Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.790.0020.816Factor Xa inhibitor

0.342 0.004 CHEMBL3548561

0.66 0.002 CHEMBL3550091

0.297 0.004 CHEMBL3549528

0.548 0.003 CHEMBL3549716

0.816 0.002 CHEMBL3548175

0.719 0.002 CHEMBL3550090

0.457 0.003 CHEMBL4525768

CHEMBL3548175
0.570.0030.57Factor X inhibitor

0.483 0.004 CHEMBL3548561

0.488 0.004 CHEMBL3550091

0.206 0.005 CHEMBL3549528

0.427 0.004 CHEMBL3549716

0.346 0.004 CHEMBL3548175

0.509 0.004 CHEMBL3550090

0.361 0.004 CHEMBL4525768

0.3990.0160.661Anticoagulant

0.372 0.019 CHEMBL3548561

0.389 0.017 CHEMBL3550091

0.385 0.018 CHEMBL3549528

0.391 0.017 CHEMBL3549716

0.661 0.005 CHEMBL3548175

0.407 0.016 CHEMBL3550090

0.337 0.023 CHEMBL4525768

CHEMBL3548175
0.4010.060.557Toll-Like receptor 7 agonist

0.557 0.023 CHEMBL3548561

0.365 0.075 CHEMBL3550091

0.421 0.052 CHEMBL3549528

0.464 0.04 CHEMBL3549716

0.412 0.055 CHEMBL3548175

0.369 0.073 CHEMBL3550090

CHEMBL3548561
0.3970.0610.554Toll-Like receptor agonist

0.554 0.023 CHEMBL3548561

0.361 0.077 CHEMBL3550091

0.422 0.052 CHEMBL3549528

0.461 0.04 CHEMBL3549716

0.407 0.058 CHEMBL3548175

0.364 0.075 CHEMBL3550090

CHEMBL3548561
0.3960.0670.56Antiobesity

0.56 0.026 CHEMBL3548561

0.349 0.088 CHEMBL3550091

0.404 0.064 CHEMBL3549716

0.413 0.061 CHEMBL3548175

0.473 0.043 CHEMBL3550090

0.208 0.199 CHEMBL4525768

CHEMBL3548561
0.2930.0050.344Glutamate (mGluR) agonist

0.331 0.005 CHEMBL3548561

0.295 0.005 CHEMBL3550091

0.058 0.048 CHEMBL3549528

0.344 0.005 CHEMBL3549716

0.144 0.015 CHEMBL3548175

0.211 0.008 CHEMBL3550090

0.192 0.01 CHEMBL4525768

CHEMBL3549716
0.2570.0050.257Interleukin 2 antagonist

0.245 0.005 CHEMBL3548561

0.247 0.005 CHEMBL3550091

0.15 0.018 CHEMBL3549528

0.225 0.005 CHEMBL3549716

0.198 0.008 CHEMBL3548175

0.243 0.005 CHEMBL3550090

0.206 0.007 CHEMBL4525768

0.2220.0080.468Glutamate receptor agonist

0.41 0.004 CHEMBL3548561

0.215 0.009 CHEMBL3550091

0.468 0.004 CHEMBL3549716

0.104 0.035 CHEMBL3550090

CHEMBL3549716
0.1740.0150.176Rho-associated kinase inhibitor

0.081 0.046 CHEMBL3548561

0.165 0.016 CHEMBL3550091

0.116 0.028 CHEMBL3549716

0.072 0.053 CHEMBL3548175

0.176 0.015 CHEMBL3550090

0.093 0.038 CHEMBL4525768

CHEMBL3550090
0.2960.1390.296MAP kinase kinase 6 inhibitor

0.268 0.169 CHEMBL3548561

0.268 0.169 CHEMBL3550091

0.265 0.172 CHEMBL3549716

0.243 0.2 CHEMBL3548175

0.296 0.139 CHEMBL3550090

0.1650.0090.165CC chemokine 6 receptor antagonist

0.165 0.01 CHEMBL3548561

0.145 0.03 CHEMBL3550091

0.156 0.016 CHEMBL3549528

0.153 0.019 CHEMBL3549716

0.156 0.016 CHEMBL3548175

0.162 0.011 CHEMBL3550090

0.144 0.032 CHEMBL4525768

0.2260.0770.244MAP-kinase-activated kinase 5 inhibitor

0.2 0.103 CHEMBL3550091

0.183 0.127 CHEMBL3549716

0.244 0.063 CHEMBL3550090

CHEMBL3550090
0.250.1080.253Nootropic

0.242 0.115 CHEMBL3550091

0.226 0.129 CHEMBL3549716

0.215 0.14 CHEMBL3548175

0.253 0.106 CHEMBL3550090

CHEMBL3550090
0.1450.0180.165Rho-associated kinase II inhibitor

0.165 0.015 CHEMBL3548561

0.133 0.021 CHEMBL3550091

0.082 0.044 CHEMBL3549716

0.125 0.023 CHEMBL3550090

0.074 0.052 CHEMBL4525768

CHEMBL3548561
0.1190.0060.119Factor IXa inhibitor

0.11 0.008 CHEMBL3548561

0.111 0.008 CHEMBL3550091

0.118 0.006 CHEMBL3549528

0.111 0.008 CHEMBL3549716

0.096 0.011 CHEMBL3548175

0.113 0.007 CHEMBL3550090

0.1 0.01 CHEMBL4525768

0.2870.1750.54Cyclophilin D inhibitor

0.54 0.04 CHEMBL3548561

0.278 0.182 CHEMBL3550091

0.276 0.185 CHEMBL3549528

0.409 0.086 CHEMBL3549716

0.324 0.142 CHEMBL3550090

CHEMBL3548561
0.2670.1690.42Analgesic

0.246 0.186 CHEMBL3550091

0.252 0.181 CHEMBL3549716

0.42 0.076 CHEMBL3548175

CHEMBL3548175
0.1330.0390.167Cyclin-dependent kinase 9 inhibitor

0.089 0.076 CHEMBL3550091

0.167 0.029 CHEMBL3550090

CHEMBL3550090
0.1580.0670.169Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.155 0.069 CHEMBL3550091

0.138 0.086 CHEMBL3549716

0.169 0.059 CHEMBL3550090

CHEMBL3550090
0.0980.0270.1Glutamate (mGluR group I) antagonist

0.097 0.028 CHEMBL3550091

0.1 0.026 CHEMBL3549716

0.078 0.039 CHEMBL3550090

CHEMBL3549716
0.1140.0510.117Chemokine receptor antagonist

0.093 0.07 CHEMBL3550091

0.117 0.05 CHEMBL3550090

CHEMBL3550090
0.0740.0140.075Chemokine receptor agonist

0.068 0.019 CHEMBL3548561

0.075 0.013 CHEMBL3550091

0.054 0.032 CHEMBL3548175

0.074 0.014 CHEMBL3550090

0.044 0.04 CHEMBL4525768

CHEMBL3550091
0.0910.0320.099CDK1/cyclin B1 inhibitor

0.069 0.049 CHEMBL3548561

0.094 0.031 CHEMBL3550091

0.071 0.047 CHEMBL3549716

0.061 0.059 CHEMBL3548175

0.099 0.029 CHEMBL3550090

CHEMBL3550090
0.1330.0770.151Aurora-C kinase inhibitor

0.151 0.049 CHEMBL3550091

0.128 0.088 CHEMBL3549716

0.14 0.064 CHEMBL3550090

0.117 0.114 CHEMBL4525768

CHEMBL3550091
0.0650.0190.065Glutamate (mGluR5) antagonist

0.064 0.02 CHEMBL3550091

0.058 0.024 CHEMBL3549716

0.049 0.03 CHEMBL3550090

0.1250.0810.14Cyclin-dependent kinase 7 inhibitor

0.126 0.079 CHEMBL3550091

0.14 0.067 CHEMBL3550090

CHEMBL3550090
0.2090.1660.345Antithrombotic

0.344 0.067 CHEMBL3548561

0.345 0.066 CHEMBL3549528

0.313 0.08 CHEMBL3549716

0.198 0.18 CHEMBL3550090

CHEMBL3549528
0.0690.0290.071Cyclin H inhibitor

0.054 0.048 CHEMBL3548561

0.07 0.028 CHEMBL3550091

0.062 0.037 CHEMBL3549716

0.055 0.046 CHEMBL3548175

0.071 0.027 CHEMBL3550090

0.058 0.042 CHEMBL4525768

CHEMBL3550090
0.0690.030.069Corticotropin releasing factor 2 receptor antagonist

0.066 0.035 CHEMBL3550091

0.063 0.04 CHEMBL3550090

0.0560.0250.113Glutamate (mGluR group I) agonist

0.089 0.01 CHEMBL3550091

0.113 0.007 CHEMBL3549716

CHEMBL3549716
0.080.0490.114Glutamate (mGluR) antagonist

0.075 0.054 CHEMBL3550091

0.114 0.028 CHEMBL3549716

CHEMBL3549716
0.0560.0280.06Phosphodiesterase 7A inhibitor

0.06 0.022 CHEMBL3548561

0.048 0.045 CHEMBL3550091

0.054 0.031 CHEMBL3550090

CHEMBL3548561
0.0650.0380.132Neuraminidase inhibitor

0.104 0.014 CHEMBL3548561

0.062 0.041 CHEMBL3550091

0.064 0.038 CHEMBL3549528

0.132 0.008 CHEMBL3549716

0.057 0.047 CHEMBL3548175

0.069 0.034 CHEMBL3550090

CHEMBL3549716
0.0660.040.137Neuraminidase (influenza) inhibitor

0.095 0.018 CHEMBL3548561

0.063 0.047 CHEMBL3550091

0.068 0.038 CHEMBL3549528

0.137 0.009 CHEMBL3549716

0.063 0.047 CHEMBL3548175

0.069 0.036 CHEMBL3550090

CHEMBL3549716
0.0410.0150.041CXC chemokine receptor agonist

0.039 0.018 CHEMBL3548561

0.041 0.013 CHEMBL3550091

0.041 0.015 CHEMBL3550090

0.0330.0080.033Hexokinase stimulant

0.02 0.013 CHEMBL3550091

0.023 0.012 CHEMBL3549716

0.025 0.01 CHEMBL3550090

0.050.0260.092Glutamate (mGluR5) agonist

0.047 0.03 CHEMBL3550091

0.092 0.008 CHEMBL3549716

CHEMBL3549716
0.0480.0260.052Baculoviral IAP repeat-containing protein inhibitor

0.052 0.015 CHEMBL3550091

0.044 0.041 CHEMBL3549716

0.048 0.027 CHEMBL3550090

CHEMBL3550091
0.0640.0420.064Phosphodiesterase VII inhibitor

0.063 0.043 CHEMBL3548561

0.030.0130.035 Hydroxytryptamine 1F agonist

0.028 0.015 CHEMBL3550091

0.1390.1250.139Cyclin-dependent kinase 3 inhibitor

0.139 0.126 CHEMBL3550091

0.0610.0480.063Prolactin release inhibitor

0.063 0.039 CHEMBL3548561

CHEMBL3548561
0.0570.050.094Tyk2 inhibitor

0.094 0.03 CHEMBL3550091

0.064 0.045 CHEMBL3550090

CHEMBL3550091
0.0410.040.072Neuraminidase (Influenza A) inhibitor

0.064 0.01 CHEMBL3548561

0.044 0.034 CHEMBL3549528

0.072 0.006 CHEMBL3549716

0.043 0.037 CHEMBL3550090

CHEMBL3549716
0.0410.040.041Dipeptidyl peptidase IV inhibitor
0.0090.0090.01Baculoviral IAP repeat-containing protein 2 inhibitor

0.01 0.005 CHEMBL3550091

CHEMBL3550091
0.0640.0650.105Rho-associated kinase I inhibitor

0.068 0.06 CHEMBL3550091

0.105 0.029 CHEMBL3550090

CHEMBL3550090
0.0770.0880.084MAP kinase 9 inhibitor

0.084 0.078 CHEMBL3550091

CHEMBL3550091
0.060.090.085ALK inhibitor

0.085 0.054 CHEMBL3550091

CHEMBL3550091
0.0290.0830.037Integrin alpha1beta1 antagonist

0.036 0.034 CHEMBL3548561

0.037 0.029 CHEMBL3550091

CHEMBL3550091
0.0390.0940.078Lipase inhibitor

0.078 0.045 CHEMBL3548561

CHEMBL3548561
0.0070.1520.03Diacylglycerol O-acyltransferase 1 inhibitor

0.03 0.019 CHEMBL3549716

CHEMBL3549716
0.0460.210.117Glutamate receptor antagonist

0.117 0.078 CHEMBL3549716

CHEMBL3549716
0.0490.2410.136Thrombolytic

0.127 0.102 CHEMBL3548561

0.136 0.093 CHEMBL3549528

CHEMBL3549528
0.1170.3240.249Peptidyltransferase inhibitor

0.249 0.051 CHEMBL3549528

CHEMBL3549528
0.0190.2270.141Myc inhibitor

0.141 0.005 CHEMBL3550090

CHEMBL3550090
0.0620.3360.143Polo-like kinase-3 inhibitor

0.143 0.092 CHEMBL3548175

CHEMBL3548175
0.0040.5250.021Adenosine A1 receptor agonist

0.021 0.02 CHEMBL3549528

CHEMBL3549528
0.0210.5910.145Cell wall synthesis inhibitor

0.145 0.07 CHEMBL3548561

CHEMBL3548561
0.0170.6190.459Platelet antagonist

0.459 0.018 CHEMBL3548175

CHEMBL3548175
0.0110.740.327Platelet aggregation inhibitor

0.327 0.03 CHEMBL3548175

CHEMBL3548175
0.0050.7630.239Protein-tyrosine phosphatase inhibitor

0.239 0.034 CHEMBL3548561

CHEMBL3548561
0.010.8150.295Angiogenesis stimulant

0.295 0.051 CHEMBL3549528

CHEMBL3549528
0.0030.9540.103Protein-tyrosine phosphatase 1B inhibitor

0.103 0.075 CHEMBL3548561

CHEMBL3548561
Ext Pa Pi Pmax Activity Other Results ID Pa_max