| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.759 | 0.002 | 0.759 | Nav1.1 sodium channel blocker | 0.626 0.003 CHEMBL1908020 0.166 0.027 CHEMBL3544522 0.644 0.003 CHEMBL1908021 0.655 0.003 CHEMBL3544888 0.555 0.003 CHEMBL3638281 0.325 0.007 CHEMBL3544887 0.606 0.003 CHEMBL3548560 0.516 0.004 CHEMBL3544501 | ||
| 0.732 | 0.005 | 0.732 | Anticonvulsant | 0.513 0.011 CHEMBL1908020 0.544 0.009 CHEMBL1908021 0.533 0.01 CHEMBL3544888 0.422 0.019 CHEMBL3638281 0.495 0.012 CHEMBL3548560 0.306 0.039 CHEMBL3544501 | ||
| 0.598 | 0.003 | 0.598 | Aldose reductase inhibitor | 0.521 0.003 CHEMBL1908020 0.177 0.009 CHEMBL3544522 0.534 0.003 CHEMBL1908021 0.551 0.003 CHEMBL3544888 0.397 0.004 CHEMBL3638281 0.382 0.004 CHEMBL3544887 0.527 0.003 CHEMBL3548560 0.048 0.04 CHEMBL3544524 0.438 0.004 CHEMBL3544501 | ||
| 0.534 | 0.006 | 0.564 | Anesthetic general | 0.546 0.005 CHEMBL1908020 0.465 0.01 CHEMBL3544522 0.564 0.005 CHEMBL1908021 0.557 0.005 CHEMBL3544888 0.551 0.005 CHEMBL3638281 0.409 0.015 CHEMBL3544523 0.539 0.006 CHEMBL3544887 0.537 0.006 CHEMBL3548560 0.371 0.02 CHEMBL3544524 0.528 0.006 CHEMBL3544501 | CHEMBL1908021 | |
| 0.536 | 0.028 | 0.714 | Aldehyde oxidase inhibitor | 0.705 0.008 CHEMBL1908020 0.69 0.009 CHEMBL1908021 0.687 0.009 CHEMBL3544888 0.417 0.044 CHEMBL3638281 0.311 0.063 CHEMBL3544523 0.698 0.008 CHEMBL3548560 0.642 0.014 CHEMBL3544524 0.714 0.007 CHEMBL3544501 | CHEMBL3544501 | |
| 0.483 | 0.031 | 0.514 | GABA C receptor rho-3 antagonist | 0.483 0.031 CHEMBL1908020 0.514 0.022 CHEMBL1908021 0.51 0.023 CHEMBL3544888 0.26 0.145 CHEMBL3638281 0.327 0.099 CHEMBL3544523 0.424 0.051 CHEMBL3548560 0.495 0.027 CHEMBL3544524 0.239 0.165 CHEMBL3544501 | CHEMBL1908021 | |
| 0.433 | 0.005 | 0.554 | Tumour necrosis factor antagonist | 0.443 0.005 CHEMBL1908020 0.42 0.005 CHEMBL1908021 0.426 0.005 CHEMBL3544888 0.362 0.009 CHEMBL3638281 0.199 0.054 CHEMBL3544887 0.448 0.005 CHEMBL3548560 0.554 0.004 CHEMBL3544501 | CHEMBL3544501 | |
| 0.486 | 0.066 | 0.747 | Caspase 9 stimulant | 0.598 0.036 CHEMBL1908020 0.499 0.06 CHEMBL3544522 0.563 0.042 CHEMBL1908021 0.567 0.041 CHEMBL3544888 0.425 0.097 CHEMBL3638281 0.529 0.05 CHEMBL3544887 0.625 0.033 CHEMBL3548560 0.415 0.102 CHEMBL3544524 0.747 0.018 CHEMBL3544501 | CHEMBL3544501 | |
| 0.467 | 0.051 | 0.467 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.324 0.182 CHEMBL1908020 0.351 0.149 CHEMBL1908021 0.348 0.153 CHEMBL3544888 0.307 0.203 CHEMBL3638281 0.397 0.103 CHEMBL3544523 0.324 0.182 CHEMBL3548560 0.432 0.074 CHEMBL3544524 | ||
| 0.347 | 0.024 | 0.379 | RNA-directed DNA polymerase inhibitor | 0.354 0.023 CHEMBL1908020 0.242 0.055 CHEMBL3544522 0.363 0.022 CHEMBL1908021 0.377 0.021 CHEMBL3544888 0.314 0.029 CHEMBL3638281 0.192 0.112 CHEMBL3544523 0.285 0.035 CHEMBL3544887 0.379 0.02 CHEMBL3548560 0.264 0.042 CHEMBL3544524 0.344 0.025 CHEMBL3544501 | CHEMBL3548560 | |
| 0.299 | 0.004 | 0.299 | Phosphodiesterase 7B inhibitor | 0.207 0.009 CHEMBL1908020 0.213 0.009 CHEMBL1908021 0.217 0.009 CHEMBL3544888 0.181 0.013 CHEMBL3638281 0.207 0.009 CHEMBL3548560 0.191 0.011 CHEMBL3544501 | ||
| 0.346 | 0.054 | 0.509 | Spasmolytic | 0.393 0.041 CHEMBL1908020 0.337 0.057 CHEMBL3544522 0.388 0.043 CHEMBL1908021 0.378 0.045 CHEMBL3544888 0.248 0.092 CHEMBL3638281 0.509 0.022 CHEMBL3544887 0.412 0.038 CHEMBL3548560 0.172 0.143 CHEMBL3544524 0.434 0.034 CHEMBL3544501 | CHEMBL3544887 | |
| 0.275 | 0.003 | 0.275 | Phosphodiesterase VII inhibitor | 0.146 0.005 CHEMBL1908020 0.149 0.004 CHEMBL1908021 0.155 0.004 CHEMBL3544888 0.126 0.005 CHEMBL3638281 0.148 0.004 CHEMBL3548560 0.132 0.005 CHEMBL3544501 | ||
| 0.311 | 0.052 | 0.311 | Cardiotonic | 0.229 0.097 CHEMBL1908020 0.229 0.097 CHEMBL1908021 0.235 0.093 CHEMBL3544888 0.24 0.09 CHEMBL3638281 0.253 0.08 CHEMBL3548560 0.246 0.085 CHEMBL3544501 | ||
| 0.268 | 0.012 | 0.45 | UDP-glucose 4-epimerase inhibitor | 0.243 0.014 CHEMBL1908020 0.439 0.004 CHEMBL3544522 0.278 0.011 CHEMBL1908021 0.298 0.01 CHEMBL3544888 0.3 0.01 CHEMBL3638281 0.121 0.042 CHEMBL3544523 0.45 0.004 CHEMBL3544887 0.243 0.014 CHEMBL3548560 0.205 0.017 CHEMBL3544524 0.132 0.036 CHEMBL3544501 | CHEMBL3544887 | |
| 0.366 | 0.111 | 0.802 | Cyclophilin D inhibitor | 0.373 0.107 CHEMBL1908020 0.627 0.023 CHEMBL3544522 0.385 0.099 CHEMBL1908021 0.402 0.09 CHEMBL3544888 0.376 0.105 CHEMBL3638281 0.802 0.007 CHEMBL3544887 0.398 0.092 CHEMBL3548560 0.241 0.223 CHEMBL3544524 0.289 0.172 CHEMBL3544501 | CHEMBL3544887 | |
| 0.257 | 0.007 | 0.38 | Alcohol dehydrogenase inhibitor | 0.378 0.004 CHEMBL1908020 0.087 0.068 CHEMBL3544522 0.364 0.004 CHEMBL1908021 0.38 0.004 CHEMBL3544888 0.145 0.022 CHEMBL3638281 0.085 0.071 CHEMBL3544523 0.273 0.006 CHEMBL3544887 0.339 0.005 CHEMBL3548560 0.192 0.013 CHEMBL3544524 0.222 0.01 CHEMBL3544501 | CHEMBL3544888 | |
| 0.287 | 0.04 | 0.579 | Tyrosine 3 hydroxylase inhibitor | 0.333 0.02 CHEMBL1908020 0.356 0.015 CHEMBL1908021 0.355 0.015 CHEMBL3544888 0.206 0.125 CHEMBL3638281 0.399 0.008 CHEMBL3544523 0.333 0.02 CHEMBL3548560 0.579 0.003 CHEMBL3544524 0.283 0.042 CHEMBL3544501 | CHEMBL3544524 | |
| 0.279 | 0.037 | 0.338 | Growth hormone agonist | 0.265 0.04 CHEMBL1908020 0.29 0.034 CHEMBL1908021 0.293 0.034 CHEMBL3544888 0.25 0.043 CHEMBL3638281 0.236 0.047 CHEMBL3544523 0.237 0.047 CHEMBL3548560 0.338 0.025 CHEMBL3544524 0.181 0.067 CHEMBL3544501 | CHEMBL3544524 | |
| 0.368 | 0.13 | 0.471 | DNA directed DNA polymerase inhibitor | 0.382 0.123 CHEMBL1908020 0.394 0.118 CHEMBL1908021 0.392 0.119 CHEMBL3544888 0.433 0.103 CHEMBL3548560 0.471 0.091 CHEMBL3544501 | CHEMBL3544501 | |
| 0.31 | 0.076 | 0.597 | Immunostimulant | 0.334 0.069 CHEMBL1908020 0.493 0.03 CHEMBL3544522 0.35 0.064 CHEMBL1908021 0.357 0.062 CHEMBL3544888 0.416 0.045 CHEMBL3638281 0.159 0.147 CHEMBL3544523 0.597 0.017 CHEMBL3544887 0.325 0.072 CHEMBL3548560 0.235 0.103 CHEMBL3544524 0.264 0.091 CHEMBL3544501 | CHEMBL3544887 | |
| 0.268 | 0.039 | 0.421 | Peptidyltransferase inhibitor | 0.273 0.036 CHEMBL1908020 0.384 0.008 CHEMBL3544522 0.284 0.031 CHEMBL1908021 0.289 0.029 CHEMBL3544888 0.335 0.015 CHEMBL3638281 0.258 0.045 CHEMBL3544523 0.421 0.005 CHEMBL3544887 0.28 0.033 CHEMBL3548560 0.293 0.027 CHEMBL3544524 0.253 0.049 CHEMBL3544501 | CHEMBL3544887 | |
| 0.277 | 0.052 | 0.451 | DNA synthesis inhibitor | 0.279 0.051 CHEMBL1908020 0.39 0.023 CHEMBL3544522 0.29 0.047 CHEMBL1908021 0.307 0.041 CHEMBL3544888 0.332 0.034 CHEMBL3638281 0.249 0.067 CHEMBL3544523 0.451 0.017 CHEMBL3544887 0.257 0.062 CHEMBL3548560 0.311 0.04 CHEMBL3544524 0.216 0.099 CHEMBL3544501 | CHEMBL3544887 | |
| 0.281 | 0.058 | 0.572 | Superoxide dismutase inhibitor | 0.358 0.035 CHEMBL1908020 0.355 0.035 CHEMBL1908021 0.349 0.037 CHEMBL3544888 0.2 0.118 CHEMBL3638281 0.572 0.008 CHEMBL3544523 0.393 0.028 CHEMBL3548560 0.572 0.008 CHEMBL3544524 0.452 0.019 CHEMBL3544501 | CHEMBL3544524 | |
| 0.231 | 0.012 | 0.231 | Nav1.6 sodium channel blocker | 0.183 0.027 CHEMBL1908020 0.189 0.024 CHEMBL1908021 0.188 0.024 CHEMBL3544888 0.121 0.094 CHEMBL3638281 0.168 0.037 CHEMBL3548560 0.153 0.05 CHEMBL3544501 | ||
| 0.234 | 0.016 | 0.486 | Ferrochelatase inhibitor | 0.103 0.068 CHEMBL1908020 0.121 0.053 CHEMBL1908021 0.136 0.044 CHEMBL3544888 0.101 0.07 CHEMBL3638281 0.311 0.007 CHEMBL3544523 0.103 0.068 CHEMBL3548560 0.486 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.267 | 0.056 | 0.42 | Cyclic AMP phosphodiesterase inhibitor | 0.293 0.045 CHEMBL1908020 0.213 0.084 CHEMBL3544522 0.271 0.054 CHEMBL1908021 0.278 0.051 CHEMBL3544888 0.229 0.075 CHEMBL3638281 0.42 0.014 CHEMBL3544887 0.31 0.038 CHEMBL3548560 0.343 0.027 CHEMBL3544501 | CHEMBL3544887 | |
| 0.258 | 0.046 | 0.575 | Peroxidase inhibitor | 0.46 0.013 CHEMBL1908020 0.453 0.014 CHEMBL1908021 0.458 0.013 CHEMBL3544888 0.127 0.093 CHEMBL3638281 0.548 0.006 CHEMBL3544523 0.462 0.013 CHEMBL3548560 0.575 0.005 CHEMBL3544524 0.353 0.028 CHEMBL3544501 | CHEMBL3544524 | |
| 0.212 | 0.014 | 0.361 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.15 0.027 CHEMBL1908020 0.229 0.012 CHEMBL3544522 0.174 0.02 CHEMBL1908021 0.181 0.019 CHEMBL3544888 0.18 0.019 CHEMBL3638281 0.211 0.014 CHEMBL3544523 0.251 0.01 CHEMBL3544887 0.15 0.027 CHEMBL3548560 0.361 0.004 CHEMBL3544524 0.091 0.064 CHEMBL3544501 | CHEMBL3544524 | |
| 0.323 | 0.125 | 0.754 | Analgesic | 0.267 0.168 CHEMBL1908020 0.284 0.154 CHEMBL1908021 0.286 0.153 CHEMBL3544888 0.241 0.191 CHEMBL3544523 0.754 0.009 CHEMBL3544524 | CHEMBL3544524 | |
| 0.251 | 0.055 | 0.251 | Neuropeptide Y2 antagonist | 0.241 0.065 CHEMBL1908020 0.251 0.056 CHEMBL1908021 0.247 0.059 CHEMBL3544888 0.202 0.115 CHEMBL3544523 0.212 0.1 CHEMBL3548560 0.194 0.13 CHEMBL3544524 0.176 0.169 CHEMBL3544501 | ||
| 0.279 | 0.085 | 0.279 | Nootropic | |||
| 0.22 | 0.029 | 0.64 | Alpha-N-acetylglucosaminidase inhibitor | 0.15 0.055 CHEMBL1908020 0.418 0.008 CHEMBL3544522 0.171 0.045 CHEMBL1908021 0.194 0.036 CHEMBL3544888 0.261 0.021 CHEMBL3638281 0.422 0.008 CHEMBL3544523 0.297 0.016 CHEMBL3544887 0.15 0.055 CHEMBL3548560 0.64 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.219 | 0.028 | 0.219 | Nav1.2 sodium channel blocker | 0.164 0.049 CHEMBL1908020 0.178 0.043 CHEMBL1908021 0.171 0.046 CHEMBL3544888 0.139 0.064 CHEMBL3548560 0.118 0.086 CHEMBL3544501 | ||
| 0.187 | 0.004 | 0.187 | Cathepsin E inhibitor | 0.126 0.008 CHEMBL1908020 0.072 0.028 CHEMBL3544522 0.132 0.007 CHEMBL1908021 0.136 0.006 CHEMBL3544888 0.115 0.01 CHEMBL3638281 0.069 0.03 CHEMBL3544887 0.123 0.008 CHEMBL3548560 0.102 0.013 CHEMBL3544501 | ||
| 0.178 | 0.003 | 0.178 | Phosphodiesterase 7A inhibitor | 0.108 0.004 CHEMBL1908020 0.112 0.004 CHEMBL1908021 0.117 0.004 CHEMBL3544888 0.093 0.005 CHEMBL3638281 0.11 0.004 CHEMBL3548560 0.094 0.005 CHEMBL3544501 | ||
| 0.251 | 0.078 | 0.289 | Gastrin inhibitor | 0.199 0.151 CHEMBL1908021 0.195 0.157 CHEMBL3544888 0.287 0.042 CHEMBL3544523 0.289 0.041 CHEMBL3544524 | CHEMBL3544524 | |
| 0.193 | 0.022 | 0.667 | GABA C receptor agonist | 0.142 0.037 CHEMBL1908020 0.162 0.03 CHEMBL1908021 0.185 0.023 CHEMBL3544888 0.112 0.056 CHEMBL3638281 0.425 0.005 CHEMBL3544523 0.142 0.037 CHEMBL3548560 0.667 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.198 | 0.03 | 0.208 | GABA C receptor rho-2 antagonist | 0.194 0.032 CHEMBL1908020 0.194 0.032 CHEMBL1908021 0.19 0.035 CHEMBL3544888 0.139 0.09 CHEMBL3544523 0.169 0.051 CHEMBL3548560 0.208 0.025 CHEMBL3544524 0.162 0.059 CHEMBL3544501 | CHEMBL3544524 | |
| 0.194 | 0.027 | 0.194 | Nav1.3 sodium channel blocker | 0.132 0.062 CHEMBL1908020 0.144 0.052 CHEMBL1908021 0.14 0.055 CHEMBL3544888 0.117 0.077 CHEMBL3548560 | ||
| 0.223 | 0.056 | 0.277 | Nitric-oxide synthase stimulant | 0.244 0.037 CHEMBL1908020 0.232 0.047 CHEMBL3544522 0.236 0.043 CHEMBL1908021 0.245 0.036 CHEMBL3544888 0.204 0.082 CHEMBL3638281 0.213 0.069 CHEMBL3544523 0.232 0.047 CHEMBL3544887 0.249 0.033 CHEMBL3548560 0.277 0.018 CHEMBL3544524 0.249 0.033 CHEMBL3544501 | CHEMBL3544524 | |
| 0.248 | 0.083 | 0.465 | 5 Hydroxytryptamine uptake stimulant | 0.244 0.087 CHEMBL1908020 0.244 0.087 CHEMBL1908021 0.241 0.09 CHEMBL3544888 0.188 0.177 CHEMBL3638281 0.308 0.041 CHEMBL3544523 0.283 0.055 CHEMBL3548560 0.465 0.006 CHEMBL3544524 0.273 0.061 CHEMBL3544501 | CHEMBL3544524 | |
| 0.319 | 0.155 | 0.425 | DNA polymerase beta inhibitor | 0.327 0.151 CHEMBL1908020 0.337 0.145 CHEMBL1908021 0.332 0.148 CHEMBL3544888 0.374 0.129 CHEMBL3548560 0.425 0.11 CHEMBL3544501 | CHEMBL3544501 | |
| 0.239 | 0.075 | 0.396 | Vasodilator | 0.262 0.063 CHEMBL1908020 0.29 0.052 CHEMBL3544522 0.263 0.063 CHEMBL1908021 0.27 0.059 CHEMBL3544888 0.179 0.122 CHEMBL3638281 0.396 0.024 CHEMBL3544887 0.291 0.051 CHEMBL3548560 0.295 0.05 CHEMBL3544501 | CHEMBL3544887 | |
| 0.314 | 0.15 | 0.514 | 5 Hydroxytryptamine release inhibitor | 0.338 0.126 CHEMBL1908020 0.305 0.16 CHEMBL3544522 0.337 0.127 CHEMBL1908021 0.336 0.127 CHEMBL3544888 0.325 0.138 CHEMBL3544523 0.399 0.079 CHEMBL3544887 0.296 0.169 CHEMBL3548560 0.514 0.028 CHEMBL3544524 0.278 0.191 CHEMBL3544501 | CHEMBL3544524 | |
| 0.25 | 0.089 | 0.561 | 5 Hydroxytryptamine release stimulant | 0.282 0.076 CHEMBL1908020 0.262 0.083 CHEMBL1908021 0.252 0.088 CHEMBL3544888 0.281 0.076 CHEMBL3544523 0.164 0.16 CHEMBL3544887 0.221 0.105 CHEMBL3548560 0.561 0.019 CHEMBL3544524 0.238 0.095 CHEMBL3544501 | CHEMBL3544524 | |
| 0.158 | 0.009 | 0.158 | Phosphodiesterase III inhibitor | 0.141 0.011 CHEMBL1908020 0.119 0.016 CHEMBL1908021 0.127 0.013 CHEMBL3544888 0.138 0.012 CHEMBL3548560 0.152 0.01 CHEMBL3544501 | ||
| 0.15 | 0.009 | 0.297 | Biliverdin reductase inhibitor | 0.087 0.023 CHEMBL1908020 0.077 0.028 CHEMBL3544522 0.101 0.018 CHEMBL1908021 0.117 0.014 CHEMBL3544888 0.137 0.011 CHEMBL3638281 0.168 0.008 CHEMBL3544523 0.064 0.036 CHEMBL3544887 0.087 0.023 CHEMBL3548560 0.297 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.153 | 0.017 | 0.295 | NADH dehydrogenase inhibitor | 0.15 0.018 CHEMBL1908020 0.292 0.007 CHEMBL3544522 0.152 0.017 CHEMBL1908021 0.168 0.014 CHEMBL3544888 0.163 0.015 CHEMBL3638281 0.131 0.023 CHEMBL3544523 0.295 0.007 CHEMBL3544887 0.15 0.018 CHEMBL3548560 0.228 0.009 CHEMBL3544524 0.109 0.035 CHEMBL3544501 | CHEMBL3544887 | |
| 0.137 | 0.003 | 0.137 | Calcitonin gene-related peptide antagonist | 0.076 0.004 CHEMBL1908020 0.078 0.004 CHEMBL1908021 0.08 0.004 CHEMBL3544888 0.071 0.004 CHEMBL3638281 0.033 0.014 CHEMBL3544887 0.074 0.004 CHEMBL3548560 0.064 0.005 CHEMBL3544501 | ||
| 0.158 | 0.025 | 0.327 | DNA repair enzyme inhibitor | 0.152 0.03 CHEMBL1908020 0.23 0.006 CHEMBL3544522 0.156 0.027 CHEMBL1908021 0.156 0.026 CHEMBL3544888 0.134 0.05 CHEMBL3638281 0.327 0.004 CHEMBL3544887 0.154 0.028 CHEMBL3548560 0.126 0.062 CHEMBL3544524 0.154 0.028 CHEMBL3544501 | CHEMBL3544887 | |
| 0.131 | 0.003 | 0.131 | Calcitonin gene-related peptide 1 receptor antagonist | 0.088 0.004 CHEMBL1908020 0.099 0.004 CHEMBL1908021 0.102 0.004 CHEMBL3544888 0.043 0.005 CHEMBL3638281 0.077 0.004 CHEMBL3548560 0.021 0.008 CHEMBL3544501 | ||
| 0.132 | 0.004 | 0.132 | Phospholipase D inhibitor | 0.102 0.013 CHEMBL1908020 0.11 0.01 CHEMBL1908021 0.109 0.01 CHEMBL3544888 0.098 0.016 CHEMBL3638281 0.081 0.034 CHEMBL3544523 0.097 0.017 CHEMBL3548560 0.102 0.013 CHEMBL3544524 | ||
| 0.268 | 0.143 | 0.472 | Histamine release inhibitor | 0.377 0.087 CHEMBL1908020 0.45 0.05 CHEMBL3544522 0.361 0.095 CHEMBL1908021 0.358 0.096 CHEMBL3544888 0.279 0.136 CHEMBL3544523 0.472 0.04 CHEMBL3544887 0.396 0.078 CHEMBL3548560 0.457 0.047 CHEMBL3544524 0.348 0.101 CHEMBL3544501 | CHEMBL3544887 | |
| 0.157 | 0.032 | 0.157 | 5 Hydroxytryptamine 3A agonist | 0.144 0.039 CHEMBL1908020 0.137 0.043 CHEMBL1908021 0.136 0.044 CHEMBL3544888 0.113 0.062 CHEMBL3548560 0.091 0.088 CHEMBL3544524 | ||
| 0.147 | 0.025 | 0.147 | DNA directed RNA polymerase inhibitor | 0.098 0.059 CHEMBL1908020 0.106 0.05 CHEMBL1908021 0.109 0.046 CHEMBL3544888 0.1 0.057 CHEMBL3638281 0.104 0.052 CHEMBL3548560 | ||
| 0.194 | 0.072 | 0.199 | 5 Hydroxytryptamine 3E antagonist | 0.199 0.063 CHEMBL3544524 | CHEMBL3544524 | |
| 0.229 | 0.118 | 0.348 | Insulysin inhibitor | 0.238 0.108 CHEMBL1908020 0.249 0.097 CHEMBL1908021 0.246 0.1 CHEMBL3544888 0.293 0.063 CHEMBL3544523 0.239 0.107 CHEMBL3548560 0.348 0.035 CHEMBL3544524 0.205 0.149 CHEMBL3544501 | CHEMBL3544524 | |
| 0.171 | 0.06 | 0.171 | Cyclin-dependent kinase 8 inhibitor | 0.129 0.104 CHEMBL1908020 0.135 0.097 CHEMBL1908021 0.141 0.089 CHEMBL3544888 0.131 0.101 CHEMBL3548560 | ||
| 0.14 | 0.029 | 0.265 | HIV-1 integrase (Overall Integration) inhibitor | 0.145 0.027 CHEMBL1908020 0.158 0.023 CHEMBL1908021 0.153 0.024 CHEMBL3544888 0.088 0.067 CHEMBL3638281 0.175 0.017 CHEMBL3544523 0.184 0.015 CHEMBL3548560 0.265 0.004 CHEMBL3544524 0.123 0.038 CHEMBL3544501 | CHEMBL3544524 | |
| 0.171 | 0.06 | 0.226 | Neurotensin receptor agonist | 0.199 0.035 CHEMBL1908020 0.197 0.036 CHEMBL1908021 0.198 0.035 CHEMBL3544888 0.18 0.049 CHEMBL3544523 0.177 0.053 CHEMBL3548560 0.226 0.026 CHEMBL3544524 0.182 0.048 CHEMBL3544501 | CHEMBL3544524 | |
| 0.127 | 0.019 | 0.127 | Bromodomain-containing protein 2 inhibitor | 0.092 0.053 CHEMBL1908020 0.091 0.054 CHEMBL1908021 0.094 0.049 CHEMBL3544888 0.09 0.055 CHEMBL3548560 0.081 0.075 CHEMBL3544501 | ||
| 0.252 | 0.145 | 0.371 | Calcium channel activator | 0.226 0.177 CHEMBL1908020 0.237 0.163 CHEMBL1908021 0.233 0.168 CHEMBL3544888 0.227 0.175 CHEMBL3544523 0.371 0.037 CHEMBL3544524 0.258 0.138 CHEMBL3544501 | CHEMBL3544524 | |
| 0.161 | 0.055 | 0.214 | Mannose-6-phosphate isomerase inhibitor | 0.149 0.065 CHEMBL1908020 0.161 0.055 CHEMBL3544522 0.157 0.059 CHEMBL1908021 0.152 0.062 CHEMBL3544888 0.121 0.098 CHEMBL3638281 0.167 0.051 CHEMBL3544887 0.185 0.039 CHEMBL3548560 0.214 0.024 CHEMBL3544524 0.173 0.047 CHEMBL3544501 | CHEMBL3544524 | |
| 0.156 | 0.05 | 0.156 | Sodium channel (voltage-gated) blocker | |||
| 0.148 | 0.047 | 0.184 | Ca2+-transporting ATPase inhibitor | 0.141 0.068 CHEMBL1908020 0.151 0.041 CHEMBL3544522 0.146 0.054 CHEMBL1908021 0.147 0.049 CHEMBL3544888 0.148 0.046 CHEMBL3638281 0.152 0.039 CHEMBL3544523 0.141 0.07 CHEMBL3544887 0.141 0.068 CHEMBL3548560 0.184 0.005 CHEMBL3544524 0.129 0.126 CHEMBL3544501 | CHEMBL3544524 | |
| 0.112 | 0.013 | 0.112 | Secretase beta inhibitor | 0.088 0.027 CHEMBL1908020 0.089 0.026 CHEMBL1908021 0.09 0.025 CHEMBL3544888 0.072 0.047 CHEMBL3638281 0.087 0.028 CHEMBL3548560 0.065 0.06 CHEMBL3544524 0.072 0.046 CHEMBL3544501 | ||
| 0.126 | 0.027 | 0.134 | Metalloproteinase-2 inhibitor | 0.124 0.028 CHEMBL1908020 0.134 0.024 CHEMBL1908021 0.134 0.024 CHEMBL3544888 0.074 0.06 CHEMBL3638281 0.127 0.026 CHEMBL3548560 0.077 0.055 CHEMBL3544524 0.114 0.032 CHEMBL3544501 | CHEMBL3544888 | |
| 0.174 | 0.075 | 0.396 | Succinate dehydrogenase inhibitor | 0.186 0.062 CHEMBL1908020 0.184 0.064 CHEMBL1908021 0.186 0.061 CHEMBL3544888 0.256 0.02 CHEMBL3544523 0.205 0.045 CHEMBL3548560 0.396 0.004 CHEMBL3544524 0.204 0.046 CHEMBL3544501 | CHEMBL3544524 | |
| 0.122 | 0.024 | 0.131 | Metalloproteinase-9 inhibitor | 0.121 0.024 CHEMBL1908020 0.131 0.021 CHEMBL1908021 0.131 0.021 CHEMBL3544888 0.068 0.059 CHEMBL3638281 0.126 0.023 CHEMBL3548560 0.117 0.026 CHEMBL3544501 | CHEMBL3544888 | |
| 0.14 | 0.045 | 0.279 | Cystathionine beta-synthase inhibitor | 0.259 0.014 CHEMBL1908020 0.132 0.05 CHEMBL3544522 0.244 0.016 CHEMBL1908021 0.249 0.015 CHEMBL3544888 0.113 0.064 CHEMBL3638281 0.15 0.04 CHEMBL3544523 0.193 0.026 CHEMBL3544887 0.261 0.014 CHEMBL3548560 0.279 0.012 CHEMBL3544524 0.234 0.018 CHEMBL3544501 | CHEMBL3544524 | |
| 0.108 | 0.013 | 0.156 | NMDA receptor glycine site agonist | 0.083 0.026 CHEMBL1908020 0.09 0.022 CHEMBL1908021 0.09 0.022 CHEMBL3544888 0.156 0.004 CHEMBL3544523 0.083 0.026 CHEMBL3548560 0.139 0.005 CHEMBL3544524 | CHEMBL3544523 | |
| 0.128 | 0.034 | 0.238 | GABA C receptor rho-1 antagonist | 0.111 0.049 CHEMBL1908020 0.115 0.045 CHEMBL1908021 0.115 0.044 CHEMBL3544888 0.143 0.024 CHEMBL3544523 0.095 0.069 CHEMBL3548560 0.238 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.119 | 0.028 | 0.119 | Phosphodiesterase I inhibitor | 0.109 0.035 CHEMBL1908020 0.107 0.037 CHEMBL1908021 0.109 0.035 CHEMBL3544888 0.095 0.051 CHEMBL3638281 0.107 0.037 CHEMBL3548560 0.118 0.028 CHEMBL3544501 | ||
| 0.104 | 0.013 | 0.121 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.074 0.023 CHEMBL1908020 0.107 0.013 CHEMBL3544522 0.083 0.019 CHEMBL1908021 0.087 0.018 CHEMBL3544888 0.117 0.011 CHEMBL3638281 0.067 0.028 CHEMBL3544523 0.098 0.015 CHEMBL3544887 0.074 0.023 CHEMBL3548560 0.121 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.104 | 0.015 | 0.104 | Collagenase 3 inhibitor | 0.077 0.026 CHEMBL1908020 0.085 0.022 CHEMBL1908021 0.086 0.021 CHEMBL3544888 0.075 0.028 CHEMBL3548560 0.072 0.03 CHEMBL3544501 | ||
| 0.095 | 0.011 | 0.095 | Phosphodiesterase 1A inhibitor | 0.066 0.03 CHEMBL1908020 0.067 0.028 CHEMBL1908021 0.067 0.027 CHEMBL3544888 0.065 0.031 CHEMBL3548560 0.059 0.043 CHEMBL3544501 | ||
| 0.122 | 0.039 | 0.292 | Creatine kinase inhibitor | 0.21 0.009 CHEMBL1908020 0.2 0.01 CHEMBL1908021 0.203 0.01 CHEMBL3544888 0.112 0.048 CHEMBL3638281 0.153 0.023 CHEMBL3544523 0.209 0.009 CHEMBL3548560 0.292 0.004 CHEMBL3544524 0.117 0.043 CHEMBL3544501 | CHEMBL3544524 | |
| 0.09 | 0.007 | 0.098 | Dihydroorotate oxidase inhibitor | 0.085 0.008 CHEMBL1908020 0.094 0.006 CHEMBL1908021 0.098 0.005 CHEMBL3544888 0.057 0.034 CHEMBL3638281 0.092 0.006 CHEMBL3548560 0.061 0.027 CHEMBL3544524 0.059 0.03 CHEMBL3544501 | CHEMBL3544888 | |
| 0.1 | 0.021 | 0.331 | Carbamoyl phosphate synthetase inhibitor | 0.074 0.032 CHEMBL1908020 0.071 0.034 CHEMBL3544522 0.084 0.027 CHEMBL1908021 0.094 0.023 CHEMBL3544888 0.109 0.018 CHEMBL3638281 0.331 0.004 CHEMBL3544523 0.074 0.032 CHEMBL3548560 0.295 0.004 CHEMBL3544524 | CHEMBL3544523 | |
| 0.126 | 0.047 | 0.271 | GABA C receptor antagonist | 0.111 0.062 CHEMBL1908020 0.119 0.054 CHEMBL1908021 0.122 0.05 CHEMBL3544888 0.148 0.031 CHEMBL3544523 0.098 0.082 CHEMBL3548560 0.271 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.116 | 0.04 | 0.2 | Electrolyte absorption antagonist | 0.089 0.076 CHEMBL1908021 0.091 0.072 CHEMBL3544888 0.2 0.008 CHEMBL3544523 0.184 0.01 CHEMBL3544524 | CHEMBL3544523 | |
| 0.095 | 0.021 | 0.227 | NMDA receptor agonist | 0.071 0.035 CHEMBL1908020 0.08 0.029 CHEMBL1908021 0.081 0.028 CHEMBL3544888 0.227 0.004 CHEMBL3544523 0.066 0.039 CHEMBL3548560 0.198 0.005 CHEMBL3544524 | CHEMBL3544523 | |
| 0.119 | 0.045 | 0.319 | Adenylate kinase inhibitor | 0.094 0.078 CHEMBL1908020 0.101 0.066 CHEMBL3544522 0.102 0.064 CHEMBL1908021 0.108 0.056 CHEMBL3544888 0.124 0.04 CHEMBL3638281 0.302 0.007 CHEMBL3544523 0.094 0.078 CHEMBL3548560 0.319 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.102 | 0.029 | 0.179 | Keratolytic | 0.17 0.011 CHEMBL1908020 0.176 0.011 CHEMBL1908021 0.179 0.01 CHEMBL3544888 0.087 0.04 CHEMBL3638281 0.148 0.015 CHEMBL3544523 0.168 0.012 CHEMBL3548560 0.169 0.012 CHEMBL3544524 0.177 0.011 CHEMBL3544501 | CHEMBL3544888 | |
| 0.104 | 0.03 | 0.273 | Phosphofructokinase-1 inhibitor | 0.089 0.036 CHEMBL1908020 0.206 0.01 CHEMBL3544522 0.102 0.031 CHEMBL1908021 0.117 0.026 CHEMBL3544888 0.12 0.025 CHEMBL3638281 0.168 0.015 CHEMBL3544523 0.198 0.011 CHEMBL3544887 0.089 0.036 CHEMBL3548560 0.273 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.093 | 0.021 | 0.249 | Argininosuccinate synthase inhibitor | 0.064 0.034 CHEMBL1908020 0.049 0.048 CHEMBL3544522 0.074 0.028 CHEMBL1908021 0.08 0.025 CHEMBL3544888 0.093 0.021 CHEMBL3638281 0.155 0.011 CHEMBL3544523 0.064 0.034 CHEMBL3548560 0.249 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.106 | 0.035 | 0.117 | Interleukin 5 antagonist | 0.112 0.03 CHEMBL1908020 0.117 0.026 CHEMBL1908021 0.117 0.026 CHEMBL3544888 0.091 0.053 CHEMBL3638281 0.107 0.034 CHEMBL3544887 0.096 0.046 CHEMBL3548560 0.089 0.057 CHEMBL3544501 | CHEMBL3544888 | |
| 0.086 | 0.015 | 0.086 | Phosphodiesterase 1C inhibitor | 0.076 0.022 CHEMBL1908020 0.077 0.022 CHEMBL1908021 0.077 0.021 CHEMBL3544888 0.078 0.021 CHEMBL3548560 0.075 0.024 CHEMBL3544501 | ||
| 0.089 | 0.018 | 0.132 | Glutamate (mGluR7) antagonist | 0.084 0.023 CHEMBL1908020 0.084 0.023 CHEMBL1908021 0.082 0.025 CHEMBL3544888 0.081 0.027 CHEMBL3544523 0.077 0.032 CHEMBL3548560 0.132 0.004 CHEMBL3544524 0.078 0.03 CHEMBL3544501 | CHEMBL3544524 | |
| 0.108 | 0.041 | 0.375 | Triose-phosphate isomerase inhibitor | 0.089 0.061 CHEMBL1908020 0.216 0.009 CHEMBL3544522 0.098 0.05 CHEMBL1908021 0.102 0.046 CHEMBL3544888 0.105 0.043 CHEMBL3638281 0.211 0.01 CHEMBL3544523 0.186 0.013 CHEMBL3544887 0.089 0.061 CHEMBL3548560 0.375 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.099 | 0.033 | 0.127 | Glycine receptor antagonist | 0.078 0.061 CHEMBL1908020 0.11 0.024 CHEMBL3544522 0.079 0.059 CHEMBL1908021 0.078 0.06 CHEMBL3544888 0.096 0.036 CHEMBL3638281 0.086 0.048 CHEMBL3544523 0.127 0.015 CHEMBL3544887 0.078 0.061 CHEMBL3548560 0.099 0.033 CHEMBL3544524 | CHEMBL3544887 | |
| 0.069 | 0.004 | 0.079 | Uridine phosphorylase inhibitor | 0.059 0.005 CHEMBL1908020 0.06 0.005 CHEMBL3544522 0.066 0.005 CHEMBL1908021 0.064 0.005 CHEMBL3544888 0.066 0.005 CHEMBL3638281 0.024 0.023 CHEMBL3544523 0.079 0.004 CHEMBL3544887 0.059 0.005 CHEMBL3548560 0.05 0.008 CHEMBL3544524 0.043 0.01 CHEMBL3544501 | CHEMBL3544887 | |
| 0.082 | 0.017 | 0.082 | MDM2 inhibitor | 0.066 0.052 CHEMBL1908020 0.07 0.039 CHEMBL1908021 0.069 0.04 CHEMBL3544888 0.072 0.034 CHEMBL3638281 0.073 0.031 CHEMBL3544523 0.067 0.047 CHEMBL3548560 0.082 0.018 CHEMBL3544524 | ||
| 0.091 | 0.026 | 0.091 | Neutrophil collagenase inhibitor | 0.08 0.032 CHEMBL1908020 0.088 0.027 CHEMBL1908021 0.088 0.027 CHEMBL3544888 0.086 0.028 CHEMBL3548560 0.057 0.055 CHEMBL3544524 0.07 0.039 CHEMBL3544501 | ||
| 0.083 | 0.021 | 0.083 | Phosphodiesterase 1B inhibitor | 0.071 0.03 CHEMBL1908020 0.07 0.03 CHEMBL1908021 0.072 0.029 CHEMBL3544888 0.068 0.033 CHEMBL3548560 0.076 0.025 CHEMBL3544501 | ||
| 0.091 | 0.031 | 0.091 | Matrix metalloproteinase inhibitor | 0.083 0.035 CHEMBL1908020 0.091 0.031 CHEMBL1908021 0.091 0.031 CHEMBL3544888 0.085 0.034 CHEMBL3548560 0.078 0.038 CHEMBL3544501 | ||
| 0.132 | 0.072 | 0.132 | Sodium channel blocker | |||
| 0.096 | 0.038 | 0.113 | Alpha 1a adrenoreceptor antagonist | 0.071 0.05 CHEMBL1908020 0.067 0.052 CHEMBL1908021 0.063 0.055 CHEMBL3544888 0.073 0.049 CHEMBL3548560 0.113 0.031 CHEMBL3544501 | CHEMBL3544501 | |
| 0.169 | 0.11 | 0.271 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.215 0.061 CHEMBL1908020 0.164 0.118 CHEMBL3544522 0.213 0.062 CHEMBL1908021 0.212 0.063 CHEMBL3544888 0.169 0.11 CHEMBL3638281 0.154 0.14 CHEMBL3544523 0.155 0.137 CHEMBL3544887 0.216 0.06 CHEMBL3548560 0.271 0.034 CHEMBL3544524 0.222 0.057 CHEMBL3544501 | CHEMBL3544524 | |
| 0.186 | 0.128 | 0.257 | DNA damaging | 0.21 0.108 CHEMBL1908020 0.185 0.129 CHEMBL3544522 0.194 0.12 CHEMBL1908021 0.195 0.12 CHEMBL3544888 0.186 0.127 CHEMBL3638281 0.164 0.152 CHEMBL3544523 0.22 0.101 CHEMBL3544887 0.224 0.097 CHEMBL3548560 0.165 0.151 CHEMBL3544524 0.257 0.077 CHEMBL3544501 | CHEMBL3544501 | |
| 0.086 | 0.029 | 0.086 | Acetylcholine M5 receptor agonist | |||
| 0.153 | 0.097 | 0.154 | 3C-like protease (Human coronavirus) inhibitor | 0.154 0.095 CHEMBL3544524 | CHEMBL3544524 | |
| 0.081 | 0.026 | 0.081 | Cannabinoid CB1 receptor antagonist | |||
| 0.139 | 0.083 | 0.201 | Adenylate cyclase stimulant | 0.158 0.05 CHEMBL1908020 0.156 0.053 CHEMBL1908021 0.16 0.048 CHEMBL3544888 0.162 0.044 CHEMBL3638281 0.166 0.039 CHEMBL3544523 0.166 0.039 CHEMBL3548560 0.201 0.013 CHEMBL3544524 0.15 0.063 CHEMBL3544501 | CHEMBL3544524 | |
| 0.079 | 0.025 | 0.784 | Alcohol oxidase inhibitor | 0.122 0.014 CHEMBL1908020 0.151 0.01 CHEMBL1908021 0.165 0.009 CHEMBL3544888 0.083 0.023 CHEMBL3638281 0.609 0.003 CHEMBL3544523 0.084 0.023 CHEMBL3548560 0.784 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.107 | 0.054 | 0.142 | Anabolic | 0.128 0.033 CHEMBL1908020 0.122 0.038 CHEMBL1908021 0.128 0.033 CHEMBL3544888 0.142 0.022 CHEMBL3638281 0.096 0.068 CHEMBL3544523 0.118 0.041 CHEMBL3548560 0.135 0.027 CHEMBL3544524 | CHEMBL3638281 | |
| 0.077 | 0.024 | 0.096 | Carbonic anhydrase VB inhibitor | 0.086 0.02 CHEMBL1908020 0.095 0.017 CHEMBL1908021 0.096 0.017 CHEMBL3544888 0.089 0.019 CHEMBL3548560 0.084 0.021 CHEMBL3544524 0.061 0.034 CHEMBL3544501 | CHEMBL3544888 | |
| 0.057 | 0.005 | 0.062 | Protein kinase (CK2) beta inhibitor | 0.061 0.005 CHEMBL1908020 0.06 0.005 CHEMBL1908021 0.062 0.005 CHEMBL3544888 0.031 0.029 CHEMBL3638281 0.062 0.005 CHEMBL3548560 0.033 0.023 CHEMBL3544501 | CHEMBL3548560 | |
| 0.078 | 0.027 | 0.541 | Glutamate (mGluR6) antagonist | 0.063 0.057 CHEMBL1908020 0.062 0.061 CHEMBL3544522 0.068 0.045 CHEMBL1908021 0.069 0.043 CHEMBL3544888 0.07 0.04 CHEMBL3638281 0.163 0.003 CHEMBL3544523 0.063 0.057 CHEMBL3548560 0.541 0.001 CHEMBL3544524 | CHEMBL3544524 | |
| 0.063 | 0.013 | 0.064 | Thymidine kinase inhibitor | 0.049 0.02 CHEMBL1908020 0.052 0.018 CHEMBL1908021 0.052 0.018 CHEMBL3544888 0.064 0.012 CHEMBL3638281 0.048 0.02 CHEMBL3548560 0.039 0.032 CHEMBL3544524 | CHEMBL3638281 | |
| 0.084 | 0.035 | 0.417 | Phenylalanine 4-hydroxylase inhibitor | 0.117 0.019 CHEMBL1908020 0.135 0.014 CHEMBL1908021 0.133 0.015 CHEMBL3544888 0.063 0.054 CHEMBL3638281 0.18 0.008 CHEMBL3544523 0.132 0.015 CHEMBL3548560 0.417 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.076 | 0.028 | 0.1 | NMDA 2C receptor antagonist | 0.095 0.018 CHEMBL1908020 0.095 0.018 CHEMBL1908021 0.093 0.018 CHEMBL3544888 0.073 0.03 CHEMBL3548560 0.1 0.016 CHEMBL3544524 | CHEMBL3544524 | |
| 0.056 | 0.009 | 0.1 | Kainate receptor agonist | 0.047 0.017 CHEMBL1908020 0.051 0.013 CHEMBL1908021 0.053 0.011 CHEMBL3544888 0.05 0.014 CHEMBL3638281 0.063 0.006 CHEMBL3544523 0.047 0.017 CHEMBL3548560 0.1 0.003 CHEMBL3544524 0.038 0.036 CHEMBL3544501 | CHEMBL3544524 | |
| 0.088 | 0.042 | 0.101 | CC chemokine 5 receptor agonist | 0.101 0.021 CHEMBL1908020 0.097 0.026 CHEMBL1908021 0.095 0.028 CHEMBL3544888 0.089 0.039 CHEMBL3548560 0.08 0.066 CHEMBL3544524 | CHEMBL1908020 | |
| 0.148 | 0.104 | 0.277 | ATPase inhibitor | 0.148 0.104 CHEMBL1908020 0.21 0.03 CHEMBL3544522 0.154 0.094 CHEMBL1908021 0.154 0.095 CHEMBL3544888 0.202 0.035 CHEMBL3638281 0.168 0.074 CHEMBL3544523 0.277 0.009 CHEMBL3544887 0.154 0.095 CHEMBL3548560 0.166 0.077 CHEMBL3544524 0.157 0.089 CHEMBL3544501 | CHEMBL3544887 | |
| 0.107 | 0.063 | 0.24 | DOPA decarboxylase inhibitor | 0.153 0.02 CHEMBL1908020 0.145 0.024 CHEMBL1908021 0.153 0.02 CHEMBL3544888 0.154 0.019 CHEMBL3544523 0.156 0.018 CHEMBL3548560 0.24 0.004 CHEMBL3544524 0.122 0.042 CHEMBL3544501 | CHEMBL3544524 | |
| 0.048 | 0.004 | 0.048 | Nicotinic acid receptor 2 antagonist | 0.04 0.005 CHEMBL1908020 0.041 0.005 CHEMBL1908021 0.043 0.005 CHEMBL3544888 0.024 0.023 CHEMBL3638281 0.036 0.007 CHEMBL3548560 0.027 0.017 CHEMBL3544524 | ||
| 0.049 | 0.005 | 0.049 | Nociceptin (N/OFQ) receptor agonist | 0.02 0.015 CHEMBL1908020 0.024 0.012 CHEMBL1908021 0.024 0.012 CHEMBL3544888 | ||
| 0.079 | 0.037 | 0.095 | Carbonic anhydrase VA inhibitor | 0.089 0.031 CHEMBL1908020 0.095 0.027 CHEMBL1908021 0.095 0.027 CHEMBL3544888 0.09 0.03 CHEMBL3548560 0.089 0.03 CHEMBL3544524 0.081 0.036 CHEMBL3544501 | CHEMBL3544888 | |
| 0.043 | 0.006 | 0.043 | Thymidine phosphorylase inhibitor | 0.031 0.01 CHEMBL1908020 0.034 0.009 CHEMBL1908021 0.037 0.008 CHEMBL3544888 0.035 0.008 CHEMBL3638281 0.033 0.009 CHEMBL3548560 | ||
| 0.081 | 0.044 | 0.366 | Glutamate decarboxylase inhibitor | 0.101 0.029 CHEMBL1908020 0.113 0.023 CHEMBL1908021 0.118 0.021 CHEMBL3544888 0.287 0.004 CHEMBL3544523 0.104 0.027 CHEMBL3548560 0.366 0.003 CHEMBL3544524 0.064 0.063 CHEMBL3544501 | CHEMBL3544524 | |
| 0.083 | 0.045 | 0.501 | Porphobilinogen synthase inhibitor | 0.088 0.042 CHEMBL1908020 0.107 0.033 CHEMBL1908021 0.117 0.029 CHEMBL3544888 0.178 0.015 CHEMBL3544523 0.088 0.042 CHEMBL3548560 0.501 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.078 | 0.041 | 0.078 | Cannabinoid receptor antagonist | |||
| 0.137 | 0.101 | 0.169 | CF transmembrane conductance regulator agonist | 0.15 0.077 CHEMBL1908020 0.164 0.055 CHEMBL1908021 0.166 0.052 CHEMBL3544888 0.128 0.122 CHEMBL3548560 0.169 0.048 CHEMBL3544524 | CHEMBL3544524 | |
| 0.178 | 0.141 | 0.368 | Interleukin agonist | 0.321 0.038 CHEMBL3544522 0.164 0.154 CHEMBL1908021 0.166 0.152 CHEMBL3544888 0.239 0.087 CHEMBL3544523 0.301 0.047 CHEMBL3544887 0.18 0.139 CHEMBL3548560 0.368 0.024 CHEMBL3544524 | CHEMBL3544524 | |
| 0.05 | 0.014 | 0.073 | Nicotinic acid receptor agonist | 0.069 0.009 CHEMBL1908020 0.071 0.008 CHEMBL1908021 0.073 0.008 CHEMBL3544888 0.045 0.017 CHEMBL3548560 | CHEMBL3544888 | |
| 0.107 | 0.072 | 0.109 | Acetylcholine release stimulant | 0.109 0.067 CHEMBL3544524 | CHEMBL3544524 | |
| 0.089 | 0.054 | 0.132 | Granulocyte macrophage colony stimulating factor agonist | 0.09 0.051 CHEMBL1908020 0.087 0.058 CHEMBL1908021 0.086 0.06 CHEMBL3544888 0.092 0.048 CHEMBL3544523 0.104 0.03 CHEMBL3548560 0.132 0.01 CHEMBL3544524 0.124 0.013 CHEMBL3544501 | CHEMBL3544524 | |
| 0.059 | 0.025 | 0.059 | Bombesin 2 receptor antagonist | 0.052 0.031 CHEMBL1908020 0.055 0.027 CHEMBL1908021 0.056 0.027 CHEMBL3544888 0.047 0.039 CHEMBL3548560 0.055 0.028 CHEMBL3544524 | ||
| 0.063 | 0.03 | 0.085 | Ryanodine receptor antagonist | 0.072 0.015 CHEMBL1908020 0.068 0.021 CHEMBL1908021 0.069 0.018 CHEMBL3544888 0.056 0.052 CHEMBL3638281 0.072 0.015 CHEMBL3548560 0.063 0.029 CHEMBL3544524 0.085 0.006 CHEMBL3544501 | CHEMBL3544501 | |
| 0.083 | 0.051 | 0.12 | Alpha 1 adrenoreceptor antagonist | 0.068 0.061 CHEMBL3548560 0.12 0.037 CHEMBL3544501 | CHEMBL3544501 | |
| 0.051 | 0.02 | 0.051 | Nicotinic acid receptor 1 agonist | 0.038 0.031 CHEMBL1908021 0.038 0.031 CHEMBL3544888 | ||
| 0.078 | 0.047 | 0.323 | Glutamate dehydrogenase inhibitor | 0.072 0.054 CHEMBL1908021 0.077 0.048 CHEMBL3544888 0.077 0.048 CHEMBL3638281 0.323 0.005 CHEMBL3544523 0.309 0.005 CHEMBL3544524 | CHEMBL3544523 | |
| 0.072 | 0.041 | 0.094 | Carbonic anhydrase V inhibitor | 0.084 0.033 CHEMBL1908020 0.093 0.029 CHEMBL1908021 0.094 0.029 CHEMBL3544888 0.087 0.032 CHEMBL3548560 0.088 0.032 CHEMBL3544524 0.075 0.039 CHEMBL3544501 | CHEMBL3544888 | |
| 0.058 | 0.028 | 0.295 | Aconitate hydratase inhibitor | 0.25 0.003 CHEMBL3544523 0.295 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.06 | 0.031 | 0.214 | Ornithine carbamoyltransferase inhibitor | 0.049 0.041 CHEMBL3544888 0.056 0.034 CHEMBL3638281 0.214 0.006 CHEMBL3544523 0.194 0.007 CHEMBL3544524 | CHEMBL3544523 | |
| 0.075 | 0.046 | 0.148 | Glycine receptor agonist | 0.066 0.063 CHEMBL1908020 0.079 0.04 CHEMBL3544522 0.073 0.049 CHEMBL1908021 0.074 0.047 CHEMBL3544888 0.074 0.048 CHEMBL3638281 0.073 0.049 CHEMBL3544523 0.066 0.063 CHEMBL3548560 0.148 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.127 | 0.099 | 0.127 | Acetylcholine M1 receptor antagonist | 0.117 0.113 CHEMBL1908020 0.125 0.101 CHEMBL1908021 0.124 0.103 CHEMBL3544888 0.116 0.114 CHEMBL3548560 | ||
| 0.04 | 0.012 | 0.04 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.024 0.023 CHEMBL1908021 0.027 0.02 CHEMBL3544888 0.033 0.015 CHEMBL3638281 0.03 0.018 CHEMBL3544524 | ||
| 0.06 | 0.033 | 0.06 | Matrix metalloproteinase (membrane-type) inhibitor | 0.053 0.042 CHEMBL1908020 0.056 0.037 CHEMBL1908021 0.056 0.037 CHEMBL3544888 0.054 0.039 CHEMBL3548560 0.052 0.043 CHEMBL3544524 0.05 0.046 CHEMBL3544501 | ||
| 0.049 | 0.022 | 0.126 | Glutamate (mGluR4) antagonist | 0.064 0.012 CHEMBL3544523 0.126 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.051 | 0.026 | 0.057 | Thymidylate synthase inhibitor | 0.046 0.033 CHEMBL1908021 0.049 0.029 CHEMBL3544888 0.045 0.034 CHEMBL3544523 0.057 0.02 CHEMBL3544524 | CHEMBL3544524 | |
| 0.059 | 0.034 | 0.065 | Pregnane X receptor antagonist | 0.053 0.05 CHEMBL1908020 0.056 0.042 CHEMBL1908021 0.058 0.036 CHEMBL3544888 0.053 0.05 CHEMBL3548560 0.065 0.021 CHEMBL3544524 0.053 0.052 CHEMBL3544501 | CHEMBL3544524 | |
| 0.033 | 0.008 | 0.033 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.027 0.016 CHEMBL1908020 0.028 0.014 CHEMBL1908021 0.028 0.015 CHEMBL3544888 0.033 0.008 CHEMBL3638281 0.027 0.016 CHEMBL3548560 | ||
| 0.083 | 0.059 | 0.139 | D-Ala-D-Ala ligase inhibitor | 0.107 0.022 CHEMBL1908020 0.105 0.024 CHEMBL1908021 0.104 0.025 CHEMBL3544888 0.107 0.022 CHEMBL3544523 0.109 0.02 CHEMBL3548560 0.139 0.007 CHEMBL3544524 0.097 0.033 CHEMBL3544501 | CHEMBL3544524 | |
| 0.093 | 0.07 | 0.253 | Aminopeptidase B inhibitor | 0.092 0.071 CHEMBL1908021 0.093 0.07 CHEMBL3544888 0.247 0.013 CHEMBL3544523 0.253 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.031 | 0.008 | 0.031 | Acid ceramidase inhibitor | |||
| 0.028 | 0.005 | 0.028 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.022 0.011 CHEMBL1908020 0.023 0.01 CHEMBL1908021 0.022 0.011 CHEMBL3544888 0.027 0.005 CHEMBL3638281 0.022 0.011 CHEMBL3548560 | ||
| 0.033 | 0.01 | 0.033 | DNA polymerase III inhibitor | 0.027 0.023 CHEMBL3544888 | ||
| 0.041 | 0.018 | 0.151 | Fumarate hydratase inhibitor | 0.032 0.026 CHEMBL1908021 0.035 0.023 CHEMBL3544888 0.042 0.017 CHEMBL3638281 0.059 0.011 CHEMBL3544523 0.151 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.105 | 0.083 | 0.227 | Alkylator | 0.122 0.066 CHEMBL1908020 0.154 0.045 CHEMBL3544522 0.116 0.072 CHEMBL1908021 0.121 0.067 CHEMBL3544888 0.14 0.052 CHEMBL3638281 0.121 0.068 CHEMBL3544523 0.227 0.02 CHEMBL3544887 0.117 0.071 CHEMBL3548560 0.112 0.075 CHEMBL3544524 0.123 0.066 CHEMBL3544501 | CHEMBL3544887 | |
| 0.128 | 0.106 | 0.197 | Sphingosine 1-phosphate receptor 5 antagonist | 0.122 0.119 CHEMBL1908021 0.124 0.113 CHEMBL3544888 0.157 0.051 CHEMBL3544523 0.126 0.11 CHEMBL3548560 0.197 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.041 | 0.02 | 0.05 | Nicotinic acid receptor 2 agonist | 0.046 0.016 CHEMBL1908020 0.048 0.015 CHEMBL1908021 0.05 0.014 CHEMBL3544888 0.037 0.024 CHEMBL3548560 | CHEMBL3544888 | |
| 0.071 | 0.05 | 0.39 | Histidine decarboxylase inhibitor | 0.13 0.023 CHEMBL1908020 0.129 0.023 CHEMBL1908021 0.142 0.021 CHEMBL3544888 0.355 0.005 CHEMBL3544523 0.126 0.024 CHEMBL3548560 0.39 0.004 CHEMBL3544524 0.091 0.036 CHEMBL3544501 | CHEMBL3544524 | |
| 0.196 | 0.176 | 0.224 | Thioredoxin glutathione reductase inhibitor | 0.199 0.174 CHEMBL1908021 0.196 0.176 CHEMBL3544888 0.212 0.162 CHEMBL3548560 0.224 0.153 CHEMBL3544501 | CHEMBL3544501 | |
| 0.037 | 0.019 | 0.037 | Purinergic P2Y2 antagonist | 0.031 0.028 CHEMBL1908020 0.033 0.024 CHEMBL1908021 0.033 0.024 CHEMBL3544888 | ||
| 0.053 | 0.035 | 0.082 | NMDA 2A receptor antagonist | 0.081 0.019 CHEMBL1908020 0.082 0.019 CHEMBL1908021 0.08 0.02 CHEMBL3544888 0.057 0.031 CHEMBL3548560 0.077 0.021 CHEMBL3544524 | CHEMBL1908021 | |
| 0.087 | 0.07 | 0.151 | Prolactin inhibitor | 0.117 0.041 CHEMBL1908020 0.116 0.041 CHEMBL1908021 0.113 0.043 CHEMBL3544888 0.102 0.053 CHEMBL3544523 0.111 0.045 CHEMBL3548560 0.151 0.022 CHEMBL3544524 | CHEMBL3544524 | |
| 0.045 | 0.028 | 0.045 | Macrophage elastase inhibitor | |||
| 0.068 | 0.051 | 0.116 | HIV-1 reverse transcriptase inhibitor | 0.116 0.024 CHEMBL3544522 0.069 0.05 CHEMBL3548560 | CHEMBL3544522 | |
| 0.022 | 0.006 | 0.024 | Thyroid hormone alpha agonist | 0.023 0.005 CHEMBL1908020 0.023 0.005 CHEMBL1908021 0.024 0.005 CHEMBL3544888 0.015 0.014 CHEMBL3638281 0.024 0.005 CHEMBL3548560 0.019 0.008 CHEMBL3544501 | CHEMBL3548560 | |
| 0.152 | 0.136 | 0.153 | Histone acetyltransferase inhibitor | 0.152 0.137 CHEMBL3548560 0.153 0.135 CHEMBL3544501 | CHEMBL3544501 | |
| 0.017 | 0.002 | 0.017 | DNA topoisomerase III inhibitor | 0.01 0.004 CHEMBL1908020 0.012 0.003 CHEMBL1908021 0.012 0.003 CHEMBL3544888 0.009 0.004 CHEMBL3638281 0.01 0.004 CHEMBL3548560 | ||
| 0.058 | 0.043 | 0.088 | Androgen agonist | 0.075 0.027 CHEMBL1908020 0.07 0.031 CHEMBL1908021 0.075 0.027 CHEMBL3544888 0.088 0.02 CHEMBL3638281 0.064 0.036 CHEMBL3548560 | CHEMBL3638281 | |
| 0.053 | 0.039 | 0.053 | Cathepsin D inhibitor | |||
| 0.027 | 0.013 | 0.096 | Glutamate (mGluR1) agonist | 0.023 0.021 CHEMBL1908021 0.023 0.021 CHEMBL3544888 0.034 0.007 CHEMBL3544523 0.096 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.037 | 0.023 | 0.037 | Nociceptin (N/OFQ) receptor antagonist | |||
| 0.025 | 0.012 | 0.134 | Glutamate (mGluR1a) agonist | 0.049 0.005 CHEMBL3544523 0.134 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.099 | 0.085 | 0.143 | Adenylate cyclase inhibitor | 0.125 0.063 CHEMBL1908020 0.124 0.064 CHEMBL1908021 0.125 0.064 CHEMBL3544888 0.125 0.063 CHEMBL3638281 0.143 0.05 CHEMBL3548560 0.133 0.057 CHEMBL3544524 | CHEMBL3548560 | |
| 0.235 | 0.222 | 0.428 | Calcium channel L-type activator | 0.388 0.089 CHEMBL1908020 0.41 0.074 CHEMBL1908021 0.395 0.085 CHEMBL3544888 0.292 0.164 CHEMBL3544523 0.301 0.157 CHEMBL3548560 0.428 0.064 CHEMBL3544524 0.292 0.164 CHEMBL3544501 | CHEMBL3544524 | |
| 0.044 | 0.032 | 0.046 | Dihydroorotase inhibitor | 0.042 0.035 CHEMBL3544523 0.046 0.029 CHEMBL3548560 | CHEMBL3548560 | |
| 0.043 | 0.032 | 0.4 | Glutamate (mGluR group III) antagonist | 0.125 0.004 CHEMBL3544523 0.4 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.039 | 0.029 | 0.079 | Dopamine D5 agonist | 0.076 0.007 CHEMBL1908020 0.068 0.009 CHEMBL1908021 0.067 0.009 CHEMBL3544888 0.036 0.034 CHEMBL3544523 0.079 0.006 CHEMBL3548560 0.074 0.007 CHEMBL3544524 0.049 0.018 CHEMBL3544501 | CHEMBL3548560 | |
| 0.059 | 0.049 | 0.059 | Corticotropin releasing factor 2 receptor antagonist | |||
| 0.197 | 0.187 | 0.197 | Beta lactamase inhibitor | |||
| 0.08 | 0.072 | 0.118 | Alpha adrenoreceptor antagonist | 0.076 0.075 CHEMBL3548560 0.118 0.048 CHEMBL3544501 | CHEMBL3544501 | |
| 0.088 | 0.08 | 0.134 | Phosphodiesterase 6D inhibitor | 0.092 0.071 CHEMBL1908020 0.088 0.083 CHEMBL3544522 0.093 0.067 CHEMBL1908021 0.093 0.068 CHEMBL3544888 0.134 0.015 CHEMBL3544887 0.096 0.06 CHEMBL3548560 | CHEMBL3544887 | |
| 0.15 | 0.142 | 0.286 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.175 0.117 CHEMBL1908020 0.173 0.119 CHEMBL1908021 0.166 0.125 CHEMBL3544888 0.221 0.089 CHEMBL3548560 0.286 0.068 CHEMBL3544501 | CHEMBL3544501 | |
| 0.043 | 0.035 | 0.157 | Phosphorylase inhibitor | 0.041 0.036 CHEMBL1908020 0.072 0.019 CHEMBL3544522 0.048 0.031 CHEMBL1908021 0.048 0.032 CHEMBL3544888 0.157 0.007 CHEMBL3544887 0.039 0.038 CHEMBL3548560 | CHEMBL3544887 | |
| 0.065 | 0.057 | 0.078 | Alpha 1b adrenoreceptor antagonist | 0.078 0.047 CHEMBL3544501 | CHEMBL3544501 | |
| 0.014 | 0.007 | 0.014 | DNA polymerase III polC-type inhibitor | |||
| 0.125 | 0.119 | 0.216 | Arachidonic acid antagonist | 0.153 0.085 CHEMBL1908020 0.141 0.099 CHEMBL1908021 0.148 0.091 CHEMBL3544888 0.137 0.103 CHEMBL3638281 0.17 0.065 CHEMBL3544523 0.165 0.071 CHEMBL3548560 0.216 0.019 CHEMBL3544524 0.135 0.106 CHEMBL3544501 | CHEMBL3544524 | |
| 0.069 | 0.063 | 0.099 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.073 0.052 CHEMBL3544523 0.099 0.014 CHEMBL3544524 | CHEMBL3544524 | |
| 0.039 | 0.035 | 0.039 | Angiotensin AT1 receptor antagonist | 0.039 0.034 CHEMBL3544524 | ||
| 0.044 | 0.04 | 0.097 | Glucose-6-phosphate isomerase inhibitor | 0.069 0.013 CHEMBL3544522 0.043 0.042 CHEMBL3544888 0.056 0.022 CHEMBL3638281 0.066 0.015 CHEMBL3544523 0.06 0.019 CHEMBL3544887 0.097 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.051 | 0.048 | 0.053 | Alpha 1d adrenoreceptor antagonist | 0.053 0.046 CHEMBL3544501 | CHEMBL3544501 | |
| 0.042 | 0.038 | 0.047 | Antimetabolite | 0.042 0.039 CHEMBL3638281 0.041 0.04 CHEMBL3544523 0.047 0.034 CHEMBL3544524 | CHEMBL3544524 | |
| 0.012 | 0.009 | 0.014 | Egl nine homolog 3 inhibitor | 0.013 0.008 CHEMBL1908020 0.014 0.006 CHEMBL1908021 0.014 0.006 CHEMBL3544888 0.011 0.009 CHEMBL3548560 0.012 0.009 CHEMBL3544524 | CHEMBL3544888 | |
| 0.038 | 0.035 | 0.038 | Plasmepsin II inhibitor | |||
| 0.032 | 0.031 | 0.032 | Growth factor receptor-bound protein 2 antagonist | 0.032 0.031 CHEMBL3544888 | ||
| 0.047 | 0.046 | 0.187 | Acyl-CoA dehydrogenase inhibitor | 0.098 0.017 CHEMBL3544523 0.187 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.024 | 0.023 | 0.029 | Integrin alpha2beta1 antagonist | 0.025 0.02 CHEMBL3544523 0.029 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.036 | 0.035 | 0.036 | Aggrecanase 1 inhibitor | |||
| 0.054 | 0.053 | 0.054 | TRPA1 antagonist | |||
| 0.129 | 0.128 | 0.157 | Heat shock protein 70 antagonist | 0.137 0.089 CHEMBL1908020 0.138 0.081 CHEMBL1908021 0.138 0.082 CHEMBL3544888 0.142 0.067 CHEMBL3544887 0.139 0.079 CHEMBL3548560 0.157 0.031 CHEMBL3544524 0.138 0.081 CHEMBL3544501 | CHEMBL3544524 | |
| 0.088 | 0.088 | 0.139 | Glutamate (mGluR7) agonist | 0.098 0.065 CHEMBL3544523 0.139 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.01 | 0.013 | Purinergic P2Y2 agonist | 0.012 0.005 CHEMBL3544522 0.01 0.009 CHEMBL3638281 0.013 0.005 CHEMBL3544887 | CHEMBL3544887 | |
| 0.033 | 0.035 | 0.041 | Integrin alpha2 antagonist | 0.036 0.028 CHEMBL3544523 0.041 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.08 | 0.083 | 0.097 | Protein kinase (CK2) inhibitor | 0.086 0.076 CHEMBL1908020 0.087 0.075 CHEMBL1908021 0.09 0.073 CHEMBL3544888 0.097 0.066 CHEMBL3548560 | CHEMBL3548560 | |
| 0.038 | 0.041 | 0.059 | GABA B receptor antagonist | 0.059 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.025 | 0.038 | Thyroid hormone agonist | 0.038 0.007 CHEMBL1908020 0.035 0.009 CHEMBL1908021 0.038 0.007 CHEMBL3544888 0.036 0.008 CHEMBL3548560 0.027 0.016 CHEMBL3544524 0.024 0.023 CHEMBL3544501 | CHEMBL3544888 | |
| 0.038 | 0.042 | 0.061 | AICAR transformylase inhibitor | 0.061 0.014 CHEMBL3544524 | CHEMBL3544524 | |
| 0.089 | 0.095 | 0.192 | Mucolytic | 0.105 0.07 CHEMBL1908020 0.093 0.088 CHEMBL3544522 0.108 0.067 CHEMBL1908021 0.11 0.064 CHEMBL3544888 0.133 0.043 CHEMBL3638281 0.161 0.027 CHEMBL3544523 0.114 0.06 CHEMBL3544887 0.115 0.059 CHEMBL3548560 0.192 0.015 CHEMBL3544524 0.141 0.038 CHEMBL3544501 | CHEMBL3544524 | |
| 0.039 | 0.045 | 0.041 | Histamine H1 receptor agonist | 0.041 0.038 CHEMBL3544524 | CHEMBL3544524 | |
| 0.076 | 0.083 | 0.109 | Estrogen-related receptor beta agonist | 0.098 0.028 CHEMBL1908020 0.098 0.027 CHEMBL1908021 0.098 0.028 CHEMBL3544888 0.083 0.058 CHEMBL3544523 0.088 0.046 CHEMBL3548560 0.109 0.016 CHEMBL3544524 0.083 0.056 CHEMBL3544501 | CHEMBL3544524 | |
| 0.061 | 0.07 | 0.088 | Exportin-1 inhibitor | 0.063 0.061 CHEMBL3544523 0.088 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.06 | 0.069 | 0.196 | Aminopeptidase I inhibitor | 0.135 0.015 CHEMBL3544523 0.196 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.032 | 0.042 | 0.12 | Glutamate (mGluR8) agonist | 0.064 0.006 CHEMBL3544523 0.12 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.113 | 0.123 | 0.304 | Insulin secretagoues | 0.126 0.102 CHEMBL1908020 0.183 0.046 CHEMBL3544522 0.134 0.092 CHEMBL1908021 0.134 0.091 CHEMBL3544888 0.12 0.111 CHEMBL3638281 0.304 0.012 CHEMBL3544887 0.136 0.09 CHEMBL3548560 | CHEMBL3544887 | |
| 0.081 | 0.091 | 0.211 | Xanthine oxidase inhibitor | 0.145 0.036 CHEMBL1908020 0.088 0.074 CHEMBL3544522 0.135 0.04 CHEMBL1908021 0.141 0.038 CHEMBL3544888 0.211 0.017 CHEMBL3544887 0.15 0.034 CHEMBL3548560 0.143 0.037 CHEMBL3544501 | CHEMBL3544887 | |
| 0.038 | 0.049 | 0.048 | Adenylate cyclase 1 inhibitor | 0.048 0.029 CHEMBL3544524 | CHEMBL3544524 | |
| 0.092 | 0.103 | 0.295 | M18 aspartyl aminopeptidase inhibitor | 0.216 0.029 CHEMBL1908020 0.203 0.033 CHEMBL1908021 0.204 0.032 CHEMBL3544888 0.295 0.013 CHEMBL3548560 0.26 0.019 CHEMBL3544501 | CHEMBL3548560 | |
| 0.127 | 0.139 | 0.24 | Psychostimulant | 0.211 0.074 CHEMBL3544523 0.24 0.062 CHEMBL3544524 | CHEMBL3544524 | |
| 0.067 | 0.079 | 0.147 | Carbonic anhydrase VI inhibitor | 0.099 0.04 CHEMBL1908020 0.099 0.039 CHEMBL1908021 0.1 0.039 CHEMBL3544888 0.102 0.038 CHEMBL3548560 0.147 0.021 CHEMBL3544524 0.102 0.038 CHEMBL3544501 | CHEMBL3544524 | |
| 0.024 | 0.038 | 0.028 | Epoxide hydrolase 1 inhibitor | 0.028 0.026 CHEMBL3544524 | CHEMBL3544524 | |
| 0.008 | 0.023 | 0.014 | Carbonic anhydrase XI inhibitor | 0.014 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.031 | 0.047 | 0.066 | Membrane dipeptidase inhibitor | 0.064 0.009 CHEMBL3544523 0.066 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.03 | 0.046 | 0.045 | Oxytocin agonist | 0.037 0.035 CHEMBL1908020 0.042 0.03 CHEMBL1908021 0.045 0.028 CHEMBL3544888 0.041 0.031 CHEMBL3544524 | CHEMBL3544888 | |
| 0.088 | 0.105 | 0.113 | Factor V inhibitor | 0.106 0.057 CHEMBL3544523 0.113 0.046 CHEMBL3544524 | CHEMBL3544524 | |
| 0.109 | 0.126 | 0.162 | Sphingosine 1-phosphate receptor 2 antagonist | 0.143 0.05 CHEMBL3544523 0.162 0.027 CHEMBL3544524 | CHEMBL3544524 | |
| 0.022 | 0.039 | 0.034 | Purinergic P2Y15 antagonist | 0.034 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.021 | 0.008 | Thyroid hormone beta agonist | 0.008 0.007 CHEMBL1908020 0.008 0.007 CHEMBL3544888 0.008 0.006 CHEMBL3548560 | CHEMBL3548560 | |
| 0.097 | 0.114 | 0.176 | Cathepsin H inhibitor | 0.131 0.062 CHEMBL3544523 0.176 0.031 CHEMBL3544524 | CHEMBL3544524 | |
| 0.034 | 0.052 | 0.049 | Nerve growth factor antagonist | 0.049 0.02 CHEMBL3544524 | CHEMBL3544524 | |
| 0.057 | 0.074 | 0.103 | Cathepsin G inhibitor | 0.103 0.032 CHEMBL3544524 | CHEMBL3544524 | |
| 0.067 | 0.086 | 0.11 | NMDA receptor antagonist | 0.108 0.042 CHEMBL1908020 0.11 0.041 CHEMBL1908021 0.107 0.042 CHEMBL3544888 0.082 0.063 CHEMBL3548560 0.092 0.052 CHEMBL3544524 | CHEMBL1908021 | |
| 0.094 | 0.113 | 0.126 | Interleukin 8 antagonist | 0.105 0.085 CHEMBL1908020 0.103 0.089 CHEMBL1908021 0.101 0.093 CHEMBL3544888 0.108 0.08 CHEMBL3548560 0.126 0.054 CHEMBL3544524 | CHEMBL3544524 | |
| 0.052 | 0.071 | 0.078 | Lipase inhibitor | 0.075 0.049 CHEMBL1908020 0.077 0.046 CHEMBL1908021 0.077 0.046 CHEMBL3544888 0.078 0.045 CHEMBL3548560 0.063 0.061 CHEMBL3544501 | CHEMBL3548560 | |
| 0.045 | 0.065 | 0.057 | Fatty acid synthase inhibitor | 0.053 0.045 CHEMBL1908020 0.054 0.044 CHEMBL1908021 0.056 0.04 CHEMBL3544888 0.057 0.04 CHEMBL3548560 | CHEMBL3548560 | |
| 0.027 | 0.048 | 0.372 | Glutamate (mGluR3) antagonist | 0.112 0.004 CHEMBL3544523 0.372 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.065 | 0.087 | 0.157 | GABA B receptor agonist | 0.074 0.057 CHEMBL1908020 0.079 0.045 CHEMBL1908021 0.079 0.043 CHEMBL3544888 0.096 0.02 CHEMBL3544523 0.075 0.053 CHEMBL3548560 0.157 0.004 CHEMBL3544524 0.074 0.056 CHEMBL3544501 | CHEMBL3544524 | |
| 0.032 | 0.053 | 0.043 | Histamine H2 receptor agonist | 0.043 0.03 CHEMBL3544523 | CHEMBL3544523 | |
| 0.059 | 0.081 | 0.095 | Analgesic, opioid | 0.095 0.034 CHEMBL1908020 0.093 0.035 CHEMBL1908021 0.094 0.035 CHEMBL3544888 0.077 0.052 CHEMBL3638281 0.071 0.059 CHEMBL3548560 | CHEMBL1908020 | |
| 0.021 | 0.044 | 0.072 | Kainate receptor 2 antagonist | 0.072 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.179 | 0.202 | 0.368 | Vasodilator, coronary | 0.356 0.052 CHEMBL3544522 0.368 0.047 CHEMBL3544887 0.199 0.183 CHEMBL3548560 0.275 0.109 CHEMBL3544524 0.258 0.127 CHEMBL3544501 | CHEMBL3544887 | |
| 0.014 | 0.038 | 0.021 | Methylmalonyl-CoA mutase inhibitor | 0.021 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.056 | 0.081 | 0.101 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.099 0.038 CHEMBL1908020 0.098 0.038 CHEMBL1908021 0.095 0.04 CHEMBL3544888 0.092 0.042 CHEMBL3548560 0.088 0.045 CHEMBL3544524 0.101 0.037 CHEMBL3544501 | CHEMBL3544501 | |
| 0.009 | 0.034 | 0.032 | Carbonic anhydrase X inhibitor | 0.015 0.014 CHEMBL3544523 0.032 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.034 | 0.032 | Carbonic anhydrase VIII inhibitor | 0.015 0.014 CHEMBL3544523 0.032 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.136 | 0.161 | 0.252 | Neurotrophic factor enhancer | 0.196 0.081 CHEMBL1908020 0.189 0.088 CHEMBL1908021 0.188 0.089 CHEMBL3544888 0.151 0.136 CHEMBL3544523 0.194 0.083 CHEMBL3544887 0.203 0.074 CHEMBL3548560 0.252 0.037 CHEMBL3544524 0.188 0.089 CHEMBL3544501 | CHEMBL3544524 | |
| 0.028 | 0.055 | 0.06 | Tryptophan 5 hydroxylase inhibitor | 0.041 0.013 CHEMBL3544523 0.06 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.034 | 0.06 | 0.039 | CF transmembrane conductance regulator antagonist | 0.039 0.03 CHEMBL1908021 0.039 0.031 CHEMBL3544888 | CHEMBL3544888 | |
| 0.019 | 0.046 | 0.029 | LFA antagonist | 0.029 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.003 | 0.03 | 0.008 | Integrin alpha5beta6 antagonist | 0.008 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.03 | 0.057 | 0.063 | AMPA 4 receptor antagonist | 0.063 0.009 CHEMBL3544524 | CHEMBL3544524 | |
| 0.109 | 0.137 | 0.249 | Hexokinase inhibitor | 0.13 0.104 CHEMBL1908020 0.156 0.072 CHEMBL3544522 0.133 0.1 CHEMBL1908021 0.131 0.103 CHEMBL3544888 0.124 0.112 CHEMBL3638281 0.249 0.017 CHEMBL3544887 0.168 0.059 CHEMBL3544524 | CHEMBL3544887 | |
| 0.04 | 0.069 | 0.097 | Alpha-mannosidase inhibitor | 0.075 0.014 CHEMBL3544522 0.048 0.047 CHEMBL3638281 0.064 0.022 CHEMBL3544523 0.084 0.01 CHEMBL3544887 0.097 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.017 | 0.047 | 0.034 | Lysophosphatidic acid receptor 1 agonist | 0.023 0.022 CHEMBL3544523 0.034 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.04 | 0.015 | Purinergic P2Y1 agonist | 0.015 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.044 | 0.024 | NMDA receptor glycine site antagonist | 0.024 0.017 CHEMBL3544523 | CHEMBL3544523 | |
| 0.046 | 0.077 | 0.109 | Purinergic P2X1 antagonist | 0.071 0.031 CHEMBL3544523 0.109 0.014 CHEMBL3544524 | CHEMBL3544524 | |
| 0.051 | 0.083 | 0.117 | Carbonic anhydrase XIII inhibitor | 0.085 0.046 CHEMBL1908020 0.084 0.047 CHEMBL3544522 0.081 0.049 CHEMBL1908021 0.086 0.046 CHEMBL3544888 0.083 0.048 CHEMBL3544887 0.088 0.044 CHEMBL3548560 0.117 0.031 CHEMBL3544524 0.11 0.034 CHEMBL3544501 | CHEMBL3544524 | |
| 0.015 | 0.047 | 0.027 | Isoleucine-tRNA ligase inhibitor | 0.027 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.028 | 0.06 | 0.042 | Carbonic anhydrase VII inhibitor | 0.042 0.038 CHEMBL1908020 0.041 0.039 CHEMBL1908021 0.042 0.038 CHEMBL3544888 0.042 0.037 CHEMBL3548560 0.041 0.039 CHEMBL3544501 | CHEMBL3548560 | |
| 0.049 | 0.082 | 0.079 | Protease 3C (Human rhinovirus) inhibitor | 0.079 0.028 CHEMBL3544524 | CHEMBL3544524 | |
| 0.03 | 0.063 | 0.045 | Glutamate (mGluR group I) agonist | 0.045 0.036 CHEMBL3544524 | CHEMBL3544524 | |
| 0.005 | 0.038 | 0.048 | Glutamate (mGluR6) agonist | 0.015 0.005 CHEMBL3544523 0.048 0.002 CHEMBL3544524 | CHEMBL3544524 | |
| 0.028 | 0.062 | 0.088 | NMDA receptor subunit 3B antagonist | 0.046 0.028 CHEMBL1908020 0.045 0.029 CHEMBL1908021 0.045 0.03 CHEMBL3544888 0.088 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.024 | 0.059 | 0.069 | Glutamate (mGluR3) agonist | 0.047 0.005 CHEMBL3544523 0.069 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.061 | 0.096 | 0.076 | Vanilloid 4 agonist | 0.076 0.048 CHEMBL3544524 | CHEMBL3544524 | |
| 0.041 | 0.076 | 0.105 | Carbonic anhydrase stimulant | 0.093 0.021 CHEMBL3544523 0.105 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.032 | 0.067 | 0.075 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.045 0.021 CHEMBL3544523 0.075 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.042 | 0.036 | Kainate receptor 1 antagonist | 0.036 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.041 | 0.076 | 0.125 | Heparanase inhibitor | 0.082 0.006 CHEMBL3544522 0.125 0.003 CHEMBL3544887 0.054 0.035 CHEMBL3544524 | CHEMBL3544887 | |
| 0.165 | 0.202 | 0.464 | Cholesterol antagonist | 0.214 0.152 CHEMBL1908020 0.456 0.04 CHEMBL3544522 0.22 0.147 CHEMBL1908021 0.225 0.144 CHEMBL3544888 0.217 0.15 CHEMBL3638281 0.289 0.098 CHEMBL3544523 0.464 0.038 CHEMBL3544887 0.216 0.151 CHEMBL3548560 0.43 0.044 CHEMBL3544524 0.192 0.172 CHEMBL3544501 | CHEMBL3544887 | |
| 0.066 | 0.103 | 0.091 | MAP kinase kinase 7 inhibitor | 0.088 0.029 CHEMBL1908020 0.084 0.037 CHEMBL1908021 0.086 0.032 CHEMBL3544888 0.078 0.052 CHEMBL3548560 0.091 0.022 CHEMBL3544524 | CHEMBL3544524 | |
| 0.021 | 0.059 | 0.07 | Kainate receptor antagonist | 0.039 0.03 CHEMBL3544523 0.07 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.015 | 0.053 | 0.055 | Lysine carboxypeptidase inhibitor | 0.04 0.01 CHEMBL3544523 0.055 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.099 | 0.139 | 0.259 | Cell wall synthesis inhibitor | 0.25 0.016 CHEMBL3544522 0.168 0.049 CHEMBL3544523 0.259 0.014 CHEMBL3544887 0.187 0.036 CHEMBL3544524 | CHEMBL3544887 | |
| 0.029 | 0.069 | 0.092 | Mannosidase inhibitor | 0.073 0.011 CHEMBL3544522 0.054 0.022 CHEMBL3544523 0.083 0.008 CHEMBL3544887 0.092 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.008 | 0.049 | 0.02 | Thromboxane A2 agonist | 0.016 0.01 CHEMBL3544523 0.02 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.046 | 0.088 | 0.221 | Catalase inhibitor | 0.214 0.013 CHEMBL3544523 0.221 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.049 | 0.092 | 0.07 | Interferon inducer | 0.07 0.035 CHEMBL3544524 | CHEMBL3544524 | |
| 0.046 | 0.089 | 0.061 | Immunoglobulin Fc receptor antagonist | 0.061 0.023 CHEMBL3544524 | CHEMBL3544524 | |
| 0.055 | 0.098 | 0.179 | GABA aminotransferase inhibitor | 0.068 0.064 CHEMBL1908021 0.068 0.066 CHEMBL3544888 0.122 0.015 CHEMBL3544523 0.179 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.051 | 0.025 | Aminopeptidase A inhibitor | 0.016 0.015 CHEMBL3544523 0.025 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.055 | 0.101 | 0.145 | Ornithine decarboxylase inhibitor | 0.096 0.048 CHEMBL3544523 0.145 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.07 | 0.031 | Melatonin receptor 1A agonist | 0.031 0.03 CHEMBL3544523 | CHEMBL3544523 | |
| 0.124 | 0.172 | 0.301 | Phospholipase C inhibitor | 0.144 0.118 CHEMBL1908020 0.153 0.101 CHEMBL3544522 0.148 0.11 CHEMBL1908021 0.148 0.111 CHEMBL3544888 0.273 0.021 CHEMBL3544523 0.143 0.12 CHEMBL3548560 0.301 0.018 CHEMBL3544524 | CHEMBL3544524 | |
| 0.005 | 0.053 | 0.014 | Lysophosphatidic acid receptor 3 agonist | 0.014 0.009 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.057 | 0.021 | Telomerase stimulant | 0.021 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.019 | 0.069 | 0.085 | NMDA receptor subunit 3A antagonist | 0.085 0.01 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.065 | 0.025 | Neuraminidase (Influenza B) inhibitor | 0.025 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.075 | 0.056 | Glycine transporter 2 inhibitor | 0.056 0.027 CHEMBL3544524 | CHEMBL3544524 | |
| 0.051 | 0.103 | 0.063 | Beta 2 adrenoreceptor agonist | 0.061 0.044 CHEMBL1908020 0.063 0.039 CHEMBL1908021 0.063 0.039 CHEMBL3544888 0.06 0.049 CHEMBL3544523 0.061 0.044 CHEMBL3548560 0.06 0.05 CHEMBL3544524 | CHEMBL3544888 | |
| 0.012 | 0.065 | 0.045 | AMPA 3 receptor antagonist | 0.028 0.022 CHEMBL3544523 0.045 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.074 | 0.127 | 0.291 | AMP-activated protein kinase stimulant | 0.089 0.087 CHEMBL1908020 0.169 0.018 CHEMBL3544522 0.091 0.083 CHEMBL1908021 0.096 0.077 CHEMBL3544888 0.106 0.063 CHEMBL3638281 0.291 0.005 CHEMBL3544887 0.092 0.082 CHEMBL3548560 | CHEMBL3544887 | |
| 0.082 | 0.135 | 0.167 | Photosensitizer | 0.12 0.057 CHEMBL3544887 0.167 0.022 CHEMBL3544524 | CHEMBL3544524 | |
| 0.074 | 0.128 | 0.255 | Beta glucuronidase inhibitor | 0.109 0.057 CHEMBL1908020 0.138 0.032 CHEMBL3544522 0.107 0.06 CHEMBL1908021 0.105 0.063 CHEMBL3544888 0.255 0.008 CHEMBL3544887 0.11 0.056 CHEMBL3548560 0.113 0.053 CHEMBL3544501 | CHEMBL3544887 | |
| 0.067 | 0.121 | 0.273 | Expectorant | 0.178 0.026 CHEMBL3544522 0.087 0.086 CHEMBL1908021 0.088 0.083 CHEMBL3544888 0.134 0.042 CHEMBL3638281 0.137 0.041 CHEMBL3544523 0.273 0.01 CHEMBL3544887 0.096 0.074 CHEMBL3548560 0.187 0.023 CHEMBL3544524 0.127 0.046 CHEMBL3544501 | CHEMBL3544887 | |
| 0.018 | 0.074 | 0.025 | Complement factor 1s inhibitor | 0.025 0.018 CHEMBL3544524 | CHEMBL3544524 | |
| 0.043 | 0.101 | 0.126 | Phosphodiesterase 4D inhibitor | 0.126 0.026 CHEMBL3544501 | CHEMBL3544501 | |
| 0.05 | 0.109 | 0.061 | Transcription factor RelA inhibitor | 0.061 0.052 CHEMBL3544501 | CHEMBL3544501 | |
| 0.054 | 0.114 | 0.086 | Interferon agonist | 0.086 0.043 CHEMBL3544524 | CHEMBL3544524 | |
| 0.011 | 0.072 | 0.032 | Geranylgeranyltransferase inhibitor | 0.032 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.025 | 0.086 | 0.083 | Glutamate (mGluR8) antagonist | 0.055 0.006 CHEMBL3544523 0.083 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.091 | 0.152 | 0.172 | Sphingosine 1-phosphate receptor 4 antagonist | 0.172 0.018 CHEMBL3544524 | CHEMBL3544524 | |
| 0.02 | 0.081 | 0.045 | Dihydropteroate synthase inhibitor | 0.045 0.021 CHEMBL3544524 | CHEMBL3544524 | |
| 0.036 | 0.098 | 0.075 | NMDA 2 receptor antagonist | 0.075 0.047 CHEMBL1908020 0.075 0.047 CHEMBL1908021 0.072 0.05 CHEMBL3544888 | CHEMBL1908021 | |
| 0.015 | 0.077 | 0.03 | Vanilloid 2 agonist | 0.024 0.022 CHEMBL3544887 0.03 0.01 CHEMBL3544524 | CHEMBL3544524 | |
| 0.066 | 0.128 | 0.123 | Lanosterol 14 alpha demethylase inhibitor | 0.123 0.028 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.072 | 0.08 | Arginase inhibitor | 0.032 0.03 CHEMBL3544522 0.08 0.006 CHEMBL3544523 0.037 0.025 CHEMBL3544887 0.08 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.011 | 0.074 | 0.022 | Antibiotic Anthracycline-like | 0.021 0.009 CHEMBL3544522 0.022 0.008 CHEMBL3544887 0.019 0.013 CHEMBL3544524 | CHEMBL3544887 | |
| 0.006 | 0.069 | 0.031 | AMPA 1 receptor antagonist | 0.031 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.022 | 0.086 | 0.061 | Adenosine deaminase inhibitor | 0.061 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.026 | 0.091 | 0.064 | Xanthine dehydrogenase inhibitor | 0.059 0.039 CHEMBL1908020 0.054 0.043 CHEMBL1908021 0.057 0.041 CHEMBL3544888 0.064 0.036 CHEMBL3548560 0.052 0.045 CHEMBL3544501 | CHEMBL3548560 | |
| 0.034 | 0.1 | 0.044 | Beta adrenoreceptor agonist | 0.043 0.039 CHEMBL1908020 0.044 0.037 CHEMBL1908021 0.044 0.037 CHEMBL3544888 0.043 0.041 CHEMBL3548560 | CHEMBL3544888 | |
| 0.061 | 0.129 | 0.108 | Falcipain 3 inhibitor | 0.108 0.063 CHEMBL3544524 | CHEMBL3544524 | |
| 0.046 | 0.114 | 0.07 | Beta 3 adrenoreceptor antagonist | 0.06 0.055 CHEMBL1908020 0.061 0.053 CHEMBL1908021 0.06 0.054 CHEMBL3544888 0.061 0.053 CHEMBL3548560 0.07 0.034 CHEMBL3544524 | CHEMBL3544524 | |
| 0.028 | 0.097 | 0.068 | Lysophosphatidic acid 3 receptor antagonist | 0.068 0.016 CHEMBL3544524 | CHEMBL3544524 | |
| 0.016 | 0.086 | 0.031 | Calcitonin receptor agonist | 0.031 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.078 | 0.019 | Nicotinic acid receptor 1 antagonist | 0.019 0.009 CHEMBL3544524 | CHEMBL3544524 | |
| 0.02 | 0.092 | 0.061 | Ribonucleotide reductase inhibitor | 0.061 0.036 CHEMBL3544523 0.059 0.037 CHEMBL3544524 | CHEMBL3544523 | |
| 0.051 | 0.122 | 0.105 | Histamine N-methyltransferase inhibitor | 0.105 0.042 CHEMBL3544524 | CHEMBL3544524 | |
| 0.049 | 0.123 | 0.077 | Adrenaline antagonist | 0.077 0.071 CHEMBL3544501 | CHEMBL3544501 | |
| 0.051 | 0.126 | 0.079 | Antiadrenergic | 0.079 0.072 CHEMBL3544501 | CHEMBL3544501 | |
| 0.013 | 0.089 | 0.068 | Sodium/glucose cotransporter inhibitor | 0.03 0.011 CHEMBL3544522 0.068 0.004 CHEMBL3544887 | CHEMBL3544887 | |
| 0.049 | 0.127 | 0.088 | Myeloperoxidase inhibitor | 0.088 0.053 CHEMBL3544524 | CHEMBL3544524 | |
| 0.068 | 0.148 | 0.145 | Glutamate release inhibitor | 0.084 0.079 CHEMBL3544523 0.145 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.039 | 0.12 | 0.084 | Potassium channel intermediate-conductance Ca-activated blocker | 0.084 0.015 CHEMBL3544524 | CHEMBL3544524 | |
| 0.154 | 0.235 | 0.297 | Vasodilator, peripheral | 0.252 0.125 CHEMBL3544522 0.297 0.098 CHEMBL3544524 0.199 0.177 CHEMBL3544501 | CHEMBL3544524 | |
| 0.166 | 0.247 | 0.538 | Alpha-glucosidase inhibitor | 0.281 0.169 CHEMBL1908020 0.283 0.169 CHEMBL1908021 0.276 0.173 CHEMBL3544888 0.538 0.07 CHEMBL3544887 0.307 0.156 CHEMBL3548560 0.363 0.13 CHEMBL3544501 | CHEMBL3544887 | |
| 0.048 | 0.129 | 0.084 | Adrenaline agonist | 0.082 0.055 CHEMBL1908020 0.084 0.053 CHEMBL1908021 0.083 0.053 CHEMBL3544888 0.081 0.057 CHEMBL3548560 | CHEMBL1908021 | |
| 0.02 | 0.102 | 0.058 | Guanylate cyclase inhibitor | 0.058 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.103 | 0.186 | 0.212 | Interferon gamma antagonist | 0.129 0.112 CHEMBL1908020 0.175 0.054 CHEMBL3544522 0.127 0.118 CHEMBL3544888 0.212 0.037 CHEMBL3544887 0.129 0.112 CHEMBL3548560 0.17 0.057 CHEMBL3544524 | CHEMBL3544887 | |
| 0.03 | 0.115 | 0.06 | Dopamine beta hydroxylase inhibitor | 0.06 0.015 CHEMBL3544524 | CHEMBL3544524 | |
| 0.017 | 0.103 | 0.046 | Toll-Like receptor 2 agonist | 0.046 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.018 | 0.108 | 0.06 | Ribonucleoside-diphosphate reductase inhibitor | 0.06 0.034 CHEMBL3544523 0.058 0.035 CHEMBL3544524 | CHEMBL3544523 | |
| 0.073 | 0.163 | 0.122 | TRPA1 agonist | 0.122 0.056 CHEMBL3544524 | CHEMBL3544524 | |
| 0.052 | 0.144 | 0.157 | Bronchodilator | 0.105 0.058 CHEMBL1908020 0.094 0.071 CHEMBL1908021 0.096 0.068 CHEMBL3544888 0.104 0.059 CHEMBL3548560 0.157 0.029 CHEMBL3544501 | CHEMBL3544501 | |
| 0.018 | 0.11 | 0.04 | Carboxypeptidase B inhibitor | 0.039 0.014 CHEMBL3544523 0.04 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.081 | 0.174 | 0.205 | Protein kinase stimulant | 0.205 0.04 CHEMBL3544887 0.164 0.059 CHEMBL3544524 0.108 0.107 CHEMBL3544501 | CHEMBL3544887 | |
| 0.108 | 0.201 | 0.204 | Lipocortins synthesis antagonist | 0.142 0.117 CHEMBL1908020 0.135 0.13 CHEMBL3544522 0.163 0.088 CHEMBL3638281 0.142 0.117 CHEMBL3548560 0.204 0.054 CHEMBL3544524 | CHEMBL3544524 | |
| 0.012 | 0.107 | 0.04 | Phosphoglycerate kinase inhibitor | 0.038 0.021 CHEMBL3544523 0.04 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.012 | 0.107 | 0.063 | Carbonic anhydrase IX inhibitor | 0.063 0.036 CHEMBL3544522 | CHEMBL3544522 | |
| 0.014 | 0.109 | 0.035 | Urate transporter 1 inhibitor | 0.035 0.032 CHEMBL3544524 | CHEMBL3544524 | |
| 0.016 | 0.113 | 0.029 | Estrogen-related receptor gamma antagonist | 0.029 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.036 | 0.133 | 0.071 | Beta adrenoreceptor antagonist | 0.07 0.038 CHEMBL3544523 0.071 0.037 CHEMBL3544524 | CHEMBL3544524 | |
| 0.09 | 0.19 | 0.15 | Vanilloid 1 agonist | 0.123 0.081 CHEMBL3544523 0.15 0.038 CHEMBL3544524 0.128 0.069 CHEMBL3544501 | CHEMBL3544524 | |
| 0.071 | 0.172 | 0.244 | Aldehyde dehydrogenase inhibitor | 0.116 0.076 CHEMBL3544523 0.244 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.018 | 0.118 | 0.044 | Opioid mu receptor agonist | 0.044 0.035 CHEMBL1908020 0.043 0.036 CHEMBL1908021 0.044 0.035 CHEMBL3544888 | CHEMBL3544888 | |
| 0.043 | 0.145 | 0.075 | Phosphodiesterase 3A inhibitor | 0.075 0.064 CHEMBL3544501 | CHEMBL3544501 | |
| 0.019 | 0.121 | 0.046 | Opioid agonist | 0.046 0.045 CHEMBL1908020 0.046 0.045 CHEMBL1908021 0.046 0.045 CHEMBL3544888 | CHEMBL3544888 | |
| 0.124 | 0.227 | 0.641 | Hypoglycemic | 0.213 0.101 CHEMBL1908020 0.516 0.014 CHEMBL3544522 0.214 0.1 CHEMBL1908021 0.225 0.093 CHEMBL3544888 0.206 0.107 CHEMBL3638281 0.641 0.006 CHEMBL3544887 0.221 0.095 CHEMBL3548560 0.204 0.109 CHEMBL3544501 | CHEMBL3544887 | |
| 0.064 | 0.166 | 0.149 | Carbonic anhydrase XV inhibitor | 0.149 0.031 CHEMBL3544524 | CHEMBL3544524 | |
| 0.096 | 0.2 | 0.197 | Melanin inhibitor | 0.14 0.097 CHEMBL1908020 0.139 0.099 CHEMBL3544522 0.136 0.103 CHEMBL1908021 0.139 0.098 CHEMBL3544888 0.197 0.042 CHEMBL3544887 0.139 0.097 CHEMBL3548560 0.178 0.053 CHEMBL3544524 0.152 0.078 CHEMBL3544501 | CHEMBL3544887 | |
| 0.027 | 0.132 | 0.05 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.05 0.042 CHEMBL1908020 | CHEMBL1908020 | |
| 0.034 | 0.139 | 0.093 | Na+ K+ transporting ATPase inhibitor | 0.079 0.052 CHEMBL3544522 0.078 0.052 CHEMBL3544887 0.093 0.038 CHEMBL3544524 | CHEMBL3544524 | |
| 0.039 | 0.144 | 0.088 | CYP2A6 inhibitor | 0.088 0.043 CHEMBL3544524 | CHEMBL3544524 | |
| 0.042 | 0.151 | 0.256 | Monophenol monooxygenase inhibitor | 0.114 0.066 CHEMBL1908020 0.11 0.068 CHEMBL3544522 0.111 0.068 CHEMBL1908021 0.114 0.066 CHEMBL3544888 0.256 0.023 CHEMBL3544887 0.114 0.066 CHEMBL3548560 0.133 0.054 CHEMBL3544524 0.125 0.058 CHEMBL3544501 | CHEMBL3544887 | |
| 0.01 | 0.118 | 0.025 | Prostaglandin F2 alpha agonist | 0.025 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.06 | 0.169 | 0.346 | Amylase inhibitor | 0.117 0.083 CHEMBL1908020 0.2 0.044 CHEMBL3544522 0.11 0.088 CHEMBL1908021 0.113 0.086 CHEMBL3544888 0.346 0.013 CHEMBL3544887 0.12 0.081 CHEMBL3548560 0.207 0.042 CHEMBL3544524 0.14 0.069 CHEMBL3544501 | CHEMBL3544887 | |
| 0.017 | 0.126 | 0.058 | GABA uptake inhibitor | 0.058 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.118 | 0.029 | Dopamine D1 agonist | 0.026 0.012 CHEMBL3544887 0.029 0.009 CHEMBL3548560 0.024 0.014 CHEMBL3544501 | CHEMBL3548560 | |
| 0.057 | 0.167 | 0.102 | Bile acid receptor antagonist | 0.102 0.045 CHEMBL3544524 | CHEMBL3544524 | |
| 0.029 | 0.14 | 0.154 | Sphingosine 1-phosphate receptor 4 agonist | 0.071 0.043 CHEMBL3544523 0.154 0.008 CHEMBL3544524 | CHEMBL3544524 | |
| 0.087 | 0.2 | 0.139 | Thiol protease inhibitor | 0.139 0.081 CHEMBL3544524 | CHEMBL3544524 | |
| 0.08 | 0.194 | 0.243 | Diuretic | 0.243 0.032 CHEMBL3544523 0.157 0.072 CHEMBL3544887 0.205 0.042 CHEMBL3544524 | CHEMBL3544523 | |
| 0.01 | 0.125 | 0.037 | 5-Alpha-reductase inhibitor | 0.037 0.026 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.126 | 0.025 | Retinoid X beta receptor antagonist | 0.025 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.057 | 0.173 | 0.162 | Carbonic anhydrase III inhibitor | 0.086 0.081 CHEMBL1908020 0.086 0.081 CHEMBL3548560 0.162 0.024 CHEMBL3544524 | CHEMBL3544524 | |
| 0.032 | 0.148 | 0.075 | CD45 antagonist | 0.075 0.013 CHEMBL3544524 | CHEMBL3544524 | |
| 0.063 | 0.18 | 0.125 | Microtubule formation inhibitor | 0.1 0.09 CHEMBL3544522 0.102 0.088 CHEMBL3638281 0.123 0.057 CHEMBL3544523 0.125 0.055 CHEMBL3544524 | CHEMBL3544524 | |
| 0.069 | 0.187 | 0.18 | Toll-Like receptor 2 antagonist | 0.109 0.09 CHEMBL1908020 0.133 0.065 CHEMBL3544523 0.116 0.082 CHEMBL3548560 0.18 0.034 CHEMBL3544524 0.142 0.058 CHEMBL3544501 | CHEMBL3544524 | |
| 0.03 | 0.149 | 0.059 | Epithelial sodium channel blocker | 0.059 0.03 CHEMBL3544524 | CHEMBL3544524 | |
| 0.088 | 0.208 | 0.199 | DNA methyltransferase I inhibitor | 0.195 0.072 CHEMBL3544887 0.135 0.122 CHEMBL3548560 0.157 0.097 CHEMBL3544524 0.199 0.069 CHEMBL3544501 | CHEMBL3544501 | |
| 0.16 | 0.28 | 0.205 | MAP kinase kinase 3 inhibitor | 0.186 0.168 CHEMBL3544523 0.205 0.108 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.145 | 0.074 | Opioid mu receptor antagonist | 0.074 0.043 CHEMBL1908020 0.072 0.044 CHEMBL1908021 0.073 0.044 CHEMBL3544888 | CHEMBL1908020 | |
| 0.037 | 0.159 | 0.07 | Adenine nucleotide translocase inhibitor | 0.053 0.045 CHEMBL1908020 0.067 0.019 CHEMBL3544522 0.054 0.044 CHEMBL1908021 0.054 0.044 CHEMBL3544888 0.07 0.015 CHEMBL3544887 0.059 0.031 CHEMBL3548560 0.058 0.032 CHEMBL3544524 0.053 0.045 CHEMBL3544501 | CHEMBL3544887 | |
| 0.159 | 0.284 | 0.61 | Antibacterial | 0.586 0.021 CHEMBL3544522 0.223 0.204 CHEMBL3544888 0.336 0.11 CHEMBL3638281 0.61 0.018 CHEMBL3544887 0.217 0.21 CHEMBL3548560 | CHEMBL3544887 | |
| 0.018 | 0.144 | 0.07 | Glutamate (mGluR4) agonist | 0.07 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.14 | 0.267 | 0.568 | Antithrombotic | 0.412 0.046 CHEMBL3544522 0.192 0.188 CHEMBL3638281 0.191 0.188 CHEMBL3544523 0.568 0.02 CHEMBL3544887 0.311 0.081 CHEMBL3544524 | CHEMBL3544887 | |
| 0.028 | 0.154 | 0.045 | Topoisomerase II beta inhibitor | 0.045 0.042 CHEMBL3544524 | CHEMBL3544524 | |
| 0.014 | 0.141 | 0.051 | Geranyltranstransferase inhibitor | 0.04 0.036 CHEMBL3544523 0.051 0.021 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.14 | 0.038 | Diamine oxidase inhibitor | 0.038 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.094 | 0.228 | 0.126 | Pregnane X receptor agonist | 0.126 0.112 CHEMBL3544524 | CHEMBL3544524 | |
| 0.027 | 0.161 | 0.06 | Sphingosine kinase 2 inhibitor | 0.06 0.031 CHEMBL3544524 | CHEMBL3544524 | |
| 0.025 | 0.163 | 0.07 | Sphingosine 1-phosphate receptor 3 antagonist | 0.07 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.025 | 0.164 | 0.046 | Cytokine production stimulant | 0.046 0.041 CHEMBL3544524 | CHEMBL3544524 | |
| 0.044 | 0.186 | 0.098 | Sphingomyelinase inhibitor | 0.098 0.062 CHEMBL3544524 | CHEMBL3544524 | |
| 0.021 | 0.163 | 0.052 | Diacylglycerol O-acyltransferase inhibitor | 0.052 0.034 CHEMBL3544524 | CHEMBL3544524 | |
| 0.026 | 0.175 | 0.096 | Glutamate receptor agonist | 0.096 0.04 CHEMBL3544524 | CHEMBL3544524 | |
| 0.02 | 0.169 | 0.133 | Glutamate (mGluR group III) agonist | 0.133 0.006 CHEMBL3544524 | CHEMBL3544524 | |
| 0.083 | 0.237 | 0.21 | DNA methylase inhibitor | 0.21 0.073 CHEMBL3544887 0.167 0.103 CHEMBL3544524 0.184 0.09 CHEMBL3544501 | CHEMBL3544887 | |
| 0.011 | 0.166 | 0.034 | ATP citrate lysase inhibitor | 0.034 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.162 | 0.05 | Sodium/glucose cotransporter 2 inhibitor | 0.026 0.019 CHEMBL3544522 0.05 0.006 CHEMBL3544887 | CHEMBL3544887 | |
| 0.027 | 0.188 | 0.06 | Sphingosine kinase inhibitor | 0.06 0.039 CHEMBL3544524 | CHEMBL3544524 | |
| 0.037 | 0.199 | 0.09 | Opioid antagonist | 0.09 0.056 CHEMBL1908020 0.088 0.058 CHEMBL1908021 0.089 0.058 CHEMBL3544888 | CHEMBL1908020 | |
| 0.01 | 0.172 | 0.057 | Retinoid X alpha receptor agonist | 0.057 0.012 CHEMBL3544524 | CHEMBL3544524 | |
| 0.006 | 0.168 | 0.036 | Kynurenine 3 monooxygenase inhibitor | 0.036 0.011 CHEMBL3544524 | CHEMBL3544524 | |
| 0.008 | 0.17 | 0.039 | Free fatty acid receptor 1 antagonist | 0.039 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.016 | 0.179 | 0.04 | Retinoid X alpha receptor antagonist | 0.04 0.015 CHEMBL3544524 | CHEMBL3544524 | |
| 0.028 | 0.191 | 0.074 | Phosphodiesterase IV inhibitor | 0.074 0.068 CHEMBL3544501 | CHEMBL3544501 | |
| 0.036 | 0.201 | 0.06 | Leukotriene C antagonist | 0.06 0.029 CHEMBL3544524 | CHEMBL3544524 | |
| 0.038 | 0.204 | 0.101 | Urease inhibitor | 0.088 0.08 CHEMBL3544523 0.101 0.066 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.176 | 0.025 | Calcium-sensing receptor agonist | 0.025 0.021 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.173 | 0.069 | Glutamate (mGluR2) antagonist | 0.069 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.19 | 0.039 | Leukotriene C4 antagonist | 0.039 0.027 CHEMBL3544524 | CHEMBL3544524 | |
| 0.022 | 0.189 | 0.067 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.052 0.05 CHEMBL3544523 0.067 0.033 CHEMBL3544524 | CHEMBL3544524 | |
| 0.017 | 0.188 | 0.045 | Retinoid X receptor antagonist | 0.045 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.028 | 0.2 | 0.054 | Sphingosine 1-phosphate receptor 1 antagonist | 0.054 0.042 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.184 | 0.158 | Glutamate (mGluR group II) antagonist | 0.158 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.07 | 0.245 | 0.11 | Transcription factor STAT6 inhibitor | 0.11 0.079 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.189 | 0.094 | Glutamate (mGluR1) antagonist | 0.094 0.018 CHEMBL3544524 | CHEMBL3544524 | |
| 0.035 | 0.213 | 0.086 | Inducible nitric-oxide synthase inhibitor | 0.086 0.053 CHEMBL3544524 | CHEMBL3544524 | |
| 0.02 | 0.198 | 0.062 | Dopamine agonist | 0.062 0.05 CHEMBL3548560 | CHEMBL3548560 | |
| 0.057 | 0.236 | 0.204 | Cyclooxygenase 3 inhibitor | 0.164 0.038 CHEMBL3544522 0.204 0.017 CHEMBL3544887 0.169 0.034 CHEMBL3544524 | CHEMBL3544887 | |
| 0.105 | 0.292 | 0.245 | 12-Lipoxygenase inhibitor | 0.195 0.158 CHEMBL1908020 0.19 0.163 CHEMBL1908021 0.185 0.168 CHEMBL3544888 0.211 0.139 CHEMBL3548560 0.245 0.112 CHEMBL3544501 | CHEMBL3544501 | |
| 0.049 | 0.236 | 0.105 | Caspase 3 inhibitor | 0.105 0.084 CHEMBL3544524 | CHEMBL3544524 | |
| 0.006 | 0.194 | 0.051 | Retinoid X receptor agonist | 0.051 0.018 CHEMBL3544524 | CHEMBL3544524 | |
| 0.057 | 0.247 | 0.106 | NADPH oxidase inhibitor | 0.106 0.102 CHEMBL3544501 | CHEMBL3544501 | |
| 0.062 | 0.253 | 0.159 | Pyruvate kinase inhibitor | 0.159 0.108 CHEMBL3544524 | CHEMBL3544524 | |
| 0.038 | 0.232 | 0.154 | ATPase (Vacuolar H+) inhibitor | 0.094 0.049 CHEMBL3544522 0.154 0.007 CHEMBL3638281 0.122 0.018 CHEMBL3544887 0.083 0.071 CHEMBL3548560 0.099 0.042 CHEMBL3544501 | CHEMBL3638281 | |
| 0.01 | 0.207 | 0.033 | 1-Alkyl-2-acetylglycerophosphocholine esterase inhibitor | 0.033 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.029 | 0.229 | 0.105 | Potassium channel (Ca-activated) activator | 0.105 0.051 CHEMBL3544524 | CHEMBL3544524 | |
| 0.041 | 0.242 | 0.101 | Interleukin 1 beta converting enzyme inhibitor | 0.101 0.056 CHEMBL3544524 | CHEMBL3544524 | |
| 0.024 | 0.225 | 0.056 | Botulinum neurotoxin type A inhibitor | 0.056 0.044 CHEMBL3544524 | CHEMBL3544524 | |
| 0.04 | 0.249 | 0.107 | Glutathione S-transferase inhibitor | 0.107 0.031 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.223 | 0.044 | Carbonic anhydrase XIV inhibitor | 0.044 0.041 CHEMBL3544524 | CHEMBL3544524 | |
| 0.111 | 0.324 | 0.436 | Immunomodulator | 0.29 0.088 CHEMBL3544522 0.436 0.034 CHEMBL3544887 | CHEMBL3544887 | |
| 0.029 | 0.243 | 0.07 | Macrophage migration inhibitory factor inhibitor | 0.07 0.066 CHEMBL3544524 | CHEMBL3544524 | |
| 0.034 | 0.254 | 0.071 | Sphingosine 1-phosphate receptor antagonist | 0.071 0.069 CHEMBL3544524 | CHEMBL3544524 | |
| 0.003 | 0.223 | 0.024 | Prostaglandin H2 antagonist | 0.024 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.042 | 0.265 | 0.115 | Thioredoxin inhibitor | 0.115 0.034 CHEMBL3544887 | CHEMBL3544887 | |
| 0.02 | 0.243 | 0.056 | Thromboxane synthase inhibitor | 0.05 0.048 CHEMBL3544523 0.056 0.035 CHEMBL3544524 | CHEMBL3544524 | |
| 0.094 | 0.318 | 0.472 | Transcription factor NF kappa B inhibitor | 0.188 0.181 CHEMBL1908020 0.278 0.108 CHEMBL3544522 0.472 0.049 CHEMBL3544887 0.199 0.17 CHEMBL3548560 0.217 0.153 CHEMBL3544524 0.24 0.135 CHEMBL3544501 | CHEMBL3544887 | |
| 0.009 | 0.235 | 0.024 | ICAM 1 antagonist | 0.024 0.014 CHEMBL3544524 | CHEMBL3544524 | |
| 0.061 | 0.288 | 0.136 | Amyloid beta precursor protein antagonist | 0.136 0.118 CHEMBL3544501 | CHEMBL3544501 | |
| 0.07 | 0.3 | 0.283 | Hemostatic | 0.151 0.066 CHEMBL3544522 0.139 0.082 CHEMBL3544523 0.268 0.019 CHEMBL3544887 0.283 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.06 | 0.292 | 0.227 | Insulin sensitizer | 0.193 0.081 CHEMBL3544523 0.227 0.049 CHEMBL3544524 | CHEMBL3544524 | |
| 0.03 | 0.262 | 0.084 | Somatostatin 1 agonist | 0.084 0.047 CHEMBL3544523 | CHEMBL3544523 | |
| 0.05 | 0.285 | 0.085 | Hematopoietic | 0.085 0.059 CHEMBL3544524 | CHEMBL3544524 | |
| 0.006 | 0.24 | 0.019 | Integrin beta5 antagonist | 0.019 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.096 | 0.332 | 0.208 | Hypoxia-inducible factor 1 alpha inhibitor | 0.181 0.177 CHEMBL3638281 0.208 0.142 CHEMBL3544501 | CHEMBL3544501 | |
| 0.031 | 0.273 | 0.105 | Mediator release inhibitor | 0.105 0.065 CHEMBL3544887 | CHEMBL3544887 | |
| 0.041 | 0.289 | 0.133 | DNA polymerase I inhibitor | 0.127 0.063 CHEMBL3544522 0.133 0.059 CHEMBL3544887 0.122 0.067 CHEMBL3548560 0.111 0.075 CHEMBL3544501 | CHEMBL3544887 | |
| 0.006 | 0.264 | 0.05 | Sphingosine 1-phosphate receptor 1 agonist | 0.05 0.02 CHEMBL3544524 | CHEMBL3544524 | |
| 0.03 | 0.292 | 0.12 | Cholesterol synthesis inhibitor | 0.12 0.065 CHEMBL3544524 | CHEMBL3544524 | |
| 0.008 | 0.273 | 0.045 | Thromboxane A2 antagonist | 0.045 0.04 CHEMBL3544524 | CHEMBL3544524 | |
| 0.076 | 0.342 | 0.116 | Papain-like protease (SARS coronavirus) inhibitor | 0.116 0.093 CHEMBL1908020 0.115 0.095 CHEMBL1908021 0.113 0.102 CHEMBL3544888 0.112 0.106 CHEMBL3548560 0.113 0.102 CHEMBL3544501 | CHEMBL1908020 | |
| 0.043 | 0.311 | 0.138 | Transcription factor NF kappa B stimulant | 0.121 0.025 CHEMBL3544522 0.138 0.019 CHEMBL3544887 | CHEMBL3544887 | |
| 0.015 | 0.293 | 0.051 | Leukotriene B4 antagonist | 0.051 0.043 CHEMBL3544524 | CHEMBL3544524 | |
| 0.029 | 0.316 | 0.094 | Nitric-oxide synthase inhibitor | 0.094 0.071 CHEMBL3544524 | CHEMBL3544524 | |
| 0.009 | 0.318 | 0.05 | Sphingosine 1-phosphate receptor agonist | 0.05 0.025 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.331 | 0.031 | Toll-Like receptor 4 agonist | 0.031 0.011 CHEMBL3544522 0.031 0.01 CHEMBL3544887 | CHEMBL3544887 | |
| 0.056 | 0.384 | 0.284 | NOS3 expression enhancer | 0.132 0.095 CHEMBL1908020 0.222 0.033 CHEMBL3544522 0.125 0.105 CHEMBL1908021 0.124 0.107 CHEMBL3544888 0.284 0.02 CHEMBL3544887 0.139 0.085 CHEMBL3548560 | CHEMBL3544887 | |
| 0.076 | 0.405 | 0.138 | Death-associated protein kinase 2 inhibitor | 0.138 0.136 CHEMBL3548560 | CHEMBL3548560 | |
| 0.037 | 0.38 | 0.162 | Phospholipase A2 inhibitor | 0.162 0.064 CHEMBL3544524 | CHEMBL3544524 | |
| 0.023 | 0.369 | 0.218 | Topoisomerase II inhibitor | 0.105 0.082 CHEMBL1908020 0.147 0.051 CHEMBL3544522 0.218 0.029 CHEMBL3544887 0.1 0.086 CHEMBL3548560 0.117 0.07 CHEMBL3544501 | CHEMBL3544887 | |
| 0.051 | 0.412 | 0.149 | Non-steroidal antiinflammatory agent | 0.149 0.115 CHEMBL3544887 0.149 0.116 CHEMBL3544524 | CHEMBL3544524 | |
| 0.102 | 0.469 | 0.416 | Interleukin 2 agonist | 0.416 0.023 CHEMBL3544522 0.199 0.192 CHEMBL3638281 0.269 0.099 CHEMBL3544523 0.406 0.026 CHEMBL3544887 0.359 0.042 CHEMBL3544524 | CHEMBL3544522 | |
| 0.005 | 0.378 | 0.213 | Geranylgeranyltransferase I inhibitor | 0.213 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.383 | 0.049 | GP IIb/IIIa receptor antagonist | 0.049 0.033 CHEMBL3544524 | CHEMBL3544524 | |
| 0.039 | 0.419 | 0.283 | Platelet antagonist | 0.18 0.117 CHEMBL3544522 0.283 0.059 CHEMBL3544887 0.178 0.119 CHEMBL3544524 | CHEMBL3544887 | |
| 0.018 | 0.406 | 0.679 | Glutamate receptor antagonist | 0.327 0.008 CHEMBL3544523 0.679 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.021 | 0.434 | 0.114 | Cell adhesion molecule inhibitor | 0.078 0.055 CHEMBL3544522 0.114 0.026 CHEMBL3544887 0.083 0.05 CHEMBL3544524 | CHEMBL3544887 | |
| 0.013 | 0.435 | 0.056 | Nitric oxide donor | 0.056 0.055 CHEMBL3544887 | CHEMBL3544887 | |
| 0.01 | 0.442 | 0.047 | Neuraminidase (Influenza A) inhibitor | 0.042 0.039 CHEMBL3544522 0.047 0.028 CHEMBL3544887 | CHEMBL3544887 | |
| 0.007 | 0.448 | 0.053 | HIV-1 integrase (Strand Transfer) inhibitor | 0.053 0.047 CHEMBL3548560 | CHEMBL3548560 | |
| 0.077 | 0.52 | 0.311 | Caspase 3 stimulant | 0.206 0.161 CHEMBL1908020 0.23 0.132 CHEMBL3544522 0.256 0.107 CHEMBL3544887 0.226 0.136 CHEMBL3548560 0.311 0.073 CHEMBL3544501 | CHEMBL3544501 | |
| 0.021 | 0.468 | 0.083 | DNA helicase inhibitor | 0.058 0.032 CHEMBL3544523 0.083 0.01 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.456 | 0.072 | HIV-1 integrase (3'-Processing) inhibitor | 0.072 0.038 CHEMBL3548560 0.064 0.043 CHEMBL3544501 | CHEMBL3548560 | |
| 0.017 | 0.47 | 0.095 | DNA intercalator | 0.095 0.079 CHEMBL3544887 | CHEMBL3544887 | |
| 0.037 | 0.509 | 0.187 | Interleukin 6 antagonist | 0.187 0.049 CHEMBL3544887 | CHEMBL3544887 | |
| 0.004 | 0.491 | 0.161 | Antineoplastic antibiotic | 0.122 0.038 CHEMBL3544522 0.117 0.039 CHEMBL3638281 0.161 0.029 CHEMBL3544887 | CHEMBL3544887 | |
| 0.018 | 0.515 | 0.255 | Lipid peroxidase inhibitor | 0.122 0.091 CHEMBL1908020 0.171 0.055 CHEMBL3544522 0.113 0.101 CHEMBL1908021 0.118 0.096 CHEMBL3544888 0.255 0.026 CHEMBL3544887 0.154 0.066 CHEMBL3548560 0.158 0.063 CHEMBL3544501 | CHEMBL3544887 | |
| 0.02 | 0.565 | 0.503 | Free radical scavenger | 0.213 0.087 CHEMBL1908020 0.379 0.033 CHEMBL3544522 0.198 0.099 CHEMBL1908021 0.202 0.096 CHEMBL3544888 0.503 0.016 CHEMBL3544887 0.289 0.055 CHEMBL3548560 0.324 0.045 CHEMBL3544501 | CHEMBL3544887 | |
| 0.009 | 0.557 | 0.081 | HIV-1 integrase inhibitor | 0.081 0.037 CHEMBL3544522 0.068 0.052 CHEMBL3548560 | CHEMBL3544522 | |
| 0.037 | 0.588 | 0.391 | Hepatoprotectant | 0.336 0.021 CHEMBL3544522 0.391 0.014 CHEMBL3544887 0.136 0.126 CHEMBL3544501 | CHEMBL3544887 | |
| 0.021 | 0.581 | 0.212 | Cell adhesion inhibitor | 0.146 0.049 CHEMBL3544522 0.212 0.022 CHEMBL3544887 0.115 0.069 CHEMBL3544524 | CHEMBL3544887 | |
| 0.01 | 0.585 | 0.653 | Topoisomerase I inhibitor | 0.653 0.002 CHEMBL3544522 0.18 0.032 CHEMBL3544887 | CHEMBL3544522 | |
| 0.008 | 0.591 | 0.037 | Erythropoietin receptor agonist | 0.037 0.032 CHEMBL3544523 | CHEMBL3544523 | |
| 0.006 | 0.607 | 0.02 | Tryptophan hydroxylase 1 inhibitor | 0.02 0.007 CHEMBL3544524 | CHEMBL3544524 | |
| 0.017 | 0.619 | 0.644 | Angiogenesis stimulant | 0.543 0.009 CHEMBL3544522 0.644 0.005 CHEMBL3544887 0.195 0.097 CHEMBL3544524 | CHEMBL3544887 | |
| 0.02 | 0.627 | 0.547 | Antioxidant | 0.199 0.114 CHEMBL1908020 0.404 0.034 CHEMBL3544522 0.185 0.127 CHEMBL1908021 0.19 0.122 CHEMBL3544888 0.547 0.015 CHEMBL3544887 0.255 0.081 CHEMBL3548560 0.28 0.07 CHEMBL3544501 | CHEMBL3544887 | |
| 0.028 | 0.636 | 0.158 | Interleukin 4 antagonist | 0.158 0.043 CHEMBL3638281 0.108 0.105 CHEMBL3544887 0.107 0.105 CHEMBL3548560 0.114 0.094 CHEMBL3544501 | CHEMBL3638281 | |
| 0.004 | 0.63 | 0.045 | Protein 30S ribosomal subunit inhibitor | 0.03 0.013 CHEMBL3544522 0.045 0.009 CHEMBL3544887 | CHEMBL3544887 | |
| 0.003 | 0.631 | 0.056 | Complement C3a chemotactic receptor antagonist | 0.056 0.024 CHEMBL3544523 0.055 0.024 CHEMBL3544524 | CHEMBL3544523 | |
| 0.007 | 0.644 | 0.141 | Farnesyltransferase inhibitor | 0.141 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.656 | 0.072 | Antibiotic Aminoglycoside-like | 0.064 0.007 CHEMBL3544522 0.072 0.006 CHEMBL3544887 | CHEMBL3544887 | |
| 0.026 | 0.673 | 0.246 | Antiobesity | 0.246 0.16 CHEMBL3544522 | CHEMBL3544522 | |
| 0.019 | 0.672 | 0.061 | Caspase 9 inhibitor | 0.061 0.045 CHEMBL3544524 | CHEMBL3544524 | |
| 0.026 | 0.686 | 0.447 | Immunosuppressant | 0.346 0.089 CHEMBL3544522 0.249 0.148 CHEMBL3638281 0.447 0.048 CHEMBL3544887 | CHEMBL3544887 | |
| 0.019 | 0.689 | 0.097 | Electron transport complex I inhibitor | 0.097 0.091 CHEMBL3544501 | CHEMBL3544501 | |
| 0.013 | 0.684 | 0.037 | Integrin alpha1beta1 antagonist | 0.037 0.03 CHEMBL3544524 | CHEMBL3544524 | |
| 0.02 | 0.691 | 0.333 | Tumour necrosis factor alpha release inhibitor | 0.183 0.124 CHEMBL3544522 0.333 0.043 CHEMBL3544887 0.181 0.126 CHEMBL3544501 | CHEMBL3544887 | |
| 0.009 | 0.683 | 0.107 | Topoisomerase II alpha inhibitor | 0.066 0.065 CHEMBL3544522 0.107 0.035 CHEMBL3544887 | CHEMBL3544887 | |
| 0.041 | 0.716 | 0.327 | Sodium/bile acid cotransporter inhibitor | 0.216 0.166 CHEMBL1908020 0.223 0.158 CHEMBL3544523 0.327 0.056 CHEMBL3544524 0.202 0.185 CHEMBL3544501 | CHEMBL3544524 | |
| 0.005 | 0.685 | 0.655 | Factor VIIa inhibitor | 0.655 0.002 CHEMBL3544523 0.269 0.004 CHEMBL3544524 | CHEMBL3544523 | |
| 0.006 | 0.698 | 0.052 | Maillard reaction inhibitor | 0.052 0.041 CHEMBL3544524 | CHEMBL3544524 | |
| 0.019 | 0.715 | 0.817 | Angiogenesis inhibitor | 0.817 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.017 | 0.716 | 0.102 | Nav1.4 sodium channel blocker | 0.102 0.073 CHEMBL3544523 0.094 0.085 CHEMBL3544524 | CHEMBL3544523 | |
| 0.062 | 0.785 | 0.138 | CC chemokine 6 receptor antagonist | 0.137 0.048 CHEMBL3544522 0.138 0.046 CHEMBL3544887 | CHEMBL3544887 | |
| 0.02 | 0.751 | 0.06 | Lipocortins synthesis agonist | 0.059 0.037 CHEMBL3544522 0.06 0.035 CHEMBL3544887 | CHEMBL3544887 | |
| 0.025 | 0.756 | 0.095 | Interleukin 12 antagonist | 0.095 0.063 CHEMBL3544887 | CHEMBL3544887 | |
| 0.008 | 0.744 | 0.088 | Uric acid excretion stimulant | 0.088 0.068 CHEMBL3544887 | CHEMBL3544887 | |
| 0.03 | 0.767 | 0.112 | Folate antagonist | 0.112 0.047 CHEMBL3544524 | CHEMBL3544524 | |
| 0.006 | 0.762 | 0.033 | Estrogen-related receptor beta antagonist | 0.033 0.02 CHEMBL1908020 | CHEMBL1908020 | |
| 0.003 | 0.764 | 0.081 | Beta tubulin antagonist | 0.081 0.029 CHEMBL3544501 | CHEMBL3544501 | |
| 0.025 | 0.791 | 0.686 | Antiinflammatory | 0.436 0.118 CHEMBL3544522 0.686 0.034 CHEMBL3544887 0.365 0.162 CHEMBL3544524 | CHEMBL3544887 | |
| 0.009 | 0.788 | 0.147 | Interleukin antagonist | 0.147 0.12 CHEMBL3544523 | CHEMBL3544523 | |
| 0.005 | 0.785 | 0.065 | Neuraminidase (influenza) inhibitor | 0.065 0.042 CHEMBL3544887 | CHEMBL3544887 | |
| 0.003 | 0.787 | 0.031 | Endothelin receptor antagonist | 0.031 0.017 CHEMBL3544524 | CHEMBL3544524 | |
| 0.003 | 0.791 | 0.022 | Endothelin A receptor antagonist | 0.022 0.014 CHEMBL3544524 | CHEMBL3544524 | |
| 0.008 | 0.798 | 0.056 | Prostaglandin F2 alpha antagonist | 0.056 0.053 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.798 | 0.336 | Selectin antagonist | 0.285 0.006 CHEMBL3544522 0.336 0.004 CHEMBL3544887 | CHEMBL3544887 | |
| 0.006 | 0.8 | 0.443 | Anticoagulant | 0.129 0.101 CHEMBL3544522 0.443 0.013 CHEMBL3544523 0.164 0.07 CHEMBL3544887 0.357 0.021 CHEMBL3544524 | CHEMBL3544523 | |
| 0.003 | 0.797 | 0.032 | Prostacyclin antagonist | 0.032 0.024 CHEMBL3544524 | CHEMBL3544524 | |
| 0.007 | 0.819 | 0.058 | Trypsin inhibitor | 0.058 0.052 CHEMBL3544523 0.058 0.055 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.819 | 0.172 | Glutamate (mGluR group I) antagonist | 0.172 0.01 CHEMBL3544524 | CHEMBL3544524 | |
| 0.003 | 0.824 | 0.244 | Plasma kallikrein inhibitor | 0.244 0.004 CHEMBL3544524 | CHEMBL3544524 | |
| 0.01 | 0.841 | 0.072 | Factor IXa inhibitor | 0.072 0.019 CHEMBL3544522 0.066 0.023 CHEMBL3544887 | CHEMBL3544522 | |
| 0.011 | 0.845 | 0.049 | Vanilloid 2 antagonist | 0.049 0.045 CHEMBL3544501 | CHEMBL3544501 | |
| 0.004 | 0.843 | 0.567 | Glutamate (mGluR) antagonist | 0.17 0.014 CHEMBL3544523 0.567 0.003 CHEMBL3544524 | CHEMBL3544524 | |
| 0.013 | 0.856 | 0.465 | Apoptosis agonist | 0.455 0.089 CHEMBL3544522 0.313 0.163 CHEMBL3638281 0.465 0.086 CHEMBL3544887 0.287 0.182 CHEMBL3544501 | CHEMBL3544887 | |
| 0.005 | 0.86 | 0.066 | Sphingosine 1-phosphate receptor 5 agonist | 0.066 0.019 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.86 | 0.236 | Kallikrein inhibitor | 0.236 0.005 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.863 | 0.104 | 5-Lipoxygenase inhibitor | 0.104 0.061 CHEMBL3544523 | CHEMBL3544523 | |
| 0.02 | 0.887 | 0.358 | Apoptosis antagonist | 0.29 0.092 CHEMBL3544522 0.358 0.052 CHEMBL3544887 | CHEMBL3544887 | |
| 0.004 | 0.874 | 0.057 | Alpha tubulin antagonist | 0.057 0.033 CHEMBL3544501 | CHEMBL3544501 | |
| 0.003 | 0.885 | 0.032 | Catechol O-methyltransferase inhibitor | 0.032 0.023 CHEMBL3548560 | CHEMBL3548560 | |
| 0.004 | 0.899 | 0.041 | VCAM-1 antagonist | 0.038 0.031 CHEMBL3544523 0.041 0.023 CHEMBL3544524 | CHEMBL3544524 | |
| 0.004 | 0.899 | 0.041 | VCAM antagonist | 0.038 0.032 CHEMBL3544523 0.041 0.023 CHEMBL3544524 | CHEMBL3544524 | |
| 0.005 | 0.9 | 0.09 | Protein 50S ribosomal subunit inhibitor | 0.077 0.021 CHEMBL3544522 0.09 0.016 CHEMBL3544887 | CHEMBL3544887 | |
| 0.005 | 0.908 | 0.316 | Nitric oxide antagonist | 0.24 0.054 CHEMBL3544522 0.316 0.037 CHEMBL3544887 | CHEMBL3544887 | |
| 0.004 | 0.915 | 0.174 | Tubulin antagonist | 0.174 0.047 CHEMBL3544501 | CHEMBL3544501 | |
| 0.004 | 0.916 | 0.115 | Estrogen receptor beta antagonist | 0.115 0.039 CHEMBL1908020 0.109 0.048 CHEMBL1908021 0.111 0.045 CHEMBL3544888 | CHEMBL1908020 | |
| 0.005 | 0.92 | 0.566 | Hypolipemic | 0.566 0.008 CHEMBL3544523 0.16 0.127 CHEMBL3544887 0.398 0.025 CHEMBL3544524 | CHEMBL3544523 | |
| 0.011 | 0.928 | 0.141 | Toll-Like receptor 4 antagonist | 0.116 0.048 CHEMBL3544522 0.141 0.026 CHEMBL3544887 0.095 0.078 CHEMBL3544524 | CHEMBL3544887 | |
| 0.006 | 0.946 | 0.069 | Glucose-6-phosphate translocase inhibitor | 0.054 0.031 CHEMBL3544522 0.069 0.017 CHEMBL3544887 | CHEMBL3544887 | |
| 0.004 | 0.953 | 0.108 | Leukotriene synthesis inhibitor | 0.108 0.022 CHEMBL3544523 | CHEMBL3544523 | |
| 0.002 | 0.954 | 0.026 | Retinoid X gamma receptor antagonist | 0.026 0.022 CHEMBL3544524 | CHEMBL3544524 | |
| 0.005 | 0.962 | 0.226 | Thrombolytic | 0.214 0.045 CHEMBL3544522 0.226 0.041 CHEMBL3544887 0.18 0.062 CHEMBL3544524 | CHEMBL3544887 | |
| 0.004 | 0.962 | 0.122 | Estrogen antagonist | 0.122 0.051 CHEMBL1908020 0.115 0.065 CHEMBL1908021 0.116 0.062 CHEMBL3544888 | CHEMBL1908020 | |
| 0.005 | 0.974 | 0.294 | Platelet adhesion inhibitor | 0.203 0.069 CHEMBL3544522 0.294 0.036 CHEMBL3544887 | CHEMBL3544887 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |