| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.64 | 0.013 | 0.64 | Toll-Like receptor 7 agonist | 0.401 0.06 CHEMBL3527592 0.64 0.013 CHEMBL1630842 0.412 0.055 CHEMBL3527593 | ||
| 0.639 | 0.013 | 0.639 | Toll-Like receptor agonist | 0.406 0.058 CHEMBL3527592 0.639 0.013 CHEMBL1630842 0.419 0.053 CHEMBL3527593 | ||
| 0.531 | 0.004 | 0.559 | HIV-1 reverse transcriptase inhibitor | 0.544 0.004 CHEMBL3527592 0.531 0.004 CHEMBL1630842 0.559 0.004 CHEMBL3527593 | CHEMBL3527593 | |
| 0.492 | 0.004 | 0.492 | Phosphodiesterase IV inhibitor | 0.257 0.007 CHEMBL3527592 0.492 0.004 CHEMBL1630842 0.177 0.016 CHEMBL3527593 | ||
| 0.4 | 0.019 | 0.4 | Platelet aggregation inhibitor | 0.312 0.033 CHEMBL3527592 0.4 0.019 CHEMBL1630842 0.197 0.083 CHEMBL3527593 | ||
| 0.417 | 0.049 | 0.42 | MAP kinase kinase 6 inhibitor | 0.42 0.047 CHEMBL3527592 0.417 0.049 CHEMBL1630842 0.395 0.061 CHEMBL3527593 | CHEMBL3527592 | |
| 0.383 | 0.024 | 0.383 | Anticonvulsant | 0.206 0.078 CHEMBL3527592 0.383 0.024 CHEMBL1630842 0.235 0.063 CHEMBL3527593 | ||
| 0.318 | 0.013 | 0.318 | Phosphodiesterase inhibitor | 0.25 0.022 CHEMBL3527592 0.318 0.013 CHEMBL1630842 0.215 0.03 CHEMBL3527593 | ||
| 0.338 | 0.037 | 0.338 | Vasodilator | 0.338 0.037 CHEMBL1630842 | ||
| 0.297 | 0.009 | 0.297 | Bronchodilator | 0.118 0.046 CHEMBL3527592 0.297 0.009 CHEMBL1630842 0.133 0.038 CHEMBL3527593 | ||
| 0.255 | 0.009 | 0.268 | DNA directed RNA polymerase inhibitor | 0.223 0.011 CHEMBL3527592 0.255 0.009 CHEMBL1630842 0.268 0.008 CHEMBL3527593 | CHEMBL3527593 | |
| 0.246 | 0.017 | 0.246 | Platelet activating factor antagonist | 0.202 0.025 CHEMBL3527592 0.246 0.017 CHEMBL1630842 0.113 0.068 CHEMBL3527593 | ||
| 0.279 | 0.062 | 0.279 | Tumour necrosis factor alpha release inhibitor | 0.213 0.098 CHEMBL3527592 0.279 0.062 CHEMBL1630842 | ||
| 0.177 | 0.01 | 0.177 | Phosphodiesterase 4B inhibitor | 0.072 0.042 CHEMBL3527592 0.177 0.01 CHEMBL1630842 | ||
| 0.218 | 0.077 | 0.389 | RNA-directed DNA polymerase inhibitor | 0.275 0.038 CHEMBL3527592 0.218 0.077 CHEMBL1630842 0.389 0.019 CHEMBL3527593 | CHEMBL3527593 | |
| 0.139 | 0.008 | 0.357 | Phosphodiesterase VI inhibitor | 0.357 0.003 CHEMBL3527592 0.139 0.008 CHEMBL1630842 0.296 0.003 CHEMBL3527593 | CHEMBL3527592 | |
| 0.126 | 0.011 | 0.126 | Dopamine D4 agonist | 0.126 0.011 CHEMBL1630842 | ||
| 0.119 | 0.013 | 0.119 | Phosphodiesterase 4A inhibitor | 0.119 0.013 CHEMBL1630842 | ||
| 0.141 | 0.041 | 0.18 | GABA receptor agonist | 0.18 0.023 CHEMBL3527592 0.141 0.041 CHEMBL1630842 0.169 0.027 CHEMBL3527593 | CHEMBL3527592 | |
| 0.116 | 0.026 | 0.154 | GABA A receptor agonist | 0.154 0.015 CHEMBL3527592 0.116 0.026 CHEMBL1630842 0.116 0.026 CHEMBL3527593 | CHEMBL3527592 | |
| 0.111 | 0.023 | 0.152 | Phosphodiesterase V inhibitor | 0.152 0.01 CHEMBL3527592 0.111 0.023 CHEMBL1630842 0.139 0.013 CHEMBL3527593 | CHEMBL3527592 | |
| 0.11 | 0.022 | 0.154 | Phosphodiesterase 5A inhibitor | 0.154 0.01 CHEMBL3527592 0.11 0.022 CHEMBL1630842 0.138 0.013 CHEMBL3527593 | CHEMBL3527592 | |
| 0.106 | 0.022 | 0.106 | Benzodiazepine agonist | 0.063 0.062 CHEMBL3527592 0.106 0.022 CHEMBL1630842 | ||
| 0.119 | 0.036 | 0.171 | Hepatocyte growth factor antagonist | 0.171 0.017 CHEMBL3527592 0.119 0.036 CHEMBL1630842 0.093 0.06 CHEMBL3527593 | CHEMBL3527592 | |
| 0.105 | 0.035 | 0.105 | Phosphodiesterase 4D inhibitor | 0.067 0.058 CHEMBL3527592 0.105 0.035 CHEMBL1630842 | ||
| 0.138 | 0.071 | 0.138 | Neurotrophic factor | 0.118 0.099 CHEMBL3527592 0.138 0.071 CHEMBL1630842 | ||
| 0.081 | 0.02 | 0.081 | Phosphodiesterase 4C inhibitor | 0.057 0.038 CHEMBL3527592 0.081 0.02 CHEMBL1630842 | ||
| 0.206 | 0.15 | 0.206 | Nootropic | 0.206 0.15 CHEMBL1630842 | ||
| 0.096 | 0.043 | 0.096 | Histamine H1 receptor antagonist | 0.096 0.043 CHEMBL1630842 | ||
| 0.082 | 0.034 | 0.122 | Phosphodiesterase III inhibitor | 0.1 0.022 CHEMBL3527592 0.082 0.034 CHEMBL1630842 0.122 0.015 CHEMBL3527593 | CHEMBL3527593 | |
| 0.082 | 0.042 | 0.11 | Polo-like kinase-2 inhibitor | 0.108 0.018 CHEMBL3527592 0.082 0.042 CHEMBL1630842 0.11 0.017 CHEMBL3527593 | CHEMBL3527593 | |
| 0.051 | 0.023 | 0.055 | Benzodiazepine inverse agonist | 0.051 0.024 CHEMBL3527592 0.051 0.023 CHEMBL1630842 0.055 0.019 CHEMBL3527593 | CHEMBL3527593 | |
| 0.07 | 0.044 | 0.07 | Dopamine agonist | 0.07 0.044 CHEMBL1630842 | ||
| 0.107 | 0.081 | 0.132 | Sphingosine 1-phosphate receptor 2 agonist | 0.132 0.039 CHEMBL3527592 0.107 0.081 CHEMBL1630842 0.122 0.052 CHEMBL3527593 | CHEMBL3527592 | |
| 0.075 | 0.05 | 0.075 | MAP kinase 14 inhibitor | 0.075 0.05 CHEMBL1630842 | ||
| 0.199 | 0.177 | 0.319 | Vasodilator, peripheral | 0.199 0.177 CHEMBL1630842 0.319 0.088 CHEMBL3527593 | CHEMBL3527593 | |
| 0.055 | 0.035 | 0.059 | GABA A receptor antagonist | 0.059 0.032 CHEMBL3527592 0.055 0.035 CHEMBL1630842 0.047 0.045 CHEMBL3527593 | CHEMBL3527592 | |
| 0.051 | 0.032 | 0.063 | Adenosine A2b receptor antagonist | 0.053 0.03 CHEMBL3527592 0.051 0.032 CHEMBL1630842 0.063 0.022 CHEMBL3527593 | CHEMBL3527593 | |
| 0.123 | 0.104 | 0.155 | Death-associated protein kinase 1 inhibitor | 0.132 0.077 CHEMBL3527592 0.123 0.104 CHEMBL1630842 0.155 0.033 CHEMBL3527593 | CHEMBL3527593 | |
| 0.033 | 0.014 | 0.038 | Thiazolidinedione | 0.038 0.009 CHEMBL3527592 0.033 0.014 CHEMBL1630842 0.036 0.01 CHEMBL3527593 | CHEMBL3527592 | |
| 0.076 | 0.059 | 0.088 | MAP kinase 7 inhibitor | 0.088 0.022 CHEMBL3527592 0.076 0.059 CHEMBL1630842 0.086 0.028 CHEMBL3527593 | CHEMBL3527592 | |
| 0.027 | 0.01 | 0.033 | Phosphodiesterase 6A inhibitor | 0.033 0.005 CHEMBL3527592 0.027 0.01 CHEMBL1630842 0.03 0.007 CHEMBL3527593 | CHEMBL3527592 | |
| 0.047 | 0.03 | 0.052 | Phosphodiesterase 6C inhibitor | 0.052 0.017 CHEMBL3527592 0.047 0.03 CHEMBL1630842 0.052 0.017 CHEMBL3527593 | CHEMBL3527593 | |
| 0.058 | 0.05 | 0.076 | Adenosine A2 receptor antagonist | 0.076 0.037 CHEMBL3527592 0.058 0.05 CHEMBL1630842 0.073 0.038 CHEMBL3527593 | CHEMBL3527592 | |
| 0.045 | 0.037 | 0.066 | Proto-oncogene tyrosine-protein kinase Met inhibitor | 0.066 0.023 CHEMBL3527592 0.045 0.037 CHEMBL1630842 | CHEMBL3527592 | |
| 0.076 | 0.072 | 0.13 | Caspase 7 inhibitor | 0.13 0.012 CHEMBL3527592 0.076 0.072 CHEMBL1630842 0.109 0.02 CHEMBL3527593 | CHEMBL3527592 | |
| 0.056 | 0.053 | 0.099 | Phosphodiesterase 1A inhibitor | 0.099 0.01 CHEMBL3527592 0.056 0.053 CHEMBL1630842 0.076 0.019 CHEMBL3527593 | CHEMBL3527592 | |
| 0.049 | 0.048 | 0.107 | Bromodomain-containing protein 4 inhibitor | 0.073 0.022 CHEMBL3527592 0.049 0.048 CHEMBL1630842 0.107 0.012 CHEMBL3527593 | CHEMBL3527593 | |
| 0.085 | 0.084 | 0.102 | Interleukin 12 antagonist | 0.102 0.05 CHEMBL3527592 0.085 0.084 CHEMBL1630842 0.099 0.055 CHEMBL3527593 | CHEMBL3527592 | |
| 0.048 | 0.048 | 0.052 | GABA receptor antagonist | 0.052 0.041 CHEMBL3527592 | CHEMBL3527592 | |
| 0.12 | 0.125 | 0.148 | Polo-like kinase-3 inhibitor | 0.141 0.094 CHEMBL3527592 0.148 0.086 CHEMBL3527593 | CHEMBL3527593 | |
| 0.047 | 0.056 | 0.074 | Phosphodiesterase II inhibitor | 0.072 0.022 CHEMBL3527592 0.074 0.021 CHEMBL3527593 | CHEMBL3527593 | |
| 0.025 | 0.041 | 0.047 | Glutamate (mGluR group II) agonist | 0.047 0.017 CHEMBL3527592 | CHEMBL3527592 | |
| 0.1 | 0.117 | 0.12 | Ribosomal protein S6 kinase inhibitor | 0.12 0.09 CHEMBL3527592 0.116 0.095 CHEMBL3527593 | CHEMBL3527592 | |
| 0.022 | 0.039 | 0.044 | Glutamate (mGluR2) agonist | 0.044 0.016 CHEMBL3527592 | CHEMBL3527592 | |
| 0.038 | 0.058 | 0.062 | Phosphodiesterase 2A inhibitor | 0.061 0.023 CHEMBL3527592 0.062 0.022 CHEMBL3527593 | CHEMBL3527593 | |
| 0.177 | 0.199 | 0.21 | Angiogenesis inhibitor | 0.21 0.158 CHEMBL3527592 | CHEMBL3527592 | |
| 0.035 | 0.06 | 0.043 | Glutamate (mGluR group III) antagonist | 0.043 0.031 CHEMBL3527592 0.043 0.033 CHEMBL3527593 | CHEMBL3527593 | |
| 0.055 | 0.08 | 0.081 | Glutamate (mGluR7) antagonist | 0.081 0.027 CHEMBL3527592 | CHEMBL3527592 | |
| 0.066 | 0.092 | 0.131 | Proto-oncogene tyrosine-protein kinase Kit inhibitor | 0.131 0.04 CHEMBL3527592 | CHEMBL3527592 | |
| 0.08 | 0.109 | 0.132 | Phosphodiesterase 6D inhibitor | 0.132 0.016 CHEMBL3527592 0.126 0.02 CHEMBL3527593 | CHEMBL3527592 | |
| 0.252 | 0.284 | 0.389 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.361 0.138 CHEMBL3527592 0.389 0.111 CHEMBL3527593 | CHEMBL3527593 | |
| 0.065 | 0.103 | 0.153 | Platelet activating factor alpha antagonist | 0.153 0.029 CHEMBL3527592 | CHEMBL3527592 | |
| 0.175 | 0.213 | 0.204 | MAP kinase kinase 3 inhibitor | 0.204 0.111 CHEMBL3527592 0.192 0.146 CHEMBL3527593 | CHEMBL3527592 | |
| 0.055 | 0.097 | 0.13 | Platelet growth factor antagonist | 0.13 0.025 CHEMBL3527592 0.086 0.051 CHEMBL3527593 | CHEMBL3527592 | |
| 0.068 | 0.122 | 0.105 | Polo-like kinase-4 inhibitor | 0.105 0.072 CHEMBL3527593 | CHEMBL3527593 | |
| 0.023 | 0.079 | 0.046 | Phosphodiesterase 3B inhibitor | 0.046 0.028 CHEMBL3527593 | CHEMBL3527593 | |
| 0.034 | 0.09 | 0.075 | Glutamate (mGluR) agonist | 0.075 0.033 CHEMBL3527592 | CHEMBL3527592 | |
| 0.06 | 0.122 | 0.157 | Mediator release inhibitor | 0.135 0.036 CHEMBL3527592 0.157 0.026 CHEMBL3527593 | CHEMBL3527593 | |
| 0.03 | 0.098 | 0.054 | Adenosine A2a receptor antagonist | 0.054 0.051 CHEMBL3527592 | CHEMBL3527592 | |
| 0.023 | 0.095 | 0.037 | Acid-sensing ion channel blocker | 0.037 0.034 CHEMBL3527593 | CHEMBL3527593 | |
| 0.037 | 0.114 | 0.105 | Phosphodiesterase 1B inhibitor | 0.105 0.013 CHEMBL3527592 0.062 0.039 CHEMBL3527593 | CHEMBL3527592 | |
| 0.044 | 0.124 | 0.087 | Phosphodiesterase 1C inhibitor | 0.087 0.015 CHEMBL3527592 | CHEMBL3527592 | |
| 0.047 | 0.128 | 0.077 | ALK inhibitor | 0.077 0.064 CHEMBL3527592 0.075 0.067 CHEMBL3527593 | CHEMBL3527592 | |
| 0.066 | 0.158 | 0.084 | Toll-Like receptor 3 antagonist | 0.084 0.083 CHEMBL3527593 | CHEMBL3527593 | |
| 0.121 | 0.216 | 0.348 | Cyclic AMP phosphodiesterase inhibitor | 0.293 0.045 CHEMBL3527592 0.348 0.026 CHEMBL3527593 | CHEMBL3527593 | |
| 0.056 | 0.153 | 0.125 | Phosphodiesterase I inhibitor | 0.125 0.024 CHEMBL3527592 0.115 0.03 CHEMBL3527593 | CHEMBL3527592 | |
| 0.164 | 0.263 | 0.343 | GABA C receptor rho-3 antagonist | 0.343 0.09 CHEMBL3527592 0.315 0.106 CHEMBL3527593 | CHEMBL3527592 | |
| 0.029 | 0.142 | 0.054 | 5 Hydroxytryptamine 1B agonist | 0.054 0.035 CHEMBL3527593 | CHEMBL3527593 | |
| 0.059 | 0.175 | 0.172 | Vascular endothelial growth factor 3 antagonist | 0.172 0.053 CHEMBL3527592 | CHEMBL3527592 | |
| 0.049 | 0.165 | 0.076 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.076 0.071 CHEMBL3527593 | CHEMBL3527593 | |
| 0.055 | 0.176 | 0.125 | Bromodomain-containing protein 2 inhibitor | 0.125 0.02 CHEMBL3527592 0.114 0.027 CHEMBL3527593 | CHEMBL3527592 | |
| 0.065 | 0.186 | 0.119 | Growth factor antagonist | 0.119 0.093 CHEMBL3527592 | CHEMBL3527592 | |
| 0.093 | 0.237 | 0.139 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.139 0.094 CHEMBL3527593 | CHEMBL3527593 | |
| 0.044 | 0.23 | 0.084 | Interleukin 1 beta converting enzyme inhibitor | 0.084 0.082 CHEMBL3527592 | CHEMBL3527592 | |
| 0.068 | 0.259 | 0.123 | Aurora-C kinase inhibitor | 0.123 0.099 CHEMBL3527593 | CHEMBL3527593 | |
| 0.018 | 0.236 | 0.056 | mTOR inhibitor | 0.056 0.032 CHEMBL3527593 | CHEMBL3527593 | |
| 0.049 | 0.275 | 0.144 | Activin receptor-like kinase 2 inhibitor | 0.144 0.072 CHEMBL3527592 0.118 0.098 CHEMBL3527593 | CHEMBL3527592 | |
| 0.067 | 0.309 | 0.129 | GABA C receptor rho-2 antagonist | 0.129 0.108 CHEMBL3527592 | CHEMBL3527592 | |
| 0.015 | 0.259 | 0.085 | Glutamate receptor agonist | 0.085 0.048 CHEMBL3527592 | CHEMBL3527592 | |
| 0.145 | 0.396 | 0.207 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.207 0.147 CHEMBL3527593 | CHEMBL3527593 | |
| 0.109 | 0.386 | 0.272 | Histamine release inhibitor | 0.272 0.14 CHEMBL3527592 0.224 0.177 CHEMBL3527593 | CHEMBL3527592 | |
| 0.079 | 0.387 | 0.15 | Death-associated protein kinase 2 inhibitor | 0.15 0.106 CHEMBL3527593 | CHEMBL3527593 | |
| 0.013 | 0.364 | 0.042 | Nicotinic acid receptor 1 agonist | 0.042 0.026 CHEMBL3527593 | CHEMBL3527593 | |
| 0.082 | 0.446 | 0.143 | Cyclin-dependent kinase 3 inhibitor | 0.143 0.113 CHEMBL3527593 | CHEMBL3527593 | |
| 0.034 | 0.404 | 0.117 | Acetylcholine M1 receptor antagonist | 0.117 0.113 CHEMBL3527593 | CHEMBL3527593 | |
| 0.076 | 0.491 | 0.201 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.201 0.156 CHEMBL3527593 | CHEMBL3527593 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |