| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.716 | 0.002 | 0.716 | HIV-1 protease inhibitor | 0.686 0.002 CHEMBL3544831 0.594 0.002 CHEMBL3544832 0.5 0.003 CHEMBL3544848 0.57 0.003 CHEMBL3544628 0.662 0.002 CHEMBL317192 0.536 0.003 CHEMBL3544847 0.304 0.003 CHEMBL3544627 | ||
| 0.6 | 0.003 | 0.6 | Protease inhibitor | 0.592 0.003 CHEMBL3544831 0.513 0.004 CHEMBL3544832 0.442 0.004 CHEMBL3544848 0.522 0.004 CHEMBL3544628 0.549 0.004 CHEMBL317192 0.484 0.004 CHEMBL3544847 0.335 0.005 CHEMBL3544627 | ||
| 0.256 | 0.06 | 0.343 | Calpain inhibitor | 0.343 0.018 CHEMBL3544831 0.31 0.026 CHEMBL3544832 0.223 0.091 CHEMBL3544848 0.199 0.114 CHEMBL3544628 0.289 0.036 CHEMBL317192 | CHEMBL3544831 | |
| 0.204 | 0.024 | 0.263 | Proteasome inhibitor | 0.263 0.014 CHEMBL3544831 0.147 0.048 CHEMBL3544832 0.202 0.024 CHEMBL3544848 0.196 0.026 CHEMBL3544628 0.252 0.015 CHEMBL317192 0.155 0.044 CHEMBL3544847 0.195 0.027 CHEMBL3544627 | CHEMBL3544831 | |
| 0.129 | 0.017 | 0.145 | Alpha 2d adrenoreceptor antagonist | 0.125 0.02 CHEMBL3544832 0.145 0.01 CHEMBL3544848 0.088 0.075 CHEMBL3544628 0.127 0.019 CHEMBL317192 0.119 0.024 CHEMBL3544847 0.1 0.049 CHEMBL3544627 | CHEMBL3544848 | |
| 0.119 | 0.013 | 0.161 | Cathepsin D inhibitor | 0.161 0.007 CHEMBL3544831 0.109 0.016 CHEMBL3544832 0.118 0.013 CHEMBL3544848 0.116 0.014 CHEMBL3544628 0.127 0.011 CHEMBL317192 0.11 0.015 CHEMBL3544847 0.114 0.014 CHEMBL3544627 | CHEMBL3544831 | |
| 0.24 | 0.138 | 0.325 | Apoptosis antagonist | 0.325 0.069 CHEMBL3544831 0.239 0.139 CHEMBL3544628 0.249 0.128 CHEMBL317192 0.205 0.172 CHEMBL3544847 | CHEMBL3544831 | |
| 0.086 | 0.008 | 0.176 | Renin inhibitor | 0.176 0.004 CHEMBL3544831 0.07 0.01 CHEMBL3544832 0.08 0.009 CHEMBL3544848 0.086 0.008 CHEMBL3544628 0.094 0.007 CHEMBL317192 0.067 0.011 CHEMBL3544847 0.079 0.009 CHEMBL3544627 | CHEMBL3544831 | |
| 0.124 | 0.049 | 0.15 | Nav1.4 sodium channel blocker | 0.15 0.034 CHEMBL3544831 0.118 0.054 CHEMBL3544832 0.125 0.048 CHEMBL3544848 0.109 0.063 CHEMBL3544628 0.129 0.045 CHEMBL317192 0.121 0.051 CHEMBL3544847 0.107 0.067 CHEMBL3544627 | CHEMBL3544831 | |
| 0.085 | 0.019 | 0.109 | Cathepsin E inhibitor | 0.109 0.011 CHEMBL3544831 0.078 0.024 CHEMBL3544832 0.088 0.018 CHEMBL3544848 0.081 0.021 CHEMBL3544628 0.09 0.017 CHEMBL317192 0.078 0.023 CHEMBL3544847 0.083 0.02 CHEMBL3544627 | CHEMBL3544831 | |
| 0.086 | 0.021 | 0.116 | Human rhinovirus A protease inhibitor | 0.116 0.013 CHEMBL3544831 0.073 0.027 CHEMBL3544832 0.083 0.022 CHEMBL3544848 0.081 0.023 CHEMBL3544628 0.082 0.023 CHEMBL317192 0.066 0.031 CHEMBL3544847 0.076 0.025 CHEMBL3544627 | CHEMBL3544831 | |
| 0.16 | 0.102 | 0.16 | P-glycoprotein inhibitor | 0.158 0.105 CHEMBL3544848 0.149 0.119 CHEMBL317192 | ||
| 0.07 | 0.021 | 0.084 | Endothelin-converting enzyme inhibitor | 0.084 0.017 CHEMBL3544831 0.063 0.023 CHEMBL3544832 0.07 0.021 CHEMBL3544848 0.064 0.023 CHEMBL3544628 0.063 0.023 CHEMBL317192 0.057 0.026 CHEMBL3544847 0.063 0.023 CHEMBL3544627 | CHEMBL3544831 | |
| 0.091 | 0.045 | 0.106 | 3C-Like protease (SARS coronavirus) inhibitor | 0.106 0.028 CHEMBL3544831 0.085 0.056 CHEMBL3544832 0.087 0.052 CHEMBL3544848 0.087 0.052 CHEMBL3544628 0.093 0.041 CHEMBL317192 0.085 0.055 CHEMBL3544847 0.082 0.063 CHEMBL3544627 | CHEMBL3544831 | |
| 0.103 | 0.062 | 0.129 | Factor V inhibitor | 0.129 0.031 CHEMBL3544831 0.099 0.072 CHEMBL3544832 0.104 0.061 CHEMBL3544848 0.105 0.059 CHEMBL3544628 0.116 0.043 CHEMBL317192 0.099 0.071 CHEMBL3544847 0.106 0.057 CHEMBL3544627 | CHEMBL3544831 | |
| 0.199 | 0.16 | 0.24 | Nootropic | 0.24 0.117 CHEMBL3544831 | CHEMBL3544831 | |
| 0.07 | 0.031 | 0.093 | Caspase 9 inhibitor | 0.093 0.016 CHEMBL3544831 0.066 0.037 CHEMBL3544832 0.061 0.046 CHEMBL3544848 0.065 0.038 CHEMBL3544628 0.073 0.029 CHEMBL317192 0.067 0.036 CHEMBL3544847 | CHEMBL3544831 | |
| 0.067 | 0.03 | 0.106 | Cathepsin B inhibitor | 0.106 0.014 CHEMBL3544831 0.062 0.034 CHEMBL3544832 0.052 0.046 CHEMBL3544848 0.063 0.033 CHEMBL3544628 0.082 0.023 CHEMBL317192 0.062 0.033 CHEMBL3544847 | CHEMBL3544831 | |
| 0.045 | 0.014 | 0.081 | Caspase 2 inhibitor | 0.081 0.006 CHEMBL3544831 0.042 0.015 CHEMBL3544832 0.044 0.014 CHEMBL3544628 0.05 0.012 CHEMBL317192 0.043 0.015 CHEMBL3544847 | CHEMBL3544831 | |
| 0.074 | 0.044 | 0.13 | Secretase beta inhibitor | 0.13 0.008 CHEMBL3544831 0.095 0.021 CHEMBL3544848 0.104 0.016 CHEMBL317192 0.075 0.042 CHEMBL3544627 | CHEMBL3544831 | |
| 0.039 | 0.013 | 0.058 | Plasmepsin I inhibitor | 0.058 0.005 CHEMBL3544831 0.037 0.014 CHEMBL3544832 0.04 0.012 CHEMBL3544848 0.037 0.014 CHEMBL3544628 0.044 0.01 CHEMBL317192 0.038 0.014 CHEMBL3544847 0.038 0.014 CHEMBL3544627 | CHEMBL3544831 | |
| 0.078 | 0.054 | 0.117 | Somatostatin 1 agonist | 0.085 0.046 CHEMBL3544831 0.072 0.062 CHEMBL3544832 0.117 0.024 CHEMBL3544848 0.076 0.056 CHEMBL3544628 0.115 0.026 CHEMBL3544627 | CHEMBL3544848 | |
| 0.051 | 0.028 | 0.059 | Bombesin antagonist | 0.059 0.02 CHEMBL3544831 0.049 0.031 CHEMBL3544832 0.059 0.019 CHEMBL3544848 0.048 0.032 CHEMBL3544628 0.052 0.026 CHEMBL317192 0.049 0.03 CHEMBL3544847 0.055 0.023 CHEMBL3544627 | CHEMBL3544848 | |
| 0.078 | 0.056 | 0.116 | Chymotrypsin inhibitor | 0.116 0.027 CHEMBL3544831 0.073 0.066 CHEMBL3544832 0.076 0.06 CHEMBL3544848 0.073 0.065 CHEMBL3544628 0.087 0.046 CHEMBL317192 0.076 0.06 CHEMBL3544847 | CHEMBL3544831 | |
| 0.203 | 0.184 | 0.315 | Interleukin 2 agonist | 0.235 0.136 CHEMBL3544831 0.315 0.064 CHEMBL3544848 0.213 0.168 CHEMBL317192 0.282 0.087 CHEMBL3544627 | CHEMBL3544848 | |
| 0.064 | 0.046 | 0.088 | Glucagon-like peptide 1 agonist | 0.088 0.029 CHEMBL3544831 0.057 0.051 CHEMBL3544832 0.054 0.053 CHEMBL3544848 0.056 0.051 CHEMBL3544628 0.071 0.041 CHEMBL317192 0.06 0.048 CHEMBL3544847 | CHEMBL3544831 | |
| 0.035 | 0.018 | 0.04 | Calpain 1 inhibitor | 0.04 0.01 CHEMBL3544831 0.039 0.012 CHEMBL3544832 0.031 0.03 CHEMBL3544848 0.035 0.02 CHEMBL3544628 0.036 0.018 CHEMBL317192 0.033 0.025 CHEMBL3544847 | CHEMBL3544831 | |
| 0.057 | 0.045 | 0.086 | Bombesin 1 receptor agonist | 0.069 0.032 CHEMBL3544831 0.053 0.05 CHEMBL3544832 0.086 0.023 CHEMBL3544848 0.06 0.041 CHEMBL317192 0.054 0.049 CHEMBL3544847 0.071 0.03 CHEMBL3544627 | CHEMBL3544848 | |
| 0.037 | 0.026 | 0.046 | Bombesin 1 receptor antagonist | 0.046 0.017 CHEMBL3544831 0.034 0.029 CHEMBL3544832 0.034 0.029 CHEMBL3544848 0.038 0.024 CHEMBL317192 0.035 0.029 CHEMBL3544847 | CHEMBL3544831 | |
| 0.026 | 0.025 | 0.033 | HCV NS5A inhibitor | 0.033 0.011 CHEMBL3544831 0.026 0.023 CHEMBL317192 | CHEMBL3544831 | |
| 0.051 | 0.051 | 0.058 | Kallikrein 1 inhibitor | 0.058 0.037 CHEMBL3544831 0.053 0.047 CHEMBL317192 | CHEMBL3544831 | |
| 0.016 | 0.019 | 0.041 | Neutral endopeptidase inhibitor | 0.033 0.011 CHEMBL3544831 0.041 0.009 CHEMBL3544848 0.018 0.017 CHEMBL3544847 0.033 0.011 CHEMBL3544627 | CHEMBL3544848 | |
| 0.022 | 0.029 | 0.031 | Cathepsin K inhibitor | 0.031 0.014 CHEMBL3544831 0.025 0.022 CHEMBL317192 | CHEMBL3544831 | |
| 0.015 | 0.023 | 0.023 | Human T-cell leukemia virus type I protease inhibitor | 0.023 0.013 CHEMBL3544831 | CHEMBL3544831 | |
| 0.027 | 0.041 | 0.074 | Cathepsin L2 inhibitor | 0.074 0.012 CHEMBL3544831 0.035 0.032 CHEMBL317192 | CHEMBL3544831 | |
| 0.045 | 0.06 | 0.061 | Bombesin 3 receptor antagonist | 0.06 0.032 CHEMBL3544831 0.061 0.032 CHEMBL3544848 0.061 0.032 CHEMBL3544627 | CHEMBL3544627 | |
| 0.029 | 0.045 | 0.036 | HCV polyprotein inhibitor | 0.036 0.019 CHEMBL3544831 | CHEMBL3544831 | |
| 0.032 | 0.05 | 0.039 | Acetyl-CoA carboxylase inhibitor | 0.039 0.032 CHEMBL3544831 | CHEMBL3544831 | |
| 0.07 | 0.089 | 0.129 | Falcipain inhibitor | 0.129 0.04 CHEMBL3544831 | CHEMBL3544831 | |
| 0.046 | 0.07 | 0.06 | Protease activated receptor antagonist | 0.058 0.05 CHEMBL3544848 0.06 0.047 CHEMBL317192 0.06 0.047 CHEMBL3544627 | CHEMBL3544627 | |
| 0.026 | 0.052 | 0.034 | Tubulin agonist | 0.033 0.027 CHEMBL3544848 0.034 0.025 CHEMBL3544627 | CHEMBL3544627 | |
| 0.043 | 0.07 | 0.05 | Angiotensin-converting enzyme inhibitor | 0.05 0.048 CHEMBL3544831 0.05 0.046 CHEMBL3544848 | CHEMBL3544848 | |
| 0.036 | 0.07 | 0.11 | Aminopeptidase microsomal inhibitor | 0.079 0.026 CHEMBL3544831 0.11 0.015 CHEMBL3544848 0.073 0.029 CHEMBL317192 0.051 0.046 CHEMBL3544847 0.102 0.017 CHEMBL3544627 | CHEMBL3544848 | |
| 0.062 | 0.101 | 0.112 | Falcipain 2 inhibitor | 0.112 0.045 CHEMBL3544831 | CHEMBL3544831 | |
| 0.046 | 0.089 | 0.058 | Gonadotropin-releasing hormone receptor agonist | 0.058 0.044 CHEMBL3544848 0.057 0.046 CHEMBL3544627 | CHEMBL3544848 | |
| 0.025 | 0.068 | 0.092 | Aminopeptidase N inhibitor | 0.059 0.025 CHEMBL3544831 0.092 0.015 CHEMBL3544848 0.054 0.028 CHEMBL317192 0.084 0.016 CHEMBL3544627 | CHEMBL3544848 | |
| 0.032 | 0.076 | 0.039 | Cathepsin F inhibitor | 0.039 0.037 CHEMBL3544848 | CHEMBL3544848 | |
| 0.038 | 0.082 | 0.052 | Carbonic anhydrase II stimulant | 0.052 0.035 CHEMBL3544848 0.049 0.042 CHEMBL3544627 | CHEMBL3544848 | |
| 0.034 | 0.085 | 0.05 | Elastase inhibitor | 0.05 0.042 CHEMBL3544831 | CHEMBL3544831 | |
| 0.02 | 0.071 | 0.037 | Carbonic anhydrase I stimulant | 0.037 0.027 CHEMBL3544848 | CHEMBL3544848 | |
| 0.04 | 0.092 | 0.058 | Acetyl-CoA transferase 2 inhibitor | 0.057 0.039 CHEMBL3544848 0.058 0.036 CHEMBL3544627 | CHEMBL3544627 | |
| 0.033 | 0.094 | 0.047 | HCV NS3/NS4A protease inhibitor | 0.047 0.039 CHEMBL3544831 | CHEMBL3544831 | |
| 0.007 | 0.094 | 0.052 | Aminopeptidase P inhibitor | 0.052 0.004 CHEMBL3544848 0.05 0.004 CHEMBL3544627 | CHEMBL3544848 | |
| 0.077 | 0.164 | 0.106 | Cell adhesion inhibitor | 0.106 0.079 CHEMBL3544848 | CHEMBL3544848 | |
| 0.092 | 0.188 | 0.177 | Growth hormone agonist | 0.149 0.088 CHEMBL3544831 0.17 0.073 CHEMBL3544848 0.177 0.069 CHEMBL3544627 | CHEMBL3544627 | |
| 0.057 | 0.184 | 0.116 | Histone deacetylase class III inhibitor | 0.116 0.073 CHEMBL3544831 | CHEMBL3544831 | |
| 0.071 | 0.205 | 0.145 | Angiogenesis stimulant | 0.139 0.129 CHEMBL3544831 0.136 0.131 CHEMBL3544848 0.145 0.126 CHEMBL3544627 | CHEMBL3544627 | |
| 0.082 | 0.216 | 0.221 | Thiol protease inhibitor | 0.221 0.033 CHEMBL3544831 0.165 0.058 CHEMBL317192 | CHEMBL3544831 | |
| 0.121 | 0.277 | 0.405 | Calpain 2 inhibitor | 0.405 0.059 CHEMBL3544831 0.315 0.105 CHEMBL317192 | CHEMBL3544831 | |
| 0.055 | 0.225 | 0.103 | Microtubule formation inhibitor | 0.103 0.085 CHEMBL3544848 | CHEMBL3544848 | |
| 0.031 | 0.211 | 0.075 | Protease 3C (Human rhinovirus) inhibitor | 0.075 0.031 CHEMBL3544831 | CHEMBL3544831 | |
| 0.03 | 0.212 | 0.067 | Analgesic, opioid | 0.067 0.066 CHEMBL3544627 | CHEMBL3544627 | |
| 0.035 | 0.221 | 0.086 | Opioid antagonist | 0.086 0.062 CHEMBL3544848 0.085 0.062 CHEMBL3544627 | CHEMBL3544848 | |
| 0.005 | 0.195 | 0.175 | Follicle-stimulating hormone agonist | 0.175 0.003 CHEMBL3544832 | CHEMBL3544832 | |
| 0.07 | 0.274 | 0.134 | Interleukin antagonist | 0.134 0.132 CHEMBL3544848 | CHEMBL3544848 | |
| 0.045 | 0.258 | 0.122 | Thrombolytic | 0.122 0.108 CHEMBL3544831 | CHEMBL3544831 | |
| 0.011 | 0.242 | 0.069 | Cathepsin L inhibitor | 0.069 0.03 CHEMBL3544831 | CHEMBL3544831 | |
| 0.014 | 0.259 | 0.04 | Plasmepsin II inhibitor | 0.04 0.031 CHEMBL3544831 | CHEMBL3544831 | |
| 0.005 | 0.263 | 0.041 | Cathepsin L1 inhibitor | 0.041 0.025 CHEMBL3544831 | CHEMBL3544831 | |
| 0.006 | 0.273 | 0.059 | Ribonucleoside-diphosphate reductase inhibitor | 0.059 0.035 CHEMBL3544831 0.056 0.036 CHEMBL3544848 | CHEMBL3544831 | |
| 0.005 | 0.277 | 0.076 | Ribonucleotide reductase inhibitor | 0.076 0.028 CHEMBL3544831 0.056 0.039 CHEMBL3544848 | CHEMBL3544831 | |
| 0.008 | 0.321 | 0.102 | Follicle-stimulating hormone antagonist | 0.102 0.002 CHEMBL3544832 | CHEMBL3544832 | |
| 0.101 | 0.418 | 0.167 | Peptidyltransferase inhibitor | 0.163 0.162 CHEMBL3544848 0.167 0.154 CHEMBL3544627 | CHEMBL3544627 | |
| 0.015 | 0.335 | 0.146 | Leukotriene synthesis inhibitor | 0.146 0.01 CHEMBL3544847 | CHEMBL3544847 | |
| 0.031 | 0.4 | 0.182 | Cathepsin H inhibitor | 0.182 0.028 CHEMBL3544831 0.114 0.084 CHEMBL3544848 | CHEMBL3544831 | |
| 0.07 | 0.48 | 0.384 | Toll-Like receptor agonist | 0.298 0.112 CHEMBL3544628 0.384 0.067 CHEMBL3544847 0.333 0.091 CHEMBL3544627 | CHEMBL3544847 | |
| 0.06 | 0.472 | 0.242 | Antithrombotic | 0.242 0.133 CHEMBL3544831 | CHEMBL3544831 | |
| 0.07 | 0.484 | 0.381 | Toll-Like receptor 7 agonist | 0.295 0.113 CHEMBL3544628 0.381 0.068 CHEMBL3544847 0.323 0.096 CHEMBL3544627 | CHEMBL3544847 | |
| 0.009 | 0.425 | 0.071 | Catalase inhibitor | 0.071 0.054 CHEMBL3544831 | CHEMBL3544831 | |
| 0.019 | 0.487 | 0.086 | Interleukin 1 beta converting enzyme inhibitor | 0.086 0.079 CHEMBL3544831 | CHEMBL3544831 | |
| 0.011 | 0.484 | 0.067 | Carbonic anhydrase stimulant | 0.067 0.034 CHEMBL3544848 | CHEMBL3544848 | |
| 0.015 | 0.601 | 0.152 | Aminopeptidase B inhibitor | 0.152 0.037 CHEMBL3544848 0.138 0.043 CHEMBL3544627 | CHEMBL3544848 | |
| 0.006 | 0.621 | 0.316 | 5-Lipoxygenase inhibitor | 0.316 0.009 CHEMBL3544847 | CHEMBL3544847 | |
| 0.013 | 0.647 | 0.176 | Immunostimulant | 0.176 0.135 CHEMBL3544848 0.175 0.136 CHEMBL3544627 | CHEMBL3544848 | |
| 0.017 | 0.659 | 0.054 | Immunoglobulin Fc receptor antagonist | 0.054 0.043 CHEMBL3544848 | CHEMBL3544848 | |
| 0.007 | 0.662 | 0.081 | Aminopeptidase I inhibitor | 0.081 0.041 CHEMBL3544848 0.073 0.049 CHEMBL3544627 | CHEMBL3544848 | |
| 0.014 | 0.85 | 0.191 | Insulysin inhibitor | 0.191 0.171 CHEMBL3544848 | CHEMBL3544848 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |