Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.5430.0050.819Lck kinase inhibitor

0.637 0.004 CHEMBL3544873

0.819 0.003 CHEMBL244377

0.475 0.005 CHEMBL3544874

0.744 0.004 CHEMBL3544897

0.744 0.004 CHEMBL3544898

0.769 0.003 CHEMBL1231106

0.69 0.004 CHEMBL457723

0.69 0.004 CHEMBL3544872

CHEMBL244377
0.5420.0160.615GABA C receptor rho-3 antagonist

0.399 0.062 CHEMBL3544873

0.543 0.016 CHEMBL244377

0.507 0.024 CHEMBL3544874

0.506 0.024 CHEMBL3544897

0.506 0.024 CHEMBL3544898

0.615 0.006 CHEMBL1231106

0.443 0.044 CHEMBL457723

0.443 0.044 CHEMBL3544872

CHEMBL1231106
0.5370.020.586Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.452 0.06 CHEMBL3544873

0.586 0.009 CHEMBL244377

0.464 0.052 CHEMBL3544874

0.518 0.026 CHEMBL3544897

0.518 0.026 CHEMBL3544898

0.517 0.026 CHEMBL1231106

0.529 0.022 CHEMBL457723

0.529 0.022 CHEMBL3544872

CHEMBL244377
0.5140.0040.658Protein-tyrosine kinase Lyn inhibitor

0.419 0.006 CHEMBL3544873

0.532 0.004 CHEMBL244377

0.45 0.005 CHEMBL3544874

0.487 0.005 CHEMBL3544897

0.487 0.005 CHEMBL3544898

0.658 0.003 CHEMBL1231106

0.442 0.005 CHEMBL457723

0.442 0.005 CHEMBL3544872

CHEMBL1231106
0.510.0310.51Cholesterol antagonist

0.251 0.124 CHEMBL3544873

0.285 0.101 CHEMBL244377

0.342 0.068 CHEMBL3544874

0.184 0.18 CHEMBL3544897

0.184 0.18 CHEMBL3544898

0.271 0.111 CHEMBL1231106

0.346 0.066 CHEMBL457723

0.346 0.066 CHEMBL3544872

0.4420.0180.503DNA synthesis inhibitor

0.442 0.018 CHEMBL3544873

0.327 0.036 CHEMBL244377

0.503 0.013 CHEMBL3544874

0.385 0.024 CHEMBL3544897

0.385 0.024 CHEMBL3544898

0.448 0.017 CHEMBL1231106

0.38 0.024 CHEMBL457723

0.38 0.024 CHEMBL3544872

CHEMBL3544874
0.460.0390.46Aldehyde oxidase inhibitor

0.366 0.052 CHEMBL244377

0.249 0.082 CHEMBL3544874

0.2 0.104 CHEMBL3544897

0.2 0.104 CHEMBL3544898

0.432 0.042 CHEMBL1231106

0.186 0.113 CHEMBL457723

0.186 0.113 CHEMBL3544872

0.4170.0030.417Toll-Like receptor 7 antagonist

0.156 0.005 CHEMBL3544873

0.245 0.004 CHEMBL3544874

0.201 0.004 CHEMBL457723

0.201 0.004 CHEMBL3544872

0.4180.0040.439Catenin beta inhibitor

0.338 0.005 CHEMBL3544873

0.255 0.01 CHEMBL244377

0.263 0.009 CHEMBL3544874

0.175 0.058 CHEMBL3544897

0.175 0.058 CHEMBL3544898

0.439 0.004 CHEMBL457723

0.439 0.004 CHEMBL3544872

CHEMBL3544872
0.4580.0480.5515 Hydroxytryptamine release inhibitor

0.406 0.074 CHEMBL3544873

0.503 0.031 CHEMBL244377

0.443 0.055 CHEMBL3544874

0.482 0.038 CHEMBL3544897

0.482 0.038 CHEMBL3544898

0.551 0.019 CHEMBL1231106

0.427 0.062 CHEMBL457723

0.427 0.062 CHEMBL3544872

CHEMBL1231106
0.4490.0510.525Histamine release inhibitor

0.383 0.084 CHEMBL3544873

0.468 0.042 CHEMBL244377

0.453 0.049 CHEMBL3544874

0.471 0.04 CHEMBL3544897

0.471 0.04 CHEMBL3544898

0.525 0.021 CHEMBL1231106

0.378 0.087 CHEMBL457723

0.378 0.087 CHEMBL3544872

CHEMBL1231106
0.390.0050.39Cell adhesion inhibitor

0.149 0.047 CHEMBL3544874

0.155 0.043 CHEMBL457723

0.155 0.043 CHEMBL3544872

0.3940.0090.443Alpha-N-acetylglucosaminidase inhibitor

0.182 0.04 CHEMBL3544873

0.435 0.007 CHEMBL244377

0.248 0.023 CHEMBL3544874

0.276 0.019 CHEMBL3544897

0.276 0.019 CHEMBL3544898

0.443 0.007 CHEMBL1231106

0.3 0.016 CHEMBL457723

0.3 0.016 CHEMBL3544872

CHEMBL1231106
0.460.0780.502Caspase 9 stimulant

0.502 0.059 CHEMBL244377

0.319 0.174 CHEMBL3544874

0.368 0.132 CHEMBL3544897

0.368 0.132 CHEMBL3544898

0.468 0.074 CHEMBL1231106

0.361 0.137 CHEMBL457723

0.361 0.137 CHEMBL3544872

CHEMBL244377
0.4160.0430.4995 Hydroxytryptamine release stimulant

0.378 0.05 CHEMBL244377

0.312 0.066 CHEMBL3544874

0.271 0.08 CHEMBL3544897

0.271 0.08 CHEMBL3544898

0.499 0.027 CHEMBL1231106

0.209 0.114 CHEMBL457723

0.209 0.114 CHEMBL3544872

CHEMBL1231106
0.4020.0290.402Hypoxia-inducible factor 1 alpha inhibitor

0.285 0.074 CHEMBL3544873

0.221 0.128 CHEMBL244377

0.352 0.044 CHEMBL3544874

0.187 0.168 CHEMBL3544897

0.187 0.168 CHEMBL3544898

0.232 0.117 CHEMBL1231106

0.33 0.052 CHEMBL457723

0.33 0.052 CHEMBL3544872

0.3810.0150.563Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.345 0.021 CHEMBL3544873

0.558 0.004 CHEMBL244377

0.278 0.035 CHEMBL3544874

0.488 0.005 CHEMBL3544897

0.488 0.005 CHEMBL3544898

0.563 0.004 CHEMBL1231106

0.413 0.011 CHEMBL457723

0.413 0.011 CHEMBL3544872

CHEMBL1231106
0.3730.0150.748Src kinase inhibitor

0.483 0.007 CHEMBL3544873

0.748 0.004 CHEMBL244377

0.327 0.021 CHEMBL3544874

0.637 0.005 CHEMBL3544897

0.637 0.005 CHEMBL3544898

0.673 0.004 CHEMBL1231106

0.547 0.005 CHEMBL457723

0.547 0.005 CHEMBL3544872

CHEMBL244377
0.3470.0040.479Tyrosine-protein kinase EMT inhibitor

0.236 0.005 CHEMBL3544873

0.479 0.004 CHEMBL244377

0.189 0.005 CHEMBL3544874

0.332 0.004 CHEMBL3544897

0.332 0.004 CHEMBL3544898

0.384 0.004 CHEMBL1231106

0.338 0.004 CHEMBL457723

0.338 0.004 CHEMBL3544872

CHEMBL244377
0.3430.0050.387Ferrochelatase inhibitor

0.178 0.028 CHEMBL3544873

0.352 0.005 CHEMBL244377

0.268 0.011 CHEMBL3544874

0.274 0.01 CHEMBL3544897

0.274 0.01 CHEMBL3544898

0.387 0.004 CHEMBL1231106

0.258 0.012 CHEMBL457723

0.258 0.012 CHEMBL3544872

CHEMBL1231106
0.3390.0080.339Toll-Like receptor 9 antagonist

0.277 0.016 CHEMBL3544873

0.203 0.034 CHEMBL244377

0.299 0.013 CHEMBL3544874

0.17 0.051 CHEMBL3544897

0.17 0.051 CHEMBL3544898

0.155 0.059 CHEMBL1231106

0.321 0.01 CHEMBL457723

0.321 0.01 CHEMBL3544872

0.3530.0280.592Peroxidase inhibitor

0.23 0.052 CHEMBL3544873

0.368 0.025 CHEMBL244377

0.396 0.021 CHEMBL3544874

0.402 0.02 CHEMBL3544897

0.402 0.02 CHEMBL3544898

0.592 0.005 CHEMBL1231106

0.189 0.062 CHEMBL457723

0.189 0.062 CHEMBL3544872

CHEMBL1231106
0.3580.0460.405Aryl hydrocarbon receptor agonist

0.34 0.05 CHEMBL3544873

0.255 0.077 CHEMBL244377

0.405 0.037 CHEMBL3544874

0.285 0.066 CHEMBL3544897

0.285 0.066 CHEMBL3544898

0.374 0.043 CHEMBL1231106

0.305 0.06 CHEMBL457723

0.305 0.06 CHEMBL3544872

CHEMBL3544874
0.3330.0270.333Anesthetic general

0.155 0.108 CHEMBL3544873

0.234 0.058 CHEMBL244377

0.244 0.053 CHEMBL3544874

0.163 0.1 CHEMBL3544897

0.163 0.1 CHEMBL3544898

0.231 0.059 CHEMBL1231106

0.223 0.063 CHEMBL457723

0.223 0.063 CHEMBL3544872

0.3180.0190.318Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.194 0.077 CHEMBL3544873

0.241 0.047 CHEMBL244377

0.278 0.031 CHEMBL3544874

0.196 0.075 CHEMBL3544897

0.196 0.075 CHEMBL3544898

0.279 0.031 CHEMBL1231106

0.238 0.048 CHEMBL457723

0.238 0.048 CHEMBL3544872

0.3290.0320.3745 Hydroxytryptamine uptake stimulant

0.199 0.154 CHEMBL3544873

0.33 0.032 CHEMBL244377

0.266 0.066 CHEMBL3544874

0.263 0.069 CHEMBL3544897

0.263 0.069 CHEMBL3544898

0.374 0.019 CHEMBL1231106

0.246 0.085 CHEMBL457723

0.246 0.085 CHEMBL3544872

CHEMBL1231106
0.4010.1060.436MAP kinase 1 inhibitor

0.392 0.111 CHEMBL3544873

0.362 0.129 CHEMBL244377

0.355 0.133 CHEMBL3544874

0.317 0.162 CHEMBL3544897

0.317 0.162 CHEMBL3544898

0.297 0.183 CHEMBL1231106

0.436 0.085 CHEMBL457723

0.436 0.085 CHEMBL3544872

CHEMBL3544872
0.2950.0050.295Electron transport complex I inhibitor

0.128 0.037 CHEMBL3544874

0.124 0.041 CHEMBL457723

0.124 0.041 CHEMBL3544872

0.3460.0570.346Vasodilator, coronary

0.248 0.137 CHEMBL3544873

0.305 0.083 CHEMBL244377

0.318 0.073 CHEMBL3544874

0.283 0.102 CHEMBL3544897

0.283 0.102 CHEMBL3544898

0.339 0.061 CHEMBL1231106

0.273 0.112 CHEMBL457723

0.273 0.112 CHEMBL3544872

0.2980.0090.539GABA C receptor agonist

0.173 0.026 CHEMBL3544873

0.319 0.008 CHEMBL244377

0.295 0.01 CHEMBL3544874

0.297 0.01 CHEMBL3544897

0.297 0.01 CHEMBL3544898

0.539 0.003 CHEMBL1231106

0.187 0.023 CHEMBL457723

0.187 0.023 CHEMBL3544872

CHEMBL1231106
0.3560.0690.641Angiogenesis inhibitor

0.51 0.028 CHEMBL3544873

0.641 0.013 CHEMBL244377

0.367 0.064 CHEMBL3544874

0.589 0.018 CHEMBL3544897

0.589 0.018 CHEMBL3544898

0.5 0.03 CHEMBL1231106

0.529 0.025 CHEMBL457723

0.529 0.025 CHEMBL3544872

CHEMBL244377
0.2760.0080.276Telomerase inhibitor

0.189 0.015 CHEMBL3544873

0.249 0.009 CHEMBL244377

0.21 0.013 CHEMBL3544874

0.203 0.013 CHEMBL3544897

0.203 0.013 CHEMBL3544898

0.265 0.008 CHEMBL1231106

0.225 0.012 CHEMBL457723

0.225 0.012 CHEMBL3544872

0.3070.0390.307Cyclic AMP phosphodiesterase inhibitor

0.193 0.099 CHEMBL244377

0.21 0.086 CHEMBL3544874

0.194 0.098 CHEMBL1231106

0.191 0.101 CHEMBL457723

0.191 0.101 CHEMBL3544872

0.3410.0780.412Vasodilator, peripheral

0.318 0.088 CHEMBL244377

0.294 0.1 CHEMBL3544874

0.275 0.111 CHEMBL3544897

0.275 0.111 CHEMBL3544898

0.412 0.052 CHEMBL1231106

0.207 0.169 CHEMBL457723

0.207 0.169 CHEMBL3544872

CHEMBL1231106
0.2980.0340.336Tyrosine 3 hydroxylase inhibitor

0.191 0.153 CHEMBL3544873

0.286 0.041 CHEMBL244377

0.254 0.064 CHEMBL3544874

0.24 0.079 CHEMBL3544897

0.24 0.079 CHEMBL3544898

0.336 0.02 CHEMBL1231106

0.231 0.089 CHEMBL457723

0.231 0.089 CHEMBL3544872

CHEMBL1231106
0.2910.0350.291MAP-kinase-activated kinase 5 inhibitor

0.19 0.117 CHEMBL3544873

0.279 0.042 CHEMBL3544874

0.18 0.131 CHEMBL457723

0.18 0.131 CHEMBL3544872

0.2680.0140.677Platelet activating factor beta antagonist

0.228 0.019 CHEMBL3544873

0.49 0.005 CHEMBL244377

0.238 0.018 CHEMBL3544874

0.425 0.005 CHEMBL3544897

0.425 0.005 CHEMBL3544898

0.677 0.004 CHEMBL1231106

0.229 0.019 CHEMBL457723

0.229 0.019 CHEMBL3544872

CHEMBL1231106
0.2710.0210.35Nitric-oxide synthase stimulant

0.237 0.042 CHEMBL3544873

0.27 0.021 CHEMBL244377

0.282 0.016 CHEMBL3544874

0.277 0.018 CHEMBL3544897

0.277 0.018 CHEMBL3544898

0.35 0.005 CHEMBL1231106

0.23 0.049 CHEMBL457723

0.23 0.049 CHEMBL3544872

CHEMBL1231106
0.2610.0120.2615 Hydroxytryptamine 3E antagonist

0.193 0.074 CHEMBL3544873

0.258 0.013 CHEMBL244377

0.226 0.03 CHEMBL3544874

0.223 0.033 CHEMBL3544897

0.223 0.033 CHEMBL3544898

0.249 0.016 CHEMBL1231106

0.224 0.033 CHEMBL457723

0.224 0.033 CHEMBL3544872

0.2890.0410.293Gastrin inhibitor

0.188 0.167 CHEMBL3544873

0.293 0.038 CHEMBL244377

0.218 0.122 CHEMBL3544874

0.222 0.116 CHEMBL3544897

0.222 0.116 CHEMBL3544898

0.237 0.095 CHEMBL1231106

0.266 0.062 CHEMBL457723

0.266 0.062 CHEMBL3544872

CHEMBL244377
0.3030.0620.522Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.406 0.02 CHEMBL3544873

0.522 0.005 CHEMBL244377

0.34 0.04 CHEMBL3544874

0.505 0.007 CHEMBL3544897

0.505 0.007 CHEMBL3544898

0.506 0.007 CHEMBL1231106

0.403 0.021 CHEMBL457723

0.403 0.021 CHEMBL3544872

CHEMBL244377
0.2550.0160.255Alkylator

0.227 0.02 CHEMBL3544873

0.189 0.03 CHEMBL244377

0.245 0.017 CHEMBL3544874

0.182 0.032 CHEMBL3544897

0.182 0.032 CHEMBL3544898

0.179 0.033 CHEMBL1231106

0.235 0.018 CHEMBL457723

0.235 0.018 CHEMBL3544872

0.2460.0160.246Toll-Like receptor antagonist

0.168 0.044 CHEMBL3544873

0.116 0.091 CHEMBL244377

0.216 0.025 CHEMBL3544874

0.114 0.094 CHEMBL1231106

0.2 0.03 CHEMBL457723

0.2 0.03 CHEMBL3544872

0.2580.0280.258Tumour necrosis factor antagonist

0.208 0.049 CHEMBL3544873

0.19 0.059 CHEMBL244377

0.252 0.03 CHEMBL3544874

0.187 0.062 CHEMBL3544897

0.187 0.062 CHEMBL3544898

0.237 0.035 CHEMBL1231106

0.212 0.047 CHEMBL457723

0.212 0.047 CHEMBL3544872

0.2910.0670.291Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.159 0.132 CHEMBL3544873

0.23 0.085 CHEMBL244377

0.211 0.094 CHEMBL3544874

0.175 0.117 CHEMBL3544897

0.175 0.117 CHEMBL3544898

0.238 0.082 CHEMBL1231106

0.205 0.097 CHEMBL457723

0.205 0.097 CHEMBL3544872

0.3070.0840.362Calcium channel activator

0.338 0.058 CHEMBL244377

0.255 0.141 CHEMBL3544874

0.287 0.106 CHEMBL3544897

0.287 0.106 CHEMBL3544898

0.362 0.042 CHEMBL1231106

0.249 0.149 CHEMBL457723

0.249 0.149 CHEMBL3544872

CHEMBL1231106
0.2640.0420.45RNA-directed DNA polymerase inhibitor

0.277 0.037 CHEMBL3544873

0.284 0.035 CHEMBL244377

0.349 0.024 CHEMBL3544874

0.374 0.021 CHEMBL3544897

0.374 0.021 CHEMBL3544898

0.45 0.014 CHEMBL1231106

0.226 0.068 CHEMBL457723

0.226 0.068 CHEMBL3544872

CHEMBL1231106
0.2870.0670.294Insulysin inhibitor

0.291 0.064 CHEMBL244377

0.234 0.113 CHEMBL3544874

0.239 0.107 CHEMBL3544897

0.239 0.107 CHEMBL3544898

0.294 0.062 CHEMBL1231106

0.233 0.114 CHEMBL457723

0.233 0.114 CHEMBL3544872

CHEMBL1231106
0.2320.0160.264GABA C receptor rho-2 antagonist

0.15 0.074 CHEMBL3544873

0.24 0.014 CHEMBL244377

0.201 0.028 CHEMBL3544874

0.205 0.026 CHEMBL3544897

0.205 0.026 CHEMBL3544898

0.264 0.009 CHEMBL1231106

0.178 0.044 CHEMBL457723

0.178 0.044 CHEMBL3544872

CHEMBL1231106
0.2590.0480.259Neuropeptide Y2 antagonist

0.2 0.119 CHEMBL244377

0.207 0.107 CHEMBL3544874

0.194 0.131 CHEMBL1231106

0.22 0.089 CHEMBL457723

0.22 0.089 CHEMBL3544872

0.2220.0120.348CF transmembrane conductance regulator agonist

0.237 0.008 CHEMBL3544873

0.348 0.003 CHEMBL244377

0.193 0.026 CHEMBL3544874

0.287 0.004 CHEMBL3544897

0.287 0.004 CHEMBL3544898

0.23 0.01 CHEMBL1231106

0.277 0.005 CHEMBL457723

0.277 0.005 CHEMBL3544872

CHEMBL244377
0.2140.0080.4MAP kinase 11 inhibitor

0.307 0.005 CHEMBL3544873

0.359 0.004 CHEMBL244377

0.149 0.018 CHEMBL3544874

0.255 0.005 CHEMBL3544897

0.255 0.005 CHEMBL3544898

0.4 0.004 CHEMBL457723

0.4 0.004 CHEMBL3544872

CHEMBL3544872
0.2130.0080.864AXL receptor tyrosine kinase inhibitor

0.589 0.004 CHEMBL3544873

0.864 0.003 CHEMBL244377

0.281 0.005 CHEMBL3544874

0.834 0.003 CHEMBL3544897

0.834 0.003 CHEMBL3544898

0.857 0.003 CHEMBL1231106

0.582 0.004 CHEMBL457723

0.582 0.004 CHEMBL3544872

CHEMBL244377
0.2250.0220.233ATPase inhibitor

0.148 0.105 CHEMBL3544873

0.188 0.048 CHEMBL244377

0.207 0.032 CHEMBL3544874

0.173 0.066 CHEMBL3544897

0.173 0.066 CHEMBL3544898

0.233 0.018 CHEMBL1231106

0.164 0.079 CHEMBL457723

0.164 0.079 CHEMBL3544872

CHEMBL1231106
0.3210.1170.32115-Lipoxygenase inhibitor

0.208 0.205 CHEMBL244377

0.236 0.177 CHEMBL3544874

0.241 0.172 CHEMBL457723

0.241 0.172 CHEMBL3544872

0.2710.070.271DNA damaging

0.192 0.122 CHEMBL244377

0.251 0.08 CHEMBL3544874

0.178 0.136 CHEMBL3544897

0.178 0.136 CHEMBL3544898

0.265 0.072 CHEMBL1231106

0.17 0.145 CHEMBL457723

0.17 0.145 CHEMBL3544872

0.2650.0660.378Superoxide dismutase inhibitor

0.254 0.072 CHEMBL244377

0.21 0.107 CHEMBL3544874

0.199 0.119 CHEMBL3544897

0.199 0.119 CHEMBL3544898

0.378 0.031 CHEMBL1231106

0.174 0.15 CHEMBL457723

0.174 0.15 CHEMBL3544872

CHEMBL1231106
0.2080.0090.787Folate antagonist

0.29 0.004 CHEMBL3544873

0.161 0.019 CHEMBL244377

0.367 0.003 CHEMBL3544874

0.333 0.003 CHEMBL3544897

0.333 0.003 CHEMBL3544898

0.787 0.001 CHEMBL1231106

0.136 0.028 CHEMBL457723

0.136 0.028 CHEMBL3544872

CHEMBL1231106
0.2530.0570.253Amyloid beta aggregation inhibitor

0.165 0.098 CHEMBL457723

0.165 0.098 CHEMBL3544872

0.2130.0220.233Epidermal growth factor receptor kinase inhibitor

0.148 0.049 CHEMBL3544873

0.214 0.022 CHEMBL244377

0.159 0.043 CHEMBL3544874

0.17 0.037 CHEMBL3544897

0.17 0.037 CHEMBL3544898

0.233 0.018 CHEMBL1231106

0.176 0.034 CHEMBL457723

0.176 0.034 CHEMBL3544872

CHEMBL1231106
0.3120.1260.354Antibacterial

0.295 0.14 CHEMBL3544873

0.259 0.169 CHEMBL244377

0.348 0.103 CHEMBL3544874

0.299 0.136 CHEMBL3544897

0.299 0.136 CHEMBL3544898

0.354 0.1 CHEMBL1231106

0.254 0.173 CHEMBL457723

0.254 0.173 CHEMBL3544872

CHEMBL1231106
0.2130.0290.334Cyclin-dependent kinase 7 inhibitor

0.212 0.03 CHEMBL3544873

0.334 0.008 CHEMBL244377

0.188 0.038 CHEMBL3544874

0.291 0.014 CHEMBL3544897

0.291 0.014 CHEMBL3544898

0.323 0.009 CHEMBL1231106

0.234 0.024 CHEMBL457723

0.234 0.024 CHEMBL3544872

CHEMBL244377
0.240.0580.243Peptidyltransferase inhibitor

0.222 0.074 CHEMBL3544873

0.243 0.056 CHEMBL244377

0.218 0.078 CHEMBL3544874

0.216 0.08 CHEMBL3544897

0.216 0.08 CHEMBL3544898

0.243 0.056 CHEMBL457723

0.243 0.056 CHEMBL3544872

CHEMBL3544872
0.2170.0350.217Lipid peroxidase inhibitor

0.12 0.094 CHEMBL3544874

0.127 0.087 CHEMBL457723

0.127 0.087 CHEMBL3544872

0.2180.0360.25Succinate dehydrogenase inhibitor

0.209 0.042 CHEMBL244377

0.175 0.074 CHEMBL3544874

0.17 0.081 CHEMBL3544897

0.17 0.081 CHEMBL3544898

0.25 0.022 CHEMBL1231106

0.163 0.09 CHEMBL457723

0.163 0.09 CHEMBL3544872

CHEMBL1231106
0.1930.0160.271Adenylate kinase inhibitor

0.113 0.05 CHEMBL3544873

0.163 0.022 CHEMBL244377

0.176 0.019 CHEMBL3544874

0.149 0.027 CHEMBL3544897

0.149 0.027 CHEMBL3544898

0.271 0.009 CHEMBL1231106

0.122 0.042 CHEMBL457723

0.122 0.042 CHEMBL3544872

CHEMBL1231106
0.210.0330.363Cytokine production inhibitor

0.363 0.009 CHEMBL3544873

0.314 0.013 CHEMBL244377

0.238 0.026 CHEMBL3544874

0.343 0.01 CHEMBL3544897

0.343 0.01 CHEMBL3544898

0.205 0.034 CHEMBL1231106

0.336 0.011 CHEMBL457723

0.336 0.011 CHEMBL3544872

CHEMBL3544873
0.2330.0580.705Tyrosine kinase inhibitor

0.332 0.037 CHEMBL3544873

0.705 0.006 CHEMBL244377

0.188 0.073 CHEMBL3544874

0.542 0.014 CHEMBL3544897

0.542 0.014 CHEMBL3544898

0.535 0.015 CHEMBL1231106

0.409 0.027 CHEMBL457723

0.409 0.027 CHEMBL3544872

CHEMBL244377
0.1880.0160.279GABA C receptor antagonist

0.139 0.037 CHEMBL3544873

0.233 0.008 CHEMBL244377

0.178 0.018 CHEMBL3544874

0.214 0.01 CHEMBL3544897

0.214 0.01 CHEMBL3544898

0.279 0.005 CHEMBL1231106

0.152 0.029 CHEMBL457723

0.152 0.029 CHEMBL3544872

CHEMBL1231106
0.1870.0150.187Nav1.5 sodium channel blocker

0.138 0.036 CHEMBL3544873

0.125 0.048 CHEMBL244377

0.164 0.021 CHEMBL3544874

0.112 0.066 CHEMBL3544897

0.112 0.066 CHEMBL3544898

0.136 0.037 CHEMBL1231106

0.152 0.025 CHEMBL457723

0.152 0.025 CHEMBL3544872

0.1860.0170.974TIE antagonist

0.85 0.003 CHEMBL3544873

0.974 0.002 CHEMBL244377

0.304 0.008 CHEMBL3544874

0.945 0.003 CHEMBL3544897

0.945 0.003 CHEMBL3544898

0.69 0.004 CHEMBL1231106

0.867 0.003 CHEMBL457723

0.867 0.003 CHEMBL3544872

CHEMBL244377
0.1840.0160.973TIE-2 antagonist

0.852 0.003 CHEMBL3544873

0.973 0.002 CHEMBL244377

0.304 0.007 CHEMBL3544874

0.945 0.003 CHEMBL3544897

0.945 0.003 CHEMBL3544898

0.696 0.004 CHEMBL1231106

0.866 0.003 CHEMBL457723

0.866 0.003 CHEMBL3544872

CHEMBL244377
0.1720.0060.317Glutamate release inhibitor

0.165 0.007 CHEMBL3544873

0.143 0.012 CHEMBL244377

0.274 0.004 CHEMBL3544874

0.219 0.004 CHEMBL3544897

0.219 0.004 CHEMBL3544898

0.317 0.003 CHEMBL1231106

0.115 0.025 CHEMBL457723

0.115 0.025 CHEMBL3544872

CHEMBL1231106
0.2450.0820.327Interleukin agonist

0.245 0.083 CHEMBL244377

0.237 0.089 CHEMBL3544874

0.232 0.092 CHEMBL3544897

0.232 0.092 CHEMBL3544898

0.327 0.036 CHEMBL1231106

CHEMBL1231106
0.1750.0140.175Phosphodiesterase 7B inhibitor

0.119 0.038 CHEMBL3544873

0.17 0.015 CHEMBL3544874

0.083 0.081 CHEMBL3544897

0.083 0.081 CHEMBL3544898

0.135 0.028 CHEMBL1231106

0.107 0.049 CHEMBL457723

0.107 0.049 CHEMBL3544872

0.1730.0140.241GABA C receptor rho-1 antagonist

0.136 0.028 CHEMBL3544873

0.219 0.006 CHEMBL244377

0.165 0.016 CHEMBL3544874

0.204 0.008 CHEMBL3544897

0.204 0.008 CHEMBL3544898

0.241 0.005 CHEMBL1231106

0.148 0.022 CHEMBL457723

0.148 0.022 CHEMBL3544872

CHEMBL1231106
0.1630.0050.165Caspase 7 inhibitor

0.114 0.018 CHEMBL3544873

0.121 0.014 CHEMBL244377

0.109 0.02 CHEMBL3544874

0.084 0.053 CHEMBL3544897

0.084 0.053 CHEMBL3544898

0.079 0.064 CHEMBL1231106

0.165 0.005 CHEMBL457723

0.165 0.005 CHEMBL3544872

CHEMBL3544872
0.1920.0350.192Mannose-6-phosphate isomerase inhibitor

0.168 0.05 CHEMBL244377

0.13 0.086 CHEMBL3544874

0.118 0.105 CHEMBL3544897

0.118 0.105 CHEMBL3544898

0.179 0.043 CHEMBL1231106

0.123 0.096 CHEMBL457723

0.123 0.096 CHEMBL3544872

0.170.0140.256NADH dehydrogenase inhibitor

0.106 0.038 CHEMBL3544873

0.149 0.018 CHEMBL244377

0.154 0.017 CHEMBL3544874

0.137 0.021 CHEMBL3544897

0.137 0.021 CHEMBL3544898

0.256 0.008 CHEMBL1231106

0.114 0.032 CHEMBL457723

0.114 0.032 CHEMBL3544872

CHEMBL1231106
0.1840.0290.379Ephrin antagonist

0.129 0.045 CHEMBL3544873

0.281 0.011 CHEMBL244377

0.139 0.04 CHEMBL3544874

0.23 0.018 CHEMBL3544897

0.23 0.018 CHEMBL3544898

0.379 0.005 CHEMBL1231106

0.143 0.039 CHEMBL457723

0.143 0.039 CHEMBL3544872

CHEMBL1231106
0.1690.0140.175Ca2+-transporting ATPase inhibitor

0.133 0.103 CHEMBL3544873

0.159 0.026 CHEMBL244377

0.154 0.035 CHEMBL3544874

0.147 0.05 CHEMBL3544897

0.147 0.05 CHEMBL3544898

0.175 0.009 CHEMBL1231106

0.144 0.059 CHEMBL457723

0.144 0.059 CHEMBL3544872

CHEMBL1231106
0.1670.0120.172Interleukin 1 beta converting enzyme inhibitor

0.142 0.021 CHEMBL3544873

0.138 0.023 CHEMBL244377

0.136 0.024 CHEMBL3544874

0.105 0.051 CHEMBL3544897

0.105 0.051 CHEMBL3544898

0.103 0.054 CHEMBL1231106

0.172 0.011 CHEMBL457723

0.172 0.011 CHEMBL3544872

CHEMBL3544872
0.2680.1140.268Transcription factor NF kappa B inhibitor

0.193 0.176 CHEMBL3544873

0.232 0.141 CHEMBL244377

0.216 0.154 CHEMBL3544874

0.211 0.158 CHEMBL1231106

0.242 0.133 CHEMBL457723

0.242 0.133 CHEMBL3544872

0.1630.0090.463Phosphodiesterase 4A inhibitor

0.274 0.005 CHEMBL3544873

0.463 0.004 CHEMBL244377

0.056 0.032 CHEMBL3544874

0.31 0.005 CHEMBL3544897

0.31 0.005 CHEMBL3544898

0.048 0.036 CHEMBL1231106

0.393 0.004 CHEMBL457723

0.393 0.004 CHEMBL3544872

CHEMBL244377
0.1930.040.197Arachidonic acid antagonist

0.178 0.056 CHEMBL244377

0.157 0.08 CHEMBL3544874

0.142 0.098 CHEMBL3544897

0.142 0.098 CHEMBL3544898

0.197 0.035 CHEMBL1231106

0.136 0.105 CHEMBL457723

0.136 0.105 CHEMBL3544872

CHEMBL1231106
0.1740.0220.211UDP-glucose 4-epimerase inhibitor

0.153 0.028 CHEMBL244377

0.117 0.045 CHEMBL3544874

0.107 0.054 CHEMBL3544897

0.107 0.054 CHEMBL3544898

0.211 0.017 CHEMBL1231106

0.107 0.053 CHEMBL457723

0.107 0.053 CHEMBL3544872

CHEMBL1231106
0.1750.0240.2075 Hydroxytryptamine 3A agonist

0.169 0.026 CHEMBL244377

0.131 0.047 CHEMBL3544874

0.126 0.051 CHEMBL3544897

0.126 0.051 CHEMBL3544898

0.207 0.013 CHEMBL1231106

0.114 0.061 CHEMBL457723

0.114 0.061 CHEMBL3544872

CHEMBL1231106
0.1590.0080.184Acyl-CoA dehydrogenase inhibitor

0.074 0.025 CHEMBL3544873

0.13 0.011 CHEMBL244377

0.137 0.01 CHEMBL3544874

0.114 0.014 CHEMBL3544897

0.114 0.014 CHEMBL3544898

0.184 0.006 CHEMBL1231106

0.085 0.02 CHEMBL457723

0.085 0.02 CHEMBL3544872

CHEMBL1231106
0.2030.0540.203Lipocortins synthesis antagonist

0.19 0.063 CHEMBL3544874

0.1830.0380.204Cell wall synthesis inhibitor

0.156 0.06 CHEMBL3544873

0.195 0.032 CHEMBL244377

0.17 0.047 CHEMBL3544874

0.181 0.039 CHEMBL3544897

0.181 0.039 CHEMBL3544898

0.204 0.028 CHEMBL1231106

0.168 0.049 CHEMBL457723

0.168 0.049 CHEMBL3544872

CHEMBL1231106
0.2050.060.205Sigma receptor agonist
0.1590.0140.223Glutamate dehydrogenase inhibitor

0.1 0.031 CHEMBL3544873

0.123 0.022 CHEMBL244377

0.169 0.013 CHEMBL3544874

0.13 0.02 CHEMBL3544897

0.13 0.02 CHEMBL3544898

0.223 0.008 CHEMBL1231106

0.095 0.033 CHEMBL457723

0.095 0.033 CHEMBL3544872

CHEMBL1231106
0.1590.0160.339Electrolyte absorption antagonist

0.135 0.026 CHEMBL3544873

0.162 0.015 CHEMBL244377

0.2 0.008 CHEMBL3544874

0.201 0.008 CHEMBL3544897

0.201 0.008 CHEMBL3544898

0.339 0.004 CHEMBL1231106

0.108 0.048 CHEMBL457723

0.108 0.048 CHEMBL3544872

CHEMBL1231106
0.2070.0660.207Insulin sensitizer

0.166 0.112 CHEMBL3544874

0.168 0.109 CHEMBL1231106

0.1640.0230.164Heat shock protein 70 antagonist

0.136 0.09 CHEMBL3544873

0.16 0.028 CHEMBL244377

0.149 0.047 CHEMBL3544874

0.146 0.054 CHEMBL3544897

0.146 0.054 CHEMBL3544898

0.159 0.03 CHEMBL1231106

0.148 0.049 CHEMBL457723

0.148 0.049 CHEMBL3544872

0.160.020.178Creatine kinase inhibitor

0.134 0.031 CHEMBL244377

0.113 0.047 CHEMBL3544874

0.094 0.066 CHEMBL3544897

0.094 0.066 CHEMBL3544898

0.178 0.015 CHEMBL1231106

0.09 0.072 CHEMBL457723

0.09 0.072 CHEMBL3544872

CHEMBL1231106
0.1520.0130.167Histamine N-methyltransferase inhibitor

0.134 0.021 CHEMBL3544873

0.135 0.02 CHEMBL244377

0.167 0.009 CHEMBL3544874

0.147 0.015 CHEMBL3544897

0.147 0.015 CHEMBL3544898

0.165 0.01 CHEMBL1231106

0.123 0.028 CHEMBL457723

0.123 0.028 CHEMBL3544872

CHEMBL3544874
0.2120.0740.305MAP kinase kinase 2 inhibitor

0.21 0.076 CHEMBL3544873

0.286 0.04 CHEMBL244377

0.228 0.065 CHEMBL3544874

0.295 0.037 CHEMBL3544897

0.295 0.037 CHEMBL3544898

0.305 0.033 CHEMBL1231106

0.201 0.081 CHEMBL457723

0.201 0.081 CHEMBL3544872

CHEMBL1231106
0.1570.0190.213Porphobilinogen synthase inhibitor

0.119 0.028 CHEMBL244377

0.09 0.041 CHEMBL3544874

0.069 0.057 CHEMBL3544897

0.069 0.057 CHEMBL3544898

0.213 0.011 CHEMBL1231106

CHEMBL1231106
0.2040.0670.251I kappa B kinase epsilon inhibitor

0.187 0.083 CHEMBL3544873

0.232 0.047 CHEMBL244377

0.21 0.063 CHEMBL3544874

0.235 0.046 CHEMBL3544897

0.235 0.046 CHEMBL3544898

0.251 0.037 CHEMBL1231106

0.184 0.085 CHEMBL457723

0.184 0.085 CHEMBL3544872

CHEMBL1231106
0.1460.0110.161Phosphodiesterase 6D inhibitor

0.118 0.026 CHEMBL3544873

0.13 0.018 CHEMBL244377

0.108 0.039 CHEMBL3544874

0.096 0.06 CHEMBL3544897

0.096 0.06 CHEMBL3544898

0.161 0.008 CHEMBL457723

0.161 0.008 CHEMBL3544872

CHEMBL3544872
0.1540.0190.474p38 MAP kinase inhibitor

0.225 0.011 CHEMBL3544873

0.474 0.005 CHEMBL244377

0.217 0.012 CHEMBL3544897

0.217 0.012 CHEMBL3544898

0.423 0.005 CHEMBL457723

0.423 0.005 CHEMBL3544872

CHEMBL244377
0.1680.0330.226Protein kinase (CK2) alpha inhibitor

0.226 0.02 CHEMBL3544873

0.198 0.025 CHEMBL244377

0.18 0.029 CHEMBL3544874

0.208 0.023 CHEMBL3544897

0.208 0.023 CHEMBL3544898

0.174 0.031 CHEMBL1231106

0.215 0.022 CHEMBL457723

0.215 0.022 CHEMBL3544872

CHEMBL3544873
0.1510.0180.223Phosphofructokinase-1 inhibitor

0.102 0.031 CHEMBL3544873

0.156 0.017 CHEMBL244377

0.145 0.019 CHEMBL3544874

0.156 0.017 CHEMBL3544897

0.156 0.017 CHEMBL3544898

0.223 0.009 CHEMBL1231106

0.103 0.031 CHEMBL457723

0.103 0.031 CHEMBL3544872

CHEMBL1231106
0.1530.0210.153Prolactin inhibitor

0.124 0.036 CHEMBL244377

0.102 0.053 CHEMBL3544874

0.113 0.044 CHEMBL1231106

0.102 0.054 CHEMBL457723

0.102 0.054 CHEMBL3544872

0.2080.0760.208Psychostimulant

0.199 0.081 CHEMBL244377

0.159 0.108 CHEMBL3544874

0.149 0.117 CHEMBL3544897

0.149 0.117 CHEMBL3544898

0.184 0.09 CHEMBL1231106

0.134 0.131 CHEMBL457723

0.134 0.131 CHEMBL3544872

0.1680.0370.188Adenylate cyclase stimulant

0.138 0.084 CHEMBL3544873

0.188 0.02 CHEMBL244377

0.152 0.059 CHEMBL3544874

0.17 0.035 CHEMBL3544897

0.17 0.035 CHEMBL3544898

0.187 0.02 CHEMBL1231106

0.155 0.054 CHEMBL457723

0.155 0.054 CHEMBL3544872

CHEMBL244377
0.1820.0510.182Acetylcholine M1 receptor antagonist

0.146 0.078 CHEMBL3544874

0.121 0.106 CHEMBL1231106

0.1580.0290.511Fibroblast growth factor 1 antagonist

0.291 0.007 CHEMBL3544873

0.511 0.004 CHEMBL244377

0.182 0.021 CHEMBL3544874

0.444 0.004 CHEMBL3544897

0.444 0.004 CHEMBL3544898

0.389 0.005 CHEMBL1231106

0.292 0.006 CHEMBL457723

0.292 0.006 CHEMBL3544872

CHEMBL244377
0.2280.0990.2615 Hydroxytryptamine 1E antagonist

0.261 0.063 CHEMBL244377

0.169 0.167 CHEMBL3544874

0.212 0.117 CHEMBL3544897

0.212 0.117 CHEMBL3544898

0.224 0.104 CHEMBL1231106

0.197 0.134 CHEMBL457723

0.197 0.134 CHEMBL3544872

CHEMBL244377
0.1610.0330.322Cyclin-dependent kinase 2 inhibitor

0.212 0.022 CHEMBL3544873

0.18 0.029 CHEMBL244377

0.2 0.024 CHEMBL3544874

0.215 0.022 CHEMBL3544897

0.215 0.022 CHEMBL3544898

0.322 0.011 CHEMBL1231106

0.185 0.028 CHEMBL457723

0.185 0.028 CHEMBL3544872

CHEMBL1231106
0.1480.0210.178Triose-phosphate isomerase inhibitor

0.127 0.029 CHEMBL244377

0.1 0.047 CHEMBL3544874

0.091 0.058 CHEMBL3544897

0.091 0.058 CHEMBL3544898

0.178 0.014 CHEMBL1231106

0.088 0.063 CHEMBL457723

0.088 0.063 CHEMBL3544872

CHEMBL1231106
0.1430.0160.292Adenosine A2a receptor antagonist

0.292 0.005 CHEMBL3544873

0.14 0.016 CHEMBL244377

0.245 0.008 CHEMBL3544874

0.238 0.008 CHEMBL3544897

0.238 0.008 CHEMBL3544898

0.196 0.01 CHEMBL1231106

0.188 0.011 CHEMBL457723

0.188 0.011 CHEMBL3544872

CHEMBL3544873
0.1370.0130.21Carbamoyl phosphate synthetase inhibitor

0.077 0.03 CHEMBL3544873

0.118 0.016 CHEMBL244377

0.13 0.014 CHEMBL3544874

0.109 0.018 CHEMBL3544897

0.109 0.018 CHEMBL3544898

0.21 0.007 CHEMBL1231106

0.084 0.026 CHEMBL457723

0.084 0.026 CHEMBL3544872

CHEMBL1231106
0.1330.0080.154Alpha 2 adrenoreceptor agonist

0.117 0.011 CHEMBL3544873

0.126 0.009 CHEMBL244377

0.103 0.014 CHEMBL3544874

0.092 0.017 CHEMBL3544897

0.092 0.017 CHEMBL3544898

0.075 0.027 CHEMBL1231106

0.154 0.006 CHEMBL457723

0.154 0.006 CHEMBL3544872

CHEMBL3544872
0.140.0180.298Adenosine A2 receptor antagonist

0.298 0.005 CHEMBL3544873

0.152 0.016 CHEMBL244377

0.238 0.008 CHEMBL3544874

0.247 0.008 CHEMBL3544897

0.247 0.008 CHEMBL3544898

0.196 0.011 CHEMBL1231106

0.192 0.011 CHEMBL457723

0.192 0.011 CHEMBL3544872

CHEMBL3544873
0.1760.0550.181Neurotensin receptor agonist

0.161 0.077 CHEMBL244377

0.152 0.097 CHEMBL3544874

0.138 0.134 CHEMBL3544897

0.138 0.134 CHEMBL3544898

0.181 0.049 CHEMBL1231106

0.139 0.133 CHEMBL457723

0.139 0.133 CHEMBL3544872

CHEMBL1231106
0.1980.0790.283Neurotrophic factor enhancer

0.182 0.095 CHEMBL3544873

0.218 0.061 CHEMBL244377

0.221 0.058 CHEMBL3544874

0.244 0.042 CHEMBL3544897

0.244 0.042 CHEMBL3544898

0.283 0.023 CHEMBL1231106

0.156 0.13 CHEMBL457723

0.156 0.13 CHEMBL3544872

CHEMBL1231106
0.180.0610.196Phospholipase C inhibitor

0.167 0.077 CHEMBL244377

0.164 0.081 CHEMBL3544874

0.152 0.103 CHEMBL3544897

0.152 0.103 CHEMBL3544898

0.196 0.046 CHEMBL1231106

0.139 0.129 CHEMBL457723

0.139 0.129 CHEMBL3544872

CHEMBL1231106
0.1230.0040.123Glutamate (mGluR7) antagonist

0.067 0.049 CHEMBL3544873

0.09 0.017 CHEMBL244377

0.103 0.009 CHEMBL3544874

0.075 0.035 CHEMBL3544897

0.075 0.035 CHEMBL3544898

0.105 0.008 CHEMBL1231106

0.081 0.026 CHEMBL457723

0.081 0.026 CHEMBL3544872

0.1430.0260.143DNA directed RNA polymerase inhibitor

0.102 0.054 CHEMBL3544873

0.13 0.032 CHEMBL3544874

0.128 0.033 CHEMBL1231106

0.1 0.056 CHEMBL457723

0.1 0.056 CHEMBL3544872

0.1640.050.191Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.142 0.089 CHEMBL3544873

0.191 0.023 CHEMBL244377

0.143 0.087 CHEMBL3544874

0.164 0.05 CHEMBL3544897

0.164 0.05 CHEMBL3544898

0.167 0.046 CHEMBL1231106

0.158 0.058 CHEMBL457723

0.158 0.058 CHEMBL3544872

CHEMBL244377
0.1880.0740.332CDC-like kinase 4 inhibitor

0.25 0.046 CHEMBL3544873

0.254 0.045 CHEMBL244377

0.232 0.053 CHEMBL3544874

0.276 0.038 CHEMBL3544897

0.276 0.038 CHEMBL3544898

0.332 0.024 CHEMBL1231106

0.227 0.055 CHEMBL457723

0.227 0.055 CHEMBL3544872

CHEMBL1231106
0.1470.0330.147Photosensitizer

0.121 0.055 CHEMBL244377

0.108 0.074 CHEMBL3544874

0.131 0.045 CHEMBL1231106

0.097 0.094 CHEMBL457723

0.097 0.094 CHEMBL3544872

0.1470.0340.21Protein kinase (CK2) inhibitor

0.196 0.019 CHEMBL3544873

0.21 0.017 CHEMBL244377

0.142 0.036 CHEMBL3544874

0.197 0.019 CHEMBL3544897

0.197 0.019 CHEMBL3544898

0.149 0.033 CHEMBL1231106

0.208 0.017 CHEMBL457723

0.208 0.017 CHEMBL3544872

CHEMBL244377
0.1470.0340.147Mucolytic

0.104 0.072 CHEMBL244377

0.118 0.057 CHEMBL3544874

0.127 0.048 CHEMBL1231106

0.098 0.08 CHEMBL457723

0.098 0.08 CHEMBL3544872

0.2570.1440.257Calpain 2 inhibitor
0.150.0380.181Aminopeptidase B inhibitor

0.134 0.045 CHEMBL244377

0.13 0.047 CHEMBL3544874

0.111 0.058 CHEMBL3544897

0.111 0.058 CHEMBL3544898

0.181 0.026 CHEMBL1231106

0.093 0.07 CHEMBL457723

0.093 0.07 CHEMBL3544872

CHEMBL1231106
0.1420.030.144Transcription factor STAT6 inhibitor

0.103 0.098 CHEMBL3544873

0.144 0.028 CHEMBL244377

0.117 0.065 CHEMBL3544874

0.119 0.061 CHEMBL3544897

0.119 0.061 CHEMBL3544898

0.133 0.04 CHEMBL1231106

0.127 0.048 CHEMBL457723

0.127 0.048 CHEMBL3544872

CHEMBL244377
0.1550.0440.157Aldehyde dehydrogenase inhibitor

0.128 0.063 CHEMBL244377

0.105 0.09 CHEMBL3544874

0.157 0.043 CHEMBL1231106

CHEMBL1231106
0.1580.0490.158Sodium channel (voltage-gated) blocker

0.128 0.076 CHEMBL3544874

0.132 0.07 CHEMBL1231106

0.190.0810.52Ca2+/calmodulin-dependent protein kinase inhibitor

0.329 0.034 CHEMBL3544873

0.397 0.018 CHEMBL244377

0.301 0.043 CHEMBL3544874

0.42 0.015 CHEMBL3544897

0.42 0.015 CHEMBL3544898

0.52 0.007 CHEMBL1231106

0.277 0.049 CHEMBL457723

0.277 0.049 CHEMBL3544872

CHEMBL1231106
0.140.0330.387CDK/cyclin complex inhibitor

0.19 0.021 CHEMBL3544873

0.298 0.01 CHEMBL244377

0.152 0.029 CHEMBL3544874

0.275 0.011 CHEMBL3544897

0.275 0.011 CHEMBL3544898

0.387 0.005 CHEMBL1231106

0.186 0.021 CHEMBL457723

0.186 0.021 CHEMBL3544872

CHEMBL1231106
0.1190.0110.262Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.091 0.016 CHEMBL3544873

0.096 0.015 CHEMBL244377

0.157 0.008 CHEMBL3544874

0.128 0.01 CHEMBL3544897

0.128 0.01 CHEMBL3544898

0.262 0.005 CHEMBL1231106

0.069 0.026 CHEMBL457723

0.069 0.026 CHEMBL3544872

CHEMBL1231106
0.1240.0170.372Phenylalanine 4-hydroxylase inhibitor

0.106 0.023 CHEMBL3544873

0.114 0.02 CHEMBL244377

0.206 0.006 CHEMBL3544874

0.183 0.008 CHEMBL3544897

0.183 0.008 CHEMBL3544898

0.372 0.003 CHEMBL1231106

0.065 0.051 CHEMBL457723

0.065 0.051 CHEMBL3544872

CHEMBL1231106
0.1240.0180.498CDK1/cyclin B inhibitor

0.226 0.008 CHEMBL3544873

0.406 0.005 CHEMBL244377

0.14 0.015 CHEMBL3544874

0.371 0.005 CHEMBL3544897

0.371 0.005 CHEMBL3544898

0.498 0.004 CHEMBL1231106

0.22 0.008 CHEMBL457723

0.22 0.008 CHEMBL3544872

CHEMBL1231106
0.1870.0810.213Focal adhesion kinase 2 inhibitor

0.185 0.082 CHEMBL244377

0.181 0.087 CHEMBL3544874

0.177 0.091 CHEMBL3544897

0.177 0.091 CHEMBL3544898

0.213 0.06 CHEMBL1231106

0.15 0.132 CHEMBL457723

0.15 0.132 CHEMBL3544872

CHEMBL1231106
0.1470.0420.172Cystathionine beta-synthase inhibitor

0.123 0.056 CHEMBL244377

0.101 0.075 CHEMBL3544874

0.172 0.032 CHEMBL1231106

CHEMBL1231106
0.1330.0290.246CDC-like kinase 3 inhibitor

0.166 0.013 CHEMBL3544873

0.246 0.004 CHEMBL244377

0.125 0.037 CHEMBL3544874

0.204 0.007 CHEMBL3544897

0.204 0.007 CHEMBL3544898

0.164 0.014 CHEMBL1231106

0.184 0.009 CHEMBL457723

0.184 0.009 CHEMBL3544872

CHEMBL244377
0.1420.040.19DNA repair enzyme inhibitor

0.163 0.022 CHEMBL3544873

0.153 0.029 CHEMBL244377

0.173 0.016 CHEMBL3544874

0.184 0.012 CHEMBL3544897

0.184 0.012 CHEMBL3544898

0.19 0.01 CHEMBL1231106

0.13 0.055 CHEMBL457723

0.13 0.055 CHEMBL3544872

CHEMBL1231106
0.1160.0150.211Alcohol oxidase inhibitor

0.097 0.019 CHEMBL244377

0.072 0.028 CHEMBL3544874

0.059 0.036 CHEMBL3544897

0.059 0.036 CHEMBL3544898

0.211 0.006 CHEMBL1231106

CHEMBL1231106
0.1160.0140.186Biliverdin reductase inhibitor

0.096 0.02 CHEMBL244377

0.096 0.02 CHEMBL3544874

0.08 0.026 CHEMBL3544897

0.08 0.026 CHEMBL3544898

0.186 0.006 CHEMBL1231106

0.06 0.04 CHEMBL457723

0.06 0.04 CHEMBL3544872

CHEMBL1231106
0.1560.0560.156Neuropeptide Y1 antagonist

0.133 0.093 CHEMBL244377

0.13 0.1 CHEMBL3544874

0.136 0.088 CHEMBL1231106

0.137 0.086 CHEMBL457723

0.137 0.086 CHEMBL3544872

0.1330.0340.172Insulin receptor antagonist

0.168 0.022 CHEMBL3544873

0.163 0.024 CHEMBL244377

0.142 0.03 CHEMBL3544874

0.172 0.021 CHEMBL3544897

0.172 0.021 CHEMBL3544898

0.133 0.034 CHEMBL1231106

0.158 0.025 CHEMBL457723

0.158 0.025 CHEMBL3544872

CHEMBL3544898
0.1170.0190.179mTOR complex 2 inhibitor

0.143 0.01 CHEMBL3544873

0.131 0.013 CHEMBL244377

0.15 0.009 CHEMBL3544874

0.168 0.007 CHEMBL3544897

0.168 0.007 CHEMBL3544898

0.179 0.005 CHEMBL1231106

0.111 0.023 CHEMBL457723

0.111 0.023 CHEMBL3544872

CHEMBL1231106
0.1330.0360.29Carbonic anhydrase III inhibitor

0.141 0.032 CHEMBL3544873

0.29 0.006 CHEMBL244377

0.106 0.055 CHEMBL3544874

0.238 0.011 CHEMBL3544897

0.238 0.011 CHEMBL3544898

0.166 0.023 CHEMBL1231106

0.186 0.019 CHEMBL457723

0.186 0.019 CHEMBL3544872

CHEMBL244377
0.1070.010.147S-adenosyl-L-methionine decarboxylase inhibitor

0.093 0.019 CHEMBL3544873

0.107 0.01 CHEMBL244377

0.118 0.006 CHEMBL3544874

0.115 0.007 CHEMBL3544897

0.115 0.007 CHEMBL3544898

0.147 0.004 CHEMBL1231106

0.086 0.028 CHEMBL457723

0.086 0.028 CHEMBL3544872

CHEMBL1231106
0.1170.020.244Adenosine A1 receptor antagonist

0.244 0.008 CHEMBL3544873

0.119 0.02 CHEMBL244377

0.197 0.011 CHEMBL3544874

0.195 0.011 CHEMBL3544897

0.195 0.011 CHEMBL3544898

0.152 0.015 CHEMBL1231106

0.166 0.014 CHEMBL457723

0.166 0.014 CHEMBL3544872

CHEMBL3544873
0.1360.0390.136Alpha 2c adrenoreceptor antagonist

0.107 0.06 CHEMBL3544874

0.086 0.08 CHEMBL457723

0.086 0.08 CHEMBL3544872

0.120.0250.691Protein kinase B gamma inhibitor

0.374 0.004 CHEMBL3544873

0.691 0.003 CHEMBL244377

0.161 0.013 CHEMBL3544874

0.601 0.003 CHEMBL3544897

0.601 0.003 CHEMBL3544898

0.501 0.003 CHEMBL1231106

0.389 0.004 CHEMBL457723

0.389 0.004 CHEMBL3544872

CHEMBL244377
0.1040.010.13MAP kinase kinase 7 inhibitor

0.115 0.005 CHEMBL3544873

0.106 0.009 CHEMBL244377

0.122 0.004 CHEMBL3544874

0.122 0.004 CHEMBL3544897

0.122 0.004 CHEMBL3544898

0.13 0.004 CHEMBL1231106

0.099 0.014 CHEMBL457723

0.099 0.014 CHEMBL3544872

CHEMBL1231106
0.1080.0140.143Maillard reaction inhibitor

0.053 0.04 CHEMBL3544873

0.12 0.01 CHEMBL3544874

0.143 0.006 CHEMBL1231106

CHEMBL1231106
0.1440.0510.663Vascular endothelial growth factor 2 antagonist

0.243 0.027 CHEMBL3544873

0.663 0.005 CHEMBL244377

0.14 0.052 CHEMBL3544874

0.534 0.007 CHEMBL3544897

0.534 0.007 CHEMBL3544898

0.619 0.005 CHEMBL1231106

0.276 0.023 CHEMBL457723

0.276 0.023 CHEMBL3544872

CHEMBL244377
0.1280.0350.173UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.118 0.04 CHEMBL244377

0.083 0.075 CHEMBL3544874

0.173 0.021 CHEMBL1231106

CHEMBL1231106
0.1120.0210.165Granulocyte macrophage colony stimulating factor agonist

0.082 0.071 CHEMBL3544873

0.11 0.023 CHEMBL244377

0.111 0.023 CHEMBL3544874

0.107 0.026 CHEMBL3544897

0.107 0.026 CHEMBL3544898

0.165 0.004 CHEMBL1231106

0.084 0.064 CHEMBL457723

0.084 0.064 CHEMBL3544872

CHEMBL1231106
0.1070.0160.11Phosphodiesterase VI inhibitor

0.074 0.053 CHEMBL3544873

0.085 0.033 CHEMBL244377

0.072 0.058 CHEMBL3544874

0.11 0.015 CHEMBL457723

0.11 0.015 CHEMBL3544872

CHEMBL3544872
0.1840.0940.305Platelet aggregation inhibitor

0.252 0.051 CHEMBL244377

0.305 0.035 CHEMBL1231106

CHEMBL1231106
0.2320.1420.232Antithrombotic

0.191 0.188 CHEMBL1231106

0.1030.0130.137ZAP-70 protein tyrosine kinase inhibitor

0.083 0.031 CHEMBL3544873

0.137 0.005 CHEMBL244377

0.08 0.035 CHEMBL3544874

0.102 0.013 CHEMBL3544897

0.102 0.013 CHEMBL3544898

0.114 0.009 CHEMBL1231106

0.097 0.016 CHEMBL457723

0.097 0.016 CHEMBL3544872

CHEMBL244377
0.1450.0560.654Vascular endothelial growth factor antagonist

0.239 0.03 CHEMBL3544873

0.654 0.005 CHEMBL244377

0.143 0.057 CHEMBL3544874

0.523 0.007 CHEMBL3544897

0.523 0.007 CHEMBL3544898

0.612 0.005 CHEMBL1231106

0.266 0.026 CHEMBL457723

0.266 0.026 CHEMBL3544872

CHEMBL244377
0.1160.0280.116CYP2A6 inhibitor

0.108 0.032 CHEMBL244377

0.077 0.051 CHEMBL3544874

0.072 0.057 CHEMBL3544897

0.072 0.057 CHEMBL3544898

0.116 0.028 CHEMBL1231106

0.1520.0640.23MAP kinase 3 inhibitor

0.183 0.033 CHEMBL3544873

0.23 0.013 CHEMBL244377

0.151 0.065 CHEMBL3544874

0.228 0.013 CHEMBL3544897

0.228 0.013 CHEMBL3544898

0.19 0.028 CHEMBL1231106

0.185 0.032 CHEMBL457723

0.185 0.032 CHEMBL3544872

CHEMBL244377
0.1020.0160.138Purinergic P2X1 antagonist

0.061 0.042 CHEMBL3544873

0.114 0.013 CHEMBL244377

0.079 0.026 CHEMBL3544874

0.092 0.019 CHEMBL3544897

0.092 0.019 CHEMBL3544898

0.138 0.009 CHEMBL1231106

0.075 0.028 CHEMBL457723

0.075 0.028 CHEMBL3544872

CHEMBL1231106
0.1020.0150.102Vanilloid 4 agonist

0.094 0.022 CHEMBL244377

0.075 0.051 CHEMBL3544874

0.069 0.068 CHEMBL3544897

0.069 0.068 CHEMBL3544898

0.089 0.027 CHEMBL1231106

0.078 0.044 CHEMBL457723

0.078 0.044 CHEMBL3544872

0.1050.0190.105Estrogen-related receptor beta agonist

0.097 0.029 CHEMBL244377

0.089 0.042 CHEMBL3544874

0.083 0.057 CHEMBL3544897

0.083 0.057 CHEMBL3544898

0.097 0.028 CHEMBL1231106

0.082 0.06 CHEMBL457723

0.082 0.06 CHEMBL3544872

0.1320.0460.133Falcipain 3 inhibitor

0.133 0.045 CHEMBL244377

0.125 0.05 CHEMBL1231106

CHEMBL244377
0.110.0240.11Alpha adrenoreceptor agonist

0.069 0.047 CHEMBL3544873

0.09 0.032 CHEMBL244377

0.073 0.043 CHEMBL3544874

0.109 0.024 CHEMBL457723

0.109 0.024 CHEMBL3544872

0.1510.0660.595Protein kinase (CK1) inhibitor

0.374 0.01 CHEMBL3544873

0.455 0.005 CHEMBL244377

0.292 0.019 CHEMBL3544874

0.495 0.005 CHEMBL3544897

0.495 0.005 CHEMBL3544898

0.595 0.004 CHEMBL1231106

0.286 0.02 CHEMBL457723

0.286 0.02 CHEMBL3544872

CHEMBL1231106
0.1220.0370.169Nitric-oxide synthase inhibitor

0.109 0.047 CHEMBL3544873

0.109 0.047 CHEMBL244377

0.151 0.022 CHEMBL3544874

0.133 0.031 CHEMBL3544897

0.133 0.031 CHEMBL3544898

0.169 0.016 CHEMBL1231106

0.094 0.07 CHEMBL457723

0.094 0.07 CHEMBL3544872

CHEMBL1231106
0.1250.040.173DOPA decarboxylase inhibitor

0.116 0.05 CHEMBL244377

0.113 0.053 CHEMBL3544874

0.107 0.064 CHEMBL3544897

0.107 0.064 CHEMBL3544898

0.173 0.012 CHEMBL1231106

CHEMBL1231106
0.0980.0140.098Orexin receptor 1 antagonist

0.073 0.047 CHEMBL244377

0.068 0.061 CHEMBL3544874

0.088 0.024 CHEMBL457723

0.088 0.024 CHEMBL3544872

0.1380.0560.158Cathepsin H inhibitor

0.131 0.063 CHEMBL244377

0.11 0.09 CHEMBL3544874

0.158 0.041 CHEMBL1231106

CHEMBL1231106
0.1010.0190.219Argininosuccinate synthase inhibitor

0.059 0.037 CHEMBL3544873

0.092 0.021 CHEMBL244377

0.114 0.016 CHEMBL3544874

0.1 0.019 CHEMBL3544897

0.1 0.019 CHEMBL3544898

0.219 0.007 CHEMBL1231106

0.055 0.041 CHEMBL457723

0.055 0.041 CHEMBL3544872

CHEMBL1231106
0.1440.0620.181Nav1.6 sodium channel blocker

0.125 0.088 CHEMBL244377

0.14 0.066 CHEMBL3544874

0.123 0.092 CHEMBL3544897

0.123 0.092 CHEMBL3544898

0.181 0.027 CHEMBL1231106

CHEMBL1231106
0.1160.0350.127Glutamate (mGluR7) agonist

0.127 0.024 CHEMBL244377

0.093 0.075 CHEMBL3544874

0.101 0.057 CHEMBL3544897

0.101 0.057 CHEMBL3544898

0.112 0.039 CHEMBL1231106

0.108 0.045 CHEMBL457723

0.108 0.045 CHEMBL3544872

CHEMBL244377
0.1340.0540.348Platelet activating factor antagonist

0.282 0.013 CHEMBL244377

0.192 0.028 CHEMBL3544897

0.192 0.028 CHEMBL3544898

0.348 0.008 CHEMBL1231106

0.106 0.074 CHEMBL457723

0.106 0.074 CHEMBL3544872

CHEMBL1231106
0.20.120.2Spasmolytic

0.162 0.152 CHEMBL244377

0.2590.1790.54MAP kinase kinase 6 inhibitor

0.38 0.071 CHEMBL3544873

0.54 0.011 CHEMBL244377

0.439 0.039 CHEMBL3544897

0.439 0.039 CHEMBL3544898

0.458 0.031 CHEMBL457723

0.458 0.031 CHEMBL3544872

CHEMBL244377
0.0910.0120.091Potassium channel (Ca-activated) blocker

0.058 0.044 CHEMBL244377

0.073 0.024 CHEMBL457723

0.073 0.024 CHEMBL3544872

0.1530.0750.294Diuretic

0.168 0.062 CHEMBL3544873

0.181 0.053 CHEMBL244377

0.195 0.046 CHEMBL3544874

0.24 0.032 CHEMBL3544897

0.24 0.032 CHEMBL3544898

0.294 0.023 CHEMBL1231106

0.124 0.1 CHEMBL457723

0.124 0.1 CHEMBL3544872

CHEMBL1231106
0.1140.0360.127Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.102 0.044 CHEMBL3544873

0.092 0.054 CHEMBL244377

0.127 0.031 CHEMBL3544874

0.097 0.048 CHEMBL3544897

0.097 0.048 CHEMBL3544898

0.116 0.035 CHEMBL1231106

0.096 0.049 CHEMBL457723

0.096 0.049 CHEMBL3544872

CHEMBL3544874
0.0910.0130.091Phosphodiesterase II inhibitor

0.05 0.048 CHEMBL457723

0.05 0.048 CHEMBL3544872

0.1060.0290.124Histamine H2 receptor antagonist

0.09 0.047 CHEMBL3544873

0.124 0.019 CHEMBL244377

0.098 0.037 CHEMBL3544874

0.114 0.024 CHEMBL3544897

0.114 0.024 CHEMBL3544898

0.117 0.023 CHEMBL1231106

0.098 0.037 CHEMBL457723

0.098 0.037 CHEMBL3544872

CHEMBL244377
0.1080.0310.116Inducible nitric-oxide synthase inhibitor

0.077 0.067 CHEMBL244377

0.104 0.034 CHEMBL3544874

0.116 0.026 CHEMBL1231106

CHEMBL1231106
0.1030.0260.206Interferon agonist

0.122 0.017 CHEMBL3544873

0.102 0.027 CHEMBL244377

0.157 0.009 CHEMBL3544874

0.15 0.01 CHEMBL3544897

0.15 0.01 CHEMBL3544898

0.206 0.005 CHEMBL1231106

0.086 0.043 CHEMBL457723

0.086 0.043 CHEMBL3544872

CHEMBL1231106
0.080.0040.08Corticotropin releasing factor 1 receptor antagonist

0.024 0.014 CHEMBL3544874

0.035 0.009 CHEMBL457723

0.035 0.009 CHEMBL3544872

0.1070.0320.222ErbB-2 antagonist

0.12 0.028 CHEMBL244377

0.07 0.059 CHEMBL3544874

0.081 0.047 CHEMBL3544897

0.081 0.047 CHEMBL3544898

0.222 0.008 CHEMBL1231106

CHEMBL1231106
0.0830.0080.083CXC chemokine 1 receptor antagonist

0.049 0.039 CHEMBL3544873

0.061 0.02 CHEMBL3544874

0.061 0.021 CHEMBL457723

0.061 0.021 CHEMBL3544872

0.0890.0150.096Exportin-1 inhibitor

0.073 0.036 CHEMBL244377

0.068 0.049 CHEMBL3544874

0.096 0.011 CHEMBL1231106

CHEMBL1231106
0.1210.0470.124Acetylcholine release stimulant

0.102 0.083 CHEMBL244377

0.124 0.042 CHEMBL1231106

CHEMBL1231106
0.0780.0040.115Protein kinase (CK2) beta inhibitor

0.077 0.004 CHEMBL3544873

0.115 0.003 CHEMBL244377

0.053 0.006 CHEMBL3544874

0.081 0.004 CHEMBL3544897

0.081 0.004 CHEMBL3544898

0.056 0.005 CHEMBL1231106

0.111 0.003 CHEMBL457723

0.111 0.003 CHEMBL3544872

CHEMBL244377
0.090.0180.09Orexin receptor antagonist

0.06 0.059 CHEMBL244377

0.078 0.03 CHEMBL457723

0.078 0.03 CHEMBL3544872

0.0850.0130.085Glucosylceramidase inhibitor

0.083 0.014 CHEMBL244377

0.052 0.044 CHEMBL3544874

0.05 0.048 CHEMBL3544897

0.05 0.048 CHEMBL3544898

0.067 0.024 CHEMBL1231106

0.074 0.019 CHEMBL457723

0.074 0.019 CHEMBL3544872

0.1150.0440.122Anabolic

0.107 0.054 CHEMBL244377

0.086 0.085 CHEMBL3544874

0.122 0.038 CHEMBL1231106

CHEMBL1231106
0.1110.040.141Lanosterol 14 alpha demethylase inhibitor

0.089 0.073 CHEMBL244377

0.1 0.055 CHEMBL3544874

0.141 0.015 CHEMBL1231106

CHEMBL1231106
0.1160.0450.116Sphingomyelinase inhibitor

0.114 0.046 CHEMBL244377

0.097 0.063 CHEMBL1231106

0.1950.1240.29Immunostimulant

0.181 0.132 CHEMBL3544873

0.194 0.124 CHEMBL244377

0.231 0.104 CHEMBL3544874

0.229 0.105 CHEMBL3544897

0.229 0.105 CHEMBL3544898

0.29 0.081 CHEMBL1231106

CHEMBL1231106
0.0750.0050.116Dihydrofolate reductase inhibitor

0.092 0.004 CHEMBL3544873

0.059 0.011 CHEMBL244377

0.116 0.003 CHEMBL3544874

0.091 0.004 CHEMBL3544897

0.091 0.004 CHEMBL3544898

0.114 0.003 CHEMBL1231106

0.061 0.01 CHEMBL457723

0.061 0.01 CHEMBL3544872

CHEMBL3544874
0.1350.0640.324Cyclin-dependent kinase inhibitor

0.233 0.03 CHEMBL3544873

0.324 0.017 CHEMBL244377

0.162 0.051 CHEMBL3544874

0.306 0.019 CHEMBL3544897

0.306 0.019 CHEMBL3544898

0.311 0.019 CHEMBL1231106

0.228 0.031 CHEMBL457723

0.228 0.031 CHEMBL3544872

CHEMBL244377
0.1490.0790.157Interferon gamma antagonist

0.132 0.106 CHEMBL244377

0.157 0.07 CHEMBL1231106

CHEMBL1231106
0.0830.0130.083Phosphodiesterase 2A inhibitor
0.0990.030.14Glutamate decarboxylase inhibitor

0.09 0.036 CHEMBL244377

0.078 0.046 CHEMBL3544874

0.068 0.057 CHEMBL3544897

0.068 0.057 CHEMBL3544898

0.14 0.015 CHEMBL1231106

CHEMBL1231106
0.0890.0210.0925 Hydroxytryptamine 3 agonist

0.075 0.031 CHEMBL244377

0.068 0.038 CHEMBL3544874

0.057 0.054 CHEMBL3544897

0.057 0.054 CHEMBL3544898

0.092 0.019 CHEMBL1231106

CHEMBL1231106
0.0810.0130.108Aconitate hydratase inhibitor

0.07 0.018 CHEMBL244377

0.057 0.029 CHEMBL3544874

0.052 0.035 CHEMBL3544897

0.052 0.035 CHEMBL3544898

0.108 0.007 CHEMBL1231106

CHEMBL1231106
0.1360.0690.696RET inhibitor

0.301 0.022 CHEMBL3544873

0.667 0.004 CHEMBL244377

0.163 0.055 CHEMBL3544874

0.558 0.005 CHEMBL3544897

0.558 0.005 CHEMBL3544898

0.696 0.004 CHEMBL1231106

0.307 0.021 CHEMBL457723

0.307 0.021 CHEMBL3544872

CHEMBL1231106
0.0980.0320.1Focal adhesion kinase 1 inhibitor

0.1 0.03 CHEMBL244377

0.069 0.064 CHEMBL1231106

CHEMBL244377
0.0820.0160.082Corticotropin releasing factor 2 receptor antagonist

0.071 0.027 CHEMBL244377

0.061 0.044 CHEMBL3544874

0.076 0.021 CHEMBL1231106

0.06 0.046 CHEMBL457723

0.06 0.046 CHEMBL3544872

0.0750.0090.12Histamine H2 receptor agonist

0.07 0.01 CHEMBL3544873

0.078 0.008 CHEMBL244377

0.094 0.005 CHEMBL3544874

0.096 0.004 CHEMBL3544897

0.096 0.004 CHEMBL3544898

0.12 0.003 CHEMBL1231106

0.052 0.02 CHEMBL457723

0.052 0.02 CHEMBL3544872

CHEMBL1231106
0.0950.0290.167Adenosine A3 receptor antagonist

0.163 0.011 CHEMBL3544873

0.134 0.015 CHEMBL244377

0.115 0.02 CHEMBL3544874

0.167 0.011 CHEMBL3544897

0.167 0.011 CHEMBL3544898

0.115 0.02 CHEMBL1231106

0.132 0.015 CHEMBL457723

0.132 0.015 CHEMBL3544872

CHEMBL3544898
0.1350.0690.135Sodium channel blocker

0.114 0.092 CHEMBL3544874

0.121 0.082 CHEMBL1231106

0.0980.0330.207Histidine decarboxylase inhibitor

0.111 0.028 CHEMBL244377

0.073 0.048 CHEMBL3544874

0.078 0.044 CHEMBL3544897

0.078 0.044 CHEMBL3544898

0.207 0.012 CHEMBL1231106

CHEMBL1231106
0.0760.0110.076Potassium channel small-conductance Ca-activated blocker

0.048 0.027 CHEMBL3544873

0.049 0.026 CHEMBL244377

0.06 0.017 CHEMBL3544874

0.045 0.031 CHEMBL1231106

0.062 0.016 CHEMBL457723

0.062 0.016 CHEMBL3544872

0.0730.0090.092Immunoglobulin Fc receptor antagonist

0.066 0.014 CHEMBL3544873

0.083 0.005 CHEMBL244377

0.074 0.008 CHEMBL3544874

0.083 0.005 CHEMBL3544897

0.083 0.005 CHEMBL3544898

0.092 0.004 CHEMBL1231106

0.066 0.015 CHEMBL457723

0.066 0.015 CHEMBL3544872

CHEMBL1231106
0.0740.010.08Glucose-6-phosphate isomerase inhibitor

0.067 0.014 CHEMBL244377

0.052 0.026 CHEMBL3544874

0.05 0.029 CHEMBL3544897

0.05 0.029 CHEMBL3544898

0.08 0.009 CHEMBL1231106

0.05 0.029 CHEMBL457723

0.05 0.029 CHEMBL3544872

CHEMBL1231106
0.090.0270.09Nav1.7 sodium channel blocker

0.065 0.05 CHEMBL3544874

0.066 0.049 CHEMBL1231106

0.1070.0430.107Alpha 2 adrenoreceptor antagonist

0.085 0.06 CHEMBL244377

0.104 0.045 CHEMBL457723

0.104 0.045 CHEMBL3544872

0.1080.0450.168Alcohol dehydrogenase inhibitor

0.094 0.06 CHEMBL244377

0.11 0.042 CHEMBL3544874

0.094 0.059 CHEMBL3544897

0.094 0.059 CHEMBL3544898

0.168 0.016 CHEMBL1231106

CHEMBL1231106
0.0890.0260.113GABA B receptor agonist

0.077 0.048 CHEMBL244377

0.092 0.024 CHEMBL3544874

0.077 0.047 CHEMBL3544897

0.077 0.047 CHEMBL3544898

0.113 0.01 CHEMBL1231106

CHEMBL1231106
0.0820.020.082Cyclin-dependent kinase 6 inhibitor

0.053 0.05 CHEMBL3544873

0.081 0.021 CHEMBL244377

0.068 0.032 CHEMBL3544874

0.066 0.035 CHEMBL3544897

0.066 0.035 CHEMBL3544898

0.077 0.024 CHEMBL1231106

0.07 0.031 CHEMBL457723

0.07 0.031 CHEMBL3544872

0.0830.0210.151Interferon inducer

0.099 0.013 CHEMBL3544873

0.082 0.022 CHEMBL244377

0.119 0.008 CHEMBL3544874

0.116 0.008 CHEMBL3544897

0.116 0.008 CHEMBL3544898

0.151 0.005 CHEMBL1231106

0.07 0.034 CHEMBL457723

0.07 0.034 CHEMBL3544872

CHEMBL1231106
0.0940.0320.117Aminopeptidase I inhibitor

0.085 0.038 CHEMBL244377

0.076 0.047 CHEMBL3544874

0.067 0.057 CHEMBL3544897

0.067 0.057 CHEMBL3544898

0.117 0.02 CHEMBL1231106

CHEMBL1231106
0.070.010.072CC chemokine 4 receptor antagonist

0.05 0.028 CHEMBL3544873

0.067 0.012 CHEMBL244377

0.049 0.029 CHEMBL3544874

0.046 0.035 CHEMBL3544897

0.046 0.035 CHEMBL3544898

0.046 0.034 CHEMBL1231106

0.072 0.009 CHEMBL457723

0.072 0.009 CHEMBL3544872

CHEMBL3544872
0.0660.0050.066Histamine H1 receptor agonist

0.046 0.024 CHEMBL3544873

0.061 0.008 CHEMBL244377

0.059 0.009 CHEMBL3544874

0.053 0.014 CHEMBL3544897

0.053 0.014 CHEMBL3544898

0.064 0.006 CHEMBL1231106

0.054 0.014 CHEMBL457723

0.054 0.014 CHEMBL3544872

0.1190.0590.119Alpha 2b adrenoreceptor antagonist

0.1 0.075 CHEMBL244377

0.088 0.087 CHEMBL457723

0.088 0.087 CHEMBL3544872

0.1140.0550.114Expectorant

0.091 0.08 CHEMBL3544874

0.102 0.067 CHEMBL1231106

0.0950.0360.099Na+ K+ transporting ATPase inhibitor

0.088 0.043 CHEMBL244377

0.075 0.055 CHEMBL3544874

0.067 0.063 CHEMBL3544897

0.067 0.063 CHEMBL3544898

0.099 0.033 CHEMBL1231106

CHEMBL1231106
0.120.0610.125 Hydroxytryptamine 2B antagonist

0.11 0.071 CHEMBL3544873

0.105 0.077 CHEMBL244377

0.12 0.06 CHEMBL3544874

0.106 0.076 CHEMBL3544897

0.106 0.076 CHEMBL3544898

0.107 0.075 CHEMBL1231106

0.109 0.073 CHEMBL457723

0.109 0.073 CHEMBL3544872

0.0730.0150.077Alpha-mannosidase inhibitor

0.056 0.033 CHEMBL3544873

0.075 0.014 CHEMBL244377

0.064 0.022 CHEMBL3544874

0.065 0.021 CHEMBL3544897

0.065 0.021 CHEMBL3544898

0.077 0.013 CHEMBL1231106

0.064 0.022 CHEMBL457723

0.064 0.022 CHEMBL3544872

CHEMBL1231106
0.1440.0860.225Cyclin-dependent kinase 8 inhibitor

0.192 0.041 CHEMBL3544873

0.207 0.031 CHEMBL244377

0.166 0.064 CHEMBL3544874

0.225 0.023 CHEMBL3544897

0.225 0.023 CHEMBL3544898

0.187 0.045 CHEMBL1231106

0.177 0.054 CHEMBL457723

0.177 0.054 CHEMBL3544872

CHEMBL3544898
0.1130.0550.113AMP-activated protein kinase stimulant

0.098 0.072 CHEMBL1231106

0.0710.0130.071Glutamate (mGluR5) agonist

0.047 0.03 CHEMBL244377

0.055 0.021 CHEMBL457723

0.055 0.021 CHEMBL3544872

0.1280.070.128Antibacterial (Helicobacter pylori)

0.113 0.092 CHEMBL244377

0.1080.050.108Estrogen receptor beta antagonist
0.0950.0370.095Glycine receptor antagonist

0.086 0.047 CHEMBL244377

0.092 0.04 CHEMBL1231106

0.0720.0150.072Glutamate (mGluR group I) agonist

0.049 0.031 CHEMBL244377

0.059 0.023 CHEMBL457723

0.059 0.023 CHEMBL3544872

0.070.0140.07Squalene epoxidase inhibitor
0.120.0630.12Calcium channel N-type blocker

0.102 0.091 CHEMBL244377

0.11 0.077 CHEMBL457723

0.11 0.077 CHEMBL3544872

0.1060.0490.227HIV-1 integrase (Overall Integration) inhibitor

0.104 0.051 CHEMBL244377

0.125 0.037 CHEMBL3544874

0.122 0.038 CHEMBL3544897

0.122 0.038 CHEMBL3544898

0.227 0.007 CHEMBL1231106

CHEMBL1231106
0.1140.0580.141Protein kinase C gamma inhibitor

0.102 0.073 CHEMBL3544873

0.131 0.044 CHEMBL244377

0.12 0.052 CHEMBL3544874

0.134 0.042 CHEMBL3544897

0.134 0.042 CHEMBL3544898

0.141 0.037 CHEMBL1231106

0.1 0.076 CHEMBL457723

0.1 0.076 CHEMBL3544872

CHEMBL1231106
0.0910.0350.091CC chemokine 5 receptor agonist

0.084 0.052 CHEMBL244377

0.083 0.054 CHEMBL1231106

0.060.0050.06DNA topoisomerase IV inhibitor

0.033 0.014 CHEMBL3544874

0.034 0.013 CHEMBL457723

0.034 0.013 CHEMBL3544872

0.2030.1480.20312-Lipoxygenase inhibitor
0.10.0450.155Phosphodiesterase IV inhibitor

0.094 0.05 CHEMBL3544873

0.136 0.027 CHEMBL244377

0.081 0.061 CHEMBL3544897

0.081 0.061 CHEMBL3544898

0.155 0.021 CHEMBL457723

0.155 0.021 CHEMBL3544872

CHEMBL3544872
0.0780.0230.086Carbonic anhydrase VB inhibitor

0.077 0.024 CHEMBL244377

0.057 0.038 CHEMBL3544874

0.054 0.041 CHEMBL3544897

0.054 0.041 CHEMBL3544898

0.086 0.02 CHEMBL1231106

0.052 0.043 CHEMBL457723

0.052 0.043 CHEMBL3544872

CHEMBL1231106
0.1080.0550.121Gastric antisecretory

0.121 0.042 CHEMBL244377

0.09 0.078 CHEMBL1231106

CHEMBL244377
0.1370.0850.145Cytidine deaminase inhibitor

0.145 0.079 CHEMBL1231106

CHEMBL1231106
0.1050.0540.353CDK2/cyclin A inhibitor

0.171 0.02 CHEMBL3544873

0.227 0.011 CHEMBL244377

0.142 0.029 CHEMBL3544874

0.252 0.009 CHEMBL3544897

0.252 0.009 CHEMBL3544898

0.353 0.005 CHEMBL1231106

0.146 0.028 CHEMBL457723

0.146 0.028 CHEMBL3544872

CHEMBL1231106
0.0610.0090.071Diamine oxidase inhibitor

0.05 0.015 CHEMBL3544873

0.067 0.007 CHEMBL244377

0.065 0.008 CHEMBL3544874

0.069 0.007 CHEMBL3544897

0.069 0.007 CHEMBL3544898

0.071 0.006 CHEMBL1231106

0.048 0.016 CHEMBL457723

0.048 0.016 CHEMBL3544872

CHEMBL1231106
0.0840.0340.151Carbonic anhydrase VA inhibitor

0.082 0.035 CHEMBL3544873

0.151 0.01 CHEMBL244377

0.066 0.051 CHEMBL3544874

0.12 0.018 CHEMBL3544897

0.12 0.018 CHEMBL3544898

0.098 0.026 CHEMBL1231106

0.11 0.021 CHEMBL457723

0.11 0.021 CHEMBL3544872

CHEMBL244377
0.1260.0760.126NADPH oxidase inhibitor

0.119 0.084 CHEMBL1231106

0.1150.0660.147Microtubule formation inhibitor

0.147 0.039 CHEMBL244377

0.11 0.074 CHEMBL3544897

0.11 0.074 CHEMBL3544898

0.12 0.061 CHEMBL1231106

0.11 0.074 CHEMBL457723

0.11 0.074 CHEMBL3544872

CHEMBL244377
0.060.010.104Inosine monophosphate dehydrogenase inhibitor

0.072 0.008 CHEMBL3544873

0.097 0.005 CHEMBL244377

0.044 0.019 CHEMBL3544874

0.066 0.009 CHEMBL3544897

0.066 0.009 CHEMBL3544898

0.04 0.022 CHEMBL1231106

0.104 0.005 CHEMBL457723

0.104 0.005 CHEMBL3544872

CHEMBL3544872
0.0750.0260.075Glutamate (mGluR1) antagonist

0.07 0.03 CHEMBL244377

0.067 0.033 CHEMBL457723

0.067 0.033 CHEMBL3544872

0.060.0110.062Guanylate cyclase inhibitor

0.041 0.032 CHEMBL244377

0.039 0.035 CHEMBL3544874

0.062 0.01 CHEMBL1231106

CHEMBL1231106
0.0570.0080.057Integrin alpha2 antagonist

0.042 0.018 CHEMBL3544874

0.041 0.019 CHEMBL457723

0.041 0.019 CHEMBL3544872

0.0590.0110.07Alpha 1d adrenoreceptor agonist

0.07 0.007 CHEMBL244377

0.04 0.026 CHEMBL3544897

0.04 0.026 CHEMBL3544898

0.063 0.01 CHEMBL1231106

0.041 0.024 CHEMBL457723

0.041 0.024 CHEMBL3544872

CHEMBL244377
0.1180.0690.118Acetylcholine muscarinic antagonist
0.0730.0250.073Acetylcholine muscarinic agonist

0.048 0.045 CHEMBL244377

0.049 0.044 CHEMBL3544874

0.0630.0150.071Mannosidase inhibitor

0.044 0.034 CHEMBL3544873

0.066 0.014 CHEMBL244377

0.054 0.022 CHEMBL3544874

0.056 0.02 CHEMBL3544897

0.056 0.02 CHEMBL3544898

0.071 0.011 CHEMBL1231106

0.052 0.023 CHEMBL457723

0.052 0.023 CHEMBL3544872

CHEMBL1231106
0.2020.1550.202Prostaglandin dehydrogenase inhibitor
0.0520.0050.091Tryptophan 5 hydroxylase inhibitor

0.079 0.003 CHEMBL3544873

0.065 0.004 CHEMBL244377

0.071 0.003 CHEMBL3544874

0.091 0.003 CHEMBL3544897

0.091 0.003 CHEMBL3544898

0.091 0.003 CHEMBL1231106

0.058 0.004 CHEMBL457723

0.058 0.004 CHEMBL3544872

CHEMBL1231106
0.070.0230.102Prolactin release inhibitor

0.08 0.011 CHEMBL3544873

0.085 0.008 CHEMBL244377

0.081 0.01 CHEMBL3544874

0.092 0.006 CHEMBL3544897

0.092 0.006 CHEMBL3544898

0.102 0.004 CHEMBL1231106

0.072 0.02 CHEMBL457723

0.072 0.02 CHEMBL3544872

CHEMBL1231106
0.0710.0240.071Phosphodiesterase 1A inhibitor

0.065 0.031 CHEMBL244377

0.061 0.038 CHEMBL3544874

0.057 0.049 CHEMBL3544897

0.057 0.049 CHEMBL3544898

0.07 0.025 CHEMBL1231106

0.0810.0330.085Phospholipase D inhibitor

0.073 0.046 CHEMBL244377

0.085 0.027 CHEMBL1231106

CHEMBL1231106
0.130.0830.145Protein kinase stimulant

0.145 0.072 CHEMBL244377

0.122 0.091 CHEMBL1231106

CHEMBL244377
0.1250.0780.153Phosphodiesterase inhibitor

0.113 0.09 CHEMBL244377

0.153 0.056 CHEMBL457723

0.153 0.056 CHEMBL3544872

CHEMBL3544872
0.1340.0880.137Pregnane X receptor agonist

0.137 0.081 CHEMBL244377

0.129 0.103 CHEMBL1231106

CHEMBL244377
0.0860.040.086Estrogen receptor alpha antagonist
0.0710.0250.147Ornithine carbamoyltransferase inhibitor

0.046 0.043 CHEMBL3544873

0.067 0.027 CHEMBL244377

0.079 0.022 CHEMBL3544874

0.071 0.025 CHEMBL3544897

0.071 0.025 CHEMBL3544898

0.147 0.01 CHEMBL1231106

CHEMBL1231106
0.090.0440.135D-Ala-D-Ala ligase inhibitor

0.086 0.054 CHEMBL3544873

0.099 0.03 CHEMBL244377

0.099 0.031 CHEMBL3544874

0.107 0.022 CHEMBL3544897

0.107 0.022 CHEMBL3544898

0.135 0.008 CHEMBL1231106

0.079 0.071 CHEMBL457723

0.079 0.071 CHEMBL3544872

CHEMBL1231106
0.0670.0210.0675 Hydroxytryptamine 2 agonist

0.046 0.043 CHEMBL457723

0.046 0.043 CHEMBL3544872

0.0660.0210.099Epithelial sodium channel blocker

0.052 0.045 CHEMBL3544873

0.064 0.024 CHEMBL244377

0.072 0.017 CHEMBL3544874

0.068 0.02 CHEMBL3544897

0.068 0.02 CHEMBL3544898

0.099 0.007 CHEMBL1231106

CHEMBL1231106
0.1690.1240.169Antiamyloidogenic
0.0660.0220.234Histamine agonist

0.154 0.005 CHEMBL3544873

0.129 0.006 CHEMBL244377

0.119 0.007 CHEMBL3544874

0.234 0.004 CHEMBL3544897

0.234 0.004 CHEMBL3544898

0.146 0.005 CHEMBL1231106

0.086 0.012 CHEMBL457723

0.086 0.012 CHEMBL3544872

CHEMBL3544898
0.0750.0310.113Glutamate (mGluR6) antagonist

0.073 0.034 CHEMBL244377

0.075 0.031 CHEMBL3544874

0.071 0.038 CHEMBL3544897

0.071 0.038 CHEMBL3544898

0.113 0.007 CHEMBL1231106

CHEMBL1231106
0.0560.0120.056Nociceptin (N/OFQ) receptor antagonist

0.046 0.016 CHEMBL457723

0.046 0.016 CHEMBL3544872

0.0870.0430.112Nicotinic alpha4beta2 receptor antagonist

0.093 0.038 CHEMBL244377

0.081 0.049 CHEMBL3544874

0.086 0.044 CHEMBL3544897

0.086 0.044 CHEMBL3544898

0.112 0.022 CHEMBL1231106

CHEMBL1231106
0.0590.0160.065Dopamine beta hydroxylase inhibitor

0.051 0.029 CHEMBL244377

0.051 0.029 CHEMBL3544874

0.065 0.011 CHEMBL1231106

CHEMBL1231106
0.0580.0150.093Cytokine production stimulant

0.048 0.034 CHEMBL3544873

0.048 0.033 CHEMBL244377

0.069 0.007 CHEMBL3544874

0.056 0.018 CHEMBL3544897

0.056 0.018 CHEMBL3544898

0.093 0.004 CHEMBL1231106

CHEMBL1231106
0.0950.0520.095Calcium antagonist

0.077 0.066 CHEMBL244377

0.088 0.057 CHEMBL1231106

0.1530.1110.573Clk dual-specificity kinase inhibitor

0.421 0.016 CHEMBL3544873

0.422 0.015 CHEMBL244377

0.343 0.029 CHEMBL3544874

0.502 0.007 CHEMBL3544897

0.502 0.007 CHEMBL3544898

0.573 0.005 CHEMBL1231106

0.317 0.035 CHEMBL457723

0.317 0.035 CHEMBL3544872

CHEMBL1231106
0.1450.1030.259LIM domain kinase 1 inhibitor

0.189 0.068 CHEMBL3544873

0.217 0.055 CHEMBL244377

0.198 0.064 CHEMBL3544874

0.258 0.034 CHEMBL3544897

0.258 0.034 CHEMBL3544898

0.259 0.034 CHEMBL1231106

0.144 0.104 CHEMBL457723

0.144 0.104 CHEMBL3544872

CHEMBL1231106
0.0630.0210.063Acetylcholine M1 receptor agonist

0.037 0.036 CHEMBL244377

0.038 0.035 CHEMBL457723

0.038 0.035 CHEMBL3544872

0.0530.0110.057Kainate receptor agonist

0.054 0.01 CHEMBL244377

0.046 0.02 CHEMBL3544874

0.045 0.021 CHEMBL3544897

0.045 0.021 CHEMBL3544898

0.057 0.009 CHEMBL1231106

0.045 0.02 CHEMBL457723

0.045 0.02 CHEMBL3544872

CHEMBL1231106
0.0730.0310.081Carbonic anhydrase IX inhibitor

0.058 0.038 CHEMBL3544873

0.069 0.033 CHEMBL244377

0.051 0.042 CHEMBL3544874

0.052 0.041 CHEMBL1231106

0.081 0.026 CHEMBL457723

0.081 0.026 CHEMBL3544872

CHEMBL3544872
0.0780.0360.078Acetylcholine M5 receptor agonist

0.061 0.055 CHEMBL1231106

0.0590.0180.092Thymidylate synthase inhibitor

0.073 0.01 CHEMBL3544873

0.061 0.016 CHEMBL244377

0.081 0.007 CHEMBL3544874

0.082 0.007 CHEMBL3544897

0.082 0.007 CHEMBL3544898

0.092 0.005 CHEMBL1231106

0.051 0.026 CHEMBL457723

0.051 0.026 CHEMBL3544872

CHEMBL1231106
0.0870.0450.087NAD(P)H dehydrogenase (quinone) inhibitor

0.069 0.062 CHEMBL244377

0.086 0.046 CHEMBL1231106

0.070.0290.07Calcium channel P-type blocker

0.061 0.054 CHEMBL244377

0.066 0.036 CHEMBL1231106

0.0570.0160.061Geranyltranstransferase inhibitor

0.061 0.013 CHEMBL244377

0.042 0.034 CHEMBL3544897

0.042 0.034 CHEMBL3544898

0.056 0.017 CHEMBL1231106

0.042 0.033 CHEMBL457723

0.042 0.033 CHEMBL3544872

CHEMBL244377
0.0630.0220.151Adenosine A2b receptor antagonist

0.151 0.006 CHEMBL3544873

0.087 0.012 CHEMBL244377

0.097 0.01 CHEMBL3544874

0.138 0.007 CHEMBL3544897

0.138 0.007 CHEMBL3544898

0.095 0.011 CHEMBL1231106

0.094 0.011 CHEMBL457723

0.094 0.011 CHEMBL3544872

CHEMBL3544873
0.0540.0140.054Nerve growth factor antagonist

0.053 0.015 CHEMBL244377

0.039 0.037 CHEMBL3544874

0.04 0.035 CHEMBL3544897

0.04 0.035 CHEMBL3544898

0.052 0.016 CHEMBL1231106

0.039 0.038 CHEMBL457723

0.039 0.038 CHEMBL3544872

0.1130.0720.239Interleukin 8 antagonist

0.176 0.021 CHEMBL3544873

0.211 0.01 CHEMBL244377

0.132 0.048 CHEMBL3544874

0.239 0.007 CHEMBL3544897

0.239 0.007 CHEMBL3544898

0.181 0.019 CHEMBL1231106

0.153 0.032 CHEMBL457723

0.153 0.032 CHEMBL3544872

CHEMBL3544898
0.0620.0220.093Potassium channel (Inward rectifier) blocker

0.052 0.031 CHEMBL3544873

0.093 0.008 CHEMBL244377

0.066 0.02 CHEMBL3544897

0.066 0.02 CHEMBL3544898

0.048 0.037 CHEMBL1231106

0.079 0.013 CHEMBL457723

0.079 0.013 CHEMBL3544872

CHEMBL244377
0.0690.0290.182Cyclin H inhibitor

0.102 0.007 CHEMBL3544873

0.182 0.003 CHEMBL244377

0.129 0.004 CHEMBL3544897

0.129 0.004 CHEMBL3544898

0.054 0.047 CHEMBL1231106

0.128 0.004 CHEMBL457723

0.128 0.004 CHEMBL3544872

CHEMBL244377
0.1030.0630.226Carbonic anhydrase XV inhibitor

0.107 0.059 CHEMBL244377

0.126 0.042 CHEMBL3544874

0.127 0.041 CHEMBL3544897

0.127 0.041 CHEMBL3544898

0.226 0.015 CHEMBL1231106

CHEMBL1231106
0.0770.0370.162Carbonic anhydrase V inhibitor

0.073 0.04 CHEMBL3544873

0.162 0.012 CHEMBL244377

0.058 0.056 CHEMBL3544874

0.124 0.02 CHEMBL3544897

0.124 0.02 CHEMBL3544898

0.098 0.028 CHEMBL1231106

0.109 0.024 CHEMBL457723

0.109 0.024 CHEMBL3544872

CHEMBL244377
0.0440.0050.044Integrin alpha2beta1 antagonist

0.025 0.022 CHEMBL244377

0.033 0.01 CHEMBL3544874

0.024 0.023 CHEMBL1231106

0.031 0.012 CHEMBL457723

0.031 0.012 CHEMBL3544872

0.0830.0430.107GABA aminotransferase inhibitor

0.078 0.05 CHEMBL244377

0.078 0.049 CHEMBL3544874

0.071 0.059 CHEMBL3544897

0.071 0.059 CHEMBL3544898

0.107 0.023 CHEMBL1231106

CHEMBL1231106
0.0450.0070.045Adenosine uptake inhibitor

0.036 0.021 CHEMBL3544873

0.043 0.008 CHEMBL244377

0.037 0.017 CHEMBL3544874

0.036 0.02 CHEMBL3544897

0.036 0.02 CHEMBL3544898

0.036 0.02 CHEMBL1231106

0.042 0.009 CHEMBL457723

0.042 0.009 CHEMBL3544872

0.0680.030.093Cyclin D1 inhibitor

0.057 0.048 CHEMBL3544873

0.086 0.014 CHEMBL244377

0.066 0.034 CHEMBL3544874

0.082 0.016 CHEMBL3544897

0.082 0.016 CHEMBL3544898

0.093 0.01 CHEMBL1231106

0.061 0.041 CHEMBL457723

0.061 0.041 CHEMBL3544872

CHEMBL1231106
0.0510.0140.0743-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.044 0.023 CHEMBL3544873

0.063 0.006 CHEMBL244377

0.051 0.014 CHEMBL3544874

0.061 0.007 CHEMBL3544897

0.061 0.007 CHEMBL3544898

0.074 0.004 CHEMBL1231106

0.045 0.021 CHEMBL457723

0.045 0.021 CHEMBL3544872

CHEMBL1231106
0.0490.0120.0492,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0840.0470.205Carbonic anhydrase XIII inhibitor

0.089 0.044 CHEMBL3544873

0.205 0.013 CHEMBL244377

0.154 0.021 CHEMBL3544897

0.154 0.021 CHEMBL3544898

0.118 0.03 CHEMBL1231106

0.122 0.029 CHEMBL457723

0.122 0.029 CHEMBL3544872

CHEMBL244377
0.0520.0160.145Dihydropteroate synthase inhibitor

0.086 0.005 CHEMBL3544873

0.077 0.007 CHEMBL244377

0.092 0.005 CHEMBL3544874

0.139 0.004 CHEMBL3544897

0.139 0.004 CHEMBL3544898

0.145 0.004 CHEMBL1231106

0.051 0.016 CHEMBL457723

0.051 0.016 CHEMBL3544872

CHEMBL1231106
0.0570.0210.212Histamine H4 receptor antagonist

0.141 0.004 CHEMBL3544873

0.104 0.005 CHEMBL244377

0.09 0.006 CHEMBL3544874

0.212 0.003 CHEMBL3544897

0.212 0.003 CHEMBL3544898

0.098 0.005 CHEMBL1231106

0.08 0.008 CHEMBL457723

0.08 0.008 CHEMBL3544872

CHEMBL3544898
0.050.0140.097Fumarate hydratase inhibitor

0.039 0.019 CHEMBL244377

0.048 0.014 CHEMBL3544874

0.039 0.019 CHEMBL3544897

0.039 0.019 CHEMBL3544898

0.097 0.005 CHEMBL1231106

CHEMBL1231106
0.0610.0250.112Proto-oncogene tyrosine-protein kinase Met inhibitor

0.06 0.026 CHEMBL244377

0.043 0.039 CHEMBL3544874

0.046 0.036 CHEMBL3544897

0.046 0.036 CHEMBL3544898

0.112 0.007 CHEMBL1231106

CHEMBL1231106
0.0560.0210.073Adenylate cyclase 1 inhibitor

0.069 0.012 CHEMBL244377

0.044 0.036 CHEMBL3544897

0.044 0.036 CHEMBL3544898

0.073 0.01 CHEMBL1231106

CHEMBL1231106
0.090.0550.09Acetylcholine agonist

0.075 0.073 CHEMBL244377

0.0490.0140.049Orexin receptor 2 antagonist
0.0650.030.065Cyclin E1 inhibitor

0.043 0.041 CHEMBL3544873

0.064 0.03 CHEMBL457723

0.064 0.03 CHEMBL3544872

0.0530.0190.104AICAR transformylase inhibitor

0.054 0.018 CHEMBL3544873

0.048 0.024 CHEMBL244377

0.075 0.008 CHEMBL3544874

0.068 0.011 CHEMBL3544897

0.068 0.011 CHEMBL3544898

0.104 0.005 CHEMBL1231106

CHEMBL1231106
0.0460.0120.065Potassium channel small-conductance Ca-activated activator

0.06 0.008 CHEMBL244377

0.035 0.018 CHEMBL3544874

0.043 0.013 CHEMBL3544897

0.043 0.013 CHEMBL3544898

0.065 0.008 CHEMBL1231106

0.034 0.019 CHEMBL457723

0.034 0.019 CHEMBL3544872

CHEMBL1231106
0.0650.0320.07Carbonic anhydrase I inhibitor

0.05 0.043 CHEMBL3544873

0.064 0.032 CHEMBL244377

0.049 0.044 CHEMBL3544874

0.052 0.041 CHEMBL1231106

0.07 0.029 CHEMBL457723

0.07 0.029 CHEMBL3544872

CHEMBL3544872
0.050.0170.05Alpha 1L adrenoreceptor agonist
0.1080.0750.108TRPA1 agonist

0.098 0.092 CHEMBL1231106

0.0380.0050.064Inosine monophosphate dehydrogenase 2 inhibitor

0.049 0.005 CHEMBL3544873

0.057 0.004 CHEMBL244377

0.027 0.009 CHEMBL3544874

0.043 0.005 CHEMBL3544897

0.043 0.005 CHEMBL3544898

0.021 0.012 CHEMBL1231106

0.064 0.004 CHEMBL457723

0.064 0.004 CHEMBL3544872

CHEMBL3544872
0.0430.0110.043Liver X receptor beta antagonist
0.040.0070.05Purinergic P2Y15 antagonist

0.031 0.015 CHEMBL3544873

0.039 0.007 CHEMBL244377

0.039 0.008 CHEMBL3544874

0.038 0.008 CHEMBL3544897

0.038 0.008 CHEMBL3544898

0.05 0.004 CHEMBL1231106

0.032 0.014 CHEMBL457723

0.032 0.014 CHEMBL3544872

CHEMBL1231106
0.0710.0390.118Potassium channel (ATP-sensitive) blocker

0.085 0.024 CHEMBL3544873

0.118 0.009 CHEMBL244377

0.069 0.043 CHEMBL3544874

0.113 0.011 CHEMBL3544897

0.113 0.011 CHEMBL3544898

0.085 0.024 CHEMBL1231106

0.09 0.02 CHEMBL457723

0.09 0.02 CHEMBL3544872

CHEMBL244377
0.0760.0440.099Glycine receptor agonist

0.099 0.021 CHEMBL1231106

CHEMBL1231106
0.0430.0110.082Hypoxanthine phosphoribosyltransferase inhibitor

0.039 0.013 CHEMBL3544873

0.039 0.013 CHEMBL244377

0.057 0.007 CHEMBL3544874

0.052 0.008 CHEMBL3544897

0.052 0.008 CHEMBL3544898

0.082 0.004 CHEMBL1231106

0.027 0.02 CHEMBL457723

0.027 0.02 CHEMBL3544872

CHEMBL1231106
0.130.10.167Sphingosine 1-phosphate receptor 5 antagonist

0.135 0.089 CHEMBL244377

0.167 0.037 CHEMBL1231106

CHEMBL1231106
0.0390.0080.042Nicotinic alpha4beta2 receptor agonist

0.042 0.007 CHEMBL244377

0.027 0.022 CHEMBL3544874

0.029 0.019 CHEMBL3544897

0.029 0.019 CHEMBL3544898

0.032 0.015 CHEMBL1231106

0.034 0.012 CHEMBL457723

0.034 0.012 CHEMBL3544872

CHEMBL244377
0.050.020.094Glutamate (mGluR1a) antagonist

0.066 0.012 CHEMBL3544873

0.094 0.005 CHEMBL244377

0.047 0.023 CHEMBL3544874

0.088 0.007 CHEMBL3544897

0.088 0.007 CHEMBL3544898

0.057 0.016 CHEMBL1231106

0.072 0.01 CHEMBL457723

0.072 0.01 CHEMBL3544872

CHEMBL244377
0.0670.0370.075Transcription factor RelA inhibitor

0.061 0.052 CHEMBL3544874

0.075 0.023 CHEMBL1231106

CHEMBL1231106
0.0970.0670.221Cyclin-dependent kinase 9 inhibitor

0.163 0.03 CHEMBL3544873

0.155 0.032 CHEMBL244377

0.136 0.039 CHEMBL3544874

0.221 0.018 CHEMBL3544897

0.221 0.018 CHEMBL3544898

0.184 0.026 CHEMBL1231106

0.111 0.052 CHEMBL457723

0.111 0.052 CHEMBL3544872

CHEMBL3544898
0.1040.0740.231MAP kinase 13 inhibitor

0.227 0.014 CHEMBL3544873

0.221 0.016 CHEMBL244377

0.128 0.049 CHEMBL3544874

0.219 0.016 CHEMBL3544897

0.219 0.016 CHEMBL3544898

0.113 0.063 CHEMBL1231106

0.231 0.014 CHEMBL457723

0.231 0.014 CHEMBL3544872

CHEMBL3544872
0.1140.0840.12Cyclooxygenase 3 inhibitor

0.12 0.077 CHEMBL1231106

CHEMBL1231106
0.0670.0370.067Cyclin E inhibitor

0.051 0.047 CHEMBL3544873

0.066 0.038 CHEMBL457723

0.066 0.038 CHEMBL3544872

0.0340.0040.034Alpha 2c adrenoreceptor agonist

0.024 0.007 CHEMBL3544873

0.023 0.008 CHEMBL244377

0.031 0.005 CHEMBL3544874

0.02 0.011 CHEMBL3544897

0.02 0.011 CHEMBL3544898

0.026 0.006 CHEMBL1231106

0.027 0.005 CHEMBL457723

0.027 0.005 CHEMBL3544872

0.0650.0350.109Carbonic anhydrase stimulant

0.069 0.032 CHEMBL244377

0.067 0.033 CHEMBL3544874

0.07 0.032 CHEMBL3544897

0.07 0.032 CHEMBL3544898

0.109 0.016 CHEMBL1231106

CHEMBL1231106
0.040.010.04Nicotinic alpha3beta4 receptor agonist

0.033 0.017 CHEMBL244377

0.027 0.025 CHEMBL3544874

0.037 0.012 CHEMBL1231106

0.0450.0160.131Phosphoglycerate kinase inhibitor

0.102 0.007 CHEMBL3544873

0.097 0.007 CHEMBL244377

0.068 0.01 CHEMBL3544874

0.131 0.005 CHEMBL3544897

0.131 0.005 CHEMBL3544898

0.103 0.007 CHEMBL1231106

0.072 0.009 CHEMBL457723

0.072 0.009 CHEMBL3544872

CHEMBL3544898
0.1070.0780.107Cholesterol synthesis inhibitor
0.0880.0590.088Bromodomain-containing protein 2 inhibitor

0.084 0.068 CHEMBL244377

0.086 0.062 CHEMBL1231106

0.0870.0580.137Insulin growth factor antagonist

0.089 0.055 CHEMBL3544873

0.137 0.026 CHEMBL244377

0.076 0.072 CHEMBL3544874

0.12 0.034 CHEMBL3544897

0.12 0.034 CHEMBL3544898

0.102 0.045 CHEMBL1231106

0.105 0.043 CHEMBL457723

0.105 0.043 CHEMBL3544872

CHEMBL244377
0.0730.0450.126Secretase beta inhibitor

0.068 0.054 CHEMBL244377

0.089 0.026 CHEMBL3544874

0.083 0.032 CHEMBL3544897

0.083 0.032 CHEMBL3544898

0.126 0.009 CHEMBL1231106

CHEMBL1231106
0.1190.090.119Vanilloid 1 agonist

0.114 0.103 CHEMBL244377

0.118 0.093 CHEMBL1231106

0.0460.0180.046Vascular adhesion protein 1 inhibitor

0.037 0.03 CHEMBL244377

0.046 0.019 CHEMBL1231106

0.110.0820.219MAP kinase 12 inhibitor

0.211 0.019 CHEMBL3544873

0.21 0.02 CHEMBL244377

0.127 0.061 CHEMBL3544874

0.203 0.022 CHEMBL3544897

0.203 0.022 CHEMBL3544898

0.114 0.078 CHEMBL1231106

0.219 0.017 CHEMBL457723

0.219 0.017 CHEMBL3544872

CHEMBL3544872
0.0470.0190.047Heme oxygenase inhibitor

0.045 0.022 CHEMBL1231106

0.0620.0340.067Carbonic anhydrase II inhibitor

0.063 0.033 CHEMBL244377

0.049 0.045 CHEMBL1231106

0.067 0.031 CHEMBL457723

0.067 0.031 CHEMBL3544872

CHEMBL3544872
0.0720.0440.076Protein kinase C beta inhibitor

0.076 0.036 CHEMBL244377

0.066 0.057 CHEMBL3544897

0.066 0.057 CHEMBL3544898

0.073 0.041 CHEMBL1231106

CHEMBL244377
0.0620.0350.075Cyclin A1 inhibitor

0.062 0.035 CHEMBL3544873

0.064 0.031 CHEMBL244377

0.066 0.028 CHEMBL3544874

0.067 0.026 CHEMBL3544897

0.067 0.026 CHEMBL3544898

0.075 0.017 CHEMBL1231106

0.059 0.041 CHEMBL457723

0.059 0.041 CHEMBL3544872

CHEMBL1231106
0.1210.0940.15Sphingosine 1-phosphate receptor 2 antagonist

0.129 0.075 CHEMBL244377

0.15 0.041 CHEMBL1231106

CHEMBL1231106
0.1940.1670.194Thyroid hormone antagonist
0.1070.0810.156Beta amyloid protein antagonist

0.118 0.069 CHEMBL244377

0.106 0.082 CHEMBL3544897

0.106 0.082 CHEMBL3544898

0.156 0.036 CHEMBL1231106

CHEMBL1231106
0.0330.0070.033Protease (Human cytomegalovirus) inhibitor

0.024 0.012 CHEMBL244377

0.0820.0550.233Carbonic anhydrase VI inhibitor

0.119 0.03 CHEMBL3544873

0.232 0.01 CHEMBL244377

0.085 0.052 CHEMBL3544874

0.233 0.01 CHEMBL3544897

0.233 0.01 CHEMBL3544898

0.183 0.015 CHEMBL1231106

0.118 0.03 CHEMBL457723

0.118 0.03 CHEMBL3544872

CHEMBL3544898
0.0640.0380.067Histone deacetylase SIRT3 inhibitor

0.067 0.033 CHEMBL244377

0.058 0.056 CHEMBL3544897

0.058 0.056 CHEMBL3544898

0.064 0.039 CHEMBL1231106

0.059 0.051 CHEMBL457723

0.059 0.051 CHEMBL3544872

CHEMBL244377
0.0830.0570.13Insulin like growth factor 1 antagonist

0.086 0.054 CHEMBL3544873

0.13 0.026 CHEMBL244377

0.074 0.071 CHEMBL3544874

0.112 0.033 CHEMBL3544897

0.112 0.033 CHEMBL3544898

0.096 0.045 CHEMBL1231106

0.1 0.042 CHEMBL457723

0.1 0.042 CHEMBL3544872

CHEMBL244377
0.0430.0180.07Glutamate (mGluR8) agonist

0.043 0.019 CHEMBL244377

0.042 0.02 CHEMBL3544874

0.04 0.022 CHEMBL3544897

0.04 0.022 CHEMBL3544898

0.07 0.005 CHEMBL1231106

CHEMBL1231106
0.1150.090.158Nav1.2 sodium channel blocker

0.115 0.09 CHEMBL3544874

0.158 0.052 CHEMBL1231106

CHEMBL1231106
0.0920.0670.131MAP kinase kinase 1 inhibitor

0.122 0.033 CHEMBL244377

0.088 0.073 CHEMBL3544874

0.116 0.038 CHEMBL3544897

0.116 0.038 CHEMBL3544898

0.131 0.026 CHEMBL1231106

CHEMBL1231106
0.0320.0070.032Vanilloid 2 agonist

0.029 0.011 CHEMBL244377

0.025 0.019 CHEMBL3544874

0.03 0.009 CHEMBL1231106

0.0520.0280.079Adenosine deaminase inhibitor

0.051 0.029 CHEMBL3544873

0.057 0.023 CHEMBL244377

0.063 0.018 CHEMBL3544874

0.066 0.016 CHEMBL3544897

0.066 0.016 CHEMBL3544898

0.079 0.009 CHEMBL1231106

CHEMBL1231106
0.0330.0090.038Hedgehog signaling activator

0.038 0.005 CHEMBL244377

0.027 0.02 CHEMBL3544874

0.032 0.01 CHEMBL3544897

0.032 0.01 CHEMBL3544898

0.032 0.01 CHEMBL1231106

0.03 0.012 CHEMBL457723

0.03 0.012 CHEMBL3544872

CHEMBL244377
0.0360.0120.036CDK4/cyclin D3 inhibitor

0.033 0.014 CHEMBL3544874

0.032 0.016 CHEMBL1231106

0.0670.0430.133Fibroblast growth factor 2 antagonist

0.109 0.021 CHEMBL3544873

0.107 0.022 CHEMBL244377

0.087 0.03 CHEMBL3544874

0.133 0.014 CHEMBL3544897

0.133 0.014 CHEMBL3544898

0.104 0.023 CHEMBL1231106

0.085 0.031 CHEMBL457723

0.085 0.031 CHEMBL3544872

CHEMBL3544898
0.0670.0430.177Tyk2 inhibitor

0.062 0.047 CHEMBL3544873

0.177 0.01 CHEMBL244377

0.094 0.03 CHEMBL3544897

0.094 0.03 CHEMBL3544898

0.11 0.024 CHEMBL457723

0.11 0.024 CHEMBL3544872

CHEMBL244377
0.0340.010.034Estrogen-related receptor gamma antagonist

0.028 0.021 CHEMBL244377

0.029 0.018 CHEMBL1231106

0.0580.0350.059Pregnane X receptor antagonist

0.054 0.049 CHEMBL244377

0.059 0.033 CHEMBL1231106

CHEMBL1231106
0.0960.0720.105Urease inhibitor

0.105 0.061 CHEMBL244377

CHEMBL244377
0.2110.1880.511Toll-Like receptor agonist

0.511 0.03 CHEMBL3544873

0.214 0.185 CHEMBL244377

0.454 0.042 CHEMBL3544874

0.451 0.043 CHEMBL3544897

0.451 0.043 CHEMBL3544898

0.415 0.054 CHEMBL1231106

0.357 0.079 CHEMBL457723

0.357 0.079 CHEMBL3544872

CHEMBL3544873
0.0340.0110.034CXC chemokine 2 receptor antagonist

0.032 0.012 CHEMBL244377

0.024 0.023 CHEMBL3544874

0.028 0.016 CHEMBL1231106

0.025 0.02 CHEMBL457723

0.025 0.02 CHEMBL3544872

0.1080.0850.108Cholinergic antagonist
0.1260.1040.126Thiol protease inhibitor

0.121 0.115 CHEMBL1231106

0.1940.1720.682Immunomodulator

0.588 0.013 CHEMBL3544873

0.357 0.057 CHEMBL244377

0.553 0.016 CHEMBL3544874

0.62 0.01 CHEMBL3544897

0.62 0.01 CHEMBL3544898

0.682 0.006 CHEMBL1231106

0.367 0.054 CHEMBL457723

0.367 0.054 CHEMBL3544872

CHEMBL1231106
0.1230.1010.132CC chemokine 6 receptor antagonist

0.132 0.063 CHEMBL244377

CHEMBL244377
0.0640.0430.158Cyclin A2 inhibitor

0.139 0.015 CHEMBL3544873

0.11 0.021 CHEMBL244377

0.097 0.025 CHEMBL3544874

0.158 0.013 CHEMBL3544897

0.158 0.013 CHEMBL3544898

0.102 0.024 CHEMBL1231106

0.099 0.025 CHEMBL457723

0.099 0.025 CHEMBL3544872

CHEMBL3544898
0.0780.0570.078Acetylcholine nicotinic antagonist
0.0440.0230.078Dopamine D5 agonist

0.045 0.022 CHEMBL244377

0.04 0.028 CHEMBL3544874

0.039 0.029 CHEMBL3544897

0.039 0.029 CHEMBL3544898

0.078 0.006 CHEMBL1231106

CHEMBL1231106
0.1110.090.116Sphingosine 1-phosphate receptor 4 antagonist

0.116 0.08 CHEMBL244377

0.113 0.086 CHEMBL1231106

CHEMBL244377
0.1060.0850.106Acetylcholine antagonist
0.0470.0260.057Oxytocin agonist

0.046 0.027 CHEMBL244377

0.039 0.033 CHEMBL3544874

0.039 0.033 CHEMBL3544897

0.039 0.033 CHEMBL3544898

0.057 0.019 CHEMBL1231106

CHEMBL1231106
0.0590.0390.086EphB4 antagonist

0.069 0.03 CHEMBL3544873

0.085 0.022 CHEMBL244377

0.061 0.037 CHEMBL3544874

0.086 0.021 CHEMBL3544897

0.086 0.021 CHEMBL3544898

0.071 0.029 CHEMBL1231106

0.068 0.031 CHEMBL457723

0.068 0.031 CHEMBL3544872

CHEMBL3544898
0.0630.0440.063Carbonic anhydrase inhibitor

0.063 0.044 CHEMBL244377

0.063 0.044 CHEMBL457723

0.063 0.044 CHEMBL3544872

0.0290.010.03Adenosine kinase inhibitor

0.019 0.017 CHEMBL3544873

0.03 0.01 CHEMBL3544874

0.02 0.016 CHEMBL1231106

0.019 0.018 CHEMBL457723

0.019 0.018 CHEMBL3544872

CHEMBL3544874
0.0830.0640.116Ornithine decarboxylase inhibitor

0.116 0.029 CHEMBL1231106

CHEMBL1231106
0.0560.0370.084Sphingosine kinase 2 inhibitor

0.051 0.046 CHEMBL244377

0.084 0.013 CHEMBL1231106

CHEMBL1231106
0.0510.0320.051Topoisomerase II beta inhibitor

0.045 0.043 CHEMBL244377

0.048 0.035 CHEMBL1231106

0.0670.0480.165CDC7 inhibitor

0.126 0.014 CHEMBL3544873

0.107 0.02 CHEMBL244377

0.107 0.02 CHEMBL3544874

0.165 0.008 CHEMBL3544897

0.165 0.008 CHEMBL3544898

0.151 0.01 CHEMBL1231106

0.084 0.033 CHEMBL457723

0.084 0.033 CHEMBL3544872

CHEMBL3544898
0.060.0410.074Androgen agonist

0.074 0.027 CHEMBL244377

0.058 0.044 CHEMBL1231106

CHEMBL244377
0.0820.0630.185Myeloperoxidase inhibitor

0.096 0.04 CHEMBL3544873

0.095 0.041 CHEMBL244377

0.117 0.021 CHEMBL3544874

0.136 0.014 CHEMBL3544897

0.136 0.014 CHEMBL3544898

0.185 0.006 CHEMBL1231106

CHEMBL1231106
0.1180.0990.166Activin receptor-like kinase 2 inhibitor

0.145 0.071 CHEMBL244377

0.119 0.097 CHEMBL3544874

0.144 0.072 CHEMBL3544897

0.144 0.072 CHEMBL3544898

0.166 0.055 CHEMBL1231106

CHEMBL1231106
0.0540.0350.056Carbonic anhydrase XII inhibitor

0.048 0.04 CHEMBL244377

0.056 0.035 CHEMBL457723

0.056 0.035 CHEMBL3544872

CHEMBL3544872
0.030.0120.032Glucosylceramidase stimulant

0.032 0.009 CHEMBL244377

0.029 0.015 CHEMBL457723

0.029 0.015 CHEMBL3544872

CHEMBL244377
0.0330.0150.033Integrin alpha4 antagonist
0.0430.0250.063Thymidine kinase inhibitor

0.046 0.022 CHEMBL244377

0.041 0.029 CHEMBL3544874

0.042 0.026 CHEMBL3544897

0.042 0.026 CHEMBL3544898

0.063 0.013 CHEMBL1231106

CHEMBL1231106
0.0690.0510.069Amidase inhibitor
0.0410.0230.041CF transmembrane conductance regulator antagonist
0.0890.0720.13Xanthine oxidase inhibitor

0.089 0.072 CHEMBL3544874

0.13 0.042 CHEMBL1231106

CHEMBL1231106
0.0220.0050.201Tryptophan hydroxylase 1 inhibitor

0.037 0.003 CHEMBL3544873

0.029 0.004 CHEMBL244377

0.041 0.003 CHEMBL3544874

0.055 0.002 CHEMBL3544897

0.055 0.002 CHEMBL3544898

0.201 0.001 CHEMBL1231106

0.023 0.005 CHEMBL457723

0.023 0.005 CHEMBL3544872

CHEMBL1231106
0.0410.0250.048Membrane dipeptidase inhibitor

0.039 0.027 CHEMBL244377

0.048 0.017 CHEMBL1231106

CHEMBL1231106
0.0390.0230.059Arginase inhibitor

0.048 0.016 CHEMBL244377

0.04 0.022 CHEMBL3544874

0.048 0.016 CHEMBL3544897

0.048 0.016 CHEMBL3544898

0.059 0.011 CHEMBL1231106

CHEMBL1231106
0.0780.0620.084Neuropeptide Y antagonist

0.084 0.052 CHEMBL457723

0.084 0.052 CHEMBL3544872

CHEMBL3544872
0.10.0840.1Calcium channel (voltage-sensitive) blocker
0.0240.0080.047Toll-Like receptor 8 agonist

0.047 0.004 CHEMBL3544873

0.024 0.008 CHEMBL244377

0.043 0.004 CHEMBL3544874

0.04 0.004 CHEMBL3544897

0.04 0.004 CHEMBL3544898

0.045 0.004 CHEMBL1231106

0.025 0.007 CHEMBL457723

0.025 0.007 CHEMBL3544872

CHEMBL3544873
0.0740.0580.114Fibroblast growth factor 3 antagonist

0.103 0.031 CHEMBL3544873

0.099 0.033 CHEMBL244377

0.083 0.047 CHEMBL3544874

0.114 0.026 CHEMBL3544897

0.114 0.026 CHEMBL3544898

0.086 0.044 CHEMBL1231106

0.091 0.039 CHEMBL457723

0.091 0.039 CHEMBL3544872

CHEMBL3544898
0.0340.0180.073Endothelial nitric-oxide synthase inhibitor

0.038 0.014 CHEMBL3544873

0.039 0.014 CHEMBL244377

0.054 0.008 CHEMBL3544874

0.06 0.007 CHEMBL3544897

0.06 0.007 CHEMBL3544898

0.073 0.005 CHEMBL1231106

CHEMBL1231106
0.0580.0430.058Gonadotropin-releasing hormone receptor agonist

0.055 0.052 CHEMBL3544874

0.060.0450.0765 Hydroxytryptamine 5A antagonist

0.076 0.026 CHEMBL244377

0.067 0.035 CHEMBL3544897

0.067 0.035 CHEMBL3544898

0.061 0.044 CHEMBL1231106

0.059 0.047 CHEMBL457723

0.059 0.047 CHEMBL3544872

CHEMBL244377
0.0710.0560.078Alpha 2a adrenoreceptor antagonist

0.078 0.05 CHEMBL244377

0.073 0.054 CHEMBL457723

0.073 0.054 CHEMBL3544872

CHEMBL244377
0.1840.1690.184Thyroid hormone beta antagonist
0.0460.0310.227CDK7/cyclin H inhibitor

0.054 0.02 CHEMBL3544873

0.227 0.004 CHEMBL244377

0.079 0.008 CHEMBL3544897

0.079 0.008 CHEMBL3544898

0.083 0.007 CHEMBL457723

0.083 0.007 CHEMBL3544872

CHEMBL244377
0.0630.0480.064Aryl hydrocarbon receptor antagonist

0.064 0.046 CHEMBL244377

CHEMBL244377
0.0720.0570.072Potassium channel (Tandem pore domain) blocker

0.069 0.068 CHEMBL1231106

0.0990.0850.19Adenylate cyclase inhibitor

0.098 0.086 CHEMBL3544873

0.136 0.055 CHEMBL244377

0.13 0.06 CHEMBL3544874

0.159 0.039 CHEMBL3544897

0.159 0.039 CHEMBL3544898

0.19 0.027 CHEMBL1231106

CHEMBL1231106
0.0510.0370.089mTOR inhibitor

0.089 0.014 CHEMBL3544873

0.064 0.025 CHEMBL244377

0.069 0.023 CHEMBL3544874

0.086 0.015 CHEMBL3544897

0.086 0.015 CHEMBL3544898

0.063 0.026 CHEMBL1231106

0.067 0.024 CHEMBL457723

0.067 0.024 CHEMBL3544872

CHEMBL3544873
0.0220.0080.028Alpha 2a adrenoreceptor agonist

0.028 0.005 CHEMBL244377

0.025 0.006 CHEMBL1231106

CHEMBL244377
0.0660.0520.067MDM2 inhibitor

0.067 0.047 CHEMBL1231106

CHEMBL1231106
0.0590.0450.059Bcl-xL inhibitor
0.0440.030.051Glutamate (mGluR group III) antagonist

0.051 0.02 CHEMBL1231106

CHEMBL1231106
0.0380.0240.038Delayed rectifier potassium channel blocker

0.036 0.028 CHEMBL244377

0.0340.0210.043Melatonin receptor 1A agonist

0.037 0.017 CHEMBL244377

0.031 0.028 CHEMBL3544874

0.033 0.024 CHEMBL3544897

0.033 0.024 CHEMBL3544898

0.043 0.011 CHEMBL1231106

CHEMBL1231106
0.0560.0430.082Fibroblast growth factor 4 antagonist

0.069 0.028 CHEMBL3544873

0.082 0.017 CHEMBL244377

0.054 0.046 CHEMBL3544874

0.077 0.02 CHEMBL3544897

0.077 0.02 CHEMBL3544898

0.052 0.049 CHEMBL1231106

0.071 0.025 CHEMBL457723

0.071 0.025 CHEMBL3544872

CHEMBL244377
0.0280.0150.031Thymidine kinase (Herpes simplex virus 1) inhibitor

0.028 0.014 CHEMBL244377

0.031 0.01 CHEMBL1231106

CHEMBL1231106
0.0550.0430.065Alpha 1 adrenoreceptor agonist

0.065 0.032 CHEMBL244377

0.061 0.035 CHEMBL457723

0.061 0.035 CHEMBL3544872

CHEMBL244377
0.0580.0450.114CDK2/cyclin E inhibitor

0.062 0.04 CHEMBL3544873

0.096 0.024 CHEMBL244377

0.055 0.048 CHEMBL3544874

0.081 0.03 CHEMBL3544897

0.081 0.03 CHEMBL3544898

0.114 0.019 CHEMBL1231106

0.067 0.037 CHEMBL457723

0.067 0.037 CHEMBL3544872

CHEMBL1231106
0.020.0080.032Adenosine A2a receptor agonist

0.032 0.005 CHEMBL3544873

0.027 0.006 CHEMBL244377

0.025 0.006 CHEMBL3544874

0.032 0.005 CHEMBL3544897

0.032 0.005 CHEMBL3544898

0.028 0.006 CHEMBL1231106

0.027 0.006 CHEMBL457723

0.027 0.006 CHEMBL3544872

CHEMBL3544898
0.0180.0050.018Antibiotic Tetracycline-like

0.015 0.01 CHEMBL3544874

0.015 0.01 CHEMBL457723

0.015 0.01 CHEMBL3544872

0.0330.0210.033Bradykinin B2 receptor antagonist
0.0270.0140.034Complement factor 1s inhibitor

0.026 0.017 CHEMBL244377

0.034 0.005 CHEMBL1231106

CHEMBL1231106
0.0540.0410.06Dihydroorotate oxidase inhibitor

0.06 0.029 CHEMBL244377

0.06 0.029 CHEMBL1231106

CHEMBL1231106
0.020.0080.027Carbonic anhydrase VIII inhibitor

0.027 0.005 CHEMBL244377

0.018 0.01 CHEMBL3544897

0.018 0.01 CHEMBL3544898

0.027 0.005 CHEMBL1231106

0.016 0.013 CHEMBL457723

0.016 0.013 CHEMBL3544872

CHEMBL1231106
0.020.0080.027Carbonic anhydrase X inhibitor

0.027 0.005 CHEMBL244377

0.018 0.01 CHEMBL3544897

0.018 0.01 CHEMBL3544898

0.027 0.005 CHEMBL1231106

0.016 0.013 CHEMBL457723

0.016 0.013 CHEMBL3544872

CHEMBL1231106
0.1110.0990.111Calcium channel blocker
0.0240.0130.068Glutamate (mGluR1a) agonist

0.035 0.007 CHEMBL244377

0.025 0.013 CHEMBL3544897

0.025 0.013 CHEMBL3544898

0.068 0.004 CHEMBL1231106

CHEMBL1231106
0.0690.0570.069Vanilloid antagonist
0.0210.010.114Histamine H4 receptor agonist

0.086 0.003 CHEMBL3544873

0.065 0.004 CHEMBL244377

0.055 0.004 CHEMBL3544874

0.114 0.003 CHEMBL3544897

0.114 0.003 CHEMBL3544898

0.063 0.004 CHEMBL1231106

0.042 0.005 CHEMBL457723

0.042 0.005 CHEMBL3544872

CHEMBL3544898
0.0680.0570.099Catalase inhibitor

0.069 0.055 CHEMBL244377

0.099 0.039 CHEMBL1231106

CHEMBL1231106
0.0540.0430.0545 Hydroxytryptamine 7 agonist
0.0260.0160.031Acid ceramidase inhibitor

0.027 0.014 CHEMBL244377

0.024 0.022 CHEMBL3544874

0.025 0.021 CHEMBL3544897

0.025 0.021 CHEMBL3544898

0.031 0.008 CHEMBL1231106

CHEMBL1231106
0.0220.0110.023Thymidine kinase (Herpes simplex virus 2) inhibitor

0.023 0.009 CHEMBL244377

0.022 0.01 CHEMBL1231106

CHEMBL244377
0.0190.0090.027Adenosine A2 receptor agonist

0.027 0.006 CHEMBL3544873

0.022 0.007 CHEMBL244377

0.022 0.007 CHEMBL3544874

0.026 0.006 CHEMBL3544897

0.026 0.006 CHEMBL3544898

0.023 0.007 CHEMBL1231106

0.023 0.007 CHEMBL457723

0.023 0.007 CHEMBL3544872

CHEMBL3544873
0.020.010.043Cyclin T1 inhibitor

0.029 0.005 CHEMBL3544873

0.029 0.005 CHEMBL244377

0.03 0.005 CHEMBL3544874

0.039 0.004 CHEMBL3544897

0.039 0.004 CHEMBL3544898

0.043 0.003 CHEMBL1231106

0.019 0.011 CHEMBL457723

0.019 0.011 CHEMBL3544872

CHEMBL1231106
0.0390.0290.081Protein kinase (CK1) epsilon inhibitor

0.054 0.011 CHEMBL3544873

0.066 0.007 CHEMBL244377

0.044 0.018 CHEMBL3544874

0.081 0.005 CHEMBL3544897

0.081 0.005 CHEMBL3544898

0.063 0.008 CHEMBL1231106

0.046 0.017 CHEMBL457723

0.046 0.017 CHEMBL3544872

CHEMBL3544898
0.0280.0180.028Myristoyl transferase inhibitor
0.0380.0290.038GABA uptake inhibitor

0.037 0.031 CHEMBL244377

0.036 0.032 CHEMBL1231106

0.0190.010.023Methylmalonyl-CoA mutase inhibitor

0.018 0.014 CHEMBL244377

0.018 0.013 CHEMBL3544874

0.023 0.005 CHEMBL1231106

CHEMBL1231106
0.1010.0910.583Protein kinase (CK1) delta inhibitor

0.291 0.013 CHEMBL3544873

0.457 0.005 CHEMBL244377

0.22 0.023 CHEMBL3544874

0.496 0.005 CHEMBL3544897

0.496 0.005 CHEMBL3544898

0.583 0.004 CHEMBL1231106

0.2 0.029 CHEMBL457723

0.2 0.029 CHEMBL3544872

CHEMBL1231106
0.0840.0750.145Polo-like kinase-1 inhibitor

0.084 0.075 CHEMBL3544873

0.145 0.018 CHEMBL244377

0.122 0.029 CHEMBL3544897

0.122 0.029 CHEMBL3544898

0.097 0.05 CHEMBL1231106

0.099 0.047 CHEMBL457723

0.099 0.047 CHEMBL3544872

CHEMBL244377
0.0310.0220.031LIM domain kinase 2 inhibitor
0.0150.0070.0151-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor

0.013 0.009 CHEMBL244377

0.012 0.011 CHEMBL1231106

0.0640.0550.296CDK1/cyclin B1 inhibitor

0.194 0.009 CHEMBL3544873

0.296 0.004 CHEMBL244377

0.088 0.034 CHEMBL3544874

0.269 0.005 CHEMBL3544897

0.269 0.005 CHEMBL3544898

0.197 0.009 CHEMBL1231106

0.196 0.009 CHEMBL457723

0.196 0.009 CHEMBL3544872

CHEMBL244377
0.0170.0090.024Purinergic P2Y1 agonist

0.015 0.011 CHEMBL3544873

0.017 0.009 CHEMBL244377

0.018 0.008 CHEMBL3544874

0.019 0.008 CHEMBL3544897

0.019 0.008 CHEMBL3544898

0.024 0.005 CHEMBL1231106

0.014 0.013 CHEMBL457723

0.014 0.013 CHEMBL3544872

CHEMBL1231106
0.110.1030.39Growth factor antagonist

0.142 0.074 CHEMBL3544873

0.39 0.018 CHEMBL244377

0.243 0.036 CHEMBL3544897

0.243 0.036 CHEMBL3544898

0.218 0.042 CHEMBL1231106

0.173 0.056 CHEMBL457723

0.173 0.056 CHEMBL3544872

CHEMBL244377
0.0540.0470.075 Hydroxytryptamine 5 antagonist

0.07 0.026 CHEMBL244377

0.061 0.035 CHEMBL3544897

0.061 0.035 CHEMBL3544898

0.055 0.045 CHEMBL1231106

0.054 0.047 CHEMBL457723

0.054 0.047 CHEMBL3544872

CHEMBL244377
0.030.0230.03Cholesterol ester transfer protein antagonist
0.0450.0380.045Cholesterol esterase inhibitor
0.050.0430.058Nicotinic alpha3beta2 receptor antagonist

0.058 0.029 CHEMBL244377

CHEMBL244377
0.1360.1290.2263C-like protease (Human coronavirus) inhibitor

0.226 0.038 CHEMBL1231106

CHEMBL1231106
0.0340.0280.034Ceramide glucosyltransferase inhibitor
0.0550.0480.135Cyclin A inhibitor

0.117 0.018 CHEMBL3544873

0.098 0.024 CHEMBL244377

0.083 0.03 CHEMBL3544874

0.135 0.015 CHEMBL3544897

0.135 0.015 CHEMBL3544898

0.091 0.026 CHEMBL1231106

0.085 0.029 CHEMBL457723

0.085 0.029 CHEMBL3544872

CHEMBL3544898
0.0560.050.061Potassium channel intermediate-conductance Ca-activated blocker

0.061 0.04 CHEMBL244377

0.057 0.049 CHEMBL1231106

CHEMBL244377
0.0810.0750.115Pim-3 kinase inhibitor

0.084 0.069 CHEMBL3544873

0.098 0.048 CHEMBL3544874

0.093 0.053 CHEMBL3544897

0.093 0.053 CHEMBL3544898

0.115 0.034 CHEMBL1231106

CHEMBL1231106
0.0190.0130.021Antibiotic Anthracycline-like

0.018 0.015 CHEMBL244377

0.021 0.009 CHEMBL1231106

CHEMBL1231106
0.0810.0750.1Phosphodiesterase I inhibitor

0.1 0.045 CHEMBL1231106

CHEMBL1231106
0.0430.0370.103Antimetabolite

0.042 0.038 CHEMBL3544873

0.069 0.022 CHEMBL3544874

0.056 0.028 CHEMBL3544897

0.056 0.028 CHEMBL3544898

0.103 0.016 CHEMBL1231106

CHEMBL1231106
0.010.0050.01Corticotropin releasing factor antagonist
0.0550.050.0555 Hydroxytryptamine 7 antagonist
0.0830.0780.126Protein kinase C zeta inhibitor

0.088 0.068 CHEMBL3544873

0.098 0.053 CHEMBL244377

0.1 0.051 CHEMBL3544874

0.117 0.035 CHEMBL3544897

0.117 0.035 CHEMBL3544898

0.126 0.029 CHEMBL1231106

CHEMBL1231106
0.0250.0210.037Lysine carboxypeptidase inhibitor

0.026 0.02 CHEMBL244377

0.037 0.012 CHEMBL1231106

CHEMBL1231106
0.0170.0120.021Telomerase stimulant

0.021 0.007 CHEMBL1231106

CHEMBL1231106
0.0450.040.045Benzodiazepine antagonist
0.0590.0540.07Protease 3C (Human rhinovirus) inhibitor

0.07 0.036 CHEMBL1231106

CHEMBL1231106
0.0640.0590.064Phosphodiesterase V inhibitor
0.0250.0210.04Thymidine phosphorylase inhibitor

0.025 0.021 CHEMBL244377

0.026 0.019 CHEMBL3544874

0.025 0.02 CHEMBL3544897

0.025 0.02 CHEMBL3544898

0.04 0.006 CHEMBL1231106

CHEMBL1231106
0.2020.1980.463Toll-Like receptor 7 agonist

0.463 0.04 CHEMBL3544873

0.203 0.197 CHEMBL244377

0.396 0.061 CHEMBL3544874

0.395 0.062 CHEMBL3544897

0.395 0.062 CHEMBL3544898

0.306 0.106 CHEMBL1231106

0.344 0.085 CHEMBL457723

0.344 0.085 CHEMBL3544872

CHEMBL3544873
0.0130.0090.014Cyclin D2 inhibitor

0.014 0.007 CHEMBL244377

0.014 0.008 CHEMBL1231106

CHEMBL1231106
0.0380.0340.038Liver X receptor alpha agonist
0.0470.0430.081Potassium channel (Inward rectifier) activator

0.081 0.008 CHEMBL244377

0.054 0.027 CHEMBL3544897

0.054 0.027 CHEMBL3544898

0.058 0.023 CHEMBL1231106

0.052 0.033 CHEMBL457723

0.052 0.033 CHEMBL3544872

CHEMBL244377
0.0160.0120.017Nicotinic alpha4 receptor agonist

0.017 0.011 CHEMBL1231106

CHEMBL1231106
0.0270.0240.0285 Hydroxytryptamine 6 agonist

0.028 0.021 CHEMBL244377

CHEMBL244377
0.0190.0160.024Imidazoline I1 receptor antagonist

0.023 0.012 CHEMBL244377

0.024 0.011 CHEMBL1231106

CHEMBL1231106
0.0660.0630.066Acetylcholine M4 receptor antagonist
0.0450.0420.078Potassium channel (ATP-sensitive) activator

0.078 0.007 CHEMBL244377

0.052 0.026 CHEMBL3544897

0.052 0.026 CHEMBL3544898

0.055 0.022 CHEMBL1231106

0.049 0.031 CHEMBL457723

0.049 0.031 CHEMBL3544872

CHEMBL244377
0.0360.0340.036Histone deacetylase 9 inhibitor
0.0250.0230.036Uridine phosphorylase inhibitor

0.036 0.014 CHEMBL1231106

CHEMBL1231106
0.0270.0250.029MAP3K8 inhibitor

0.029 0.02 CHEMBL244377

0.029 0.019 CHEMBL1231106

CHEMBL1231106
0.020.0180.027Neuraminidase (Influenza B) inhibitor

0.022 0.013 CHEMBL244377

0.021 0.015 CHEMBL3544897

0.021 0.015 CHEMBL3544898

0.027 0.005 CHEMBL1231106

CHEMBL1231106
0.0190.0180.022Factor XIII inhibitor

0.022 0.011 CHEMBL244377

0.021 0.013 CHEMBL1231106

CHEMBL244377
0.070.0690.217Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.099 0.036 CHEMBL244377

0.085 0.046 CHEMBL3544874

0.111 0.03 CHEMBL3544897

0.111 0.03 CHEMBL3544898

0.217 0.005 CHEMBL1231106

CHEMBL1231106
0.0460.0450.046Protein 50S ribosomal subunit inhibitor
0.0650.0640.065ErbB-4 antagonist
0.0550.0540.063Ryanodine receptor antagonist

0.063 0.03 CHEMBL1231106

CHEMBL1231106
0.0230.0220.025Lysophosphatidic acid receptor 1 agonist

0.024 0.02 CHEMBL244377

0.025 0.018 CHEMBL1231106

CHEMBL1231106
0.0350.0350.043Toll-Like receptor 2 agonist

0.043 0.027 CHEMBL244377

0.037 0.033 CHEMBL1231106

CHEMBL244377
0.0310.030.0311-Alkyl-2-acetylglycerophosphocholine esterase inhibitor
0.0440.0440.051NMDA 2A receptor antagonist

0.051 0.037 CHEMBL244377

CHEMBL244377
0.030.030.047Glutamate (mGluR3) agonist

0.031 0.024 CHEMBL244377

0.032 0.024 CHEMBL3544874

0.033 0.02 CHEMBL3544897

0.033 0.02 CHEMBL3544898

0.047 0.006 CHEMBL1231106

CHEMBL1231106
0.0120.0120.013Lysophosphatidic acid receptor 3 agonist

0.013 0.01 CHEMBL1231106

CHEMBL1231106
0.1330.1330.144Pyruvate kinase inhibitor

0.144 0.12 CHEMBL1231106

CHEMBL1231106
0.0150.0160.022CDK2/cyclin A3 inhibitor

0.018 0.008 CHEMBL3544873

0.02 0.005 CHEMBL244377

0.016 0.011 CHEMBL3544874

0.022 0.004 CHEMBL3544897

0.022 0.004 CHEMBL3544898

0.02 0.005 CHEMBL1231106

0.016 0.011 CHEMBL457723

0.016 0.011 CHEMBL3544872

CHEMBL3544898
0.1180.1210.175Hexokinase inhibitor

0.122 0.115 CHEMBL244377

0.175 0.053 CHEMBL1231106

CHEMBL1231106
0.0240.0270.028LFA antagonist

0.026 0.022 CHEMBL244377

0.028 0.019 CHEMBL1231106

CHEMBL1231106
0.0530.0560.068NMDA 2C receptor antagonist

0.067 0.036 CHEMBL244377

0.068 0.035 CHEMBL1231106

CHEMBL1231106
0.0210.0240.047Purinergic P2X agonist

0.023 0.022 CHEMBL3544874

0.047 0.01 CHEMBL1231106

CHEMBL1231106
0.0090.0120.011Imidazoline I2 receptor antagonist

0.01 0.009 CHEMBL244377

0.011 0.008 CHEMBL1231106

CHEMBL1231106
0.0120.0160.016NMDA receptor phencyclidine site antagonist

0.016 0.01 CHEMBL244377

CHEMBL244377
0.0220.0250.033Glutamate (mGluR1) agonist

0.025 0.016 CHEMBL244377

0.033 0.008 CHEMBL1231106

CHEMBL1231106
0.0140.0180.019Adenosine A3 receptor agonist

0.018 0.01 CHEMBL3544873

0.019 0.009 CHEMBL244377

0.019 0.01 CHEMBL3544897

0.019 0.01 CHEMBL3544898

0.018 0.01 CHEMBL457723

0.018 0.01 CHEMBL3544872

CHEMBL3544898
0.0390.0420.05Glutamate (mGluR4) antagonist

0.05 0.02 CHEMBL1231106

CHEMBL1231106
0.0620.0660.108Epoxide hydrolase inhibitor

0.108 0.021 CHEMBL244377

0.067 0.058 CHEMBL3544897

0.067 0.058 CHEMBL3544898

0.098 0.026 CHEMBL457723

0.098 0.026 CHEMBL3544872

CHEMBL244377
0.0060.0090.015DNA topoisomerase III inhibitor

0.007 0.005 CHEMBL244377

0.007 0.006 CHEMBL3544874

0.008 0.004 CHEMBL3544897

0.008 0.004 CHEMBL3544898

0.015 0.003 CHEMBL1231106

CHEMBL1231106
0.0080.0120.01Purinergic P2Y2 agonist

0.01 0.009 CHEMBL1231106

CHEMBL1231106
0.0430.0480.052Lysophosphatidic acid 3 receptor antagonist

0.047 0.041 CHEMBL244377

0.052 0.033 CHEMBL1231106

CHEMBL1231106
0.060.0650.253MAP kinase 14 inhibitor

0.143 0.02 CHEMBL3544873

0.253 0.008 CHEMBL244377

0.138 0.022 CHEMBL3544897

0.138 0.022 CHEMBL3544898

0.232 0.009 CHEMBL457723

0.232 0.009 CHEMBL3544872

CHEMBL244377
0.050.0560.073Botulinum neurotoxin type A inhibitor

0.064 0.032 CHEMBL244377

0.064 0.032 CHEMBL3544897

0.064 0.032 CHEMBL3544898

0.073 0.022 CHEMBL1231106

CHEMBL1231106
0.1440.150.192Histone acetyltransferase inhibitor

0.174 0.108 CHEMBL244377

0.192 0.082 CHEMBL1231106

CHEMBL1231106
0.0090.0150.019Purine nucleoside phosphorylase inhibitor

0.012 0.007 CHEMBL3544874

0.013 0.007 CHEMBL3544897

0.013 0.007 CHEMBL3544898

0.019 0.003 CHEMBL1231106

CHEMBL1231106
0.0470.0530.065 Hydroxytryptamine 6 antagonist

0.06 0.036 CHEMBL244377

0.057 0.039 CHEMBL3544897

0.057 0.039 CHEMBL3544898

0.052 0.046 CHEMBL1231106

CHEMBL244377
0.0260.0330.034Calcitonin receptor agonist

0.034 0.023 CHEMBL1231106

CHEMBL1231106
0.0380.0450.07Fructose-1,6-bisphosphatase inhibitor

0.043 0.034 CHEMBL244377

0.044 0.033 CHEMBL3544897

0.044 0.033 CHEMBL3544898

0.07 0.012 CHEMBL1231106

CHEMBL1231106
0.0190.0270.032Isoleucine-tRNA ligase inhibitor

0.022 0.017 CHEMBL3544874

0.032 0.005 CHEMBL1231106

CHEMBL1231106
0.0080.0170.018Glutamate (mGluR6) agonist

0.018 0.005 CHEMBL1231106

CHEMBL1231106
0.0090.0180.012Carbonic anhydrase XI inhibitor

0.012 0.01 CHEMBL244377

0.012 0.009 CHEMBL1231106

CHEMBL1231106
0.0180.0270.021Glutaminyl-peptide cyclotransferase inhibitor

0.021 0.017 CHEMBL244377

0.021 0.017 CHEMBL1231106

CHEMBL1231106
0.0340.0430.0375 Hydroxytryptamine 2B agonist

0.037 0.031 CHEMBL1231106

CHEMBL1231106
0.0460.0550.07Lysine-specific demethylase 1A inhibitor

0.059 0.029 CHEMBL244377

0.049 0.047 CHEMBL3544874

0.061 0.026 CHEMBL3544897

0.061 0.026 CHEMBL3544898

0.07 0.018 CHEMBL1231106

CHEMBL1231106
0.0040.0130.006CC chemokine 6 receptor agonist

0.006 0.005 CHEMBL1231106

CHEMBL1231106
0.1720.1820.242Transcription factor STAT inhibitor

0.242 0.093 CHEMBL244377

0.192 0.15 CHEMBL1231106

CHEMBL244377
0.0550.0650.064Phosphodiesterase 1C inhibitor

0.064 0.039 CHEMBL1231106

CHEMBL1231106
0.0530.0640.072Sphingosine 1-phosphate receptor 4 agonist

0.072 0.042 CHEMBL1231106

CHEMBL1231106
0.0150.0270.021Alpha 2b adrenoreceptor agonist

0.021 0.009 CHEMBL1231106

CHEMBL1231106
0.0250.0370.031Methionyl aminopeptidase 1 inhibitor

0.031 0.024 CHEMBL244377

0.031 0.023 CHEMBL1231106

CHEMBL1231106
0.0540.0660.0835 Hydroxytryptamine 3A antagonist

0.083 0.029 CHEMBL244377

0.069 0.043 CHEMBL3544897

0.069 0.043 CHEMBL3544898

0.064 0.049 CHEMBL1231106

CHEMBL244377
0.0290.0420.057Glutamate (mGluR3) antagonist

0.057 0.009 CHEMBL1231106

CHEMBL1231106
0.050.0630.123Heat shock protein 90 beta antagonist

0.075 0.024 CHEMBL3544873

0.073 0.025 CHEMBL244377

0.077 0.023 CHEMBL3544874

0.111 0.008 CHEMBL3544897

0.111 0.008 CHEMBL3544898

0.123 0.006 CHEMBL1231106

CHEMBL1231106
0.1360.150.277Potassium channel blocker

0.277 0.054 CHEMBL244377

0.166 0.119 CHEMBL457723

0.166 0.119 CHEMBL3544872

CHEMBL244377
0.0410.0550.062Bombesin 2 receptor antagonist

0.062 0.023 CHEMBL1231106

CHEMBL1231106
0.0130.0290.02Complement factor D inhibitor

0.02 0.009 CHEMBL1231106

CHEMBL1231106
0.0530.0690.065Syk tyrosine kinase inhibitor

0.065 0.054 CHEMBL244377

CHEMBL244377
0.0490.0650.069Sphingosine kinase inhibitor

0.069 0.026 CHEMBL1231106

CHEMBL1231106
0.020.0370.025Nicotinic acid receptor 2 antagonist

0.025 0.021 CHEMBL1231106

CHEMBL1231106
0.0660.0830.108Bcr-Abl kinase inhibitor

0.108 0.034 CHEMBL244377

0.086 0.057 CHEMBL3544897

0.086 0.057 CHEMBL3544898

0.088 0.054 CHEMBL457723

0.088 0.054 CHEMBL3544872

CHEMBL244377
0.0460.0640.085NMDA receptor glycine site agonist

0.085 0.025 CHEMBL244377

0.063 0.043 CHEMBL3544897

0.063 0.043 CHEMBL3544898

0.074 0.033 CHEMBL1231106

CHEMBL244377
0.0380.0550.043Dipeptidyl peptidase IV inhibitor

0.043 0.032 CHEMBL1231106

CHEMBL1231106
0.0380.0560.059Aldosterone antagonist

0.059 0.02 CHEMBL1231106

CHEMBL1231106
0.0210.0390.032Thrombin receptor antagonist

0.032 0.016 CHEMBL1231106

CHEMBL1231106
0.1190.1380.135Melanin inhibitor

0.135 0.106 CHEMBL1231106

CHEMBL1231106
0.0260.0450.034Carboxypeptidase B inhibitor

0.034 0.021 CHEMBL1231106

CHEMBL1231106
0.0590.0780.074Glutamate receptor agonist

0.074 0.059 CHEMBL1231106

CHEMBL1231106
0.0560.0760.075Cathepsin G inhibitor

0.075 0.048 CHEMBL1231106

CHEMBL1231106
0.030.0510.041Potassium channel Kv1.1 blocker

0.041 0.021 CHEMBL244377

0.037 0.029 CHEMBL1231106

CHEMBL244377
0.0450.0650.451Phosphatidylinositol kinase inhibitor

0.235 0.007 CHEMBL3544873

0.108 0.019 CHEMBL244377

0.195 0.009 CHEMBL3544874

0.312 0.005 CHEMBL3544897

0.312 0.005 CHEMBL3544898

0.451 0.004 CHEMBL1231106

0.093 0.023 CHEMBL457723

0.093 0.023 CHEMBL3544872

CHEMBL1231106
0.0490.070.078NMDA receptor agonist

0.078 0.03 CHEMBL244377

0.061 0.046 CHEMBL3544897

0.061 0.046 CHEMBL3544898

0.072 0.034 CHEMBL1231106

CHEMBL244377
0.0110.0320.016Nicotinic acid receptor 1 antagonist

0.016 0.015 CHEMBL1231106

CHEMBL1231106
0.0310.0520.036AMPA 4 receptor antagonist

0.036 0.035 CHEMBL1231106

CHEMBL1231106
0.0450.0670.073MAP kinase kinase 9 inhibitor

0.073 0.019 CHEMBL244377

0.053 0.045 CHEMBL3544897

0.053 0.045 CHEMBL3544898

0.055 0.039 CHEMBL457723

0.055 0.039 CHEMBL3544872

CHEMBL244377
0.0310.0530.041NMDA receptor subunit 3B antagonist

0.041 0.034 CHEMBL244377

CHEMBL244377
0.0410.0640.0493(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.049 0.045 CHEMBL1231106

CHEMBL1231106
0.0320.0560.045Sphingosine kinase 1 inhibitor

0.045 0.023 CHEMBL1231106

CHEMBL1231106
0.1860.210.267Ca2+/calmodulin-dependent kinase IV inhibitor

0.204 0.154 CHEMBL3544873

0.267 0.047 CHEMBL244377

0.22 0.116 CHEMBL3544897

0.22 0.116 CHEMBL3544898

0.237 0.085 CHEMBL457723

0.237 0.085 CHEMBL3544872

CHEMBL244377
0.0290.0530.036MAP3K5 inhibitor

0.036 0.033 CHEMBL244377

0.036 0.032 CHEMBL1231106

CHEMBL1231106
0.0240.0480.0385 Hydroxytryptamine 3B antagonist

0.038 0.022 CHEMBL244377

CHEMBL244377
0.0260.0510.04ATR kinase inhibitor

0.031 0.028 CHEMBL3544873

0.035 0.019 CHEMBL244377

0.04 0.012 CHEMBL3544897

0.04 0.012 CHEMBL3544898

0.038 0.015 CHEMBL1231106

CHEMBL3544898
0.0440.0690.133Phosphodiesterase VII inhibitor

0.091 0.017 CHEMBL3544873

0.133 0.005 CHEMBL244377

0.113 0.008 CHEMBL3544897

0.113 0.008 CHEMBL3544898

0.075 0.03 CHEMBL1231106

0.101 0.012 CHEMBL457723

0.101 0.012 CHEMBL3544872

CHEMBL244377
0.0160.0410.028Fructose-1,6-bisphosphatase 1 inhibitor

0.028 0.009 CHEMBL1231106

CHEMBL1231106
0.0930.1180.132Toll-Like receptor 2 antagonist

0.132 0.066 CHEMBL1231106

CHEMBL1231106
0.060.0870.072Acetylcholine nicotinic agonist

0.072 0.069 CHEMBL244377

CHEMBL244377
0.0610.0880.078Keratolytic

0.078 0.051 CHEMBL1231106

CHEMBL1231106
0.0330.060.31Phosphatidylinositol 3-kinase alpha inhibitor

0.227 0.006 CHEMBL3544873

0.121 0.013 CHEMBL244377

0.168 0.009 CHEMBL3544874

0.285 0.005 CHEMBL3544897

0.285 0.005 CHEMBL3544898

0.31 0.005 CHEMBL1231106

0.101 0.016 CHEMBL457723

0.101 0.016 CHEMBL3544872

CHEMBL1231106
0.0870.1150.121Nav1.3 sodium channel blocker

0.121 0.073 CHEMBL1231106

CHEMBL1231106
0.0570.0860.086Leucine-rich repeat kinase 2 inhibitor

0.086 0.052 CHEMBL244377

CHEMBL244377
0.0420.070.05Dipeptidyl peptidase inhibitor

0.05 0.043 CHEMBL1231106

CHEMBL1231106
0.030.060.093Aggrecanase 1 inhibitor

0.093 0.005 CHEMBL244377

0.041 0.024 CHEMBL3544897

0.041 0.024 CHEMBL3544898

0.045 0.018 CHEMBL457723

0.045 0.018 CHEMBL3544872

CHEMBL244377
0.0330.0640.083Carbonic anhydrase XIV inhibitor

0.083 0.016 CHEMBL244377

0.063 0.023 CHEMBL3544897

0.063 0.023 CHEMBL3544898

0.058 0.026 CHEMBL1231106

0.044 0.041 CHEMBL457723

0.044 0.041 CHEMBL3544872

CHEMBL244377
0.0690.10.128Potassium channel activator

0.128 0.028 CHEMBL244377

0.081 0.074 CHEMBL3544897

0.081 0.074 CHEMBL3544898

CHEMBL244377
0.0270.0580.083CDK5/p25 inhibitor

0.039 0.031 CHEMBL244377

0.036 0.035 CHEMBL3544874

0.054 0.018 CHEMBL3544897

0.054 0.018 CHEMBL3544898

0.083 0.009 CHEMBL1231106

CHEMBL1231106
0.0250.0570.085Glutamate (mGluR4) agonist

0.033 0.025 CHEMBL3544874

0.039 0.016 CHEMBL3544897

0.039 0.016 CHEMBL3544898

0.085 0.005 CHEMBL1231106

CHEMBL1231106
0.030.0620.142Glutamate (mGluR group III) agonist

0.04 0.034 CHEMBL244377

0.049 0.024 CHEMBL3544874

0.08 0.013 CHEMBL3544897

0.08 0.013 CHEMBL3544898

0.142 0.005 CHEMBL1231106

CHEMBL1231106
0.030.0630.047Ribonucleoside-diphosphate reductase inhibitor

0.047 0.043 CHEMBL1231106

CHEMBL1231106
0.030.0640.049Ribonucleotide reductase inhibitor

0.049 0.043 CHEMBL1231106

CHEMBL1231106
0.0180.0520.0275 Hydroxytryptamine 4 agonist

0.027 0.01 CHEMBL244377

0.025 0.014 CHEMBL3544897

0.025 0.014 CHEMBL3544898

CHEMBL244377
0.0390.0750.096CXC chemokine 4 receptor antagonist

0.096 0.026 CHEMBL244377

0.056 0.045 CHEMBL3544897

0.056 0.045 CHEMBL3544898

0.053 0.048 CHEMBL457723

0.053 0.048 CHEMBL3544872

CHEMBL244377
0.0250.0640.043Antibiotic Aminoglycoside-like

0.039 0.022 CHEMBL3544873

0.043 0.018 CHEMBL244377

0.043 0.018 CHEMBL3544897

0.043 0.018 CHEMBL3544898

0.038 0.023 CHEMBL457723

0.038 0.023 CHEMBL3544872

CHEMBL3544898
0.0220.0610.052Carbonic anhydrase IV inhibitor

0.052 0.024 CHEMBL244377

CHEMBL244377
0.1070.1480.155Hemostatic

0.143 0.077 CHEMBL244377

0.119 0.117 CHEMBL3544897

0.119 0.117 CHEMBL3544898

0.155 0.062 CHEMBL1231106

CHEMBL1231106
0.0320.0730.096Xanthine dehydrogenase inhibitor

0.063 0.036 CHEMBL3544897

0.063 0.036 CHEMBL3544898

0.096 0.017 CHEMBL1231106

CHEMBL1231106
0.0290.0720.045Plasmepsin II inhibitor

0.045 0.023 CHEMBL1231106

CHEMBL1231106
0.1130.1570.23DNA methyltransferase I inhibitor

0.133 0.126 CHEMBL3544874

0.136 0.121 CHEMBL3544897

0.136 0.121 CHEMBL3544898

0.23 0.055 CHEMBL1231106

CHEMBL1231106
0.0640.1120.084Antihistaminic

0.084 0.072 CHEMBL3544897

0.084 0.072 CHEMBL3544898

0.083 0.074 CHEMBL1231106

CHEMBL3544898
0.0580.1080.188I kappa B kinase inhibitor

0.129 0.022 CHEMBL3544873

0.146 0.017 CHEMBL244377

0.079 0.063 CHEMBL3544874

0.188 0.009 CHEMBL3544897

0.188 0.009 CHEMBL3544898

0.112 0.03 CHEMBL1231106

0.097 0.041 CHEMBL457723

0.097 0.041 CHEMBL3544872

CHEMBL3544898
0.1140.1640.206Antipruritic

0.136 0.112 CHEMBL3544873

0.161 0.083 CHEMBL244377

0.145 0.101 CHEMBL3544874

0.206 0.045 CHEMBL3544897

0.206 0.045 CHEMBL3544898

0.205 0.046 CHEMBL1231106

CHEMBL3544898
0.0770.1270.138Amylase inhibitor

0.138 0.07 CHEMBL1231106

CHEMBL1231106
0.0320.0830.056Toll-Like receptor 8 antagonist

0.056 0.034 CHEMBL1231106

CHEMBL1231106
0.1130.1650.251DNA methylase inhibitor

0.152 0.115 CHEMBL244377

0.145 0.121 CHEMBL3544874

0.195 0.082 CHEMBL3544897

0.195 0.082 CHEMBL3544898

0.251 0.048 CHEMBL1231106

CHEMBL1231106
0.040.0910.079NMDA 2 receptor antagonist

0.079 0.044 CHEMBL244377

CHEMBL244377
0.0320.0840.058Neuropeptide Y5 antagonist

0.048 0.039 CHEMBL244377

0.058 0.031 CHEMBL457723

0.058 0.031 CHEMBL3544872

CHEMBL3544872
0.0210.0750.039Purinergic P2Y antagonist

0.039 0.038 CHEMBL244377

CHEMBL244377
0.0560.1110.082Potassium channel (Ca-activated) activator

0.082 0.072 CHEMBL244377

CHEMBL244377
0.0770.1320.17MAP kinase kinase inhibitor

0.149 0.052 CHEMBL244377

0.17 0.041 CHEMBL3544897

0.17 0.041 CHEMBL3544898

0.162 0.045 CHEMBL1231106

CHEMBL3544898
0.0540.1090.075Histamine antagonist

0.075 0.07 CHEMBL3544897

0.075 0.07 CHEMBL3544898

0.073 0.072 CHEMBL1231106

CHEMBL3544898
0.0440.10.113I kappa B kinase 2 inhibitor

0.071 0.031 CHEMBL3544873

0.093 0.015 CHEMBL244377

0.113 0.009 CHEMBL3544897

0.113 0.009 CHEMBL3544898

0.078 0.024 CHEMBL1231106

0.06 0.047 CHEMBL457723

0.06 0.047 CHEMBL3544872

CHEMBL3544898
0.0150.0740.035Nicotinic acid receptor agonist

0.035 0.026 CHEMBL1231106

CHEMBL1231106
0.1170.1770.792Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.43 0.021 CHEMBL3544873

0.328 0.041 CHEMBL244377

0.417 0.023 CHEMBL3544874

0.564 0.008 CHEMBL3544897

0.564 0.008 CHEMBL3544898

0.792 0.004 CHEMBL1231106

0.213 0.085 CHEMBL457723

0.213 0.085 CHEMBL3544872

CHEMBL1231106
0.0450.1080.102Rho-associated kinase I inhibitor

0.069 0.058 CHEMBL3544873

0.08 0.046 CHEMBL244377

0.102 0.03 CHEMBL3544897

0.102 0.03 CHEMBL3544898

0.094 0.035 CHEMBL1231106

CHEMBL3544898
0.0090.0730.124O6-alkylguanine-DNA alkyltransferase inhibitor

0.026 0.004 CHEMBL3544873

0.032 0.003 CHEMBL3544874

0.033 0.003 CHEMBL3544897

0.033 0.003 CHEMBL3544898

0.124 0.001 CHEMBL1231106

CHEMBL1231106
0.0360.10.22Cyclin B1 inhibitor

0.084 0.019 CHEMBL3544873

0.163 0.005 CHEMBL244377

0.058 0.046 CHEMBL3544874

0.147 0.005 CHEMBL3544897

0.147 0.005 CHEMBL3544898

0.22 0.004 CHEMBL1231106

0.078 0.023 CHEMBL457723

0.078 0.023 CHEMBL3544872

CHEMBL1231106
0.1480.2140.223Transcription factor STAT3 inhibitor

0.223 0.108 CHEMBL244377

0.179 0.166 CHEMBL1231106

CHEMBL244377
0.030.0960.063CDK4/cyclin D inhibitor

0.063 0.035 CHEMBL244377

0.054 0.047 CHEMBL3544897

0.054 0.047 CHEMBL3544898

0.057 0.042 CHEMBL1231106

CHEMBL244377
0.0970.1640.259Heat shock protein 90 antagonist

0.124 0.107 CHEMBL3544873

0.119 0.116 CHEMBL244377

0.162 0.062 CHEMBL3544874

0.197 0.039 CHEMBL3544897

0.197 0.039 CHEMBL3544898

0.259 0.018 CHEMBL1231106

CHEMBL1231106
0.0290.0960.04GABA B receptor antagonist

0.04 0.035 CHEMBL1231106

CHEMBL1231106
0.060.1310.111Granulocyte macrophage colony stimulating factor antagonist

0.101 0.07 CHEMBL244377

0.111 0.06 CHEMBL3544897

0.111 0.06 CHEMBL3544898

0.098 0.074 CHEMBL1231106

CHEMBL3544898
0.0310.1020.052Pim-2 kinase inhibitor

0.052 0.041 CHEMBL1231106

CHEMBL1231106
0.0180.0910.047Carbonic anhydrase VII inhibitor

0.047 0.031 CHEMBL244377

CHEMBL244377
0.0510.1240.082MAO A inhibitor

0.082 0.079 CHEMBL244377

CHEMBL244377
0.0380.1140.067Janus tyrosine kinase 2 inhibitor

0.065 0.06 CHEMBL244377

0.067 0.058 CHEMBL1231106

CHEMBL1231106
0.0270.1030.455Raf kinase C inhibitor

0.175 0.012 CHEMBL3544873

0.455 0.004 CHEMBL244377

0.26 0.006 CHEMBL3544897

0.26 0.006 CHEMBL3544898

0.323 0.005 CHEMBL457723

0.323 0.005 CHEMBL3544872

CHEMBL244377
0.0980.1760.246Heat shock protein 90 alpha antagonist

0.149 0.088 CHEMBL3544874

0.166 0.072 CHEMBL3544897

0.166 0.072 CHEMBL3544898

0.246 0.028 CHEMBL1231106

CHEMBL1231106
0.0270.1070.182Cyclin B2 inhibitor

0.074 0.018 CHEMBL3544873

0.152 0.005 CHEMBL244377

0.135 0.005 CHEMBL3544897

0.135 0.005 CHEMBL3544898

0.182 0.004 CHEMBL1231106

0.07 0.022 CHEMBL457723

0.07 0.022 CHEMBL3544872

CHEMBL1231106
0.0260.1070.225Phosphatidylinositol 3-kinase beta inhibitor

0.087 0.015 CHEMBL3544873

0.097 0.013 CHEMBL3544874

0.114 0.01 CHEMBL3544897

0.114 0.01 CHEMBL3544898

0.225 0.005 CHEMBL1231106

CHEMBL1231106
0.0070.090.026Aggrecanase 2 inhibitor

0.026 0.012 CHEMBL244377

CHEMBL244377
0.1340.2270.364MAP kinase kinase 5 inhibitor

0.259 0.005 CHEMBL3544873

0.364 0.003 CHEMBL244377

0.307 0.004 CHEMBL3544897

0.307 0.004 CHEMBL3544898

0.29 0.004 CHEMBL457723

0.29 0.004 CHEMBL3544872

CHEMBL244377
0.0650.160.612T cell inhibitor

0.443 0.004 CHEMBL3544873

0.612 0.003 CHEMBL244377

0.081 0.063 CHEMBL3544874

0.535 0.003 CHEMBL3544897

0.535 0.003 CHEMBL3544898

0.085 0.049 CHEMBL1231106

0.488 0.004 CHEMBL457723

0.488 0.004 CHEMBL3544872

CHEMBL244377
0.0890.1830.483Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.276 0.039 CHEMBL3544873

0.296 0.032 CHEMBL244377

0.231 0.055 CHEMBL3544874

0.367 0.016 CHEMBL3544897

0.367 0.016 CHEMBL3544898

0.483 0.006 CHEMBL1231106

0.171 0.08 CHEMBL457723

0.171 0.08 CHEMBL3544872

CHEMBL1231106
0.0360.1320.185Cyclin B3 inhibitor

0.121 0.021 CHEMBL244377

0.12 0.021 CHEMBL3544897

0.12 0.021 CHEMBL3544898

0.185 0.008 CHEMBL1231106

CHEMBL1231106
0.0270.1230.129Phosphatidylinositol 3-kinase gamma inhibitor

0.074 0.023 CHEMBL3544873

0.071 0.024 CHEMBL3544874

0.094 0.016 CHEMBL3544897

0.094 0.016 CHEMBL3544898

0.129 0.011 CHEMBL1231106

CHEMBL1231106
0.0510.1490.1Mediator release inhibitor

0.1 0.07 CHEMBL244377

CHEMBL244377
0.0260.1240.115Janus tyrosine kinase 3 inhibitor

0.115 0.028 CHEMBL244377

0.062 0.06 CHEMBL3544897

0.062 0.06 CHEMBL3544898

CHEMBL244377
0.0490.1480.095MAP kinase kinase kinase inhibitor

0.095 0.072 CHEMBL1231106

CHEMBL1231106
0.0560.1560.157Aurora-B kinase inhibitor

0.11 0.072 CHEMBL3544873

0.134 0.055 CHEMBL244377

0.157 0.044 CHEMBL3544897

0.157 0.044 CHEMBL3544898

0.101 0.081 CHEMBL1231106

0.096 0.088 CHEMBL457723

0.096 0.088 CHEMBL3544872

CHEMBL3544898
0.0270.1270.186Cyclin B inhibitor

0.073 0.019 CHEMBL3544873

0.166 0.005 CHEMBL244377

0.146 0.005 CHEMBL3544897

0.146 0.005 CHEMBL3544898

0.186 0.004 CHEMBL1231106

0.069 0.023 CHEMBL457723

0.069 0.023 CHEMBL3544872

CHEMBL1231106
0.0560.1560.21c-Src kinase inhibitor

0.152 0.054 CHEMBL3544873

0.21 0.033 CHEMBL244377

0.201 0.035 CHEMBL3544897

0.201 0.035 CHEMBL3544898

0.165 0.048 CHEMBL1231106

0.146 0.057 CHEMBL457723

0.146 0.057 CHEMBL3544872

CHEMBL244377
0.0580.1620.194Thioredoxin inhibitor

0.097 0.052 CHEMBL3544874

0.093 0.057 CHEMBL3544897

0.093 0.057 CHEMBL3544898

0.194 0.009 CHEMBL1231106

CHEMBL1231106
0.0740.180.449Protein kinase C nu inhibitor

0.2 0.047 CHEMBL3544873

0.302 0.024 CHEMBL244377

0.172 0.059 CHEMBL3544874

0.362 0.014 CHEMBL3544897

0.362 0.014 CHEMBL3544898

0.449 0.006 CHEMBL1231106

0.122 0.09 CHEMBL457723

0.122 0.09 CHEMBL3544872

CHEMBL1231106
0.0290.1360.062Cyclin-dependent kinase 4 inhibitor

0.062 0.049 CHEMBL244377

CHEMBL244377
0.0410.1490.325Cyclin-dependent kinase 1 inhibitor

0.156 0.039 CHEMBL3544873

0.318 0.01 CHEMBL244377

0.293 0.012 CHEMBL3544897

0.293 0.012 CHEMBL3544898

0.325 0.01 CHEMBL1231106

0.139 0.046 CHEMBL457723

0.139 0.046 CHEMBL3544872

CHEMBL1231106
0.10.2090.787Dyrk kinase inhibitor

0.399 0.026 CHEMBL3544873

0.313 0.048 CHEMBL244377

0.39 0.028 CHEMBL3544874

0.552 0.009 CHEMBL3544897

0.552 0.009 CHEMBL3544898

0.787 0.004 CHEMBL1231106

0.193 0.102 CHEMBL457723

0.193 0.102 CHEMBL3544872

CHEMBL1231106
0.060.1710.115TRKA antagonist

0.107 0.08 CHEMBL244377

0.115 0.071 CHEMBL3544897

0.115 0.071 CHEMBL3544898

0.108 0.079 CHEMBL1231106

CHEMBL3544898
0.0490.1670.13Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.13 0.06 CHEMBL244377

0.102 0.084 CHEMBL3544897

0.102 0.084 CHEMBL3544898

0.105 0.082 CHEMBL457723

0.105 0.082 CHEMBL3544872

CHEMBL244377
0.0490.1660.129Abl kinase inhibitor

0.129 0.06 CHEMBL244377

0.102 0.084 CHEMBL3544897

0.102 0.084 CHEMBL3544898

0.105 0.081 CHEMBL457723

0.105 0.081 CHEMBL3544872

CHEMBL244377
0.0210.1390.445Raf kinase B inhibitor

0.158 0.013 CHEMBL3544873

0.445 0.004 CHEMBL244377

0.274 0.006 CHEMBL3544897

0.274 0.006 CHEMBL3544898

0.261 0.006 CHEMBL457723

0.261 0.006 CHEMBL3544872

CHEMBL244377
0.0570.1770.109Thioredoxin reductase inhibitor

0.109 0.022 CHEMBL1231106

CHEMBL1231106
0.0480.170.17Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.098 0.04 CHEMBL3544873

0.17 0.01 CHEMBL244377

0.15 0.014 CHEMBL3544897

0.15 0.014 CHEMBL3544898

0.141 0.017 CHEMBL1231106

0.099 0.039 CHEMBL457723

0.099 0.039 CHEMBL3544872

CHEMBL244377
0.0480.1750.227Glycogen synthase kinase-3 inhibitor

0.134 0.053 CHEMBL244377

0.119 0.062 CHEMBL3544897

0.119 0.062 CHEMBL3544898

0.227 0.026 CHEMBL1231106

CHEMBL1231106
0.0050.1310.02Sodium/hydrogen exchanger inhibitor

0.02 0.008 CHEMBL1231106

CHEMBL1231106
0.0590.1910.119Tyrosine-protein kinase receptor antagonist

0.108 0.099 CHEMBL244377

0.119 0.088 CHEMBL3544897

0.119 0.088 CHEMBL3544898

0.111 0.095 CHEMBL1231106

CHEMBL3544898
0.0380.1720.371I kappa B kinase 1 inhibitor

0.269 0.004 CHEMBL3544873

0.35 0.004 CHEMBL244377

0.098 0.024 CHEMBL3544874

0.371 0.004 CHEMBL3544897

0.371 0.004 CHEMBL3544898

0.234 0.005 CHEMBL1231106

0.228 0.005 CHEMBL457723

0.228 0.005 CHEMBL3544872

CHEMBL3544898
0.0210.1560.153CDK9/cyclin T1 inhibitor

0.062 0.038 CHEMBL3544873

0.134 0.012 CHEMBL244377

0.133 0.012 CHEMBL3544897

0.133 0.012 CHEMBL3544898

0.153 0.01 CHEMBL1231106

0.051 0.05 CHEMBL457723

0.051 0.05 CHEMBL3544872

CHEMBL1231106
0.0250.1650.116Phosphodiesterase 7A inhibitor

0.064 0.016 CHEMBL3544873

0.116 0.004 CHEMBL244377

0.089 0.005 CHEMBL3544897

0.089 0.005 CHEMBL3544898

0.056 0.028 CHEMBL1231106

0.072 0.01 CHEMBL457723

0.072 0.01 CHEMBL3544872

CHEMBL244377
0.0260.1660.508Raf kinase inhibitor

0.179 0.015 CHEMBL3544873

0.508 0.004 CHEMBL244377

0.316 0.006 CHEMBL3544897

0.316 0.006 CHEMBL3544898

0.282 0.007 CHEMBL457723

0.282 0.007 CHEMBL3544872

CHEMBL244377
0.0350.1750.519Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.222 0.015 CHEMBL3544873

0.519 0.005 CHEMBL244377

0.363 0.006 CHEMBL3544897

0.363 0.006 CHEMBL3544898

0.29 0.009 CHEMBL457723

0.29 0.009 CHEMBL3544872

CHEMBL244377
0.0420.1830.288Vascular endothelial growth factor 1 antagonist

0.167 0.035 CHEMBL244377

0.113 0.058 CHEMBL3544897

0.113 0.058 CHEMBL3544898

0.288 0.012 CHEMBL1231106

CHEMBL1231106
0.0490.190.141Glycogen synthase kinase-3 alpha inhibitor

0.103 0.101 CHEMBL244377

0.106 0.097 CHEMBL3544897

0.106 0.097 CHEMBL3544898

0.141 0.072 CHEMBL1231106

CHEMBL1231106
0.0580.210.281Toll-Like receptor 3 antagonist

0.099 0.052 CHEMBL3544873

0.152 0.014 CHEMBL3544874

0.147 0.015 CHEMBL3544897

0.147 0.015 CHEMBL3544898

0.281 0.004 CHEMBL1231106

CHEMBL1231106
0.030.1910.122MAP kinase 10 inhibitor

0.122 0.023 CHEMBL244377

0.072 0.062 CHEMBL3544897

0.072 0.062 CHEMBL3544898

0.087 0.044 CHEMBL457723

0.087 0.044 CHEMBL3544872

CHEMBL244377
0.0850.2510.535Death-associated protein kinase 3 inhibitor

0.25 0.053 CHEMBL3544873

0.365 0.023 CHEMBL244377

0.208 0.07 CHEMBL3544874

0.426 0.013 CHEMBL3544897

0.426 0.013 CHEMBL3544898

0.535 0.005 CHEMBL1231106

0.16 0.108 CHEMBL457723

0.16 0.108 CHEMBL3544872

CHEMBL1231106
0.030.1960.108Polo-like kinase-2 inhibitor

0.108 0.019 CHEMBL244377

CHEMBL244377
0.0290.1980.382Aurora-A kinase inhibitor

0.129 0.05 CHEMBL3544873

0.382 0.008 CHEMBL244377

0.243 0.019 CHEMBL3544897

0.243 0.019 CHEMBL3544898

0.093 0.072 CHEMBL1231106

0.174 0.032 CHEMBL457723

0.174 0.032 CHEMBL3544872

CHEMBL244377
0.0060.1780.017Adenosine A2b receptor agonist

0.014 0.011 CHEMBL244377

0.016 0.009 CHEMBL3544897

0.016 0.009 CHEMBL3544898

0.017 0.007 CHEMBL1231106

CHEMBL1231106
0.040.2130.121MAP kinase 8 inhibitor

0.087 0.078 CHEMBL3544873

0.121 0.043 CHEMBL244377

0.109 0.052 CHEMBL3544897

0.109 0.052 CHEMBL3544898

0.091 0.071 CHEMBL1231106

0.088 0.075 CHEMBL457723

0.088 0.075 CHEMBL3544872

CHEMBL244377
0.0140.1910.38Phosphatidylinositol 3-kinase delta inhibitor

0.109 0.018 CHEMBL3544873

0.137 0.013 CHEMBL3544874

0.153 0.01 CHEMBL3544897

0.153 0.01 CHEMBL3544898

0.38 0.004 CHEMBL1231106

CHEMBL1231106
0.030.2070.442Tyrosine-protein kinase receptor FLT3 inhibitor

0.142 0.056 CHEMBL3544873

0.442 0.008 CHEMBL244377

0.273 0.023 CHEMBL3544897

0.273 0.023 CHEMBL3544898

0.206 0.035 CHEMBL457723

0.206 0.035 CHEMBL3544872

CHEMBL244377
0.0380.2150.077Phosphodiesterase VIII inhibitor

0.077 0.039 CHEMBL1231106

CHEMBL1231106
0.0240.2010.115CDK2/cyclin E2 inhibitor

0.115 0.024 CHEMBL244377

0.102 0.027 CHEMBL3544897

0.102 0.027 CHEMBL3544898

0.111 0.025 CHEMBL1231106

CHEMBL244377
0.0540.2350.351Ca2+/calmodulin-dependent kinase II delta inhibitor

0.163 0.059 CHEMBL244377

0.22 0.04 CHEMBL3544897

0.22 0.04 CHEMBL3544898

0.351 0.01 CHEMBL1231106

CHEMBL1231106
0.0610.2460.697Protein kinase (CK1) gamma 1 inhibitor

0.31 0.018 CHEMBL3544873

0.273 0.024 CHEMBL244377

0.325 0.016 CHEMBL3544874

0.497 0.005 CHEMBL3544897

0.497 0.005 CHEMBL3544898

0.697 0.003 CHEMBL1231106

CHEMBL1231106
0.030.2180.078ALK inhibitor

0.078 0.062 CHEMBL244377

CHEMBL244377
0.0020.1910.122Phosphoribosylglycinamide formyltransferase inhibitor

0.01 0.004 CHEMBL3544874

0.009 0.004 CHEMBL3544897

0.009 0.004 CHEMBL3544898

0.122 0.001 CHEMBL1231106

CHEMBL1231106
0.0040.1960.022Prokineticin receptor 1 antagonist

0.022 0.005 CHEMBL1231106

CHEMBL1231106
0.0110.2050.028Granulocyte colony stimulating factor receptor agonist

0.028 0.004 CHEMBL1231106

CHEMBL1231106
0.0920.2860.252MAP kinase kinase 4 inhibitor

0.155 0.052 CHEMBL3544873

0.172 0.031 CHEMBL3544874

0.177 0.027 CHEMBL3544897

0.177 0.027 CHEMBL3544898

0.252 0.005 CHEMBL1231106

CHEMBL1231106
0.0470.250.496CDC-like kinase 1 inhibitor

0.303 0.01 CHEMBL3544873

0.324 0.008 CHEMBL244377

0.237 0.021 CHEMBL3544874

0.412 0.004 CHEMBL3544897

0.412 0.004 CHEMBL3544898

0.496 0.004 CHEMBL1231106

0.186 0.044 CHEMBL457723

0.186 0.044 CHEMBL3544872

CHEMBL1231106
0.0130.2190.068Bruton tyrosine kinase inhibitor

0.068 0.027 CHEMBL1231106

CHEMBL1231106
0.0270.2340.202Protein kinase A inhibitor

0.094 0.05 CHEMBL3544873

0.08 0.06 CHEMBL244377

0.09 0.052 CHEMBL3544874

0.145 0.026 CHEMBL3544897

0.145 0.026 CHEMBL3544898

0.202 0.013 CHEMBL1231106

CHEMBL1231106
0.0810.2930.255Streptokinase A inhibitor

0.255 0.1 CHEMBL1231106

CHEMBL1231106
0.0630.2790.106Factor V inhibitor

0.106 0.057 CHEMBL1231106

CHEMBL1231106
0.0160.2460.054H+/K+-transporting ATPase inhibitor

0.054 0.032 CHEMBL244377

CHEMBL244377
0.0250.2550.095Platelet activating factor alpha antagonist

0.095 0.063 CHEMBL244377

0.085 0.074 CHEMBL3544897

0.085 0.074 CHEMBL3544898

0.086 0.073 CHEMBL1231106

CHEMBL244377
0.0060.2360.096Histamine H3 receptor agonist

0.024 0.023 CHEMBL3544874

0.029 0.018 CHEMBL3544897

0.029 0.018 CHEMBL3544898

0.096 0.006 CHEMBL1231106

CHEMBL1231106
0.0430.2750.66Protein kinase (CK1) gamma 2 inhibitor

0.223 0.026 CHEMBL3544873

0.213 0.028 CHEMBL244377

0.226 0.025 CHEMBL3544874

0.357 0.005 CHEMBL3544897

0.357 0.005 CHEMBL3544898

0.66 0.003 CHEMBL1231106

CHEMBL1231106
0.0280.270.147Glycogen synthase kinase-3 beta inhibitor

0.12 0.061 CHEMBL244377

0.147 0.045 CHEMBL1231106

CHEMBL1231106
0.0220.2640.159Platelet growth factor antagonist

0.079 0.058 CHEMBL3544873

0.14 0.022 CHEMBL244377

0.151 0.019 CHEMBL3544897

0.151 0.019 CHEMBL3544898

0.159 0.017 CHEMBL1231106

CHEMBL1231106
0.0040.2540.1685 Lipoxygenase activating protein inhibitor

0.016 0.006 CHEMBL3544873

0.03 0.004 CHEMBL3544874

0.026 0.004 CHEMBL3544897

0.026 0.004 CHEMBL3544898

0.168 0.002 CHEMBL1231106

CHEMBL1231106
0.0550.3070.491Protein kinase (CK1) gamma 3 inhibitor

0.225 0.035 CHEMBL3544873

0.278 0.021 CHEMBL244377

0.185 0.057 CHEMBL3544874

0.361 0.009 CHEMBL3544897

0.361 0.009 CHEMBL3544898

0.491 0.005 CHEMBL1231106

0.145 0.095 CHEMBL457723

0.145 0.095 CHEMBL3544872

CHEMBL1231106
0.0530.310.149CDK3/cyclin E inhibitor

0.149 0.027 CHEMBL244377

0.126 0.048 CHEMBL3544897

0.126 0.048 CHEMBL3544898

0.121 0.054 CHEMBL1231106

CHEMBL244377
0.1340.4140.295MAP kinase kinase 3 inhibitor

0.254 0.028 CHEMBL3544873

0.295 0.008 CHEMBL244377

0.205 0.109 CHEMBL3544874

0.295 0.008 CHEMBL3544897

0.295 0.008 CHEMBL3544898

0.24 0.042 CHEMBL1231106

0.243 0.039 CHEMBL457723

0.243 0.039 CHEMBL3544872

CHEMBL3544898
0.0550.3390.36Antimitotic

0.164 0.109 CHEMBL3544873

0.36 0.03 CHEMBL244377

0.269 0.053 CHEMBL3544897

0.269 0.053 CHEMBL3544898

0.205 0.081 CHEMBL457723

0.205 0.081 CHEMBL3544872

CHEMBL244377
0.0340.3190.226Ribosomal protein S6 kinase inhibitor

0.122 0.088 CHEMBL3544873

0.126 0.084 CHEMBL244377

0.183 0.045 CHEMBL3544897

0.183 0.045 CHEMBL3544898

0.226 0.027 CHEMBL1231106

CHEMBL1231106
0.0310.3550.549Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.184 0.071 CHEMBL3544873

0.195 0.066 CHEMBL244377

0.228 0.052 CHEMBL3544874

0.393 0.019 CHEMBL3544897

0.393 0.019 CHEMBL3544898

0.549 0.005 CHEMBL1231106

CHEMBL1231106
0.0270.3530.656Protein kinase (CK1) gamma inhibitor

0.223 0.037 CHEMBL3544873

0.23 0.035 CHEMBL244377

0.218 0.038 CHEMBL3544874

0.403 0.007 CHEMBL3544897

0.403 0.007 CHEMBL3544898

0.656 0.004 CHEMBL1231106

CHEMBL1231106
0.0090.3370.054Purinergic P2X3 antagonist

0.054 0.01 CHEMBL1231106

CHEMBL1231106
0.0280.3570.419CDC-like kinase 2 inhibitor

0.197 0.068 CHEMBL3544873

0.346 0.021 CHEMBL244377

0.368 0.018 CHEMBL3544897

0.368 0.018 CHEMBL3544898

0.419 0.011 CHEMBL1231106

0.134 0.105 CHEMBL457723

0.134 0.105 CHEMBL3544872

CHEMBL1231106
0.0540.3890.296Polo-like kinase-3 inhibitor

0.208 0.041 CHEMBL244377

0.232 0.03 CHEMBL3544897

0.232 0.03 CHEMBL3544898

0.296 0.012 CHEMBL1231106

CHEMBL1231106
0.0750.4120.174Death-associated protein kinase 2 inhibitor

0.174 0.062 CHEMBL244377

CHEMBL244377
0.0460.3840.132Transforming growth factor beta 3 antagonist

0.083 0.055 CHEMBL3544873

0.132 0.007 CHEMBL244377

0.102 0.022 CHEMBL3544897

0.102 0.022 CHEMBL3544898

0.097 0.027 CHEMBL457723

0.097 0.027 CHEMBL3544872

CHEMBL244377
0.0450.390.123Aurora-C kinase inhibitor

0.123 0.1 CHEMBL244377

CHEMBL244377
0.0130.3960.304Purinergic P2X2 antagonist

0.216 0.004 CHEMBL3544873

0.192 0.005 CHEMBL244377

0.193 0.005 CHEMBL3544874

0.26 0.003 CHEMBL3544897

0.26 0.003 CHEMBL3544898

0.304 0.002 CHEMBL1231106

0.132 0.016 CHEMBL457723

0.132 0.016 CHEMBL3544872

CHEMBL1231106
0.0260.4130.303Proto-oncogene tyrosine-protein kinase Yes inhibitor

0.151 0.06 CHEMBL3544873

0.254 0.028 CHEMBL244377

0.303 0.017 CHEMBL3544897

0.303 0.017 CHEMBL3544898

0.292 0.019 CHEMBL1231106

CHEMBL3544898
0.0110.4070.341Cyclin-dependent kinase 5 inhibitor

0.147 0.042 CHEMBL3544873

0.237 0.016 CHEMBL244377

0.287 0.011 CHEMBL3544897

0.287 0.011 CHEMBL3544898

0.341 0.007 CHEMBL1231106

0.098 0.077 CHEMBL457723

0.098 0.077 CHEMBL3544872

CHEMBL1231106
0.0420.4560.165Tumour necrosis factor alpha release inhibitor

0.165 0.139 CHEMBL244377

0.16 0.146 CHEMBL457723

0.16 0.146 CHEMBL3544872

CHEMBL244377
0.0220.440.229Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.158 0.067 CHEMBL244377

0.177 0.055 CHEMBL3544897

0.177 0.055 CHEMBL3544898

0.229 0.031 CHEMBL1231106

CHEMBL1231106
0.0110.4490.171Rho-associated kinase inhibitor

0.082 0.044 CHEMBL3544897

0.082 0.044 CHEMBL3544898

0.171 0.015 CHEMBL1231106

CHEMBL1231106
0.0080.4470.131Proto-oncogene tyrosine-protein kinase Kit inhibitor

0.131 0.04 CHEMBL244377

0.109 0.05 CHEMBL3544897

0.109 0.05 CHEMBL3544898

CHEMBL244377
0.0320.4820.205Amyloid beta precursor protein antagonist

0.205 0.054 CHEMBL244377

0.143 0.11 CHEMBL3544897

0.143 0.11 CHEMBL3544898

0.155 0.096 CHEMBL457723

0.155 0.096 CHEMBL3544872

CHEMBL244377
0.0310.4930.111Activin receptor-like kinase 4 inhibitor

0.108 0.07 CHEMBL3544897

0.108 0.07 CHEMBL3544898

0.111 0.065 CHEMBL1231106

CHEMBL1231106
0.0080.5080.112Pim-1 kinase inhibitor

0.112 0.047 CHEMBL1231106

CHEMBL1231106
0.0250.5280.177Nav1.4 sodium channel blocker

0.097 0.081 CHEMBL3544874

0.177 0.025 CHEMBL1231106

CHEMBL1231106
0.0110.5160.093MAP kinase kinase 10 inhibitor

0.093 0.021 CHEMBL244377

CHEMBL244377
0.0240.5440.446Ca2+/calmodulin-dependent kinase II beta inhibitor

0.141 0.14 CHEMBL244377

0.156 0.121 CHEMBL3544874

0.262 0.047 CHEMBL3544897

0.262 0.047 CHEMBL3544898

0.446 0.011 CHEMBL1231106

CHEMBL1231106
0.0110.5540.046Guanylate cyclase stimulant

0.046 0.025 CHEMBL1231106

CHEMBL1231106
0.0050.5610.286Growth hormone secretagogue receptor antagonist

0.055 0.015 CHEMBL3544874

0.036 0.024 CHEMBL3544897

0.036 0.024 CHEMBL3544898

0.286 0.004 CHEMBL1231106

CHEMBL1231106
0.0090.5740.109Protein kinase B beta inhibitor

0.08 0.043 CHEMBL3544897

0.08 0.043 CHEMBL3544898

0.109 0.02 CHEMBL1231106

CHEMBL1231106
0.030.5990.681Interleukin 4 antagonist

0.216 0.018 CHEMBL3544873

0.265 0.011 CHEMBL3544874

0.331 0.007 CHEMBL3544897

0.331 0.007 CHEMBL3544898

0.681 0.003 CHEMBL1231106

CHEMBL1231106
0.0310.6130.131Interleukin 2 antagonist

0.131 0.031 CHEMBL244377

CHEMBL244377
0.010.5960.15TRKB antagonist

0.15 0.047 CHEMBL1231106

CHEMBL1231106
0.0070.6050.084Rho-associated kinase II inhibitor

0.084 0.042 CHEMBL1231106

CHEMBL1231106
0.0090.6130.139Polo-like kinase-4 inhibitor

0.139 0.043 CHEMBL1231106

CHEMBL1231106
0.0560.6680.209Cyclin-dependent kinase 3 inhibitor

0.209 0.029 CHEMBL244377

0.139 0.125 CHEMBL457723

0.139 0.125 CHEMBL3544872

CHEMBL244377
0.0410.6540.389Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.17 0.119 CHEMBL3544874

0.238 0.067 CHEMBL3544897

0.238 0.067 CHEMBL3544898

0.389 0.017 CHEMBL1231106

CHEMBL1231106
0.0220.6660.276mTOR complex 1 inhibitor

0.113 0.038 CHEMBL3544873

0.12 0.029 CHEMBL3544874

0.145 0.013 CHEMBL3544897

0.145 0.013 CHEMBL3544898

0.276 0.004 CHEMBL1231106

CHEMBL1231106
0.0110.6650.501Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.156 0.115 CHEMBL3544874

0.247 0.047 CHEMBL3544897

0.247 0.047 CHEMBL3544898

0.501 0.005 CHEMBL1231106

CHEMBL1231106
0.0140.6690.482Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.141 0.083 CHEMBL3544874

0.148 0.079 CHEMBL3544897

0.148 0.079 CHEMBL3544898

0.482 0.005 CHEMBL1231106

CHEMBL1231106
0.0050.6890.188Check point kinase 2 inhibitor

0.116 0.052 CHEMBL3544897

0.116 0.052 CHEMBL3544898

0.188 0.02 CHEMBL1231106

CHEMBL1231106
0.0050.7070.063Protein kinase B alpha inhibitor

0.063 0.056 CHEMBL1231106

CHEMBL1231106
0.0070.710.126Vascular endothelial growth factor 3 antagonist

0.126 0.089 CHEMBL244377

0.117 0.098 CHEMBL3544897

0.117 0.098 CHEMBL3544898

CHEMBL244377
0.0060.7130.302MAP kinase 9 inhibitor

0.086 0.075 CHEMBL3544873

0.302 0.012 CHEMBL244377

0.246 0.016 CHEMBL3544897

0.246 0.016 CHEMBL3544898

0.092 0.069 CHEMBL1231106

CHEMBL244377
0.020.7510.258Immunosuppressant

0.222 0.174 CHEMBL244377

0.258 0.142 CHEMBL3544897

0.258 0.142 CHEMBL3544898

CHEMBL3544898
0.0090.7520.183TRKC antagonist

0.183 0.077 CHEMBL1231106

CHEMBL1231106
0.0040.750.043Factor VIIa inhibitor

0.043 0.023 CHEMBL244377

0.041 0.024 CHEMBL3544897

0.041 0.024 CHEMBL3544898

CHEMBL244377
0.0230.80.13Interleukin 12 antagonist

0.13 0.021 CHEMBL1231106

CHEMBL1231106
0.0040.790.067Urokinase inhibitor

0.067 0.025 CHEMBL1231106

CHEMBL1231106
0.0110.8030.151Interleukin 6 antagonist

0.151 0.088 CHEMBL244377

CHEMBL244377
0.0160.8090.167MAP3K9 inhibitor

0.167 0.038 CHEMBL1231106

CHEMBL1231106
0.0090.8040.138Factor XII inhibitor

0.138 0.016 CHEMBL1231106

CHEMBL1231106
0.0270.8250.152Growth factor agonist

0.152 0.137 CHEMBL3544897

0.152 0.137 CHEMBL3544898

CHEMBL3544898
0.0120.8120.048Carbonic anhydrase II stimulant

0.048 0.045 CHEMBL1231106

CHEMBL1231106
0.0060.8510.05Nicotinic acid receptor 1 agonist

0.05 0.02 CHEMBL1231106

CHEMBL1231106
0.0050.8580.106Aminoacyl-tRNA synthetase inhibitor

0.08 0.078 CHEMBL3544897

0.08 0.078 CHEMBL3544898

0.106 0.039 CHEMBL1231106

CHEMBL1231106
0.0130.8960.321Interleukin 5 antagonist

0.087 0.059 CHEMBL3544873

0.111 0.031 CHEMBL3544874

0.131 0.017 CHEMBL3544897

0.131 0.017 CHEMBL3544898

0.321 0.004 CHEMBL1231106

CHEMBL1231106
0.0090.9050.055CC chemokine receptor 2B antagonist

0.055 0.024 CHEMBL244377

0.047 0.038 CHEMBL3544897

0.047 0.038 CHEMBL3544898

CHEMBL244377
0.0080.9540.073Factor IXa inhibitor

0.073 0.019 CHEMBL1231106

CHEMBL1231106
Ext Pa Pi Pmax Activity Other Results ID Pa_max