| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.89 | 0.001 | 0.89 | Angiotensin-converting enzyme inhibitor | 0.765 0.001 CHEMBL2158192 | ||
| 0.803 | 0.001 | 0.803 | Neutral endopeptidase inhibitor | 0.706 0.001 CHEMBL2158192 | ||
| 0.725 | 0.003 | 0.725 | Chelator | 0.676 0.003 CHEMBL2158192 | ||
| 0.706 | 0.002 | 0.706 | Expectorant | 0.545 0.003 CHEMBL2158192 | ||
| 0.702 | 0.001 | 0.702 | Mucolytic | 0.521 0.002 CHEMBL2158192 | ||
| 0.659 | 0.001 | 0.659 | Angiotensin-converting enzyme 2 inhibitor | 0.469 0.001 CHEMBL2158192 | ||
| 0.63 | 0.004 | 0.63 | Hepatoprotectant | 0.4 0.013 CHEMBL2158192 | ||
| 0.586 | 0.005 | 0.586 | Peroxidase inhibitor | 0.565 0.005 CHEMBL2158192 | ||
| 0.566 | 0.002 | 0.828 | Glutamate decarboxylase inhibitor | 0.828 0.002 CHEMBL2158192 | CHEMBL2158192 | |
| 0.56 | 0.009 | 0.56 | Tumour necrosis factor alpha release inhibitor | |||
| 0.549 | 0.003 | 0.549 | Aminopeptidase B inhibitor | 0.435 0.004 CHEMBL2158192 | ||
| 0.48 | 0.006 | 0.625 | Alpha-N-acetylglucosaminidase inhibitor | 0.625 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.471 | 0.005 | 0.471 | Sodium/bile acid cotransporter inhibitor | 0.303 0.076 CHEMBL2158192 | ||
| 0.46 | 0.017 | 0.526 | Superoxide dismutase inhibitor | 0.526 0.011 CHEMBL2158192 | CHEMBL2158192 | |
| 0.405 | 0.003 | 0.417 | Endothelin-converting enzyme inhibitor | 0.417 0.002 CHEMBL2158192 | CHEMBL2158192 | |
| 0.402 | 0.011 | 0.473 | Thrombolytic | 0.473 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.391 | 0.004 | 0.575 | Porphobilinogen synthase inhibitor | 0.575 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.394 | 0.011 | 0.394 | Phospholipase C inhibitor | 0.349 0.014 CHEMBL2158192 | ||
| 0.373 | 0.027 | 0.38 | Angiogenesis stimulant | 0.38 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.372 | 0.028 | 0.372 | Insulysin inhibitor | 0.344 0.036 CHEMBL2158192 | ||
| 0.375 | 0.034 | 0.375 | Cardiotonic | 0.244 0.087 CHEMBL2158192 | ||
| 0.339 | 0.002 | 0.339 | Aminopeptidase I inhibitor | 0.295 0.003 CHEMBL2158192 | ||
| 0.383 | 0.055 | 0.383 | Immunostimulant | 0.32 0.073 CHEMBL2158192 | ||
| 0.368 | 0.042 | 0.368 | Antioxidant | 0.263 0.077 CHEMBL2158192 | ||
| 0.331 | 0.005 | 0.371 | Catalase inhibitor | 0.371 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.331 | 0.005 | 0.331 | Histidine decarboxylase inhibitor | 0.313 0.006 CHEMBL2158192 | ||
| 0.33 | 0.005 | 0.404 | Alcohol dehydrogenase inhibitor | 0.404 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.372 | 0.056 | 0.513 | Cholesterol antagonist | 0.513 0.031 CHEMBL2158192 | CHEMBL2158192 | |
| 0.315 | 0.02 | 0.315 | Peptidyltransferase inhibitor | |||
| 0.3 | 0.011 | 0.47 | Succinate dehydrogenase inhibitor | 0.47 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.308 | 0.021 | 0.308 | Diuretic | 0.277 0.026 CHEMBL2158192 | ||
| 0.342 | 0.057 | 0.687 | Aldehyde oxidase inhibitor | 0.687 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.282 | 0.008 | 0.326 | Adenylate kinase inhibitor | 0.326 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.304 | 0.031 | 0.334 | Tyrosine 3 hydroxylase inhibitor | 0.334 0.02 CHEMBL2158192 | CHEMBL2158192 | |
| 0.297 | 0.029 | 0.648 | Dual specificity phosphatase 3 inhibitor | 0.648 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.27 | 0.004 | 0.363 | Phenylalanine 4-hydroxylase inhibitor | 0.363 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.291 | 0.03 | 0.317 | DNA methyltransferase I inhibitor | 0.317 0.021 CHEMBL2158192 | CHEMBL2158192 | |
| 0.325 | 0.074 | 0.367 | Antithrombotic | 0.367 0.059 CHEMBL2158192 | CHEMBL2158192 | |
| 0.266 | 0.017 | 0.363 | M17 leucyl aminopeptidase inhibitor | 0.363 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.254 | 0.013 | 0.4 | GABA C receptor agonist | 0.4 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.241 | 0.008 | 0.324 | Glutamate dehydrogenase inhibitor | 0.324 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.329 | 0.097 | 0.329 | Calpain 2 inhibitor | 0.27 0.135 CHEMBL2158192 | ||
| 0.266 | 0.04 | 0.296 | DNA methylase inhibitor | 0.296 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.229 | 0.007 | 0.229 | Matrix metalloproteinase inhibitor | 0.13 0.017 CHEMBL2158192 | ||
| 0.229 | 0.017 | 0.356 | Ferrochelatase inhibitor | 0.356 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.271 | 0.06 | 0.351 | Free radical scavenger | 0.351 0.039 CHEMBL2158192 | CHEMBL2158192 | |
| 0.263 | 0.057 | 0.28 | Interleukin antagonist | 0.28 0.052 CHEMBL2158192 | CHEMBL2158192 | |
| 0.293 | 0.093 | 0.334 | Vasodilator, coronary | 0.334 0.064 CHEMBL2158192 | CHEMBL2158192 | |
| 0.207 | 0.01 | 0.249 | HIV-1 integrase (Overall Integration) inhibitor | 0.249 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.199 | 0.007 | 0.199 | Ornithine carbamoyltransferase inhibitor | 0.194 0.007 CHEMBL2158192 | ||
| 0.31 | 0.118 | 0.338 | Histamine release inhibitor | 0.338 0.105 CHEMBL2158192 | CHEMBL2158192 | |
| 0.233 | 0.042 | 0.601 | Dual specificity phosphatase inhibitor | 0.601 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.252 | 0.063 | 0.252 | Calpain inhibitor | 0.23 0.084 CHEMBL2158192 | ||
| 0.186 | 0.003 | 0.186 | Protocollagen prolyl hydroxylase inhibitor | |||
| 0.182 | 0.004 | 0.182 | Collagenase inhibitor | 0.135 0.004 CHEMBL2158192 | ||
| 0.18 | 0.005 | 0.181 | NMDA receptor agonist | 0.181 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.18 | 0.007 | 0.18 | Glutathione S-transferase inhibitor | 0.129 0.018 CHEMBL2158192 | ||
| 0.247 | 0.083 | 0.247 | Gastrin inhibitor | 0.218 0.122 CHEMBL2158192 | ||
| 0.157 | 0.003 | 0.169 | Lysine carboxypeptidase inhibitor | 0.169 0.002 CHEMBL2158192 | CHEMBL2158192 | |
| 0.159 | 0.006 | 0.159 | Aminopeptidase microsomal inhibitor | 0.142 0.009 CHEMBL2158192 | ||
| 0.163 | 0.013 | 0.163 | Metalloproteinase-9 inhibitor | 0.152 0.015 CHEMBL2158192 | ||
| 0.161 | 0.011 | 0.161 | Neutrophil collagenase inhibitor | 0.093 0.025 CHEMBL2158192 | ||
| 0.154 | 0.018 | 0.154 | Metalloproteinase-2 inhibitor | 0.128 0.026 CHEMBL2158192 | ||
| 0.14 | 0.006 | 0.14 | Aminopeptidase N inhibitor | 0.123 0.009 CHEMBL2158192 | ||
| 0.224 | 0.09 | 0.254 | DNA synthesis inhibitor | 0.254 0.064 CHEMBL2158192 | CHEMBL2158192 | |
| 0.13 | 0.005 | 0.13 | Botulinum neurotoxin type A inhibitor | 0.091 0.012 CHEMBL2158192 | ||
| 0.177 | 0.056 | 0.188 | Phospholipase A2 inhibitor | 0.188 0.049 CHEMBL2158192 | CHEMBL2158192 | |
| 0.162 | 0.041 | 0.188 | Aldehyde dehydrogenase inhibitor | 0.188 0.031 CHEMBL2158192 | CHEMBL2158192 | |
| 0.125 | 0.004 | 0.187 | Vanilloid 2 antagonist | 0.187 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.131 | 0.011 | 0.143 | Acyl-CoA dehydrogenase inhibitor | 0.143 0.01 CHEMBL2158192 | CHEMBL2158192 | |
| 0.184 | 0.066 | 0.184 | Growth hormone agonist | 0.14 0.095 CHEMBL2158192 | ||
| 0.173 | 0.058 | 0.185 | Neurotensin receptor agonist | 0.185 0.045 CHEMBL2158192 | CHEMBL2158192 | |
| 0.121 | 0.007 | 0.263 | Macrophage elastase inhibitor | 0.263 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.133 | 0.02 | 0.181 | Lanosterol 14 alpha demethylase inhibitor | 0.181 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.131 | 0.022 | 0.251 | Phosphofructokinase-1 inhibitor | 0.251 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.116 | 0.01 | 0.116 | Matrix metalloproteinase 1 inhibitor | 0.093 0.015 CHEMBL2158192 | ||
| 0.107 | 0.003 | 0.107 | Membrane dipeptidase inhibitor | 0.09 0.004 CHEMBL2158192 | ||
| 0.115 | 0.012 | 0.115 | Matrix metalloproteinase (membrane-type) inhibitor | 0.097 0.015 CHEMBL2158192 | ||
| 0.253 | 0.151 | 0.373 | GABA C receptor rho-3 antagonist | 0.373 0.074 CHEMBL2158192 | CHEMBL2158192 | |
| 0.129 | 0.031 | 0.148 | Anabolic | 0.148 0.019 CHEMBL2158192 | CHEMBL2158192 | |
| 0.107 | 0.011 | 0.107 | Phospholipase D inhibitor | 0.093 0.019 CHEMBL2158192 | ||
| 0.099 | 0.003 | 0.269 | AMPA receptor agonist | 0.269 0.002 CHEMBL2158192 | CHEMBL2158192 | |
| 0.155 | 0.061 | 0.194 | Cell wall synthesis inhibitor | 0.194 0.033 CHEMBL2158192 | CHEMBL2158192 | |
| 0.115 | 0.031 | 0.167 | NADH dehydrogenase inhibitor | 0.167 0.014 CHEMBL2158192 | CHEMBL2158192 | |
| 0.157 | 0.074 | 0.157 | Anticoagulant | |||
| 0.088 | 0.007 | 0.11 | Leukotriene A4 hydrolase inhibitor | 0.11 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.115 | 0.035 | 0.233 | Triose-phosphate isomerase inhibitor | 0.233 0.008 CHEMBL2158192 | CHEMBL2158192 | |
| 0.088 | 0.009 | 0.099 | Alpha-mannosidase inhibitor | 0.099 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.135 | 0.056 | 0.135 | Adenylate cyclase inhibitor | 0.135 0.056 CHEMBL2158192 | ||
| 0.088 | 0.009 | 0.088 | Farnesyltransferase inhibitor | 0.086 0.01 CHEMBL2158192 | ||
| 0.121 | 0.043 | 0.149 | Carbonic anhydrase III inhibitor | 0.149 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.146 | 0.069 | 0.167 | Adenylate cyclase stimulant | 0.167 0.039 CHEMBL2158192 | CHEMBL2158192 | |
| 0.096 | 0.02 | 0.096 | Ribonucleoside-diphosphate reductase inhibitor | 0.067 0.031 CHEMBL2158192 | ||
| 0.096 | 0.022 | 0.096 | Ribonucleotide reductase inhibitor | 0.068 0.032 CHEMBL2158192 | ||
| 0.08 | 0.009 | 0.094 | Mannosidase inhibitor | 0.094 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.223 | 0.152 | 0.225 | Interleukin 2 agonist | 0.225 0.149 CHEMBL2158192 | CHEMBL2158192 | |
| 0.084 | 0.016 | 0.084 | Toll-Like receptor 2 agonist | 0.052 0.023 CHEMBL2158192 | ||
| 0.119 | 0.053 | 0.176 | GABA C receptor antagonist | 0.176 0.019 CHEMBL2158192 | CHEMBL2158192 | |
| 0.067 | 0.003 | 0.067 | Aminopeptidase A inhibitor | 0.043 0.004 CHEMBL2158192 | ||
| 0.13 | 0.066 | 0.13 | Vanilloid 1 agonist | |||
| 0.083 | 0.019 | 0.187 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.187 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.075 | 0.013 | 0.075 | Carbonic anhydrase IV inhibitor | 0.04 0.033 CHEMBL2158192 | ||
| 0.065 | 0.006 | 0.065 | Peptide deformylase inhibitor | 0.044 0.012 CHEMBL2158192 | ||
| 0.085 | 0.026 | 0.171 | Carbamoyl phosphate synthetase inhibitor | 0.171 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.082 | 0.024 | 0.27 | Alcohol oxidase inhibitor | 0.27 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.061 | 0.004 | 0.078 | Carboxypeptidase B inhibitor | 0.078 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.065 | 0.009 | 0.065 | Arginase inhibitor | 0.065 0.009 CHEMBL2158192 | ||
| 0.166 | 0.112 | 0.166 | Insulin sensitizer | 0.155 0.127 CHEMBL2158192 | ||
| 0.085 | 0.032 | 0.085 | Carbonic anhydrase inhibitor | 0.063 0.044 CHEMBL2158192 | ||
| 0.077 | 0.028 | 0.162 | Biliverdin reductase inhibitor | 0.162 0.008 CHEMBL2158192 | CHEMBL2158192 | |
| 0.064 | 0.017 | 0.065 | Immunoglobulin Fc receptor antagonist | 0.065 0.016 CHEMBL2158192 | CHEMBL2158192 | |
| 0.057 | 0.013 | 0.137 | Integrin alpha5beta1 antagonist | 0.137 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.054 | 0.013 | 0.071 | AMPA 4 receptor antagonist | 0.071 0.008 CHEMBL2158192 | CHEMBL2158192 | |
| 0.058 | 0.018 | 0.058 | Erythropoietin receptor agonist | |||
| 0.121 | 0.081 | 0.225 | Amylase inhibitor | 0.225 0.036 CHEMBL2158192 | CHEMBL2158192 | |
| 0.065 | 0.026 | 0.065 | GP IIb/IIIa receptor antagonist | |||
| 0.125 | 0.088 | 0.145 | Lipid peroxidase inhibitor | 0.145 0.072 CHEMBL2158192 | CHEMBL2158192 | |
| 0.102 | 0.065 | 0.102 | Factor V inhibitor | |||
| 0.057 | 0.023 | 0.057 | HCV NS3/NS4A protease inhibitor | 0.052 0.029 CHEMBL2158192 | ||
| 0.084 | 0.051 | 0.084 | Glycine receptor antagonist | |||
| 0.093 | 0.062 | 0.199 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.199 0.016 CHEMBL2158192 | CHEMBL2158192 | |
| 0.096 | 0.065 | 0.162 | UDP-glucose 4-epimerase inhibitor | 0.162 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.071 | 0.041 | 0.071 | Glucagon-like peptide 1 agonist | |||
| 0.064 | 0.034 | 0.151 | Argininosuccinate synthase inhibitor | 0.151 0.011 CHEMBL2158192 | CHEMBL2158192 | |
| 0.065 | 0.036 | 0.095 | Collagenase 3 inhibitor | 0.095 0.017 CHEMBL2158192 | CHEMBL2158192 | |
| 0.084 | 0.055 | 0.09 | Estrogen-related receptor beta agonist | 0.09 0.041 CHEMBL2158192 | CHEMBL2158192 | |
| 0.059 | 0.032 | 0.064 | Leukotriene C antagonist | 0.064 0.021 CHEMBL2158192 | CHEMBL2158192 | |
| 0.193 | 0.167 | 0.274 | 5 Hydroxytryptamine uptake stimulant | 0.274 0.06 CHEMBL2158192 | CHEMBL2158192 | |
| 0.089 | 0.064 | 0.126 | Thioredoxin inhibitor | 0.126 0.027 CHEMBL2158192 | CHEMBL2158192 | |
| 0.077 | 0.053 | 0.15 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.15 0.019 CHEMBL2158192 | CHEMBL2158192 | |
| 0.026 | 0.003 | 0.029 | Methylmalonyl-CoA mutase inhibitor | 0.029 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.075 | 0.053 | 0.088 | GABA B receptor agonist | 0.088 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.051 | 0.029 | 0.097 | Glucose-6-phosphate isomerase inhibitor | 0.097 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.126 | 0.105 | 0.126 | Thiol protease inhibitor | |||
| 0.03 | 0.011 | 0.031 | Lysophosphatidic acid receptor 1 agonist | 0.031 0.01 CHEMBL2158192 | CHEMBL2158192 | |
| 0.093 | 0.074 | 0.131 | GABA C receptor rho-1 antagonist | 0.131 0.031 CHEMBL2158192 | CHEMBL2158192 | |
| 0.024 | 0.006 | 0.073 | N-Acetylated alpha-linked acidic dipeptidase inhibitor | 0.073 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.066 | 0.048 | 0.113 | Glutamate (mGluR6) antagonist | 0.113 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.18 | 0.163 | 0.361 | Lipoxygenase inhibitor | 0.361 0.048 CHEMBL2158192 | CHEMBL2158192 | |
| 0.037 | 0.021 | 0.085 | Fumarate hydratase inhibitor | 0.085 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.082 | 0.065 | 0.082 | Vanilloid agonist | |||
| 0.038 | 0.022 | 0.06 | p53 inhibitor | 0.06 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.048 | 0.032 | 0.061 | Adenosine deaminase inhibitor | 0.061 0.02 CHEMBL2158192 | CHEMBL2158192 | |
| 0.077 | 0.061 | 0.091 | Carbonic anhydrase VI inhibitor | 0.091 0.045 CHEMBL2158192 | CHEMBL2158192 | |
| 0.027 | 0.012 | 0.033 | Aminopeptidase P inhibitor | 0.033 0.008 CHEMBL2158192 | CHEMBL2158192 | |
| 0.131 | 0.117 | 0.169 | Ca2+-transporting ATPase inhibitor | 0.169 0.014 CHEMBL2158192 | CHEMBL2158192 | |
| 0.018 | 0.004 | 0.036 | Carboxypeptidase B2 inhibitor | 0.036 0.003 CHEMBL2158192 | CHEMBL2158192 | |
| 0.154 | 0.141 | 0.242 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.242 0.046 CHEMBL2158192 | CHEMBL2158192 | |
| 0.03 | 0.018 | 0.03 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.03 0.017 CHEMBL2158192 | ||
| 0.043 | 0.031 | 0.074 | Glutamate (mGluR4) antagonist | 0.074 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.046 | 0.034 | 0.046 | Thymidylate synthase inhibitor | 0.041 0.04 CHEMBL2158192 | ||
| 0.182 | 0.171 | 0.214 | 12-Lipoxygenase inhibitor | 0.214 0.136 CHEMBL2158192 | CHEMBL2158192 | |
| 0.053 | 0.041 | 0.053 | Carbonic anhydrase II inhibitor | |||
| 0.045 | 0.035 | 0.053 | Antimetabolite | 0.053 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.047 | 0.037 | 0.047 | Metalloproteinase-3 inhibitor | 0.046 0.037 CHEMBL2158192 | ||
| 0.112 | 0.102 | 0.112 | Histone deacetylase SIRT1 inhibitor | |||
| 0.053 | 0.045 | 0.053 | Adenine nucleotide translocase inhibitor | |||
| 0.048 | 0.043 | 0.12 | Aconitate hydratase inhibitor | 0.12 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.079 | 0.075 | 0.079 | Hematopoietic | |||
| 0.024 | 0.02 | 0.024 | Histone deacetylase class IIb inhibitor | |||
| 0.023 | 0.02 | 0.023 | Histone deacetylase 6 inhibitor | |||
| 0.086 | 0.083 | 0.137 | Electrolyte absorption antagonist | 0.137 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.037 | 0.034 | 0.042 | Leukotriene C4 antagonist | 0.042 0.019 CHEMBL2158192 | CHEMBL2158192 | |
| 0.052 | 0.051 | 0.052 | Carbonic anhydrase stimulant | |||
| 0.015 | 0.014 | 0.023 | Carbonic anhydrase VIII inhibitor | 0.023 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.015 | 0.014 | 0.023 | Carbonic anhydrase X inhibitor | 0.023 0.006 CHEMBL2158192 | CHEMBL2158192 | |
| 0.033 | 0.033 | 0.088 | Glutamate (mGluR3) antagonist | 0.088 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.034 | 0.035 | 0.065 | Glutamate (mGluR8) agonist | 0.065 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.049 | 0.052 | 0.056 | DNA helicase inhibitor | 0.056 0.034 CHEMBL2158192 | CHEMBL2158192 | |
| 0.022 | 0.025 | 0.036 | CXC chemokine 2 receptor antagonist | 0.036 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.112 | 0.116 | 0.211 | Mannose-6-phosphate isomerase inhibitor | 0.211 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.037 | 0.042 | 0.06 | Kainate receptor agonist | 0.06 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.118 | 0.129 | 0.205 | Arachidonic acid antagonist | 0.205 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.041 | 0.053 | 0.054 | Lysophosphatidic acid 3 receptor antagonist | 0.054 0.03 CHEMBL2158192 | CHEMBL2158192 | |
| 0.097 | 0.111 | 0.103 | Toll-Like receptor 2 antagonist | 0.103 0.1 CHEMBL2158192 | CHEMBL2158192 | |
| 0.074 | 0.088 | 0.117 | D-Ala-D-Ala ligase inhibitor | 0.117 0.015 CHEMBL2158192 | CHEMBL2158192 | |
| 0.008 | 0.022 | 0.017 | Lysophosphatidic acid receptor 3 agonist | 0.017 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.077 | 0.093 | 0.104 | Monophenol monooxygenase inhibitor | 0.104 0.073 CHEMBL2158192 | CHEMBL2158192 | |
| 0.258 | 0.275 | 0.311 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.311 0.198 CHEMBL2158192 | CHEMBL2158192 | |
| 0.053 | 0.07 | 0.06 | Protease 3C (Human rhinovirus) inhibitor | 0.06 0.053 CHEMBL2158192 | CHEMBL2158192 | |
| 0.061 | 0.078 | 0.089 | Glycine receptor agonist | 0.089 0.028 CHEMBL2158192 | CHEMBL2158192 | |
| 0.161 | 0.178 | 0.189 | Nitric-oxide synthase stimulant | 0.189 0.108 CHEMBL2158192 | CHEMBL2158192 | |
| 0.027 | 0.045 | 0.041 | Glutamate (mGluR3) agonist | 0.041 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.076 | 0.095 | 0.149 | Creatine kinase inhibitor | 0.149 0.024 CHEMBL2158192 | CHEMBL2158192 | |
| 0.06 | 0.079 | 0.086 | MDM2 inhibitor | 0.086 0.014 CHEMBL2158192 | CHEMBL2158192 | |
| 0.05 | 0.07 | 0.344 | Peroxisome proliferator-activated receptor gamma agonist | 0.344 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.108 | 0.13 | 0.214 | Protein-tyrosine phosphatase inhibitor | 0.214 0.042 CHEMBL2158192 | CHEMBL2158192 | |
| 0.036 | 0.058 | 0.066 | Glutamate (mGluR group III) antagonist | 0.066 0.01 CHEMBL2158192 | CHEMBL2158192 | |
| 0.079 | 0.103 | 0.097 | Bile acid receptor antagonist | 0.097 0.056 CHEMBL2158192 | CHEMBL2158192 | |
| 0.006 | 0.031 | 0.017 | Glutamate (mGluR6) agonist | 0.017 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.012 | 0.04 | 0.111 | Integrin alphaVbeta1 antagonist | 0.111 0.004 CHEMBL2158192 | CHEMBL2158192 | |
| 0.076 | 0.105 | 0.137 | Xanthine oxidase inhibitor | 0.137 0.04 CHEMBL2158192 | CHEMBL2158192 | |
| 0.009 | 0.039 | 0.017 | Thromboxane A2 agonist | 0.017 0.008 CHEMBL2158192 | CHEMBL2158192 | |
| 0.034 | 0.064 | 0.05 | Carbonic anhydrase VB inhibitor | 0.05 0.045 CHEMBL2158192 | CHEMBL2158192 | |
| 0.134 | 0.165 | 0.156 | Neurotrophic factor enhancer | 0.156 0.13 CHEMBL2158192 | CHEMBL2158192 | |
| 0.111 | 0.147 | 0.153 | GABA C receptor rho-2 antagonist | 0.153 0.07 CHEMBL2158192 | CHEMBL2158192 | |
| 0.027 | 0.067 | 0.041 | Glutamate (mGluR8) antagonist | 0.041 0.016 CHEMBL2158192 | CHEMBL2158192 | |
| 0.104 | 0.144 | 0.209 | Insulin secretagoues | 0.209 0.032 CHEMBL2158192 | CHEMBL2158192 | |
| 0.01 | 0.051 | 0.019 | Telomerase stimulant | 0.019 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.054 | 0.098 | 0.194 | CDC25A inhibitor | 0.194 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.081 | 0.126 | 0.138 | DOPA decarboxylase inhibitor | 0.138 0.028 CHEMBL2158192 | CHEMBL2158192 | |
| 0.083 | 0.129 | 0.118 | Photosensitizer | 0.118 0.059 CHEMBL2158192 | CHEMBL2158192 | |
| 0.184 | 0.231 | 0.367 | 15-Lipoxygenase inhibitor | 0.367 0.09 CHEMBL2158192 | CHEMBL2158192 | |
| 0.023 | 0.07 | 0.047 | Carbonic anhydrase IX inhibitor | 0.047 0.045 CHEMBL2158192 | CHEMBL2158192 | |
| 0.013 | 0.062 | 0.022 | Prostaglandin F2 alpha agonist | 0.022 0.016 CHEMBL2158192 | CHEMBL2158192 | |
| 0.046 | 0.095 | 0.079 | Carbonic anhydrase XIII inhibitor | 0.079 0.051 CHEMBL2158192 | CHEMBL2158192 | |
| 0.018 | 0.07 | 0.047 | Retinoid X alpha receptor agonist | 0.047 0.016 CHEMBL2158192 | CHEMBL2158192 | |
| 0.007 | 0.059 | 0.024 | VLA-4 antagonist | 0.024 0.02 CHEMBL2158192 | CHEMBL2158192 | |
| 0.016 | 0.069 | 0.026 | Vanilloid 2 agonist | 0.026 0.017 CHEMBL2158192 | CHEMBL2158192 | |
| 0.055 | 0.108 | 0.081 | Peroxisome proliferator-activated receptor gamma antagonist | 0.081 0.032 CHEMBL2158192 | CHEMBL2158192 | |
| 0.074 | 0.129 | 0.117 | Cholesterol synthesis inhibitor | 0.117 0.068 CHEMBL2158192 | CHEMBL2158192 | |
| 0.074 | 0.129 | 0.28 | Histone deacetylase class III inhibitor | 0.28 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.024 | 0.08 | 0.063 | Guanylate cyclase inhibitor | 0.063 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.081 | 0.139 | 0.11 | Cyclooxygenase 3 inhibitor | 0.11 0.089 CHEMBL2158192 | CHEMBL2158192 | |
| 0.027 | 0.084 | 0.047 | Dihydroorotase inhibitor | 0.047 0.027 CHEMBL2158192 | CHEMBL2158192 | |
| 0.062 | 0.121 | 0.084 | Sphingomyelinase inhibitor | 0.084 0.081 CHEMBL2158192 | CHEMBL2158192 | |
| 0.051 | 0.111 | 0.079 | Ornithine decarboxylase inhibitor | 0.079 0.068 CHEMBL2158192 | CHEMBL2158192 | |
| 0.03 | 0.091 | 0.059 | Diacylglycerol O-acyltransferase inhibitor | 0.059 0.026 CHEMBL2158192 | CHEMBL2158192 | |
| 0.021 | 0.082 | 0.063 | Peroxisome proliferator-activated receptor alpha agonist | 0.063 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.029 | 0.09 | 0.046 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.046 0.02 CHEMBL2158192 | CHEMBL2158192 | |
| 0.038 | 0.1 | 0.111 | HIV-1 reverse transcriptase inhibitor | 0.111 0.025 CHEMBL2158192 | CHEMBL2158192 | |
| 0.01 | 0.074 | 0.024 | Retinoid X gamma receptor agonist | 0.024 0.015 CHEMBL2158192 | CHEMBL2158192 | |
| 0.032 | 0.098 | 0.05 | Dopamine beta hydroxylase inhibitor | 0.05 0.031 CHEMBL2158192 | CHEMBL2158192 | |
| 0.065 | 0.131 | 0.095 | Granulocyte macrophage colony stimulating factor agonist | 0.095 0.042 CHEMBL2158192 | CHEMBL2158192 | |
| 0.049 | 0.117 | 0.076 | GABA aminotransferase inhibitor | 0.076 0.052 CHEMBL2158192 | CHEMBL2158192 | |
| 0.052 | 0.125 | 0.076 | Keratolytic | 0.076 0.054 CHEMBL2158192 | CHEMBL2158192 | |
| 0.008 | 0.082 | 0.021 | Retinoid X beta receptor agonist | 0.021 0.015 CHEMBL2158192 | CHEMBL2158192 | |
| 0.212 | 0.287 | 0.346 | 5 Hydroxytryptamine release inhibitor | 0.346 0.119 CHEMBL2158192 | CHEMBL2158192 | |
| 0.133 | 0.211 | 0.319 | Hypoglycemic | 0.319 0.047 CHEMBL2158192 | CHEMBL2158192 | |
| 0.012 | 0.089 | 0.022 | Retinoid X beta receptor antagonist | 0.022 0.011 CHEMBL2158192 | CHEMBL2158192 | |
| 0.02 | 0.1 | 0.038 | GABA uptake inhibitor | 0.038 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.141 | 0.223 | 0.225 | RNA-directed DNA polymerase inhibitor | 0.225 0.069 CHEMBL2158192 | CHEMBL2158192 | |
| 0.08 | 0.163 | 0.116 | Interleukin 8 antagonist | 0.116 0.067 CHEMBL2158192 | CHEMBL2158192 | |
| 0.011 | 0.097 | 0.041 | Retinoid X receptor agonist | 0.041 0.022 CHEMBL2158192 | CHEMBL2158192 | |
| 0.082 | 0.17 | 0.157 | Protein kinase stimulant | 0.157 0.064 CHEMBL2158192 | CHEMBL2158192 | |
| 0.109 | 0.196 | 0.163 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.163 0.127 CHEMBL2158192 | CHEMBL2158192 | |
| 0.033 | 0.127 | 0.054 | Thromboxane synthase inhibitor | 0.054 0.039 CHEMBL2158192 | CHEMBL2158192 | |
| 0.107 | 0.206 | 0.182 | Interleukin agonist | 0.182 0.138 CHEMBL2158192 | CHEMBL2158192 | |
| 0.076 | 0.176 | 0.128 | Cytidine deaminase inhibitor | 0.128 0.093 CHEMBL2158192 | CHEMBL2158192 | |
| 0.035 | 0.139 | 0.076 | Purinergic P2X1 antagonist | 0.076 0.027 CHEMBL2158192 | CHEMBL2158192 | |
| 0.051 | 0.158 | 0.087 | Prolactin inhibitor | 0.087 0.071 CHEMBL2158192 | CHEMBL2158192 | |
| 0.141 | 0.257 | 0.271 | Vasodilator, peripheral | 0.271 0.113 CHEMBL2158192 | CHEMBL2158192 | |
| 0.043 | 0.168 | 0.064 | Exportin-1 inhibitor | 0.064 0.059 CHEMBL2158192 | CHEMBL2158192 | |
| 0.031 | 0.157 | 0.071 | Na+ K+ transporting ATPase inhibitor | 0.071 0.059 CHEMBL2158192 | CHEMBL2158192 | |
| 0.13 | 0.256 | 0.211 | Hypoxia-inducible factor 1 alpha inhibitor | 0.211 0.139 CHEMBL2158192 | CHEMBL2158192 | |
| 0.018 | 0.144 | 0.033 | Retinoid X alpha receptor antagonist | 0.033 0.026 CHEMBL2158192 | CHEMBL2158192 | |
| 0.01 | 0.138 | 0.077 | Urate transporter 1 inhibitor | 0.077 0.009 CHEMBL2158192 | CHEMBL2158192 | |
| 0.061 | 0.192 | 0.091 | Toll-Like receptor 4 antagonist | 0.091 0.086 CHEMBL2158192 | CHEMBL2158192 | |
| 0.019 | 0.154 | 0.037 | Retinoid X receptor antagonist | 0.037 0.029 CHEMBL2158192 | CHEMBL2158192 | |
| 0.046 | 0.193 | 0.275 | Uric acid excretion stimulant | 0.275 0.005 CHEMBL2158192 | CHEMBL2158192 | |
| 0.048 | 0.198 | 0.147 | Cystathionine beta-synthase inhibitor | 0.147 0.042 CHEMBL2158192 | CHEMBL2158192 | |
| 0.008 | 0.161 | 0.03 | Peroxisome proliferator-activated receptor delta agonist | 0.03 0.028 CHEMBL2158192 | CHEMBL2158192 | |
| 0.11 | 0.275 | 0.244 | Thioredoxin glutathione reductase inhibitor | 0.244 0.138 CHEMBL2158192 | CHEMBL2158192 | |
| 0.086 | 0.254 | 0.137 | Interferon gamma antagonist | 0.137 0.098 CHEMBL2158192 | CHEMBL2158192 | |
| 0.049 | 0.22 | 0.198 | Cyclooxygenase 1 inhibitor | 0.198 0.035 CHEMBL2158192 | CHEMBL2158192 | |
| 0.036 | 0.209 | 0.079 | Inducible nitric-oxide synthase inhibitor | 0.079 0.063 CHEMBL2158192 | CHEMBL2158192 | |
| 0.107 | 0.294 | 0.179 | 5 Hydroxytryptamine release stimulant | 0.179 0.141 CHEMBL2158192 | CHEMBL2158192 | |
| 0.089 | 0.284 | 0.141 | Lipocortins synthesis antagonist | 0.141 0.119 CHEMBL2158192 | CHEMBL2158192 | |
| 0.006 | 0.21 | 0.027 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.027 0.021 CHEMBL2158192 | CHEMBL2158192 | |
| 0.029 | 0.236 | 0.07 | Glutamate (mGluR7) antagonist | 0.07 0.042 CHEMBL2158192 | CHEMBL2158192 | |
| 0.085 | 0.294 | 0.198 | Prostaglandin dehydrogenase inhibitor | 0.198 0.158 CHEMBL2158192 | CHEMBL2158192 | |
| 0.021 | 0.243 | 0.09 | CDC25B inhibitor | 0.09 0.021 CHEMBL2158192 | CHEMBL2158192 | |
| 0.029 | 0.253 | 0.346 | 5-Lipoxygenase inhibitor | 0.346 0.007 CHEMBL2158192 | CHEMBL2158192 | |
| 0.107 | 0.382 | 0.215 | Antibacterial | 0.215 0.212 CHEMBL2158192 | CHEMBL2158192 | |
| 0.113 | 0.391 | 0.233 | Calcium channel activator | 0.233 0.168 CHEMBL2158192 | CHEMBL2158192 | |
| 0.038 | 0.476 | 0.227 | Streptokinase A inhibitor | 0.227 0.117 CHEMBL2158192 | CHEMBL2158192 | |
| 0.057 | 0.613 | 0.37 | Cyclophilin D inhibitor | 0.37 0.109 CHEMBL2158192 | CHEMBL2158192 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |