| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.79 | 0.002 | 0.816 | Factor Xa inhibitor | 0.342 0.004 CHEMBL3548561 0.66 0.002 CHEMBL3550091 0.297 0.004 CHEMBL3549528 0.548 0.003 CHEMBL3549716 0.816 0.002 CHEMBL3548175 0.719 0.002 CHEMBL3550090 0.457 0.003 CHEMBL4525768 | CHEMBL3548175 | |
| 0.57 | 0.003 | 0.57 | Factor X inhibitor | 0.483 0.004 CHEMBL3548561 0.488 0.004 CHEMBL3550091 0.206 0.005 CHEMBL3549528 0.427 0.004 CHEMBL3549716 0.346 0.004 CHEMBL3548175 0.509 0.004 CHEMBL3550090 0.361 0.004 CHEMBL4525768 | ||
| 0.399 | 0.016 | 0.661 | Anticoagulant | 0.372 0.019 CHEMBL3548561 0.389 0.017 CHEMBL3550091 0.385 0.018 CHEMBL3549528 0.391 0.017 CHEMBL3549716 0.661 0.005 CHEMBL3548175 0.407 0.016 CHEMBL3550090 0.337 0.023 CHEMBL4525768 | CHEMBL3548175 | |
| 0.401 | 0.06 | 0.557 | Toll-Like receptor 7 agonist | 0.557 0.023 CHEMBL3548561 0.365 0.075 CHEMBL3550091 0.421 0.052 CHEMBL3549528 0.464 0.04 CHEMBL3549716 0.412 0.055 CHEMBL3548175 0.369 0.073 CHEMBL3550090 | CHEMBL3548561 | |
| 0.397 | 0.061 | 0.554 | Toll-Like receptor agonist | 0.554 0.023 CHEMBL3548561 0.361 0.077 CHEMBL3550091 0.422 0.052 CHEMBL3549528 0.461 0.04 CHEMBL3549716 0.407 0.058 CHEMBL3548175 0.364 0.075 CHEMBL3550090 | CHEMBL3548561 | |
| 0.396 | 0.067 | 0.56 | Antiobesity | 0.56 0.026 CHEMBL3548561 0.349 0.088 CHEMBL3550091 0.404 0.064 CHEMBL3549716 0.413 0.061 CHEMBL3548175 0.473 0.043 CHEMBL3550090 0.208 0.199 CHEMBL4525768 | CHEMBL3548561 | |
| 0.293 | 0.005 | 0.344 | Glutamate (mGluR) agonist | 0.331 0.005 CHEMBL3548561 0.295 0.005 CHEMBL3550091 0.058 0.048 CHEMBL3549528 0.344 0.005 CHEMBL3549716 0.144 0.015 CHEMBL3548175 0.211 0.008 CHEMBL3550090 0.192 0.01 CHEMBL4525768 | CHEMBL3549716 | |
| 0.257 | 0.005 | 0.257 | Interleukin 2 antagonist | 0.245 0.005 CHEMBL3548561 0.247 0.005 CHEMBL3550091 0.15 0.018 CHEMBL3549528 0.225 0.005 CHEMBL3549716 0.198 0.008 CHEMBL3548175 0.243 0.005 CHEMBL3550090 0.206 0.007 CHEMBL4525768 | ||
| 0.222 | 0.008 | 0.468 | Glutamate receptor agonist | 0.41 0.004 CHEMBL3548561 0.215 0.009 CHEMBL3550091 0.468 0.004 CHEMBL3549716 0.104 0.035 CHEMBL3550090 | CHEMBL3549716 | |
| 0.174 | 0.015 | 0.176 | Rho-associated kinase inhibitor | 0.081 0.046 CHEMBL3548561 0.165 0.016 CHEMBL3550091 0.116 0.028 CHEMBL3549716 0.072 0.053 CHEMBL3548175 0.176 0.015 CHEMBL3550090 0.093 0.038 CHEMBL4525768 | CHEMBL3550090 | |
| 0.296 | 0.139 | 0.296 | MAP kinase kinase 6 inhibitor | 0.268 0.169 CHEMBL3548561 0.268 0.169 CHEMBL3550091 0.265 0.172 CHEMBL3549716 0.243 0.2 CHEMBL3548175 0.296 0.139 CHEMBL3550090 | ||
| 0.165 | 0.009 | 0.165 | CC chemokine 6 receptor antagonist | 0.165 0.01 CHEMBL3548561 0.145 0.03 CHEMBL3550091 0.156 0.016 CHEMBL3549528 0.153 0.019 CHEMBL3549716 0.156 0.016 CHEMBL3548175 0.162 0.011 CHEMBL3550090 0.144 0.032 CHEMBL4525768 | ||
| 0.226 | 0.077 | 0.244 | MAP-kinase-activated kinase 5 inhibitor | 0.2 0.103 CHEMBL3550091 0.183 0.127 CHEMBL3549716 0.244 0.063 CHEMBL3550090 | CHEMBL3550090 | |
| 0.25 | 0.108 | 0.253 | Nootropic | 0.242 0.115 CHEMBL3550091 0.226 0.129 CHEMBL3549716 0.215 0.14 CHEMBL3548175 0.253 0.106 CHEMBL3550090 | CHEMBL3550090 | |
| 0.145 | 0.018 | 0.165 | Rho-associated kinase II inhibitor | 0.165 0.015 CHEMBL3548561 0.133 0.021 CHEMBL3550091 0.082 0.044 CHEMBL3549716 0.125 0.023 CHEMBL3550090 0.074 0.052 CHEMBL4525768 | CHEMBL3548561 | |
| 0.119 | 0.006 | 0.119 | Factor IXa inhibitor | 0.11 0.008 CHEMBL3548561 0.111 0.008 CHEMBL3550091 0.118 0.006 CHEMBL3549528 0.111 0.008 CHEMBL3549716 0.096 0.011 CHEMBL3548175 0.113 0.007 CHEMBL3550090 0.1 0.01 CHEMBL4525768 | ||
| 0.287 | 0.175 | 0.54 | Cyclophilin D inhibitor | 0.54 0.04 CHEMBL3548561 0.278 0.182 CHEMBL3550091 0.276 0.185 CHEMBL3549528 0.409 0.086 CHEMBL3549716 0.324 0.142 CHEMBL3550090 | CHEMBL3548561 | |
| 0.267 | 0.169 | 0.42 | Analgesic | 0.246 0.186 CHEMBL3550091 0.252 0.181 CHEMBL3549716 0.42 0.076 CHEMBL3548175 | CHEMBL3548175 | |
| 0.133 | 0.039 | 0.167 | Cyclin-dependent kinase 9 inhibitor | 0.089 0.076 CHEMBL3550091 0.167 0.029 CHEMBL3550090 | CHEMBL3550090 | |
| 0.158 | 0.067 | 0.169 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.155 0.069 CHEMBL3550091 0.138 0.086 CHEMBL3549716 0.169 0.059 CHEMBL3550090 | CHEMBL3550090 | |
| 0.098 | 0.027 | 0.1 | Glutamate (mGluR group I) antagonist | 0.097 0.028 CHEMBL3550091 0.1 0.026 CHEMBL3549716 0.078 0.039 CHEMBL3550090 | CHEMBL3549716 | |
| 0.114 | 0.051 | 0.117 | Chemokine receptor antagonist | 0.093 0.07 CHEMBL3550091 0.117 0.05 CHEMBL3550090 | CHEMBL3550090 | |
| 0.074 | 0.014 | 0.075 | Chemokine receptor agonist | 0.068 0.019 CHEMBL3548561 0.075 0.013 CHEMBL3550091 0.054 0.032 CHEMBL3548175 0.074 0.014 CHEMBL3550090 0.044 0.04 CHEMBL4525768 | CHEMBL3550091 | |
| 0.091 | 0.032 | 0.099 | CDK1/cyclin B1 inhibitor | 0.069 0.049 CHEMBL3548561 0.094 0.031 CHEMBL3550091 0.071 0.047 CHEMBL3549716 0.061 0.059 CHEMBL3548175 0.099 0.029 CHEMBL3550090 | CHEMBL3550090 | |
| 0.133 | 0.077 | 0.151 | Aurora-C kinase inhibitor | 0.151 0.049 CHEMBL3550091 0.128 0.088 CHEMBL3549716 0.14 0.064 CHEMBL3550090 0.117 0.114 CHEMBL4525768 | CHEMBL3550091 | |
| 0.065 | 0.019 | 0.065 | Glutamate (mGluR5) antagonist | 0.064 0.02 CHEMBL3550091 0.058 0.024 CHEMBL3549716 0.049 0.03 CHEMBL3550090 | ||
| 0.125 | 0.081 | 0.14 | Cyclin-dependent kinase 7 inhibitor | 0.126 0.079 CHEMBL3550091 0.14 0.067 CHEMBL3550090 | CHEMBL3550090 | |
| 0.209 | 0.166 | 0.345 | Antithrombotic | 0.344 0.067 CHEMBL3548561 0.345 0.066 CHEMBL3549528 0.313 0.08 CHEMBL3549716 0.198 0.18 CHEMBL3550090 | CHEMBL3549528 | |
| 0.069 | 0.029 | 0.071 | Cyclin H inhibitor | 0.054 0.048 CHEMBL3548561 0.07 0.028 CHEMBL3550091 0.062 0.037 CHEMBL3549716 0.055 0.046 CHEMBL3548175 0.071 0.027 CHEMBL3550090 0.058 0.042 CHEMBL4525768 | CHEMBL3550090 | |
| 0.069 | 0.03 | 0.069 | Corticotropin releasing factor 2 receptor antagonist | 0.066 0.035 CHEMBL3550091 0.063 0.04 CHEMBL3550090 | ||
| 0.056 | 0.025 | 0.113 | Glutamate (mGluR group I) agonist | 0.089 0.01 CHEMBL3550091 0.113 0.007 CHEMBL3549716 | CHEMBL3549716 | |
| 0.08 | 0.049 | 0.114 | Glutamate (mGluR) antagonist | 0.075 0.054 CHEMBL3550091 0.114 0.028 CHEMBL3549716 | CHEMBL3549716 | |
| 0.056 | 0.028 | 0.06 | Phosphodiesterase 7A inhibitor | 0.06 0.022 CHEMBL3548561 0.048 0.045 CHEMBL3550091 0.054 0.031 CHEMBL3550090 | CHEMBL3548561 | |
| 0.065 | 0.038 | 0.132 | Neuraminidase inhibitor | 0.104 0.014 CHEMBL3548561 0.062 0.041 CHEMBL3550091 0.064 0.038 CHEMBL3549528 0.132 0.008 CHEMBL3549716 0.057 0.047 CHEMBL3548175 0.069 0.034 CHEMBL3550090 | CHEMBL3549716 | |
| 0.066 | 0.04 | 0.137 | Neuraminidase (influenza) inhibitor | 0.095 0.018 CHEMBL3548561 0.063 0.047 CHEMBL3550091 0.068 0.038 CHEMBL3549528 0.137 0.009 CHEMBL3549716 0.063 0.047 CHEMBL3548175 0.069 0.036 CHEMBL3550090 | CHEMBL3549716 | |
| 0.041 | 0.015 | 0.041 | CXC chemokine receptor agonist | 0.039 0.018 CHEMBL3548561 0.041 0.013 CHEMBL3550091 0.041 0.015 CHEMBL3550090 | ||
| 0.033 | 0.008 | 0.033 | Hexokinase stimulant | 0.02 0.013 CHEMBL3550091 0.023 0.012 CHEMBL3549716 0.025 0.01 CHEMBL3550090 | ||
| 0.05 | 0.026 | 0.092 | Glutamate (mGluR5) agonist | 0.047 0.03 CHEMBL3550091 0.092 0.008 CHEMBL3549716 | CHEMBL3549716 | |
| 0.048 | 0.026 | 0.052 | Baculoviral IAP repeat-containing protein inhibitor | 0.052 0.015 CHEMBL3550091 0.044 0.041 CHEMBL3549716 0.048 0.027 CHEMBL3550090 | CHEMBL3550091 | |
| 0.064 | 0.042 | 0.064 | Phosphodiesterase VII inhibitor | 0.063 0.043 CHEMBL3548561 | ||
| 0.03 | 0.013 | 0.03 | 5 Hydroxytryptamine 1F agonist | 0.028 0.015 CHEMBL3550091 | ||
| 0.139 | 0.125 | 0.139 | Cyclin-dependent kinase 3 inhibitor | 0.139 0.126 CHEMBL3550091 | ||
| 0.061 | 0.048 | 0.063 | Prolactin release inhibitor | 0.063 0.039 CHEMBL3548561 | CHEMBL3548561 | |
| 0.057 | 0.05 | 0.094 | Tyk2 inhibitor | 0.094 0.03 CHEMBL3550091 0.064 0.045 CHEMBL3550090 | CHEMBL3550091 | |
| 0.041 | 0.04 | 0.072 | Neuraminidase (Influenza A) inhibitor | 0.064 0.01 CHEMBL3548561 0.044 0.034 CHEMBL3549528 0.072 0.006 CHEMBL3549716 0.043 0.037 CHEMBL3550090 | CHEMBL3549716 | |
| 0.041 | 0.04 | 0.041 | Dipeptidyl peptidase IV inhibitor | |||
| 0.009 | 0.009 | 0.01 | Baculoviral IAP repeat-containing protein 2 inhibitor | 0.01 0.005 CHEMBL3550091 | CHEMBL3550091 | |
| 0.064 | 0.065 | 0.105 | Rho-associated kinase I inhibitor | 0.068 0.06 CHEMBL3550091 0.105 0.029 CHEMBL3550090 | CHEMBL3550090 | |
| 0.077 | 0.088 | 0.084 | MAP kinase 9 inhibitor | 0.084 0.078 CHEMBL3550091 | CHEMBL3550091 | |
| 0.06 | 0.09 | 0.085 | ALK inhibitor | 0.085 0.054 CHEMBL3550091 | CHEMBL3550091 | |
| 0.029 | 0.083 | 0.037 | Integrin alpha1beta1 antagonist | 0.036 0.034 CHEMBL3548561 0.037 0.029 CHEMBL3550091 | CHEMBL3550091 | |
| 0.039 | 0.094 | 0.078 | Lipase inhibitor | 0.078 0.045 CHEMBL3548561 | CHEMBL3548561 | |
| 0.007 | 0.152 | 0.03 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.03 0.019 CHEMBL3549716 | CHEMBL3549716 | |
| 0.046 | 0.21 | 0.117 | Glutamate receptor antagonist | 0.117 0.078 CHEMBL3549716 | CHEMBL3549716 | |
| 0.049 | 0.241 | 0.136 | Thrombolytic | 0.127 0.102 CHEMBL3548561 0.136 0.093 CHEMBL3549528 | CHEMBL3549528 | |
| 0.117 | 0.324 | 0.249 | Peptidyltransferase inhibitor | 0.249 0.051 CHEMBL3549528 | CHEMBL3549528 | |
| 0.019 | 0.227 | 0.141 | Myc inhibitor | 0.141 0.005 CHEMBL3550090 | CHEMBL3550090 | |
| 0.062 | 0.336 | 0.143 | Polo-like kinase-3 inhibitor | 0.143 0.092 CHEMBL3548175 | CHEMBL3548175 | |
| 0.004 | 0.525 | 0.021 | Adenosine A1 receptor agonist | 0.021 0.02 CHEMBL3549528 | CHEMBL3549528 | |
| 0.021 | 0.591 | 0.145 | Cell wall synthesis inhibitor | 0.145 0.07 CHEMBL3548561 | CHEMBL3548561 | |
| 0.017 | 0.619 | 0.459 | Platelet antagonist | 0.459 0.018 CHEMBL3548175 | CHEMBL3548175 | |
| 0.011 | 0.74 | 0.327 | Platelet aggregation inhibitor | 0.327 0.03 CHEMBL3548175 | CHEMBL3548175 | |
| 0.005 | 0.763 | 0.239 | Protein-tyrosine phosphatase inhibitor | 0.239 0.034 CHEMBL3548561 | CHEMBL3548561 | |
| 0.01 | 0.815 | 0.295 | Angiogenesis stimulant | 0.295 0.051 CHEMBL3549528 | CHEMBL3549528 | |
| 0.003 | 0.954 | 0.103 | Protein-tyrosine phosphatase 1B inhibitor | 0.103 0.075 CHEMBL3548561 | CHEMBL3548561 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |