033 CHEMBL3542352 | CHEMBL3542350 | |
| 0.007 | 0.721 | 0.145 | Gastric antisecretory | 0.094 0.073 CHEMBL3542349 0.145 0.029 CHEMBL3542351 0.104 0.061 CHEMBL3542352 0.13 0.037 CHEMBL3988902 | CHEMBL3542351 | |
| 0.004 | 0.718 | 0.048 | Glutamate (mGluR2) agonist | 0.048 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.722 | 0.054 | Sphingosine 1-phosphate receptor 5 agonist | 0.054 0.037 CHEMBL3542352 | CHEMBL3542352 | |
| 0.003 | 0.719 | 0.112 | Acyl-CoA dehydrogenase inhibitor | 0.112 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.017 | 0.735 | 0.132 | Lanosterol 14 alpha demethylase inhibitor | 0.112 0.04 CHEMBL3542349 0.118 0.032 CHEMBL3542350 0.132 0.02 CHEMBL3542351 0.129 0.023 CHEMBL3542352 | CHEMBL3542351 | |
| 0.016 | 0.734 | 0.173 | Cytokine production inhibitor | 0.173 0.047 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.724 | 0.052 | CF transmembrane conductance regulator antagonist | 0.04 0.026 CHEMBL3542350 0.052 0.007 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.726 | 0.354 | Cystathionine beta-synthase inhibitor | 0.146 0.042 CHEMBL3542349 0.117 0.06 CHEMBL3542350 0.354 0.006 CHEMBL3542351 0.125 0.055 CHEMBL3542352 | CHEMBL3542351 | |
| 0.006 | 0.725 | 0.071 | Adenosine deaminase inhibitor | 0.071 0.013 CHEMBL3542351 0.043 0.037 CHEMBL3542352 | CHEMBL3542351 | |
| 0.01 | 0.73 | 0.09 | Prolactin inhibitor | 0.09 0.066 CHEMBL3542351 | CHEMBL3542351 | |
| 0.013 | 0.735 | 0.113 | Bile acid receptor antagonist | 0.113 0.027 CHEMBL3542351 0.09 0.074 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.728 | 0.061 | Histone deacetylase inhibitor | 0.058 0.057 CHEMBL3542350 0.061 0.052 CHEMBL3542352 | CHEMBL3542352 | |
| 0.008 | 0.732 | 0.07 | Cyclin B3 inhibitor | 0.07 0.046 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.727 | 0.021 | Toll-Like receptor 8 agonist | 0.021 0.012 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.727 | 0.228 | AMPA receptor antagonist | 0.228 0.004 CHEMBL3542349 0.225 0.004 CHEMBL3542351 0.051 0.03 CHEMBL3988901 0.109 0.01 CHEMBL3542352 | CHEMBL3542349 | |
| 0.027 | 0.753 | 0.209 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.209 0.147 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.731 | 0.295 | Vascular endothelial growth factor 2 antagonist | 0.295 0.021 CHEMBL3542350 | CHEMBL3542350 | |
| 0.022 | 0.748 | 0.234 | Adenylate kinase inhibitor | 0.102 0.065 CHEMBL3542349 0.093 0.079 CHEMBL3988903 0.234 0.011 CHEMBL3542351 0.096 0.075 CHEMBL3988901 0.119 0.045 CHEMBL3542352 | CHEMBL3542351 | |
| 0.007 | 0.734 | 0.308 | Vascular endothelial growth factor antagonist | 0.308 0.021 CHEMBL3542350 | CHEMBL3542350 | |
| 0.012 | 0.74 | 0.123 | Carbonic anhydrase VI inhibitor | 0.123 0.028 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.733 | 0.242 | LIM domain kinase 1 inhibitor | 0.242 0.042 CHEMBL3542349 0.187 0.07 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.732 | 0.09 | Amidase inhibitor | 0.09 0.03 CHEMBL3542350 0.077 0.04 CHEMBL3542351 0.081 0.036 CHEMBL3542352 | CHEMBL3542350 | |
| 0.004 | 0.734 | 0.073 | Adrenaline agonist | 0.073 0.067 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.736 | 0.279 | RET inhibitor | 0.279 0.026 CHEMBL3542350 | CHEMBL3542350 | |
| 0.013 | 0.748 | 0.153 | Acetylcholine release stimulant | 0.145 0.02 CHEMBL3542349 0.119 0.049 CHEMBL3542350 0.153 0.015 CHEMBL3542351 0.118 0.052 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.739 | 0.049 | Carbonic anhydrase XIV inhibitor | 0.049 0.034 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.742 | 0.051 | AICAR transformylase inhibitor | 0.045 0.029 CHEMBL3542351 0.051 0.021 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.741 | 0.425 | Alcohol dehydrogenase inhibitor | 0.191 0.013 CHEMBL3542349 0.425 0.004 CHEMBL3542351 0.142 0.023 CHEMBL3988901 0.254 0.007 CHEMBL3542352 0.104 0.049 CHEMBL3988902 | CHEMBL3542351 | |
| 0.001 | 0.738 | 0.024 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.024 0.01 CHEMBL3542349 | CHEMBL3542349 | |
| 0.012 | 0.75 | 0.261 | Antibacterial (Helicobacter pylori) | 0.24 0.013 CHEMBL3542349 0.162 0.038 CHEMBL3542351 0.162 0.038 CHEMBL3988901 0.123 0.077 CHEMBL3542352 0.261 0.01 CHEMBL3988902 | CHEMBL3988902 | |
| 0.018 | 0.757 | 0.101 | Phosphodiesterase 7B inhibitor | 0.101 0.055 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.744 | 0.411 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.411 0.01 CHEMBL3542350 | CHEMBL3542350 | |
| 0.004 | 0.745 | 0.046 | Glutamate (mGluR5) antagonist | 0.046 0.034 CHEMBL3542349 0.042 0.039 CHEMBL3542350 | CHEMBL3542349 | |
| 0.049 | 0.792 | 0.211 | Heat shock protein 70 antagonist | 0.143 0.064 CHEMBL3542349 0.211 0.005 CHEMBL3542351 0.142 0.068 CHEMBL3542352 | CHEMBL3542351 | |
| 0.004 | 0.747 | 0.11 | Thromboxane synthase inhibitor | 0.11 0.005 CHEMBL3542351 0.093 0.008 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.748 | 0.346 | TRKB antagonist | 0.346 0.007 CHEMBL3542350 | CHEMBL3542350 | |
| 0.005 | 0.751 | 0.091 | Glutamate (mGluR) antagonist | 0.076 0.053 CHEMBL3542349 0.091 0.04 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.75 | 0.067 | GABA B receptor antagonist | 0.067 0.009 CHEMBL3542349 0.063 0.011 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.749 | 0.024 | Calcium-sensing receptor agonist | 0.024 0.023 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.75 | 0.075 | NMDA receptor glycine site agonist | 0.075 0.032 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.753 | 0.082 | NMDA receptor agonist | 0.082 0.027 CHEMBL3542351 0.056 0.054 CHEMBL3988901 0.059 0.049 CHEMBL3542352 0.06 0.047 CHEMBL3988902 | CHEMBL3542351 | |
| 0.002 | 0.751 | 0.052 | Inosine monophosphate dehydrogenase inhibitor | 0.052 0.014 CHEMBL3542349 | CHEMBL3542349 | |
| 0.006 | 0.754 | 0.128 | Growth factor antagonist | 0.127 0.086 CHEMBL3542349 0.128 0.085 CHEMBL3542350 | CHEMBL3542350 | |
| 0.005 | 0.753 | 0.231 | Protein kinase C gamma inhibitor | 0.179 0.019 CHEMBL3542349 0.231 0.009 CHEMBL3542351 0.11 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.755 | 0.053 | Glucosylceramidase inhibitor | 0.053 0.042 CHEMBL3542351 | CHEMBL3542351 | |
| 0.011 | 0.762 | 0.097 | Anabolic | 0.093 0.073 CHEMBL3542349 0.097 0.067 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.755 | 0.058 | AMPA 4 receptor antagonist | 0.058 0.011 CHEMBL3542351 0.041 0.024 CHEMBL3988901 | CHEMBL3542351 | |
| 0.004 | 0.756 | 0.126 | Macrophage colony-stimulating factor 1 receptor antagonist | 0.126 0.02 CHEMBL3542350 | CHEMBL3542350 | |
| 0.034 | 0.787 | 0.16 | MAP kinase kinase 4 inhibitor | 0.16 0.045 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.757 | 0.077 | Transforming growth factor beta 1 antagonist | 0.077 0.016 CHEMBL3542349 0.044 0.041 CHEMBL3542352 | CHEMBL3542349 | |
| 0.009 | 0.763 | 0.189 | Keratolytic | 0.189 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.756 | 0.123 | Kynurenine 3 monooxygenase inhibitor | 0.037 0.011 CHEMBL3542350 0.123 0.003 CHEMBL3542351 | CHEMBL3542351 | |
| 0.04 | 0.795 | 0.304 | Tyrosine 3 hydroxylase inhibitor | 0.206 0.126 CHEMBL3542349 0.247 0.071 CHEMBL3542351 0.304 0.031 CHEMBL3542352 | CHEMBL3542352 | |
| 0.01 | 0.766 | 0.193 | Potassium channel (Ca-activated) activator | 0.193 0.016 CHEMBL3542351 0.097 0.058 CHEMBL3542352 | CHEMBL3542351 | |
| 0.016 | 0.773 | 0.087 | Transcription factor RelA inhibitor | 0.087 0.012 CHEMBL3542349 0.078 0.019 CHEMBL3542350 0.086 0.013 CHEMBL3542351 | CHEMBL3542349 | |
| 0.005 | 0.763 | 0.191 | Mcl-1 antagonist | 0.191 0.061 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.766 | 0.053 | Sphingosine 1-phosphate receptor 1 antagonist | 0.053 0.044 CHEMBL3542352 | CHEMBL3542352 | |
| 0.025 | 0.786 | 0.65 | Histamine release inhibitor | 0.302 0.122 CHEMBL3542349 0.65 0.007 CHEMBL3542351 0.488 0.033 CHEMBL3988901 0.499 0.029 CHEMBL3542352 0.44 0.055 CHEMBL3988902 | CHEMBL3542351 | |
| 0.019 | 0.781 | 0.175 | Interferon gamma antagonist | 0.157 0.069 CHEMBL3542349 0.175 0.053 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.765 | 0.095 | Thymidylate synthase inhibitor | 0.051 0.026 CHEMBL3542351 0.066 0.013 CHEMBL3988901 0.095 0.005 CHEMBL3542352 0.049 0.029 CHEMBL3988902 | CHEMBL3542352 | |
| 0.007 | 0.77 | 0.248 | Uric acid excretion stimulant | 0.248 0.007 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.768 | 0.432 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.432 0.021 CHEMBL3542349 0.211 0.086 CHEMBL3542350 0.306 0.049 CHEMBL3542351 | CHEMBL3542349 | |
| 0.011 | 0.775 | 0.064 | Exportin-1 inhibitor | 0.064 0.059 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.768 | 0.08 | Potassium channel (ATP-sensitive) blocker | 0.08 0.028 CHEMBL3542349 0.075 0.034 CHEMBL3542351 | CHEMBL3542349 | |
| 0.012 | 0.777 | 0.709 | Aldehyde oxidase inhibitor | 0.709 0.008 CHEMBL3542349 0.653 0.013 CHEMBL3542351 0.267 0.076 CHEMBL3542352 | CHEMBL3542349 | |
| 0.006 | 0.775 | 0.047 | Vanilloid 3 antagonist | 0.041 0.02 CHEMBL3542349 0.047 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.776 | 0.157 | Phospholipase D inhibitor | 0.085 0.028 CHEMBL3542349 0.109 0.01 CHEMBL3542351 0.157 0.003 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.775 | 0.239 | ErbB-2 antagonist | 0.239 0.007 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.771 | 0.039 | Nicotinic acid receptor 1 antagonist | 0.039 0.003 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.771 | 0.027 | Prostaglandin EP2 agonist | 0.027 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.773 | 0.04 | Alpha 2b adrenoreceptor agonist | 0.04 0.004 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.775 | 0.163 | Protein kinase C zeta inhibitor | 0.163 0.017 CHEMBL3542349 0.119 0.033 CHEMBL3542351 | CHEMBL3542349 | |
| 0.017 | 0.789 | 0.095 | Glutamate (mGluR7) agonist | 0.091 0.081 CHEMBL3542351 0.095 0.072 CHEMBL3542352 | CHEMBL3542352 | |
| 0.002 | 0.774 | 0.089 | Carbonic anhydrase VB inhibitor | 0.089 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.776 | 0.166 | Diuretic | 0.164 0.065 CHEMBL3542351 0.166 0.064 CHEMBL3988901 0.164 0.066 CHEMBL3542352 | CHEMBL3988901 | |
| 0.004 | 0.779 | 0.414 | Dyrk kinase inhibitor | 0.414 0.024 CHEMBL3542349 0.209 0.094 CHEMBL3542350 0.3 0.053 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.78 | 0.064 | DNA-dependent protein kinase inhibitor | 0.064 0.013 CHEMBL3542349 | CHEMBL3542349 | |
| 0.027 | 0.804 | 0.616 | GABA C receptor rho-3 antagonist | 0.556 0.013 CHEMBL3542349 0.502 0.025 CHEMBL3542350 0.581 0.01 CHEMBL3542351 0.616 0.006 CHEMBL3542352 | CHEMBL3542352 | |
| 0.006 | 0.783 | 0.097 | Fatty acid synthase inhibitor | 0.053 0.045 CHEMBL3542349 0.097 0.012 CHEMBL3542351 0.052 0.047 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.778 | 0.045 | Prostaglandin H2 antagonist | 0.045 0.004 CHEMBL3542351 0.027 0.016 CHEMBL3542352 | CHEMBL3542351 | |
| 0.012 | 0.79 | 0.341 | DNA methylase inhibitor | 0.157 0.111 CHEMBL3542349 0.298 0.028 CHEMBL3542351 0.337 0.019 CHEMBL3988901 0.246 0.05 CHEMBL3542352 0.341 0.018 CHEMBL3988902 | CHEMBL3988902 | |
| 0.004 | 0.783 | 0.082 | CDC7 inhibitor | 0.064 0.051 CHEMBL3542349 0.082 0.034 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.784 | 0.03 | Glucosylceramidase stimulant | 0.03 0.012 CHEMBL3542349 0.026 0.024 CHEMBL3542352 | CHEMBL3542349 | |
| 0.007 | 0.787 | 0.212 | Histamine N-methyltransferase inhibitor | 0.143 0.017 CHEMBL3542349 0.093 0.052 CHEMBL3542350 0.212 0.005 CHEMBL3542351 0.095 0.051 CHEMBL3988901 0.106 0.04 CHEMBL3542352 0.086 0.06 CHEMBL3988902 | CHEMBL3542351 | |
| 0.03 | 0.811 | 0.166 | MAP-kinase-activated kinase 5 inhibitor | 0.166 0.155 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.785 | 0.058 | Epithelial sodium channel blocker | 0.058 0.032 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.786 | 0.046 | Phosphodiesterase 4A inhibitor | 0.046 0.038 CHEMBL3542350 | CHEMBL3542350 | |
| 0.003 | 0.785 | 0.098 | Rho-associated kinase I inhibitor | 0.098 0.033 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.787 | 0.136 | Glutamate (mGluR7) antagonist | 0.109 0.007 CHEMBL3542349 0.11 0.006 CHEMBL3542350 0.136 0.004 CHEMBL3542351 0.075 0.034 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.786 | 0.061 | Carbamoyl phosphate synthetase inhibitor | 0.061 0.042 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.793 | 0.163 | Glutamate dehydrogenase inhibitor | 0.095 0.033 CHEMBL3542349 0.163 0.014 CHEMBL3542351 0.103 0.029 CHEMBL3988901 0.081 0.044 CHEMBL3542352 0.092 0.035 CHEMBL3988902 | CHEMBL3542351 | |
| 0.006 | 0.79 | 0.437 | Ferrochelatase inhibitor | 0.148 0.038 CHEMBL3542349 0.437 0.003 CHEMBL3542351 0.176 0.029 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.785 | 0.035 | Phosphoglycerate kinase inhibitor | 0.035 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.794 | 0.325 | DNA methyltransferase I inhibitor | 0.149 0.105 CHEMBL3542349 0.3 0.026 CHEMBL3542351 0.289 0.03 CHEMBL3988901 0.235 0.053 CHEMBL3542352 0.325 0.019 CHEMBL3988902 | CHEMBL3988902 | |
| 0.003 | 0.787 | 0.073 | Leukotriene C antagonist | 0.073 0.012 CHEMBL3542351 0.061 0.028 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.786 | 0.028 | Epoxide hydrolase 1 inhibitor | 0.028 0.027 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.79 | 0.029 | Prostaglandin agonist | 0.029 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.011 | 0.8 | 0.239 | Triose-phosphate isomerase inhibitor | 0.087 0.064 CHEMBL3542349 0.102 0.046 CHEMBL3988903 0.239 0.008 CHEMBL3542351 0.083 0.071 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.792 | 0.115 | Pim-2 kinase inhibitor | 0.115 0.012 CHEMBL3542349 | CHEMBL3542349 | |
| 0 | 0.79 | 0.135 | Egl nine homolog 3 inhibitor | 0.057 0.003 CHEMBL3542351 0.135 0.002 CHEMBL3542352 | CHEMBL3542352 | |
| 0.009 | 0.802 | 0.111 | Adenylate cyclase inhibitor | 0.111 0.075 CHEMBL3542352 | CHEMBL3542352 | |
| 0.01 | 0.804 | 0.155 | Sphingosine 1-phosphate receptor 4 antagonist | 0.155 0.029 CHEMBL3542349 0.155 0.029 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.796 | 0.025 | Myristoyl transferase inhibitor | 0.025 0.023 CHEMBL3542349 | CHEMBL3542349 | |
| 0.007 | 0.802 | 0.348 | Cholinergic | 0.348 0.013 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.797 | 0.18 | Egl nine homolog 1 inhibitor | 0.063 0.003 CHEMBL3542351 0.18 0.002 CHEMBL3542352 | CHEMBL3542352 | |
| 0.007 | 0.803 | 0.314 | Mannose-6-phosphate isomerase inhibitor | 0.269 0.009 CHEMBL3542349 0.167 0.051 CHEMBL3542350 0.314 0.005 CHEMBL3542351 0.174 0.046 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.799 | 0.065 | Thromboxane A2 antagonist | 0.065 0.025 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.8 | 0.112 | Glutamate (mGluR4) agonist | 0.039 0.017 CHEMBL3542349 0.037 0.019 CHEMBL3542350 0.112 0.004 CHEMBL3542351 0.038 0.018 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.802 | 0.16 | MAO inhibitor | 0.16 0.056 CHEMBL3542349 | CHEMBL3542349 | |
| 0.004 | 0.804 | 0.17 | Glutamate (mGluR group III) agonist | 0.048 0.025 CHEMBL3542349 0.045 0.028 CHEMBL3542350 0.17 0.004 CHEMBL3542351 0.074 0.014 CHEMBL3542352 0.051 0.023 CHEMBL3988902 | CHEMBL3542351 | |
| 0.005 | 0.806 | 0.091 | Pregnane X receptor antagonist | 0.091 0.004 CHEMBL3542349 0.083 0.005 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.804 | 0.256 | Protein kinase (CK2) alpha inhibitor | 0.256 0.015 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.804 | 0.062 | DNA gyrase subunit B inhibitor | 0.062 0.008 CHEMBL3542351 0.052 0.012 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.803 | 0.022 | Prostaglandin E2 agonist | 0.022 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.807 | 0.085 | Carbonic anhydrase VA inhibitor | 0.085 0.033 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.808 | 0.067 | NMDA 2C receptor antagonist | 0.067 0.037 CHEMBL3542351 | CHEMBL3542351 | |
| 0 | 0.806 | 0.007 | Integrin alpha5beta6 antagonist | 0.007 0.004 CHEMBL3542352 | CHEMBL3542352 | |
| 0.009 | 0.816 | 0.208 | Interleukin 8 antagonist | 0.208 0.011 CHEMBL3542349 0.166 0.025 CHEMBL3542351 0.107 0.082 CHEMBL3542352 | CHEMBL3542349 | |
| 0.003 | 0.81 | 0.056 | Squalene epoxidase inhibitor | 0.056 0.024 CHEMBL3542349 | CHEMBL3542349 | |
| 0.008 | 0.817 | 0.141 | Purinergic P2X1 antagonist | 0.118 0.012 CHEMBL3542349 0.141 0.008 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.81 | 0.083 | Kainate receptor antagonist | 0.037 0.032 CHEMBL3542349 0.083 0.009 CHEMBL3542351 0.036 0.033 CHEMBL3988901 | CHEMBL3542351 | |
| 0.002 | 0.812 | 0.053 | Acetylcholine M2 receptor antagonist | 0.053 0.051 CHEMBL3542350 | CHEMBL3542350 | |
| 0.004 | 0.814 | 0.077 | Sphingosine 1-phosphate receptor antagonist | 0.076 0.054 CHEMBL3542350 0.073 0.062 CHEMBL3542351 0.077 0.052 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.815 | 0.19 | Spasmolytic | 0.17 0.145 CHEMBL3542349 0.19 0.129 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.812 | 0.028 | MAP3K8 inhibitor | 0.028 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.813 | 0.064 | Kainate receptor 2 antagonist | 0.051 0.015 CHEMBL3542349 0.064 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.814 | 0.051 | Histamine H1 receptor agonist | 0.051 0.016 CHEMBL3542349 0.041 0.038 CHEMBL3542351 | CHEMBL3542349 | |
| 0.001 | 0.814 | 0.053 | Carbonic anhydrase IV inhibitor | 0.053 0.023 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.818 | 0.054 | Heat shock protein 90 beta antagonist | 0.054 0.053 CHEMBL3542352 | CHEMBL3542352 | |
| 0.002 | 0.816 | 0.18 | Pim-3 kinase inhibitor | 0.18 0.011 CHEMBL3542349 0.09 0.058 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.816 | 0.07 | Thromboxane antagonist | 0.07 0.026 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.818 | 0.088 | Protein kinase (CK2) beta inhibitor | 0.041 0.011 CHEMBL3542349 0.088 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.817 | 0.215 | Xanthine dehydrogenase inhibitor | 0.131 0.009 CHEMBL3542349 0.215 0.004 CHEMBL3542351 0.057 0.041 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.817 | 0.063 | GABA uptake inhibitor | 0.063 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.82 | 0.066 | Heparanase inhibitor | 0.066 0.015 CHEMBL3542351 0.056 0.03 CHEMBL3542352 | CHEMBL3542351 | |
| 0.006 | 0.822 | 0.186 | Arachidonic acid antagonist | 0.13 0.112 CHEMBL3542349 0.186 0.047 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.818 | 0.043 | Alpha 2c adrenoreceptor agonist | 0.025 0.006 CHEMBL3542349 0.043 0.004 CHEMBL3542350 | CHEMBL3542350 | |
| 0.005 | 0.824 | 0.074 | Potassium channel (Tandem pore domain) blocker | 0.074 0.051 CHEMBL3542352 | CHEMBL3542352 | |
| 0.008 | 0.827 | 0.082 | MDM2 inhibitor | 0.082 0.017 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.825 | 0.155 | Epidermal growth factor receptor kinase inhibitor | 0.155 0.045 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.822 | 0.047 | Leukotriene C4 antagonist | 0.047 0.013 CHEMBL3542351 0.037 0.032 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.822 | 0.077 | Aryl hydrocarbon receptor antagonist | 0.077 0.029 CHEMBL3542349 0.063 0.048 CHEMBL3542351 | CHEMBL3542349 | |
| 0.004 | 0.824 | 0.162 | Phosphodiesterase 4D inhibitor | 0.162 0.016 CHEMBL3542350 0.088 0.043 CHEMBL3542351 | CHEMBL3542350 | |
| 0.002 | 0.823 | 0.042 | Histamine H2 receptor agonist | 0.042 0.031 CHEMBL3542349 | CHEMBL3542349 | |
| 0.005 | 0.827 | 0.281 | 12-Lipoxygenase inhibitor | 0.264 0.101 CHEMBL3542349 0.281 0.091 CHEMBL3542351 | CHEMBL3542351 | |
| 0.03 | 0.855 | 0.403 | Calcium channel activator | 0.319 0.074 CHEMBL3542349 0.283 0.109 CHEMBL3542350 0.403 0.023 CHEMBL3542351 0.252 0.145 CHEMBL3542352 | CHEMBL3542351 | |
| 0.006 | 0.833 | 0.105 | Carbonic anhydrase XIII inhibitor | 0.105 0.035 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.83 | 0.035 | ICAM 1 antagonist | 0.024 0.014 CHEMBL3542349 0.023 0.016 CHEMBL3542351 0.035 0.005 CHEMBL3542352 | CHEMBL3542352 | |
| 0.005 | 0.834 | 0.106 | Phosphodiesterase inhibitor | 0.106 0.099 CHEMBL3542350 | CHEMBL3542350 | |
| 0.009 | 0.838 | 0.355 | Cyclic AMP phosphodiesterase inhibitor | 0.154 0.146 CHEMBL3542349 0.181 0.11 CHEMBL3542350 0.355 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.834 | 0.177 | Alkaline phosphatase inhibitor | 0.154 0.057 CHEMBL3542349 0.177 0.044 CHEMBL3542351 0.135 0.071 CHEMBL3542352 | CHEMBL3542351 | |
| 0.008 | 0.842 | 0.24 | Electrolyte absorption antagonist | 0.094 0.067 CHEMBL3542349 0.24 0.005 CHEMBL3542351 0.136 0.026 CHEMBL3542352 0.114 0.041 CHEMBL3988902 | CHEMBL3542351 | |
| 0.006 | 0.84 | 0.142 | Nav1.6 sodium channel blocker | 0.122 0.093 CHEMBL3542349 0.142 0.064 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.836 | 0.089 | Glycine transporter 2 inhibitor | 0.089 0.015 CHEMBL3988901 0.076 0.019 CHEMBL3542352 | CHEMBL3988901 | |
| 0.004 | 0.838 | 0.09 | Glycine receptor antagonist | 0.09 0.042 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.838 | 0.045 | Nicotinic acid receptor 2 antagonist | 0.045 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.841 | 0.115 | Urease inhibitor | 0.115 0.05 CHEMBL3542351 0.105 0.061 CHEMBL3542352 | CHEMBL3542351 | |
| 0.042 | 0.881 | 0.621 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.621 0.005 CHEMBL3542349 0.44 0.068 CHEMBL3542350 0.557 0.014 CHEMBL3542351 0.463 0.053 CHEMBL3542352 | CHEMBL3542349 | |
| 0.001 | 0.84 | 0.072 | Guanylate cyclase inhibitor | 0.04 0.034 CHEMBL3542349 0.072 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.842 | 0.122 | Phosphofructokinase-1 inhibitor | 0.106 0.029 CHEMBL3542349 0.122 0.025 CHEMBL3542351 | CHEMBL3542351 | |
| 0.014 | 0.854 | 0.179 | Amylase inhibitor | 0.179 0.052 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.847 | 0.296 | Beta glucuronidase inhibitor | 0.245 0.009 CHEMBL3542349 0.296 0.006 CHEMBL3542350 0.171 0.018 CHEMBL3542351 | CHEMBL3542350 | |
| 0.007 | 0.847 | 0.073 | Phosphodiesterase VI inhibitor | 0.073 0.055 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.846 | 0.091 | Myeloperoxidase inhibitor | 0.091 0.047 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.849 | 0.26 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.172 0.105 CHEMBL3542350 0.26 0.038 CHEMBL3542351 0.166 0.114 CHEMBL3542352 | CHEMBL3542351 | |
| 0.004 | 0.846 | 0.074 | Adenosine A3 receptor antagonist | 0.072 0.055 CHEMBL3542349 0.074 0.053 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.844 | 0.23 | Biliverdin reductase inhibitor | 0.23 0.005 CHEMBL3542351 0.06 0.041 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.845 | 0.041 | Dihydrofolate reductase inhibitor | 0.04 0.039 CHEMBL3542351 0.041 0.038 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.848 | 0.131 | Activin receptor-like kinase 2 inhibitor | 0.131 0.084 CHEMBL3542349 0.12 0.096 CHEMBL3542350 0.121 0.095 CHEMBL3542351 | CHEMBL3542349 | |
| 0 | 0.845 | 0.018 | Thrombopoietin agonist | 0.018 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.014 | 0.859 | 0.164 | MAP kinase 3 inhibitor | 0.128 0.112 CHEMBL3542349 0.164 0.049 CHEMBL3542351 0.138 0.09 CHEMBL3542352 | CHEMBL3542351 | |
| 0.007 | 0.852 | 0.234 | Xanthine oxidase inhibitor | 0.2 0.019 CHEMBL3542349 0.234 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.846 | 0.072 | Free fatty acid receptor 1 antagonist | 0.033 0.024 CHEMBL3542349 0.072 0.004 CHEMBL3542351 0.032 0.027 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.847 | 0.048 | CDK5/p25 inhibitor | 0.048 0.023 CHEMBL3542349 | CHEMBL3542349 | |
| 0.011 | 0.857 | 0.267 | Cyclophilin D inhibitor | 0.267 0.194 CHEMBL3542351 0.267 0.194 CHEMBL3542352 | CHEMBL3542352 | |
| 0.001 | 0.848 | 0.037 | Protein kinase (CK1) epsilon inhibitor | 0.037 0.033 CHEMBL3542349 | CHEMBL3542349 | |
| 0.009 | 0.856 | 0.096 | mTOR complex 2 inhibitor | 0.084 0.059 CHEMBL3542349 0.096 0.039 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.849 | 0.058 | Farnesoid X receptor agonist | 0.058 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.85 | 0.254 | Protein kinase (CK2) inhibitor | 0.083 0.08 CHEMBL3542349 0.254 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.85 | 0.162 | Argininosuccinate synthase inhibitor | 0.162 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.859 | 0.163 | HIV-1 integrase (Overall Integration) inhibitor | 0.163 0.021 CHEMBL3542351 0.133 0.032 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.853 | 0.122 | Cyclooxygenase 2 inhibitor | 0.122 0.077 CHEMBL3542350 | CHEMBL3542350 | |
| 0 | 0.85 | 0.033 | Kainate receptor 1 antagonist | 0.033 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.854 | 0.111 | Protein kinase C beta inhibitor | 0.1 0.014 CHEMBL3542349 0.111 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.851 | 0.025 | NMDA receptor glycine site antagonist | 0.025 0.016 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.853 | 0.018 | CC chemokine 9 receptor antagonist | 0.018 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.855 | 0.163 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.16 0.016 CHEMBL3542349 0.163 0.015 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.858 | 0.21 | Glutamate receptor antagonist | 0.143 0.056 CHEMBL3542349 0.21 0.023 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.855 | 0.077 | NMDA receptor subunit 3B antagonist | 0.077 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.858 | 0.416 | GABA C receptor agonist | 0.12 0.049 CHEMBL3542349 0.095 0.072 CHEMBL3542350 0.416 0.005 CHEMBL3542351 0.21 0.019 CHEMBL3542352 | CHEMBL3542351 | |
| 0.004 | 0.858 | 0.079 | Potassium channel intermediate-conductance Ca-activated blocker | 0.061 0.04 CHEMBL3542349 0.079 0.018 CHEMBL3542350 0.079 0.018 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.857 | 0.047 | Liver X receptor beta antagonist | 0.047 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.861 | 0.047 | Glucose-6-phosphate isomerase inhibitor | 0.047 0.035 CHEMBL3542351 | CHEMBL3542351 | |
| 0.008 | 0.864 | 0.094 | MAP kinase kinase 7 inhibitor | 0.094 0.019 CHEMBL3542351 0.075 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.006 | 0.862 | 0.054 | Potassium channel small-conductance Ca-activated blocker | 0.054 0.022 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.858 | 0.114 | MAO B inhibitor | 0.114 0.054 CHEMBL3542349 | CHEMBL3542349 | |
| 0.004 | 0.861 | 0.043 | Kainate receptor agonist | 0.043 0.024 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.86 | 0.079 | Na+ K+ transporting ATPase inhibitor | 0.079 0.051 CHEMBL3542350 | CHEMBL3542350 | |
| 0.005 | 0.864 | 0.273 | UDP-glucose 4-epimerase inhibitor | 0.11 0.051 CHEMBL3542349 0.273 0.012 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.86 | 0.025 | Integrin beta2 antagonist | 0.025 0.004 CHEMBL3542352 | CHEMBL3542352 | |
| 0.007 | 0.867 | 0.134 | Antipruritic | 0.134 0.116 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.863 | 0.113 | Diacylglycerol O-acyltransferase inhibitor | 0.097 0.008 CHEMBL3542351 0.113 0.005 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.865 | 0.39 | Pyruvate kinase inhibitor | 0.372 0.027 CHEMBL3542349 0.31 0.045 CHEMBL3542350 0.39 0.022 CHEMBL3542351 0.15 0.115 CHEMBL3542352 | CHEMBL3542351 | |
| 0.006 | 0.867 | 0.117 | Glycine receptor agonist | 0.068 0.059 CHEMBL3542350 0.117 0.014 CHEMBL3542351 0.067 0.062 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.864 | 0.078 | Prostaglandin-E synthase inhibitor | 0.078 0.04 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.864 | 0.102 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.102 0.016 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.868 | 0.286 | Succinate dehydrogenase inhibitor | 0.161 0.094 CHEMBL3542349 0.286 0.013 CHEMBL3542351 0.17 0.081 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.868 | 0.045 | Nicotinic acid receptor 1 agonist | 0.045 0.023 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.869 | 0.132 | Sphingosine 1-phosphate receptor 2 antagonist | 0.132 0.069 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.869 | 0.188 | Glycogen synthase kinase-3 alpha inhibitor | 0.129 0.079 CHEMBL3542349 0.152 0.065 CHEMBL3542350 0.188 0.045 CHEMBL3542351 | CHEMBL3542351 | |
| 0.009 | 0.876 | 0.207 | NADH dehydrogenase inhibitor | 0.081 0.072 CHEMBL3542349 0.207 0.01 CHEMBL3542351 0.096 0.049 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.871 | 0.038 | Complement factor 1s inhibitor | 0.038 0.004 CHEMBL3542349 0.024 0.021 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.87 | 0.141 | Dihydroorotase inhibitor | 0.141 0.004 CHEMBL3542351 0.042 0.034 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.869 | 0.045 | Acetylcholine M4 receptor agonist | 0.045 0.013 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.87 | 0.042 | Sphingosine 1-phosphate receptor agonist | 0.042 0.034 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.872 | 0.087 | Syk tyrosine kinase inhibitor | 0.087 0.035 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.874 | 0.179 | MAP kinase kinase 2 inhibitor | 0.179 0.097 CHEMBL3542351 0.146 0.125 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.872 | 0.051 | Dihydropteroate synthase inhibitor | 0.051 0.016 CHEMBL3542351 0.037 0.031 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.872 | 0.155 | Urate transporter 1 inhibitor | 0.155 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.875 | 0.227 | Cytidine deaminase inhibitor | 0.169 0.063 CHEMBL3542350 0.227 0.036 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.877 | 0.263 | Toll-Like receptor antagonist | 0.263 0.012 CHEMBL3542349 0.117 0.089 CHEMBL3542351 0.112 0.098 CHEMBL3988902 | CHEMBL3542349 | |
| 0.002 | 0.874 | 0.049 | Liver X receptor alpha agonist | 0.049 0.02 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.877 | 0.119 | Cyclooxygenase inhibitor | 0.119 0.1 CHEMBL3542350 | CHEMBL3542350 | |
| 0.004 | 0.876 | 0.108 | Bromodomain-containing protein 2 inhibitor | 0.089 0.056 CHEMBL3542349 0.103 0.037 CHEMBL3542350 0.108 0.032 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.875 | 0.114 | Cyclin-dependent kinase 9 inhibitor | 0.114 0.049 CHEMBL3542349 0.085 0.084 CHEMBL3542350 | CHEMBL3542349 | |
| 0.012 | 0.885 | 0.232 | Histone acetyltransferase inhibitor | 0.193 0.081 CHEMBL3542349 0.177 0.104 CHEMBL3542350 0.232 0.035 CHEMBL3542351 0.184 0.094 CHEMBL3542352 | CHEMBL3542351 | |
| 0.009 | 0.883 | 0.114 | Phosphodiesterase 6D inhibitor | 0.114 0.031 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.876 | 0.079 | Nerve growth factor antagonist | 0.044 0.027 CHEMBL3542349 0.079 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.01 | 0.887 | 0.118 | D-Ala-D-Ala ligase inhibitor | 0.118 0.014 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.879 | 0.036 | Liver X receptor beta agonist | 0.036 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.879 | 0.079 | Glutamate (mGluR3) antagonist | 0.079 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.88 | 0.057 | Glutamate (mGluR group I) agonist | 0.057 0.025 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.883 | 0.359 | GABA receptor agonist | 0.287 0.007 CHEMBL3542349 0.359 0.005 CHEMBL3542350 0.164 0.029 CHEMBL3542351 0.116 0.06 CHEMBL3542352 | CHEMBL3542350 | |
| 0.002 | 0.881 | 0.116 | GABA receptor antagonist | 0.116 0.013 CHEMBL3542349 0.059 0.033 CHEMBL3542351 | CHEMBL3542349 | |
| 0.001 | 0.881 | 0.042 | Alpha 1d adrenoreceptor agonist | 0.042 0.023 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.884 | 0.312 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.162 0.129 CHEMBL3542350 0.312 0.061 CHEMBL3542351 0.156 0.135 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.885 | 0.056 | Glutamate (mGluR8) agonist | 0.056 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.885 | 0.07 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.07 0.021 CHEMBL3542349 0.062 0.027 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.885 | 0.075 | Purinergic P2X4 antagonist | 0.075 0.008 CHEMBL3542349 0.052 0.022 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.884 | 0.697 | Aryl hydrocarbon receptor agonist | 0.697 0.009 CHEMBL3542349 0.418 0.034 CHEMBL3542350 0.42 0.034 CHEMBL3542351 0.177 0.116 CHEMBL3542352 | CHEMBL3542349 | |
| 0.003 | 0.886 | 0.059 | Dopamine beta hydroxylase inhibitor | 0.047 0.036 CHEMBL3542349 0.059 0.016 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.888 | 0.189 | 5 Hydroxytryptamine 1E antagonist | 0.189 0.143 CHEMBL3542349 | CHEMBL3542349 | |
| 0.002 | 0.886 | 0.095 | Alpha 2 adrenoreceptor agonist | 0.057 0.046 CHEMBL3542349 0.095 0.016 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.887 | 0.179 | Tyrosine-protein kinase receptor antagonist | 0.179 0.05 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.885 | 0.073 | Retinoid X receptor agonist | 0.073 0.009 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.887 | 0.116 | GABA A receptor antagonist | 0.116 0.013 CHEMBL3542349 0.054 0.036 CHEMBL3542351 | CHEMBL3542349 | |
| 0.005 | 0.89 | 0.065 | Phosphodiesterase 1A inhibitor | 0.065 0.031 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.887 | 0.135 | Sphingosine 1-phosphate receptor 4 agonist | 0.135 0.012 CHEMBL3542349 0.061 0.053 CHEMBL3542351 0.115 0.018 CHEMBL3542352 | CHEMBL3542349 | |
| 0.022 | 0.908 | 0.104 | Glutamate release inhibitor | 0.104 0.037 CHEMBL3542351 | CHEMBL3542351 | |
| 0.007 | 0.894 | 0.321 | Transcription factor inhibitor | 0.261 0.179 CHEMBL3542349 0.321 0.144 CHEMBL3542350 0.225 0.205 CHEMBL3542351 | CHEMBL3542350 | |
| 0.004 | 0.891 | 0.078 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.078 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.889 | 0.168 | Benzodiazepine agonist | 0.133 0.012 CHEMBL3542349 0.168 0.005 CHEMBL3542350 0.073 0.047 CHEMBL3542351 | CHEMBL3542350 | |
| 0.003 | 0.891 | 0.056 | Ryanodine receptor antagonist | 0.056 0.049 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.889 | 0.169 | Dihydroorotate dehydrogenase inhibitor | 0.062 0.027 CHEMBL3542349 0.169 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0 | 0.888 | 0.035 | Alpha 2a adrenoreceptor agonist | 0.035 0.005 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.889 | 0.051 | NMDA receptor subunit 3A antagonist | 0.051 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.011 | 0.899 | 0.296 | Hexokinase inhibitor | 0.296 0.011 CHEMBL3542351 0.13 0.105 CHEMBL3542352 | CHEMBL3542351 | |
| 0.005 | 0.893 | 0.22 | Thioredoxin glutathione reductase inhibitor | 0.22 0.155 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.892 | 0.344 | GABA A receptor agonist | 0.268 0.005 CHEMBL3542349 0.344 0.004 CHEMBL3542350 0.113 0.028 CHEMBL3542351 0.079 0.066 CHEMBL3542352 | CHEMBL3542350 | |
| 0.002 | 0.892 | 0.091 | NMDA receptor antagonist | 0.091 0.053 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.894 | 0.251 | Creatine kinase inhibitor | 0.1 0.059 CHEMBL3542349 0.251 0.005 CHEMBL3542351 0.085 0.079 CHEMBL3542352 | CHEMBL3542351 | |
| 0.004 | 0.895 | 0.119 | Glutamate (mGluR4) antagonist | 0.053 0.018 CHEMBL3542349 0.119 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.895 | 0.092 | Bcr-Abl kinase inhibitor | 0.092 0.049 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.896 | 0.194 | Focal adhesion kinase 2 inhibitor | 0.194 0.074 CHEMBL3542349 0.151 0.129 CHEMBL3542350 0.188 0.079 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.897 | 0.14 | Cyclin-dependent kinase 8 inhibitor | 0.128 0.105 CHEMBL3542349 0.14 0.09 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.896 | 0.264 | Lipoxygenase inhibitor | 0.193 0.148 CHEMBL3542349 0.264 0.091 CHEMBL3542350 0.247 0.102 CHEMBL3542351 | CHEMBL3542350 | |
| 0.002 | 0.896 | 0.066 | Orexin receptor antagonist | 0.066 0.046 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.895 | 0.02 | Glutamate (mGluR1a) agonist | 0.02 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.895 | 0.034 | Orexin receptor 2 antagonist | 0.034 0.028 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.895 | 0.047 | Glycine transporter inhibitor | 0.047 0.034 CHEMBL3542352 | CHEMBL3542352 | |
| 0.001 | 0.895 | 0.031 | Retinoid X beta receptor antagonist | 0.031 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.896 | 0.035 | Carnitine palmitoyltransferase inhibitor | 0.035 0.023 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.897 | 0.075 | RNA-directed RNA polymerase inhibitor | 0.075 0.007 CHEMBL3542351 0.046 0.015 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.898 | 0.203 | Glutamate receptor agonist | 0.104 0.035 CHEMBL3542349 0.203 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.9 | 0.177 | Nitric-oxide synthase inhibitor | 0.177 0.014 CHEMBL3988901 0.092 0.073 CHEMBL3988902 | CHEMBL3988901 | |
| 0.001 | 0.898 | 0.079 | NMDA 2 receptor antagonist | 0.079 0.044 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.899 | 0.091 | Nicotinic alpha4beta2 receptor antagonist | 0.085 0.045 CHEMBL3542349 0.085 0.045 CHEMBL3542350 0.091 0.039 CHEMBL3542351 | CHEMBL3542351 | |
| 0.006 | 0.904 | 0.443 | Hypoxia-inducible factor 1 alpha inhibitor | 0.239 0.111 CHEMBL3542349 0.443 0.021 CHEMBL3542350 0.348 0.045 CHEMBL3542351 0.34 0.048 CHEMBL3542352 | CHEMBL3542350 | |
| 0.033 | 0.931 | 0.217 | 5 Hydroxytryptamine 3E antagonist | 0.217 0.039 CHEMBL3542349 0.173 0.126 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.901 | 0.089 | Histamine H1 receptor antagonist | 0.089 0.049 CHEMBL3542351 | CHEMBL3542351 | |
| 0.011 | 0.91 | 0.171 | CF transmembrane conductance regulator agonist | 0.157 0.064 CHEMBL3542349 0.171 0.045 CHEMBL3542351 0.157 0.064 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.9 | 0.084 | Retinoid X alpha receptor agonist | 0.084 0.007 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.902 | 0.083 | Orexin receptor 1 antagonist | 0.083 0.031 CHEMBL3542349 0.077 0.04 CHEMBL3542350 | CHEMBL3542349 | |
| 0.002 | 0.903 | 0.072 | Phosphodiesterase 4B inhibitor | 0.072 0.042 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.904 | 0.052 | Retinoid X alpha receptor antagonist | 0.052 0.005 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.903 | 0.039 | Calcium release-activated channel blocker | 0.039 0.016 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.905 | 0.151 | MAP kinase kinase 1 inhibitor | 0.151 0.016 CHEMBL3542350 0.11 0.046 CHEMBL3542351 | CHEMBL3542350 | |
| 0.008 | 0.91 | 0.168 | DNA repair enzyme inhibitor | 0.168 0.019 CHEMBL3542350 0.131 0.053 CHEMBL3542351 | CHEMBL3542350 | |
| 0.008 | 0.911 | 0.172 | NADPH oxidase inhibitor | 0.172 0.043 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.907 | 0.06 | Retinoid X receptor antagonist | 0.06 0.006 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.906 | 0.107 | Granulocyte macrophage colony stimulating factor antagonist | 0.107 0.064 CHEMBL3542350 | CHEMBL3542350 | |
| 0.006 | 0.911 | 0.219 | Cell wall synthesis inhibitor | 0.154 0.062 CHEMBL3542350 0.199 0.03 CHEMBL3542351 0.195 0.032 CHEMBL3988901 0.127 0.09 CHEMBL3542352 0.219 0.023 CHEMBL3988902 | CHEMBL3988902 | |
| 0.002 | 0.907 | 0.137 | Nicotinic acid receptor agonist | 0.044 0.018 CHEMBL3542349 0.137 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.91 | 0.099 | Glutamate (mGluR6) antagonist | 0.099 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.908 | 0.098 | Alpha adrenoreceptor agonist | 0.098 0.029 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.908 | 0.067 | Stearoyl-CoA desaturase inhibitor | 0.067 0.015 CHEMBL3542352 | CHEMBL3542352 | |
| 0.004 | 0.912 | 0.134 | 5 Hydroxytryptamine 3 agonist | 0.134 0.006 CHEMBL3542349 0.072 0.034 CHEMBL3542351 | CHEMBL3542349 | |
| 0 | 0.909 | 0.027 | Nicotinic alpha3beta4 receptor agonist | 0.027 0.026 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.912 | 0.142 | Glutamate (mGluR group III) antagonist | 0.056 0.015 CHEMBL3542349 0.142 0.004 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.911 | 0.035 | Carnitine palmitoyltransferase 1 inhibitor | 0.035 0.022 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.911 | 0.037 | LFA antagonist | 0.031 0.014 CHEMBL3542351 0.037 0.009 CHEMBL3542352 | CHEMBL3542352 | |
| 0.008 | 0.919 | 0.287 | Antiinflammatory | 0.287 0.228 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.916 | 0.206 | Thyroid hormone antagonist | 0.206 0.157 CHEMBL3542352 | CHEMBL3542352 | |
| 0.003 | 0.915 | 0.257 | I kappa B kinase epsilon inhibitor | 0.141 0.129 CHEMBL3542350 0.257 0.034 CHEMBL3542351 0.137 0.134 CHEMBL3542352 | CHEMBL3542351 | |
| 0.003 | 0.915 | 0.26 | Heat shock protein 90 alpha antagonist | 0.26 0.023 CHEMBL3542349 0.185 0.059 CHEMBL3542350 0.228 0.035 CHEMBL3542351 0.133 0.107 CHEMBL3542352 | CHEMBL3542349 | |
| 0.003 | 0.915 | 0.083 | Phosphodiesterase 1C inhibitor | 0.083 0.017 CHEMBL3542351 | CHEMBL3542351 | |
| 0.005 | 0.917 | 0.195 | Thyroid hormone beta antagonist | 0.195 0.158 CHEMBL3542352 | CHEMBL3542352 | |
| 0 | 0.913 | 0.031 | Uridine phosphorylase inhibitor | 0.031 0.017 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.915 | 0.175 | Phosphodiesterase IV inhibitor | 0.175 0.017 CHEMBL3542350 0.105 0.041 CHEMBL3542351 | CHEMBL3542350 | |
| 0.003 | 0.917 | 0.203 | Anticonvulsant | 0.203 0.08 CHEMBL3542350 0.146 0.135 CHEMBL3542352 | CHEMBL3542350 | |
| 0.002 | 0.917 | 0.047 | Potassium channel (ATP-sensitive) activator | 0.047 0.035 CHEMBL3542349 | CHEMBL3542349 | |
| 0.002 | 0.917 | 0.05 | Potassium channel (Inward rectifier) activator | 0.05 0.037 CHEMBL3542349 | CHEMBL3542349 | |
| 0.004 | 0.919 | 0.237 | Non-steroidal antiinflammatory agent | 0.237 0.049 CHEMBL3542351 0.146 0.121 CHEMBL3542352 | CHEMBL3542351 | |
| 0.002 | 0.917 | 0.085 | Acetylcholine nicotinic agonist | 0.085 0.05 CHEMBL3542349 0.081 0.056 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.918 | 0.188 | Toll-Like receptor 9 antagonist | 0.188 0.041 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.919 | 0.1 | Cholinergic antagonist | 0.1 0.096 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.918 | 0.062 | Nicotinic alpha7 receptor agonist | 0.062 0.03 CHEMBL3542349 | CHEMBL3542349 | |
| 0.002 | 0.92 | 0.171 | MAP kinase kinase inhibitor | 0.171 0.04 CHEMBL3542350 0.128 0.067 CHEMBL3542351 | CHEMBL3542350 | |
| 0.005 | 0.923 | 0.065 | Phosphodiesterase 1B inhibitor | 0.065 0.035 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.922 | 0.18 | Heat shock protein 90 antagonist | 0.18 0.049 CHEMBL3542349 0.133 0.093 CHEMBL3542350 0.151 0.074 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.922 | 0.324 | DNA polymerase beta inhibitor | 0.324 0.153 CHEMBL3542349 0.219 0.211 CHEMBL3542350 0.236 0.201 CHEMBL3542351 | CHEMBL3542349 | |
| 0.005 | 0.924 | 0.376 | MAP kinase 1 inhibitor | 0.376 0.121 CHEMBL3542349 0.328 0.152 CHEMBL3542350 0.314 0.166 CHEMBL3542351 0.281 0.201 CHEMBL3542352 | CHEMBL3542349 | |
| 0.001 | 0.92 | 0.06 | HCV NS5B polymerase inhibitor | 0.06 0.008 CHEMBL3542351 0.032 0.021 CHEMBL3542352 | CHEMBL3542351 | |
| 0.001 | 0.921 | 0.053 | Nicotinic neuronal receptor agonist | 0.053 0.042 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.921 | 0.07 | Acetylcholine M5 receptor agonist | 0.07 0.044 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.921 | 0.045 | Fructose-1,6-bisphosphatase inhibitor | 0.045 0.031 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.922 | 0.048 | Glutamate (mGluR5) agonist | 0.048 0.028 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.923 | 0.056 | Alpha 1 adrenoreceptor agonist | 0.056 0.042 CHEMBL3542350 | CHEMBL3542350 | |
| 0.003 | 0.926 | 0.143 | Pregnane X receptor agonist | 0.138 0.078 CHEMBL3542349 0.143 0.067 CHEMBL3542350 0.134 0.09 CHEMBL3542351 | CHEMBL3542350 | |
| 0.002 | 0.925 | 0.137 | Inducible nitric-oxide synthase inhibitor | 0.137 0.019 CHEMBL3988901 0.074 0.073 CHEMBL3988902 | CHEMBL3988901 | |
| 0.001 | 0.924 | 0.042 | Glutamate (mGluR2) antagonist | 0.042 0.011 CHEMBL3542351 | CHEMBL3542351 | |
| 0.004 | 0.928 | 0.097 | Phosphodiesterase I inhibitor | 0.097 0.049 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.926 | 0.064 | Glutamate (mGluR group II) antagonist | 0.064 0.01 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.929 | 0.1 | 5 Hydroxytryptamine 3A agonist | 0.1 0.076 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.931 | 0.183 | Sphingosine 1-phosphate receptor 5 antagonist | 0.183 0.021 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.929 | 0.095 | 5 Hydroxytryptamine 1D antagonist | 0.095 0.024 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.932 | 0.172 | Acetylcholine M1 receptor antagonist | 0.172 0.057 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.93 | 0.129 | Aromatase inhibitor | 0.129 0.016 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.93 | 0.064 | 5 Hydroxytryptamine 1B antagonist | 0.064 0.046 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.931 | 0.058 | Dopamine D3 antagonist | 0.058 0.047 CHEMBL3542349 | CHEMBL3542349 | |
| 0.003 | 0.933 | 0.249 | Alpha-glucosidase inhibitor | 0.244 0.191 CHEMBL3542349 0.249 0.188 CHEMBL3542350 | CHEMBL3542350 | |
| 0.004 | 0.934 | 0.068 | Dihydroorotate oxidase inhibitor | 0.068 0.019 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.933 | 0.076 | Acetylcholine M5 receptor antagonist | 0.076 0.026 CHEMBL3542350 | CHEMBL3542350 | |
| 0.001 | 0.933 | 0.118 | Acetylcholine muscarinic agonist | 0.118 0.014 CHEMBL3542350 | CHEMBL3542350 | |
| 0.002 | 0.936 | 0.202 | Acetylcholine agonist | 0.202 0.014 CHEMBL3542350 | CHEMBL3542350 | |
| 0.003 | 0.938 | 0.28 | DNA directed DNA polymerase inhibitor | 0.28 0.173 CHEMBL3542349 0.22 0.212 CHEMBL3542351 | CHEMBL3542349 | |
| 0.002 | 0.937 | 0.184 | Prostaglandin dehydrogenase inhibitor | 0.184 0.168 CHEMBL3542349 | CHEMBL3542349 | |
| 0.001 | 0.937 | 0.074 | Acetylcholine M1 receptor agonist | 0.074 0.018 CHEMBL3542350 | CHEMBL3542350 | |
| 0.01 | 0.947 | 0.182 | Ca2+-transporting ATPase inhibitor | 0.14 0.072 CHEMBL3542349 0.182 0.006 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.939 | 0.127 | Acetylcholine M4 receptor antagonist | 0.091 0.036 CHEMBL3542349 0.127 0.016 CHEMBL3542350 | CHEMBL3542350 | |
| 0.009 | 0.947 | 0.255 | RNA-directed DNA polymerase inhibitor | 0.192 0.112 CHEMBL3542349 0.255 0.047 CHEMBL3542351 | CHEMBL3542351 | |
| 0.001 | 0.943 | 0.052 | Purinergic P2Y antagonist | 0.052 0.025 CHEMBL3542351 | CHEMBL3542351 | |
| 0.003 | 0.947 | 0.347 | 15-Lipoxygenase inhibitor | 0.347 0.101 CHEMBL3542349 0.298 0.134 CHEMBL3542350 0.313 0.123 CHEMBL3542351 | CHEMBL3542349 | |
| 0.003 | 0.957 | 0.143 | AMP-activated protein kinase stimulant | 0.143 0.033 CHEMBL3542351 | CHEMBL3542351 | |
| 0.002 | 0.96 | 0.07 | Estrogen receptor alpha antagonist | 0.07 0.068 CHEMBL3542349 | CHEMBL3542349 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |