| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.782 | 0.001 | 0.782 | Orexin receptor antagonist | 0.394 0.002 CHEMBL3527303 0.084 0.023 CHEMBL3526735 0.298 0.002 CHEMBL3542347 0.211 0.003 CHEMBL3542348 0.329 0.002 CHEMBL3526736 0.181 0.004 CHEMBL3527503 0.157 0.004 CHEMBL3527393 0.247 0.003 CHEMBL3526808 | ||
| 0.679 | 0.013 | 0.783 | Antiobesity | 0.783 0.006 CHEMBL3527303 0.343 0.09 CHEMBL3526735 0.578 0.023 CHEMBL3542347 0.518 0.034 CHEMBL3542348 0.536 0.03 CHEMBL3526736 0.708 0.01 CHEMBL3527503 0.44 0.052 CHEMBL3527393 0.648 0.015 CHEMBL3526808 | CHEMBL3527303 | |
| 0.61 | 0.001 | 0.61 | Orexin receptor 1 antagonist | 0.315 0.002 CHEMBL3527303 0.224 0.003 CHEMBL3542347 0.171 0.004 CHEMBL3542348 0.241 0.003 CHEMBL3526736 0.141 0.005 CHEMBL3527503 0.154 0.004 CHEMBL3527393 0.22 0.003 CHEMBL3526808 | ||
| 0.401 | 0.001 | 0.401 | Orexin receptor 2 antagonist | 0.234 0.002 CHEMBL3527303 0.143 0.003 CHEMBL3542347 0.093 0.005 CHEMBL3542348 0.143 0.003 CHEMBL3526736 0.07 0.008 CHEMBL3527503 0.085 0.005 CHEMBL3527393 0.162 0.003 CHEMBL3526808 | ||
| 0.292 | 0.049 | 0.292 | Potassium channel blocker | |||
| 0.141 | 0.012 | 0.165 | Alpha 2d adrenoreceptor antagonist | 0.165 0.005 CHEMBL3527303 0.111 0.032 CHEMBL3526735 0.138 0.013 CHEMBL3542347 0.134 0.015 CHEMBL3542348 0.136 0.014 CHEMBL3526736 0.132 0.016 CHEMBL3527503 0.136 0.014 CHEMBL3527393 0.148 0.01 CHEMBL3526808 | CHEMBL3527303 | |
| 0.145 | 0.029 | 0.145 | CC chemokine 6 receptor antagonist | 0.128 0.077 CHEMBL3527303 0.134 0.056 CHEMBL3526735 0.122 0.109 CHEMBL3542348 0.122 0.106 CHEMBL3526736 0.122 0.108 CHEMBL3527503 0.131 0.069 CHEMBL3526808 | ||
| 0.096 | 0.012 | 0.096 | Enoyl-[acyl-carrier-protein] reductase inhibitor | |||
| 0.086 | 0.007 | 0.086 | Potassium channel subfamily K member 3 blocker | 0.082 0.008 CHEMBL3527303 0.046 0.013 CHEMBL3542347 0.057 0.01 CHEMBL3542348 0.053 0.011 CHEMBL3526736 0.057 0.01 CHEMBL3527503 0.03 0.021 CHEMBL3526808 | ||
| 0.128 | 0.054 | 0.128 | Calcium channel N-type blocker | 0.114 0.072 CHEMBL3527303 | ||
| 0.088 | 0.019 | 0.088 | Potassium channel (Tandem pore domain) blocker | 0.081 0.032 CHEMBL3527303 | ||
| 0.128 | 0.063 | 0.154 | Papain-like protease (SARS coronavirus) inhibitor | 0.154 0.031 CHEMBL3542348 0.122 0.076 CHEMBL3526736 0.151 0.033 CHEMBL3527503 | CHEMBL3542348 | |
| 0.222 | 0.162 | 0.382 | Vasodilator, coronary | 0.382 0.041 CHEMBL3526735 | CHEMBL3526735 | |
| 0.086 | 0.037 | 0.103 | Lipase inhibitor | 0.103 0.025 CHEMBL3526735 0.073 0.051 CHEMBL3542348 | CHEMBL3526735 | |
| 0.22 | 0.173 | 0.22 | Beta lactamase inhibitor | 0.193 0.19 CHEMBL3526736 | ||
| 0.147 | 0.105 | 0.147 | Amyloid beta precursor protein antagonist | |||
| 0.051 | 0.011 | 0.051 | Glucose-6-phosphate dehydrogenase inhibitor | 0.043 0.017 CHEMBL3527303 0.05 0.011 CHEMBL3542347 0.05 0.012 CHEMBL3542348 0.051 0.011 CHEMBL3526736 0.051 0.011 CHEMBL3527503 | ||
| 0.206 | 0.167 | 0.206 | Thioredoxin glutathione reductase inhibitor | |||
| 0.059 | 0.02 | 0.063 | Neurokinin 3 antagonist | 0.063 0.017 CHEMBL3527303 0.039 0.037 CHEMBL3542347 0.044 0.032 CHEMBL3526736 0.046 0.03 CHEMBL3526808 | CHEMBL3527303 | |
| 0.076 | 0.042 | 0.142 | Glutamate (mGluR group I) antagonist | 0.142 0.015 CHEMBL3527303 0.083 0.035 CHEMBL3526808 | CHEMBL3527303 | |
| 0.057 | 0.024 | 0.104 | Glutamate (mGluR5) antagonist | 0.104 0.009 CHEMBL3527303 0.047 0.033 CHEMBL3527393 0.063 0.02 CHEMBL3526808 | CHEMBL3527303 | |
| 0.205 | 0.182 | 0.215 | Ca(v)3.3 blocker | 0.215 0.16 CHEMBL3527303 | CHEMBL3527303 | |
| 0.037 | 0.018 | 0.048 | Tubulin agonist | 0.048 0.009 CHEMBL3527303 0.033 0.026 CHEMBL3526735 0.039 0.016 CHEMBL3542347 0.039 0.017 CHEMBL3542348 0.04 0.015 CHEMBL3526736 0.04 0.015 CHEMBL3527503 0.041 0.014 CHEMBL3527393 0.043 0.012 CHEMBL3526808 | CHEMBL3527303 | |
| 0.061 | 0.044 | 0.178 | Glutamate (mGluR) agonist | 0.178 0.011 CHEMBL3527303 0.064 0.042 CHEMBL3527503 0.058 0.047 CHEMBL3527393 0.129 0.017 CHEMBL3526808 | CHEMBL3527303 | |
| 0.048 | 0.033 | 0.126 | Glutamate (mGluR group I) agonist | 0.126 0.005 CHEMBL3527303 0.048 0.032 CHEMBL3526808 | CHEMBL3527303 | |
| 0.06 | 0.045 | 0.06 | Dopamine D3 antagonist | |||
| 0.222 | 0.208 | 0.222 | Transcription factor inhibitor | |||
| 0.079 | 0.067 | 0.079 | Acetylcholine agonist | |||
| 0.068 | 0.056 | 0.068 | Dopamine antagonist | |||
| 0.052 | 0.04 | 0.052 | Nicotinic alpha7 receptor agonist | |||
| 0.08 | 0.069 | 0.105 | 3C-Like protease (SARS coronavirus) inhibitor | 0.105 0.029 CHEMBL3542348 | CHEMBL3542348 | |
| 0.204 | 0.196 | 0.446 | Toll-Like receptor 7 agonist | 0.295 0.113 CHEMBL3527303 0.321 0.098 CHEMBL3526735 0.251 0.147 CHEMBL3542347 0.261 0.138 CHEMBL3542348 0.446 0.044 CHEMBL3527503 0.307 0.105 CHEMBL3526808 | CHEMBL3527503 | |
| 0.043 | 0.041 | 0.043 | Purinergic P2X antagonist | 0.043 0.041 CHEMBL3526808 | ||
| 0.013 | 0.014 | 0.034 | Dipeptidyl peptidase IX inhibitor | 0.034 0.005 CHEMBL3527303 | CHEMBL3527303 | |
| 0.039 | 0.045 | 0.055 | CDK7/cyclin H inhibitor | 0.055 0.019 CHEMBL3527303 | CHEMBL3527303 | |
| 0.213 | 0.221 | 0.426 | Analgesic | 0.308 0.135 CHEMBL3527303 0.221 0.212 CHEMBL3542348 0.252 0.181 CHEMBL3527503 0.286 0.152 CHEMBL3527393 0.426 0.074 CHEMBL3526808 | CHEMBL3526808 | |
| 0.011 | 0.022 | 0.025 | Dipeptidyl peptidase VIII inhibitor | 0.025 0.005 CHEMBL3527303 | CHEMBL3527303 | |
| 0.196 | 0.207 | 0.44 | Toll-Like receptor agonist | 0.293 0.115 CHEMBL3527303 0.328 0.094 CHEMBL3526735 0.244 0.154 CHEMBL3542347 0.252 0.146 CHEMBL3542348 0.44 0.046 CHEMBL3527503 0.306 0.107 CHEMBL3526808 | CHEMBL3527503 | |
| 0.061 | 0.075 | 0.134 | Glutamate (mGluR) antagonist | 0.134 0.021 CHEMBL3527303 0.095 0.038 CHEMBL3526808 | CHEMBL3527303 | |
| 0.044 | 0.061 | 0.181 | Dipeptidyl peptidase inhibitor | 0.181 0.004 CHEMBL3527303 | CHEMBL3527303 | |
| 0.068 | 0.093 | 0.092 | Phosphodiesterase 11A inhibitor | 0.092 0.04 CHEMBL3527303 | CHEMBL3527303 | |
| 0.068 | 0.093 | 0.092 | Phosphodiesterase XI inhibitor | 0.092 0.04 CHEMBL3527303 | CHEMBL3527303 | |
| 0.106 | 0.147 | 0.12 | NOS3 expression enhancer | 0.12 0.116 CHEMBL3526808 | CHEMBL3526808 | |
| 0.023 | 0.073 | 0.039 | Opioid kappa receptor agonist | 0.039 0.035 CHEMBL3526808 | CHEMBL3526808 | |
| 0.171 | 0.223 | 0.189 | Caspase 3 stimulant | 0.189 0.186 CHEMBL3526735 | CHEMBL3526735 | |
| 0.033 | 0.09 | 0.151 | Dipeptidyl peptidase IV inhibitor | 0.151 0.004 CHEMBL3527303 | CHEMBL3527303 | |
| 0.007 | 0.065 | 0.012 | Integrin alphaLbeta2 antagonist | 0.012 0.011 CHEMBL3526735 | CHEMBL3526735 | |
| 0.02 | 0.085 | 0.034 | RNA-directed RNA polymerase inhibitor | 0.034 0.024 CHEMBL3526735 | CHEMBL3526735 | |
| 0.07 | 0.157 | 0.108 | Glutamate (mGluR7) agonist | 0.108 0.045 CHEMBL3527303 | CHEMBL3527303 | |
| 0.099 | 0.186 | 0.157 | Dual specificity phosphatase inhibitor | 0.157 0.087 CHEMBL3526735 | CHEMBL3526735 | |
| 0.023 | 0.111 | 0.08 | Glutamate (mGluR5) agonist | 0.08 0.01 CHEMBL3527303 0.046 0.032 CHEMBL3526808 | CHEMBL3527303 | |
| 0.02 | 0.113 | 0.039 | Vanilloid 4 antagonist | 0.039 0.012 CHEMBL3527303 | CHEMBL3527303 | |
| 0.074 | 0.202 | 0.215 | Protein-tyrosine phosphatase inhibitor | 0.215 0.041 CHEMBL3526735 0.125 0.108 CHEMBL3527503 | CHEMBL3526735 | |
| 0.071 | 0.199 | 0.154 | Histone deacetylase SIRT1 inhibitor | 0.154 0.059 CHEMBL3526735 | CHEMBL3526735 | |
| 0.046 | 0.175 | 0.061 | Prolactin release inhibitor | 0.061 0.049 CHEMBL3527303 | CHEMBL3527303 | |
| 0.039 | 0.179 | 0.074 | Bcl-xL inhibitor | 0.074 0.016 CHEMBL3527303 | CHEMBL3527303 | |
| 0.034 | 0.176 | 0.076 | Analgesic, opioid | 0.076 0.053 CHEMBL3527393 | CHEMBL3527393 | |
| 0.077 | 0.234 | 0.106 | Sphingosine 1-phosphate receptor 2 agonist | 0.106 0.085 CHEMBL3526808 | CHEMBL3526808 | |
| 0.028 | 0.185 | 0.095 | CDC25B inhibitor | 0.095 0.018 CHEMBL3526735 | CHEMBL3526735 | |
| 0.013 | 0.184 | 0.039 | Dipeptidyl peptidase II inhibitor | 0.039 0.015 CHEMBL3527303 | CHEMBL3527303 | |
| 0.076 | 0.251 | 0.187 | Platelet adhesion inhibitor | 0.187 0.078 CHEMBL3526735 | CHEMBL3526735 | |
| 0.035 | 0.222 | 0.061 | Caspase 9 inhibitor | 0.061 0.046 CHEMBL3526735 | CHEMBL3526735 | |
| 0.006 | 0.198 | 0.026 | Integrin alphaVbeta3 antagonist | 0.026 0.01 CHEMBL3526735 | CHEMBL3526735 | |
| 0.04 | 0.233 | 0.183 | Glutamate receptor antagonist | 0.183 0.031 CHEMBL3527303 0.125 0.069 CHEMBL3526808 | CHEMBL3527303 | |
| 0.059 | 0.254 | 0.12 | Anticoagulant | 0.12 0.112 CHEMBL3527303 | CHEMBL3527303 | |
| 0.005 | 0.227 | 0.021 | Histone deacetylase 3 inhibitor | 0.021 0.019 CHEMBL3526735 | CHEMBL3526735 | |
| 0.1 | 0.324 | 0.183 | Transcription factor STAT3 inhibitor | 0.183 0.159 CHEMBL3526735 | CHEMBL3526735 | |
| 0.051 | 0.276 | 0.08 | Hematopoietic | 0.08 0.074 CHEMBL3526735 | CHEMBL3526735 | |
| 0.025 | 0.25 | 0.066 | CDC25A inhibitor | 0.066 0.064 CHEMBL3526735 | CHEMBL3526735 | |
| 0.025 | 0.262 | 0.131 | Protein-tyrosine phosphatase 1B inhibitor | 0.131 0.055 CHEMBL3526735 | CHEMBL3526735 | |
| 0.061 | 0.31 | 0.126 | Factor V inhibitor | 0.102 0.065 CHEMBL3526735 0.126 0.033 CHEMBL3542348 | CHEMBL3542348 | |
| 0.021 | 0.271 | 0.055 | Integrin alpha1beta1 antagonist | 0.055 0.005 CHEMBL3526735 | CHEMBL3526735 | |
| 0.027 | 0.277 | 0.059 | Bcl2 antagonist | 0.059 0.057 CHEMBL3527303 | CHEMBL3527303 | |
| 0.136 | 0.389 | 0.391 | Cyclophilin D inhibitor | 0.281 0.18 CHEMBL3526735 0.391 0.096 CHEMBL3527503 | CHEMBL3527503 | |
| 0.025 | 0.295 | 0.111 | HIV-1 integrase inhibitor | 0.111 0.019 CHEMBL3527393 | CHEMBL3527393 | |
| 0.012 | 0.301 | 0.13 | Glutamate receptor agonist | 0.13 0.023 CHEMBL3527303 0.088 0.046 CHEMBL3526808 | CHEMBL3527303 | |
| 0.005 | 0.301 | 0.046 | Integrin antagonist | 0.046 0.029 CHEMBL3526735 | CHEMBL3526735 | |
| 0.022 | 0.356 | 0.084 | Protease inhibitor | 0.084 0.081 CHEMBL3526735 | CHEMBL3526735 | |
| 0.024 | 0.365 | 0.055 | DNA helicase inhibitor | 0.055 0.037 CHEMBL3527503 | CHEMBL3527503 | |
| 0.029 | 0.379 | 0.133 | Thrombolytic | 0.133 0.096 CHEMBL3526735 | CHEMBL3526735 | |
| 0.102 | 0.469 | 0.294 | Interleukin 2 agonist | 0.201 0.188 CHEMBL3527303 0.231 0.141 CHEMBL3526735 0.294 0.078 CHEMBL3527503 | CHEMBL3527503 | |
| 0.013 | 0.388 | 0.051 | Sphingosine 1-phosphate receptor 5 agonist | 0.051 0.044 CHEMBL3526735 | CHEMBL3526735 | |
| 0.004 | 0.428 | 0.023 | Prostaglandin D2 antagonist | 0.023 0.015 CHEMBL3527503 | CHEMBL3527503 | |
| 0.011 | 0.468 | 0.102 | Protein kinase B alpha inhibitor | 0.102 0.029 CHEMBL3542347 | CHEMBL3542347 | |
| 0.005 | 0.476 | 0.142 | Antineoplastic antibiotic | 0.142 0.033 CHEMBL3542347 | CHEMBL3542347 | |
| 0.005 | 0.477 | 0.058 | Prostaglandin antagonist | 0.058 0.033 CHEMBL3527503 | CHEMBL3527503 | |
| 0.073 | 0.554 | 0.423 | Apoptosis agonist | 0.423 0.103 CHEMBL3542347 | CHEMBL3542347 | |
| 0.027 | 0.515 | 0.133 | Cell adhesion inhibitor | 0.133 0.057 CHEMBL3526735 | CHEMBL3526735 | |
| 0.015 | 0.515 | 0.085 | Cell adhesion molecule inhibitor | 0.085 0.047 CHEMBL3526735 | CHEMBL3526735 | |
| 0.059 | 0.596 | 0.169 | Catenin beta inhibitor | 0.169 0.068 CHEMBL3526735 | CHEMBL3526735 | |
| 0.024 | 0.609 | 0.104 | Photosensitizer | 0.104 0.081 CHEMBL3526735 | CHEMBL3526735 | |
| 0.023 | 0.611 | 0.143 | Thiol protease inhibitor | 0.143 0.076 CHEMBL3526735 | CHEMBL3526735 | |
| 0.059 | 0.651 | 0.259 | Antiinflammatory | 0.259 0.256 CHEMBL3542348 | CHEMBL3542348 | |
| 0.012 | 0.618 | 0.121 | Interleukin 1 beta converting enzyme inhibitor | 0.121 0.034 CHEMBL3526735 | CHEMBL3526735 | |
| 0.035 | 0.664 | 0.127 | Folate antagonist | 0.127 0.033 CHEMBL3526735 | CHEMBL3526735 | |
| 0.008 | 0.643 | 0.051 | Protein 50S ribosomal subunit inhibitor | 0.051 0.039 CHEMBL3542348 | CHEMBL3542348 | |
| 0.005 | 0.659 | 0.075 | Sphingosine 1-phosphate receptor 4 agonist | 0.075 0.04 CHEMBL3526735 | CHEMBL3526735 | |
| 0.025 | 0.689 | 0.2 | Immunosuppressant | 0.2 0.197 CHEMBL3542347 | CHEMBL3542347 | |
| 0.003 | 0.689 | 0.028 | 1,3-Beta-glucan synthase inhibitor | 0.028 0.019 CHEMBL3527393 | CHEMBL3527393 | |
| 0.012 | 0.702 | 0.128 | Bone formation stimulant | 0.128 0.078 CHEMBL3526735 | CHEMBL3526735 | |
| 0.008 | 0.745 | 0.235 | Platelet antagonist | 0.235 0.079 CHEMBL3526735 | CHEMBL3526735 | |
| 0.004 | 0.745 | 0.061 | HIV-1 integrase (3'-Processing) inhibitor | 0.061 0.046 CHEMBL3527393 | CHEMBL3527393 | |
| 0.004 | 0.762 | 0.07 | HIV-1 integrase (Strand Transfer) inhibitor | 0.07 0.036 CHEMBL3527393 | CHEMBL3527393 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |