Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.640.0130.64Toll-Like receptor 7 agonist

0.401 0.06 CHEMBL3527592

0.64 0.013 CHEMBL1630842

0.412 0.055 CHEMBL3527593

0.6390.0130.639Toll-Like receptor agonist

0.406 0.058 CHEMBL3527592

0.639 0.013 CHEMBL1630842

0.419 0.053 CHEMBL3527593

0.5310.0040.559HIV-1 reverse transcriptase inhibitor

0.544 0.004 CHEMBL3527592

0.531 0.004 CHEMBL1630842

0.559 0.004 CHEMBL3527593

CHEMBL3527593
0.4920.0040.492Phosphodiesterase IV inhibitor

0.257 0.007 CHEMBL3527592

0.492 0.004 CHEMBL1630842

0.177 0.016 CHEMBL3527593

0.40.0190.4Platelet aggregation inhibitor

0.312 0.033 CHEMBL3527592

0.4 0.019 CHEMBL1630842

0.197 0.083 CHEMBL3527593

0.4170.0490.42MAP kinase kinase 6 inhibitor

0.42 0.047 CHEMBL3527592

0.417 0.049 CHEMBL1630842

0.395 0.061 CHEMBL3527593

CHEMBL3527592
0.3830.0240.383Anticonvulsant

0.206 0.078 CHEMBL3527592

0.383 0.024 CHEMBL1630842

0.235 0.063 CHEMBL3527593

0.3180.0130.318Phosphodiesterase inhibitor

0.25 0.022 CHEMBL3527592

0.318 0.013 CHEMBL1630842

0.215 0.03 CHEMBL3527593

0.3380.0370.338Vasodilator

0.338 0.037 CHEMBL1630842

0.2970.0090.297Bronchodilator

0.118 0.046 CHEMBL3527592

0.297 0.009 CHEMBL1630842

0.133 0.038 CHEMBL3527593

0.2550.0090.268DNA directed RNA polymerase inhibitor

0.223 0.011 CHEMBL3527592

0.255 0.009 CHEMBL1630842

0.268 0.008 CHEMBL3527593

CHEMBL3527593
0.2460.0170.246Platelet activating factor antagonist

0.202 0.025 CHEMBL3527592

0.246 0.017 CHEMBL1630842

0.113 0.068 CHEMBL3527593

0.2790.0620.279Tumour necrosis factor alpha release inhibitor

0.213 0.098 CHEMBL3527592

0.279 0.062 CHEMBL1630842

0.1770.010.177Phosphodiesterase 4B inhibitor

0.072 0.042 CHEMBL3527592

0.177 0.01 CHEMBL1630842

0.2180.0770.389RNA-directed DNA polymerase inhibitor

0.275 0.038 CHEMBL3527592

0.218 0.077 CHEMBL1630842

0.389 0.019 CHEMBL3527593

CHEMBL3527593
0.1390.0080.357Phosphodiesterase VI inhibitor

0.357 0.003 CHEMBL3527592

0.139 0.008 CHEMBL1630842

0.296 0.003 CHEMBL3527593

CHEMBL3527592
0.1260.0110.126Dopamine D4 agonist

0.126 0.011 CHEMBL1630842

0.1190.0130.119Phosphodiesterase 4A inhibitor

0.119 0.013 CHEMBL1630842

0.1410.0410.18GABA receptor agonist

0.18 0.023 CHEMBL3527592

0.141 0.041 CHEMBL1630842

0.169 0.027 CHEMBL3527593

CHEMBL3527592
0.1160.0260.154GABA A receptor agonist

0.154 0.015 CHEMBL3527592

0.116 0.026 CHEMBL1630842

0.116 0.026 CHEMBL3527593

CHEMBL3527592
0.1110.0230.152Phosphodiesterase V inhibitor

0.152 0.01 CHEMBL3527592

0.111 0.023 CHEMBL1630842

0.139 0.013 CHEMBL3527593

CHEMBL3527592
0.110.0220.154Phosphodiesterase 5A inhibitor

0.154 0.01 CHEMBL3527592

0.11 0.022 CHEMBL1630842

0.138 0.013 CHEMBL3527593

CHEMBL3527592
0.1060.0220.106Benzodiazepine agonist

0.063 0.062 CHEMBL3527592

0.106 0.022 CHEMBL1630842

0.1190.0360.171Hepatocyte growth factor antagonist

0.171 0.017 CHEMBL3527592

0.119 0.036 CHEMBL1630842

0.093 0.06 CHEMBL3527593

CHEMBL3527592
0.1050.0350.105Phosphodiesterase 4D inhibitor

0.067 0.058 CHEMBL3527592

0.105 0.035 CHEMBL1630842

0.1380.0710.138Neurotrophic factor

0.118 0.099 CHEMBL3527592

0.138 0.071 CHEMBL1630842

0.0810.020.081Phosphodiesterase 4C inhibitor

0.057 0.038 CHEMBL3527592

0.081 0.02 CHEMBL1630842

0.2060.150.206Nootropic

0.206 0.15 CHEMBL1630842

0.0960.0430.096Histamine H1 receptor antagonist

0.096 0.043 CHEMBL1630842

0.0820.0340.122Phosphodiesterase III inhibitor

0.1 0.022 CHEMBL3527592

0.082 0.034 CHEMBL1630842

0.122 0.015 CHEMBL3527593

CHEMBL3527593
0.0820.0420.11Polo-like kinase-2 inhibitor

0.108 0.018 CHEMBL3527592

0.082 0.042 CHEMBL1630842

0.11 0.017 CHEMBL3527593

CHEMBL3527593
0.0510.0230.055Benzodiazepine inverse agonist

0.051 0.024 CHEMBL3527592

0.051 0.023 CHEMBL1630842

0.055 0.019 CHEMBL3527593

CHEMBL3527593
0.070.0440.07Dopamine agonist

0.07 0.044 CHEMBL1630842

0.1070.0810.132Sphingosine 1-phosphate receptor 2 agonist

0.132 0.039 CHEMBL3527592

0.107 0.081 CHEMBL1630842

0.122 0.052 CHEMBL3527593

CHEMBL3527592
0.0750.050.075MAP kinase 14 inhibitor

0.075 0.05 CHEMBL1630842

0.1990.1770.319Vasodilator, peripheral

0.199 0.177 CHEMBL1630842

0.319 0.088 CHEMBL3527593

CHEMBL3527593
0.0550.0350.059GABA A receptor antagonist

0.059 0.032 CHEMBL3527592

0.055 0.035 CHEMBL1630842

0.047 0.045 CHEMBL3527593

CHEMBL3527592
0.0510.0320.063Adenosine A2b receptor antagonist

0.053 0.03 CHEMBL3527592

0.051 0.032 CHEMBL1630842

0.063 0.022 CHEMBL3527593

CHEMBL3527593
0.1230.1040.155Death-associated protein kinase 1 inhibitor

0.132 0.077 CHEMBL3527592

0.123 0.104 CHEMBL1630842

0.155 0.033 CHEMBL3527593

CHEMBL3527593
0.0330.0140.038Thiazolidinedione

0.038 0.009 CHEMBL3527592

0.033 0.014 CHEMBL1630842

0.036 0.01 CHEMBL3527593

CHEMBL3527592
0.0760.0590.088MAP kinase 7 inhibitor

0.088 0.022 CHEMBL3527592

0.076 0.059 CHEMBL1630842

0.086 0.028 CHEMBL3527593

CHEMBL3527592
0.0270.010.033Phosphodiesterase 6A inhibitor

0.033 0.005 CHEMBL3527592

0.027 0.01 CHEMBL1630842

0.03 0.007 CHEMBL3527593

CHEMBL3527592
0.0470.030.052Phosphodiesterase 6C inhibitor

0.052 0.017 CHEMBL3527592

0.047 0.03 CHEMBL1630842

0.052 0.017 CHEMBL3527593

CHEMBL3527593
0.0580.050.076Adenosine A2 receptor antagonist

0.076 0.037 CHEMBL3527592

0.058 0.05 CHEMBL1630842

0.073 0.038 CHEMBL3527593

CHEMBL3527592
0.0450.0370.066Proto-oncogene tyrosine-protein kinase Met inhibitor

0.066 0.023 CHEMBL3527592

0.045 0.037 CHEMBL1630842

CHEMBL3527592
0.0760.0720.13Caspase 7 inhibitor

0.13 0.012 CHEMBL3527592

0.076 0.072 CHEMBL1630842

0.109 0.02 CHEMBL3527593

CHEMBL3527592
0.0560.0530.099Phosphodiesterase 1A inhibitor

0.099 0.01 CHEMBL3527592

0.056 0.053 CHEMBL1630842

0.076 0.019 CHEMBL3527593

CHEMBL3527592
0.0490.0480.107Bromodomain-containing protein 4 inhibitor

0.073 0.022 CHEMBL3527592

0.049 0.048 CHEMBL1630842

0.107 0.012 CHEMBL3527593

CHEMBL3527593
0.0850.0840.102Interleukin 12 antagonist

0.102 0.05 CHEMBL3527592

0.085 0.084 CHEMBL1630842

0.099 0.055 CHEMBL3527593

CHEMBL3527592
0.0480.0480.052GABA receptor antagonist

0.052 0.041 CHEMBL3527592

CHEMBL3527592
0.120.1250.148Polo-like kinase-3 inhibitor

0.141 0.094 CHEMBL3527592

0.148 0.086 CHEMBL3527593

CHEMBL3527593
0.0470.0560.074Phosphodiesterase II inhibitor

0.072 0.022 CHEMBL3527592

0.074 0.021 CHEMBL3527593

CHEMBL3527593
0.0250.0410.047Glutamate (mGluR group II) agonist

0.047 0.017 CHEMBL3527592

CHEMBL3527592
0.10.1170.12Ribosomal protein S6 kinase inhibitor

0.12 0.09 CHEMBL3527592

0.116 0.095 CHEMBL3527593

CHEMBL3527592
0.0220.0390.044Glutamate (mGluR2) agonist

0.044 0.016 CHEMBL3527592

CHEMBL3527592
0.0380.0580.062Phosphodiesterase 2A inhibitor

0.061 0.023 CHEMBL3527592

0.062 0.022 CHEMBL3527593

CHEMBL3527593
0.1770.1990.21Angiogenesis inhibitor

0.21 0.158 CHEMBL3527592

CHEMBL3527592
0.0350.060.043Glutamate (mGluR group III) antagonist

0.043 0.031 CHEMBL3527592

0.043 0.033 CHEMBL3527593

CHEMBL3527593
0.0550.080.081Glutamate (mGluR7) antagonist

0.081 0.027 CHEMBL3527592

CHEMBL3527592
0.0660.0920.131Proto-oncogene tyrosine-protein kinase Kit inhibitor

0.131 0.04 CHEMBL3527592

CHEMBL3527592
0.080.1090.132Phosphodiesterase 6D inhibitor

0.132 0.016 CHEMBL3527592

0.126 0.02 CHEMBL3527593

CHEMBL3527592
0.2520.2840.389Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.361 0.138 CHEMBL3527592

0.389 0.111 CHEMBL3527593

CHEMBL3527593
0.0650.1030.153Platelet activating factor alpha antagonist

0.153 0.029 CHEMBL3527592

CHEMBL3527592
0.1750.2130.204MAP kinase kinase 3 inhibitor

0.204 0.111 CHEMBL3527592

0.192 0.146 CHEMBL3527593

CHEMBL3527592
0.0550.0970.13Platelet growth factor antagonist

0.13 0.025 CHEMBL3527592

0.086 0.051 CHEMBL3527593

CHEMBL3527592
0.0680.1220.105Polo-like kinase-4 inhibitor

0.105 0.072 CHEMBL3527593

CHEMBL3527593
0.0230.0790.046Phosphodiesterase 3B inhibitor

0.046 0.028 CHEMBL3527593

CHEMBL3527593
0.0340.090.075Glutamate (mGluR) agonist

0.075 0.033 CHEMBL3527592

CHEMBL3527592
0.060.1220.157Mediator release inhibitor

0.135 0.036 CHEMBL3527592

0.157 0.026 CHEMBL3527593

CHEMBL3527593
0.030.0980.054Adenosine A2a receptor antagonist

0.054 0.051 CHEMBL3527592

CHEMBL3527592
0.0230.0950.037Acid-sensing ion channel blocker

0.037 0.034 CHEMBL3527593

CHEMBL3527593
0.0370.1140.105Phosphodiesterase 1B inhibitor

0.105 0.013 CHEMBL3527592

0.062 0.039 CHEMBL3527593

CHEMBL3527592
0.0440.1240.087Phosphodiesterase 1C inhibitor

0.087 0.015 CHEMBL3527592

CHEMBL3527592
0.0470.1280.077ALK inhibitor

0.077 0.064 CHEMBL3527592

0.075 0.067 CHEMBL3527593

CHEMBL3527592
0.0660.1580.084Toll-Like receptor 3 antagonist

0.084 0.083 CHEMBL3527593

CHEMBL3527593
0.1210.2160.348Cyclic AMP phosphodiesterase inhibitor

0.293 0.045 CHEMBL3527592

0.348 0.026 CHEMBL3527593

CHEMBL3527593
0.0560.1530.125Phosphodiesterase I inhibitor

0.125 0.024 CHEMBL3527592

0.115 0.03 CHEMBL3527593

CHEMBL3527592
0.1640.2630.343GABA C receptor rho-3 antagonist

0.343 0.09 CHEMBL3527592

0.315 0.106 CHEMBL3527593

CHEMBL3527592
0.0290.1420.0545 Hydroxytryptamine 1B agonist

0.054 0.035 CHEMBL3527593

CHEMBL3527593
0.0590.1750.172Vascular endothelial growth factor 3 antagonist

0.172 0.053 CHEMBL3527592

CHEMBL3527592
0.0490.1650.076Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.076 0.071 CHEMBL3527593

CHEMBL3527593
0.0550.1760.125Bromodomain-containing protein 2 inhibitor

0.125 0.02 CHEMBL3527592

0.114 0.027 CHEMBL3527593

CHEMBL3527592
0.0650.1860.119Growth factor antagonist

0.119 0.093 CHEMBL3527592

CHEMBL3527592
0.0930.2370.139Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.139 0.094 CHEMBL3527593

CHEMBL3527593
0.0440.230.084Interleukin 1 beta converting enzyme inhibitor

0.084 0.082 CHEMBL3527592

CHEMBL3527592
0.0680.2590.123Aurora-C kinase inhibitor

0.123 0.099 CHEMBL3527593

CHEMBL3527593
0.0180.2360.056mTOR inhibitor

0.056 0.032 CHEMBL3527593

CHEMBL3527593
0.0490.2750.144Activin receptor-like kinase 2 inhibitor

0.144 0.072 CHEMBL3527592

0.118 0.098 CHEMBL3527593

CHEMBL3527592
0.0670.3090.129GABA C receptor rho-2 antagonist

0.129 0.108 CHEMBL3527592

CHEMBL3527592
0.0150.2590.085Glutamate receptor agonist

0.085 0.048 CHEMBL3527592

CHEMBL3527592
0.1450.3960.207Ca2+/calmodulin-dependent kinase IV inhibitor

0.207 0.147 CHEMBL3527593

CHEMBL3527593
0.1090.3860.272Histamine release inhibitor

0.272 0.14 CHEMBL3527592

0.224 0.177 CHEMBL3527593

CHEMBL3527592
0.0790.3870.15Death-associated protein kinase 2 inhibitor

0.15 0.106 CHEMBL3527593

CHEMBL3527593
0.0130.3640.042Nicotinic acid receptor 1 agonist

0.042 0.026 CHEMBL3527593

CHEMBL3527593
0.0820.4460.143Cyclin-dependent kinase 3 inhibitor

0.143 0.113 CHEMBL3527593

CHEMBL3527593
0.0340.4040.117Acetylcholine M1 receptor antagonist

0.117 0.113 CHEMBL3527593

CHEMBL3527593
0.0760.4910.201Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.201 0.156 CHEMBL3527593

CHEMBL3527593
Ext Pa Pi Pmax Activity Other Results ID Pa_max