| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.846 | 0.003 | 0.846 | Cyclooxygenase inhibitor | 0.776 0.003 CHEMBL745 0.766 0.003 CHEMBL743 0.608 0.004 CHEMBL3544878 | ||
| 0.82 | 0.003 | 0.82 | Cyclooxygenase 2 inhibitor | 0.738 0.003 CHEMBL745 0.722 0.003 CHEMBL743 0.544 0.004 CHEMBL3544878 | ||
| 0.811 | 0.003 | 0.98 | Non-steroidal antiinflammatory agent | 0.838 0.003 CHEMBL745 0.886 0.003 CHEMBL743 0.98 0.002 CHEMBL3544878 | CHEMBL3544878 | |
| 0.78 | 0.003 | 0.78 | Cyclooxygenase 1 inhibitor | 0.732 0.004 CHEMBL745 0.727 0.004 CHEMBL743 0.577 0.004 CHEMBL3544878 | ||
| 0.681 | 0.002 | 0.932 | Carbonic anhydrase XV inhibitor | 0.929 0.001 CHEMBL745 0.932 0.001 CHEMBL743 0.257 0.011 CHEMBL3544878 | CHEMBL743 | |
| 0.593 | 0.003 | 0.758 | Carbonic anhydrase III inhibitor | 0.722 0.002 CHEMBL745 0.758 0.002 CHEMBL743 0.478 0.003 CHEMBL3544878 | CHEMBL743 | |
| 0.537 | 0.003 | 0.811 | Carbonic anhydrase VI inhibitor | 0.811 0.002 CHEMBL745 0.807 0.002 CHEMBL743 0.474 0.003 CHEMBL3544878 | CHEMBL745 | |
| 0.51 | 0.003 | 0.555 | Carbonic anhydrase IX inhibitor | 0.495 0.003 CHEMBL745 0.526 0.003 CHEMBL743 0.555 0.003 CHEMBL3544878 | CHEMBL3544878 | |
| 0.567 | 0.063 | 0.818 | Antiinflammatory | 0.631 0.045 CHEMBL745 0.611 0.05 CHEMBL743 0.818 0.013 CHEMBL3544878 | CHEMBL3544878 | |
| 0.464 | 0.003 | 0.568 | Carbonic anhydrase inhibitor | 0.467 0.003 CHEMBL745 0.537 0.003 CHEMBL743 0.568 0.003 CHEMBL3544878 | CHEMBL3544878 | |
| 0.479 | 0.056 | 0.479 | Analgesic | 0.411 0.08 CHEMBL745 0.429 0.073 CHEMBL743 0.257 0.177 CHEMBL3544878 | ||
| 0.422 | 0.012 | 0.548 | Diuretic | 0.306 0.021 CHEMBL745 0.548 0.005 CHEMBL743 0.5 0.008 CHEMBL3544878 | CHEMBL743 | |
| 0.414 | 0.004 | 0.57 | Carbonic anhydrase XII inhibitor | 0.397 0.004 CHEMBL745 0.479 0.003 CHEMBL743 0.57 0.003 CHEMBL3544878 | CHEMBL3544878 | |
| 0.403 | 0.004 | 0.66 | Carbonic anhydrase XIII inhibitor | 0.66 0.003 CHEMBL745 0.66 0.003 CHEMBL743 0.395 0.004 CHEMBL3544878 | CHEMBL743 | |
| 0.401 | 0.004 | 0.401 | Sodium channel (voltage-gated) blocker | 0.37 0.005 CHEMBL745 0.288 0.009 CHEMBL743 | ||
| 0.399 | 0.005 | 0.399 | Alkaline phosphatase inhibitor | 0.296 0.012 CHEMBL745 0.397 0.005 CHEMBL743 0.36 0.007 CHEMBL3544878 | ||
| 0.386 | 0.002 | 0.525 | Carbonic anhydrase VB inhibitor | 0.525 0.002 CHEMBL745 0.462 0.002 CHEMBL743 0.077 0.024 CHEMBL3544878 | CHEMBL745 | |
| 0.377 | 0.005 | 0.377 | Sodium channel blocker | 0.329 0.008 CHEMBL745 0.223 0.025 CHEMBL743 | ||
| 0.35 | 0.005 | 0.357 | Cyclin-dependent kinase 3 inhibitor | 0.357 0.005 CHEMBL745 0.325 0.006 CHEMBL743 0.215 0.026 CHEMBL3544878 | CHEMBL745 | |
| 0.392 | 0.047 | 0.469 | Caspase 3 stimulant | 0.426 0.037 CHEMBL745 0.361 0.056 CHEMBL743 0.469 0.025 CHEMBL3544878 | CHEMBL3544878 | |
| 0.337 | 0.004 | 0.413 | Carbonic anhydrase I inhibitor | 0.323 0.004 CHEMBL745 0.413 0.003 CHEMBL743 0.329 0.004 CHEMBL3544878 | CHEMBL743 | |
| 0.373 | 0.044 | 0.421 | Lipoxygenase inhibitor | 0.421 0.032 CHEMBL745 0.406 0.036 CHEMBL743 | CHEMBL745 | |
| 0.333 | 0.004 | 0.378 | Carbonic anhydrase II inhibitor | 0.324 0.004 CHEMBL745 0.378 0.003 CHEMBL743 0.335 0.004 CHEMBL3544878 | CHEMBL743 | |
| 0.329 | 0.004 | 0.329 | Interleukin 2 antagonist | 0.247 0.005 CHEMBL745 0.264 0.005 CHEMBL743 0.168 0.012 CHEMBL3544878 | ||
| 0.319 | 0.003 | 0.465 | Carbonic anhydrase V inhibitor | 0.465 0.003 CHEMBL745 0.394 0.003 CHEMBL743 0.091 0.03 CHEMBL3544878 | CHEMBL745 | |
| 0.297 | 0.003 | 0.401 | Carbonic anhydrase VA inhibitor | 0.401 0.003 CHEMBL745 0.369 0.003 CHEMBL743 0.101 0.024 CHEMBL3544878 | CHEMBL745 | |
| 0.25 | 0.004 | 0.25 | Nav1.7 sodium channel blocker | 0.219 0.005 CHEMBL745 0.132 0.014 CHEMBL743 | ||
| 0.298 | 0.055 | 0.326 | Transcription factor STAT3 inhibitor | 0.272 0.068 CHEMBL745 0.326 0.042 CHEMBL743 0.2 0.133 CHEMBL3544878 | CHEMBL743 | |
| 0.277 | 0.044 | 0.277 | EphB2 antagonist | 0.158 0.122 CHEMBL745 0.201 0.087 CHEMBL743 | ||
| 0.218 | 0.005 | 0.241 | Interleukin 5 antagonist | 0.232 0.005 CHEMBL745 0.241 0.005 CHEMBL743 0.158 0.009 CHEMBL3544878 | CHEMBL743 | |
| 0.277 | 0.069 | 0.289 | Transcription factor STAT inhibitor | 0.23 0.102 CHEMBL745 0.289 0.063 CHEMBL743 | CHEMBL743 | |
| 0.276 | 0.071 | 0.276 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.215 0.091 CHEMBL743 | ||
| 0.206 | 0.007 | 0.412 | Electrolyte absorption antagonist | 0.165 0.014 CHEMBL745 0.412 0.003 CHEMBL743 | CHEMBL743 | |
| 0.213 | 0.014 | 0.213 | Ca(v)2.2 blocker | 0.131 0.035 CHEMBL745 0.134 0.034 CHEMBL743 | ||
| 0.216 | 0.021 | 0.223 | 5-Lipoxygenase inhibitor | 0.223 0.02 CHEMBL745 0.22 0.021 CHEMBL743 | CHEMBL745 | |
| 0.21 | 0.02 | 0.249 | Interleukin 4 antagonist | 0.207 0.02 CHEMBL745 0.249 0.013 CHEMBL743 0.225 0.017 CHEMBL3544878 | CHEMBL743 | |
| 0.233 | 0.047 | 0.233 | Focal adhesion kinase 2 inhibitor | 0.149 0.133 CHEMBL745 0.172 0.097 CHEMBL743 | ||
| 0.202 | 0.02 | 0.205 | CF transmembrane conductance regulator agonist | 0.205 0.019 CHEMBL745 0.149 0.078 CHEMBL743 0.148 0.08 CHEMBL3544878 | CHEMBL745 | |
| 0.221 | 0.044 | 0.221 | Histone acetyltransferase inhibitor | 0.16 0.125 CHEMBL745 0.213 0.051 CHEMBL743 | ||
| 0.174 | 0.007 | 0.18 | Factor Xa inhibitor | 0.118 0.011 CHEMBL745 0.163 0.008 CHEMBL743 0.18 0.007 CHEMBL3544878 | CHEMBL3544878 | |
| 0.166 | 0.006 | 0.166 | Factor X inhibitor | 0.125 0.008 CHEMBL745 0.129 0.008 CHEMBL743 0.059 0.018 CHEMBL3544878 | ||
| 0.165 | 0.005 | 0.228 | Carbonic anhydrase VII inhibitor | 0.155 0.006 CHEMBL745 0.228 0.004 CHEMBL743 0.052 0.025 CHEMBL3544878 | CHEMBL743 | |
| 0.158 | 0.013 | 0.158 | Nav1.8 sodium channel blocker | 0.142 0.015 CHEMBL745 0.155 0.013 CHEMBL743 | ||
| 0.144 | 0.005 | 0.144 | Aldosterone antagonist | 0.06 0.02 CHEMBL745 0.097 0.008 CHEMBL743 | ||
| 0.163 | 0.025 | 0.187 | Heat shock protein 70 antagonist | 0.158 0.03 CHEMBL745 0.187 0.009 CHEMBL743 0.153 0.039 CHEMBL3544878 | CHEMBL743 | |
| 0.144 | 0.013 | 0.17 | Prostaglandin-E synthase inhibitor | 0.134 0.015 CHEMBL745 0.17 0.009 CHEMBL743 | CHEMBL743 | |
| 0.16 | 0.038 | 0.16 | Pregnane X receptor agonist | 0.132 0.094 CHEMBL745 | ||
| 0.129 | 0.01 | 0.129 | Cannabinoid CB1 receptor antagonist | 0.08 0.027 CHEMBL745 | ||
| 0.124 | 0.005 | 0.148 | Carbonic anhydrase IV inhibitor | 0.128 0.004 CHEMBL745 0.148 0.004 CHEMBL743 0.04 0.033 CHEMBL3544878 | CHEMBL743 | |
| 0.123 | 0.007 | 0.424 | Carbonic anhydrase XIV inhibitor | 0.249 0.004 CHEMBL745 0.323 0.003 CHEMBL743 0.424 0.003 CHEMBL3544878 | CHEMBL3544878 | |
| 0.134 | 0.019 | 0.159 | Phosphodiesterase 3A inhibitor | 0.159 0.014 CHEMBL745 0.092 0.04 CHEMBL743 | CHEMBL745 | |
| 0.168 | 0.054 | 0.168 | Activin receptor-like kinase 2 inhibitor | 0.148 0.068 CHEMBL745 | ||
| 0.132 | 0.021 | 0.152 | I kappa B kinase inhibitor | 0.152 0.016 CHEMBL745 0.126 0.024 CHEMBL743 | CHEMBL745 | |
| 0.148 | 0.039 | 0.148 | Calcium channel N-type blocker | 0.103 0.089 CHEMBL745 0.113 0.073 CHEMBL743 | ||
| 0.272 | 0.164 | 0.272 | MAP kinase kinase 6 inhibitor | 0.234 0.213 CHEMBL743 | ||
| 0.145 | 0.043 | 0.145 | Cyclin-dependent kinase 1 inhibitor | 0.129 0.05 CHEMBL745 0.088 0.075 CHEMBL743 | ||
| 0.104 | 0.005 | 0.104 | Purinergic P2X4 antagonist | 0.094 0.005 CHEMBL745 0.091 0.005 CHEMBL743 | ||
| 0.133 | 0.034 | 0.133 | CDK2/cyclin A inhibitor | 0.113 0.048 CHEMBL745 0.096 0.061 CHEMBL743 | ||
| 0.114 | 0.014 | 0.114 | Potassium channel Kv1.5 blocker | 0.068 0.03 CHEMBL745 0.05 0.048 CHEMBL743 | ||
| 0.12 | 0.022 | 0.12 | Cannabinoid receptor antagonist | |||
| 0.104 | 0.011 | 0.12 | I kappa B kinase 2 inhibitor | 0.12 0.008 CHEMBL745 0.092 0.016 CHEMBL743 | CHEMBL745 | |
| 0.136 | 0.044 | 0.136 | Cyclin-dependent kinase 2 inhibitor | 0.107 0.063 CHEMBL745 0.093 0.078 CHEMBL743 | ||
| 0.147 | 0.058 | 0.147 | Nav1.6 sodium channel blocker | 0.117 0.101 CHEMBL745 | ||
| 0.13 | 0.041 | 0.13 | Sphingosine 1-phosphate receptor 2 agonist | 0.114 0.066 CHEMBL745 0.108 0.079 CHEMBL743 | ||
| 0.103 | 0.02 | 0.103 | Ca(v)3.1 blocker | 0.079 0.064 CHEMBL745 0.08 0.059 CHEMBL743 | ||
| 0.147 | 0.067 | 0.163 | MAP kinase kinase 4 inhibitor | 0.146 0.07 CHEMBL745 0.163 0.04 CHEMBL743 | CHEMBL743 | |
| 0.098 | 0.024 | 0.098 | CC chemokine 5 receptor agonist | |||
| 0.152 | 0.078 | 0.301 | Anticoagulant | 0.163 0.07 CHEMBL745 0.194 0.055 CHEMBL743 0.301 0.028 CHEMBL3544878 | CHEMBL3544878 | |
| 0.124 | 0.05 | 0.124 | CDK3/cyclin E inhibitor | 0.123 0.052 CHEMBL745 0.123 0.051 CHEMBL743 | ||
| 0.243 | 0.17 | 0.243 | 15-Lipoxygenase inhibitor | 0.226 0.186 CHEMBL743 | ||
| 0.109 | 0.038 | 0.148 | Phosphodiesterase 6D inhibitor | 0.1 0.051 CHEMBL745 0.1 0.051 CHEMBL743 0.148 0.01 CHEMBL3544878 | CHEMBL3544878 | |
| 0.113 | 0.046 | 0.179 | Creatine kinase inhibitor | 0.091 0.07 CHEMBL745 0.179 0.014 CHEMBL743 | CHEMBL743 | |
| 0.078 | 0.012 | 0.078 | Mineralocorticoid receptor antagonist | 0.06 0.02 CHEMBL745 0.07 0.014 CHEMBL743 | ||
| 0.082 | 0.017 | 0.082 | Cyclin H inhibitor | 0.069 0.03 CHEMBL745 0.065 0.034 CHEMBL743 | ||
| 0.11 | 0.045 | 0.113 | Phosphodiesterase 7B inhibitor | 0.089 0.071 CHEMBL745 0.113 0.043 CHEMBL743 | CHEMBL743 | |
| 0.064 | 0.005 | 0.064 | AMPA receptor agonist | 0.064 0.005 CHEMBL745 0.063 0.005 CHEMBL743 0.038 0.02 CHEMBL3544878 | ||
| 0.081 | 0.022 | 0.096 | Nitric oxide donor | 0.081 0.021 CHEMBL745 0.085 0.018 CHEMBL743 0.096 0.011 CHEMBL3544878 | CHEMBL3544878 | |
| 0.227 | 0.17 | 0.307 | Toll-Like receptor 7 agonist | 0.307 0.106 CHEMBL745 0.306 0.106 CHEMBL743 | CHEMBL745 | |
| 0.098 | 0.043 | 0.098 | Bromodomain-containing protein 2 inhibitor | |||
| 0.149 | 0.095 | 0.159 | Antipruritic | 0.159 0.084 CHEMBL743 | CHEMBL743 | |
| 0.203 | 0.151 | 0.203 | Thyroid hormone beta antagonist | |||
| 0.058 | 0.006 | 0.125 | Liver X receptor beta antagonist | 0.125 0.003 CHEMBL745 0.079 0.004 CHEMBL743 | CHEMBL745 | |
| 0.123 | 0.072 | 0.123 | Cathepsin H inhibitor | 0.121 0.074 CHEMBL743 | ||
| 0.132 | 0.083 | 0.14 | Mannose-6-phosphate isomerase inhibitor | 0.12 0.1 CHEMBL745 0.14 0.074 CHEMBL743 0.134 0.08 CHEMBL3544878 | CHEMBL743 | |
| 0.085 | 0.037 | 0.092 | Epoxide hydrolase inhibitor | 0.064 0.062 CHEMBL745 0.092 0.03 CHEMBL743 | CHEMBL743 | |
| 0.072 | 0.027 | 0.072 | Transcription factor RelA inhibitor | |||
| 0.055 | 0.009 | 0.122 | Liver X receptor beta agonist | 0.122 0.004 CHEMBL745 0.063 0.008 CHEMBL743 | CHEMBL745 | |
| 0.081 | 0.036 | 0.094 | Phosphodiesterase 4B inhibitor | 0.094 0.028 CHEMBL745 0.091 0.029 CHEMBL743 | CHEMBL745 | |
| 0.134 | 0.092 | 0.164 | Sphingosine 1-phosphate receptor 5 antagonist | 0.164 0.041 CHEMBL743 | CHEMBL743 | |
| 0.062 | 0.02 | 0.062 | Carbonic anhydrase II stimulant | 0.053 0.033 CHEMBL745 0.055 0.03 CHEMBL743 | ||
| 0.067 | 0.027 | 0.067 | Ca(v)3.2 blocker | |||
| 0.052 | 0.014 | 0.052 | Glucocorticoid antagonist | 0.032 0.023 CHEMBL745 0.029 0.024 CHEMBL743 | ||
| 0.279 | 0.243 | 0.279 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | |||
| 0.046 | 0.011 | 0.073 | Liver X receptor antagonist | 0.073 0.006 CHEMBL745 0.049 0.01 CHEMBL743 | CHEMBL745 | |
| 0.151 | 0.117 | 0.17 | Interleukin antagonist | 0.155 0.114 CHEMBL745 0.17 0.104 CHEMBL743 | CHEMBL743 | |
| 0.08 | 0.046 | 0.088 | Sphingosine 1-phosphate receptor antagonist | 0.085 0.037 CHEMBL745 0.088 0.033 CHEMBL743 | CHEMBL743 | |
| 0.075 | 0.042 | 0.075 | ZAP-70 protein tyrosine kinase inhibitor | 0.065 0.054 CHEMBL745 | ||
| 0.093 | 0.062 | 0.201 | Potassium channel (Ca-activated) activator | 0.201 0.014 CHEMBL743 | CHEMBL743 | |
| 0.052 | 0.021 | 0.07 | Liver X receptor agonist | 0.07 0.013 CHEMBL745 0.051 0.022 CHEMBL743 | CHEMBL745 | |
| 0.137 | 0.108 | 0.212 | Dual specificity phosphatase 3 inhibitor | 0.155 0.092 CHEMBL745 0.212 0.055 CHEMBL743 | CHEMBL743 | |
| 0.069 | 0.04 | 0.069 | Aryl hydrocarbon receptor antagonist | |||
| 0.214 | 0.185 | 0.303 | Toll-Like receptor agonist | 0.303 0.109 CHEMBL745 0.292 0.116 CHEMBL743 | CHEMBL745 | |
| 0.064 | 0.036 | 0.064 | Carbonic anhydrase stimulant | |||
| 0.059 | 0.032 | 0.07 | Sphingosine 1-phosphate receptor 1 antagonist | 0.07 0.018 CHEMBL745 0.065 0.022 CHEMBL743 | CHEMBL745 | |
| 0.176 | 0.15 | 0.176 | Streptokinase A inhibitor | |||
| 0.121 | 0.095 | 0.126 | Sphingosine 1-phosphate receptor 2 antagonist | 0.126 0.083 CHEMBL743 | CHEMBL743 | |
| 0.227 | 0.203 | 0.227 | Transcription factor inhibitor | |||
| 0.063 | 0.042 | 0.063 | Cyclin A inhibitor | |||
| 0.096 | 0.078 | 0.114 | Factor V inhibitor | 0.096 0.078 CHEMBL745 0.114 0.045 CHEMBL743 | CHEMBL743 | |
| 0.093 | 0.075 | 0.093 | Urease inhibitor | 0.088 0.08 CHEMBL743 | ||
| 0.032 | 0.016 | 0.048 | Liver X receptor alpha antagonist | 0.048 0.006 CHEMBL745 0.035 0.012 CHEMBL743 | CHEMBL745 | |
| 0.061 | 0.046 | 0.061 | Cyclin A2 inhibitor | |||
| 0.1 | 0.085 | 0.1 | Nav1.5 sodium channel blocker | |||
| 0.04 | 0.025 | 0.055 | Glutamate (mGluR group II) antagonist | 0.052 0.015 CHEMBL745 0.055 0.013 CHEMBL743 | CHEMBL743 | |
| 0.122 | 0.107 | 0.142 | CC chemokine 6 receptor antagonist | 0.132 0.064 CHEMBL743 0.142 0.035 CHEMBL3544878 | CHEMBL3544878 | |
| 0.187 | 0.173 | 0.187 | Thyroid hormone antagonist | |||
| 0.22 | 0.21 | 0.22 | DNA polymerase beta inhibitor | |||
| 0.03 | 0.02 | 0.037 | Glutamate (mGluR2) antagonist | 0.037 0.013 CHEMBL745 0.035 0.015 CHEMBL743 | CHEMBL745 | |
| 0.021 | 0.011 | 0.021 | Factor IX inhibitor | 0.017 0.015 CHEMBL745 0.018 0.013 CHEMBL743 | ||
| 0.071 | 0.062 | 0.071 | CC chemokine receptor antagonist | |||
| 0.014 | 0.007 | 0.02 | Carbonic anhydrase XI inhibitor | 0.02 0.004 CHEMBL743 | CHEMBL743 | |
| 0.032 | 0.025 | 0.032 | Calcium release-activated channel blocker | |||
| 0.038 | 0.032 | 0.039 | Phenylethanolamine N methyltransferase inhibitor | 0.039 0.031 CHEMBL745 | CHEMBL745 | |
| 0.113 | 0.107 | 0.113 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | |||
| 0.062 | 0.057 | 0.065 | CDK1/cyclin B1 inhibitor | 0.065 0.054 CHEMBL745 | CHEMBL745 | |
| 0.034 | 0.03 | 0.084 | Glutamate (mGluR3) antagonist | 0.048 0.014 CHEMBL745 0.084 0.005 CHEMBL743 | CHEMBL743 | |
| 0.068 | 0.064 | 0.068 | S-adenosyl-L-methionine decarboxylase inhibitor | |||
| 0.057 | 0.054 | 0.058 | Heme oxygenase stimulant | 0.058 0.053 CHEMBL743 | CHEMBL743 | |
| 0.107 | 0.105 | 0.107 | Calcium channel blocker | |||
| 0.014 | 0.017 | 0.03 | Carbonic anhydrase X inhibitor | 0.03 0.004 CHEMBL743 | CHEMBL743 | |
| 0.014 | 0.017 | 0.03 | Carbonic anhydrase VIII inhibitor | 0.03 0.004 CHEMBL743 | CHEMBL743 | |
| 0.06 | 0.063 | 0.062 | MAP kinase kinase 8 inhibitor | 0.062 0.059 CHEMBL745 | CHEMBL745 | |
| 0.033 | 0.036 | 0.07 | Urate transporter 1 inhibitor | 0.07 0.01 CHEMBL743 | CHEMBL743 | |
| 0.192 | 0.199 | 0.301 | Sodium/bile acid cotransporter inhibitor | 0.215 0.168 CHEMBL745 0.301 0.078 CHEMBL743 0.197 0.192 CHEMBL3544878 | CHEMBL743 | |
| 0.135 | 0.144 | 0.14 | Neurotensin receptor agonist | 0.14 0.13 CHEMBL743 | CHEMBL743 | |
| 0.011 | 0.02 | 0.015 | G-protein-coupled receptor 120 agonist | 0.015 0.014 CHEMBL745 | CHEMBL745 | |
| 0.13 | 0.141 | 0.18 | ATPase inhibitor | 0.18 0.058 CHEMBL3544878 | CHEMBL3544878 | |
| 0.031 | 0.048 | 0.053 | Liver X receptor alpha agonist | 0.053 0.017 CHEMBL745 | CHEMBL745 | |
| 0.122 | 0.139 | 0.173 | Amyloid beta precursor protein antagonist | 0.173 0.079 CHEMBL743 | CHEMBL743 | |
| 0.053 | 0.073 | 0.059 | Trypsin inhibitor | 0.059 0.052 CHEMBL743 | CHEMBL743 | |
| 0.01 | 0.03 | 0.04 | Prostaglandin EP1 antagonist | 0.018 0.015 CHEMBL745 0.04 0.008 CHEMBL743 | CHEMBL743 | |
| 0.018 | 0.046 | 0.023 | Glutamate (mGluR1) agonist | 0.023 0.022 CHEMBL743 | CHEMBL743 | |
| 0.068 | 0.104 | 0.093 | Aminoacyl-tRNA synthetase inhibitor | 0.093 0.054 CHEMBL745 0.086 0.066 CHEMBL743 | CHEMBL745 | |
| 0.023 | 0.066 | 0.042 | Dihydropteroate synthase inhibitor | 0.042 0.024 CHEMBL743 | CHEMBL743 | |
| 0.019 | 0.068 | 0.037 | TRPM8 blocker | 0.037 0.028 CHEMBL743 | CHEMBL743 | |
| 0.103 | 0.159 | 0.335 | Hemostatic | 0.13 0.095 CHEMBL745 0.136 0.086 CHEMBL743 0.335 0.013 CHEMBL3544878 | CHEMBL3544878 | |
| 0.049 | 0.106 | 0.073 | Phosphodiesterase IV inhibitor | 0.073 0.07 CHEMBL745 | CHEMBL745 | |
| 0.119 | 0.176 | 0.285 | Aldehyde oxidase inhibitor | 0.285 0.071 CHEMBL743 | CHEMBL743 | |
| 0.106 | 0.168 | 0.168 | Dual specificity phosphatase inhibitor | 0.168 0.076 CHEMBL743 | CHEMBL743 | |
| 0.033 | 0.096 | 0.081 | Factor IXa inhibitor | 0.081 0.016 CHEMBL3544878 | CHEMBL3544878 | |
| 0.027 | 0.091 | 0.042 | AICAR transformylase inhibitor | 0.042 0.034 CHEMBL743 | CHEMBL743 | |
| 0.028 | 0.098 | 0.042 | Guanylate cyclase stimulant | 0.042 0.034 CHEMBL743 | CHEMBL743 | |
| 0.042 | 0.135 | 0.075 | Potassium channel large-conductance Ca-activated activator | 0.075 0.039 CHEMBL743 | CHEMBL743 | |
| 0.088 | 0.187 | 0.165 | Hexokinase inhibitor | 0.164 0.064 CHEMBL743 0.165 0.063 CHEMBL3544878 | CHEMBL3544878 | |
| 0.019 | 0.134 | 0.073 | Prostaglandin E2 antagonist | 0.073 0.022 CHEMBL743 | CHEMBL743 | |
| 0.056 | 0.173 | 0.082 | Thioredoxin inhibitor | 0.082 0.077 CHEMBL3544878 | CHEMBL3544878 | |
| 0.014 | 0.138 | 0.042 | AMPA receptor antagonist | 0.042 0.041 CHEMBL743 | CHEMBL743 | |
| 0.01 | 0.137 | 0.029 | Sodium/glucose cotransporter inhibitor | 0.029 0.013 CHEMBL3544878 | CHEMBL3544878 | |
| 0.055 | 0.193 | 0.087 | ABCA1 expression enhancer | 0.087 0.07 CHEMBL743 | CHEMBL743 | |
| 0.144 | 0.284 | 0.227 | Antiobesity | 0.227 0.18 CHEMBL3544878 | CHEMBL3544878 | |
| 0.127 | 0.273 | 0.333 | Peptidyltransferase inhibitor | 0.165 0.157 CHEMBL743 0.333 0.015 CHEMBL3544878 | CHEMBL3544878 | |
| 0.046 | 0.192 | 0.127 | Uric acid excretion stimulant | 0.127 0.034 CHEMBL743 0.121 0.037 CHEMBL3544878 | CHEMBL743 | |
| 0.052 | 0.207 | 0.223 | Amylase inhibitor | 0.223 0.036 CHEMBL3544878 | CHEMBL3544878 | |
| 0.063 | 0.231 | 0.14 | Mcl-1 antagonist | 0.14 0.1 CHEMBL743 | CHEMBL743 | |
| 0.035 | 0.204 | 0.1 | Protein kinase (CK2) alpha inhibitor | 0.1 0.077 CHEMBL743 | CHEMBL743 | |
| 0.043 | 0.22 | 0.093 | Ferrochelatase inhibitor | 0.093 0.079 CHEMBL743 | CHEMBL743 | |
| 0.122 | 0.299 | 0.472 | Alpha-glucosidase inhibitor | 0.472 0.089 CHEMBL3544878 | CHEMBL3544878 | |
| 0.099 | 0.307 | 0.521 | Transcription factor NF kappa B inhibitor | 0.521 0.041 CHEMBL3544878 | CHEMBL3544878 | |
| 0.009 | 0.24 | 0.028 | Purinergic P2Y14 antagonist | 0.028 0.024 CHEMBL743 | CHEMBL743 | |
| 0.067 | 0.336 | 0.351 | Tumour necrosis factor alpha release inhibitor | 0.351 0.038 CHEMBL3544878 | CHEMBL3544878 | |
| 0.032 | 0.322 | 0.224 | AMP-activated protein kinase stimulant | 0.224 0.008 CHEMBL3544878 | CHEMBL3544878 | |
| 0.072 | 0.392 | 0.155 | Lipocortins synthesis antagonist | 0.155 0.098 CHEMBL743 | CHEMBL743 | |
| 0.051 | 0.372 | 0.37 | Platelet adhesion inhibitor | 0.37 0.015 CHEMBL3544878 | CHEMBL3544878 | |
| 0.034 | 0.374 | 0.088 | NADH dehydrogenase inhibitor | 0.088 0.059 CHEMBL3544878 | CHEMBL3544878 | |
| 0.027 | 0.388 | 0.112 | Beta glucuronidase inhibitor | 0.112 0.054 CHEMBL3544878 | CHEMBL3544878 | |
| 0.103 | 0.464 | 0.5 | Apoptosis agonist | 0.5 0.074 CHEMBL3544878 | CHEMBL3544878 | |
| 0.078 | 0.443 | 0.373 | Immunomodulator | 0.373 0.052 CHEMBL3544878 | CHEMBL3544878 | |
| 0.053 | 0.452 | 0.133 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.133 0.109 CHEMBL743 | CHEMBL743 | |
| 0.048 | 0.461 | 0.179 | NOS3 expression enhancer | 0.179 0.05 CHEMBL3544878 | CHEMBL3544878 | |
| 0.068 | 0.487 | 0.202 | Histamine release inhibitor | 0.202 0.2 CHEMBL3544878 | CHEMBL3544878 | |
| 0.058 | 0.48 | 0.518 | Antithrombotic | 0.518 0.027 CHEMBL3544878 | CHEMBL3544878 | |
| 0.029 | 0.497 | 0.236 | Platelet antagonist | 0.236 0.079 CHEMBL3544878 | CHEMBL3544878 | |
| 0.008 | 0.488 | 0.113 | Protein-tyrosine phosphatase 1B inhibitor | 0.113 0.068 CHEMBL3544878 | CHEMBL3544878 | |
| 0.026 | 0.519 | 0.402 | Free radical scavenger | 0.402 0.028 CHEMBL3544878 | CHEMBL3544878 | |
| 0.024 | 0.538 | 0.148 | Cell wall synthesis inhibitor | 0.148 0.068 CHEMBL3544878 | CHEMBL3544878 | |
| 0.014 | 0.533 | 0.14 | Protein-tyrosine phosphatase inhibitor | 0.14 0.089 CHEMBL3544878 | CHEMBL3544878 | |
| 0.046 | 0.568 | 0.498 | Antibacterial | 0.498 0.041 CHEMBL3544878 | CHEMBL3544878 | |
| 0.007 | 0.532 | 0.038 | Retinoic acid alpha receptor agonist | 0.038 0.03 CHEMBL743 | CHEMBL743 | |
| 0.063 | 0.594 | 0.393 | Apoptosis antagonist | 0.393 0.04 CHEMBL3544878 | CHEMBL3544878 | |
| 0.025 | 0.558 | 0.141 | Toll-Like receptor 4 antagonist | 0.141 0.026 CHEMBL3544878 | CHEMBL3544878 | |
| 0.026 | 0.575 | 0.183 | Insulin secretagoues | 0.183 0.046 CHEMBL3544878 | CHEMBL3544878 | |
| 0.024 | 0.739 | 0.121 | Transcription factor NF kappa B stimulant | 0.121 0.025 CHEMBL3544878 | CHEMBL3544878 | |
| 0.007 | 0.742 | 0.063 | Protein 50S ribosomal subunit inhibitor | 0.063 0.028 CHEMBL3544878 | CHEMBL3544878 | |
| 0.009 | 0.761 | 0.051 | Glucose-6-phosphate translocase inhibitor | 0.051 0.037 CHEMBL3544878 | CHEMBL3544878 | |
| 0.008 | 0.762 | 0.191 | Immunostimulant | 0.191 0.126 CHEMBL3544878 | CHEMBL3544878 | |
| 0.02 | 0.795 | 0.361 | Hypoglycemic | 0.361 0.035 CHEMBL3544878 | CHEMBL3544878 | |
| 0.019 | 0.796 | 0.539 | Cyclophilin D inhibitor | 0.539 0.04 CHEMBL3544878 | CHEMBL3544878 | |
| 0.015 | 0.826 | 0.312 | Immunosuppressant | 0.312 0.107 CHEMBL3544878 | CHEMBL3544878 | |
| 0.007 | 0.844 | 0.171 | Thrombolytic | 0.171 0.067 CHEMBL3544878 | CHEMBL3544878 | |
| 0.005 | 0.844 | 0.37 | Antioxidant | 0.37 0.041 CHEMBL3544878 | CHEMBL3544878 | |
| 0.039 | 0.909 | 0.365 | Interleukin 2 agonist | 0.365 0.039 CHEMBL3544878 | CHEMBL3544878 | |
| 0.003 | 0.883 | 0.234 | Selectin antagonist | 0.234 0.009 CHEMBL3544878 | CHEMBL3544878 | |
| 0.011 | 0.952 | 0.305 | Hepatoprotectant | 0.305 0.028 CHEMBL3544878 | CHEMBL3544878 | |
| 0.005 | 0.952 | 0.165 | Vasodilator | 0.165 0.137 CHEMBL3544878 | CHEMBL3544878 | |
| 0.004 | 0.952 | 0.242 | Nitric oxide antagonist | 0.242 0.054 CHEMBL3544878 | CHEMBL3544878 | |
| 0.003 | 0.979 | 0.048 | Antibiotic Aminoglycoside-like | 0.048 0.014 CHEMBL3544878 | CHEMBL3544878 | |
| 0.004 | 0.991 | 0.428 | Angiogenesis stimulant | 0.428 0.018 CHEMBL3544878 | CHEMBL3544878 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |