Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9610.0030.961Phosphatidylinositol 3-kinase alpha inhibitor

0.83 0.003 CHEMBL3526762

0.960.0030.96Phosphatidylinositol kinase inhibitor

0.838 0.003 CHEMBL3526762

0.9460.0030.946Phosphatidylinositol 3-kinase gamma inhibitor

0.803 0.003 CHEMBL3526762

0.7720.0010.772mTOR inhibitor

0.707 0.001 CHEMBL3526762

0.5050.0310.505Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.381 0.119 CHEMBL3526762

0.3680.0210.368EphB2 antagonist

0.261 0.051 CHEMBL3526762

0.3350.0020.335mTOR complex 2 inhibitor

0.272 0.003 CHEMBL3526762

0.3280.0030.328mTOR complex 1 inhibitor

0.27 0.004 CHEMBL3526762

0.2650.0180.265Activin receptor-like kinase 2 inhibitor

0.131 0.084 CHEMBL3526762

0.2920.0490.292Potassium channel blocker

0.254 0.065 CHEMBL3526762

0.2730.0390.273TRKC antagonist

0.167 0.088 CHEMBL3526762

0.3290.1090.329MAP kinase kinase 6 inhibitor

0.263 0.174 CHEMBL3526762

0.2380.0190.238Cyclin-dependent kinase 8 inhibitor

0.163 0.067 CHEMBL3526762

0.2630.0530.263Ca2+/calmodulin-dependent protein kinase inhibitor

0.137 0.126 CHEMBL3526762

0.2520.060.252Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.157 0.134 CHEMBL3526762

0.1960.0050.196Phosphatidylinositol 3-kinase beta inhibitor

0.102 0.012 CHEMBL3526762

0.2350.0540.235Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.126 0.119 CHEMBL3526762

0.2010.0230.201MAP kinase 3 inhibitor

0.189 0.029 CHEMBL3526762

0.2250.0520.225Focal adhesion kinase 2 inhibitor
0.2360.0690.236MAP-kinase-activated kinase 5 inhibitor

0.181 0.131 CHEMBL3526762

0.2420.0770.242Ca2+/calmodulin-dependent kinase IV inhibitor

0.206 0.149 CHEMBL3526762

0.2010.0440.201Polo-like kinase-3 inhibitor
0.2190.070.219MAP kinase kinase 2 inhibitor
0.1650.0180.165Vanilloid antagonist

0.139 0.023 CHEMBL3526762

0.1790.0320.179TRKB antagonist

0.112 0.084 CHEMBL3526762

0.2620.1150.262Angiogenesis inhibitor

0.19 0.182 CHEMBL3526762

0.2510.1060.251Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.188 0.172 CHEMBL3526762

0.1890.0450.189Tyrosine-protein kinase receptor antagonist
0.1480.0040.148Potassium channel (Inward rectifier) blocker

0.094 0.008 CHEMBL3526762

0.1490.0110.149Phosphatidylinositol 3-kinase delta inhibitor

0.073 0.028 CHEMBL3526762

0.1530.0210.153Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.09 0.057 CHEMBL3526762

0.1450.0130.145Phosphodiesterase 4B inhibitor
0.140.0160.14Tyk2 inhibitor

0.065 0.045 CHEMBL3526762

0.1460.0320.146EphA2 antagonist

0.112 0.062 CHEMBL3526762

0.1310.020.131Interleukin 12 antagonist

0.112 0.038 CHEMBL3526762

0.1180.0110.118Polo-like kinase-2 inhibitor

0.084 0.041 CHEMBL3526762

0.1570.050.157Tyrosine-protein kinase receptor FLT3 inhibitor
0.1560.050.156Protein kinase (CK1) delta inhibitor
0.1430.0390.143Ephrin antagonist

0.09 0.073 CHEMBL3526762

0.1180.0140.118EphB4 antagonist

0.054 0.045 CHEMBL3526762

0.2060.1060.206MAP kinase kinase 3 inhibitor

0.187 0.165 CHEMBL3526762

0.1730.0790.173MAP kinase kinase 5 inhibitor
0.1810.0880.181I kappa B kinase epsilon inhibitor
0.1650.0740.165Protein kinase (CK1) gamma 3 inhibitor
0.1440.0580.144Aurora-C kinase inhibitor

0.126 0.092 CHEMBL3526762

0.1780.0960.178Ca2+/calmodulin-dependent kinase II beta inhibitor
0.1280.050.1285 Hydroxytryptamine 3A agonist
0.1470.0710.147Protein kinase (CK1) gamma 1 inhibitor
0.0840.0090.084DNA-dependent protein kinase inhibitor

0.055 0.018 CHEMBL3526762

0.2090.1350.209Gastrin inhibitor
0.0910.0190.091Orexin receptor 1 antagonist
0.140.070.14Cytokine production inhibitor
0.1420.0720.142Protein kinase (CK1) gamma inhibitor
0.1420.0730.142Protein kinase (CK1) inhibitor
0.1270.0590.127Aurora-B kinase inhibitor
0.0770.0170.183Glucosylceramidase inhibitor

0.183 0.003 CHEMBL3526762

CHEMBL3526762
0.120.0650.12Protein kinase (CK1) gamma 2 inhibitor
0.1660.1110.166Proto-oncogene tyrosine-protein kinase Fyn inhibitor
0.060.0050.06ATR kinase inhibitor
0.1110.0590.111Vascular endothelial growth factor 1 antagonist
0.0980.0480.098Polo-like kinase-1 inhibitor
0.1130.0630.113Polo-like kinase-4 inhibitor
0.0930.0460.093TIE antagonist
0.0530.0070.053ATM kinase inhibitor

0.047 0.01 CHEMBL3526762

0.0910.0460.091TIE-2 antagonist
0.0480.0050.048Potassium channel (Inward rectifier) 1 blocker

0.043 0.005 CHEMBL3526762

0.0760.0330.076Adenosine A2a receptor antagonist

0.058 0.047 CHEMBL3526762

0.1460.1040.146CDC-like kinase 4 inhibitor
0.1310.0910.131Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor
0.1080.0690.108Interleukin 2 antagonist
0.0860.0480.086Transforming growth factor beta 3 antagonist
0.0910.0530.091Phosphodiesterase IV inhibitor
0.0730.0350.073Raf kinase C inhibitor
0.0760.0390.076Vanilloid 1 antagonist
0.0710.0330.071Janus tyrosine kinase 1 inhibitor
0.1350.0980.135Tyrosine kinase inhibitor
0.0730.0360.073Orexin receptor antagonist
0.080.0450.08Rho-associated kinase II inhibitor
0.0840.0540.084Leucine-rich repeat kinase 2 inhibitor
0.1140.0840.114RET inhibitor
0.0690.0410.069Adenosine A2 receptor antagonist
0.1960.1690.196Immunomodulator

0.193 0.173 CHEMBL3526762

0.1090.0840.109MAP kinase 12 inhibitor
0.0750.0510.075Janus tyrosine kinase 2 inhibitor
0.1050.0820.105TRKA antagonist
0.0220.0050.022Granulocyte colony stimulating factor receptor agonist

0.019 0.012 CHEMBL3526762

0.0380.0230.038Orexin receptor 2 antagonist
0.0690.0550.069Epoxide hydrolase inhibitor
0.1230.1130.123Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.0760.0660.076Insulin like growth factor 1 antagonist
0.0780.070.078Insulin growth factor antagonist
0.1080.1020.108DNA repair enzyme inhibitor

0.107 0.103 CHEMBL3526762

0.0540.0480.054Protein kinase C iota inhibitor
0.050.0440.05Alpha 1L adrenoreceptor antagonist
0.020.0540.029Potassium channel subfamily K member 3 blocker

0.029 0.023 CHEMBL3526762

CHEMBL3526762
0.0240.0660.047Purinergic P2Y antagonist

0.047 0.029 CHEMBL3526762

CHEMBL3526762
0.2240.2980.263Antiinflammatory

0.263 0.252 CHEMBL3526762

CHEMBL3526762
0.0080.3990.09NMDA 2B receptor antagonist

0.09 0.018 CHEMBL3526762

CHEMBL3526762
0.0030.6770.0291,3-Beta-glucan synthase inhibitor

0.029 0.017 CHEMBL3526762

CHEMBL3526762
Ext Pa Pi Pmax Activity Other Results ID Pa_max