| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.968 | 0.001 | 0.968 | Glutamate decarboxylase inhibitor | 0.898 0.001 CHEMBL3544532 0.908 0.001 CHEMBL3544531 0.587 0.002 CHEMBL3544554 | ||
| 0.962 | 0.002 | 0.962 | Interleukin antagonist | 0.696 0.004 CHEMBL3544532 0.684 0.005 CHEMBL3544531 0.306 0.047 CHEMBL3544554 | ||
| 0.931 | 0.001 | 0.931 | Superoxide dismutase inhibitor | 0.793 0.003 CHEMBL3544532 0.696 0.004 CHEMBL3544531 0.754 0.004 CHEMBL3544554 | ||
| 0.846 | 0.002 | 0.846 | Chelator | 0.69 0.003 CHEMBL3544532 0.702 0.003 CHEMBL3544531 0.641 0.003 CHEMBL3544554 | ||
| 0.832 | 0.001 | 0.832 | T cell inhibitor | 0.69 0.002 CHEMBL3544532 0.541 0.003 CHEMBL3544531 0.639 0.003 CHEMBL3544554 | ||
| 0.797 | 0.001 | 0.867 | Adenine nucleotide translocase inhibitor | 0.824 0.001 CHEMBL3544532 0.76 0.001 CHEMBL3544531 0.867 0 CHEMBL3544554 | CHEMBL3544554 | |
| 0.758 | 0.004 | 0.758 | Hypoglycemic | 0.664 0.005 CHEMBL3544532 0.552 0.011 CHEMBL3544531 0.609 0.008 CHEMBL3544554 | ||
| 0.74 | 0.004 | 0.74 | Vasodilator | 0.664 0.005 CHEMBL3544532 0.712 0.004 CHEMBL3544531 0.626 0.005 CHEMBL3544554 | ||
| 0.714 | 0.002 | 0.714 | Aminopeptidase B inhibitor | 0.427 0.004 CHEMBL3544532 0.439 0.004 CHEMBL3544531 0.443 0.004 CHEMBL3544554 | ||
| 0.685 | 0.003 | 0.685 | Peroxidase inhibitor | 0.565 0.005 CHEMBL3544532 0.575 0.005 CHEMBL3544531 0.448 0.014 CHEMBL3544554 | ||
| 0.659 | 0.007 | 0.659 | Immunosuppressant | 0.542 0.022 CHEMBL3544532 0.379 0.072 CHEMBL3544531 0.654 0.007 CHEMBL3544554 | ||
| 0.637 | 0.002 | 0.637 | Aminoacyl-tRNA synthetase inhibitor | 0.487 0.003 CHEMBL3544532 0.437 0.004 CHEMBL3544531 0.453 0.003 CHEMBL3544554 | ||
| 0.604 | 0.002 | 0.604 | Alcohol dehydrogenase inhibitor | 0.332 0.005 CHEMBL3544532 0.403 0.004 CHEMBL3544531 0.221 0.01 CHEMBL3544554 | ||
| 0.616 | 0.017 | 0.616 | Aldehyde oxidase inhibitor | 0.525 0.029 CHEMBL3544532 0.363 0.053 CHEMBL3544531 0.412 0.045 CHEMBL3544554 | ||
| 0.581 | 0.003 | 0.581 | Glutamate dehydrogenase inhibitor | 0.51 0.003 CHEMBL3544532 0.41 0.004 CHEMBL3544531 0.289 0.006 CHEMBL3544554 | ||
| 0.551 | 0.002 | 0.551 | Phenylalanine 4-hydroxylase inhibitor | 0.349 0.004 CHEMBL3544532 0.361 0.003 CHEMBL3544531 0.469 0.003 CHEMBL3544554 | ||
| 0.568 | 0.021 | 0.615 | Immunostimulant | 0.558 0.022 CHEMBL3544532 0.615 0.015 CHEMBL3544531 0.498 0.029 CHEMBL3544554 | CHEMBL3544531 | |
| 0.537 | 0.005 | 0.634 | Alpha-N-acetylglucosaminidase inhibitor | 0.634 0.004 CHEMBL3544532 0.397 0.009 CHEMBL3544531 0.489 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.502 | 0.003 | 0.502 | Histidine decarboxylase inhibitor | 0.441 0.003 CHEMBL3544532 0.435 0.003 CHEMBL3544531 0.252 0.009 CHEMBL3544554 | ||
| 0.489 | 0.005 | 0.581 | 5 Hydroxytryptamine uptake stimulant | 0.542 0.004 CHEMBL3544532 0.437 0.009 CHEMBL3544531 0.581 0.003 CHEMBL3544554 | CHEMBL3544554 | |
| 0.469 | 0.003 | 0.469 | Integrin alpha5beta1 antagonist | 0.076 0.007 CHEMBL3544532 0.05 0.018 CHEMBL3544531 0.046 0.022 CHEMBL3544554 | ||
| 0.464 | 0.004 | 0.544 | Tyrosine 3 hydroxylase inhibitor | 0.543 0.004 CHEMBL3544532 0.377 0.011 CHEMBL3544531 0.544 0.004 CHEMBL3544554 | CHEMBL3544554 | |
| 0.433 | 0.003 | 0.459 | Ornithine carbamoyltransferase inhibitor | 0.356 0.004 CHEMBL3544532 0.459 0.003 CHEMBL3544531 0.337 0.004 CHEMBL3544554 | CHEMBL3544531 | |
| 0.43 | 0.009 | 0.43 | Bone formation stimulant | 0.132 0.075 CHEMBL3544532 0.106 0.099 CHEMBL3544554 | ||
| 0.426 | 0.009 | 0.426 | Phospholipase C inhibitor | 0.302 0.018 CHEMBL3544532 0.295 0.019 CHEMBL3544531 0.303 0.018 CHEMBL3544554 | ||
| 0.412 | 0.005 | 0.5 | GABA C receptor agonist | 0.5 0.004 CHEMBL3544532 0.286 0.01 CHEMBL3544531 0.368 0.006 CHEMBL3544554 | CHEMBL3544532 | |
| 0.407 | 0.004 | 0.407 | Porphobilinogen synthase inhibitor | 0.314 0.005 CHEMBL3544532 0.142 0.022 CHEMBL3544531 0.246 0.008 CHEMBL3544554 | ||
| 0.391 | 0.004 | 0.391 | Catalase inhibitor | 0.341 0.005 CHEMBL3544532 0.339 0.005 CHEMBL3544531 0.218 0.012 CHEMBL3544554 | ||
| 0.405 | 0.026 | 0.439 | Interleukin 2 agonist | 0.439 0.018 CHEMBL3544532 0.372 0.037 CHEMBL3544531 0.398 0.028 CHEMBL3544554 | CHEMBL3544532 | |
| 0.42 | 0.042 | 0.534 | 5 Hydroxytryptamine release stimulant | 0.534 0.022 CHEMBL3544532 0.237 0.096 CHEMBL3544531 0.519 0.024 CHEMBL3544554 | CHEMBL3544532 | |
| 0.37 | 0.005 | 0.37 | Succinate dehydrogenase inhibitor | 0.328 0.007 CHEMBL3544532 0.277 0.015 CHEMBL3544531 0.233 0.029 CHEMBL3544554 | ||
| 0.366 | 0.004 | 0.366 | Adenylate kinase inhibitor | 0.364 0.004 CHEMBL3544532 0.318 0.006 CHEMBL3544531 0.273 0.008 CHEMBL3544554 | ||
| 0.335 | 0.004 | 0.335 | GP IIb/IIIa receptor antagonist | 0.146 0.011 CHEMBL3544532 0.063 0.026 CHEMBL3544531 0.07 0.024 CHEMBL3544554 | ||
| 0.356 | 0.032 | 0.356 | Insulysin inhibitor | 0.336 0.039 CHEMBL3544532 0.279 0.073 CHEMBL3544531 0.297 0.06 CHEMBL3544554 | ||
| 0.326 | 0.007 | 0.381 | Expectorant | 0.24 0.014 CHEMBL3544532 0.381 0.005 CHEMBL3544531 0.231 0.015 CHEMBL3544554 | CHEMBL3544531 | |
| 0.323 | 0.004 | 0.383 | Mucolytic | 0.25 0.006 CHEMBL3544532 0.383 0.003 CHEMBL3544531 0.235 0.008 CHEMBL3544554 | CHEMBL3544531 | |
| 0.338 | 0.021 | 0.485 | Hepatoprotectant | 0.272 0.038 CHEMBL3544532 0.485 0.008 CHEMBL3544531 0.255 0.042 CHEMBL3544554 | CHEMBL3544531 | |
| 0.331 | 0.038 | 0.331 | Angiogenesis stimulant | 0.303 0.048 CHEMBL3544532 0.241 0.074 CHEMBL3544531 0.314 0.044 CHEMBL3544554 | ||
| 0.299 | 0.008 | 0.359 | Ferrochelatase inhibitor | 0.359 0.004 CHEMBL3544532 0.207 0.021 CHEMBL3544531 0.269 0.011 CHEMBL3544554 | CHEMBL3544532 | |
| 0.291 | 0.004 | 0.375 | Carbamoyl phosphate synthetase inhibitor | 0.375 0.003 CHEMBL3544532 0.277 0.005 CHEMBL3544531 0.258 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.287 | 0.003 | 0.287 | Aminopeptidase I inhibitor | 0.225 0.005 CHEMBL3544532 0.191 0.008 CHEMBL3544531 0.183 0.008 CHEMBL3544554 | ||
| 0.288 | 0.004 | 0.386 | Argininosuccinate synthase inhibitor | 0.386 0.003 CHEMBL3544532 0.263 0.005 CHEMBL3544531 0.264 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.299 | 0.024 | 0.299 | Thrombolytic | 0.27 0.029 CHEMBL3544532 0.208 0.048 CHEMBL3544531 0.249 0.034 CHEMBL3544554 | ||
| 0.273 | 0.003 | 0.363 | Kinesin antagonist | 0.301 0.003 CHEMBL3544532 0.363 0.002 CHEMBL3544531 0.327 0.003 CHEMBL3544554 | CHEMBL3544531 | |
| 0.273 | 0.003 | 0.363 | Kinesin-like protein 1 inhibitor | 0.301 0.003 CHEMBL3544532 0.363 0.002 CHEMBL3544531 0.327 0.003 CHEMBL3544554 | CHEMBL3544531 | |
| 0.276 | 0.008 | 0.412 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.412 0.004 CHEMBL3544532 0.306 0.006 CHEMBL3544531 0.259 0.009 CHEMBL3544554 | CHEMBL3544532 | |
| 0.275 | 0.006 | 0.277 | Phosphofructokinase-1 inhibitor | 0.277 0.006 CHEMBL3544532 0.195 0.012 CHEMBL3544531 0.181 0.013 CHEMBL3544554 | CHEMBL3544532 | |
| 0.308 | 0.041 | 0.308 | DNA synthesis inhibitor | 0.3 0.043 CHEMBL3544532 0.219 0.096 CHEMBL3544531 0.288 0.048 CHEMBL3544554 | ||
| 0.263 | 0.004 | 0.263 | Angiotensin-converting enzyme inhibitor | 0.08 0.013 CHEMBL3544532 0.106 0.008 CHEMBL3544531 0.074 0.016 CHEMBL3544554 | ||
| 0.33 | 0.074 | 0.392 | Cholesterol antagonist | 0.392 0.051 CHEMBL3544532 0.357 0.062 CHEMBL3544531 0.258 0.12 CHEMBL3544554 | CHEMBL3544532 | |
| 0.251 | 0.005 | 0.253 | Integrin antagonist | 0.253 0.005 CHEMBL3544532 0.224 0.006 CHEMBL3544531 0.116 0.014 CHEMBL3544554 | CHEMBL3544532 | |
| 0.316 | 0.075 | 0.335 | Vasodilator, coronary | 0.335 0.063 CHEMBL3544532 0.193 0.188 CHEMBL3544531 0.268 0.117 CHEMBL3544554 | CHEMBL3544532 | |
| 0.291 | 0.053 | 0.347 | Interleukin agonist | 0.347 0.03 CHEMBL3544532 0.219 0.103 CHEMBL3544531 0.273 0.063 CHEMBL3544554 | CHEMBL3544532 | |
| 0.274 | 0.038 | 0.417 | Growth hormone agonist | 0.329 0.027 CHEMBL3544532 0.257 0.042 CHEMBL3544531 0.417 0.014 CHEMBL3544554 | CHEMBL3544554 | |
| 0.349 | 0.116 | 0.418 | 5 Hydroxytryptamine release inhibitor | 0.418 0.068 CHEMBL3544532 0.269 0.202 CHEMBL3544531 0.343 0.121 CHEMBL3544554 | CHEMBL3544532 | |
| 0.226 | 0.003 | 0.226 | Angiotensin-converting enzyme 2 inhibitor | 0.019 0.01 CHEMBL3544532 0.016 0.014 CHEMBL3544554 | ||
| 0.244 | 0.022 | 0.244 | Neurotensin receptor agonist | 0.223 0.026 CHEMBL3544532 0.167 0.067 CHEMBL3544531 0.211 0.03 CHEMBL3544554 | ||
| 0.281 | 0.059 | 0.421 | Platelet antagonist | 0.295 0.054 CHEMBL3544532 0.281 0.059 CHEMBL3544531 0.421 0.023 CHEMBL3544554 | CHEMBL3544554 | |
| 0.217 | 0.004 | 0.217 | Endothelin-converting enzyme inhibitor | 0.151 0.009 CHEMBL3544532 0.141 0.01 CHEMBL3544531 0.053 0.028 CHEMBL3544554 | ||
| 0.209 | 0.004 | 0.263 | NMDA receptor agonist | 0.225 0.004 CHEMBL3544532 0.263 0.004 CHEMBL3544531 0.217 0.004 CHEMBL3544554 | CHEMBL3544531 | |
| 0.207 | 0.003 | 0.207 | Neutral endopeptidase inhibitor | 0.027 0.013 CHEMBL3544532 0.08 0.005 CHEMBL3544531 0.019 0.016 CHEMBL3544554 | ||
| 0.232 | 0.033 | 0.232 | Amylase inhibitor | 0.162 0.059 CHEMBL3544532 0.122 0.08 CHEMBL3544531 0.209 0.041 CHEMBL3544554 | ||
| 0.332 | 0.136 | 0.524 | Cyclophilin D inhibitor | 0.356 0.118 CHEMBL3544532 0.524 0.044 CHEMBL3544554 | CHEMBL3544554 | |
| 0.247 | 0.053 | 0.288 | Peptidyltransferase inhibitor | 0.275 0.035 CHEMBL3544532 0.236 0.061 CHEMBL3544531 0.288 0.029 CHEMBL3544554 | CHEMBL3544554 | |
| 0.288 | 0.097 | 0.442 | Antithrombotic | 0.393 0.051 CHEMBL3544532 0.346 0.066 CHEMBL3544531 0.442 0.04 CHEMBL3544554 | CHEMBL3544554 | |
| 0.19 | 0.007 | 0.534 | Alcohol oxidase inhibitor | 0.534 0.003 CHEMBL3544532 0.152 0.01 CHEMBL3544531 0.155 0.01 CHEMBL3544554 | CHEMBL3544532 | |
| 0.183 | 0.01 | 0.21 | DOPA decarboxylase inhibitor | 0.21 0.005 CHEMBL3544532 0.148 0.023 CHEMBL3544531 0.18 0.01 CHEMBL3544554 | CHEMBL3544532 | |
| 0.189 | 0.027 | 0.238 | Cystathionine beta-synthase inhibitor | 0.238 0.017 CHEMBL3544532 0.127 0.053 CHEMBL3544531 0.179 0.03 CHEMBL3544554 | CHEMBL3544532 | |
| 0.165 | 0.003 | 0.214 | Glutamate (mGluR6) antagonist | 0.214 0.003 CHEMBL3544532 0.132 0.004 CHEMBL3544531 0.171 0.003 CHEMBL3544554 | CHEMBL3544532 | |
| 0.169 | 0.009 | 0.169 | Glutathione S-transferase inhibitor | 0.142 0.014 CHEMBL3544532 0.114 0.026 CHEMBL3544531 0.154 0.011 CHEMBL3544554 | ||
| 0.187 | 0.036 | 0.232 | Cell wall synthesis inhibitor | 0.228 0.021 CHEMBL3544532 0.216 0.024 CHEMBL3544531 0.232 0.02 CHEMBL3544554 | CHEMBL3544554 | |
| 0.183 | 0.032 | 0.219 | Aldehyde dehydrogenase inhibitor | 0.164 0.04 CHEMBL3544532 0.147 0.049 CHEMBL3544531 0.219 0.024 CHEMBL3544554 | CHEMBL3544554 | |
| 0.16 | 0.012 | 0.16 | Matrix metalloproteinase inhibitor | 0.069 0.045 CHEMBL3544532 0.124 0.019 CHEMBL3544554 | ||
| 0.177 | 0.032 | 0.265 | Cell adhesion inhibitor | 0.265 0.013 CHEMBL3544532 0.107 0.078 CHEMBL3544531 0.207 0.023 CHEMBL3544554 | CHEMBL3544532 | |
| 0.161 | 0.017 | 0.266 | Triose-phosphate isomerase inhibitor | 0.266 0.006 CHEMBL3544532 0.143 0.022 CHEMBL3544531 0.214 0.009 CHEMBL3544554 | CHEMBL3544532 | |
| 0.174 | 0.031 | 0.187 | Adenylate cyclase stimulant | 0.182 0.024 CHEMBL3544532 0.145 0.072 CHEMBL3544531 0.187 0.02 CHEMBL3544554 | CHEMBL3544554 | |
| 0.183 | 0.04 | 0.183 | Mannose-6-phosphate isomerase inhibitor | 0.149 0.065 CHEMBL3544532 0.136 0.079 CHEMBL3544531 | ||
| 0.153 | 0.01 | 0.22 | Ornithine decarboxylase inhibitor | 0.22 0.004 CHEMBL3544532 0.162 0.008 CHEMBL3544531 0.162 0.008 CHEMBL3544554 | CHEMBL3544532 | |
| 0.146 | 0.008 | 0.64 | Aminopeptidase microsomal inhibitor | 0.307 0.003 CHEMBL3544532 0.64 0.002 CHEMBL3544531 0.097 0.018 CHEMBL3544554 | CHEMBL3544531 | |
| 0.22 | 0.083 | 0.22 | Free radical scavenger | 0.195 0.102 CHEMBL3544531 | ||
| 0.2 | 0.073 | 0.269 | Insulin sensitizer | 0.269 0.025 CHEMBL3544532 0.244 0.038 CHEMBL3544531 0.255 0.031 CHEMBL3544554 | CHEMBL3544532 | |
| 0.125 | 0.004 | 0.189 | Fumarate hydratase inhibitor | 0.189 0.003 CHEMBL3544532 0.077 0.007 CHEMBL3544531 0.105 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.122 | 0.003 | 0.122 | Lysine carboxypeptidase inhibitor | 0.063 0.006 CHEMBL3544532 0.052 0.007 CHEMBL3544531 0.046 0.009 CHEMBL3544554 | ||
| 0.127 | 0.008 | 0.623 | Aminopeptidase N inhibitor | 0.286 0.003 CHEMBL3544532 0.623 0.002 CHEMBL3544531 0.076 0.018 CHEMBL3544554 | CHEMBL3544531 | |
| 0.116 | 0.004 | 0.139 | Nitric oxide donor | 0.125 0.004 CHEMBL3544532 0.125 0.004 CHEMBL3544531 0.139 0.003 CHEMBL3544554 | CHEMBL3544554 | |
| 0.124 | 0.013 | 0.207 | Biliverdin reductase inhibitor | 0.207 0.005 CHEMBL3544532 0.107 0.017 CHEMBL3544531 0.108 0.016 CHEMBL3544554 | CHEMBL3544532 | |
| 0.123 | 0.012 | 0.157 | Glycine receptor agonist | 0.157 0.006 CHEMBL3544532 0.11 0.016 CHEMBL3544531 0.112 0.015 CHEMBL3544554 | CHEMBL3544532 | |
| 0.224 | 0.114 | 0.27 | Gastrin inhibitor | 0.27 0.058 CHEMBL3544532 0.203 0.144 CHEMBL3544531 0.252 0.077 CHEMBL3544554 | CHEMBL3544532 | |
| 0.114 | 0.005 | 0.114 | Leukotriene A4 hydrolase inhibitor | 0.033 0.029 CHEMBL3544532 0.068 0.012 CHEMBL3544531 | ||
| 0.143 | 0.034 | 0.18 | GABA C receptor antagonist | 0.18 0.018 CHEMBL3544532 0.122 0.05 CHEMBL3544531 0.127 0.046 CHEMBL3544554 | CHEMBL3544532 | |
| 0.189 | 0.082 | 0.189 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.156 0.136 CHEMBL3544532 | ||
| 0.121 | 0.013 | 0.158 | Toll-Like receptor 2 agonist | 0.098 0.015 CHEMBL3544532 0.072 0.018 CHEMBL3544531 0.158 0.01 CHEMBL3544554 | CHEMBL3544554 | |
| 0.131 | 0.024 | 0.159 | NADH dehydrogenase inhibitor | 0.159 0.016 CHEMBL3544532 0.099 0.045 CHEMBL3544531 0.119 0.029 CHEMBL3544554 | CHEMBL3544532 | |
| 0.11 | 0.003 | 0.11 | Arginase inhibitor | 0.086 0.005 CHEMBL3544532 0.078 0.006 CHEMBL3544531 0.084 0.005 CHEMBL3544554 | ||
| 0.109 | 0.003 | 0.138 | Kainate receptor agonist | 0.138 0.002 CHEMBL3544532 0.081 0.004 CHEMBL3544531 0.101 0.003 CHEMBL3544554 | CHEMBL3544532 | |
| 0.13 | 0.024 | 0.13 | Opioid delta receptor antagonist | 0.115 0.027 CHEMBL3544532 0.07 0.04 CHEMBL3544531 0.074 0.038 CHEMBL3544554 | ||
| 0.15 | 0.044 | 0.158 | Ca2+-transporting ATPase inhibitor | 0.158 0.026 CHEMBL3544532 0.137 0.087 CHEMBL3544531 0.148 0.047 CHEMBL3544554 | CHEMBL3544532 | |
| 0.168 | 0.063 | 0.168 | Diuretic | 0.14 0.086 CHEMBL3544532 0.134 0.09 CHEMBL3544554 | ||
| 0.116 | 0.012 | 0.116 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.077 0.022 CHEMBL3544532 0.055 0.041 CHEMBL3544554 | ||
| 0.151 | 0.046 | 0.221 | Alkylator | 0.153 0.045 CHEMBL3544532 0.221 0.021 CHEMBL3544531 0.137 0.054 CHEMBL3544554 | CHEMBL3544531 | |
| 0.137 | 0.034 | 0.137 | Carbonic anhydrase III inhibitor | 0.092 0.071 CHEMBL3544532 | ||
| 0.133 | 0.031 | 0.22 | Uric acid excretion stimulant | 0.22 0.01 CHEMBL3544532 0.216 0.011 CHEMBL3544531 0.138 0.028 CHEMBL3544554 | CHEMBL3544532 | |
| 0.106 | 0.005 | 0.106 | Vanilloid 2 antagonist | |||
| 0.131 | 0.031 | 0.177 | Folate antagonist | 0.177 0.014 CHEMBL3544532 0.168 0.017 CHEMBL3544531 0.159 0.019 CHEMBL3544554 | CHEMBL3544532 | |
| 0.264 | 0.164 | 0.465 | Antibacterial | 0.465 0.051 CHEMBL3544532 0.423 0.067 CHEMBL3544531 0.372 0.09 CHEMBL3544554 | CHEMBL3544532 | |
| 0.101 | 0.003 | 0.122 | Glutamate (mGluR8) agonist | 0.122 0.002 CHEMBL3544532 0.088 0.004 CHEMBL3544531 0.098 0.003 CHEMBL3544554 | CHEMBL3544532 | |
| 0.131 | 0.033 | 0.199 | Creatine kinase inhibitor | 0.199 0.011 CHEMBL3544532 0.157 0.021 CHEMBL3544531 0.117 0.043 CHEMBL3544554 | CHEMBL3544532 | |
| 0.131 | 0.033 | 0.131 | HIV-1 integrase (Overall Integration) inhibitor | 0.107 0.049 CHEMBL3544532 | ||
| 0.103 | 0.006 | 0.103 | Alpha-mannosidase inhibitor | 0.084 0.01 CHEMBL3544532 0.077 0.013 CHEMBL3544531 0.076 0.013 CHEMBL3544554 | ||
| 0.101 | 0.005 | 0.117 | Collagenase inhibitor | 0.048 0.037 CHEMBL3544532 0.117 0.005 CHEMBL3544554 | CHEMBL3544554 | |
| 0.112 | 0.017 | 0.112 | Ribonucleoside-diphosphate reductase inhibitor | 0.087 0.023 CHEMBL3544532 0.071 0.028 CHEMBL3544531 0.053 0.038 CHEMBL3544554 | ||
| 0.099 | 0.004 | 0.099 | Glutamate (mGluR3) antagonist | 0.099 0.004 CHEMBL3544532 0.042 0.019 CHEMBL3544531 0.071 0.006 CHEMBL3544554 | ||
| 0.098 | 0.004 | 0.121 | Membrane dipeptidase inhibitor | 0.088 0.004 CHEMBL3544532 0.121 0.003 CHEMBL3544531 0.087 0.004 CHEMBL3544554 | CHEMBL3544531 | |
| 0.1 | 0.006 | 0.1 | Mannosidase inhibitor | 0.07 0.011 CHEMBL3544532 0.065 0.014 CHEMBL3544531 0.06 0.017 CHEMBL3544554 | ||
| 0.126 | 0.034 | 0.126 | Anabolic | 0.116 0.044 CHEMBL3544532 0.094 0.071 CHEMBL3544554 | ||
| 0.11 | 0.018 | 0.11 | Ribonucleotide reductase inhibitor | 0.087 0.024 CHEMBL3544532 0.072 0.03 CHEMBL3544531 0.053 0.04 CHEMBL3544554 | ||
| 0.146 | 0.055 | 0.18 | Toll-Like receptor 2 antagonist | 0.18 0.034 CHEMBL3544532 0.141 0.059 CHEMBL3544531 0.145 0.056 CHEMBL3544554 | CHEMBL3544532 | |
| 0.193 | 0.102 | 0.221 | Nitric-oxide synthase stimulant | 0.221 0.059 CHEMBL3544532 0.168 0.157 CHEMBL3544531 0.189 0.11 CHEMBL3544554 | CHEMBL3544532 | |
| 0.142 | 0.052 | 0.198 | Cathepsin H inhibitor | 0.198 0.023 CHEMBL3544532 0.131 0.062 CHEMBL3544531 0.165 0.036 CHEMBL3544554 | CHEMBL3544532 | |
| 0.125 | 0.036 | 0.157 | GABA C receptor rho-1 antagonist | 0.157 0.018 CHEMBL3544532 0.088 0.082 CHEMBL3544531 0.112 0.048 CHEMBL3544554 | CHEMBL3544532 | |
| 0.108 | 0.018 | 0.108 | Glucagon-like peptide 1 agonist | 0.096 0.024 CHEMBL3544532 0.072 0.04 CHEMBL3544531 0.101 0.021 CHEMBL3544554 | ||
| 0.104 | 0.015 | 0.137 | Acyl-CoA dehydrogenase inhibitor | 0.137 0.01 CHEMBL3544532 0.108 0.014 CHEMBL3544531 0.107 0.015 CHEMBL3544554 | CHEMBL3544532 | |
| 0.094 | 0.006 | 0.156 | VLA-4 antagonist | 0.156 0.004 CHEMBL3544532 0.099 0.006 CHEMBL3544531 0.099 0.006 CHEMBL3544554 | CHEMBL3544532 | |
| 0.161 | 0.075 | 0.194 | Arachidonic acid antagonist | 0.183 0.05 CHEMBL3544532 0.14 0.1 CHEMBL3544531 0.194 0.038 CHEMBL3544554 | CHEMBL3544554 | |
| 0.084 | 0.005 | 0.084 | Vitronectin receptor antagonist | 0.026 0.012 CHEMBL3544532 | ||
| 0.167 | 0.088 | 0.257 | DNA methyltransferase I inhibitor | 0.205 0.067 CHEMBL3544532 0.257 0.044 CHEMBL3544531 0.188 0.075 CHEMBL3544554 | CHEMBL3544531 | |
| 0.087 | 0.008 | 0.087 | HCV NS3/NS4A protease inhibitor | 0.056 0.025 CHEMBL3544532 0.059 0.022 CHEMBL3544554 | ||
| 0.093 | 0.015 | 0.109 | Glutamate (mGluR7) antagonist | 0.109 0.007 CHEMBL3544532 0.07 0.043 CHEMBL3544531 0.085 0.022 CHEMBL3544554 | CHEMBL3544532 | |
| 0.103 | 0.025 | 0.13 | GABA aminotransferase inhibitor | 0.13 0.013 CHEMBL3544532 0.08 0.047 CHEMBL3544531 0.099 0.028 CHEMBL3544554 | CHEMBL3544532 | |
| 0.106 | 0.03 | 0.106 | Metalloproteinase-9 inhibitor | 0.069 0.056 CHEMBL3544532 0.106 0.03 CHEMBL3544554 | ||
| 0.128 | 0.052 | 0.238 | Interleukin 8 antagonist | 0.238 0.007 CHEMBL3544532 0.168 0.024 CHEMBL3544531 0.164 0.026 CHEMBL3544554 | CHEMBL3544532 | |
| 0.087 | 0.011 | 0.111 | Aconitate hydratase inhibitor | 0.111 0.007 CHEMBL3544532 0.062 0.024 CHEMBL3544531 0.077 0.015 CHEMBL3544554 | CHEMBL3544532 | |
| 0.116 | 0.041 | 0.19 | Prolactin inhibitor | 0.148 0.023 CHEMBL3544532 0.087 0.07 CHEMBL3544531 0.19 0.01 CHEMBL3544554 | CHEMBL3544554 | |
| 0.129 | 0.056 | 0.129 | Monophenol monooxygenase inhibitor | 0.096 0.079 CHEMBL3544532 0.1 0.076 CHEMBL3544531 | ||
| 0.189 | 0.117 | 0.198 | RNA-directed DNA polymerase inhibitor | 0.185 0.124 CHEMBL3544532 0.198 0.103 CHEMBL3544554 | CHEMBL3544554 | |
| 0.095 | 0.025 | 0.127 | Sirtuin 1 inhibitor | 0.085 0.031 CHEMBL3544532 0.063 0.054 CHEMBL3544531 0.127 0.012 CHEMBL3544554 | CHEMBL3544554 | |
| 0.102 | 0.033 | 0.145 | Somatostatin 1 agonist | 0.145 0.015 CHEMBL3544532 0.124 0.022 CHEMBL3544531 | CHEMBL3544532 | |
| 0.236 | 0.167 | 0.306 | GABA C receptor rho-3 antagonist | 0.306 0.112 CHEMBL3544532 0.206 0.2 CHEMBL3544554 | CHEMBL3544532 | |
| 0.235 | 0.167 | 0.448 | Histamine release inhibitor | 0.422 0.064 CHEMBL3544532 0.268 0.143 CHEMBL3544531 0.448 0.051 CHEMBL3544554 | CHEMBL3544554 | |
| 0.11 | 0.042 | 0.119 | Lanosterol 14 alpha demethylase inhibitor | 0.1 0.056 CHEMBL3544532 0.119 0.031 CHEMBL3544554 | CHEMBL3544554 | |
| 0.08 | 0.012 | 0.102 | Farnesyltransferase inhibitor | 0.074 0.014 CHEMBL3544532 0.092 0.009 CHEMBL3544531 0.102 0.007 CHEMBL3544554 | CHEMBL3544554 | |
| 0.167 | 0.103 | 0.26 | DNA methylase inhibitor | 0.214 0.07 CHEMBL3544532 0.26 0.043 CHEMBL3544531 0.188 0.087 CHEMBL3544554 | CHEMBL3544531 | |
| 0.188 | 0.124 | 0.217 | Antioxidant | 0.217 0.103 CHEMBL3544531 | CHEMBL3544531 | |
| 0.088 | 0.024 | 0.088 | Phospholipase D inhibitor | 0.067 0.059 CHEMBL3544532 | ||
| 0.087 | 0.023 | 0.112 | Carbonic anhydrase stimulant | 0.112 0.016 CHEMBL3544532 0.061 0.04 CHEMBL3544531 0.087 0.023 CHEMBL3544554 | CHEMBL3544532 | |
| 0.071 | 0.009 | 0.196 | Integrin alpha4 antagonist | 0.183 0.004 CHEMBL3544532 0.196 0.004 CHEMBL3544531 0.094 0.007 CHEMBL3544554 | CHEMBL3544531 | |
| 0.106 | 0.044 | 0.106 | Opioid antagonist | 0.098 0.049 CHEMBL3544532 0.082 0.066 CHEMBL3544554 | ||
| 0.066 | 0.004 | 0.075 | Glutamate (mGluR8) antagonist | 0.075 0.004 CHEMBL3544532 0.057 0.006 CHEMBL3544531 0.064 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.061 | 0.005 | 0.104 | Integrin beta7 antagonist | 0.104 0.004 CHEMBL3544532 0.067 0.005 CHEMBL3544531 0.081 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.122 | 0.066 | 0.154 | Adenylate cyclase inhibitor | 0.154 0.042 CHEMBL3544532 0.149 0.046 CHEMBL3544554 | CHEMBL3544532 | |
| 0.162 | 0.106 | 0.162 | Pyruvate kinase inhibitor | |||
| 0.09 | 0.035 | 0.09 | Opioid mu receptor antagonist | 0.079 0.04 CHEMBL3544532 | ||
| 0.071 | 0.017 | 0.086 | Complement C3a chemotactic receptor antagonist | 0.086 0.012 CHEMBL3544532 0.056 0.024 CHEMBL3544531 0.07 0.017 CHEMBL3544554 | CHEMBL3544532 | |
| 0.081 | 0.027 | 0.129 | NMDA receptor glycine site agonist | 0.125 0.008 CHEMBL3544532 0.074 0.033 CHEMBL3544531 0.129 0.006 CHEMBL3544554 | CHEMBL3544554 | |
| 0.183 | 0.13 | 0.183 | Calpain inhibitor | |||
| 0.095 | 0.042 | 0.097 | Factor XII inhibitor | 0.097 0.041 CHEMBL3544532 0.079 0.069 CHEMBL3544531 0.095 0.042 CHEMBL3544554 | CHEMBL3544532 | |
| 0.057 | 0.004 | 0.175 | Glutamate (mGluR1a) agonist | 0.146 0.003 CHEMBL3544532 0.175 0.002 CHEMBL3544531 0.079 0.004 CHEMBL3544554 | CHEMBL3544531 | |
| 0.062 | 0.01 | 0.085 | AMPA 4 receptor antagonist | 0.076 0.007 CHEMBL3544532 0.038 0.03 CHEMBL3544531 0.085 0.006 CHEMBL3544554 | CHEMBL3544554 | |
| 0.064 | 0.012 | 0.098 | Glutamate (mGluR4) antagonist | 0.098 0.005 CHEMBL3544532 0.044 0.029 CHEMBL3544531 0.089 0.007 CHEMBL3544554 | CHEMBL3544532 | |
| 0.067 | 0.016 | 0.067 | Adenosine deaminase inhibitor | 0.055 0.025 CHEMBL3544532 0.047 0.033 CHEMBL3544531 0.057 0.023 CHEMBL3544554 | ||
| 0.107 | 0.056 | 0.116 | Factor V inhibitor | 0.116 0.043 CHEMBL3544532 0.105 0.058 CHEMBL3544531 0.102 0.064 CHEMBL3544554 | CHEMBL3544532 | |
| 0.08 | 0.031 | 0.08 | Neutrophil collagenase inhibitor | 0.062 0.048 CHEMBL3544554 | ||
| 0.072 | 0.023 | 0.072 | Matrix metalloproteinase (membrane-type) inhibitor | 0.053 0.041 CHEMBL3544532 0.056 0.037 CHEMBL3544554 | ||
| 0.052 | 0.004 | 0.065 | Glutamate (mGluR3) agonist | 0.063 0.004 CHEMBL3544532 0.045 0.006 CHEMBL3544531 0.065 0.003 CHEMBL3544554 | CHEMBL3544554 | |
| 0.063 | 0.016 | 0.084 | Glucose-6-phosphate isomerase inhibitor | 0.084 0.008 CHEMBL3544532 0.058 0.02 CHEMBL3544531 0.059 0.02 CHEMBL3544554 | CHEMBL3544532 | |
| 0.051 | 0.005 | 0.088 | Integrin alpha4beta7 antagonist | 0.088 0.004 CHEMBL3544532 0.039 0.006 CHEMBL3544531 0.06 0.005 CHEMBL3544554 | CHEMBL3544532 | |
| 0.05 | 0.005 | 0.061 | Tryptophan 5 hydroxylase inhibitor | 0.061 0.004 CHEMBL3544532 0.039 0.018 CHEMBL3544531 0.055 0.004 CHEMBL3544554 | CHEMBL3544532 | |
| 0.092 | 0.048 | 0.106 | Granulocyte macrophage colony stimulating factor agonist | 0.106 0.027 CHEMBL3544532 0.085 0.062 CHEMBL3544554 | CHEMBL3544532 | |
| 0.058 | 0.014 | 0.088 | Glutamate (mGluR group III) antagonist | 0.088 0.006 CHEMBL3544532 0.041 0.037 CHEMBL3544531 0.075 0.008 CHEMBL3544554 | CHEMBL3544532 | |
| 0.061 | 0.018 | 0.077 | Glutamate (mGluR group III) agonist | 0.077 0.014 CHEMBL3544532 0.044 0.028 CHEMBL3544531 0.057 0.02 CHEMBL3544554 | CHEMBL3544532 | |
| 0.05 | 0.007 | 0.05 | Carboxypeptidase B inhibitor | 0.039 0.013 CHEMBL3544532 0.034 0.02 CHEMBL3544531 0.034 0.021 CHEMBL3544554 | ||
| 0.069 | 0.026 | 0.069 | Botulinum neurotoxin type A inhibitor | 0.056 0.044 CHEMBL3544532 0.06 0.038 CHEMBL3544554 | ||
| 0.046 | 0.004 | 0.067 | Aminopeptidase A inhibitor | 0.037 0.005 CHEMBL3544532 0.067 0.003 CHEMBL3544531 0.033 0.006 CHEMBL3544554 | CHEMBL3544531 | |
| 0.068 | 0.027 | 0.068 | Matrix metalloproteinase 1 inhibitor | 0.057 0.034 CHEMBL3544554 | ||
| 0.1 | 0.06 | 0.193 | Nitric-oxide synthase inhibitor | 0.142 0.026 CHEMBL3544532 0.193 0.01 CHEMBL3544531 0.159 0.019 CHEMBL3544554 | CHEMBL3544531 | |
| 0.137 | 0.098 | 0.159 | Interferon gamma antagonist | 0.159 0.067 CHEMBL3544532 0.142 0.089 CHEMBL3544554 | CHEMBL3544532 | |
| 0.062 | 0.023 | 0.062 | Metalloproteinase-3 inhibitor | 0.045 0.04 CHEMBL3544532 0.051 0.032 CHEMBL3544554 | ||
| 0.089 | 0.051 | 0.102 | Hematopoietic | 0.102 0.034 CHEMBL3544532 0.093 0.044 CHEMBL3544554 | CHEMBL3544532 | |
| 0.043 | 0.005 | 0.043 | Aminopeptidase P inhibitor | 0.026 0.013 CHEMBL3544532 0.021 0.019 CHEMBL3544531 0.021 0.019 CHEMBL3544554 | ||
| 0.098 | 0.06 | 0.099 | Electrolyte absorption antagonist | 0.099 0.059 CHEMBL3544532 | CHEMBL3544532 | |
| 0.042 | 0.005 | 0.144 | Glutamate (mGluR1) agonist | 0.125 0.003 CHEMBL3544532 0.144 0.003 CHEMBL3544531 0.053 0.005 CHEMBL3544554 | CHEMBL3544531 | |
| 0.051 | 0.015 | 0.081 | Kainate receptor 2 antagonist | 0.076 0.007 CHEMBL3544532 0.081 0.006 CHEMBL3544554 | CHEMBL3544554 | |
| 0.1 | 0.065 | 0.119 | Protease inhibitor | 0.119 0.048 CHEMBL3544532 0.115 0.052 CHEMBL3544554 | CHEMBL3544532 | |
| 0.083 | 0.049 | 0.118 | Metalloproteinase-2 inhibitor | 0.076 0.057 CHEMBL3544532 0.118 0.03 CHEMBL3544554 | CHEMBL3544554 | |
| 0.115 | 0.083 | 0.174 | Cyclooxygenase 3 inhibitor | 0.174 0.031 CHEMBL3544532 0.167 0.035 CHEMBL3544531 0.162 0.038 CHEMBL3544554 | CHEMBL3544532 | |
| 0.07 | 0.038 | 0.083 | MDM2 inhibitor | 0.078 0.023 CHEMBL3544532 0.065 0.056 CHEMBL3544531 0.083 0.017 CHEMBL3544554 | CHEMBL3544554 | |
| 0.034 | 0.003 | 0.051 | Glutamate (mGluR6) agonist | 0.051 0.002 CHEMBL3544532 0.04 0.003 CHEMBL3544531 0.033 0.003 CHEMBL3544554 | CHEMBL3544532 | |
| 0.096 | 0.065 | 0.15 | UDP-glucose 4-epimerase inhibitor | 0.15 0.029 CHEMBL3544532 0.127 0.039 CHEMBL3544531 0.086 0.079 CHEMBL3544554 | CHEMBL3544532 | |
| 0.13 | 0.099 | 0.157 | Sphingosine 1-phosphate receptor 5 antagonist | 0.157 0.05 CHEMBL3544532 0.14 0.08 CHEMBL3544554 | CHEMBL3544532 | |
| 0.097 | 0.066 | 0.116 | Glutamate (mGluR7) agonist | 0.116 0.035 CHEMBL3544532 0.115 0.036 CHEMBL3544554 | CHEMBL3544532 | |
| 0.107 | 0.076 | 0.131 | Photosensitizer | 0.131 0.046 CHEMBL3544532 0.128 0.049 CHEMBL3544554 | CHEMBL3544532 | |
| 0.121 | 0.091 | 0.133 | Protein kinase stimulant | 0.133 0.081 CHEMBL3544532 | CHEMBL3544532 | |
| 0.047 | 0.018 | 0.056 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.056 0.01 CHEMBL3544532 0.045 0.022 CHEMBL3544554 | CHEMBL3544532 | |
| 0.079 | 0.05 | 0.104 | Keratolytic | 0.1 0.03 CHEMBL3544532 0.104 0.028 CHEMBL3544554 | CHEMBL3544554 | |
| 0.129 | 0.102 | 0.137 | Phospholipase A2 inhibitor | 0.137 0.089 CHEMBL3544532 0.129 0.102 CHEMBL3544554 | CHEMBL3544532 | |
| 0.042 | 0.015 | 0.05 | AMPA receptor agonist | 0.05 0.009 CHEMBL3544532 0.037 0.022 CHEMBL3544531 0.05 0.009 CHEMBL3544554 | CHEMBL3544554 | |
| 0.071 | 0.044 | 0.109 | Sphingosine 1-phosphate receptor 4 agonist | 0.108 0.021 CHEMBL3544532 0.109 0.021 CHEMBL3544554 | CHEMBL3544554 | |
| 0.041 | 0.015 | 0.045 | Glutamate (mGluR4) agonist | 0.045 0.013 CHEMBL3544532 0.033 0.026 CHEMBL3544554 | CHEMBL3544532 | |
| 0.076 | 0.05 | 0.091 | GABA B receptor agonist | 0.091 0.025 CHEMBL3544532 0.071 0.066 CHEMBL3544531 0.076 0.05 CHEMBL3544554 | CHEMBL3544532 | |
| 0.049 | 0.023 | 0.049 | Growth hormone release inhibitor | 0.043 0.028 CHEMBL3544532 0.037 0.036 CHEMBL3544531 | ||
| 0.03 | 0.005 | 0.03 | N-Acetylated alpha-linked acidic dipeptidase inhibitor | 0.013 0.012 CHEMBL3544532 0.015 0.01 CHEMBL3544531 | ||
| 0.053 | 0.029 | 0.069 | Antimetabolite | 0.069 0.022 CHEMBL3544532 0.068 0.022 CHEMBL3544531 0.056 0.028 CHEMBL3544554 | CHEMBL3544532 | |
| 0.027 | 0.004 | 0.031 | Tryptophan hydroxylase 1 inhibitor | 0.031 0.003 CHEMBL3544532 0.023 0.005 CHEMBL3544531 0.027 0.004 CHEMBL3544554 | CHEMBL3544532 | |
| 0.051 | 0.028 | 0.071 | Neurotensin receptor antagonist | 0.071 0.02 CHEMBL3544532 0.041 0.036 CHEMBL3544531 0.043 0.034 CHEMBL3544554 | CHEMBL3544532 | |
| 0.088 | 0.066 | 0.122 | Glutamate release inhibitor | 0.122 0.02 CHEMBL3544532 0.086 0.073 CHEMBL3544531 0.113 0.028 CHEMBL3544554 | CHEMBL3544532 | |
| 0.048 | 0.026 | 0.048 | Macrophage elastase inhibitor | 0.04 0.034 CHEMBL3544532 0.042 0.031 CHEMBL3544554 | ||
| 0.046 | 0.024 | 0.073 | Kainate receptor antagonist | 0.073 0.011 CHEMBL3544532 0.071 0.012 CHEMBL3544554 | CHEMBL3544532 | |
| 0.041 | 0.019 | 0.053 | Integrin alpha1beta1 antagonist | 0.046 0.011 CHEMBL3544532 0.038 0.027 CHEMBL3544531 0.053 0.006 CHEMBL3544554 | CHEMBL3544554 | |
| 0.081 | 0.06 | 0.176 | Inducible nitric-oxide synthase inhibitor | 0.102 0.035 CHEMBL3544532 0.176 0.011 CHEMBL3544531 0.116 0.026 CHEMBL3544554 | CHEMBL3544531 | |
| 0.067 | 0.047 | 0.091 | Leukotriene synthesis inhibitor | 0.091 0.031 CHEMBL3544532 0.089 0.032 CHEMBL3544554 | CHEMBL3544532 | |
| 0.041 | 0.021 | 0.044 | VCAM-1 antagonist | 0.044 0.015 CHEMBL3544532 0.041 0.021 CHEMBL3544554 | CHEMBL3544532 | |
| 0.052 | 0.032 | 0.063 | Lysophosphatidic acid 3 receptor antagonist | 0.063 0.019 CHEMBL3544532 0.046 0.043 CHEMBL3544531 0.057 0.026 CHEMBL3544554 | CHEMBL3544532 | |
| 0.041 | 0.022 | 0.044 | VCAM antagonist | 0.044 0.016 CHEMBL3544532 0.041 0.021 CHEMBL3544554 | CHEMBL3544532 | |
| 0.116 | 0.097 | 0.146 | Vanilloid 1 agonist | 0.146 0.043 CHEMBL3544532 0.126 0.073 CHEMBL3544531 0.13 0.065 CHEMBL3544554 | CHEMBL3544532 | |
| 0.035 | 0.017 | 0.049 | Peptide deformylase inhibitor | 0.049 0.01 CHEMBL3544554 | CHEMBL3544554 | |
| 0.076 | 0.059 | 0.131 | Cell adhesion molecule inhibitor | 0.131 0.02 CHEMBL3544532 0.105 0.031 CHEMBL3544554 | CHEMBL3544532 | |
| 0.033 | 0.016 | 0.033 | Bradykinin B2 receptor agonist | 0.026 0.022 CHEMBL3544532 | ||
| 0.022 | 0.006 | 0.025 | Telomerase stimulant | 0.025 0.004 CHEMBL3544532 0.018 0.011 CHEMBL3544531 0.021 0.007 CHEMBL3544554 | CHEMBL3544532 | |
| 0.035 | 0.019 | 0.035 | Somatostatin agonist | |||
| 0.058 | 0.043 | 0.068 | Collagenase 3 inhibitor | 0.068 0.034 CHEMBL3544554 | CHEMBL3544554 | |
| 0.047 | 0.032 | 0.056 | Thymidylate synthase inhibitor | 0.056 0.02 CHEMBL3544532 0.051 0.026 CHEMBL3544531 0.049 0.029 CHEMBL3544554 | CHEMBL3544532 | |
| 0.051 | 0.037 | 0.059 | Carbonic anhydrase II stimulant | 0.059 0.024 CHEMBL3544532 0.051 0.037 CHEMBL3544554 | CHEMBL3544532 | |
| 0.044 | 0.031 | 0.054 | AICAR transformylase inhibitor | 0.054 0.018 CHEMBL3544532 0.044 0.031 CHEMBL3544554 | CHEMBL3544532 | |
| 0.025 | 0.013 | 0.044 | Kainate receptor 1 antagonist | 0.044 0.006 CHEMBL3544532 0.023 0.013 CHEMBL3544554 | CHEMBL3544532 | |
| 0.035 | 0.023 | 0.052 | Calcitonin receptor agonist | 0.052 0.016 CHEMBL3544532 0.032 0.025 CHEMBL3544531 0.032 0.025 CHEMBL3544554 | CHEMBL3544532 | |
| 0.087 | 0.076 | 0.087 | Xanthine oxidase inhibitor | |||
| 0.074 | 0.063 | 0.074 | Interferon agonist | 0.073 0.065 CHEMBL3544532 | ||
| 0.026 | 0.016 | 0.027 | Lysophosphatidic acid receptor 1 agonist | 0.027 0.014 CHEMBL3544532 0.025 0.017 CHEMBL3544554 | CHEMBL3544532 | |
| 0.037 | 0.027 | 0.047 | Carbonic anhydrase I stimulant | 0.047 0.018 CHEMBL3544532 0.035 0.029 CHEMBL3544554 | CHEMBL3544532 | |
| 0.094 | 0.085 | 0.186 | Nav1.4 sodium channel blocker | 0.186 0.022 CHEMBL3544532 0.16 0.03 CHEMBL3544531 0.185 0.023 CHEMBL3544554 | CHEMBL3544532 | |
| 0.053 | 0.044 | 0.055 | Immunoglobulin Fc receptor antagonist | 0.055 0.037 CHEMBL3544532 | CHEMBL3544532 | |
| 0.026 | 0.017 | 0.03 | Vanilloid 2 agonist | 0.03 0.01 CHEMBL3544532 0.024 0.021 CHEMBL3544554 | CHEMBL3544532 | |
| 0.022 | 0.013 | 0.022 | Geranylgeranyltransferase I inhibitor | |||
| 0.041 | 0.032 | 0.041 | Guanylate cyclase inhibitor | |||
| 0.088 | 0.08 | 0.088 | Urease inhibitor | |||
| 0.023 | 0.015 | 0.023 | Geranylgeranyltransferase inhibitor | |||
| 0.017 | 0.009 | 0.019 | Purinergic P2Y1 agonist | 0.017 0.009 CHEMBL3544532 0.014 0.013 CHEMBL3544531 0.019 0.007 CHEMBL3544554 | CHEMBL3544554 | |
| 0.013 | 0.006 | 0.013 | Carboxypeptidase B2 inhibitor | |||
| 0.017 | 0.011 | 0.022 | Carbonic anhydrase X inhibitor | 0.022 0.007 CHEMBL3544532 0.017 0.011 CHEMBL3544531 0.019 0.009 CHEMBL3544554 | CHEMBL3544532 | |
| 0.017 | 0.011 | 0.022 | Carbonic anhydrase VIII inhibitor | 0.022 0.007 CHEMBL3544532 0.017 0.011 CHEMBL3544531 0.019 0.009 CHEMBL3544554 | CHEMBL3544532 | |
| 0.121 | 0.115 | 0.165 | Thiol protease inhibitor | 0.165 0.058 CHEMBL3544532 0.151 0.068 CHEMBL3544531 0.146 0.073 CHEMBL3544554 | CHEMBL3544532 | |
| 0.028 | 0.022 | 0.039 | AMPA 2 receptor antagonist | 0.039 0.015 CHEMBL3544532 0.028 0.022 CHEMBL3544554 | CHEMBL3544532 | |
| 0.022 | 0.017 | 0.027 | Isoleucine-tRNA ligase inhibitor | 0.026 0.009 CHEMBL3544532 0.021 0.019 CHEMBL3544531 0.027 0.008 CHEMBL3544554 | CHEMBL3544554 | |
| 0.046 | 0.041 | 0.06 | Cytokine production stimulant | 0.047 0.037 CHEMBL3544532 0.06 0.013 CHEMBL3544554 | CHEMBL3544554 | |
| 0.068 | 0.064 | 0.08 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.08 0.038 CHEMBL3544532 0.072 0.055 CHEMBL3544554 | CHEMBL3544532 | |
| 0.109 | 0.106 | 0.202 | Histone deacetylase SIRT1 inhibitor | 0.129 0.081 CHEMBL3544532 0.202 0.029 CHEMBL3544554 | CHEMBL3544554 | |
| 0.029 | 0.026 | 0.05 | Prostacyclin antagonist | 0.048 0.014 CHEMBL3544532 0.05 0.013 CHEMBL3544554 | CHEMBL3544554 | |
| 0.037 | 0.035 | 0.048 | Oxytocin agonist | 0.048 0.025 CHEMBL3544532 | CHEMBL3544532 | |
| 0.086 | 0.085 | 0.101 | Bile acid receptor antagonist | 0.101 0.047 CHEMBL3544532 | CHEMBL3544532 | |
| 0.012 | 0.011 | 0.013 | Lysophosphatidic acid receptor 3 agonist | 0.013 0.01 CHEMBL3544532 0.012 0.011 CHEMBL3544554 | CHEMBL3544532 | |
| 0.029 | 0.028 | 0.05 | Dipeptidyl peptidase II inhibitor | 0.038 0.016 CHEMBL3544532 0.05 0.009 CHEMBL3544554 | CHEMBL3544554 | |
| 0.025 | 0.024 | 0.038 | AMPA 3 receptor antagonist | 0.038 0.015 CHEMBL3544532 | CHEMBL3544532 | |
| 0.133 | 0.133 | 0.263 | Psychostimulant | 0.263 0.054 CHEMBL3544532 0.184 0.09 CHEMBL3544554 | CHEMBL3544532 | |
| 0.027 | 0.027 | 0.034 | Caspase 2 inhibitor | 0.034 0.02 CHEMBL3544532 | CHEMBL3544532 | |
| 0.017 | 0.017 | 0.019 | Methylmalonyl-CoA mutase inhibitor | 0.019 0.012 CHEMBL3544532 0.017 0.016 CHEMBL3544531 0.017 0.016 CHEMBL3544554 | CHEMBL3544532 | |
| 0.025 | 0.027 | 0.027 | Baculoviral IAP repeat-containing protein 4 inhibitor | 0.027 0.019 CHEMBL3544532 | CHEMBL3544532 | |
| 0.116 | 0.118 | 0.373 | Anticoagulant | 0.367 0.019 CHEMBL3544532 0.269 0.034 CHEMBL3544531 0.373 0.019 CHEMBL3544554 | CHEMBL3544554 | |
| 0.014 | 0.018 | 0.019 | Kainate receptor 3 antagonist | 0.019 0.01 CHEMBL3544532 | CHEMBL3544532 | |
| 0.018 | 0.023 | 0.022 | Neuraminidase (Influenza B) inhibitor | 0.022 0.013 CHEMBL3544532 | CHEMBL3544532 | |
| 0.128 | 0.133 | 0.151 | Heat shock protein 70 antagonist | 0.142 0.069 CHEMBL3544532 0.151 0.043 CHEMBL3544554 | CHEMBL3544554 | |
| 0.031 | 0.036 | 0.032 | Growth factor receptor-bound protein 2 antagonist | 0.032 0.031 CHEMBL3544554 | CHEMBL3544554 | |
| 0.021 | 0.028 | 0.052 | Urotensin II agonist | 0.052 0.006 CHEMBL3544532 0.034 0.012 CHEMBL3544531 | CHEMBL3544532 | |
| 0.051 | 0.06 | 0.057 | Purinergic P2X1 antagonist | 0.057 0.048 CHEMBL3544532 | CHEMBL3544532 | |
| 0.015 | 0.024 | 0.019 | Integrin alphaVbeta1 antagonist | 0.019 0.013 CHEMBL3544532 | CHEMBL3544532 | |
| 0.034 | 0.045 | 0.042 | NMDA receptor subunit 3B antagonist | 0.042 0.032 CHEMBL3544532 | CHEMBL3544532 | |
| 0.014 | 0.025 | 0.022 | Kainate receptor 5 antagonist | 0.022 0.014 CHEMBL3544532 | CHEMBL3544532 | |
| 0.028 | 0.04 | 0.032 | p53 inhibitor | 0.032 0.029 CHEMBL3544554 | CHEMBL3544554 | |
| 0.041 | 0.053 | 0.048 | Bombesin 2 receptor antagonist | 0.048 0.036 CHEMBL3544532 0.046 0.039 CHEMBL3544554 | CHEMBL3544532 | |
| 0.016 | 0.028 | 0.022 | Integrin alphaVbeta3 antagonist | 0.022 0.015 CHEMBL3544532 | CHEMBL3544532 | |
| 0.02 | 0.034 | 0.026 | Thyroid hormone agonist | 0.026 0.018 CHEMBL3544532 | CHEMBL3544532 | |
| 0.029 | 0.043 | 0.042 | Cholecystokinin B agonist | 0.037 0.026 CHEMBL3544532 0.042 0.021 CHEMBL3544554 | CHEMBL3544554 | |
| 0.027 | 0.041 | 0.039 | NMDA receptor subunit 3A antagonist | 0.039 0.026 CHEMBL3544532 | CHEMBL3544532 | |
| 0.06 | 0.073 | 0.073 | Exportin-1 inhibitor | 0.073 0.037 CHEMBL3544532 0.065 0.055 CHEMBL3544554 | CHEMBL3544532 | |
| 0.014 | 0.029 | 0.027 | Integrin beta5 antagonist | 0.027 0.01 CHEMBL3544532 | CHEMBL3544532 | |
| 0.048 | 0.065 | 0.061 | NMDA 2C receptor antagonist | 0.061 0.044 CHEMBL3544532 | CHEMBL3544532 | |
| 0.022 | 0.039 | 0.027 | Purinergic P2Y15 antagonist | 0.027 0.024 CHEMBL3544532 | CHEMBL3544532 | |
| 0.012 | 0.029 | 0.019 | Integrin beta3 antagonist | 0.019 0.014 CHEMBL3544532 | CHEMBL3544532 | |
| 0.03 | 0.047 | 0.039 | Dopamine D5 agonist | 0.039 0.03 CHEMBL3544532 | CHEMBL3544532 | |
| 0.052 | 0.069 | 0.063 | Caspase 9 inhibitor | 0.06 0.047 CHEMBL3544532 0.063 0.041 CHEMBL3544554 | CHEMBL3544554 | |
| 0.091 | 0.108 | 0.135 | Microtubule formation inhibitor | 0.135 0.047 CHEMBL3544532 0.135 0.046 CHEMBL3544531 0.116 0.065 CHEMBL3544554 | CHEMBL3544531 | |
| 0.113 | 0.131 | 0.159 | Hemostatic | 0.159 0.058 CHEMBL3544532 0.13 0.096 CHEMBL3544554 | CHEMBL3544532 | |
| 0.119 | 0.138 | 0.139 | Melanin inhibitor | 0.139 0.099 CHEMBL3544532 | CHEMBL3544532 | |
| 0.025 | 0.045 | 0.067 | Somatostatin 1 antagonist | 0.067 0.012 CHEMBL3544532 0.052 0.019 CHEMBL3544531 | CHEMBL3544532 | |
| 0.026 | 0.048 | 0.031 | Angiotensin II receptor antagonist | 0.031 0.03 CHEMBL3544554 | CHEMBL3544554 | |
| 0.073 | 0.095 | 0.09 | D-Ala-D-Ala ligase inhibitor | 0.082 0.062 CHEMBL3544532 0.09 0.045 CHEMBL3544554 | CHEMBL3544554 | |
| 0.059 | 0.082 | 0.128 | Analgesic, opioid | 0.128 0.02 CHEMBL3544531 | CHEMBL3544531 | |
| 0.012 | 0.035 | 0.025 | Human T-cell leukemia virus type I protease inhibitor | 0.025 0.011 CHEMBL3544554 | CHEMBL3544554 | |
| 0.107 | 0.132 | 0.132 | Sphingosine 1-phosphate receptor 2 antagonist | 0.132 0.07 CHEMBL3544532 0.116 0.107 CHEMBL3544554 | CHEMBL3544532 | |
| 0.027 | 0.053 | 0.064 | Erythropoietin receptor agonist | 0.058 0.018 CHEMBL3544532 0.043 0.026 CHEMBL3544531 0.064 0.016 CHEMBL3544554 | CHEMBL3544554 | |
| 0.06 | 0.086 | 0.067 | Peroxisome proliferator-activated receptor gamma antagonist | 0.067 0.062 CHEMBL3544532 0.066 0.063 CHEMBL3544554 | CHEMBL3544532 | |
| 0.05 | 0.078 | 0.072 | Protease 3C (Human rhinovirus) inhibitor | 0.072 0.035 CHEMBL3544532 0.072 0.034 CHEMBL3544554 | CHEMBL3544554 | |
| 0.012 | 0.04 | 0.025 | AMPA 1 receptor antagonist | 0.025 0.024 CHEMBL3544532 | CHEMBL3544532 | |
| 0.171 | 0.201 | 0.234 | Immunomodulator | 0.234 0.128 CHEMBL3544531 | CHEMBL3544531 | |
| 0.18 | 0.211 | 0.267 | Apoptosis antagonist | 0.267 0.112 CHEMBL3544532 0.195 0.186 CHEMBL3544531 | CHEMBL3544532 | |
| 0.003 | 0.036 | 0.01 | Neurokinin 3 agonist | 0.01 0.009 CHEMBL3544554 | CHEMBL3544554 | |
| 0.051 | 0.084 | 0.069 | Na+ K+ transporting ATPase inhibitor | 0.069 0.061 CHEMBL3544532 | CHEMBL3544532 | |
| 0.052 | 0.086 | 0.096 | Cathepsin G inhibitor | 0.096 0.035 CHEMBL3544532 | CHEMBL3544532 | |
| 0.014 | 0.048 | 0.028 | Somatostatin 4 antagonist | 0.028 0.013 CHEMBL3544532 | CHEMBL3544532 | |
| 0.017 | 0.054 | 0.034 | Calcium-sensing receptor agonist | 0.026 0.019 CHEMBL3544532 0.034 0.01 CHEMBL3544531 | CHEMBL3544531 | |
| 0.026 | 0.063 | 0.042 | Glycine transporter 2 inhibitor | 0.042 0.036 CHEMBL3544532 0.04 0.038 CHEMBL3544554 | CHEMBL3544532 | |
| 0.071 | 0.108 | 0.079 | Estrogen-related receptor beta agonist | 0.079 0.071 CHEMBL3544532 | CHEMBL3544532 | |
| 0.24 | 0.279 | 0.7 | Antiinflammatory | 0.7 0.031 CHEMBL3544532 0.686 0.033 CHEMBL3544531 | CHEMBL3544532 | |
| 0.088 | 0.133 | 0.172 | Lipid peroxidase inhibitor | 0.11 0.104 CHEMBL3544532 0.172 0.054 CHEMBL3544531 | CHEMBL3544531 | |
| 0.025 | 0.071 | 0.053 | NMDA 2A receptor antagonist | 0.044 0.043 CHEMBL3544532 0.053 0.035 CHEMBL3544554 | CHEMBL3544554 | |
| 0.01 | 0.058 | 0.051 | Somatostatin 5 antagonist | 0.051 0.013 CHEMBL3544532 0.03 0.023 CHEMBL3544531 | CHEMBL3544532 | |
| 0.162 | 0.211 | 0.284 | Transcription factor NF kappa B inhibitor | 0.202 0.167 CHEMBL3544532 0.284 0.104 CHEMBL3544531 | CHEMBL3544531 | |
| 0.041 | 0.092 | 0.06 | DNA helicase inhibitor | 0.06 0.028 CHEMBL3544531 | CHEMBL3544531 | |
| 0.056 | 0.111 | 0.074 | Glycine receptor antagonist | 0.074 0.068 CHEMBL3544532 | CHEMBL3544532 | |
| 0.009 | 0.067 | 0.046 | Somatostatin 2 antagonist | 0.046 0.016 CHEMBL3544532 0.046 0.016 CHEMBL3544531 | CHEMBL3544531 | |
| 0.108 | 0.168 | 0.236 | Anesthetic general | 0.229 0.06 CHEMBL3544532 0.181 0.086 CHEMBL3544531 0.236 0.057 CHEMBL3544554 | CHEMBL3544554 | |
| 0.03 | 0.091 | 0.077 | Maillard reaction inhibitor | 0.077 0.026 CHEMBL3544532 | CHEMBL3544532 | |
| 0.012 | 0.075 | 0.035 | Endothelial nitric-oxide synthase inhibitor | 0.035 0.017 CHEMBL3544554 | CHEMBL3544554 | |
| 0.239 | 0.306 | 0.293 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.293 0.223 CHEMBL3544532 | CHEMBL3544532 | |
| 0.103 | 0.17 | 0.127 | GABA C receptor rho-2 antagonist | 0.127 0.112 CHEMBL3544532 | CHEMBL3544532 | |
| 0.031 | 0.1 | 0.067 | Dipeptidyl peptidase IV inhibitor | 0.067 0.01 CHEMBL3544532 0.065 0.011 CHEMBL3544531 0.046 0.026 CHEMBL3544554 | CHEMBL3544532 | |
| 0.089 | 0.159 | 0.112 | Sphingosine 1-phosphate receptor 4 antagonist | 0.112 0.089 CHEMBL3544532 0.11 0.093 CHEMBL3544554 | CHEMBL3544532 | |
| 0.153 | 0.222 | 0.178 | Neuropeptide Y2 antagonist | 0.178 0.165 CHEMBL3544532 | CHEMBL3544532 | |
| 0.024 | 0.097 | 0.058 | Neurokinin 2 agonist | 0.058 0.014 CHEMBL3544554 | CHEMBL3544554 | |
| 0.019 | 0.095 | 0.055 | HIV-1 protease inhibitor | 0.055 0.016 CHEMBL3544554 | CHEMBL3544554 | |
| 0.156 | 0.233 | 0.233 | Vasodilator, peripheral | 0.233 0.141 CHEMBL3544532 0.212 0.163 CHEMBL3544554 | CHEMBL3544532 | |
| 0.034 | 0.12 | 0.074 | Dipeptidyl peptidase inhibitor | 0.074 0.016 CHEMBL3544532 0.07 0.018 CHEMBL3544531 0.054 0.034 CHEMBL3544554 | CHEMBL3544532 | |
| 0.048 | 0.134 | 0.089 | Histamine N-methyltransferase inhibitor | 0.089 0.057 CHEMBL3544554 | CHEMBL3544554 | |
| 0.018 | 0.107 | 0.039 | Angiotensin AT1 receptor antagonist | 0.039 0.036 CHEMBL3544554 | CHEMBL3544554 | |
| 0.156 | 0.257 | 0.256 | Sodium/bile acid cotransporter inhibitor | 0.213 0.171 CHEMBL3544532 0.256 0.122 CHEMBL3544554 | CHEMBL3544554 | |
| 0.144 | 0.249 | 0.17 | 5 Hydroxytryptamine 3E antagonist | 0.17 0.137 CHEMBL3544554 | CHEMBL3544554 | |
| 0.106 | 0.222 | 0.147 | Neurotrophic factor enhancer | 0.147 0.142 CHEMBL3544554 | CHEMBL3544554 | |
| 0.016 | 0.134 | 0.034 | Somatostatin 5 agonist | 0.034 0.025 CHEMBL3544532 | CHEMBL3544532 | |
| 0.039 | 0.177 | 0.054 | Lipocortins synthesis agonist | 0.054 0.051 CHEMBL3544554 | CHEMBL3544554 | |
| 0.02 | 0.182 | 0.048 | Microtubule stabilization | 0.048 0.031 CHEMBL3544531 | CHEMBL3544531 | |
| 0.101 | 0.276 | 0.212 | DNA damaging | 0.212 0.106 CHEMBL3544532 0.189 0.125 CHEMBL3544531 | CHEMBL3544532 | |
| 0.032 | 0.218 | 0.067 | Secretase beta inhibitor | 0.067 0.056 CHEMBL3544554 | CHEMBL3544554 | |
| 0.018 | 0.205 | 0.078 | Baculoviral IAP repeat-containing protein inhibitor | 0.078 0.004 CHEMBL3544554 | CHEMBL3544554 | |
| 0.025 | 0.226 | 0.071 | Bombesin 1 receptor agonist | 0.071 0.031 CHEMBL3544554 | CHEMBL3544554 | |
| 0.043 | 0.252 | 0.126 | Histone deacetylase class III inhibitor | 0.126 0.065 CHEMBL3544554 | CHEMBL3544554 | |
| 0.042 | 0.262 | 0.145 | Thioredoxin inhibitor | 0.145 0.018 CHEMBL3544532 0.109 0.039 CHEMBL3544531 | CHEMBL3544532 | |
| 0.072 | 0.291 | 0.144 | Insulin secretagoues | 0.144 0.081 CHEMBL3544554 | CHEMBL3544554 | |
| 0.067 | 0.295 | 0.195 | Platelet adhesion inhibitor | 0.195 0.074 CHEMBL3544532 | CHEMBL3544532 | |
| 0.023 | 0.263 | 0.066 | Thrombin inhibitor | 0.066 0.061 CHEMBL3544554 | CHEMBL3544554 | |
| 0.135 | 0.39 | 0.714 | Apoptosis agonist | 0.284 0.184 CHEMBL3544532 0.366 0.13 CHEMBL3544531 0.714 0.028 CHEMBL3544554 | CHEMBL3544554 | |
| 0.015 | 0.271 | 0.027 | Vasopressin 1A agonist | 0.027 0.025 CHEMBL3544532 | CHEMBL3544532 | |
| 0.063 | 0.348 | 0.153 | Non-steroidal antiinflammatory agent | 0.153 0.111 CHEMBL3544554 | CHEMBL3544554 | |
| 0.008 | 0.318 | 0.051 | Baculoviral IAP repeat-containing protein 3 inhibitor | 0.051 0.003 CHEMBL3544554 | CHEMBL3544554 | |
| 0.086 | 0.466 | 0.278 | Analgesic | 0.278 0.159 CHEMBL3544531 | CHEMBL3544531 | |
| 0.004 | 0.555 | 0.326 | Beta tubulin antagonist | 0.326 0.005 CHEMBL3544554 | CHEMBL3544554 | |
| 0.003 | 0.631 | 0.012 | Baculoviral IAP repeat-containing protein 2 inhibitor | 0.012 0.004 CHEMBL3544554 | CHEMBL3544554 | |
| 0.005 | 0.879 | 0.155 | Tubulin antagonist | 0.155 0.056 CHEMBL3544554 | CHEMBL3544554 | |
| 0.005 | 0.901 | 0.576 | Tumour necrosis factor alpha release inhibitor | 0.557 0.01 CHEMBL3544532 0.576 0.009 CHEMBL3544531 | CHEMBL3544531 | |
| 0.01 | 0.92 | 0.184 | ErbB-3 antagonist | 0.184 0.012 CHEMBL3544531 | CHEMBL3544531 | |
| 0.019 | 0.952 | 0.154 | NOS3 expression enhancer | 0.154 0.068 CHEMBL3544531 | CHEMBL3544531 | |
| 0.004 | 0.959 | 0.409 | Antimitotic | 0.409 0.022 CHEMBL3544531 | CHEMBL3544531 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |