| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.525 | 0.005 | 0.563 | Insulin secretagoues | 0.306 0.012 CHEMBL3527366 0.504 0.005 CHEMBL4525741 0.563 0.004 CHEMBL3526588 0.493 0.005 CHEMBL4525742 0.469 0.005 CHEMBL3526452 0.382 0.007 CHEMBL4525743 0.198 0.037 CHEMBL4525744 0.331 0.009 CHEMBL3526587 | CHEMBL3526588 | |
| 0.327 | 0.036 | 0.432 | Interleukin agonist | 0.31 0.043 CHEMBL3527366 0.356 0.027 CHEMBL4525741 0.432 0.015 CHEMBL3526588 0.348 0.03 CHEMBL4525742 0.33 0.035 CHEMBL3526452 0.174 0.145 CHEMBL4525743 0.322 0.038 CHEMBL3526587 | CHEMBL3526588 | |
| 0.348 | 0.088 | 0.4 | Antiobesity | 0.322 0.102 CHEMBL4525741 0.353 0.086 CHEMBL3526588 0.344 0.09 CHEMBL4525742 0.4 0.065 CHEMBL3526452 | CHEMBL3526452 | |
| 0.328 | 0.075 | 0.609 | Cholesterol antagonist | 0.33 0.073 CHEMBL3527366 0.283 0.103 CHEMBL4525741 0.609 0.017 CHEMBL3526588 0.326 0.076 CHEMBL4525742 0.347 0.066 CHEMBL3526452 0.222 0.146 CHEMBL4525744 0.51 0.031 CHEMBL3526587 | CHEMBL3526588 | |
| 0.321 | 0.072 | 0.424 | Calcium channel activator | 0.3 0.091 CHEMBL3527366 0.424 0.017 CHEMBL4525741 0.28 0.113 CHEMBL4525742 0.296 0.096 CHEMBL3526452 | CHEMBL4525741 | |
| 0.263 | 0.044 | 0.263 | Neuropeptide Y2 antagonist | 0.21 0.103 CHEMBL3527366 0.201 0.118 CHEMBL4525741 0.247 0.06 CHEMBL4525742 0.224 0.084 CHEMBL3526587 | ||
| 0.293 | 0.079 | 0.429 | Interleukin 2 agonist | 0.301 0.073 CHEMBL3527366 0.252 0.116 CHEMBL4525741 0.429 0.02 CHEMBL3526588 0.346 0.047 CHEMBL4525742 0.318 0.062 CHEMBL3526452 0.251 0.117 CHEMBL4525743 0.239 0.131 CHEMBL4525744 0.322 0.059 CHEMBL3526587 | CHEMBL3526588 | |
| 0.339 | 0.126 | 0.367 | Calcium channel L-type activator | 0.367 0.105 CHEMBL3527366 0.321 0.14 CHEMBL4525741 0.349 0.118 CHEMBL4525742 0.262 0.193 CHEMBL3526452 0.266 0.188 CHEMBL4525743 | CHEMBL3527366 | |
| 0.296 | 0.09 | 0.682 | Antithrombotic | 0.269 0.112 CHEMBL3527366 0.277 0.106 CHEMBL4525741 0.682 0.009 CHEMBL3526588 0.277 0.106 CHEMBL4525742 0.317 0.078 CHEMBL3526452 0.295 0.091 CHEMBL4525744 0.453 0.037 CHEMBL3526587 | CHEMBL3526588 | |
| 0.276 | 0.074 | 0.34 | Insulysin inhibitor | 0.217 0.133 CHEMBL3527366 0.34 0.038 CHEMBL4525742 0.263 0.085 CHEMBL3526587 | CHEMBL4525742 | |
| 0.333 | 0.131 | 0.409 | 5 Hydroxytryptamine release inhibitor | 0.409 0.073 CHEMBL3527366 0.268 0.204 CHEMBL4525742 0.246 0.233 CHEMBL4525744 0.338 0.126 CHEMBL3526587 | CHEMBL3527366 | |
| 0.263 | 0.065 | 0.349 | Gastrin inhibitor | 0.28 0.048 CHEMBL3527366 0.207 0.139 CHEMBL4525741 0.275 0.053 CHEMBL4525742 0.213 0.129 CHEMBL3526452 0.195 0.156 CHEMBL4525744 0.349 0.011 CHEMBL3526587 | CHEMBL3526587 | |
| 0.268 | 0.083 | 0.464 | Spasmolytic | 0.192 0.127 CHEMBL3527366 0.216 0.108 CHEMBL4525741 0.464 0.028 CHEMBL3526588 0.22 0.105 CHEMBL4525742 0.352 0.052 CHEMBL3526452 0.169 0.146 CHEMBL3526587 | CHEMBL3526588 | |
| 0.264 | 0.08 | 0.264 | Ca(v)3.3 blocker | 0.254 0.095 CHEMBL3527366 0.255 0.094 CHEMBL4525741 0.237 0.121 CHEMBL4525742 0.221 0.15 CHEMBL3526452 0.221 0.15 CHEMBL4525743 0.246 0.107 CHEMBL4525744 0.253 0.097 CHEMBL3526587 | ||
| 0.255 | 0.074 | 0.474 | Hypoglycemic | 0.227 0.091 CHEMBL3527366 0.228 0.091 CHEMBL4525741 0.474 0.018 CHEMBL3526588 0.21 0.104 CHEMBL4525742 0.264 0.069 CHEMBL3526452 0.242 0.082 CHEMBL4525743 0.245 0.08 CHEMBL3526587 | CHEMBL3526588 | |
| 0.256 | 0.079 | 0.333 | Transcription factor STAT3 inhibitor | 0.222 0.109 CHEMBL3527366 0.333 0.039 CHEMBL4525742 0.191 0.147 CHEMBL3526452 0.197 0.138 CHEMBL4525743 0.193 0.144 CHEMBL3526587 | CHEMBL4525742 | |
| 0.319 | 0.146 | 0.59 | Cyclophilin D inhibitor | 0.381 0.102 CHEMBL4525741 0.59 0.029 CHEMBL3526588 0.279 0.182 CHEMBL4525742 0.386 0.099 CHEMBL3526452 0.278 0.183 CHEMBL3526587 | CHEMBL3526588 | |
| 0.199 | 0.035 | 0.224 | Neurotensin receptor agonist | 0.206 0.032 CHEMBL3527366 0.224 0.026 CHEMBL4525742 0.14 0.13 CHEMBL3526452 0.149 0.103 CHEMBL4525744 0.216 0.028 CHEMBL3526587 | CHEMBL4525742 | |
| 0.219 | 0.056 | 0.308 | Insulin sensitizer | 0.26 0.029 CHEMBL3527366 0.189 0.085 CHEMBL4525741 0.158 0.123 CHEMBL4525742 0.199 0.075 CHEMBL3526452 0.181 0.094 CHEMBL4525744 0.308 0.014 CHEMBL3526587 | CHEMBL3526587 | |
| 0.205 | 0.042 | 0.218 | Diuretic | 0.21 0.04 CHEMBL3527366 0.13 0.094 CHEMBL4525741 0.176 0.057 CHEMBL3526588 0.178 0.055 CHEMBL4525742 0.166 0.064 CHEMBL3526452 0.117 0.109 CHEMBL4525743 0.218 0.038 CHEMBL3526587 | CHEMBL3526587 | |
| 0.269 | 0.108 | 0.356 | Sodium/bile acid cotransporter inhibitor | 0.282 0.096 CHEMBL3527366 0.239 0.14 CHEMBL4525741 0.309 0.071 CHEMBL4525742 0.312 0.069 CHEMBL3526452 0.228 0.153 CHEMBL4525743 0.284 0.094 CHEMBL4525744 0.356 0.036 CHEMBL3526587 | CHEMBL3526587 | |
| 0.171 | 0.017 | 0.249 | Caspase 3 inhibitor | 0.167 0.018 CHEMBL3527366 0.111 0.074 CHEMBL4525741 0.171 0.017 CHEMBL4525742 0.128 0.048 CHEMBL3526452 0.237 0.005 CHEMBL4525744 0.249 0.005 CHEMBL3526587 | CHEMBL3526587 | |
| 0.266 | 0.112 | 0.434 | Apoptosis antagonist | 0.291 0.091 CHEMBL3527366 0.201 0.177 CHEMBL4525741 0.434 0.03 CHEMBL3526588 0.284 0.097 CHEMBL4525742 0.276 0.103 CHEMBL3526452 0.24 0.138 CHEMBL4525743 0.297 0.087 CHEMBL4525744 0.342 0.06 CHEMBL3526587 | CHEMBL3526588 | |
| 0.155 | 0.008 | 0.165 | Prostaglandin E2 antagonist | 0.165 0.007 CHEMBL3527366 0.103 0.014 CHEMBL4525741 0.106 0.013 CHEMBL4525742 0.11 0.013 CHEMBL3526452 0.073 0.022 CHEMBL4525743 0.088 0.017 CHEMBL4525744 0.163 0.008 CHEMBL3526587 | CHEMBL3527366 | |
| 0.183 | 0.037 | 0.261 | Anesthetic local | 0.261 0.018 CHEMBL3527366 0.144 0.052 CHEMBL4525741 0.106 0.077 CHEMBL4525742 0.145 0.051 CHEMBL3526452 0.114 0.071 CHEMBL4525743 0.246 0.021 CHEMBL4525744 0.228 0.025 CHEMBL3526587 | CHEMBL3527366 | |
| 0.188 | 0.044 | 0.244 | Thiol protease inhibitor | 0.18 0.048 CHEMBL3527366 0.197 0.04 CHEMBL4525742 0.244 0.028 CHEMBL4525744 0.239 0.029 CHEMBL3526587 | CHEMBL4525744 | |
| 0.23 | 0.09 | 0.261 | Tyrosine 3 hydroxylase inhibitor | 0.244 0.075 CHEMBL3527366 0.217 0.108 CHEMBL4525741 0.261 0.058 CHEMBL4525742 0.211 0.118 CHEMBL3526587 | CHEMBL4525742 | |
| 0.144 | 0.006 | 0.168 | Neuraminidase inhibitor | 0.168 0.005 CHEMBL3527366 0.088 0.02 CHEMBL4525741 0.14 0.007 CHEMBL3526588 0.159 0.005 CHEMBL4525742 0.148 0.006 CHEMBL3526452 0.128 0.009 CHEMBL4525743 0.139 0.007 CHEMBL4525744 0.147 0.006 CHEMBL3526587 | CHEMBL3527366 | |
| 0.271 | 0.134 | 0.408 | Calpain 2 inhibitor | 0.266 0.138 CHEMBL3527366 0.408 0.057 CHEMBL4525744 0.29 0.121 CHEMBL3526587 | CHEMBL4525744 | |
| 0.161 | 0.039 | 0.263 | Cyclooxygenase 3 inhibitor | 0.207 0.016 CHEMBL3527366 0.115 0.083 CHEMBL4525741 0.263 0.008 CHEMBL3526588 0.155 0.044 CHEMBL4525742 0.164 0.038 CHEMBL3526452 0.102 0.1 CHEMBL4525744 0.182 0.027 CHEMBL3526587 | CHEMBL3526588 | |
| 0.227 | 0.105 | 0.339 | Transcription factor STAT inhibitor | 0.193 0.149 CHEMBL3527366 0.339 0.038 CHEMBL4525742 0.196 0.144 CHEMBL3526452 | CHEMBL4525742 | |
| 0.129 | 0.01 | 0.167 | Neuraminidase (influenza) inhibitor | 0.167 0.006 CHEMBL3527366 0.077 0.028 CHEMBL4525741 0.143 0.008 CHEMBL3526588 0.156 0.007 CHEMBL4525742 0.136 0.009 CHEMBL3526452 0.121 0.012 CHEMBL4525743 0.135 0.009 CHEMBL4525744 0.142 0.008 CHEMBL3526587 | CHEMBL3527366 | |
| 0.263 | 0.146 | 0.392 | Histamine release inhibitor | 0.384 0.084 CHEMBL3527366 0.274 0.139 CHEMBL3526588 0.206 0.194 CHEMBL4525742 0.392 0.08 CHEMBL3526587 | CHEMBL3526587 | |
| 0.157 | 0.043 | 0.246 | Cell adhesion inhibitor | 0.161 0.04 CHEMBL3527366 0.118 0.066 CHEMBL4525741 0.239 0.016 CHEMBL3526588 0.17 0.035 CHEMBL4525742 0.169 0.036 CHEMBL3526452 0.12 0.065 CHEMBL4525744 0.246 0.015 CHEMBL3526587 | CHEMBL3526587 | |
| 0.173 | 0.06 | 0.224 | Protein-tyrosine phosphatase inhibitor | 0.211 0.043 CHEMBL3527366 0.172 0.061 CHEMBL4525741 0.185 0.053 CHEMBL3526588 0.2 0.046 CHEMBL4525742 0.156 0.072 CHEMBL3526452 0.155 0.074 CHEMBL4525744 0.224 0.038 CHEMBL3526587 | CHEMBL3526587 | |
| 0.203 | 0.098 | 0.369 | Platelet antagonist | 0.199 0.101 CHEMBL3527366 0.19 0.109 CHEMBL4525741 0.3 0.053 CHEMBL3526588 0.183 0.115 CHEMBL4525742 0.217 0.09 CHEMBL3526452 0.166 0.129 CHEMBL4525744 0.369 0.034 CHEMBL3526587 | CHEMBL3526587 | |
| 0.165 | 0.062 | 0.282 | Phospholipase A2 inhibitor | 0.209 0.038 CHEMBL3527366 0.157 0.068 CHEMBL4525741 0.143 0.082 CHEMBL4525742 0.208 0.038 CHEMBL4525744 0.282 0.016 CHEMBL3526587 | CHEMBL3526587 | |
| 0.149 | 0.066 | 0.149 | Neuropeptide Y1 antagonist | 0.136 0.088 CHEMBL4525742 | ||
| 0.09 | 0.01 | 0.114 | Melanocortin 4 antagonist | 0.054 0.021 CHEMBL4525741 0.05 0.023 CHEMBL3526588 0.114 0.008 CHEMBL4525742 0.075 0.013 CHEMBL3526452 0.07 0.015 CHEMBL4525743 | CHEMBL4525742 | |
| 0.195 | 0.118 | 0.268 | Calpain inhibitor | 0.221 0.094 CHEMBL3527366 0.18 0.135 CHEMBL4525742 0.268 0.05 CHEMBL4525744 0.224 0.09 CHEMBL3526587 | CHEMBL4525744 | |
| 0.131 | 0.057 | 0.158 | Proteasome inhibitor | 0.131 0.058 CHEMBL3527366 0.095 0.094 CHEMBL4525741 0.158 0.042 CHEMBL4525742 0.15 0.046 CHEMBL4525744 0.136 0.054 CHEMBL3526587 | CHEMBL4525742 | |
| 0.169 | 0.095 | 0.238 | Anesthetic general | 0.227 0.061 CHEMBL3527366 0.238 0.056 CHEMBL4525741 0.21 0.069 CHEMBL3526588 0.177 0.089 CHEMBL4525742 0.161 0.103 CHEMBL3526452 0.162 0.101 CHEMBL4525743 0.187 0.082 CHEMBL3526587 | CHEMBL4525741 | |
| 0.104 | 0.032 | 0.179 | Cell adhesion molecule inhibitor | 0.108 0.029 CHEMBL3527366 0.084 0.049 CHEMBL4525741 0.156 0.014 CHEMBL3526588 0.11 0.028 CHEMBL4525742 0.119 0.024 CHEMBL3526452 0.081 0.052 CHEMBL4525744 0.179 0.011 CHEMBL3526587 | CHEMBL3526587 | |
| 0.151 | 0.079 | 0.248 | Anticoagulant | 0.168 0.067 CHEMBL3527366 0.134 0.095 CHEMBL4525741 0.248 0.039 CHEMBL3526588 0.155 0.076 CHEMBL4525742 0.142 0.088 CHEMBL3526452 0.206 0.051 CHEMBL4525743 0.188 0.058 CHEMBL4525744 0.224 0.045 CHEMBL3526587 | CHEMBL3526588 | |
| 0.134 | 0.062 | 0.149 | Antibacterial (Helicobacter pylori) | 0.114 0.091 CHEMBL3527366 0.132 0.065 CHEMBL4525742 0.118 0.085 CHEMBL3526452 0.149 0.047 CHEMBL3526587 | CHEMBL3526587 | |
| 0.252 | 0.181 | 0.288 | Analgesic | 0.22 0.214 CHEMBL4525741 0.261 0.174 CHEMBL4525742 0.288 0.151 CHEMBL3526452 | CHEMBL3526452 | |
| 0.081 | 0.014 | 0.099 | Melanocortin antagonist | 0.052 0.027 CHEMBL4525741 0.05 0.03 CHEMBL3526588 0.099 0.012 CHEMBL4525742 0.066 0.018 CHEMBL3526452 0.062 0.02 CHEMBL4525743 | CHEMBL4525742 | |
| 0.072 | 0.006 | 0.082 | Neuraminidase (Influenza A) inhibitor | 0.082 0.005 CHEMBL3527366 0.056 0.016 CHEMBL4525741 0.073 0.006 CHEMBL3526588 0.077 0.005 CHEMBL4525742 0.069 0.007 CHEMBL3526452 0.062 0.011 CHEMBL4525743 0.066 0.009 CHEMBL4525744 0.071 0.007 CHEMBL3526587 | CHEMBL3527366 | |
| 0.073 | 0.013 | 0.082 | Adenine nucleotide translocase inhibitor | 0.082 0.008 CHEMBL3527366 0.065 0.02 CHEMBL4525741 0.074 0.012 CHEMBL3526588 0.079 0.009 CHEMBL4525742 0.069 0.016 CHEMBL3526452 0.07 0.015 CHEMBL4525743 0.074 0.012 CHEMBL4525744 0.082 0.008 CHEMBL3526587 | CHEMBL3526587 | |
| 0.066 | 0.008 | 0.105 | Prostaglandin EP3 antagonist | 0.081 0.007 CHEMBL3527366 0.047 0.011 CHEMBL4525741 0.065 0.008 CHEMBL4525742 0.05 0.01 CHEMBL3526452 0.041 0.014 CHEMBL4525743 0.043 0.013 CHEMBL4525744 0.105 0.005 CHEMBL3526587 | CHEMBL3526587 | |
| 0.088 | 0.04 | 0.093 | Ca(v)3.1 blocker | 0.093 0.031 CHEMBL4525742 | CHEMBL4525742 | |
| 0.136 | 0.088 | 0.151 | Sphingosine 1-phosphate receptor 5 antagonist | 0.131 0.098 CHEMBL3527366 0.151 0.059 CHEMBL3526587 | CHEMBL3526587 | |
| 0.124 | 0.078 | 0.14 | Vanilloid 1 agonist | 0.114 0.102 CHEMBL3527366 0.112 0.109 CHEMBL4525741 0.124 0.077 CHEMBL3526588 0.134 0.059 CHEMBL4525742 0.113 0.107 CHEMBL3526452 0.14 0.05 CHEMBL3526587 | CHEMBL3526587 | |
| 0.098 | 0.06 | 0.16 | Interleukin 1 beta converting enzyme inhibitor | 0.122 0.034 CHEMBL3527366 0.087 0.078 CHEMBL4525742 0.156 0.015 CHEMBL4525744 0.16 0.014 CHEMBL3526587 | CHEMBL3526587 | |
| 0.066 | 0.028 | 0.109 | Prostaglandin antagonist | 0.057 0.034 CHEMBL3527366 0.047 0.043 CHEMBL4525741 0.109 0.015 CHEMBL3526587 | CHEMBL3526587 | |
| 0.12 | 0.086 | 0.151 | Interleukin 4 antagonist | 0.111 0.099 CHEMBL3527366 0.115 0.092 CHEMBL4525741 0.131 0.07 CHEMBL3526588 0.151 0.049 CHEMBL4525742 0.123 0.081 CHEMBL3526452 0.111 0.1 CHEMBL3526587 | CHEMBL4525742 | |
| 0.086 | 0.053 | 0.115 | 3C-Like protease (SARS coronavirus) inhibitor | 0.086 0.053 CHEMBL3527366 0.093 0.042 CHEMBL4525742 0.079 0.071 CHEMBL3526452 0.115 0.022 CHEMBL4525744 0.08 0.07 CHEMBL3526587 | CHEMBL4525744 | |
| 0.145 | 0.113 | 0.215 | Lipocortins synthesis antagonist | 0.215 0.048 CHEMBL3527366 0.157 0.095 CHEMBL4525741 0.153 0.1 CHEMBL4525742 0.181 0.07 CHEMBL3526452 0.192 0.061 CHEMBL3526587 | CHEMBL3527366 | |
| 0.071 | 0.04 | 0.075 | Potassium channel (ATP-sensitive) blocker | 0.075 0.033 CHEMBL3527366 0.073 0.036 CHEMBL4525741 | CHEMBL3527366 | |
| 0.13 | 0.1 | 0.23 | Thrombolytic | 0.127 0.102 CHEMBL3527366 0.23 0.039 CHEMBL3526588 0.144 0.087 CHEMBL4525742 0.151 0.081 CHEMBL3526452 0.187 0.058 CHEMBL3526587 | CHEMBL3526588 | |
| 0.102 | 0.076 | 0.154 | Protein-tyrosine phosphatase 1B inhibitor | 0.135 0.052 CHEMBL3527366 0.104 0.075 CHEMBL4525741 0.139 0.05 CHEMBL3526588 0.118 0.064 CHEMBL4525742 0.094 0.085 CHEMBL3526452 0.097 0.081 CHEMBL4525744 0.154 0.044 CHEMBL3526587 | CHEMBL3526587 | |
| 0.048 | 0.022 | 0.054 | GHS receptor agonist | 0.054 0.017 CHEMBL4525742 | CHEMBL4525742 | |
| 0.204 | 0.179 | 0.374 | Vasodilator, coronary | 0.214 0.17 CHEMBL4525741 0.374 0.044 CHEMBL3526588 | CHEMBL3526588 | |
| 0.111 | 0.088 | 0.154 | Toll-Like receptor 2 antagonist | 0.154 0.05 CHEMBL4525742 0.142 0.059 CHEMBL3526587 | CHEMBL4525742 | |
| 0.036 | 0.012 | 0.077 | Prostaglandin EP4 antagonist | 0.023 0.022 CHEMBL4525741 0.031 0.015 CHEMBL3526452 0.077 0.005 CHEMBL3526587 | CHEMBL3526587 | |
| 0.028 | 0.005 | 0.043 | Neuraminidase (Influenza B) inhibitor | 0.043 0.003 CHEMBL3527366 0.028 0.005 CHEMBL4525742 0.024 0.009 CHEMBL3526452 0.026 0.007 CHEMBL4525744 0.029 0.005 CHEMBL3526587 | CHEMBL3527366 | |
| 0.115 | 0.093 | 0.115 | Calcium channel blocker | |||
| 0.137 | 0.117 | 0.175 | Amyloid beta precursor protein antagonist | 0.175 0.077 CHEMBL3527366 0.149 0.103 CHEMBL4525742 | CHEMBL3527366 | |
| 0.109 | 0.09 | 0.144 | M17 leucyl aminopeptidase inhibitor | 0.144 0.059 CHEMBL3527366 0.131 0.069 CHEMBL3526587 | CHEMBL3527366 | |
| 0.171 | 0.153 | 0.236 | Superoxide dismutase inhibitor | 0.236 0.084 CHEMBL3527366 0.185 0.136 CHEMBL4525742 0.184 0.136 CHEMBL4525744 | CHEMBL3527366 | |
| 0.1 | 0.084 | 0.1 | Calcium channel (voltage-sensitive) blocker | |||
| 0.054 | 0.039 | 0.077 | Matrix metalloproteinase (membrane-type) inhibitor | 0.072 0.023 CHEMBL3527366 0.051 0.044 CHEMBL4525742 0.077 0.021 CHEMBL3526587 | CHEMBL3526587 | |
| 0.036 | 0.023 | 0.036 | Tryptophan 5 hydroxylase inhibitor | |||
| 0.081 | 0.068 | 0.09 | Vanilloid agonist | 0.082 0.065 CHEMBL3527366 0.09 0.046 CHEMBL4525742 0.088 0.05 CHEMBL3526587 | CHEMBL4525742 | |
| 0.031 | 0.02 | 0.031 | Potassium channel subfamily K member 3 blocker | 0.031 0.02 CHEMBL4525741 0.029 0.023 CHEMBL4525742 | ||
| 0.068 | 0.056 | 0.093 | Aminopeptidase I inhibitor | 0.08 0.042 CHEMBL3527366 0.093 0.032 CHEMBL4525742 0.068 0.056 CHEMBL3526587 | CHEMBL4525742 | |
| 0.059 | 0.048 | 0.089 | Prostaglandin F2 alpha antagonist | 0.056 0.054 CHEMBL3527366 0.057 0.052 CHEMBL4525742 0.065 0.039 CHEMBL3526452 0.089 0.017 CHEMBL3526587 | CHEMBL3526587 | |
| 0.053 | 0.042 | 0.067 | DNA helicase inhibitor | 0.059 0.03 CHEMBL3527366 0.052 0.044 CHEMBL4525741 0.067 0.019 CHEMBL4525742 0.058 0.031 CHEMBL3526587 | CHEMBL4525742 | |
| 0.04 | 0.031 | 0.14 | Integrin antagonist | 0.044 0.029 CHEMBL3527366 0.052 0.027 CHEMBL4525742 0.14 0.011 CHEMBL3526587 | CHEMBL3526587 | |
| 0.027 | 0.018 | 0.034 | Urotensin II agonist | 0.029 0.016 CHEMBL3527366 0.034 0.013 CHEMBL4525742 0.033 0.013 CHEMBL3526587 | CHEMBL4525742 | |
| 0.04 | 0.031 | 0.044 | Acetyl-CoA carboxylase inhibitor | 0.041 0.029 CHEMBL4525741 0.044 0.026 CHEMBL3526452 | CHEMBL3526452 | |
| 0.06 | 0.052 | 0.066 | Protease 3C (Human rhinovirus) inhibitor | 0.066 0.043 CHEMBL3527366 | CHEMBL3527366 | |
| 0.086 | 0.078 | 0.106 | Protease inhibitor | 0.106 0.061 CHEMBL3527366 0.092 0.072 CHEMBL4525742 0.09 0.074 CHEMBL3526452 0.086 0.079 CHEMBL4525743 0.1 0.065 CHEMBL4525744 0.095 0.07 CHEMBL3526587 | CHEMBL3527366 | |
| 0.067 | 0.061 | 0.098 | Peroxisome proliferator-activated receptor gamma antagonist | 0.081 0.032 CHEMBL3527366 0.068 0.058 CHEMBL4525741 0.098 0.016 CHEMBL3526587 | CHEMBL3526587 | |
| 0.014 | 0.01 | 0.018 | Integrin beta6 antagonist | 0.015 0.008 CHEMBL3527366 0.013 0.012 CHEMBL4525741 0.016 0.007 CHEMBL4525742 0.014 0.012 CHEMBL3526452 0.014 0.011 CHEMBL4525744 0.018 0.005 CHEMBL3526587 | CHEMBL3526587 | |
| 0.191 | 0.187 | 0.315 | Vasodilator, peripheral | 0.19 0.188 CHEMBL4525741 0.315 0.09 CHEMBL3526588 | CHEMBL3526588 | |
| 0.103 | 0.101 | 0.136 | Cathepsin H inhibitor | 0.136 0.058 CHEMBL3527366 0.135 0.058 CHEMBL4525742 0.115 0.082 CHEMBL4525744 | CHEMBL3527366 | |
| 0.071 | 0.069 | 0.091 | Sphingosine 1-phosphate receptor antagonist | 0.091 0.029 CHEMBL3526587 | CHEMBL3526587 | |
| 0.016 | 0.015 | 0.016 | Tryptophan hydroxylase 1 inhibitor | |||
| 0.03 | 0.03 | 0.05 | Kainate receptor 2 antagonist | 0.031 0.03 CHEMBL3527366 0.044 0.019 CHEMBL4525742 0.05 0.016 CHEMBL3526587 | CHEMBL3526587 | |
| 0.037 | 0.037 | 0.083 | Leukocyte elastase inhibitor | 0.038 0.036 CHEMBL3527366 0.083 0.012 CHEMBL4525743 | CHEMBL4525743 | |
| 0.018 | 0.018 | 0.034 | Caspase 8 inhibitor | 0.02 0.012 CHEMBL3527366 0.026 0.007 CHEMBL4525744 0.034 0.004 CHEMBL3526587 | CHEMBL3526587 | |
| 0.02 | 0.022 | 0.025 | Beta 1 adrenoreceptor agonist | 0.025 0.012 CHEMBL3527366 0.022 0.017 CHEMBL4525742 0.022 0.017 CHEMBL3526587 | CHEMBL3527366 | |
| 0.081 | 0.083 | 0.132 | ABCA1 expression enhancer | 0.094 0.058 CHEMBL3527366 0.096 0.056 CHEMBL4525741 0.132 0.024 CHEMBL4525744 | CHEMBL4525744 | |
| 0.012 | 0.014 | 0.075 | Integrin alpha4beta1 antagonist | 0.015 0.011 CHEMBL4525742 0.075 0.004 CHEMBL3526587 | CHEMBL3526587 | |
| 0.137 | 0.14 | 0.167 | Catenin beta inhibitor | 0.15 0.105 CHEMBL3527366 0.164 0.076 CHEMBL4525742 0.167 0.072 CHEMBL3526587 | CHEMBL3526587 | |
| 0.032 | 0.035 | 0.107 | Factor VIIa inhibitor | 0.107 0.011 CHEMBL3527366 0.059 0.018 CHEMBL4525744 0.091 0.013 CHEMBL3526587 | CHEMBL3527366 | |
| 0.019 | 0.022 | 0.062 | Integrin alpha4 antagonist | 0.021 0.02 CHEMBL3527366 0.026 0.017 CHEMBL4525742 0.062 0.009 CHEMBL3526587 | CHEMBL3526587 | |
| 0.035 | 0.038 | 0.037 | Integrin alpha1beta1 antagonist | 0.037 0.031 CHEMBL4525742 0.036 0.035 CHEMBL3526587 | CHEMBL4525742 | |
| 0.046 | 0.049 | 0.05 | Factor III inhibitor | 0.049 0.037 CHEMBL3527366 0.05 0.033 CHEMBL4525742 | CHEMBL4525742 | |
| 0.042 | 0.047 | 0.046 | Beta adrenoreceptor agonist | 0.046 0.027 CHEMBL3527366 0.045 0.03 CHEMBL4525742 0.046 0.028 CHEMBL3526587 | CHEMBL3526587 | |
| 0.076 | 0.082 | 0.118 | Estrogen-related receptor beta agonist | 0.118 0.011 CHEMBL3527366 0.085 0.053 CHEMBL4525742 0.082 0.062 CHEMBL3526587 | CHEMBL3527366 | |
| 0.134 | 0.142 | 0.294 | Non-steroidal antiinflammatory agent | 0.144 0.123 CHEMBL3527366 0.294 0.029 CHEMBL3526588 0.154 0.11 CHEMBL4525742 0.142 0.127 CHEMBL3526587 | CHEMBL3526588 | |
| 0.047 | 0.055 | 0.066 | Cathepsin L inhibitor | 0.061 0.037 CHEMBL4525742 0.066 0.033 CHEMBL4525744 | CHEMBL4525744 | |
| 0.027 | 0.035 | 0.042 | Leukotriene A4 hydrolase inhibitor | 0.042 0.024 CHEMBL3526587 | CHEMBL3526587 | |
| 0.077 | 0.086 | 0.137 | Aminopeptidase B inhibitor | 0.134 0.045 CHEMBL3527366 0.113 0.057 CHEMBL4525742 0.111 0.058 CHEMBL4525744 0.137 0.044 CHEMBL3526587 | CHEMBL3526587 | |
| 0.15 | 0.159 | 0.37 | Tumour necrosis factor alpha release inhibitor | 0.37 0.033 CHEMBL3526588 0.195 0.114 CHEMBL3526452 | CHEMBL3526588 | |
| 0.017 | 0.026 | 0.046 | VLA-4 antagonist | 0.022 0.021 CHEMBL4525742 0.046 0.014 CHEMBL3526587 | CHEMBL3526587 | |
| 0.036 | 0.045 | 0.041 | VCAM-1 antagonist | 0.038 0.033 CHEMBL3527366 0.037 0.035 CHEMBL4525742 0.037 0.035 CHEMBL4525744 0.041 0.021 CHEMBL3526587 | CHEMBL3526587 | |
| 0.035 | 0.046 | 0.041 | VCAM antagonist | 0.038 0.033 CHEMBL3527366 0.037 0.035 CHEMBL4525742 0.037 0.036 CHEMBL4525744 0.041 0.021 CHEMBL3526587 | CHEMBL3526587 | |
| 0.05 | 0.061 | 0.058 | Immunoglobulin Fc receptor antagonist | 0.058 0.029 CHEMBL3527366 | CHEMBL3527366 | |
| 0.043 | 0.055 | 0.062 | Aminopeptidase microsomal inhibitor | 0.062 0.038 CHEMBL3527366 0.05 0.047 CHEMBL4525742 0.05 0.047 CHEMBL4525743 0.06 0.039 CHEMBL3526587 | CHEMBL3527366 | |
| 0.057 | 0.069 | 0.286 | Catalase inhibitor | 0.153 0.025 CHEMBL3527366 0.286 0.006 CHEMBL4525744 0.258 0.008 CHEMBL3526587 | CHEMBL4525744 | |
| 0.014 | 0.027 | 0.02 | Integrin alphaVbeta1 antagonist | 0.02 0.012 CHEMBL3526587 | CHEMBL3526587 | |
| 0.077 | 0.09 | 0.083 | Uric acid excretion stimulant | 0.083 0.078 CHEMBL3526588 0.083 0.077 CHEMBL4525742 | CHEMBL4525742 | |
| 0.008 | 0.023 | 0.011 | 3C-Like protease (MERS coronavirus) inhibitor | 0.011 0.009 CHEMBL4525744 | CHEMBL4525744 | |
| 0.029 | 0.044 | 0.036 | Cholecystokinin B agonist | 0.036 0.028 CHEMBL3526587 | CHEMBL3526587 | |
| 0.056 | 0.071 | 0.064 | Beta 2 adrenoreceptor agonist | 0.064 0.033 CHEMBL3527366 0.064 0.035 CHEMBL4525742 0.059 0.055 CHEMBL3526452 0.061 0.047 CHEMBL3526587 | CHEMBL4525742 | |
| 0.136 | 0.153 | 0.359 | Hypolipemic | 0.282 0.055 CHEMBL3527366 0.174 0.115 CHEMBL4525741 0.217 0.083 CHEMBL3526588 0.159 0.128 CHEMBL3526452 0.222 0.081 CHEMBL4525744 0.359 0.033 CHEMBL3526587 | CHEMBL3526587 | |
| 0.01 | 0.027 | 0.018 | Cholecystokinin A agonist | 0.018 0.009 CHEMBL4525743 | CHEMBL4525743 | |
| 0.027 | 0.045 | 0.042 | Glutamate (mGluR3) agonist | 0.042 0.008 CHEMBL3527366 0.032 0.023 CHEMBL3526587 | CHEMBL3527366 | |
| 0.04 | 0.059 | 0.052 | Bombesin 2 receptor antagonist | 0.052 0.03 CHEMBL4525742 | CHEMBL4525742 | |
| 0.015 | 0.034 | 0.025 | Integrin alphaVbeta3 antagonist | 0.025 0.011 CHEMBL3526587 | CHEMBL3526587 | |
| 0.015 | 0.034 | 0.022 | CC chemokine 1 receptor antagonist | 0.022 0.018 CHEMBL4525741 | CHEMBL4525741 | |
| 0.065 | 0.084 | 0.297 | Chymotrypsin inhibitor | 0.072 0.066 CHEMBL3527366 0.297 0.004 CHEMBL4525743 | CHEMBL4525743 | |
| 0.044 | 0.065 | 0.064 | Cathepsin B inhibitor | 0.064 0.032 CHEMBL4525744 | CHEMBL4525744 | |
| 0.108 | 0.129 | 0.16 | Sphingosine 1-phosphate receptor 2 antagonist | 0.16 0.03 CHEMBL3526587 | CHEMBL3526587 | |
| 0.047 | 0.07 | 0.072 | Matrix metalloproteinase inhibitor | 0.072 0.042 CHEMBL3527366 0.072 0.042 CHEMBL3526587 | CHEMBL3526587 | |
| 0.063 | 0.086 | 0.085 | Adrenaline agonist | 0.085 0.051 CHEMBL4525742 | CHEMBL4525742 | |
| 0.009 | 0.033 | 0.017 | Cholecystokinin agonist | 0.017 0.015 CHEMBL4525743 | CHEMBL4525743 | |
| 0.03 | 0.055 | 0.045 | Aminopeptidase N inhibitor | 0.045 0.037 CHEMBL3527366 0.043 0.039 CHEMBL3526587 | CHEMBL3527366 | |
| 0.092 | 0.117 | 0.135 | Bone formation stimulant | 0.135 0.072 CHEMBL3526587 | CHEMBL3526587 | |
| 0.05 | 0.076 | 0.066 | Caspase 9 inhibitor | 0.064 0.04 CHEMBL4525744 0.066 0.037 CHEMBL3526587 | CHEMBL3526587 | |
| 0.125 | 0.151 | 0.136 | Heat shock protein 70 antagonist | 0.13 0.122 CHEMBL3527366 0.136 0.091 CHEMBL4525742 0.134 0.102 CHEMBL3526587 | CHEMBL4525742 | |
| 0.028 | 0.055 | 0.033 | Calcium-independent phospholipase A2 inhibitor | 0.033 0.026 CHEMBL3526587 | CHEMBL3526587 | |
| 0.029 | 0.057 | 0.065 | GP IIb/IIIa receptor antagonist | 0.065 0.026 CHEMBL3526587 | CHEMBL3526587 | |
| 0.126 | 0.158 | 0.16 | P-glycoprotein inhibitor | 0.16 0.102 CHEMBL3526588 | CHEMBL3526588 | |
| 0.044 | 0.079 | 0.093 | Peroxisome proliferator-activated receptor gamma agonist | 0.059 0.058 CHEMBL3527366 0.093 0.032 CHEMBL3526587 | CHEMBL3526587 | |
| 0.168 | 0.204 | 0.558 | Transcription factor NF kappa B inhibitor | 0.237 0.137 CHEMBL3527366 0.558 0.037 CHEMBL3526588 0.206 0.163 CHEMBL4525742 0.192 0.177 CHEMBL4525744 0.229 0.143 CHEMBL3526587 | CHEMBL3526588 | |
| 0.03 | 0.067 | 0.038 | Plasmepsin II inhibitor | 0.038 0.036 CHEMBL3527366 | CHEMBL3527366 | |
| 0.074 | 0.112 | 0.093 | Xanthine oxidase inhibitor | 0.093 0.067 CHEMBL3526588 | CHEMBL3526588 | |
| 0.027 | 0.066 | 0.093 | Peroxisome proliferator-activated receptor alpha agonist | 0.093 0.014 CHEMBL3526587 | CHEMBL3526587 | |
| 0.076 | 0.117 | 0.229 | Carbonic anhydrase XV inhibitor | 0.229 0.014 CHEMBL3527366 0.094 0.076 CHEMBL3526587 | CHEMBL3527366 | |
| 0.009 | 0.051 | 0.019 | Vitronectin receptor antagonist | 0.019 0.016 CHEMBL3526587 | CHEMBL3526587 | |
| 0.021 | 0.062 | 0.035 | Calpain 1 inhibitor | 0.035 0.019 CHEMBL4525744 | CHEMBL4525744 | |
| 0.043 | 0.084 | 0.059 | Sphingosine 1-phosphate receptor 1 antagonist | 0.059 0.031 CHEMBL3526587 | CHEMBL3526587 | |
| 0.023 | 0.065 | 0.033 | Peroxisome proliferator-activated receptor delta antagonist | 0.033 0.024 CHEMBL3526587 | CHEMBL3526587 | |
| 0.178 | 0.22 | 0.383 | Immunosuppressant | 0.383 0.07 CHEMBL3526588 0.256 0.143 CHEMBL3526452 0.222 0.175 CHEMBL4525744 0.249 0.148 CHEMBL3526587 | CHEMBL3526588 | |
| 0.103 | 0.148 | 0.118 | Farnesoid X receptor antagonist | 0.118 0.108 CHEMBL3526587 | CHEMBL3526587 | |
| 0.059 | 0.104 | 0.103 | NMDA receptor antagonist | 0.08 0.066 CHEMBL3527366 0.103 0.045 CHEMBL4525742 0.081 0.064 CHEMBL3526587 | CHEMBL4525742 | |
| 0.107 | 0.153 | 0.465 | Angiogenesis stimulant | 0.231 0.079 CHEMBL3527366 0.465 0.014 CHEMBL3526588 0.139 0.13 CHEMBL4525742 0.169 0.111 CHEMBL3526452 0.222 0.083 CHEMBL3526587 | CHEMBL3526588 | |
| 0.032 | 0.081 | 0.064 | Prostaglandin EP2 antagonist | 0.064 0.037 CHEMBL3526587 | CHEMBL3526587 | |
| 0.092 | 0.141 | 0.142 | Protein kinase stimulant | 0.12 0.092 CHEMBL3527366 0.142 0.074 CHEMBL3526588 0.123 0.089 CHEMBL4525742 0.111 0.103 CHEMBL3526452 | CHEMBL3526588 | |
| 0.066 | 0.118 | 0.139 | Falcipain 3 inhibitor | 0.139 0.042 CHEMBL4525742 | CHEMBL4525742 | |
| 0.012 | 0.065 | 0.03 | Endothelin receptor antagonist | 0.03 0.018 CHEMBL4525744 | CHEMBL4525744 | |
| 0.034 | 0.086 | 0.123 | Elastase inhibitor | 0.123 0.005 CHEMBL4525743 | CHEMBL4525743 | |
| 0.081 | 0.136 | 0.16 | Factor V inhibitor | 0.096 0.079 CHEMBL4525741 0.16 0.014 CHEMBL4525744 0.102 0.064 CHEMBL3526587 | CHEMBL4525744 | |
| 0.06 | 0.116 | 0.085 | Falcipain inhibitor | 0.085 0.068 CHEMBL4525742 0.079 0.075 CHEMBL4525744 | CHEMBL4525742 | |
| 0.037 | 0.093 | 0.067 | Sphingosine 1-phosphate receptor 3 antagonist | 0.067 0.029 CHEMBL3526587 | CHEMBL3526587 | |
| 0.058 | 0.116 | 0.082 | Falcipain 2 inhibitor | 0.082 0.067 CHEMBL4525742 | CHEMBL4525742 | |
| 0.068 | 0.127 | 0.088 | Potassium channel (Voltage-sensitive) activator | 0.088 0.071 CHEMBL4525741 | CHEMBL4525741 | |
| 0.042 | 0.101 | 0.065 | CDC25B inhibitor | 0.065 0.044 CHEMBL4525744 0.061 0.049 CHEMBL3526587 | CHEMBL4525744 | |
| 0.062 | 0.124 | 0.1 | Aminoacyl-tRNA synthetase inhibitor | 0.1 0.045 CHEMBL3526587 | CHEMBL3526587 | |
| 0.099 | 0.164 | 0.126 | Dual specificity phosphatase 3 inhibitor | 0.126 0.12 CHEMBL3526587 | CHEMBL3526587 | |
| 0.016 | 0.082 | 0.056 | Kainate receptor antagonist | 0.056 0.018 CHEMBL3527366 0.041 0.028 CHEMBL3526587 | CHEMBL3527366 | |
| 0.063 | 0.129 | 0.094 | ATPase (Vacuolar H+) inhibitor | 0.094 0.049 CHEMBL3526588 0.08 0.077 CHEMBL3526452 | CHEMBL3526588 | |
| 0.228 | 0.294 | 0.632 | Antiinflammatory | 0.263 0.252 CHEMBL4525741 0.632 0.045 CHEMBL3526588 0.316 0.2 CHEMBL4525742 0.34 0.18 CHEMBL3526452 | CHEMBL3526588 | |
| 0.078 | 0.144 | 0.104 | Alpha-N-acetylglucosaminidase inhibitor | 0.104 0.096 CHEMBL4525742 | CHEMBL4525742 | |
| 0.049 | 0.116 | 0.075 | Metalloproteinase-2 inhibitor | 0.075 0.058 CHEMBL3526587 | CHEMBL3526587 | |
| 0.085 | 0.153 | 0.129 | Histone deacetylase SIRT1 inhibitor | 0.125 0.085 CHEMBL4525742 0.129 0.081 CHEMBL3526587 | CHEMBL3526587 | |
| 0.005 | 0.076 | 0.019 | Endothelin B receptor antagonist | 0.019 0.013 CHEMBL4525744 | CHEMBL4525744 | |
| 0.103 | 0.175 | 0.145 | Dual specificity phosphatase inhibitor | 0.145 0.1 CHEMBL3526587 | CHEMBL3526587 | |
| 0.042 | 0.115 | 0.065 | Cathepsin G inhibitor | 0.065 0.06 CHEMBL4525743 | CHEMBL4525743 | |
| 0.04 | 0.114 | 0.053 | Kallikrein 1 inhibitor | 0.053 0.047 CHEMBL4525743 | CHEMBL4525743 | |
| 0.04 | 0.116 | 0.129 | Elastase 1 inhibitor | 0.129 0.009 CHEMBL4525743 | CHEMBL4525743 | |
| 0.015 | 0.091 | 0.022 | Vitamin D receptor antagonist | 0.022 0.015 CHEMBL4525741 | CHEMBL4525741 | |
| 0.02 | 0.097 | 0.061 | Ribonucleoside-diphosphate reductase inhibitor | 0.05 0.04 CHEMBL4525742 0.061 0.034 CHEMBL3526587 | CHEMBL3526587 | |
| 0.117 | 0.195 | 0.154 | Phospholipase C inhibitor | 0.154 0.098 CHEMBL4525742 0.145 0.118 CHEMBL3526587 | CHEMBL4525742 | |
| 0.042 | 0.122 | 0.06 | Leukotriene C antagonist | 0.06 0.028 CHEMBL3526587 | CHEMBL3526587 | |
| 0.034 | 0.114 | 0.063 | Lipase inhibitor | 0.063 0.061 CHEMBL3526588 | CHEMBL3526588 | |
| 0.114 | 0.196 | 0.448 | Immunostimulant | 0.219 0.11 CHEMBL3527366 0.448 0.037 CHEMBL3526588 0.16 0.147 CHEMBL4525742 0.207 0.116 CHEMBL3526452 0.165 0.143 CHEMBL4525744 0.279 0.085 CHEMBL3526587 | CHEMBL3526588 | |
| 0.018 | 0.101 | 0.062 | Ribonucleotide reductase inhibitor | 0.049 0.043 CHEMBL4525742 0.062 0.035 CHEMBL3526587 | CHEMBL3526587 | |
| 0.064 | 0.148 | 0.13 | DNA polymerase I inhibitor | 0.13 0.061 CHEMBL3526588 0.11 0.076 CHEMBL3526587 | CHEMBL3526588 | |
| 0.026 | 0.111 | 0.064 | Lysophosphatidic acid 3 receptor antagonist | 0.051 0.034 CHEMBL3527366 0.064 0.018 CHEMBL3526587 | CHEMBL3526587 | |
| 0.045 | 0.132 | 0.078 | Trypsin inhibitor | 0.078 0.028 CHEMBL4525743 | CHEMBL4525743 | |
| 0.029 | 0.117 | 0.049 | Leukotriene B4 antagonist | 0.049 0.046 CHEMBL3526587 | CHEMBL3526587 | |
| 0.164 | 0.254 | 0.279 | Toll-Like receptor 7 agonist | 0.218 0.18 CHEMBL3527366 0.246 0.151 CHEMBL3526452 0.279 0.124 CHEMBL3526587 | CHEMBL3526587 | |
| 0.023 | 0.115 | 0.06 | Plasmin inhibitor | 0.06 0.028 CHEMBL4525743 | CHEMBL4525743 | |
| 0.069 | 0.162 | 0.092 | Glutamate (mGluR7) agonist | 0.092 0.079 CHEMBL3526587 | CHEMBL3526587 | |
| 0.027 | 0.123 | 0.221 | Selectin antagonist | 0.221 0.009 CHEMBL3526588 | CHEMBL3526588 | |
| 0.031 | 0.127 | 0.074 | Leukotriene antagonist | 0.074 0.036 CHEMBL3526587 | CHEMBL3526587 | |
| 0.064 | 0.161 | 0.105 | Mucolytic | 0.105 0.07 CHEMBL3527366 | CHEMBL3527366 | |
| 0.017 | 0.115 | 0.038 | Opioid kappa receptor agonist | 0.038 0.037 CHEMBL3526452 | CHEMBL3526452 | |
| 0.1 | 0.198 | 0.146 | Interferon gamma antagonist | 0.146 0.084 CHEMBL4525741 0.131 0.11 CHEMBL3526588 0.133 0.106 CHEMBL4525742 | CHEMBL4525741 | |
| 0.16 | 0.26 | 0.294 | Toll-Like receptor agonist | 0.221 0.178 CHEMBL3527366 0.242 0.156 CHEMBL3526452 0.294 0.115 CHEMBL3526587 | CHEMBL3526587 | |
| 0.091 | 0.192 | 0.199 | Growth hormone agonist | 0.132 0.104 CHEMBL4525742 0.199 0.059 CHEMBL3526587 | CHEMBL3526587 | |
| 0.026 | 0.127 | 0.037 | Leukotriene C4 antagonist | 0.037 0.034 CHEMBL3526587 | CHEMBL3526587 | |
| 0.106 | 0.207 | 0.259 | Antiamyloidogenic | 0.259 0.067 CHEMBL3526588 0.187 0.109 CHEMBL4525742 0.181 0.114 CHEMBL3526587 | CHEMBL3526588 | |
| 0.087 | 0.189 | 0.118 | Sigma receptor agonist | 0.118 0.117 CHEMBL3526452 | CHEMBL3526452 | |
| 0.033 | 0.136 | 0.051 | Sphingosine 1-phosphate receptor 5 agonist | 0.051 0.044 CHEMBL3526587 | CHEMBL3526587 | |
| 0.039 | 0.145 | 0.064 | Epoxide hydrolase inhibitor | 0.064 0.062 CHEMBL3526587 | CHEMBL3526587 | |
| 0.029 | 0.135 | 0.057 | Nitric oxide donor | 0.057 0.053 CHEMBL3526588 | CHEMBL3526588 | |
| 0.022 | 0.131 | 0.067 | Protein 50S ribosomal subunit inhibitor | 0.067 0.026 CHEMBL3526588 | CHEMBL3526588 | |
| 0.012 | 0.121 | 0.035 | 1,3-Beta-glucan synthase inhibitor | 0.031 0.012 CHEMBL3526452 0.035 0.007 CHEMBL4525743 | CHEMBL4525743 | |
| 0.023 | 0.134 | 0.043 | Microtubule stabilization | 0.043 0.037 CHEMBL3526588 | CHEMBL3526588 | |
| 0.111 | 0.225 | 0.329 | Vasodilator | 0.172 0.13 CHEMBL3527366 0.29 0.052 CHEMBL3526588 0.329 0.039 CHEMBL4525743 0.207 0.099 CHEMBL3526587 | CHEMBL4525743 | |
| 0.133 | 0.249 | 0.29 | Peptidyltransferase inhibitor | 0.163 0.162 CHEMBL3527366 0.29 0.028 CHEMBL3526588 0.176 0.135 CHEMBL3526452 0.174 0.139 CHEMBL3526587 | CHEMBL3526588 | |
| 0.028 | 0.15 | 0.073 | Heparanase inhibitor | 0.064 0.018 CHEMBL3526588 0.057 0.028 CHEMBL4525744 0.073 0.01 CHEMBL3526587 | CHEMBL3526587 | |
| 0.052 | 0.175 | 0.094 | Chelator | 0.092 0.089 CHEMBL4525742 0.094 0.087 CHEMBL3526587 | CHEMBL3526587 | |
| 0.129 | 0.253 | 0.23 | DNA synthesis inhibitor | 0.23 0.083 CHEMBL3526588 0.182 0.15 CHEMBL4525742 | CHEMBL3526588 | |
| 0.086 | 0.212 | 0.339 | Platelet adhesion inhibitor | 0.339 0.022 CHEMBL3526588 | CHEMBL3526588 | |
| 0.103 | 0.232 | 0.177 | ATPase inhibitor | 0.177 0.061 CHEMBL3526588 | CHEMBL3526588 | |
| 0.047 | 0.177 | 0.138 | Expectorant | 0.087 0.086 CHEMBL3527366 0.138 0.04 CHEMBL3526588 | CHEMBL3526588 | |
| 0.055 | 0.186 | 0.115 | Transcription factor NF kappa B stimulant | 0.115 0.028 CHEMBL3526588 | CHEMBL3526588 | |
| 0.045 | 0.179 | 0.079 | Antineoplastic alkaloid | 0.079 0.067 CHEMBL4525741 | CHEMBL4525741 | |
| 0.155 | 0.291 | 0.52 | Antibacterial | 0.321 0.12 CHEMBL3527366 0.52 0.035 CHEMBL3526588 0.297 0.138 CHEMBL4525742 0.259 0.169 CHEMBL3526452 0.289 0.143 CHEMBL4525743 0.345 0.105 CHEMBL4525744 0.22 0.207 CHEMBL3526587 | CHEMBL3526588 | |
| 0.055 | 0.193 | 0.105 | Histone deacetylase class III inhibitor | 0.105 0.084 CHEMBL3526587 | CHEMBL3526587 | |
| 0.018 | 0.158 | 0.099 | Plasminogen activator inhibitor | 0.099 0.016 CHEMBL4525743 | CHEMBL4525743 | |
| 0.042 | 0.193 | 0.095 | Mediator release inhibitor | 0.095 0.076 CHEMBL3526588 | CHEMBL3526588 | |
| 0.097 | 0.249 | 0.16 | Succinate dehydrogenase inhibitor | 0.16 0.096 CHEMBL3527366 0.148 0.116 CHEMBL4525744 0.16 0.095 CHEMBL3526587 | CHEMBL3526587 | |
| 0.057 | 0.211 | 0.134 | Toll-Like receptor 4 antagonist | 0.134 0.032 CHEMBL3526588 | CHEMBL3526588 | |
| 0.099 | 0.255 | 0.374 | Antioxidant | 0.374 0.04 CHEMBL3526588 | CHEMBL3526588 | |
| 0.027 | 0.19 | 0.049 | Parathyroid hormone antagonist | 0.049 0.022 CHEMBL4525741 | CHEMBL4525741 | |
| 0.1 | 0.264 | 0.203 | Cardiotonic | 0.203 0.116 CHEMBL4525743 | CHEMBL4525743 | |
| 0.088 | 0.255 | 0.35 | Free radical scavenger | 0.35 0.039 CHEMBL3526588 0.149 0.146 CHEMBL4525742 | CHEMBL3526588 | |
| 0.052 | 0.222 | 0.184 | Lipid peroxidase inhibitor | 0.184 0.048 CHEMBL3526588 | CHEMBL3526588 | |
| 0.018 | 0.191 | 0.048 | Antibiotic Aminoglycoside-like | 0.048 0.015 CHEMBL3526588 | CHEMBL3526588 | |
| 0.178 | 0.357 | 0.315 | Caspase 9 stimulant | 0.315 0.178 CHEMBL4525741 0.279 0.218 CHEMBL3526588 | CHEMBL4525741 | |
| 0.015 | 0.197 | 0.044 | Carbonic anhydrase XIV inhibitor | 0.044 0.04 CHEMBL3527366 | CHEMBL3527366 | |
| 0.069 | 0.252 | 0.119 | Sphingosine 1-phosphate receptor 4 antagonist | 0.119 0.073 CHEMBL3526587 | CHEMBL3526587 | |
| 0.075 | 0.259 | 0.296 | Hepatoprotectant | 0.296 0.031 CHEMBL3526588 | CHEMBL3526588 | |
| 0.019 | 0.204 | 0.049 | Alpha-mannosidase inhibitor | 0.049 0.045 CHEMBL3526588 | CHEMBL3526588 | |
| 0.056 | 0.254 | 0.139 | Amyloid beta aggregation inhibitor | 0.139 0.117 CHEMBL3526587 | CHEMBL3526587 | |
| 0.026 | 0.226 | 0.065 | NMDA receptor agonist | 0.065 0.041 CHEMBL3526587 | CHEMBL3526587 | |
| 0.051 | 0.255 | 0.106 | Microtubule formation inhibitor | 0.106 0.08 CHEMBL3526588 | CHEMBL3526588 | |
| 0.077 | 0.282 | 0.21 | Platelet aggregation inhibitor | 0.21 0.074 CHEMBL3526587 | CHEMBL3526587 | |
| 0.029 | 0.236 | 0.071 | GABA aminotransferase inhibitor | 0.071 0.059 CHEMBL3527366 0.07 0.062 CHEMBL3526587 | CHEMBL3527366 | |
| 0.13 | 0.338 | 0.249 | Caspase 3 stimulant | 0.249 0.113 CHEMBL3526588 | CHEMBL3526588 | |
| 0.015 | 0.223 | 0.08 | Antineoplastic antibiotic | 0.08 0.057 CHEMBL3526588 | CHEMBL3526588 | |
| 0.022 | 0.232 | 0.047 | Glucose-6-phosphate translocase inhibitor | 0.047 0.046 CHEMBL3526588 | CHEMBL3526588 | |
| 0.081 | 0.293 | 0.134 | Papain-like protease (SARS coronavirus) inhibitor | 0.134 0.054 CHEMBL4525741 0.113 0.103 CHEMBL4525742 | CHEMBL4525741 | |
| 0.069 | 0.283 | 0.25 | Nitric oxide antagonist | 0.25 0.052 CHEMBL3526588 | CHEMBL3526588 | |
| 0.115 | 0.336 | 0.17 | MAP kinase kinase 5 inhibitor | 0.17 0.085 CHEMBL4525741 | CHEMBL4525741 | |
| 0.058 | 0.281 | 0.116 | Folate antagonist | 0.116 0.042 CHEMBL3526587 | CHEMBL3526587 | |
| 0.134 | 0.361 | 0.234 | 5 Hydroxytryptamine uptake stimulant | 0.234 0.098 CHEMBL4525742 0.194 0.164 CHEMBL3526587 | CHEMBL4525742 | |
| 0.033 | 0.275 | 0.088 | Kallikrein 7 inhibitor | 0.088 0.008 CHEMBL4525743 | CHEMBL4525743 | |
| 0.052 | 0.335 | 0.146 | Interleukin antagonist | 0.146 0.12 CHEMBL3526587 | CHEMBL3526587 | |
| 0.126 | 0.409 | 0.422 | Apoptosis agonist | 0.422 0.103 CHEMBL3526588 | CHEMBL3526588 | |
| 0.039 | 0.38 | 0.116 | Cell wall synthesis inhibitor | 0.116 0.106 CHEMBL3526588 | CHEMBL3526588 | |
| 0.027 | 0.374 | 0.112 | AMP-activated protein kinase stimulant | 0.112 0.057 CHEMBL3526588 | CHEMBL3526588 | |
| 0.016 | 0.372 | 0.079 | Rho-associated kinase II inhibitor | 0.079 0.046 CHEMBL3527366 | CHEMBL3527366 | |
| 0.079 | 0.441 | 0.267 | Immunomodulator | 0.267 0.102 CHEMBL3526588 | CHEMBL3526588 | |
| 0.049 | 0.451 | 0.121 | NOS3 expression enhancer | 0.121 0.114 CHEMBL3526588 | CHEMBL3526588 | |
| 0.041 | 0.468 | 0.305 | Alpha-glucosidase inhibitor | 0.305 0.157 CHEMBL3526588 | CHEMBL3526588 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |