| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.961 | 0.003 | 0.961 | Phosphatidylinositol 3-kinase alpha inhibitor | 0.83 0.003 CHEMBL3526762 | ||
| 0.96 | 0.003 | 0.96 | Phosphatidylinositol kinase inhibitor | 0.838 0.003 CHEMBL3526762 | ||
| 0.946 | 0.003 | 0.946 | Phosphatidylinositol 3-kinase gamma inhibitor | 0.803 0.003 CHEMBL3526762 | ||
| 0.772 | 0.001 | 0.772 | mTOR inhibitor | 0.707 0.001 CHEMBL3526762 | ||
| 0.505 | 0.031 | 0.505 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.381 0.119 CHEMBL3526762 | ||
| 0.368 | 0.021 | 0.368 | EphB2 antagonist | 0.261 0.051 CHEMBL3526762 | ||
| 0.335 | 0.002 | 0.335 | mTOR complex 2 inhibitor | 0.272 0.003 CHEMBL3526762 | ||
| 0.328 | 0.003 | 0.328 | mTOR complex 1 inhibitor | 0.27 0.004 CHEMBL3526762 | ||
| 0.265 | 0.018 | 0.265 | Activin receptor-like kinase 2 inhibitor | 0.131 0.084 CHEMBL3526762 | ||
| 0.292 | 0.049 | 0.292 | Potassium channel blocker | 0.254 0.065 CHEMBL3526762 | ||
| 0.273 | 0.039 | 0.273 | TRKC antagonist | 0.167 0.088 CHEMBL3526762 | ||
| 0.329 | 0.109 | 0.329 | MAP kinase kinase 6 inhibitor | 0.263 0.174 CHEMBL3526762 | ||
| 0.238 | 0.019 | 0.238 | Cyclin-dependent kinase 8 inhibitor | 0.163 0.067 CHEMBL3526762 | ||
| 0.263 | 0.053 | 0.263 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.137 0.126 CHEMBL3526762 | ||
| 0.252 | 0.06 | 0.252 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.157 0.134 CHEMBL3526762 | ||
| 0.196 | 0.005 | 0.196 | Phosphatidylinositol 3-kinase beta inhibitor | 0.102 0.012 CHEMBL3526762 | ||
| 0.235 | 0.054 | 0.235 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.126 0.119 CHEMBL3526762 | ||
| 0.201 | 0.023 | 0.201 | MAP kinase 3 inhibitor | 0.189 0.029 CHEMBL3526762 | ||
| 0.225 | 0.052 | 0.225 | Focal adhesion kinase 2 inhibitor | |||
| 0.236 | 0.069 | 0.236 | MAP-kinase-activated kinase 5 inhibitor | 0.181 0.131 CHEMBL3526762 | ||
| 0.242 | 0.077 | 0.242 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.206 0.149 CHEMBL3526762 | ||
| 0.201 | 0.044 | 0.201 | Polo-like kinase-3 inhibitor | |||
| 0.219 | 0.07 | 0.219 | MAP kinase kinase 2 inhibitor | |||
| 0.165 | 0.018 | 0.165 | Vanilloid antagonist | 0.139 0.023 CHEMBL3526762 | ||
| 0.179 | 0.032 | 0.179 | TRKB antagonist | 0.112 0.084 CHEMBL3526762 | ||
| 0.262 | 0.115 | 0.262 | Angiogenesis inhibitor | 0.19 0.182 CHEMBL3526762 | ||
| 0.251 | 0.106 | 0.251 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.188 0.172 CHEMBL3526762 | ||
| 0.189 | 0.045 | 0.189 | Tyrosine-protein kinase receptor antagonist | |||
| 0.148 | 0.004 | 0.148 | Potassium channel (Inward rectifier) blocker | 0.094 0.008 CHEMBL3526762 | ||
| 0.149 | 0.011 | 0.149 | Phosphatidylinositol 3-kinase delta inhibitor | 0.073 0.028 CHEMBL3526762 | ||
| 0.153 | 0.021 | 0.153 | Interleukin-1 receptor-associated protein kinase 4 inhibitor | 0.09 0.057 CHEMBL3526762 | ||
| 0.145 | 0.013 | 0.145 | Phosphodiesterase 4B inhibitor | |||
| 0.14 | 0.016 | 0.14 | Tyk2 inhibitor | 0.065 0.045 CHEMBL3526762 | ||
| 0.146 | 0.032 | 0.146 | EphA2 antagonist | 0.112 0.062 CHEMBL3526762 | ||
| 0.131 | 0.02 | 0.131 | Interleukin 12 antagonist | 0.112 0.038 CHEMBL3526762 | ||
| 0.118 | 0.011 | 0.118 | Polo-like kinase-2 inhibitor | 0.084 0.041 CHEMBL3526762 | ||
| 0.157 | 0.05 | 0.157 | Tyrosine-protein kinase receptor FLT3 inhibitor | |||
| 0.156 | 0.05 | 0.156 | Protein kinase (CK1) delta inhibitor | |||
| 0.143 | 0.039 | 0.143 | Ephrin antagonist | 0.09 0.073 CHEMBL3526762 | ||
| 0.118 | 0.014 | 0.118 | EphB4 antagonist | 0.054 0.045 CHEMBL3526762 | ||
| 0.206 | 0.106 | 0.206 | MAP kinase kinase 3 inhibitor | 0.187 0.165 CHEMBL3526762 | ||
| 0.173 | 0.079 | 0.173 | MAP kinase kinase 5 inhibitor | |||
| 0.181 | 0.088 | 0.181 | I kappa B kinase epsilon inhibitor | |||
| 0.165 | 0.074 | 0.165 | Protein kinase (CK1) gamma 3 inhibitor | |||
| 0.144 | 0.058 | 0.144 | Aurora-C kinase inhibitor | 0.126 0.092 CHEMBL3526762 | ||
| 0.178 | 0.096 | 0.178 | Ca2+/calmodulin-dependent kinase II beta inhibitor | |||
| 0.128 | 0.05 | 0.128 | 5 Hydroxytryptamine 3A agonist | |||
| 0.147 | 0.071 | 0.147 | Protein kinase (CK1) gamma 1 inhibitor | |||
| 0.084 | 0.009 | 0.084 | DNA-dependent protein kinase inhibitor | 0.055 0.018 CHEMBL3526762 | ||
| 0.209 | 0.135 | 0.209 | Gastrin inhibitor | |||
| 0.091 | 0.019 | 0.091 | Orexin receptor 1 antagonist | |||
| 0.14 | 0.07 | 0.14 | Cytokine production inhibitor | |||
| 0.142 | 0.072 | 0.142 | Protein kinase (CK1) gamma inhibitor | |||
| 0.142 | 0.073 | 0.142 | Protein kinase (CK1) inhibitor | |||
| 0.127 | 0.059 | 0.127 | Aurora-B kinase inhibitor | |||
| 0.077 | 0.017 | 0.183 | Glucosylceramidase inhibitor | 0.183 0.003 CHEMBL3526762 | CHEMBL3526762 | |
| 0.12 | 0.065 | 0.12 | Protein kinase (CK1) gamma 2 inhibitor | |||
| 0.166 | 0.111 | 0.166 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | |||
| 0.06 | 0.005 | 0.06 | ATR kinase inhibitor | |||
| 0.111 | 0.059 | 0.111 | Vascular endothelial growth factor 1 antagonist | |||
| 0.098 | 0.048 | 0.098 | Polo-like kinase-1 inhibitor | |||
| 0.113 | 0.063 | 0.113 | Polo-like kinase-4 inhibitor | |||
| 0.093 | 0.046 | 0.093 | TIE antagonist | |||
| 0.053 | 0.007 | 0.053 | ATM kinase inhibitor | 0.047 0.01 CHEMBL3526762 | ||
| 0.091 | 0.046 | 0.091 | TIE-2 antagonist | |||
| 0.048 | 0.005 | 0.048 | Potassium channel (Inward rectifier) 1 blocker | 0.043 0.005 CHEMBL3526762 | ||
| 0.076 | 0.033 | 0.076 | Adenosine A2a receptor antagonist | 0.058 0.047 CHEMBL3526762 | ||
| 0.146 | 0.104 | 0.146 | CDC-like kinase 4 inhibitor | |||
| 0.131 | 0.091 | 0.131 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | |||
| 0.108 | 0.069 | 0.108 | Interleukin 2 antagonist | |||
| 0.086 | 0.048 | 0.086 | Transforming growth factor beta 3 antagonist | |||
| 0.091 | 0.053 | 0.091 | Phosphodiesterase IV inhibitor | |||
| 0.073 | 0.035 | 0.073 | Raf kinase C inhibitor | |||
| 0.076 | 0.039 | 0.076 | Vanilloid 1 antagonist | |||
| 0.071 | 0.033 | 0.071 | Janus tyrosine kinase 1 inhibitor | |||
| 0.135 | 0.098 | 0.135 | Tyrosine kinase inhibitor | |||
| 0.073 | 0.036 | 0.073 | Orexin receptor antagonist | |||
| 0.08 | 0.045 | 0.08 | Rho-associated kinase II inhibitor | |||
| 0.084 | 0.054 | 0.084 | Leucine-rich repeat kinase 2 inhibitor | |||
| 0.114 | 0.084 | 0.114 | RET inhibitor | |||
| 0.069 | 0.041 | 0.069 | Adenosine A2 receptor antagonist | |||
| 0.196 | 0.169 | 0.196 | Immunomodulator | 0.193 0.173 CHEMBL3526762 | ||
| 0.109 | 0.084 | 0.109 | MAP kinase 12 inhibitor | |||
| 0.075 | 0.051 | 0.075 | Janus tyrosine kinase 2 inhibitor | |||
| 0.105 | 0.082 | 0.105 | TRKA antagonist | |||
| 0.022 | 0.005 | 0.022 | Granulocyte colony stimulating factor receptor agonist | 0.019 0.012 CHEMBL3526762 | ||
| 0.038 | 0.023 | 0.038 | Orexin receptor 2 antagonist | |||
| 0.069 | 0.055 | 0.069 | Epoxide hydrolase inhibitor | |||
| 0.123 | 0.113 | 0.123 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | |||
| 0.076 | 0.066 | 0.076 | Insulin like growth factor 1 antagonist | |||
| 0.078 | 0.07 | 0.078 | Insulin growth factor antagonist | |||
| 0.108 | 0.102 | 0.108 | DNA repair enzyme inhibitor | 0.107 0.103 CHEMBL3526762 | ||
| 0.054 | 0.048 | 0.054 | Protein kinase C iota inhibitor | |||
| 0.05 | 0.044 | 0.05 | Alpha 1L adrenoreceptor antagonist | |||
| 0.02 | 0.054 | 0.029 | Potassium channel subfamily K member 3 blocker | 0.029 0.023 CHEMBL3526762 | CHEMBL3526762 | |
| 0.024 | 0.066 | 0.047 | Purinergic P2Y antagonist | 0.047 0.029 CHEMBL3526762 | CHEMBL3526762 | |
| 0.224 | 0.298 | 0.263 | Antiinflammatory | 0.263 0.252 CHEMBL3526762 | CHEMBL3526762 | |
| 0.008 | 0.399 | 0.09 | NMDA 2B receptor antagonist | 0.09 0.018 CHEMBL3526762 | CHEMBL3526762 | |
| 0.003 | 0.677 | 0.029 | 1,3-Beta-glucan synthase inhibitor | 0.029 0.017 CHEMBL3526762 | CHEMBL3526762 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |