| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.719 | 0.002 | 0.735 | Interleukin 8 antagonist | 0.735 0.002 CHEMBL1031 0.376 0.004 CHEMBL1033 0.67 0.003 CHEMBL1030 0.593 0.003 CHEMBL1035 0.644 0.003 CHEMBL1032 | CHEMBL1031 | |
| 0.717 | 0.028 | 0.72 | Antiinflammatory | 0.707 0.029 CHEMBL1031 0.602 0.053 CHEMBL1033 0.709 0.029 CHEMBL1030 0.647 0.041 CHEMBL1035 0.72 0.027 CHEMBL1032 | CHEMBL1032 | |
| 0.622 | 0.004 | 0.622 | Non-steroidal antiinflammatory agent | 0.62 0.004 CHEMBL1031 0.52 0.006 CHEMBL1033 0.578 0.005 CHEMBL1030 0.535 0.005 CHEMBL1035 0.578 0.005 CHEMBL1032 | ||
| 0.585 | 0.002 | 0.617 | Cyclooxygenase 3 inhibitor | 0.617 0.002 CHEMBL1031 0.492 0.003 CHEMBL1033 0.56 0.003 CHEMBL1030 0.547 0.003 CHEMBL1035 0.568 0.003 CHEMBL1032 | CHEMBL1031 | |
| 0.566 | 0.004 | 0.566 | Cyclooxygenase 1 inhibitor | 0.533 0.005 CHEMBL1031 0.431 0.006 CHEMBL1033 0.532 0.005 CHEMBL1030 0.483 0.005 CHEMBL1035 0.538 0.005 CHEMBL1032 | ||
| 0.513 | 0.019 | 0.517 | Interleukin antagonist | 0.517 0.018 CHEMBL1031 0.348 0.039 CHEMBL1033 0.506 0.019 CHEMBL1030 0.444 0.025 CHEMBL1035 0.504 0.019 CHEMBL1032 | CHEMBL1031 | |
| 0.511 | 0.031 | 0.647 | Aldehyde oxidase inhibitor | 0.647 0.013 CHEMBL1031 0.384 0.049 CHEMBL1033 0.559 0.025 CHEMBL1030 0.471 0.037 CHEMBL1035 0.593 0.02 CHEMBL1032 | CHEMBL1031 | |
| 0.454 | 0.011 | 0.454 | Anesthetic general | 0.453 0.011 CHEMBL1031 0.315 0.03 CHEMBL1033 0.415 0.015 CHEMBL1030 0.372 0.02 CHEMBL1035 0.396 0.017 CHEMBL1032 | ||
| 0.481 | 0.039 | 0.481 | 5 Hydroxytryptamine release inhibitor | 0.474 0.041 CHEMBL1031 0.349 0.116 CHEMBL1033 0.449 0.052 CHEMBL1030 0.408 0.073 CHEMBL1035 0.435 0.059 CHEMBL1032 | ||
| 0.437 | 0.004 | 0.437 | Prostaglandin antagonist | 0.302 0.005 CHEMBL1031 0.162 0.009 CHEMBL1033 0.301 0.005 CHEMBL1030 0.247 0.005 CHEMBL1035 0.303 0.005 CHEMBL1032 | ||
| 0.433 | 0.006 | 0.433 | Cyclooxygenase inhibitor | 0.403 0.007 CHEMBL1031 0.338 0.012 CHEMBL1033 0.401 0.007 CHEMBL1030 0.384 0.008 CHEMBL1035 0.404 0.007 CHEMBL1032 | ||
| 0.366 | 0.005 | 0.366 | Succinate dehydrogenase inhibitor | 0.356 0.005 CHEMBL1031 0.296 0.011 CHEMBL1033 0.321 0.008 CHEMBL1030 0.323 0.008 CHEMBL1035 0.332 0.007 CHEMBL1032 | ||
| 0.42 | 0.065 | 0.442 | Histamine release inhibitor | 0.442 0.054 CHEMBL1031 0.251 0.154 CHEMBL1033 0.417 0.067 CHEMBL1030 0.36 0.095 CHEMBL1035 0.411 0.07 CHEMBL1032 | CHEMBL1031 | |
| 0.428 | 0.076 | 0.449 | Cyclophilin D inhibitor | 0.42 0.08 CHEMBL1031 0.277 0.184 CHEMBL1033 0.423 0.079 CHEMBL1030 0.344 0.127 CHEMBL1035 0.449 0.067 CHEMBL1032 | CHEMBL1032 | |
| 0.402 | 0.059 | 0.402 | Toll-Like receptor 7 agonist | 0.355 0.079 CHEMBL1031 0.297 0.112 CHEMBL1033 0.34 0.087 CHEMBL1030 0.276 0.126 CHEMBL1035 0.363 0.076 CHEMBL1032 | ||
| 0.375 | 0.035 | 0.377 | Interleukin 2 agonist | 0.377 0.035 CHEMBL1031 0.296 0.077 CHEMBL1033 0.37 0.037 CHEMBL1030 0.347 0.047 CHEMBL1035 0.374 0.036 CHEMBL1032 | CHEMBL1031 | |
| 0.344 | 0.004 | 0.357 | ATPase inhibitor | 0.357 0.004 CHEMBL1031 0.302 0.006 CHEMBL1033 0.354 0.004 CHEMBL1030 0.293 0.007 CHEMBL1035 0.354 0.004 CHEMBL1032 | CHEMBL1031 | |
| 0.416 | 0.077 | 0.416 | Analgesic | 0.39 0.089 CHEMBL1031 0.415 0.078 CHEMBL1030 0.276 0.161 CHEMBL1035 0.407 0.081 CHEMBL1032 | ||
| 0.397 | 0.061 | 0.397 | Toll-Like receptor agonist | 0.348 0.083 CHEMBL1031 0.291 0.116 CHEMBL1033 0.334 0.091 CHEMBL1030 0.269 0.132 CHEMBL1035 0.356 0.079 CHEMBL1032 | ||
| 0.357 | 0.024 | 0.372 | Cyclic AMP phosphodiesterase inhibitor | 0.372 0.021 CHEMBL1031 0.274 0.053 CHEMBL1033 0.324 0.033 CHEMBL1030 0.272 0.054 CHEMBL1035 0.344 0.027 CHEMBL1032 | CHEMBL1031 | |
| 0.371 | 0.045 | 0.499 | Lipoxygenase inhibitor | 0.499 0.019 CHEMBL1031 0.479 0.021 CHEMBL1033 0.435 0.029 CHEMBL1030 0.403 0.037 CHEMBL1035 0.464 0.024 CHEMBL1032 | CHEMBL1031 | |
| 0.339 | 0.013 | 0.339 | Gastrin inhibitor | 0.293 0.038 CHEMBL1031 0.225 0.112 CHEMBL1033 0.29 0.04 CHEMBL1030 0.271 0.057 CHEMBL1035 0.275 0.053 CHEMBL1032 | ||
| 0.32 | 0.011 | 0.32 | Cyclooxygenase 2 inhibitor | 0.298 0.014 CHEMBL1031 0.247 0.02 CHEMBL1033 0.297 0.014 CHEMBL1030 0.288 0.015 CHEMBL1035 0.298 0.014 CHEMBL1032 | ||
| 0.316 | 0.008 | 0.316 | GABA C receptor agonist | 0.218 0.017 CHEMBL1031 0.098 0.069 CHEMBL1033 0.249 0.014 CHEMBL1030 0.19 0.022 CHEMBL1035 0.249 0.014 CHEMBL1032 | ||
| 0.35 | 0.05 | 0.35 | Calcium channel activator | 0.347 0.052 CHEMBL1031 0.315 0.078 CHEMBL1033 0.314 0.078 CHEMBL1030 0.296 0.096 CHEMBL1035 0.317 0.076 CHEMBL1032 | ||
| 0.29 | 0.008 | 0.29 | Ferrochelatase inhibitor | 0.125 0.051 CHEMBL1031 0.169 0.031 CHEMBL1030 0.12 0.053 CHEMBL1035 0.14 0.042 CHEMBL1032 | ||
| 0.345 | 0.066 | 0.379 | Cholesterol antagonist | 0.379 0.054 CHEMBL1031 0.23 0.14 CHEMBL1033 0.322 0.078 CHEMBL1030 0.305 0.088 CHEMBL1035 0.332 0.072 CHEMBL1032 | CHEMBL1031 | |
| 0.328 | 0.055 | 0.364 | Sodium/bile acid cotransporter inhibitor | 0.362 0.033 CHEMBL1031 0.326 0.057 CHEMBL1033 0.352 0.038 CHEMBL1030 0.33 0.054 CHEMBL1035 0.364 0.032 CHEMBL1032 | CHEMBL1032 | |
| 0.31 | 0.04 | 0.31 | 5 Hydroxytryptamine uptake stimulant | 0.305 0.042 CHEMBL1031 0.236 0.096 CHEMBL1033 0.266 0.066 CHEMBL1030 0.281 0.056 CHEMBL1035 0.267 0.066 CHEMBL1032 | ||
| 0.269 | 0.003 | 0.27 | Arachidonic acid antagonist | 0.27 0.003 CHEMBL1031 0.244 0.007 CHEMBL1033 0.263 0.004 CHEMBL1030 0.264 0.004 CHEMBL1035 0.267 0.004 CHEMBL1032 | CHEMBL1031 | |
| 0.271 | 0.006 | 0.286 | Potassium channel (Ca-activated) activator | 0.286 0.005 CHEMBL1031 0.147 0.029 CHEMBL1033 0.274 0.006 CHEMBL1030 0.239 0.009 CHEMBL1035 0.249 0.008 CHEMBL1032 | CHEMBL1031 | |
| 0.293 | 0.037 | 0.358 | Tyrosine 3 hydroxylase inhibitor | 0.358 0.014 CHEMBL1031 0.239 0.08 CHEMBL1033 0.339 0.019 CHEMBL1030 0.288 0.039 CHEMBL1035 0.357 0.014 CHEMBL1032 | CHEMBL1031 | |
| 0.281 | 0.029 | 0.281 | Src kinase inhibitor | 0.246 0.037 CHEMBL1031 0.201 0.054 CHEMBL1033 0.24 0.039 CHEMBL1030 0.263 0.033 CHEMBL1035 0.236 0.04 CHEMBL1032 | ||
| 0.271 | 0.02 | 0.271 | Lck kinase inhibitor | 0.23 0.03 CHEMBL1031 0.194 0.043 CHEMBL1033 0.225 0.031 CHEMBL1030 0.211 0.036 CHEMBL1035 0.219 0.033 CHEMBL1032 | ||
| 0.253 | 0.004 | 0.253 | Prostaglandin D2 antagonist | 0.138 0.004 CHEMBL1031 0.064 0.005 CHEMBL1033 0.142 0.004 CHEMBL1030 0.109 0.005 CHEMBL1035 0.142 0.004 CHEMBL1032 | ||
| 0.291 | 0.053 | 0.291 | Interleukin agonist | 0.284 0.056 CHEMBL1031 0.253 0.077 CHEMBL1030 0.226 0.098 CHEMBL1035 0.268 0.066 CHEMBL1032 | ||
| 0.255 | 0.022 | 0.268 | Phospholipase A2 inhibitor | 0.268 0.019 CHEMBL1031 0.203 0.041 CHEMBL1033 0.255 0.022 CHEMBL1030 0.268 0.019 CHEMBL1035 0.256 0.022 CHEMBL1032 | CHEMBL1035 | |
| 0.236 | 0.005 | 0.236 | Electrolyte absorption antagonist | 0.156 0.017 CHEMBL1031 0.107 0.049 CHEMBL1033 0.191 0.009 CHEMBL1030 0.154 0.018 CHEMBL1035 0.167 0.014 CHEMBL1032 | ||
| 0.246 | 0.024 | 0.246 | Alpha-N-acetylglucosaminidase inhibitor | 0.14 0.061 CHEMBL1031 0.18 0.041 CHEMBL1030 0.139 0.062 CHEMBL1035 0.16 0.05 CHEMBL1032 | ||
| 0.228 | 0.007 | 0.228 | HIV-1 integrase (Overall Integration) inhibitor | 0.228 0.007 CHEMBL1031 0.116 0.042 CHEMBL1033 0.198 0.012 CHEMBL1030 0.206 0.01 CHEMBL1035 0.197 0.012 CHEMBL1032 | ||
| 0.24 | 0.021 | 0.24 | Insulin secretagoues | 0.232 0.024 CHEMBL1031 0.145 0.08 CHEMBL1033 0.215 0.029 CHEMBL1030 0.174 0.053 CHEMBL1035 0.227 0.025 CHEMBL1032 | ||
| 0.32 | 0.103 | 0.371 | GABA C receptor rho-3 antagonist | 0.371 0.075 CHEMBL1031 0.32 0.103 CHEMBL1030 0.268 0.139 CHEMBL1035 0.321 0.102 CHEMBL1032 | CHEMBL1031 | |
| 0.222 | 0.013 | 0.222 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.136 0.031 CHEMBL1031 0.092 0.063 CHEMBL1033 0.176 0.02 CHEMBL1030 0.137 0.031 CHEMBL1035 0.151 0.026 CHEMBL1032 | ||
| 0.227 | 0.024 | 0.227 | Interleukin 1 antagonist | 0.211 0.029 CHEMBL1031 0.14 0.065 CHEMBL1033 0.188 0.038 CHEMBL1030 0.157 0.053 CHEMBL1035 0.189 0.038 CHEMBL1032 | ||
| 0.294 | 0.092 | 0.294 | Antithrombotic | 0.293 0.093 CHEMBL1031 0.261 0.118 CHEMBL1033 0.284 0.099 CHEMBL1030 0.286 0.098 CHEMBL1035 0.29 0.095 CHEMBL1032 | ||
| 0.214 | 0.012 | 0.308 | Histidine decarboxylase inhibitor | 0.308 0.006 CHEMBL1031 0.114 0.027 CHEMBL1033 0.259 0.008 CHEMBL1030 0.187 0.014 CHEMBL1035 0.294 0.007 CHEMBL1032 | CHEMBL1031 | |
| 0.207 | 0.005 | 0.207 | Prostaglandin-E synthase inhibitor | 0.186 0.007 CHEMBL1031 0.078 0.04 CHEMBL1033 0.174 0.008 CHEMBL1030 0.134 0.015 CHEMBL1035 0.159 0.01 CHEMBL1032 | ||
| 0.203 | 0.005 | 0.203 | NMDA receptor agonist | 0.142 0.009 CHEMBL1031 0.065 0.041 CHEMBL1033 0.148 0.008 CHEMBL1030 0.125 0.012 CHEMBL1035 0.126 0.012 CHEMBL1032 | ||
| 0.195 | 0.008 | 0.195 | Interleukin 2 antagonist | 0.159 0.015 CHEMBL1031 0.121 0.043 CHEMBL1033 0.155 0.016 CHEMBL1030 0.167 0.013 CHEMBL1035 0.147 0.02 CHEMBL1032 | ||
| 0.27 | 0.089 | 0.315 | Immunostimulant | 0.297 0.079 CHEMBL1031 0.165 0.143 CHEMBL1033 0.301 0.078 CHEMBL1030 0.206 0.117 CHEMBL1035 0.315 0.075 CHEMBL1032 | CHEMBL1032 | |
| 0.337 | 0.156 | 0.415 | Caspase 9 stimulant | 0.415 0.102 CHEMBL1031 0.338 0.156 CHEMBL1033 0.355 0.141 CHEMBL1030 0.299 0.195 CHEMBL1035 0.388 0.118 CHEMBL1032 | CHEMBL1031 | |
| 0.282 | 0.105 | 0.394 | Transcription factor NF kappa B inhibitor | 0.394 0.065 CHEMBL1031 0.347 0.078 CHEMBL1033 0.336 0.081 CHEMBL1030 0.305 0.091 CHEMBL1035 0.372 0.07 CHEMBL1032 | CHEMBL1031 | |
| 0.229 | 0.052 | 0.426 | Peroxidase inhibitor | 0.422 0.018 CHEMBL1031 0.122 0.098 CHEMBL1033 0.368 0.025 CHEMBL1030 0.34 0.03 CHEMBL1035 0.426 0.017 CHEMBL1032 | CHEMBL1032 | |
| 0.186 | 0.012 | 0.186 | Sphingosine 1-phosphate receptor 4 antagonist | 0.161 0.024 CHEMBL1031 0.128 0.059 CHEMBL1033 0.147 0.036 CHEMBL1030 0.168 0.02 CHEMBL1035 0.142 0.041 CHEMBL1032 | ||
| 0.177 | 0.005 | 0.177 | Sphingosine 1-phosphate receptor 4 agonist | 0.151 0.008 CHEMBL1031 0.08 0.037 CHEMBL1033 0.159 0.007 CHEMBL1030 0.126 0.014 CHEMBL1035 0.159 0.007 CHEMBL1032 | ||
| 0.231 | 0.061 | 0.249 | Platelet aggregation inhibitor | 0.178 0.099 CHEMBL1031 0.249 0.052 CHEMBL1033 0.196 0.084 CHEMBL1030 0.169 0.108 CHEMBL1035 0.203 0.079 CHEMBL1032 | CHEMBL1033 | |
| 0.172 | 0.005 | 0.221 | Bile acid receptor antagonist | 0.21 0.004 CHEMBL1031 0.137 0.01 CHEMBL1033 0.208 0.004 CHEMBL1030 0.152 0.007 CHEMBL1035 0.221 0.004 CHEMBL1032 | CHEMBL1032 | |
| 0.217 | 0.063 | 0.23 | Nitric-oxide synthase stimulant | 0.23 0.048 CHEMBL1031 0.189 0.109 CHEMBL1033 0.221 0.059 CHEMBL1030 0.196 0.095 CHEMBL1035 0.229 0.05 CHEMBL1032 | CHEMBL1031 | |
| 0.163 | 0.016 | 0.212 | DOPA decarboxylase inhibitor | 0.211 0.005 CHEMBL1031 0.121 0.044 CHEMBL1033 0.187 0.009 CHEMBL1030 0.166 0.015 CHEMBL1035 0.212 0.005 CHEMBL1032 | CHEMBL1032 | |
| 0.151 | 0.004 | 0.151 | CXC chemokine 1 receptor antagonist | 0.145 0.004 CHEMBL1031 0.085 0.007 CHEMBL1033 0.145 0.004 CHEMBL1030 0.124 0.005 CHEMBL1035 0.132 0.005 CHEMBL1032 | ||
| 0.161 | 0.017 | 0.161 | Potassium channel activator | 0.119 0.033 CHEMBL1031 0.119 0.033 CHEMBL1030 0.1 0.048 CHEMBL1035 0.103 0.044 CHEMBL1032 | ||
| 0.176 | 0.033 | 0.176 | Cell adhesion inhibitor | 0.145 0.05 CHEMBL1031 0.159 0.041 CHEMBL1033 0.132 0.057 CHEMBL1030 0.17 0.035 CHEMBL1035 0.131 0.058 CHEMBL1032 | ||
| 0.174 | 0.031 | 0.201 | Protein kinase (CK2) alpha inhibitor | 0.165 0.034 CHEMBL1031 0.174 0.031 CHEMBL1033 0.164 0.034 CHEMBL1030 0.201 0.024 CHEMBL1035 0.157 0.038 CHEMBL1032 | CHEMBL1035 | |
| 0.146 | 0.005 | 0.146 | NMDA receptor glycine site agonist | 0.113 0.011 CHEMBL1031 0.065 0.041 CHEMBL1033 0.114 0.011 CHEMBL1030 0.107 0.013 CHEMBL1035 0.101 0.016 CHEMBL1032 | ||
| 0.187 | 0.046 | 0.251 | Interferon gamma antagonist | 0.224 0.034 CHEMBL1031 0.171 0.056 CHEMBL1033 0.229 0.033 CHEMBL1030 0.172 0.055 CHEMBL1035 0.251 0.028 CHEMBL1032 | CHEMBL1032 | |
| 0.148 | 0.007 | 0.148 | Elastase 1 inhibitor | 0.133 0.009 CHEMBL1031 0.101 0.019 CHEMBL1033 0.133 0.009 CHEMBL1030 0.121 0.011 CHEMBL1035 0.128 0.01 CHEMBL1032 | ||
| 0.189 | 0.048 | 0.189 | Diuretic | 0.156 0.073 CHEMBL1031 0.17 0.061 CHEMBL1030 0.128 0.096 CHEMBL1035 0.157 0.072 CHEMBL1032 | ||
| 0.323 | 0.183 | 0.323 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | |||
| 0.171 | 0.032 | 0.273 | Cystathionine beta-synthase inhibitor | 0.273 0.012 CHEMBL1031 0.125 0.054 CHEMBL1033 0.208 0.023 CHEMBL1030 0.227 0.019 CHEMBL1035 0.246 0.016 CHEMBL1032 | CHEMBL1031 | |
| 0.171 | 0.033 | 0.171 | Sphingosine 1-phosphate receptor 5 antagonist | 0.157 0.05 CHEMBL1031 0.161 0.044 CHEMBL1030 0.142 0.076 CHEMBL1035 0.164 0.041 CHEMBL1032 | ||
| 0.167 | 0.03 | 0.167 | Interleukin 1b antagonist | 0.148 0.042 CHEMBL1031 0.129 0.056 CHEMBL1033 0.137 0.049 CHEMBL1030 0.114 0.067 CHEMBL1035 0.133 0.052 CHEMBL1032 | ||
| 0.161 | 0.024 | 0.161 | Catalase inhibitor | 0.126 0.032 CHEMBL1031 0.108 0.036 CHEMBL1030 0.075 0.051 CHEMBL1035 0.108 0.036 CHEMBL1032 | ||
| 0.256 | 0.12 | 0.308 | Thyroid hormone antagonist | 0.288 0.099 CHEMBL1031 0.275 0.108 CHEMBL1033 0.282 0.103 CHEMBL1030 0.249 0.124 CHEMBL1035 0.308 0.089 CHEMBL1032 | CHEMBL1032 | |
| 0.147 | 0.018 | 0.147 | ABCA1 expression enhancer | 0.135 0.022 CHEMBL1031 0.1 0.05 CHEMBL1033 0.133 0.023 CHEMBL1030 0.115 0.035 CHEMBL1035 0.136 0.022 CHEMBL1032 | ||
| 0.134 | 0.008 | 0.157 | NMDA receptor subunit 3B antagonist | 0.157 0.005 CHEMBL1031 0.141 0.007 CHEMBL1030 0.142 0.007 CHEMBL1035 0.112 0.009 CHEMBL1032 | CHEMBL1031 | |
| 0.15 | 0.026 | 0.15 | Adenylate kinase inhibitor | 0.111 0.052 CHEMBL1031 0.126 0.039 CHEMBL1030 0.105 0.059 CHEMBL1035 0.117 0.046 CHEMBL1032 | ||
| 0.177 | 0.056 | 0.188 | Catenin beta inhibitor | 0.188 0.043 CHEMBL1031 0.141 0.128 CHEMBL1033 0.176 0.057 CHEMBL1030 0.162 0.08 CHEMBL1035 0.174 0.061 CHEMBL1032 | CHEMBL1031 | |
| 0.233 | 0.113 | 0.239 | Insulysin inhibitor | 0.234 0.112 CHEMBL1031 0.239 0.107 CHEMBL1030 0.187 0.178 CHEMBL1035 0.222 0.126 CHEMBL1032 | CHEMBL1030 | |
| 0.146 | 0.026 | 0.177 | NMDA receptor antagonist | 0.177 0.018 CHEMBL1031 0.16 0.022 CHEMBL1030 0.109 0.041 CHEMBL1035 0.135 0.029 CHEMBL1032 | CHEMBL1031 | |
| 0.171 | 0.057 | 0.18 | Hexokinase inhibitor | 0.18 0.049 CHEMBL1031 0.137 0.095 CHEMBL1033 0.16 0.067 CHEMBL1030 0.175 0.053 CHEMBL1035 0.156 0.072 CHEMBL1032 | CHEMBL1031 | |
| 0.161 | 0.052 | 0.161 | MAP kinase 3 inhibitor | 0.133 0.099 CHEMBL1031 | ||
| 0.115 | 0.007 | 0.137 | NMDA receptor subunit 3A antagonist | 0.137 0.005 CHEMBL1031 0.122 0.006 CHEMBL1030 0.111 0.007 CHEMBL1035 0.098 0.009 CHEMBL1032 | CHEMBL1031 | |
| 0.114 | 0.006 | 0.114 | Kainate receptor antagonist | 0.069 0.013 CHEMBL1031 0.08 0.01 CHEMBL1030 0.05 0.021 CHEMBL1035 0.07 0.012 CHEMBL1032 | ||
| 0.123 | 0.016 | 0.123 | Potassium channel large-conductance Ca-activated activator | 0.123 0.016 CHEMBL1031 0.074 0.039 CHEMBL1033 0.122 0.016 CHEMBL1030 0.112 0.019 CHEMBL1035 0.112 0.019 CHEMBL1032 | ||
| 0.234 | 0.129 | 0.278 | Thyroid hormone beta antagonist | 0.263 0.11 CHEMBL1031 0.257 0.114 CHEMBL1033 0.258 0.113 CHEMBL1030 0.225 0.135 CHEMBL1035 0.278 0.1 CHEMBL1032 | CHEMBL1032 | |
| 0.122 | 0.019 | 0.129 | Peroxisome proliferator-activated receptor gamma agonist | 0.112 0.022 CHEMBL1031 0.076 0.044 CHEMBL1033 0.112 0.022 CHEMBL1030 0.085 0.037 CHEMBL1035 0.129 0.018 CHEMBL1032 | CHEMBL1032 | |
| 0.14 | 0.04 | 0.14 | CC chemokine 6 receptor antagonist | 0.137 0.047 CHEMBL1031 0.13 0.072 CHEMBL1033 0.137 0.046 CHEMBL1030 0.137 0.046 CHEMBL1035 0.133 0.059 CHEMBL1032 | ||
| 0.126 | 0.025 | 0.126 | Lanosterol 14 alpha demethylase inhibitor | 0.102 0.052 CHEMBL1031 0.099 0.057 CHEMBL1030 0.089 0.073 CHEMBL1035 | ||
| 0.119 | 0.021 | 0.163 | Glutamate decarboxylase inhibitor | 0.156 0.012 CHEMBL1031 0.066 0.06 CHEMBL1033 0.145 0.014 CHEMBL1030 0.105 0.027 CHEMBL1035 0.163 0.011 CHEMBL1032 | CHEMBL1032 | |
| 0.136 | 0.038 | 0.136 | GABA C receptor antagonist | 0.116 0.057 CHEMBL1031 0.124 0.049 CHEMBL1030 0.092 0.091 CHEMBL1035 0.114 0.059 CHEMBL1032 | ||
| 0.109 | 0.011 | 0.128 | GABA B receptor agonist | 0.128 0.005 CHEMBL1031 0.085 0.033 CHEMBL1033 0.107 0.012 CHEMBL1030 0.098 0.018 CHEMBL1035 0.113 0.01 CHEMBL1032 | CHEMBL1031 | |
| 0.124 | 0.03 | 0.124 | Triose-phosphate isomerase inhibitor | 0.09 0.059 CHEMBL1031 0.1 0.048 CHEMBL1030 0.089 0.061 CHEMBL1035 0.094 0.055 CHEMBL1032 | ||
| 0.118 | 0.026 | 0.163 | Adrenaline agonist | 0.163 0.012 CHEMBL1031 0.077 0.062 CHEMBL1033 0.147 0.015 CHEMBL1030 0.14 0.017 CHEMBL1035 0.154 0.014 CHEMBL1032 | CHEMBL1031 | |
| 0.102 | 0.01 | 0.102 | Thromboxane antagonist | 0.087 0.016 CHEMBL1031 0.048 0.043 CHEMBL1033 0.08 0.02 CHEMBL1030 0.093 0.014 CHEMBL1035 0.076 0.022 CHEMBL1032 | ||
| 0.099 | 0.008 | 0.099 | Diacylglycerol O-acyltransferase inhibitor | 0.059 0.027 CHEMBL1031 0.06 0.026 CHEMBL1030 0.046 0.042 CHEMBL1035 0.055 0.03 CHEMBL1032 | ||
| 0.145 | 0.055 | 0.145 | Ca2+-transporting ATPase inhibitor | 0.136 0.091 CHEMBL1031 0.138 0.08 CHEMBL1030 0.135 0.094 CHEMBL1035 0.134 0.1 CHEMBL1032 | ||
| 0.126 | 0.035 | 0.126 | GABA C receptor rho-1 antagonist | 0.105 0.055 CHEMBL1031 0.106 0.055 CHEMBL1030 0.099 0.064 CHEMBL1032 | ||
| 0.11 | 0.019 | 0.12 | D-Ala-D-Ala ligase inhibitor | 0.12 0.014 CHEMBL1031 0.088 0.048 CHEMBL1033 0.115 0.016 CHEMBL1030 0.112 0.018 CHEMBL1035 0.108 0.021 CHEMBL1032 | CHEMBL1031 | |
| 0.142 | 0.052 | 0.142 | Sphingosine 1-phosphate receptor 2 antagonist | 0.135 0.064 CHEMBL1031 0.136 0.063 CHEMBL1030 0.115 0.111 CHEMBL1035 0.142 0.052 CHEMBL1032 | ||
| 0.163 | 0.074 | 0.179 | Neurotensin receptor agonist | 0.179 0.051 CHEMBL1031 0.143 0.121 CHEMBL1033 0.168 0.065 CHEMBL1030 0.152 0.098 CHEMBL1035 0.169 0.064 CHEMBL1032 | CHEMBL1031 | |
| 0.131 | 0.042 | 0.146 | Protein kinase (CK2) inhibitor | 0.119 0.049 CHEMBL1031 0.11 0.055 CHEMBL1033 0.124 0.046 CHEMBL1030 0.146 0.034 CHEMBL1035 0.113 0.053 CHEMBL1032 | CHEMBL1035 | |
| 0.101 | 0.013 | 0.101 | Phosphorylase inhibitor | 0.096 0.014 CHEMBL1031 0.073 0.019 CHEMBL1030 0.055 0.028 CHEMBL1035 0.071 0.02 CHEMBL1032 | ||
| 0.146 | 0.057 | 0.203 | Farnesoid X receptor antagonist | 0.183 0.028 CHEMBL1031 0.14 0.065 CHEMBL1033 0.186 0.027 CHEMBL1030 0.141 0.064 CHEMBL1035 0.203 0.021 CHEMBL1032 | CHEMBL1032 | |
| 0.118 | 0.03 | 0.118 | NADH dehydrogenase inhibitor | 0.1 0.044 CHEMBL1031 0.103 0.041 CHEMBL1030 0.096 0.048 CHEMBL1035 0.104 0.04 CHEMBL1032 | ||
| 0.166 | 0.079 | 0.199 | Phospholipase C inhibitor | 0.187 0.054 CHEMBL1031 0.195 0.047 CHEMBL1030 0.15 0.106 CHEMBL1035 0.199 0.044 CHEMBL1032 | CHEMBL1032 | |
| 0.089 | 0.005 | 0.089 | Carnitine palmitoyltransferase 1B inhibitor | 0.07 0.011 CHEMBL1031 0.064 0.014 CHEMBL1033 0.066 0.013 CHEMBL1030 0.069 0.011 CHEMBL1035 0.065 0.014 CHEMBL1032 | ||
| 0.088 | 0.004 | 0.088 | NMDA receptor glycine site antagonist | 0.061 0.005 CHEMBL1031 0.055 0.005 CHEMBL1030 0.048 0.006 CHEMBL1035 0.046 0.007 CHEMBL1032 | ||
| 0.123 | 0.039 | 0.165 | Creatine kinase inhibitor | 0.165 0.018 CHEMBL1031 0.148 0.025 CHEMBL1030 0.128 0.035 CHEMBL1035 0.149 0.024 CHEMBL1032 | CHEMBL1031 | |
| 0.093 | 0.009 | 0.093 | Thromboxane A2 antagonist | 0.079 0.015 CHEMBL1031 0.075 0.018 CHEMBL1030 0.082 0.014 CHEMBL1035 0.071 0.021 CHEMBL1032 | ||
| 0.103 | 0.02 | 0.118 | Leukotriene antagonist | 0.118 0.016 CHEMBL1031 0.07 0.04 CHEMBL1033 0.097 0.023 CHEMBL1030 0.09 0.026 CHEMBL1035 0.104 0.02 CHEMBL1032 | CHEMBL1031 | |
| 0.1 | 0.018 | 0.121 | Aldose reductase inhibitor | 0.118 0.014 CHEMBL1031 0.083 0.022 CHEMBL1033 0.118 0.014 CHEMBL1030 0.075 0.025 CHEMBL1035 0.121 0.014 CHEMBL1032 | CHEMBL1032 | |
| 0.145 | 0.063 | 0.145 | Pregnane X receptor agonist | 0.132 0.095 CHEMBL1031 0.126 0.113 CHEMBL1030 | ||
| 0.109 | 0.029 | 0.109 | Cell adhesion molecule inhibitor | 0.081 0.052 CHEMBL1031 0.075 0.06 CHEMBL1030 0.074 0.061 CHEMBL1032 | ||
| 0.177 | 0.098 | 0.188 | Insulin sensitizer | 0.188 0.086 CHEMBL1031 0.161 0.118 CHEMBL1030 0.144 0.141 CHEMBL1035 0.172 0.104 CHEMBL1032 | CHEMBL1031 | |
| 0.087 | 0.009 | 0.087 | DNA helicase inhibitor | 0.079 0.011 CHEMBL1031 0.073 0.015 CHEMBL1033 0.079 0.012 CHEMBL1030 0.075 0.013 CHEMBL1035 0.077 0.013 CHEMBL1032 | ||
| 0.089 | 0.012 | 0.089 | MDM2 inhibitor | 0.074 0.029 CHEMBL1031 0.072 0.033 CHEMBL1030 0.071 0.035 CHEMBL1035 0.07 0.038 CHEMBL1032 | ||
| 0.132 | 0.055 | 0.154 | Cholesterol synthesis inhibitor | 0.154 0.042 CHEMBL1031 0.103 0.083 CHEMBL1033 0.126 0.06 CHEMBL1030 0.115 0.07 CHEMBL1035 0.135 0.053 CHEMBL1032 | CHEMBL1031 | |
| 0.196 | 0.122 | 0.233 | Superoxide dismutase inhibitor | 0.233 0.086 CHEMBL1031 0.186 0.134 CHEMBL1033 0.21 0.107 CHEMBL1030 0.169 0.156 CHEMBL1035 0.221 0.096 CHEMBL1032 | CHEMBL1031 | |
| 0.1 | 0.027 | 0.108 | GABA aminotransferase inhibitor | 0.108 0.022 CHEMBL1031 0.096 0.03 CHEMBL1030 0.081 0.045 CHEMBL1035 0.093 0.033 CHEMBL1032 | CHEMBL1031 | |
| 0.136 | 0.064 | 0.159 | c-Src kinase inhibitor | 0.134 0.065 CHEMBL1031 0.127 0.07 CHEMBL1030 0.159 0.05 CHEMBL1035 0.125 0.071 CHEMBL1032 | CHEMBL1035 | |
| 0.183 | 0.111 | 0.192 | ErbB-1 antagonist | 0.185 0.108 CHEMBL1031 0.192 0.099 CHEMBL1033 0.183 0.111 CHEMBL1030 0.168 0.138 CHEMBL1035 0.169 0.135 CHEMBL1032 | CHEMBL1033 | |
| 0.171 | 0.1 | 0.171 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.168 0.103 CHEMBL1031 0.156 0.114 CHEMBL1030 0.159 0.112 CHEMBL1032 | ||
| 0.122 | 0.051 | 0.122 | Aminopeptidase B inhibitor | 0.089 0.074 CHEMBL1031 0.111 0.058 CHEMBL1030 0.09 0.073 CHEMBL1032 | ||
| 0.107 | 0.037 | 0.107 | Platelet growth factor antagonist | 0.093 0.045 CHEMBL1031 0.09 0.048 CHEMBL1033 0.083 0.054 CHEMBL1030 0.083 0.054 CHEMBL1032 | ||
| 0.219 | 0.149 | 0.383 | Angiogenesis inhibitor | 0.219 0.149 CHEMBL1031 0.369 0.063 CHEMBL1033 0.22 0.148 CHEMBL1030 0.383 0.059 CHEMBL1035 0.239 0.131 CHEMBL1032 | CHEMBL1035 | |
| 0.086 | 0.017 | 0.096 | NMDA 2A receptor antagonist | 0.094 0.015 CHEMBL1031 0.096 0.014 CHEMBL1030 0.062 0.028 CHEMBL1035 0.078 0.021 CHEMBL1032 | CHEMBL1030 | |
| 0.209 | 0.141 | 0.345 | 12-Lipoxygenase inhibitor | 0.313 0.073 CHEMBL1031 0.345 0.059 CHEMBL1033 0.272 0.097 CHEMBL1030 0.268 0.099 CHEMBL1035 0.294 0.083 CHEMBL1032 | CHEMBL1033 | |
| 0.073 | 0.005 | 0.073 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.033 0.017 CHEMBL1031 0.034 0.016 CHEMBL1030 0.025 0.024 CHEMBL1035 0.032 0.017 CHEMBL1032 | ||
| 0.119 | 0.051 | 0.177 | 5-Lipoxygenase inhibitor | 0.177 0.03 CHEMBL1031 0.137 0.043 CHEMBL1033 0.154 0.036 CHEMBL1030 0.114 0.053 CHEMBL1035 0.169 0.032 CHEMBL1032 | CHEMBL1031 | |
| 0.07 | 0.003 | 0.07 | Elastase 3B inhibitor | 0.06 0.003 CHEMBL1031 0.052 0.004 CHEMBL1033 0.061 0.003 CHEMBL1030 0.06 0.004 CHEMBL1035 0.06 0.004 CHEMBL1032 | ||
| 0.07 | 0.003 | 0.07 | Elastase 3A inhibitor | 0.06 0.003 CHEMBL1031 0.052 0.004 CHEMBL1033 0.061 0.003 CHEMBL1030 0.06 0.004 CHEMBL1035 0.06 0.004 CHEMBL1032 | ||
| 0.07 | 0.003 | 0.07 | Elastase 2B inhibitor | 0.06 0.003 CHEMBL1031 0.052 0.004 CHEMBL1033 0.061 0.003 CHEMBL1030 0.06 0.004 CHEMBL1035 0.06 0.004 CHEMBL1032 | ||
| 0.115 | 0.048 | 0.115 | Gastric antisecretory | 0.108 0.056 CHEMBL1031 0.09 0.078 CHEMBL1030 0.091 0.078 CHEMBL1032 | ||
| 0.231 | 0.165 | 0.253 | Immunosuppressant | 0.23 0.166 CHEMBL1031 0.229 0.167 CHEMBL1033 0.235 0.161 CHEMBL1030 0.253 0.145 CHEMBL1035 0.231 0.165 CHEMBL1032 | CHEMBL1035 | |
| 0.152 | 0.086 | 0.153 | Interleukin 6 antagonist | 0.153 0.084 CHEMBL1031 0.139 0.107 CHEMBL1030 0.135 0.116 CHEMBL1032 | CHEMBL1031 | |
| 0.075 | 0.01 | 0.076 | Leukotriene C antagonist | 0.076 0.009 CHEMBL1031 0.054 0.046 CHEMBL1033 0.071 0.013 CHEMBL1030 0.07 0.014 CHEMBL1035 0.072 0.012 CHEMBL1032 | CHEMBL1031 | |
| 0.085 | 0.022 | 0.105 | Purinergic P2X1 antagonist | 0.084 0.023 CHEMBL1031 0.059 0.044 CHEMBL1033 0.105 0.015 CHEMBL1030 0.078 0.026 CHEMBL1035 0.097 0.017 CHEMBL1032 | CHEMBL1030 | |
| 0.088 | 0.024 | 0.088 | Peroxisome proliferator-activated receptor gamma antagonist | 0.084 0.028 CHEMBL1031 0.075 0.043 CHEMBL1033 0.082 0.031 CHEMBL1030 0.078 0.036 CHEMBL1035 0.087 0.026 CHEMBL1032 | ||
| 0.17 | 0.108 | 0.219 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.219 0.059 CHEMBL1031 0.185 0.086 CHEMBL1033 0.188 0.084 CHEMBL1030 0.192 0.079 CHEMBL1035 0.207 0.067 CHEMBL1032 | CHEMBL1031 | |
| 0.073 | 0.01 | 0.073 | Dihydroorotase inhibitor | 0.05 0.024 CHEMBL1031 0.047 0.028 CHEMBL1030 0.045 0.03 CHEMBL1035 0.044 0.031 CHEMBL1032 | ||
| 0.076 | 0.014 | 0.076 | Sphingosine 1-phosphate receptor 5 agonist | 0.062 0.023 CHEMBL1031 0.063 0.022 CHEMBL1030 0.057 0.03 CHEMBL1035 0.063 0.022 CHEMBL1032 | ||
| 0.114 | 0.052 | 0.14 | Carbonic anhydrase XV inhibitor | 0.14 0.035 CHEMBL1031 0.088 0.086 CHEMBL1033 0.125 0.043 CHEMBL1030 0.1 0.067 CHEMBL1035 0.132 0.038 CHEMBL1032 | CHEMBL1031 | |
| 0.069 | 0.008 | 0.069 | AMPA 4 receptor antagonist | 0.049 0.016 CHEMBL1031 0.054 0.013 CHEMBL1030 0.041 0.025 CHEMBL1035 0.045 0.019 CHEMBL1032 | ||
| 0.19 | 0.13 | 0.19 | 5 Hydroxytryptamine release stimulant | 0.177 0.144 CHEMBL1031 0.173 0.149 CHEMBL1030 | ||
| 0.092 | 0.032 | 0.181 | CDC25A inhibitor | 0.101 0.027 CHEMBL1031 0.141 0.014 CHEMBL1033 0.093 0.032 CHEMBL1030 0.181 0.009 CHEMBL1035 0.094 0.031 CHEMBL1032 | CHEMBL1035 | |
| 0.082 | 0.022 | 0.082 | Glutamate (mGluR6) antagonist | 0.063 0.058 CHEMBL1031 0.064 0.053 CHEMBL1030 | ||
| 0.176 | 0.117 | 0.277 | Antiamyloidogenic | 0.263 0.065 CHEMBL1031 0.221 0.086 CHEMBL1033 0.236 0.077 CHEMBL1030 0.16 0.134 CHEMBL1035 0.277 0.06 CHEMBL1032 | CHEMBL1032 | |
| 0.107 | 0.048 | 0.11 | MAP kinase kinase 1 inhibitor | 0.088 0.073 CHEMBL1031 0.108 0.047 CHEMBL1030 0.096 0.062 CHEMBL1035 0.11 0.045 CHEMBL1032 | CHEMBL1032 | |
| 0.173 | 0.115 | 0.179 | Hypolipemic | 0.172 0.117 CHEMBL1031 0.171 0.117 CHEMBL1030 0.179 0.11 CHEMBL1032 | CHEMBL1032 | |
| 0.07 | 0.012 | 0.07 | Fructose-1,6-bisphosphatase inhibitor | 0.058 0.018 CHEMBL1031 0.056 0.02 CHEMBL1030 0.042 0.036 CHEMBL1035 0.056 0.02 CHEMBL1032 | ||
| 0.089 | 0.032 | 0.129 | Phenylalanine 4-hydroxylase inhibitor | 0.129 0.016 CHEMBL1031 0.104 0.024 CHEMBL1030 0.084 0.034 CHEMBL1035 0.118 0.019 CHEMBL1032 | CHEMBL1031 | |
| 0.095 | 0.038 | 0.1 | Porphobilinogen synthase inhibitor | 0.086 0.043 CHEMBL1031 0.1 0.036 CHEMBL1030 0.08 0.047 CHEMBL1035 0.093 0.039 CHEMBL1032 | CHEMBL1030 | |
| 0.081 | 0.025 | 0.081 | Biliverdin reductase inhibitor | 0.052 0.051 CHEMBL1030 | ||
| 0.065 | 0.01 | 0.076 | Liver X receptor alpha agonist | 0.076 0.007 CHEMBL1031 0.062 0.012 CHEMBL1030 0.049 0.02 CHEMBL1035 0.065 0.01 CHEMBL1032 | CHEMBL1031 | |
| 0.081 | 0.026 | 0.081 | Prostaglandin EP2 antagonist | 0.07 0.033 CHEMBL1031 0.071 0.032 CHEMBL1030 0.055 0.046 CHEMBL1035 0.071 0.032 CHEMBL1032 | ||
| 0.129 | 0.075 | 0.213 | Amylase inhibitor | 0.213 0.04 CHEMBL1031 0.155 0.061 CHEMBL1030 0.109 0.089 CHEMBL1035 0.179 0.052 CHEMBL1032 | CHEMBL1031 | |
| 0.079 | 0.026 | 0.082 | NMDA 2C receptor antagonist | 0.082 0.024 CHEMBL1031 0.079 0.025 CHEMBL1030 0.059 0.047 CHEMBL1035 0.069 0.034 CHEMBL1032 | CHEMBL1031 | |
| 0.081 | 0.027 | 0.162 | CDC25B inhibitor | 0.088 0.022 CHEMBL1031 0.126 0.01 CHEMBL1033 0.082 0.026 CHEMBL1030 0.162 0.005 CHEMBL1035 0.082 0.026 CHEMBL1032 | CHEMBL1035 | |
| 0.066 | 0.015 | 0.066 | Heparanase inhibitor | 0.059 0.024 CHEMBL1031 0.051 0.042 CHEMBL1033 0.058 0.025 CHEMBL1030 0.055 0.032 CHEMBL1035 0.056 0.03 CHEMBL1032 | ||
| 0.06 | 0.009 | 0.06 | p53 inhibitor | 0.044 0.018 CHEMBL1031 0.038 0.022 CHEMBL1030 0.038 0.022 CHEMBL1035 0.035 0.026 CHEMBL1032 | ||
| 0.116 | 0.065 | 0.116 | Caspase 3 inhibitor | 0.107 0.08 CHEMBL1031 0.108 0.079 CHEMBL1030 0.116 0.066 CHEMBL1035 0.1 0.092 CHEMBL1032 | ||
| 0.069 | 0.019 | 0.069 | Aconitate hydratase inhibitor | 0.049 0.039 CHEMBL1030 | ||
| 0.129 | 0.078 | 0.129 | Protein-tyrosine kinase Lyn inhibitor | 0.117 0.088 CHEMBL1033 0.102 0.1 CHEMBL1030 | ||
| 0.054 | 0.005 | 0.054 | Kainate receptor 1 antagonist | 0.028 0.011 CHEMBL1031 0.034 0.009 CHEMBL1030 0.019 0.017 CHEMBL1035 0.029 0.011 CHEMBL1032 | ||
| 0.087 | 0.038 | 0.087 | Glutamate dehydrogenase inhibitor | 0.074 0.052 CHEMBL1030 0.066 0.062 CHEMBL1032 | ||
| 0.057 | 0.008 | 0.057 | Kainate receptor agonist | 0.045 0.021 CHEMBL1031 0.046 0.019 CHEMBL1030 0.044 0.023 CHEMBL1035 0.044 0.022 CHEMBL1032 | ||
| 0.105 | 0.057 | 0.112 | Folate antagonist | 0.093 0.079 CHEMBL1031 0.095 0.076 CHEMBL1033 0.112 0.047 CHEMBL1030 0.112 0.046 CHEMBL1032 | CHEMBL1032 | |
| 0.17 | 0.126 | 0.17 | Platelet antagonist | 0.148 0.147 CHEMBL1035 | ||
| 0.109 | 0.065 | 0.12 | Mucolytic | 0.118 0.056 CHEMBL1031 0.114 0.061 CHEMBL1033 0.115 0.06 CHEMBL1030 0.094 0.087 CHEMBL1035 0.12 0.054 CHEMBL1032 | CHEMBL1032 | |
| 0.086 | 0.042 | 0.117 | Keratolytic | 0.115 0.023 CHEMBL1031 0.082 0.046 CHEMBL1033 0.11 0.025 CHEMBL1030 0.082 0.046 CHEMBL1035 0.117 0.022 CHEMBL1032 | CHEMBL1032 | |
| 0.137 | 0.094 | 0.137 | GABA C receptor rho-2 antagonist | 0.136 0.095 CHEMBL1031 0.127 0.111 CHEMBL1030 | ||
| 0.056 | 0.013 | 0.056 | Kainate receptor 2 antagonist | |||
| 0.082 | 0.04 | 0.082 | Aminopeptidase I inhibitor | 0.074 0.049 CHEMBL1030 | ||
| 0.052 | 0.009 | 0.06 | Peroxisome proliferator-activated receptor delta antagonist | 0.045 0.012 CHEMBL1031 0.036 0.019 CHEMBL1033 0.051 0.009 CHEMBL1030 0.038 0.017 CHEMBL1035 0.06 0.008 CHEMBL1032 | CHEMBL1032 | |
| 0.072 | 0.03 | 0.081 | Prostaglandin F2 alpha antagonist | 0.068 0.035 CHEMBL1031 0.08 0.023 CHEMBL1030 0.057 0.051 CHEMBL1035 0.081 0.022 CHEMBL1032 | CHEMBL1032 | |
| 0.048 | 0.007 | 0.048 | Kynurenine 3 monooxygenase inhibitor | 0.024 0.022 CHEMBL1031 0.026 0.019 CHEMBL1030 | ||
| 0.065 | 0.024 | 0.065 | Dihydroorotate dehydrogenase inhibitor | 0.054 0.033 CHEMBL1031 0.05 0.037 CHEMBL1030 | ||
| 0.147 | 0.107 | 0.203 | DNA methyltransferase I inhibitor | 0.185 0.077 CHEMBL1031 0.172 0.085 CHEMBL1033 0.183 0.078 CHEMBL1030 0.203 0.067 CHEMBL1032 | CHEMBL1032 | |
| 0.074 | 0.035 | 0.074 | Potassium channel (ATP-sensitive) blocker | 0.068 0.044 CHEMBL1031 0.07 0.041 CHEMBL1030 0.066 0.049 CHEMBL1032 | ||
| 0.085 | 0.048 | 0.085 | T cell inhibitor | 0.085 0.05 CHEMBL1035 | ||
| 0.089 | 0.052 | 0.089 | Hematopoietic | 0.082 0.067 CHEMBL1031 0.082 0.067 CHEMBL1030 | ||
| 0.117 | 0.08 | 0.117 | M17 leucyl aminopeptidase inhibitor | 0.113 0.084 CHEMBL1031 0.112 0.086 CHEMBL1030 0.115 0.082 CHEMBL1032 | ||
| 0.048 | 0.012 | 0.049 | Leukotriene C4 antagonist | 0.049 0.011 CHEMBL1031 0.044 0.016 CHEMBL1030 0.044 0.016 CHEMBL1035 0.045 0.015 CHEMBL1032 | CHEMBL1031 | |
| 0.071 | 0.034 | 0.071 | Carbamoyl phosphate synthetase inhibitor | 0.055 0.048 CHEMBL1030 0.055 0.048 CHEMBL1032 | ||
| 0.043 | 0.007 | 0.05 | CXC chemokine 2 receptor antagonist | 0.041 0.008 CHEMBL1031 0.05 0.005 CHEMBL1030 0.033 0.011 CHEMBL1035 0.038 0.009 CHEMBL1032 | CHEMBL1030 | |
| 0.046 | 0.01 | 0.046 | AMPA 3 receptor antagonist | 0.029 0.021 CHEMBL1031 0.03 0.021 CHEMBL1030 | ||
| 0.2 | 0.164 | 0.2 | Immunomodulator | 0.186 0.18 CHEMBL1030 | ||
| 0.046 | 0.011 | 0.046 | Carnitine palmitoyltransferase inhibitor | 0.033 0.025 CHEMBL1031 | ||
| 0.048 | 0.013 | 0.048 | Glutamate (mGluR8) agonist | 0.039 0.023 CHEMBL1031 0.04 0.022 CHEMBL1030 0.036 0.029 CHEMBL1035 0.04 0.022 CHEMBL1032 | ||
| 0.045 | 0.011 | 0.045 | Carnitine palmitoyltransferase 1 inhibitor | 0.033 0.025 CHEMBL1031 | ||
| 0.158 | 0.124 | 0.158 | Growth factor agonist | 0.154 0.133 CHEMBL1031 0.155 0.131 CHEMBL1030 0.152 0.137 CHEMBL1032 | ||
| 0.055 | 0.021 | 0.055 | Carbonic anhydrase IV inhibitor | 0.042 0.031 CHEMBL1031 0.043 0.03 CHEMBL1030 0.039 0.034 CHEMBL1032 | ||
| 0.061 | 0.028 | 0.061 | Dihydroorotate oxidase inhibitor | 0.056 0.037 CHEMBL1031 0.054 0.041 CHEMBL1030 0.053 0.043 CHEMBL1032 | ||
| 0.037 | 0.005 | 0.037 | Complement factor 1r inhibitor | 0.032 0.009 CHEMBL1031 0.028 0.013 CHEMBL1033 0.032 0.009 CHEMBL1030 0.032 0.009 CHEMBL1035 0.03 0.01 CHEMBL1032 | ||
| 0.046 | 0.014 | 0.046 | Integrin alpha2 antagonist | |||
| 0.084 | 0.052 | 0.131 | Carbonic anhydrase VI inhibitor | 0.131 0.025 CHEMBL1031 0.104 0.037 CHEMBL1030 0.076 0.063 CHEMBL1035 0.119 0.03 CHEMBL1032 | CHEMBL1031 | |
| 0.158 | 0.127 | 0.208 | Neurotrophic factor enhancer | 0.208 0.069 CHEMBL1031 0.175 0.104 CHEMBL1030 0.15 0.137 CHEMBL1035 0.186 0.091 CHEMBL1032 | CHEMBL1031 | |
| 0.044 | 0.013 | 0.044 | AMPA 1 receptor antagonist | 0.028 0.021 CHEMBL1031 0.034 0.018 CHEMBL1030 | ||
| 0.042 | 0.012 | 0.047 | Liver X receptor beta antagonist | 0.047 0.009 CHEMBL1031 0.041 0.012 CHEMBL1030 0.037 0.014 CHEMBL1035 0.042 0.012 CHEMBL1032 | CHEMBL1031 | |
| 0.118 | 0.088 | 0.173 | Interleukin 4 antagonist | 0.163 0.04 CHEMBL1031 0.127 0.075 CHEMBL1033 0.166 0.037 CHEMBL1030 0.149 0.051 CHEMBL1035 0.173 0.033 CHEMBL1032 | CHEMBL1032 | |
| 0.043 | 0.013 | 0.043 | Liver X receptor beta agonist | 0.042 0.014 CHEMBL1031 0.03 0.029 CHEMBL1033 0.043 0.014 CHEMBL1030 0.034 0.022 CHEMBL1035 0.042 0.014 CHEMBL1032 | ||
| 0.051 | 0.023 | 0.051 | Glutamate (mGluR group III) agonist | 0.038 0.037 CHEMBL1031 | ||
| 0.096 | 0.067 | 0.146 | Carbonic anhydrase III inhibitor | 0.146 0.03 CHEMBL1031 0.117 0.047 CHEMBL1030 0.093 0.071 CHEMBL1035 0.127 0.04 CHEMBL1032 | CHEMBL1031 | |
| 0.047 | 0.018 | 0.048 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.047 0.018 CHEMBL1031 0.048 0.017 CHEMBL1030 0.044 0.023 CHEMBL1035 0.048 0.017 CHEMBL1032 | CHEMBL1032 | |
| 0.148 | 0.119 | 0.191 | DNA methylase inhibitor | 0.18 0.093 CHEMBL1031 0.162 0.107 CHEMBL1033 0.178 0.094 CHEMBL1030 0.191 0.085 CHEMBL1032 | CHEMBL1032 | |
| 0.039 | 0.011 | 0.039 | 11-Beta-hydroxysteroid dehydrogenase 2 inhibitor | 0.026 0.021 CHEMBL1031 0.031 0.016 CHEMBL1030 0.025 0.022 CHEMBL1032 | ||
| 0.04 | 0.013 | 0.053 | ATP citrate lysase inhibitor | 0.053 0.007 CHEMBL1031 0.051 0.007 CHEMBL1030 0.047 0.009 CHEMBL1035 0.053 0.007 CHEMBL1032 | CHEMBL1032 | |
| 0.094 | 0.067 | 0.114 | UDP-glucose 4-epimerase inhibitor | 0.114 0.048 CHEMBL1030 0.105 0.055 CHEMBL1032 | CHEMBL1030 | |
| 0.061 | 0.035 | 0.085 | Alcohol oxidase inhibitor | 0.077 0.026 CHEMBL1031 0.085 0.022 CHEMBL1030 0.05 0.045 CHEMBL1035 0.084 0.023 CHEMBL1032 | CHEMBL1030 | |
| 0.148 | 0.123 | 0.148 | MAP kinase kinase 2 inhibitor | |||
| 0.071 | 0.045 | 0.087 | Carbonic anhydrase VA inhibitor | 0.086 0.032 CHEMBL1031 0.081 0.036 CHEMBL1030 0.087 0.032 CHEMBL1032 | CHEMBL1032 | |
| 0.122 | 0.097 | 0.122 | Mannose-6-phosphate isomerase inhibitor | 0.117 0.105 CHEMBL1031 0.122 0.098 CHEMBL1030 0.121 0.098 CHEMBL1032 | ||
| 0.036 | 0.011 | 0.04 | Liver X receptor alpha antagonist | 0.04 0.009 CHEMBL1031 0.034 0.014 CHEMBL1033 0.037 0.011 CHEMBL1030 0.035 0.013 CHEMBL1035 0.039 0.01 CHEMBL1032 | CHEMBL1031 | |
| 0.091 | 0.066 | 0.091 | Potassium channel (Voltage-sensitive) activator | |||
| 0.082 | 0.058 | 0.094 | Glutathione S-transferase inhibitor | 0.083 0.057 CHEMBL1031 0.09 0.048 CHEMBL1030 0.094 0.043 CHEMBL1032 | CHEMBL1032 | |
| 0.04 | 0.015 | 0.04 | Tryptophan 5 hydroxylase inhibitor | |||
| 0.051 | 0.027 | 0.051 | Integrin antagonist | |||
| 0.063 | 0.039 | 0.063 | Alpha 2 adrenoreceptor agonist | 0.061 0.042 CHEMBL1031 0.056 0.048 CHEMBL1030 | ||
| 0.061 | 0.036 | 0.061 | Botulinum neurotoxin type A inhibitor | 0.057 0.043 CHEMBL1031 | ||
| 0.033 | 0.009 | 0.033 | Integrin alpha2beta1 antagonist | |||
| 0.043 | 0.019 | 0.043 | Potassium channel Kv1.1 blocker | |||
| 0.077 | 0.053 | 0.077 | Sphingosine 1-phosphate receptor antagonist | 0.071 0.068 CHEMBL1031 0.074 0.06 CHEMBL1035 | ||
| 0.068 | 0.045 | 0.068 | Phosphodiesterase 4B inhibitor | |||
| 0.039 | 0.017 | 0.039 | Glutamate (mGluR4) agonist | 0.031 0.029 CHEMBL1031 | ||
| 0.069 | 0.048 | 0.069 | Phosphofructokinase-1 inhibitor | 0.061 0.056 CHEMBL1030 0.061 0.055 CHEMBL1032 | ||
| 0.032 | 0.011 | 0.071 | Thyroid hormone agonist | 0.052 0.004 CHEMBL1031 0.025 0.02 CHEMBL1033 0.053 0.004 CHEMBL1030 0.032 0.01 CHEMBL1035 0.071 0.003 CHEMBL1032 | CHEMBL1032 | |
| 0.063 | 0.042 | 0.063 | Caspase 9 inhibitor | 0.057 0.055 CHEMBL1031 | ||
| 0.058 | 0.038 | 0.058 | Argininosuccinate synthase inhibitor | |||
| 0.034 | 0.015 | 0.034 | Integrin alpha4 antagonist | 0.024 0.019 CHEMBL1035 | ||
| 0.087 | 0.068 | 0.087 | Glutamate release inhibitor | |||
| 0.04 | 0.021 | 0.04 | Glutamate (mGluR3) antagonist | |||
| 0.093 | 0.075 | 0.109 | Urease inhibitor | 0.109 0.056 CHEMBL1031 0.107 0.059 CHEMBL1030 0.092 0.076 CHEMBL1035 0.108 0.058 CHEMBL1032 | CHEMBL1031 | |
| 0.109 | 0.091 | 0.109 | Cathepsin H inhibitor | |||
| 0.023 | 0.005 | 0.033 | Thyroid hormone alpha agonist | 0.025 0.005 CHEMBL1031 0.022 0.005 CHEMBL1033 0.03 0.004 CHEMBL1030 0.022 0.005 CHEMBL1035 0.033 0.004 CHEMBL1032 | CHEMBL1032 | |
| 0.069 | 0.052 | 0.091 | NMDA 2 receptor antagonist | 0.091 0.037 CHEMBL1031 0.086 0.04 CHEMBL1030 0.067 0.054 CHEMBL1032 | CHEMBL1031 | |
| 0.027 | 0.01 | 0.027 | Elastase 2A inhibitor | |||
| 0.027 | 0.01 | 0.027 | Elastase 2 inhibitor | |||
| 0.023 | 0.006 | 0.042 | Thyroid hormone alpha antagonist | 0.031 0.005 CHEMBL1031 0.016 0.01 CHEMBL1033 0.033 0.005 CHEMBL1030 0.021 0.007 CHEMBL1035 0.042 0.004 CHEMBL1032 | CHEMBL1032 | |
| 0.036 | 0.02 | 0.036 | Purinergic P2Y2 antagonist | 0.032 0.027 CHEMBL1031 0.031 0.027 CHEMBL1030 | ||
| 0.057 | 0.041 | 0.057 | Protein kinase C theta inhibitor | |||
| 0.051 | 0.035 | 0.051 | Lysophosphatidic acid 3 receptor antagonist | |||
| 0.034 | 0.018 | 0.037 | Liver X receptor antagonist | 0.037 0.016 CHEMBL1031 0.029 0.024 CHEMBL1033 0.034 0.018 CHEMBL1030 0.032 0.021 CHEMBL1035 0.035 0.017 CHEMBL1032 | CHEMBL1031 | |
| 0.178 | 0.163 | 0.178 | Neuropeptide Y2 antagonist | |||
| 0.054 | 0.039 | 0.076 | Maillard reaction inhibitor | 0.076 0.026 CHEMBL1031 0.068 0.03 CHEMBL1030 0.056 0.038 CHEMBL1035 0.071 0.029 CHEMBL1032 | CHEMBL1031 | |
| 0.048 | 0.033 | 0.048 | Glucose-6-phosphate isomerase inhibitor | |||
| 0.044 | 0.03 | 0.044 | Liver X receptor agonist | 0.043 0.031 CHEMBL1031 0.042 0.032 CHEMBL1030 0.043 0.03 CHEMBL1032 | ||
| 0.02 | 0.006 | 0.02 | Thromboxane A2 agonist | 0.014 0.013 CHEMBL1031 | ||
| 0.036 | 0.022 | 0.036 | 1-Alkyl-2-acetylglycerophosphocholine esterase inhibitor | 0.036 0.022 CHEMBL1031 0.031 0.03 CHEMBL1030 0.033 0.026 CHEMBL1035 0.033 0.026 CHEMBL1032 | ||
| 0.028 | 0.015 | 0.028 | Prostaglandin H2 antagonist | |||
| 0.063 | 0.05 | 0.08 | Carbonic anhydrase V inhibitor | 0.08 0.036 CHEMBL1031 0.074 0.04 CHEMBL1030 0.064 0.049 CHEMBL1035 0.08 0.035 CHEMBL1032 | CHEMBL1032 | |
| 0.022 | 0.009 | 0.022 | Integrin alpha4beta1 antagonist | 0.014 0.013 CHEMBL1031 0.016 0.011 CHEMBL1035 | ||
| 0.034 | 0.021 | 0.034 | Protein kinase (CK2) beta inhibitor | 0.032 0.027 CHEMBL1031 0.034 0.021 CHEMBL1030 0.032 0.026 CHEMBL1032 | ||
| 0.088 | 0.075 | 0.088 | Interleukin 1 beta converting enzyme inhibitor | 0.085 0.08 CHEMBL1030 | ||
| 0.113 | 0.101 | 0.145 | Protein kinase stimulant | 0.145 0.072 CHEMBL1031 0.119 0.093 CHEMBL1033 0.122 0.09 CHEMBL1030 0.124 0.088 CHEMBL1035 0.138 0.077 CHEMBL1032 | CHEMBL1031 | |
| 0.114 | 0.102 | 0.129 | Vanilloid 1 agonist | 0.129 0.068 CHEMBL1031 0.124 0.078 CHEMBL1033 0.12 0.089 CHEMBL1030 0.124 0.078 CHEMBL1035 0.127 0.073 CHEMBL1032 | CHEMBL1031 | |
| 0.036 | 0.024 | 0.036 | Glutamate (mGluR8) antagonist | |||
| 0.032 | 0.02 | 0.034 | Prostaglandin agonist | 0.03 0.022 CHEMBL1031 0.033 0.019 CHEMBL1030 0.029 0.024 CHEMBL1035 0.034 0.017 CHEMBL1032 | CHEMBL1032 | |
| 0.212 | 0.2 | 0.335 | 15-Lipoxygenase inhibitor | 0.335 0.108 CHEMBL1031 0.323 0.116 CHEMBL1033 0.274 0.147 CHEMBL1030 0.232 0.18 CHEMBL1035 0.306 0.128 CHEMBL1032 | CHEMBL1031 | |
| 0.06 | 0.05 | 0.069 | Beta 2 adrenoreceptor agonist | 0.069 0.021 CHEMBL1031 0.066 0.028 CHEMBL1030 0.068 0.023 CHEMBL1035 0.068 0.023 CHEMBL1032 | CHEMBL1031 | |
| 0.02 | 0.01 | 0.02 | Alpha 2b adrenoreceptor agonist | |||
| 0.029 | 0.019 | 0.029 | Carnitine palmitoyltransferase 1A inhibitor | |||
| 0.067 | 0.057 | 0.067 | Cathepsin G inhibitor | |||
| 0.128 | 0.119 | 0.207 | Dual specificity phosphatase 3 inhibitor | 0.163 0.086 CHEMBL1031 0.204 0.059 CHEMBL1033 0.165 0.084 CHEMBL1030 0.207 0.057 CHEMBL1035 0.168 0.082 CHEMBL1032 | CHEMBL1035 | |
| 0.042 | 0.033 | 0.042 | Glutamate (mGluR4) antagonist | |||
| 0.027 | 0.018 | 0.027 | VLA-4 antagonist | |||
| 0.033 | 0.025 | 0.033 | Fumarate hydratase inhibitor | |||
| 0.024 | 0.015 | 0.026 | Prostaglandin E2 agonist | 0.022 0.018 CHEMBL1031 0.024 0.015 CHEMBL1030 0.022 0.018 CHEMBL1035 0.026 0.014 CHEMBL1032 | CHEMBL1032 | |
| 0.044 | 0.036 | 0.044 | Thymidylate synthase inhibitor | |||
| 0.038 | 0.031 | 0.038 | VCAM-1 antagonist | |||
| 0.038 | 0.031 | 0.038 | VCAM antagonist | |||
| 0.032 | 0.024 | 0.032 | Prostacyclin antagonist | |||
| 0.051 | 0.044 | 0.051 | Thromboxane synthase inhibitor | |||
| 0.063 | 0.057 | 0.063 | ZAP-70 protein tyrosine kinase inhibitor | 0.063 0.058 CHEMBL1033 | ||
| 0.079 | 0.072 | 0.105 | Estrogen-related receptor beta agonist | 0.095 0.031 CHEMBL1031 0.083 0.058 CHEMBL1033 0.103 0.022 CHEMBL1030 0.081 0.063 CHEMBL1035 0.105 0.019 CHEMBL1032 | CHEMBL1032 | |
| 0.018 | 0.012 | 0.018 | Complement factor D inhibitor | |||
| 0.046 | 0.04 | 0.046 | Prostaglandin E2 antagonist | |||
| 0.073 | 0.068 | 0.073 | Glycine receptor antagonist | |||
| 0.067 | 0.062 | 0.1 | Carbonic anhydrase XIII inhibitor | 0.1 0.038 CHEMBL1031 0.081 0.049 CHEMBL1030 0.092 0.042 CHEMBL1032 | CHEMBL1031 | |
| 0.023 | 0.018 | 0.023 | Fructose-1,6-bisphosphatase 1 inhibitor | |||
| 0.015 | 0.011 | 0.015 | CC chemokine 10 receptor antagonist | |||
| 0.031 | 0.027 | 0.031 | Free fatty acid receptor 1 antagonist | |||
| 0.085 | 0.081 | 0.085 | MAP kinase 8 inhibitor | |||
| 0.043 | 0.04 | 0.05 | Beta adrenoreceptor agonist | 0.05 0.018 CHEMBL1031 0.048 0.023 CHEMBL1030 0.048 0.023 CHEMBL1035 0.049 0.02 CHEMBL1032 | CHEMBL1031 | |
| 0.036 | 0.033 | 0.036 | Integrin alpha1beta1 antagonist | |||
| 0.024 | 0.021 | 0.024 | Prostaglandin EP4 antagonist | |||
| 0.075 | 0.072 | 0.075 | Histamine N-methyltransferase inhibitor | |||
| 0.142 | 0.139 | 0.142 | Anticonvulsant | |||
| 0.027 | 0.024 | 0.027 | AMPA 2 receptor antagonist | |||
| 0.03 | 0.027 | 0.03 | Peroxisome proliferator-activated receptor delta agonist | 0.03 0.028 CHEMBL1032 | ||
| 0.02 | 0.017 | 0.024 | Prostaglandin EP2 agonist | 0.021 0.017 CHEMBL1030 0.024 0.015 CHEMBL1032 | CHEMBL1032 | |
| 0.031 | 0.029 | 0.031 | Retinoid X alpha receptor agonist | |||
| 0.029 | 0.027 | 0.029 | Sirtuin 2 inhibitor | |||
| 0.141 | 0.139 | 0.159 | EphB2 antagonist | 0.159 0.12 CHEMBL1030 0.156 0.124 CHEMBL1032 | CHEMBL1030 | |
| 0.042 | 0.04 | 0.042 | AMPA receptor antagonist | |||
| 0.016 | 0.014 | 0.017 | Alpha 2a adrenoreceptor agonist | 0.017 0.013 CHEMBL1031 | CHEMBL1031 | |
| 0.118 | 0.117 | 0.16 | Protein-tyrosine phosphatase inhibitor | 0.146 0.082 CHEMBL1031 0.138 0.092 CHEMBL1030 0.16 0.069 CHEMBL1035 0.143 0.086 CHEMBL1032 | CHEMBL1035 | |
| 0.041 | 0.041 | 0.042 | Peroxisome proliferator-activated receptor alpha agonist | 0.042 0.039 CHEMBL1032 | CHEMBL1032 | |
| 0.007 | 0.008 | 0.029 | Thyroid hormone beta agonist | 0.015 0.004 CHEMBL1031 0.016 0.004 CHEMBL1030 0.029 0.003 CHEMBL1032 | CHEMBL1032 | |
| 0.013 | 0.014 | 0.014 | Integrin beta6 antagonist | 0.014 0.01 CHEMBL1031 0.014 0.011 CHEMBL1030 0.014 0.01 CHEMBL1032 | CHEMBL1032 | |
| 0.121 | 0.123 | 0.138 | Adenylate cyclase stimulant | 0.138 0.084 CHEMBL1031 0.128 0.105 CHEMBL1030 0.137 0.087 CHEMBL1032 | CHEMBL1031 | |
| 0.085 | 0.088 | 0.102 | Anabolic | 0.097 0.067 CHEMBL1031 0.093 0.073 CHEMBL1030 0.102 0.06 CHEMBL1032 | CHEMBL1032 | |
| 0.091 | 0.095 | 0.101 | Multidrug resistance-associated protein 1 inhibitor | 0.101 0.076 CHEMBL1031 | CHEMBL1031 | |
| 0.161 | 0.165 | 0.182 | Peptidyltransferase inhibitor | 0.182 0.124 CHEMBL1031 0.175 0.138 CHEMBL1030 0.177 0.134 CHEMBL1032 | CHEMBL1031 | |
| 0.189 | 0.196 | 0.247 | Apoptosis antagonist | 0.247 0.13 CHEMBL1031 0.201 0.177 CHEMBL1033 0.202 0.177 CHEMBL1030 0.216 0.161 CHEMBL1035 0.218 0.159 CHEMBL1032 | CHEMBL1031 | |
| 0.068 | 0.075 | 0.074 | Phosphodiesterase IV inhibitor | 0.074 0.068 CHEMBL1031 | CHEMBL1031 | |
| 0.128 | 0.135 | 0.133 | Heat shock protein 70 antagonist | 0.133 0.104 CHEMBL1031 | CHEMBL1031 | |
| 0.031 | 0.04 | 0.036 | Urate transporter 1 inhibitor | 0.036 0.031 CHEMBL1030 | CHEMBL1030 | |
| 0.018 | 0.027 | 0.021 | Prostaglandin F2 alpha agonist | 0.021 0.018 CHEMBL1032 | CHEMBL1032 | |
| 0.082 | 0.092 | 0.107 | Interleukin 12 antagonist | 0.107 0.043 CHEMBL1031 0.098 0.057 CHEMBL1030 0.101 0.051 CHEMBL1032 | CHEMBL1031 | |
| 0.017 | 0.029 | 0.023 | Beta 1 adrenoreceptor agonist | 0.023 0.014 CHEMBL1031 | CHEMBL1031 | |
| 0.084 | 0.096 | 0.09 | EphA2 antagonist | 0.09 0.087 CHEMBL1033 | CHEMBL1033 | |
| 0.027 | 0.04 | 0.041 | Nicotinic acid receptor agonist | 0.041 0.02 CHEMBL1030 0.036 0.025 CHEMBL1032 | CHEMBL1030 | |
| 0.089 | 0.102 | 0.109 | Histone deacetylase class III inhibitor | 0.109 0.08 CHEMBL1031 | CHEMBL1031 | |
| 0.027 | 0.041 | 0.033 | Glutamate (mGluR3) agonist | 0.031 0.025 CHEMBL1030 0.033 0.02 CHEMBL1032 | CHEMBL1032 | |
| 0.09 | 0.105 | 0.177 | M18 aspartyl aminopeptidase inhibitor | 0.177 0.041 CHEMBL1031 0.124 0.067 CHEMBL1030 0.109 0.081 CHEMBL1035 0.153 0.05 CHEMBL1032 | CHEMBL1031 | |
| 0.074 | 0.091 | 0.111 | Alcohol dehydrogenase inhibitor | 0.086 0.07 CHEMBL1031 0.111 0.041 CHEMBL1030 0.109 0.043 CHEMBL1032 | CHEMBL1030 | |
| 0.084 | 0.102 | 0.104 | Toll-Like receptor 4 antagonist | 0.104 0.063 CHEMBL1031 0.094 0.08 CHEMBL1030 0.097 0.075 CHEMBL1032 | CHEMBL1031 | |
| 0.073 | 0.091 | 0.084 | Interleukin 5 antagonist | 0.079 0.075 CHEMBL1031 0.084 0.065 CHEMBL1030 0.08 0.073 CHEMBL1032 | CHEMBL1030 | |
| 0.03 | 0.048 | 0.05 | Dopamine D5 agonist | 0.05 0.017 CHEMBL1031 0.042 0.025 CHEMBL1030 0.05 0.018 CHEMBL1032 | CHEMBL1032 | |
| 0.082 | 0.103 | 0.111 | AMP-activated protein kinase stimulant | 0.097 0.074 CHEMBL1031 0.1 0.07 CHEMBL1030 0.111 0.057 CHEMBL1032 | CHEMBL1032 | |
| 0.011 | 0.033 | 0.017 | Nicotinic acid receptor 1 antagonist | 0.017 0.014 CHEMBL1030 | CHEMBL1030 | |
| 0.084 | 0.106 | 0.1 | Nav1.4 sodium channel blocker | 0.1 0.076 CHEMBL1031 0.098 0.079 CHEMBL1030 0.097 0.08 CHEMBL1032 | CHEMBL1031 | |
| 0.048 | 0.07 | 0.054 | Pregnane X receptor antagonist | 0.054 0.048 CHEMBL1030 | CHEMBL1030 | |
| 0.035 | 0.061 | 0.051 | Beta 2 adrenoreceptor antagonist | 0.051 0.035 CHEMBL1031 0.047 0.041 CHEMBL1030 0.051 0.035 CHEMBL1032 | CHEMBL1032 | |
| 0.027 | 0.054 | 0.035 | Dihydropteroate synthase inhibitor | 0.035 0.034 CHEMBL1030 | CHEMBL1030 | |
| 0.118 | 0.145 | 0.264 | Amyloid beta precursor protein antagonist | 0.147 0.105 CHEMBL1031 0.264 0.028 CHEMBL1033 0.132 0.124 CHEMBL1030 0.185 0.068 CHEMBL1035 0.14 0.113 CHEMBL1032 | CHEMBL1033 | |
| 0.087 | 0.115 | 0.107 | TRPA1 agonist | 0.107 0.075 CHEMBL1031 | CHEMBL1031 | |
| 0.086 | 0.114 | 0.111 | MAP kinase kinase inhibitor | 0.111 0.083 CHEMBL1030 0.108 0.086 CHEMBL1032 | CHEMBL1030 | |
| 0.043 | 0.072 | 0.056 | Androgen agonist | 0.056 0.047 CHEMBL1030 0.055 0.048 CHEMBL1032 | CHEMBL1030 | |
| 0.075 | 0.104 | 0.088 | Expectorant | 0.087 0.085 CHEMBL1031 0.088 0.083 CHEMBL1032 | CHEMBL1032 | |
| 0.046 | 0.079 | 0.058 | Adenine nucleotide translocase inhibitor | 0.054 0.044 CHEMBL1031 0.057 0.034 CHEMBL1030 0.058 0.032 CHEMBL1032 | CHEMBL1032 | |
| 0.115 | 0.149 | 0.199 | Dual specificity phosphatase inhibitor | 0.144 0.101 CHEMBL1031 0.192 0.059 CHEMBL1033 0.143 0.102 CHEMBL1030 0.199 0.055 CHEMBL1035 0.147 0.098 CHEMBL1032 | CHEMBL1035 | |
| 0.07 | 0.109 | 0.093 | DNA directed RNA polymerase inhibitor | 0.09 0.07 CHEMBL1030 0.093 0.065 CHEMBL1032 | CHEMBL1032 | |
| 0.049 | 0.087 | 0.066 | Phosphodiesterase 4D inhibitor | 0.066 0.059 CHEMBL1033 | CHEMBL1033 | |
| 0.116 | 0.156 | 0.14 | CF transmembrane conductance regulator agonist | 0.14 0.095 CHEMBL1031 0.132 0.113 CHEMBL1032 | CHEMBL1031 | |
| 0.039 | 0.083 | 0.059 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.059 0.04 CHEMBL1031 | CHEMBL1031 | |
| 0.089 | 0.133 | 0.127 | NADPH oxidase inhibitor | 0.127 0.074 CHEMBL1031 | CHEMBL1031 | |
| 0.049 | 0.095 | 0.078 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.078 0.053 CHEMBL1031 0.067 0.065 CHEMBL1030 0.069 0.062 CHEMBL1032 | CHEMBL1031 | |
| 0.055 | 0.102 | 0.096 | Macrophage migration inhibitory factor inhibitor | 0.096 0.037 CHEMBL1031 0.083 0.047 CHEMBL1030 0.073 0.061 CHEMBL1035 0.095 0.038 CHEMBL1032 | CHEMBL1031 | |
| 0.081 | 0.132 | 0.112 | Bone formation stimulant | 0.112 0.094 CHEMBL1031 0.105 0.1 CHEMBL1032 | CHEMBL1031 | |
| 0.043 | 0.098 | 0.064 | Beta adrenoreceptor antagonist | 0.059 0.057 CHEMBL1031 0.064 0.048 CHEMBL1032 | CHEMBL1032 | |
| 0.067 | 0.125 | 0.093 | Protein-tyrosine phosphatase 1B inhibitor | 0.092 0.087 CHEMBL1031 0.093 0.085 CHEMBL1035 | CHEMBL1035 | |
| 0.202 | 0.27 | 0.321 | Calcium channel L-type activator | 0.279 0.175 CHEMBL1031 0.321 0.14 CHEMBL1030 0.253 0.202 CHEMBL1032 | CHEMBL1030 | |
| 0.079 | 0.151 | 0.115 | Toll-Like receptor 2 antagonist | 0.115 0.083 CHEMBL1031 0.108 0.092 CHEMBL1032 | CHEMBL1031 | |
| 0.069 | 0.146 | 0.095 | Beta glucuronidase inhibitor | 0.095 0.078 CHEMBL1031 | CHEMBL1031 | |
| 0.102 | 0.18 | 0.137 | Melanin inhibitor | 0.137 0.102 CHEMBL1031 0.133 0.108 CHEMBL1032 | CHEMBL1031 | |
| 0.034 | 0.123 | 0.06 | HIV-1 integrase (3'-Processing) inhibitor | 0.06 0.047 CHEMBL1031 0.056 0.052 CHEMBL1035 0.058 0.05 CHEMBL1032 | CHEMBL1031 | |
| 0.078 | 0.193 | 0.147 | Mcl-1 antagonist | 0.124 0.12 CHEMBL1031 0.147 0.092 CHEMBL1033 0.131 0.111 CHEMBL1035 | CHEMBL1033 | |
| 0.039 | 0.165 | 0.087 | Monophenol monooxygenase inhibitor | 0.087 0.086 CHEMBL1031 | CHEMBL1031 | |
| 0.061 | 0.195 | 0.155 | Lipid peroxidase inhibitor | 0.155 0.065 CHEMBL1031 0.132 0.082 CHEMBL1033 0.121 0.093 CHEMBL1030 0.148 0.07 CHEMBL1032 | CHEMBL1031 | |
| 0.075 | 0.218 | 0.141 | Pyruvate kinase inhibitor | 0.141 0.124 CHEMBL1033 | CHEMBL1033 | |
| 0.056 | 0.201 | 0.092 | Vanilloid agonist | 0.092 0.044 CHEMBL1033 | CHEMBL1033 | |
| 0.107 | 0.264 | 0.171 | Hypoglycemic | 0.167 0.152 CHEMBL1031 0.171 0.146 CHEMBL1032 | CHEMBL1032 | |
| 0.072 | 0.256 | 0.138 | Heat shock protein 90 alpha antagonist | 0.138 0.1 CHEMBL1035 | CHEMBL1035 | |
| 0.057 | 0.25 | 0.162 | Amyloid beta aggregation inhibitor | 0.162 0.1 CHEMBL1031 0.148 0.109 CHEMBL1032 | CHEMBL1031 | |
| 0.112 | 0.312 | 0.24 | Alpha-glucosidase inhibitor | 0.24 0.193 CHEMBL1033 | CHEMBL1033 | |
| 0.003 | 0.227 | 0.034 | Estrogen receptor alpha agonist | 0.034 0.024 CHEMBL1032 | CHEMBL1032 | |
| 0.013 | 0.242 | 0.077 | Fibroblast growth factor 4 antagonist | 0.077 0.02 CHEMBL1033 0.07 0.027 CHEMBL1035 | CHEMBL1033 | |
| 0.034 | 0.265 | 0.133 | Bronchodilator | 0.133 0.038 CHEMBL1033 | CHEMBL1033 | |
| 0.073 | 0.325 | 0.21 | Antioxidant | 0.21 0.107 CHEMBL1031 0.19 0.122 CHEMBL1033 0.168 0.144 CHEMBL1030 0.209 0.108 CHEMBL1032 | CHEMBL1031 | |
| 0.087 | 0.359 | 0.198 | Hypoxia-inducible factor 1 alpha inhibitor | 0.198 0.154 CHEMBL1033 | CHEMBL1033 | |
| 0.01 | 0.285 | 0.055 | Alpha tubulin antagonist | 0.055 0.035 CHEMBL1033 | CHEMBL1033 | |
| 0.059 | 0.338 | 0.204 | Free radical scavenger | 0.204 0.094 CHEMBL1031 0.155 0.14 CHEMBL1030 0.199 0.099 CHEMBL1032 | CHEMBL1031 | |
| 0.039 | 0.367 | 0.128 | Estrogen antagonist | 0.122 0.051 CHEMBL1031 0.122 0.052 CHEMBL1030 0.111 0.073 CHEMBL1035 0.128 0.04 CHEMBL1032 | CHEMBL1032 | |
| 0.056 | 0.407 | 0.196 | Thioredoxin glutathione reductase inhibitor | 0.196 0.176 CHEMBL1033 | CHEMBL1033 | |
| 0.088 | 0.51 | 0.263 | Apoptosis agonist | 0.263 0.201 CHEMBL1033 | CHEMBL1033 | |
| 0.022 | 0.447 | 0.111 | Estrogen receptor beta antagonist | 0.106 0.053 CHEMBL1031 0.103 0.059 CHEMBL1030 0.097 0.071 CHEMBL1035 0.111 0.044 CHEMBL1032 | CHEMBL1032 | |
| 0.076 | 0.524 | 0.232 | Caspase 3 stimulant | 0.232 0.129 CHEMBL1033 | CHEMBL1033 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |