| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.993 | 0.001 | 0.993 | Renin inhibitor | 0.99 0.001 CHEMBL3507701 0.972 0.002 CHEMBL3507697 0.26 0.004 CHEMBL3507704 0.988 0.001 CHEMBL3507703 0.989 0.001 CHEMBL3507700 0.989 0.001 CHEMBL3507699 0.825 0.002 CHEMBL3507695 0.863 0.002 CHEMBL3507696 | ||
| 0.447 | 0.021 | 0.447 | Cardiotonic | 0.417 0.026 CHEMBL3507701 0.416 0.026 CHEMBL3507697 0.392 0.03 CHEMBL3507703 0.43 0.024 CHEMBL3507700 0.438 0.023 CHEMBL3507699 0.392 0.03 CHEMBL3507695 0.415 0.026 CHEMBL3507696 | ||
| 0.387 | 0.054 | 0.649 | Immunostimulant | 0.396 0.051 CHEMBL3507701 0.408 0.047 CHEMBL3507697 0.431 0.041 CHEMBL3507703 0.378 0.056 CHEMBL3507700 0.418 0.045 CHEMBL3507699 0.634 0.013 CHEMBL3507695 0.649 0.012 CHEMBL3507696 | CHEMBL3507696 | |
| 0.344 | 0.04 | 0.446 | Platelet antagonist | 0.319 0.047 CHEMBL3507701 0.446 0.02 CHEMBL3507697 0.157 0.137 CHEMBL3507704 0.335 0.042 CHEMBL3507703 0.332 0.043 CHEMBL3507700 0.343 0.04 CHEMBL3507699 0.342 0.04 CHEMBL3507695 0.362 0.035 CHEMBL3507696 | CHEMBL3507697 | |
| 0.269 | 0.007 | 0.299 | Protease inhibitor | 0.297 0.005 CHEMBL3507701 0.267 0.007 CHEMBL3507697 0.132 0.04 CHEMBL3507704 0.299 0.005 CHEMBL3507703 0.271 0.007 CHEMBL3507700 0.259 0.007 CHEMBL3507699 0.215 0.011 CHEMBL3507695 0.2 0.014 CHEMBL3507696 | CHEMBL3507703 | |
| 0.266 | 0.064 | 0.391 | Antiamyloidogenic | 0.378 0.033 CHEMBL3507701 0.342 0.041 CHEMBL3507697 0.369 0.035 CHEMBL3507703 0.258 0.068 CHEMBL3507700 0.325 0.045 CHEMBL3507699 0.391 0.03 CHEMBL3507695 0.342 0.041 CHEMBL3507696 | CHEMBL3507695 | |
| 0.24 | 0.056 | 0.252 | Platelet aggregation inhibitor | 0.252 0.05 CHEMBL3507697 0.171 0.105 CHEMBL3507704 0.229 0.062 CHEMBL3507703 0.212 0.073 CHEMBL3507700 0.207 0.077 CHEMBL3507699 | CHEMBL3507697 | |
| 0.271 | 0.113 | 0.461 | Vasodilator, coronary | 0.244 0.14 CHEMBL3507701 0.234 0.15 CHEMBL3507697 0.251 0.133 CHEMBL3507704 0.25 0.134 CHEMBL3507703 0.259 0.125 CHEMBL3507700 0.272 0.113 CHEMBL3507699 0.44 0.025 CHEMBL3507695 0.461 0.021 CHEMBL3507696 | CHEMBL3507696 | |
| 0.176 | 0.02 | 0.228 | Vanilloid 1 agonist | 0.194 0.014 CHEMBL3507701 0.17 0.023 CHEMBL3507697 0.206 0.011 CHEMBL3507704 0.149 0.039 CHEMBL3507703 0.187 0.016 CHEMBL3507700 0.191 0.014 CHEMBL3507699 0.228 0.007 CHEMBL3507695 0.221 0.008 CHEMBL3507696 | CHEMBL3507695 | |
| 0.159 | 0.007 | 0.254 | Cathepsin D inhibitor | 0.175 0.005 CHEMBL3507701 0.153 0.007 CHEMBL3507697 0.254 0.004 CHEMBL3507703 0.161 0.007 CHEMBL3507700 0.153 0.007 CHEMBL3507699 0.11 0.015 CHEMBL3507695 0.1 0.019 CHEMBL3507696 | CHEMBL3507703 | |
| 0.232 | 0.084 | 0.476 | Tumour necrosis factor alpha release inhibitor | 0.275 0.063 CHEMBL3507701 0.24 0.079 CHEMBL3507697 0.244 0.077 CHEMBL3507703 0.239 0.08 CHEMBL3507700 0.23 0.085 CHEMBL3507699 0.476 0.016 CHEMBL3507695 0.437 0.021 CHEMBL3507696 | CHEMBL3507695 | |
| 0.273 | 0.133 | 0.421 | Immunosuppressant | 0.269 0.135 CHEMBL3507701 0.295 0.118 CHEMBL3507697 0.404 0.061 CHEMBL3507704 0.227 0.169 CHEMBL3507703 0.292 0.12 CHEMBL3507700 0.285 0.125 CHEMBL3507699 0.421 0.056 CHEMBL3507695 0.42 0.056 CHEMBL3507696 | CHEMBL3507695 | |
| 0.169 | 0.036 | 0.182 | Farnesoid X receptor antagonist | 0.162 0.041 CHEMBL3507701 0.17 0.035 CHEMBL3507697 0.135 0.074 CHEMBL3507704 0.152 0.05 CHEMBL3507703 0.182 0.028 CHEMBL3507700 0.18 0.029 CHEMBL3507699 0.127 0.088 CHEMBL3507696 | CHEMBL3507700 | |
| 0.253 | 0.124 | 0.317 | Sodium/bile acid cotransporter inhibitor | 0.282 0.096 CHEMBL3507701 0.317 0.065 CHEMBL3507697 0.249 0.129 CHEMBL3507704 0.233 0.147 CHEMBL3507703 0.268 0.11 CHEMBL3507700 0.263 0.115 CHEMBL3507699 | CHEMBL3507697 | |
| 0.166 | 0.042 | 0.226 | Toll-Like receptor 2 antagonist | 0.226 0.014 CHEMBL3507701 0.187 0.03 CHEMBL3507697 0.173 0.038 CHEMBL3507703 0.152 0.051 CHEMBL3507700 0.195 0.026 CHEMBL3507699 0.132 0.066 CHEMBL3507695 | CHEMBL3507701 | |
| 0.209 | 0.09 | 0.465 | Angiogenesis stimulant | 0.246 0.072 CHEMBL3507701 0.256 0.067 CHEMBL3507697 0.216 0.086 CHEMBL3507703 0.251 0.069 CHEMBL3507700 0.236 0.077 CHEMBL3507699 0.465 0.014 CHEMBL3507695 0.441 0.016 CHEMBL3507696 | CHEMBL3507695 | |
| 0.173 | 0.058 | 0.229 | Phospholipase A2 inhibitor | 0.229 0.03 CHEMBL3507697 0.134 0.094 CHEMBL3507704 0.145 0.08 CHEMBL3507703 0.162 0.064 CHEMBL3507700 0.188 0.049 CHEMBL3507699 | CHEMBL3507697 | |
| 0.152 | 0.047 | 0.246 | Cyclooxygenase 3 inhibitor | 0.121 0.076 CHEMBL3507701 0.123 0.074 CHEMBL3507697 0.243 0.009 CHEMBL3507704 0.171 0.033 CHEMBL3507703 0.131 0.066 CHEMBL3507700 0.156 0.043 CHEMBL3507699 0.209 0.016 CHEMBL3507695 0.246 0.009 CHEMBL3507696 | CHEMBL3507696 | |
| 0.114 | 0.01 | 0.15 | Cathepsin E inhibitor | 0.126 0.008 CHEMBL3507701 0.116 0.01 CHEMBL3507697 0.15 0.005 CHEMBL3507703 0.114 0.01 CHEMBL3507700 0.109 0.011 CHEMBL3507699 0.087 0.019 CHEMBL3507695 0.08 0.022 CHEMBL3507696 | CHEMBL3507703 | |
| 0.109 | 0.015 | 0.133 | Aminopeptidase microsomal inhibitor | 0.133 0.011 CHEMBL3507701 0.118 0.013 CHEMBL3507697 0.079 0.025 CHEMBL3507703 0.109 0.015 CHEMBL3507700 0.11 0.015 CHEMBL3507699 0.074 0.028 CHEMBL3507695 0.067 0.034 CHEMBL3507696 | CHEMBL3507701 | |
| 0.135 | 0.042 | 0.238 | Mucolytic | 0.192 0.015 CHEMBL3507701 0.188 0.016 CHEMBL3507697 0.105 0.071 CHEMBL3507704 0.16 0.027 CHEMBL3507703 0.169 0.023 CHEMBL3507700 0.143 0.036 CHEMBL3507699 0.238 0.008 CHEMBL3507695 0.179 0.019 CHEMBL3507696 | CHEMBL3507695 | |
| 0.103 | 0.014 | 0.151 | Endothelin-converting enzyme inhibitor | 0.133 0.01 CHEMBL3507701 0.127 0.011 CHEMBL3507697 0.151 0.009 CHEMBL3507703 0.109 0.013 CHEMBL3507700 0.094 0.015 CHEMBL3507699 0.059 0.025 CHEMBL3507695 0.05 0.03 CHEMBL3507696 | CHEMBL3507703 | |
| 0.163 | 0.077 | 0.247 | Growth hormone agonist | 0.219 0.052 CHEMBL3507701 0.247 0.044 CHEMBL3507697 0.153 0.085 CHEMBL3507703 0.184 0.066 CHEMBL3507700 0.167 0.075 CHEMBL3507699 0.136 0.1 CHEMBL3507695 | CHEMBL3507697 | |
| 0.084 | 0.005 | 0.103 | HIV-1 protease inhibitor | 0.103 0.005 CHEMBL3507701 0.08 0.005 CHEMBL3507697 0.094 0.005 CHEMBL3507703 0.087 0.005 CHEMBL3507700 0.085 0.005 CHEMBL3507699 0.07 0.008 CHEMBL3507695 0.065 0.009 CHEMBL3507696 | CHEMBL3507701 | |
| 0.083 | 0.016 | 0.108 | Aminopeptidase N inhibitor | 0.108 0.011 CHEMBL3507701 0.094 0.014 CHEMBL3507697 0.056 0.027 CHEMBL3507703 0.084 0.016 CHEMBL3507700 0.083 0.017 CHEMBL3507699 0.052 0.029 CHEMBL3507695 0.045 0.036 CHEMBL3507696 | CHEMBL3507701 | |
| 0.094 | 0.029 | 0.123 | Matrix metalloproteinase inhibitor | 0.095 0.029 CHEMBL3507701 0.123 0.019 CHEMBL3507697 0.108 0.024 CHEMBL3507703 0.091 0.031 CHEMBL3507700 0.086 0.034 CHEMBL3507699 | CHEMBL3507697 | |
| 0.133 | 0.074 | 0.154 | Bone formation stimulant | 0.13 0.077 CHEMBL3507701 0.144 0.064 CHEMBL3507697 0.144 0.064 CHEMBL3507703 0.154 0.056 CHEMBL3507700 0.138 0.069 CHEMBL3507699 | CHEMBL3507700 | |
| 0.092 | 0.033 | 0.152 | Aminopeptidase I inhibitor | 0.134 0.016 CHEMBL3507701 0.152 0.012 CHEMBL3507697 0.117 0.02 CHEMBL3507700 0.094 0.032 CHEMBL3507699 | CHEMBL3507697 | |
| 0.163 | 0.105 | 0.163 | MAP kinase kinase 5 inhibitor | 0.154 0.135 CHEMBL3507704 0.157 0.126 CHEMBL3507703 0.156 0.13 CHEMBL3507699 | ||
| 0.218 | 0.16 | 0.413 | Interleukin 2 agonist | 0.262 0.106 CHEMBL3507701 0.282 0.087 CHEMBL3507697 0.293 0.079 CHEMBL3507704 0.224 0.151 CHEMBL3507703 0.267 0.1 CHEMBL3507700 0.231 0.141 CHEMBL3507699 0.413 0.024 CHEMBL3507695 0.389 0.031 CHEMBL3507696 | CHEMBL3507695 | |
| 0.095 | 0.039 | 0.118 | Vanilloid agonist | 0.118 0.019 CHEMBL3507701 0.095 0.04 CHEMBL3507697 0.113 0.022 CHEMBL3507704 0.086 0.056 CHEMBL3507703 0.104 0.029 CHEMBL3507700 0.107 0.026 CHEMBL3507699 0.099 0.035 CHEMBL3507695 0.092 0.044 CHEMBL3507696 | CHEMBL3507701 | |
| 0.181 | 0.127 | 0.302 | Peptidyltransferase inhibitor | 0.219 0.078 CHEMBL3507701 0.203 0.095 CHEMBL3507697 0.206 0.092 CHEMBL3507704 0.24 0.058 CHEMBL3507703 0.212 0.085 CHEMBL3507700 0.203 0.095 CHEMBL3507699 0.302 0.024 CHEMBL3507695 0.288 0.029 CHEMBL3507696 | CHEMBL3507695 | |
| 0.083 | 0.032 | 0.136 | Secretase beta inhibitor | 0.101 0.018 CHEMBL3507701 0.065 0.06 CHEMBL3507697 0.136 0.007 CHEMBL3507703 0.086 0.029 CHEMBL3507700 0.073 0.045 CHEMBL3507699 | CHEMBL3507703 | |
| 0.163 | 0.116 | 0.197 | Insulin sensitizer | 0.197 0.076 CHEMBL3507697 0.165 0.113 CHEMBL3507703 0.161 0.118 CHEMBL3507700 0.177 0.099 CHEMBL3507699 | CHEMBL3507697 | |
| 0.087 | 0.044 | 0.108 | Somatostatin 1 agonist | 0.108 0.029 CHEMBL3507701 0.087 0.044 CHEMBL3507697 0.077 0.055 CHEMBL3507703 0.09 0.041 CHEMBL3507700 0.093 0.039 CHEMBL3507699 0.081 0.05 CHEMBL3507695 0.071 0.063 CHEMBL3507696 | CHEMBL3507701 | |
| 0.099 | 0.06 | 0.166 | Sphingomyelinase inhibitor | 0.095 0.066 CHEMBL3507701 0.127 0.036 CHEMBL3507703 0.11 0.05 CHEMBL3507700 0.166 0.019 CHEMBL3507695 0.123 0.039 CHEMBL3507696 | CHEMBL3507695 | |
| 0.145 | 0.107 | 0.176 | Amyloid beta precursor protein antagonist | 0.176 0.076 CHEMBL3507701 0.148 0.104 CHEMBL3507697 0.16 0.091 CHEMBL3507703 0.158 0.092 CHEMBL3507700 0.157 0.094 CHEMBL3507699 | CHEMBL3507701 | |
| 0.047 | 0.009 | 0.059 | Plasmepsin I inhibitor | 0.051 0.007 CHEMBL3507701 0.047 0.009 CHEMBL3507697 0.059 0.005 CHEMBL3507703 0.046 0.009 CHEMBL3507700 0.045 0.01 CHEMBL3507699 0.035 0.016 CHEMBL3507695 0.032 0.019 CHEMBL3507696 | CHEMBL3507703 | |
| 0.111 | 0.074 | 0.164 | Proteasome inhibitor | 0.147 0.048 CHEMBL3507701 0.096 0.093 CHEMBL3507697 0.164 0.039 CHEMBL3507703 0.095 0.094 CHEMBL3507700 0.122 0.063 CHEMBL3507699 | CHEMBL3507703 | |
| 0.205 | 0.17 | 0.343 | Vasodilator, peripheral | 0.225 0.149 CHEMBL3507697 0.23 0.144 CHEMBL3507703 0.214 0.16 CHEMBL3507699 0.302 0.096 CHEMBL3507695 0.343 0.077 CHEMBL3507696 | CHEMBL3507696 | |
| 0.101 | 0.067 | 0.426 | Expectorant | 0.176 0.026 CHEMBL3507701 0.169 0.029 CHEMBL3507697 0.099 0.07 CHEMBL3507704 0.124 0.048 CHEMBL3507703 0.14 0.039 CHEMBL3507700 0.11 0.058 CHEMBL3507699 0.426 0.004 CHEMBL3507695 0.288 0.009 CHEMBL3507696 | CHEMBL3507695 | |
| 0.05 | 0.018 | 0.069 | Plasmepsin II inhibitor | 0.047 0.021 CHEMBL3507701 0.04 0.03 CHEMBL3507697 0.069 0.008 CHEMBL3507703 0.043 0.026 CHEMBL3507700 0.038 0.035 CHEMBL3507699 | CHEMBL3507703 | |
| 0.036 | 0.007 | 0.04 | Aminopeptidase P inhibitor | 0.04 0.005 CHEMBL3507701 0.036 0.006 CHEMBL3507697 0.036 0.007 CHEMBL3507700 0.035 0.007 CHEMBL3507699 0.027 0.013 CHEMBL3507695 0.024 0.015 CHEMBL3507696 | CHEMBL3507701 | |
| 0.058 | 0.034 | 0.065 | Matrix metalloproteinase (membrane-type) inhibitor | 0.053 0.041 CHEMBL3507701 0.062 0.03 CHEMBL3507697 0.065 0.028 CHEMBL3507703 0.052 0.043 CHEMBL3507700 0.052 0.043 CHEMBL3507699 | CHEMBL3507703 | |
| 0.194 | 0.17 | 0.531 | Cholesterol antagonist | 0.217 0.151 CHEMBL3507701 0.281 0.104 CHEMBL3507697 0.331 0.073 CHEMBL3507704 0.241 0.132 CHEMBL3507699 0.511 0.031 CHEMBL3507695 0.531 0.028 CHEMBL3507696 | CHEMBL3507696 | |
| 0.057 | 0.034 | 0.067 | Matrix metalloproteinase 1 inhibitor | 0.06 0.032 CHEMBL3507701 0.066 0.028 CHEMBL3507697 0.067 0.027 CHEMBL3507703 0.055 0.035 CHEMBL3507700 0.052 0.037 CHEMBL3507699 | CHEMBL3507703 | |
| 0.057 | 0.036 | 0.072 | Human rhinovirus A protease inhibitor | 0.07 0.028 CHEMBL3507701 0.066 0.031 CHEMBL3507697 0.072 0.027 CHEMBL3507703 0.059 0.035 CHEMBL3507700 0.056 0.038 CHEMBL3507699 | CHEMBL3507703 | |
| 0.153 | 0.134 | 0.31 | Hypolipemic | 0.164 0.124 CHEMBL3507697 0.31 0.046 CHEMBL3507704 0.149 0.138 CHEMBL3507700 0.156 0.13 CHEMBL3507699 0.154 0.133 CHEMBL3507695 0.198 0.095 CHEMBL3507696 | CHEMBL3507704 | |
| 0.05 | 0.033 | 0.061 | Bombesin 2 receptor antagonist | 0.057 0.026 CHEMBL3507701 0.061 0.024 CHEMBL3507697 0.054 0.029 CHEMBL3507703 0.05 0.033 CHEMBL3507700 0.046 0.041 CHEMBL3507699 | CHEMBL3507697 | |
| 0.054 | 0.039 | 0.059 | Angiotensin-converting enzyme inhibitor | 0.059 0.031 CHEMBL3507701 0.059 0.031 CHEMBL3507697 0.057 0.034 CHEMBL3507703 0.054 0.039 CHEMBL3507700 0.055 0.037 CHEMBL3507699 | CHEMBL3507697 | |
| 0.055 | 0.04 | 0.068 | Immunoglobulin Fc receptor antagonist | 0.068 0.013 CHEMBL3507701 0.054 0.041 CHEMBL3507703 0.058 0.03 CHEMBL3507700 | CHEMBL3507701 | |
| 0.049 | 0.035 | 0.049 | Metalloproteinase-3 inhibitor | 0.048 0.036 CHEMBL3507697 0.048 0.035 CHEMBL3507703 0.043 0.042 CHEMBL3507700 | ||
| 0.053 | 0.039 | 0.098 | Ribonucleoside-diphosphate reductase inhibitor | 0.098 0.02 CHEMBL3507701 0.079 0.025 CHEMBL3507697 0.067 0.03 CHEMBL3507703 0.064 0.032 CHEMBL3507700 0.077 0.026 CHEMBL3507699 0.054 0.038 CHEMBL3507695 | CHEMBL3507701 | |
| 0.049 | 0.035 | 0.054 | Collagenase inhibitor | 0.054 0.025 CHEMBL3507701 0.051 0.03 CHEMBL3507697 0.051 0.03 CHEMBL3507703 0.049 0.034 CHEMBL3507700 0.048 0.037 CHEMBL3507699 | CHEMBL3507701 | |
| 0.052 | 0.041 | 0.098 | Ribonucleotide reductase inhibitor | 0.098 0.021 CHEMBL3507701 0.079 0.027 CHEMBL3507697 0.068 0.032 CHEMBL3507703 0.065 0.034 CHEMBL3507700 0.077 0.028 CHEMBL3507699 0.059 0.037 CHEMBL3507695 | CHEMBL3507701 | |
| 0.046 | 0.035 | 0.056 | Bombesin antagonist | 0.049 0.031 CHEMBL3507701 0.046 0.036 CHEMBL3507697 0.056 0.022 CHEMBL3507703 0.046 0.036 CHEMBL3507700 0.046 0.037 CHEMBL3507699 | CHEMBL3507703 | |
| 0.05 | 0.043 | 0.061 | Vanilloid 2 antagonist | 0.061 0.021 CHEMBL3507701 0.05 0.043 CHEMBL3507700 0.056 0.028 CHEMBL3507699 | CHEMBL3507701 | |
| 0.081 | 0.077 | 0.117 | ATPase (Vacuolar H+) inhibitor | 0.087 0.063 CHEMBL3507701 0.081 0.076 CHEMBL3507697 0.117 0.022 CHEMBL3507704 0.086 0.064 CHEMBL3507703 0.085 0.066 CHEMBL3507699 0.114 0.024 CHEMBL3507695 0.111 0.027 CHEMBL3507696 | CHEMBL3507704 | |
| 0.019 | 0.017 | 0.027 | Neutral endopeptidase inhibitor | 0.024 0.014 CHEMBL3507701 0.027 0.013 CHEMBL3507697 0.018 0.017 CHEMBL3507700 0.018 0.017 CHEMBL3507699 | CHEMBL3507697 | |
| 0.059 | 0.058 | 0.07 | Beta adrenoreceptor antagonist | 0.07 0.039 CHEMBL3507699 | CHEMBL3507699 | |
| 0.045 | 0.046 | 0.067 | Neuropeptide agonist | 0.059 0.038 CHEMBL3507701 0.046 0.045 CHEMBL3507697 0.067 0.036 CHEMBL3507703 0.054 0.04 CHEMBL3507700 | CHEMBL3507703 | |
| 0.114 | 0.117 | 0.217 | Thrombolytic | 0.119 0.112 CHEMBL3507701 0.142 0.088 CHEMBL3507697 0.121 0.109 CHEMBL3507700 0.131 0.098 CHEMBL3507699 0.213 0.046 CHEMBL3507695 0.217 0.044 CHEMBL3507696 | CHEMBL3507696 | |
| 0.055 | 0.059 | 0.07 | Nitric oxide donor | 0.058 0.052 CHEMBL3507703 0.07 0.033 CHEMBL3507696 | CHEMBL3507696 | |
| 0.182 | 0.187 | 0.294 | Insulysin inhibitor | 0.294 0.062 CHEMBL3507701 0.257 0.09 CHEMBL3507697 0.202 0.154 CHEMBL3507703 0.217 0.133 CHEMBL3507699 | CHEMBL3507701 | |
| 0.123 | 0.132 | 0.182 | Amyloid beta aggregation inhibitor | 0.172 0.093 CHEMBL3507701 0.178 0.09 CHEMBL3507699 0.175 0.092 CHEMBL3507695 0.182 0.088 CHEMBL3507696 | CHEMBL3507696 | |
| 0.089 | 0.102 | 0.098 | Factor V inhibitor | 0.093 0.088 CHEMBL3507701 0.098 0.074 CHEMBL3507697 | CHEMBL3507697 | |
| 0.074 | 0.09 | 0.089 | 3C-Like protease (SARS coronavirus) inhibitor | 0.083 0.059 CHEMBL3507701 0.089 0.048 CHEMBL3507703 | CHEMBL3507703 | |
| 0.061 | 0.077 | 0.069 | Metalloproteinase-9 inhibitor | 0.069 0.058 CHEMBL3507701 0.069 0.057 CHEMBL3507703 | CHEMBL3507703 | |
| 0.073 | 0.089 | 0.149 | Aminopeptidase B inhibitor | 0.144 0.04 CHEMBL3507701 0.149 0.038 CHEMBL3507697 0.105 0.061 CHEMBL3507700 | CHEMBL3507697 | |
| 0.012 | 0.033 | 0.02 | Human T-cell leukemia virus type I protease inhibitor | 0.02 0.015 CHEMBL3507703 | CHEMBL3507703 | |
| 0.123 | 0.145 | 0.302 | Hepatoprotectant | 0.148 0.112 CHEMBL3507701 0.133 0.129 CHEMBL3507697 0.142 0.119 CHEMBL3507699 0.302 0.029 CHEMBL3507695 0.289 0.033 CHEMBL3507696 | CHEMBL3507695 | |
| 0.028 | 0.053 | 0.043 | Macrophage elastase inhibitor | 0.043 0.03 CHEMBL3507697 | CHEMBL3507697 | |
| 0.042 | 0.069 | 0.051 | Cathepsin B inhibitor | 0.051 0.048 CHEMBL3507703 | CHEMBL3507703 | |
| 0.13 | 0.16 | 0.174 | Neurotensin receptor agonist | 0.174 0.057 CHEMBL3507701 0.165 0.07 CHEMBL3507697 0.138 0.134 CHEMBL3507703 | CHEMBL3507701 | |
| 0.058 | 0.089 | 0.136 | Calcium antagonist | 0.136 0.027 CHEMBL3507704 | CHEMBL3507704 | |
| 0.049 | 0.081 | 0.063 | Caspase 9 inhibitor | 0.063 0.042 CHEMBL3507697 0.059 0.049 CHEMBL3507703 | CHEMBL3507697 | |
| 0.178 | 0.215 | 0.38 | Apoptosis antagonist | 0.208 0.169 CHEMBL3507701 0.223 0.154 CHEMBL3507697 0.216 0.16 CHEMBL3507704 0.217 0.159 CHEMBL3507703 0.206 0.171 CHEMBL3507699 0.38 0.044 CHEMBL3507695 0.367 0.049 CHEMBL3507696 | CHEMBL3507695 | |
| 0.056 | 0.094 | 0.08 | Metalloproteinase-2 inhibitor | 0.08 0.052 CHEMBL3507697 | CHEMBL3507697 | |
| 0.016 | 0.055 | 0.028 | Caspase 2 inhibitor | 0.028 0.026 CHEMBL3507703 | CHEMBL3507703 | |
| 0.079 | 0.118 | 0.152 | Toll-Like receptor 4 antagonist | 0.149 0.021 CHEMBL3507695 0.152 0.02 CHEMBL3507696 | CHEMBL3507696 | |
| 0.048 | 0.088 | 0.06 | Protease 3C (Human rhinovirus) inhibitor | 0.06 0.052 CHEMBL3507701 0.059 0.054 CHEMBL3507697 | CHEMBL3507701 | |
| 0.068 | 0.109 | 0.134 | Transcription factor NF kappa B stimulant | 0.134 0.02 CHEMBL3507695 0.132 0.02 CHEMBL3507696 | CHEMBL3507695 | |
| 0.019 | 0.061 | 0.028 | 1,3-Beta-glucan synthase inhibitor | 0.027 0.024 CHEMBL3507695 0.028 0.021 CHEMBL3507696 | CHEMBL3507696 | |
| 0.03 | 0.073 | 0.052 | Neuraminidase (Influenza A) inhibitor | 0.052 0.021 CHEMBL3507704 0.047 0.028 CHEMBL3507703 | CHEMBL3507704 | |
| 0.02 | 0.064 | 0.029 | Toll-Like receptor 4 agonist | 0.029 0.014 CHEMBL3507695 0.028 0.014 CHEMBL3507696 | CHEMBL3507695 | |
| 0.045 | 0.091 | 0.132 | Catalase inhibitor | 0.132 0.03 CHEMBL3507697 | CHEMBL3507697 | |
| 0.083 | 0.131 | 0.2 | Electron transport complex I inhibitor | 0.096 0.093 CHEMBL3507701 0.2 0.008 CHEMBL3507704 | CHEMBL3507704 | |
| 0.032 | 0.082 | 0.055 | Opioid delta receptor antagonist | 0.055 0.05 CHEMBL3507701 | CHEMBL3507701 | |
| 0.046 | 0.097 | 0.072 | Neuraminidase (influenza) inhibitor | 0.072 0.032 CHEMBL3507704 0.064 0.045 CHEMBL3507703 | CHEMBL3507704 | |
| 0.039 | 0.091 | 0.075 | Peroxisome proliferator-activated receptor gamma agonist | 0.075 0.045 CHEMBL3507704 | CHEMBL3507704 | |
| 0.034 | 0.087 | 0.077 | Neuraminidase inhibitor | 0.077 0.028 CHEMBL3507704 0.067 0.036 CHEMBL3507703 | CHEMBL3507704 | |
| 0.169 | 0.222 | 0.526 | Antithrombotic | 0.251 0.125 CHEMBL3507697 0.524 0.026 CHEMBL3507695 0.526 0.026 CHEMBL3507696 | CHEMBL3507696 | |
| 0.034 | 0.092 | 0.052 | Leukotriene B4 antagonist | 0.052 0.04 CHEMBL3507697 | CHEMBL3507697 | |
| 0.033 | 0.094 | 0.272 | Selectin antagonist | 0.272 0.007 CHEMBL3507695 0.266 0.007 CHEMBL3507696 | CHEMBL3507695 | |
| 0.055 | 0.12 | 0.077 | Opioid antagonist | 0.077 0.074 CHEMBL3507701 | CHEMBL3507701 | |
| 0.037 | 0.103 | 0.064 | Leukotriene antagonist | 0.064 0.046 CHEMBL3507697 | CHEMBL3507697 | |
| 0.126 | 0.197 | 0.225 | Vasodilator | 0.169 0.132 CHEMBL3507695 0.225 0.086 CHEMBL3507696 | CHEMBL3507696 | |
| 0.068 | 0.139 | 0.145 | DNA polymerase I inhibitor | 0.101 0.085 CHEMBL3507701 0.096 0.09 CHEMBL3507699 0.145 0.052 CHEMBL3507695 0.137 0.057 CHEMBL3507696 | CHEMBL3507695 | |
| 0.022 | 0.098 | 0.065 | Antibiotic Aminoglycoside-like | 0.054 0.011 CHEMBL3507704 0.065 0.007 CHEMBL3507695 0.06 0.009 CHEMBL3507696 | CHEMBL3507695 | |
| 0.108 | 0.187 | 0.145 | P-glycoprotein inhibitor | 0.145 0.124 CHEMBL3507704 | CHEMBL3507704 | |
| 0.102 | 0.181 | 0.326 | Melanin inhibitor | 0.153 0.078 CHEMBL3507701 0.146 0.087 CHEMBL3507704 0.326 0.019 CHEMBL3507695 0.213 0.036 CHEMBL3507696 | CHEMBL3507695 | |
| 0.099 | 0.179 | 0.273 | Nitric oxide antagonist | 0.128 0.122 CHEMBL3507701 0.175 0.079 CHEMBL3507704 0.273 0.046 CHEMBL3507695 0.25 0.052 CHEMBL3507696 | CHEMBL3507695 | |
| 0.017 | 0.097 | 0.032 | Melatonin 1 agonist | 0.032 0.025 CHEMBL3507703 | CHEMBL3507703 | |
| 0.039 | 0.126 | 0.065 | Cathepsin G inhibitor | 0.065 0.06 CHEMBL3507701 | CHEMBL3507701 | |
| 0.098 | 0.192 | 0.232 | Interleukin antagonist | 0.232 0.069 CHEMBL3507703 | CHEMBL3507703 | |
| 0.095 | 0.19 | 0.324 | Anesthetic general | 0.324 0.028 CHEMBL3507704 0.163 0.101 CHEMBL3507696 | CHEMBL3507704 | |
| 0.19 | 0.29 | 0.587 | Cyclophilin D inhibitor | 0.253 0.209 CHEMBL3507697 0.567 0.034 CHEMBL3507695 0.587 0.03 CHEMBL3507696 | CHEMBL3507696 | |
| 0.138 | 0.241 | 0.548 | Transcription factor NF kappa B inhibitor | 0.265 0.117 CHEMBL3507701 0.36 0.074 CHEMBL3507704 0.196 0.173 CHEMBL3507699 0.548 0.038 CHEMBL3507695 0.458 0.051 CHEMBL3507696 | CHEMBL3507695 | |
| 0.114 | 0.223 | 0.391 | Antioxidant | 0.186 0.126 CHEMBL3507701 0.176 0.136 CHEMBL3507699 0.391 0.036 CHEMBL3507695 0.369 0.041 CHEMBL3507696 | CHEMBL3507695 | |
| 0.088 | 0.197 | 0.13 | Thiol protease inhibitor | 0.13 0.097 CHEMBL3507703 | CHEMBL3507703 | |
| 0.074 | 0.186 | 0.114 | Histone deacetylase SIRT1 inhibitor | 0.114 0.098 CHEMBL3507703 | CHEMBL3507703 | |
| 0.011 | 0.126 | 0.036 | Protein 30S ribosomal subunit inhibitor | 0.022 0.019 CHEMBL3507704 0.036 0.011 CHEMBL3507695 0.031 0.012 CHEMBL3507696 | CHEMBL3507695 | |
| 0.07 | 0.189 | 0.118 | Cathepsin H inhibitor | 0.118 0.078 CHEMBL3507701 | CHEMBL3507701 | |
| 0.112 | 0.236 | 0.183 | Calpain inhibitor | 0.167 0.153 CHEMBL3507701 0.183 0.131 CHEMBL3507703 | CHEMBL3507703 | |
| 0.024 | 0.153 | 0.108 | Antineoplastic antibiotic | 0.09 0.051 CHEMBL3507704 0.108 0.043 CHEMBL3507695 0.093 0.05 CHEMBL3507696 | CHEMBL3507695 | |
| 0.111 | 0.254 | 0.389 | Hypoglycemic | 0.192 0.121 CHEMBL3507704 0.372 0.033 CHEMBL3507695 0.389 0.029 CHEMBL3507696 | CHEMBL3507696 | |
| 0.086 | 0.23 | 0.134 | Adenylate cyclase stimulant | 0.134 0.092 CHEMBL3507701 | CHEMBL3507701 | |
| 0.059 | 0.203 | 0.112 | Microtubule formation inhibitor | 0.112 0.071 CHEMBL3507704 | CHEMBL3507704 | |
| 0.112 | 0.277 | 0.398 | 5 Hydroxytryptamine release stimulant | 0.201 0.12 CHEMBL3507701 0.398 0.046 CHEMBL3507695 | CHEMBL3507695 | |
| 0.118 | 0.304 | 0.189 | Nootropic | 0.189 0.173 CHEMBL3507703 | CHEMBL3507703 | |
| 0.074 | 0.26 | 0.225 | Platelet adhesion inhibitor | 0.225 0.059 CHEMBL3507695 0.217 0.063 CHEMBL3507696 | CHEMBL3507695 | |
| 0.082 | 0.269 | 0.336 | Free radical scavenger | 0.169 0.124 CHEMBL3507701 0.336 0.042 CHEMBL3507695 0.305 0.051 CHEMBL3507696 | CHEMBL3507695 | |
| 0.032 | 0.223 | 0.073 | Interferon inducer | 0.073 0.031 CHEMBL3507696 | CHEMBL3507696 | |
| 0.032 | 0.227 | 0.091 | Interferon agonist | 0.091 0.037 CHEMBL3507696 | CHEMBL3507696 | |
| 0.048 | 0.244 | 0.079 | Interleukin 5 antagonist | 0.079 0.074 CHEMBL3507704 | CHEMBL3507704 | |
| 0.017 | 0.218 | 0.067 | Protein 50S ribosomal subunit inhibitor | 0.062 0.029 CHEMBL3507704 0.067 0.026 CHEMBL3507695 0.061 0.03 CHEMBL3507696 | CHEMBL3507695 | |
| 0.127 | 0.335 | 0.246 | Tyrosine 3 hydroxylase inhibitor | 0.246 0.072 CHEMBL3507701 0.201 0.133 CHEMBL3507697 0.194 0.146 CHEMBL3507704 | CHEMBL3507701 | |
| 0.053 | 0.267 | 0.118 | Antibacterial (Helicobacter pylori) | 0.118 0.085 CHEMBL3507704 | CHEMBL3507704 | |
| 0.058 | 0.274 | 0.247 | Protein kinase stimulant | 0.153 0.066 CHEMBL3507704 0.247 0.027 CHEMBL3507695 0.199 0.042 CHEMBL3507696 | CHEMBL3507695 | |
| 0.07 | 0.299 | 0.128 | Insulin secretagoues | 0.128 0.099 CHEMBL3507695 0.122 0.108 CHEMBL3507696 | CHEMBL3507695 | |
| 0.042 | 0.272 | 0.141 | Lipid peroxidase inhibitor | 0.141 0.074 CHEMBL3507695 0.139 0.076 CHEMBL3507696 | CHEMBL3507695 | |
| 0.015 | 0.261 | 0.082 | Alpha-mannosidase inhibitor | 0.082 0.01 CHEMBL3507695 0.074 0.014 CHEMBL3507696 | CHEMBL3507695 | |
| 0.018 | 0.272 | 0.154 | Monophenol monooxygenase inhibitor | 0.154 0.045 CHEMBL3507695 0.117 0.063 CHEMBL3507696 | CHEMBL3507695 | |
| 0.152 | 0.413 | 0.525 | Antiinflammatory | 0.525 0.078 CHEMBL3507695 0.513 0.082 CHEMBL3507696 | CHEMBL3507695 | |
| 0.019 | 0.295 | 0.074 | CDC25A inhibitor | 0.074 0.051 CHEMBL3507704 | CHEMBL3507704 | |
| 0.068 | 0.351 | 0.179 | Interferon gamma antagonist | 0.179 0.051 CHEMBL3507695 0.168 0.059 CHEMBL3507696 | CHEMBL3507695 | |
| 0.009 | 0.317 | 0.064 | Mannosidase inhibitor | 0.064 0.014 CHEMBL3507695 0.056 0.019 CHEMBL3507696 | CHEMBL3507695 | |
| 0.006 | 0.328 | 0.042 | Sodium/glucose cotransporter inhibitor | 0.042 0.006 CHEMBL3507695 0.041 0.007 CHEMBL3507696 | CHEMBL3507695 | |
| 0.072 | 0.395 | 0.184 | Superoxide dismutase inhibitor | 0.184 0.136 CHEMBL3507701 | CHEMBL3507701 | |
| 0.11 | 0.444 | 0.345 | Apoptosis agonist | 0.345 0.141 CHEMBL3507695 0.33 0.152 CHEMBL3507696 | CHEMBL3507695 | |
| 0.023 | 0.357 | 0.13 | Cholesterol synthesis inhibitor | 0.13 0.057 CHEMBL3507704 | CHEMBL3507704 | |
| 0.032 | 0.384 | 0.395 | Amylase inhibitor | 0.395 0.009 CHEMBL3507695 0.288 0.02 CHEMBL3507696 | CHEMBL3507695 | |
| 0.052 | 0.406 | 0.148 | Non-steroidal antiinflammatory agent | 0.148 0.118 CHEMBL3507695 | CHEMBL3507695 | |
| 0.004 | 0.362 | 0.034 | Sodium/glucose cotransporter 2 inhibitor | 0.034 0.01 CHEMBL3507695 0.031 0.012 CHEMBL3507696 | CHEMBL3507695 | |
| 0.049 | 0.412 | 0.13 | Interleukin 6 antagonist | 0.13 0.126 CHEMBL3507695 | CHEMBL3507695 | |
| 0.092 | 0.457 | 0.234 | Caspase 3 stimulant | 0.234 0.127 CHEMBL3507695 | CHEMBL3507695 | |
| 0.013 | 0.413 | 0.034 | Tubulin agonist | 0.034 0.024 CHEMBL3507704 | CHEMBL3507704 | |
| 0.042 | 0.459 | 0.312 | Interleukin agonist | 0.312 0.042 CHEMBL3507695 0.216 0.106 CHEMBL3507696 | CHEMBL3507695 | |
| 0.038 | 0.472 | 0.144 | Hemostatic | 0.144 0.076 CHEMBL3507695 0.138 0.084 CHEMBL3507696 | CHEMBL3507695 | |
| 0.063 | 0.513 | 0.222 | Immunomodulator | 0.21 0.152 CHEMBL3507695 0.222 0.139 CHEMBL3507696 | CHEMBL3507696 | |
| 0.048 | 0.506 | 0.21 | Neurotrophic factor enhancer | 0.21 0.067 CHEMBL3507695 | CHEMBL3507695 | |
| 0.09 | 0.597 | 0.185 | 5 Hydroxytryptamine uptake stimulant | 0.185 0.184 CHEMBL3507701 | CHEMBL3507701 | |
| 0.017 | 0.669 | 0.264 | DNA synthesis inhibitor | 0.264 0.058 CHEMBL3507695 0.191 0.137 CHEMBL3507696 | CHEMBL3507695 | |
| 0.011 | 0.789 | 0.45 | Antibacterial | 0.24 0.186 CHEMBL3507704 0.45 0.057 CHEMBL3507695 0.375 0.088 CHEMBL3507696 | CHEMBL3507695 | |
| 0.025 | 0.845 | 0.123 | NOS3 expression enhancer | 0.123 0.11 CHEMBL3507695 | CHEMBL3507695 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |