| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.936 | 0.003 | 0.936 | Anticoagulant | 0.823 0.004 CHEMBL3527225 0.817 0.004 CHEMBL3527224 0.883 0.004 CHEMBL1710849 0.809 0.004 CHEMBL3527010 0.823 0.004 CHEMBL3527226 0.871 0.004 CHEMBL3527068 | ||
| 0.809 | 0.003 | 0.809 | Thrombin inhibitor | 0.54 0.004 CHEMBL3527225 0.534 0.004 CHEMBL3527224 0.588 0.003 CHEMBL1710849 0.522 0.004 CHEMBL3527010 0.54 0.004 CHEMBL3527226 0.617 0.003 CHEMBL3527068 | ||
| 0.789 | 0.002 | 0.789 | Trypsin inhibitor | 0.584 0.003 CHEMBL3527225 0.587 0.003 CHEMBL3527224 0.616 0.003 CHEMBL1710849 0.569 0.003 CHEMBL3527010 0.584 0.003 CHEMBL3527226 0.646 0.003 CHEMBL3527068 | ||
| 0.773 | 0.003 | 0.773 | Factor X inhibitor | 0.443 0.004 CHEMBL3527225 0.445 0.004 CHEMBL3527224 0.478 0.004 CHEMBL1710849 0.428 0.004 CHEMBL3527010 0.443 0.004 CHEMBL3527226 0.521 0.004 CHEMBL3527068 | ||
| 0.752 | 0.002 | 0.752 | Trypsin I inhibitor | 0.568 0.003 CHEMBL3527225 0.579 0.003 CHEMBL3527224 0.605 0.003 CHEMBL1710849 0.564 0.003 CHEMBL3527010 0.568 0.003 CHEMBL3527226 0.623 0.003 CHEMBL3527068 | ||
| 0.722 | 0.002 | 0.722 | Plasmin inhibitor | 0.547 0.003 CHEMBL3527225 0.533 0.003 CHEMBL3527224 0.554 0.003 CHEMBL1710849 0.531 0.003 CHEMBL3527010 0.547 0.003 CHEMBL3527226 0.586 0.003 CHEMBL3527068 | ||
| 0.635 | 0.005 | 0.635 | Platelet antagonist | 0.543 0.01 CHEMBL3527225 0.56 0.009 CHEMBL3527224 0.629 0.005 CHEMBL1710849 0.554 0.009 CHEMBL3527010 0.543 0.01 CHEMBL3527226 0.574 0.008 CHEMBL3527068 | ||
| 0.564 | 0.02 | 0.606 | Antithrombotic | 0.585 0.018 CHEMBL3527225 0.577 0.019 CHEMBL3527224 0.553 0.022 CHEMBL1710849 0.606 0.016 CHEMBL3527010 0.585 0.018 CHEMBL3527226 0.606 0.016 CHEMBL3527068 | CHEMBL3527068 | |
| 0.537 | 0.005 | 0.598 | Platelet adhesion inhibitor | 0.499 0.005 CHEMBL3527225 0.505 0.005 CHEMBL3527224 0.598 0.004 CHEMBL1710849 0.481 0.006 CHEMBL3527010 0.499 0.005 CHEMBL3527226 0.525 0.005 CHEMBL3527068 | CHEMBL1710849 | |
| 0.525 | 0.004 | 0.684 | NMDA 2 receptor antagonist | 0.684 0.003 CHEMBL3527225 0.564 0.003 CHEMBL3527224 0.572 0.003 CHEMBL1710849 0.453 0.004 CHEMBL3527010 0.684 0.003 CHEMBL3527226 0.589 0.003 CHEMBL3527068 | CHEMBL3527226 | |
| 0.511 | 0.003 | 0.511 | Plasminogen activator inhibitor | 0.262 0.004 CHEMBL3527225 0.247 0.004 CHEMBL3527224 0.22 0.004 CHEMBL1710849 0.248 0.004 CHEMBL3527010 0.262 0.004 CHEMBL3527226 0.31 0.004 CHEMBL3527068 | ||
| 0.509 | 0.009 | 0.509 | Platelet aggregation inhibitor | 0.427 0.016 CHEMBL3527225 0.387 0.02 CHEMBL3527224 0.41 0.017 CHEMBL1710849 0.383 0.02 CHEMBL3527010 0.427 0.016 CHEMBL3527226 0.453 0.013 CHEMBL3527068 | ||
| 0.502 | 0.003 | 0.502 | Kallikrein 1 inhibitor | 0.249 0.004 CHEMBL3527225 0.234 0.004 CHEMBL3527224 0.253 0.004 CHEMBL1710849 0.226 0.004 CHEMBL3527010 0.249 0.004 CHEMBL3527226 0.302 0.004 CHEMBL3527068 | ||
| 0.51 | 0.012 | 0.646 | Superoxide dismutase inhibitor | 0.611 0.006 CHEMBL3527225 0.473 0.016 CHEMBL3527224 0.395 0.028 CHEMBL1710849 0.464 0.017 CHEMBL3527010 0.611 0.006 CHEMBL3527226 0.646 0.005 CHEMBL3527068 | CHEMBL3527068 | |
| 0.476 | 0.012 | 0.476 | Sigma receptor agonist | 0.452 0.015 CHEMBL3527225 0.445 0.015 CHEMBL3527224 0.357 0.029 CHEMBL1710849 0.402 0.022 CHEMBL3527010 0.452 0.015 CHEMBL3527226 0.413 0.02 CHEMBL3527068 | ||
| 0.457 | 0.003 | 0.457 | Tryptase inhibitor | 0.275 0.004 CHEMBL3527225 0.266 0.004 CHEMBL3527224 0.334 0.003 CHEMBL1710849 0.269 0.004 CHEMBL3527010 0.275 0.004 CHEMBL3527226 0.315 0.004 CHEMBL3527068 | ||
| 0.479 | 0.031 | 0.503 | 5 Hydroxytryptamine release stimulant | 0.503 0.027 CHEMBL3527225 0.309 0.067 CHEMBL3527224 0.183 0.138 CHEMBL1710849 0.415 0.043 CHEMBL3527010 0.503 0.027 CHEMBL3527226 0.422 0.041 CHEMBL3527068 | CHEMBL3527226 | |
| 0.411 | 0.004 | 0.411 | Nav1.1 sodium channel blocker | 0.356 0.005 CHEMBL3527225 0.39 0.005 CHEMBL3527224 0.291 0.009 CHEMBL1710849 0.333 0.006 CHEMBL3527010 0.356 0.005 CHEMBL3527226 0.344 0.005 CHEMBL3527068 | ||
| 0.4 | 0.008 | 0.446 | Hemostatic | 0.401 0.008 CHEMBL3527225 0.365 0.01 CHEMBL3527224 0.446 0.005 CHEMBL1710849 0.425 0.006 CHEMBL3527010 0.401 0.008 CHEMBL3527226 0.431 0.006 CHEMBL3527068 | CHEMBL1710849 | |
| 0.372 | 0.007 | 0.372 | Butyrylcholinesterase inhibitor | 0.293 0.011 CHEMBL3527225 0.249 0.015 CHEMBL3527224 0.133 0.041 CHEMBL1710849 0.294 0.011 CHEMBL3527010 0.293 0.011 CHEMBL3527226 0.306 0.01 CHEMBL3527068 | ||
| 0.35 | 0.003 | 0.35 | Factor VIIa inhibitor | 0.237 0.004 CHEMBL3527225 0.24 0.004 CHEMBL3527224 0.249 0.004 CHEMBL1710849 0.239 0.004 CHEMBL3527010 0.237 0.004 CHEMBL3527226 0.256 0.004 CHEMBL3527068 | ||
| 0.367 | 0.026 | 0.367 | Anticonvulsant | 0.191 0.09 CHEMBL3527225 0.207 0.078 CHEMBL3527224 0.194 0.087 CHEMBL1710849 0.156 0.121 CHEMBL3527010 0.191 0.09 CHEMBL3527226 0.192 0.089 CHEMBL3527068 | ||
| 0.343 | 0.005 | 0.497 | NMDA receptor antagonist | 0.497 0.004 CHEMBL3527225 0.41 0.004 CHEMBL3527224 0.36 0.005 CHEMBL1710849 0.354 0.005 CHEMBL3527010 0.497 0.004 CHEMBL3527226 0.402 0.005 CHEMBL3527068 | CHEMBL3527226 | |
| 0.351 | 0.016 | 0.406 | Tyrosine 3 hydroxylase inhibitor | 0.406 0.008 CHEMBL3527225 0.35 0.016 CHEMBL3527224 0.22 0.104 CHEMBL1710849 0.386 0.01 CHEMBL3527010 0.406 0.008 CHEMBL3527226 0.396 0.009 CHEMBL3527068 | CHEMBL3527226 | |
| 0.342 | 0.011 | 0.342 | Nav1.2 sodium channel blocker | 0.254 0.021 CHEMBL3527225 0.308 0.014 CHEMBL3527224 0.211 0.031 CHEMBL1710849 0.292 0.016 CHEMBL3527010 0.254 0.021 CHEMBL3527226 0.212 0.03 CHEMBL3527068 | ||
| 0.334 | 0.01 | 0.334 | Acetylcholine M1 receptor antagonist | 0.315 0.012 CHEMBL3527225 0.294 0.015 CHEMBL3527224 0.314 0.012 CHEMBL1710849 0.263 0.022 CHEMBL3527010 0.315 0.012 CHEMBL3527226 0.322 0.011 CHEMBL3527068 | ||
| 0.306 | 0.004 | 0.306 | Factor Xa inhibitor | 0.208 0.005 CHEMBL3527225 0.22 0.005 CHEMBL3527224 0.16 0.008 CHEMBL1710849 0.223 0.005 CHEMBL3527010 0.208 0.005 CHEMBL3527226 0.253 0.005 CHEMBL3527068 | ||
| 0.297 | 0.004 | 0.297 | Nitric-oxide synthase inhibitor | 0.209 0.008 CHEMBL3527225 0.232 0.006 CHEMBL3527224 0.166 0.017 CHEMBL1710849 0.197 0.01 CHEMBL3527010 0.209 0.008 CHEMBL3527226 0.244 0.005 CHEMBL3527068 | ||
| 0.291 | 0.005 | 0.291 | GP IIb/IIIa receptor antagonist | 0.161 0.009 CHEMBL3527225 0.14 0.012 CHEMBL3527224 0.151 0.01 CHEMBL1710849 0.137 0.012 CHEMBL3527010 0.161 0.009 CHEMBL3527226 0.176 0.008 CHEMBL3527068 | ||
| 0.333 | 0.058 | 0.593 | Aldehyde oxidase inhibitor | 0.593 0.02 CHEMBL3527225 0.48 0.036 CHEMBL3527224 0.247 0.083 CHEMBL1710849 0.57 0.023 CHEMBL3527010 0.593 0.02 CHEMBL3527226 0.567 0.023 CHEMBL3527068 | CHEMBL3527226 | |
| 0.277 | 0.003 | 0.277 | 5 Hydroxytryptamine 3 agonist | 0.195 0.004 CHEMBL3527225 0.161 0.004 CHEMBL3527224 0.115 0.01 CHEMBL1710849 0.168 0.004 CHEMBL3527010 0.195 0.004 CHEMBL3527226 0.179 0.004 CHEMBL3527068 | ||
| 0.288 | 0.016 | 0.314 | Cholinergic antagonist | 0.254 0.02 CHEMBL3527225 0.21 0.029 CHEMBL3527224 0.314 0.013 CHEMBL1710849 0.186 0.036 CHEMBL3527010 0.254 0.02 CHEMBL3527226 0.249 0.021 CHEMBL3527068 | CHEMBL1710849 | |
| 0.277 | 0.005 | 0.277 | CXC chemokine 4 receptor antagonist | 0.211 0.01 CHEMBL3527225 0.153 0.015 CHEMBL3527224 0.142 0.017 CHEMBL1710849 0.122 0.02 CHEMBL3527010 0.211 0.01 CHEMBL3527226 0.206 0.01 CHEMBL3527068 | ||
| 0.281 | 0.011 | 0.326 | Acetylcholine muscarinic antagonist | 0.256 0.014 CHEMBL3527225 0.225 0.019 CHEMBL3527224 0.326 0.007 CHEMBL1710849 0.204 0.023 CHEMBL3527010 0.256 0.014 CHEMBL3527226 0.25 0.014 CHEMBL3527068 | CHEMBL1710849 | |
| 0.285 | 0.015 | 0.311 | Acetylcholine antagonist | 0.253 0.019 CHEMBL3527225 0.21 0.028 CHEMBL3527224 0.311 0.013 CHEMBL1710849 0.185 0.035 CHEMBL3527010 0.253 0.019 CHEMBL3527226 0.248 0.021 CHEMBL3527068 | CHEMBL1710849 | |
| 0.257 | 0.005 | 0.302 | HIV-1 integrase (Overall Integration) inhibitor | 0.257 0.005 CHEMBL3527225 0.302 0.004 CHEMBL3527224 0.21 0.01 CHEMBL1710849 0.264 0.004 CHEMBL3527010 0.257 0.005 CHEMBL3527226 0.288 0.004 CHEMBL3527068 | CHEMBL3527224 | |
| 0.374 | 0.125 | 0.374 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.269 0.258 CHEMBL1710849 | ||
| 0.352 | 0.108 | 0.366 | Analgesic | 0.298 0.143 CHEMBL3527225 0.226 0.207 CHEMBL3527224 0.361 0.102 CHEMBL1710849 0.366 0.1 CHEMBL3527010 0.298 0.143 CHEMBL3527226 0.248 0.184 CHEMBL3527068 | CHEMBL3527010 | |
| 0.354 | 0.112 | 0.401 | 5 Hydroxytryptamine release inhibitor | 0.378 0.092 CHEMBL3527225 0.3 0.165 CHEMBL3527224 0.267 0.205 CHEMBL1710849 0.401 0.077 CHEMBL3527010 0.378 0.092 CHEMBL3527226 0.334 0.13 CHEMBL3527068 | CHEMBL3527010 | |
| 0.238 | 0.009 | 0.238 | 5 Hydroxytryptamine 7 antagonist | 0.121 0.021 CHEMBL3527225 0.111 0.023 CHEMBL3527224 0.108 0.024 CHEMBL3527010 0.121 0.021 CHEMBL3527226 0.107 0.024 CHEMBL3527068 | ||
| 0.247 | 0.019 | 0.247 | Sodium channel blocker | 0.178 0.042 CHEMBL3527225 0.195 0.034 CHEMBL3527224 0.135 0.069 CHEMBL1710849 0.217 0.027 CHEMBL3527010 0.178 0.042 CHEMBL3527226 0.157 0.054 CHEMBL3527068 | ||
| 0.228 | 0.004 | 0.324 | NMDA 2A receptor antagonist | 0.324 0.004 CHEMBL3527225 0.272 0.004 CHEMBL3527224 0.102 0.013 CHEMBL1710849 0.261 0.004 CHEMBL3527010 0.324 0.004 CHEMBL3527226 0.243 0.004 CHEMBL3527068 | CHEMBL3527226 | |
| 0.25 | 0.031 | 0.268 | Tumour necrosis factor antagonist | 0.268 0.025 CHEMBL3527225 0.246 0.032 CHEMBL3527224 0.215 0.045 CHEMBL3527010 0.268 0.025 CHEMBL3527226 0.251 0.03 CHEMBL3527068 | CHEMBL3527226 | |
| 0.223 | 0.004 | 0.223 | Urokinase inhibitor | 0.178 0.005 CHEMBL3527225 0.174 0.005 CHEMBL3527224 0.169 0.005 CHEMBL1710849 0.173 0.005 CHEMBL3527010 0.178 0.005 CHEMBL3527226 0.184 0.005 CHEMBL3527068 | ||
| 0.253 | 0.04 | 0.268 | P-glycoprotein inhibitor | 0.253 0.04 CHEMBL3527225 0.254 0.04 CHEMBL3527224 0.187 0.073 CHEMBL1710849 0.185 0.075 CHEMBL3527010 0.253 0.04 CHEMBL3527226 0.268 0.036 CHEMBL3527068 | CHEMBL3527068 | |
| 0.213 | 0.003 | 0.261 | Sphingosine kinase 2 inhibitor | 0.226 0.003 CHEMBL3527225 0.207 0.003 CHEMBL3527224 0.261 0.002 CHEMBL1710849 0.19 0.003 CHEMBL3527010 0.226 0.003 CHEMBL3527226 0.233 0.002 CHEMBL3527068 | CHEMBL1710849 | |
| 0.205 | 0.006 | 0.205 | Neurotensin receptor antagonist | 0.176 0.008 CHEMBL3527225 0.152 0.01 CHEMBL3527224 0.113 0.012 CHEMBL1710849 0.152 0.01 CHEMBL3527010 0.176 0.008 CHEMBL3527226 0.165 0.009 CHEMBL3527068 | ||
| 0.262 | 0.07 | 0.271 | Interleukin agonist | 0.243 0.084 CHEMBL3527225 0.203 0.118 CHEMBL3527224 0.226 0.097 CHEMBL1710849 0.235 0.09 CHEMBL3527010 0.243 0.084 CHEMBL3527226 0.271 0.065 CHEMBL3527068 | CHEMBL3527068 | |
| 0.193 | 0.008 | 0.193 | Interleukin 2 antagonist | 0.147 0.02 CHEMBL3527225 0.144 0.022 CHEMBL3527224 0.141 0.023 CHEMBL1710849 0.148 0.019 CHEMBL3527010 0.147 0.02 CHEMBL3527226 0.143 0.022 CHEMBL3527068 | ||
| 0.193 | 0.014 | 0.345 | Histidine decarboxylase inhibitor | 0.335 0.005 CHEMBL3527225 0.269 0.008 CHEMBL3527224 0.157 0.018 CHEMBL1710849 0.262 0.008 CHEMBL3527010 0.335 0.005 CHEMBL3527226 0.345 0.005 CHEMBL3527068 | CHEMBL3527068 | |
| 0.195 | 0.017 | 0.195 | 5 Hydroxytryptamine 3A agonist | 0.181 0.021 CHEMBL3527225 0.143 0.039 CHEMBL3527224 0.143 0.039 CHEMBL3527010 0.181 0.021 CHEMBL3527226 0.155 0.032 CHEMBL3527068 | ||
| 0.228 | 0.053 | 0.252 | Non-steroidal antiinflammatory agent | 0.251 0.042 CHEMBL3527225 0.211 0.062 CHEMBL3527224 0.172 0.094 CHEMBL1710849 0.222 0.056 CHEMBL3527010 0.251 0.042 CHEMBL3527226 0.252 0.042 CHEMBL3527068 | CHEMBL3527068 | |
| 0.218 | 0.044 | 0.249 | Thrombolytic | 0.223 0.042 CHEMBL3527225 0.201 0.051 CHEMBL3527224 0.188 0.058 CHEMBL1710849 0.194 0.055 CHEMBL3527010 0.223 0.042 CHEMBL3527226 0.249 0.034 CHEMBL3527068 | CHEMBL3527068 | |
| 0.183 | 0.009 | 0.183 | Sigma receptor antagonist | 0.11 0.015 CHEMBL3527225 0.093 0.017 CHEMBL3527224 0.067 0.024 CHEMBL3527010 0.11 0.015 CHEMBL3527226 0.093 0.017 CHEMBL3527068 | ||
| 0.195 | 0.034 | 0.195 | Anesthetic local | 0.139 0.054 CHEMBL3527225 0.146 0.05 CHEMBL3527224 0.139 0.054 CHEMBL1710849 0.143 0.052 CHEMBL3527010 0.139 0.054 CHEMBL3527226 0.159 0.045 CHEMBL3527068 | ||
| 0.182 | 0.024 | 0.182 | Antihistaminic | 0.086 0.069 CHEMBL3527225 0.086 0.069 CHEMBL3527226 0.087 0.069 CHEMBL3527068 | ||
| 0.174 | 0.021 | 0.201 | Protein kinase C gamma inhibitor | 0.188 0.017 CHEMBL3527225 0.157 0.028 CHEMBL3527224 0.201 0.014 CHEMBL1710849 0.169 0.023 CHEMBL3527010 0.188 0.017 CHEMBL3527226 0.177 0.02 CHEMBL3527068 | CHEMBL1710849 | |
| 0.176 | 0.023 | 0.176 | Histamine antagonist | 0.075 0.07 CHEMBL3527225 0.075 0.07 CHEMBL3527226 0.073 0.072 CHEMBL3527068 | ||
| 0.155 | 0.004 | 0.232 | Sphingosine kinase inhibitor | 0.167 0.004 CHEMBL3527225 0.19 0.003 CHEMBL3527224 0.232 0.003 CHEMBL1710849 0.157 0.004 CHEMBL3527010 0.167 0.004 CHEMBL3527226 0.181 0.003 CHEMBL3527068 | CHEMBL1710849 | |
| 0.153 | 0.004 | 0.153 | Histamine H4 receptor antagonist | 0.072 0.011 CHEMBL3527225 0.059 0.02 CHEMBL3527224 0.052 0.028 CHEMBL1710849 0.059 0.02 CHEMBL3527010 0.072 0.011 CHEMBL3527226 0.072 0.011 CHEMBL3527068 | ||
| 0.258 | 0.11 | 0.328 | Interleukin 2 agonist | 0.294 0.078 CHEMBL3527225 0.275 0.093 CHEMBL3527224 0.328 0.056 CHEMBL1710849 0.275 0.093 CHEMBL3527010 0.294 0.078 CHEMBL3527226 0.285 0.085 CHEMBL3527068 | CHEMBL1710849 | |
| 0.156 | 0.009 | 0.156 | Acetylcholine M4 receptor antagonist | 0.094 0.033 CHEMBL3527225 0.082 0.044 CHEMBL3527224 0.066 0.062 CHEMBL1710849 0.079 0.047 CHEMBL3527010 0.094 0.033 CHEMBL3527226 0.096 0.031 CHEMBL3527068 | ||
| 0.239 | 0.093 | 0.264 | 5 Hydroxytryptamine uptake stimulant | 0.232 0.101 CHEMBL3527225 0.234 0.098 CHEMBL3527224 0.224 0.111 CHEMBL1710849 0.234 0.098 CHEMBL3527010 0.232 0.101 CHEMBL3527226 0.264 0.068 CHEMBL3527068 | CHEMBL3527068 | |
| 0.277 | 0.132 | 0.319 | GABA C receptor rho-3 antagonist | 0.273 0.135 CHEMBL3527225 0.319 0.104 CHEMBL3527224 0.214 0.19 CHEMBL1710849 0.319 0.104 CHEMBL3527010 0.273 0.135 CHEMBL3527226 | CHEMBL3527010 | |
| 0.203 | 0.058 | 0.203 | 5 Hydroxytryptamine 3E antagonist | 0.163 0.161 CHEMBL3527224 0.163 0.161 CHEMBL3527010 | ||
| 0.168 | 0.028 | 0.184 | GABA C receptor agonist | 0.141 0.038 CHEMBL3527225 0.141 0.038 CHEMBL3527224 0.133 0.042 CHEMBL1710849 0.141 0.038 CHEMBL3527010 0.141 0.038 CHEMBL3527226 0.184 0.024 CHEMBL3527068 | CHEMBL3527068 | |
| 0.154 | 0.014 | 0.188 | Analgesic, opioid | 0.188 0.01 CHEMBL3527225 0.125 0.021 CHEMBL3527224 0.138 0.017 CHEMBL1710849 0.148 0.015 CHEMBL3527010 0.188 0.01 CHEMBL3527226 0.153 0.014 CHEMBL3527068 | CHEMBL3527226 | |
| 0.16 | 0.022 | 0.208 | AMP-activated protein kinase stimulant | 0.193 0.012 CHEMBL3527225 0.208 0.01 CHEMBL3527224 0.152 0.027 CHEMBL1710849 0.192 0.012 CHEMBL3527010 0.193 0.012 CHEMBL3527226 0.195 0.012 CHEMBL3527068 | CHEMBL3527224 | |
| 0.242 | 0.104 | 0.256 | Insulysin inhibitor | 0.248 0.098 CHEMBL3527225 0.221 0.128 CHEMBL3527224 0.189 0.174 CHEMBL1710849 0.211 0.141 CHEMBL3527010 0.248 0.098 CHEMBL3527226 0.256 0.09 CHEMBL3527068 | CHEMBL3527068 | |
| 0.14 | 0.004 | 0.14 | Factor XIa inhibitor | 0.105 0.005 CHEMBL3527225 0.106 0.005 CHEMBL3527224 0.088 0.007 CHEMBL1710849 0.104 0.005 CHEMBL3527010 0.105 0.005 CHEMBL3527226 0.114 0.005 CHEMBL3527068 | ||
| 0.174 | 0.04 | 0.174 | Sodium channel (voltage-gated) blocker | 0.121 0.083 CHEMBL3527225 0.127 0.077 CHEMBL3527224 0.124 0.08 CHEMBL3527010 0.121 0.083 CHEMBL3527226 0.106 0.103 CHEMBL3527068 | ||
| 0.181 | 0.049 | 0.213 | Neurotensin receptor agonist | 0.213 0.029 CHEMBL3527225 0.196 0.037 CHEMBL3527224 0.193 0.039 CHEMBL3527010 0.213 0.029 CHEMBL3527226 0.187 0.043 CHEMBL3527068 | CHEMBL3527226 | |
| 0.146 | 0.017 | 0.146 | Inducible nitric-oxide synthase inhibitor | 0.105 0.033 CHEMBL3527225 0.128 0.022 CHEMBL3527224 0.088 0.05 CHEMBL1710849 0.108 0.031 CHEMBL3527010 0.105 0.033 CHEMBL3527226 0.127 0.022 CHEMBL3527068 | ||
| 0.147 | 0.02 | 0.208 | Protein kinase C zeta inhibitor | 0.208 0.01 CHEMBL3527225 0.208 0.01 CHEMBL3527224 0.153 0.019 CHEMBL1710849 0.183 0.014 CHEMBL3527010 0.208 0.01 CHEMBL3527226 0.188 0.013 CHEMBL3527068 | CHEMBL3527226 | |
| 0.134 | 0.01 | 0.134 | Acetylcholine M5 receptor antagonist | 0.105 0.016 CHEMBL3527225 0.083 0.023 CHEMBL3527224 0.06 0.042 CHEMBL1710849 0.09 0.02 CHEMBL3527010 0.105 0.016 CHEMBL3527226 0.103 0.017 CHEMBL3527068 | ||
| 0.158 | 0.034 | 0.176 | Antiadrenergic | 0.131 0.042 CHEMBL3527225 0.176 0.029 CHEMBL3527224 0.133 0.041 CHEMBL3527010 0.131 0.042 CHEMBL3527226 0.148 0.036 CHEMBL3527068 | CHEMBL3527224 | |
| 0.126 | 0.008 | 0.126 | Kallikrein inhibitor | 0.067 0.02 CHEMBL3527225 0.067 0.02 CHEMBL3527224 0.061 0.023 CHEMBL1710849 0.062 0.022 CHEMBL3527010 0.067 0.02 CHEMBL3527226 0.071 0.018 CHEMBL3527068 | ||
| 0.197 | 0.079 | 0.256 | Neurotrophic factor enhancer | 0.256 0.035 CHEMBL3527225 0.218 0.061 CHEMBL3527224 0.252 0.038 CHEMBL3527010 0.256 0.035 CHEMBL3527226 0.255 0.036 CHEMBL3527068 | CHEMBL3527226 | |
| 0.136 | 0.02 | 0.136 | Histamine N-methyltransferase inhibitor | 0.125 0.026 CHEMBL3527225 0.106 0.041 CHEMBL3527224 0.077 0.07 CHEMBL1710849 0.113 0.035 CHEMBL3527010 0.125 0.026 CHEMBL3527226 0.106 0.041 CHEMBL3527068 | ||
| 0.122 | 0.007 | 0.129 | Protein kinase C beta inhibitor | 0.119 0.008 CHEMBL3527225 0.109 0.01 CHEMBL3527224 0.129 0.005 CHEMBL1710849 0.106 0.011 CHEMBL3527010 0.119 0.008 CHEMBL3527226 0.116 0.008 CHEMBL3527068 | CHEMBL1710849 | |
| 0.16 | 0.049 | 0.164 | Acetylcholinesterase inhibitor | 0.162 0.048 CHEMBL3527225 0.142 0.06 CHEMBL3527224 0.154 0.053 CHEMBL3527010 0.162 0.048 CHEMBL3527226 0.164 0.047 CHEMBL3527068 | CHEMBL3527068 | |
| 0.115 | 0.004 | 0.115 | Calcium channel P-type blocker | 0.09 0.009 CHEMBL3527225 0.085 0.011 CHEMBL3527224 0.099 0.005 CHEMBL1710849 0.093 0.008 CHEMBL3527010 0.09 0.009 CHEMBL3527226 0.085 0.011 CHEMBL3527068 | ||
| 0.119 | 0.011 | 0.137 | Maillard reaction inhibitor | 0.123 0.01 CHEMBL3527225 0.137 0.007 CHEMBL3527224 0.114 0.012 CHEMBL1710849 0.137 0.007 CHEMBL3527010 0.123 0.01 CHEMBL3527226 0.133 0.008 CHEMBL3527068 | CHEMBL3527010 | |
| 0.128 | 0.023 | 0.128 | Glutamate (mGluR7) agonist | 0.09 0.084 CHEMBL1710849 | ||
| 0.116 | 0.011 | 0.144 | NMDA 2C receptor antagonist | 0.144 0.007 CHEMBL3527225 0.124 0.01 CHEMBL3527224 0.092 0.019 CHEMBL3527010 0.144 0.007 CHEMBL3527226 0.114 0.012 CHEMBL3527068 | CHEMBL3527226 | |
| 0.283 | 0.179 | 0.364 | Cyclophilin D inhibitor | 0.322 0.144 CHEMBL3527225 0.323 0.143 CHEMBL3527224 0.364 0.112 CHEMBL1710849 0.342 0.128 CHEMBL3527010 0.322 0.144 CHEMBL3527226 0.347 0.125 CHEMBL3527068 | CHEMBL1710849 | |
| 0.108 | 0.004 | 0.194 | Dopamine D5 agonist | 0.194 0.002 CHEMBL3527225 0.15 0.003 CHEMBL3527224 0.055 0.014 CHEMBL1710849 0.12 0.004 CHEMBL3527010 0.194 0.002 CHEMBL3527226 0.186 0.002 CHEMBL3527068 | CHEMBL3527226 | |
| 0.139 | 0.035 | 0.139 | Nav1.5 sodium channel blocker | 0.102 0.082 CHEMBL3527225 0.102 0.082 CHEMBL3527226 0.1 0.085 CHEMBL3527068 | ||
| 0.107 | 0.004 | 0.166 | Sphingosine kinase 1 inhibitor | 0.101 0.004 CHEMBL3527225 0.127 0.004 CHEMBL3527224 0.166 0.003 CHEMBL1710849 0.111 0.004 CHEMBL3527010 0.101 0.004 CHEMBL3527226 0.117 0.004 CHEMBL3527068 | CHEMBL1710849 | |
| 0.146 | 0.046 | 0.146 | 5 Hydroxytryptamine 2 antagonist | 0.086 0.083 CHEMBL3527225 0.094 0.077 CHEMBL3527224 0.091 0.079 CHEMBL3527010 0.086 0.083 CHEMBL3527226 | ||
| 0.209 | 0.11 | 0.209 | Cardiotonic | 0.167 0.156 CHEMBL3527225 0.178 0.141 CHEMBL3527224 0.172 0.149 CHEMBL3527010 0.167 0.156 CHEMBL3527226 0.189 0.129 CHEMBL3527068 | ||
| 0.11 | 0.012 | 0.11 | Alpha 2 adrenoreceptor agonist | 0.09 0.018 CHEMBL3527225 0.094 0.017 CHEMBL3527224 0.066 0.035 CHEMBL3527010 0.09 0.018 CHEMBL3527226 0.1 0.015 CHEMBL3527068 | ||
| 0.109 | 0.013 | 0.109 | 5 Hydroxytryptamine 5 antagonist | 0.072 0.025 CHEMBL3527225 0.088 0.018 CHEMBL3527224 0.074 0.024 CHEMBL3527010 0.072 0.025 CHEMBL3527226 0.064 0.031 CHEMBL3527068 | ||
| 0.162 | 0.068 | 0.162 | Cholinergic | 0.142 0.083 CHEMBL3527225 0.121 0.106 CHEMBL3527224 0.134 0.091 CHEMBL3527010 0.142 0.083 CHEMBL3527226 0.145 0.08 CHEMBL3527068 | ||
| 0.101 | 0.007 | 0.101 | Lysine-specific demethylase 1A inhibitor | 0.091 0.009 CHEMBL3527225 0.08 0.012 CHEMBL3527224 0.101 0.006 CHEMBL3527010 0.091 0.009 CHEMBL3527226 0.093 0.008 CHEMBL3527068 | ||
| 0.151 | 0.058 | 0.189 | Bone formation stimulant | 0.189 0.039 CHEMBL3527225 0.146 0.062 CHEMBL3527224 0.155 0.055 CHEMBL3527010 0.189 0.039 CHEMBL3527226 0.174 0.044 CHEMBL3527068 | CHEMBL3527226 | |
| 0.097 | 0.004 | 0.097 | Trypsin II inhibitor | 0.07 0.006 CHEMBL3527225 0.069 0.006 CHEMBL3527224 0.075 0.005 CHEMBL1710849 0.069 0.006 CHEMBL3527010 0.07 0.006 CHEMBL3527226 0.074 0.005 CHEMBL3527068 | ||
| 0.099 | 0.007 | 0.099 | Factor VII inhibitor | 0.055 0.011 CHEMBL3527225 0.063 0.01 CHEMBL3527224 0.061 0.01 CHEMBL1710849 0.06 0.01 CHEMBL3527010 0.055 0.011 CHEMBL3527226 0.066 0.01 CHEMBL3527068 | ||
| 0.135 | 0.048 | 0.135 | 5 Hydroxytryptamine 2B antagonist | 0.101 0.083 CHEMBL3527225 0.119 0.062 CHEMBL3527224 0.101 0.083 CHEMBL3527226 | ||
| 0.09 | 0.005 | 0.09 | Plasma kallikrein inhibitor | 0.044 0.015 CHEMBL3527225 0.042 0.017 CHEMBL3527224 0.041 0.018 CHEMBL1710849 0.043 0.016 CHEMBL3527010 0.044 0.015 CHEMBL3527226 0.046 0.014 CHEMBL3527068 | ||
| 0.149 | 0.064 | 0.187 | Adenylate cyclase stimulant | 0.171 0.034 CHEMBL3527225 0.145 0.071 CHEMBL3527224 0.151 0.061 CHEMBL1710849 0.147 0.068 CHEMBL3527010 0.171 0.034 CHEMBL3527226 0.187 0.021 CHEMBL3527068 | CHEMBL3527068 | |
| 0.129 | 0.044 | 0.129 | GABA C receptor antagonist | 0.117 0.055 CHEMBL3527225 0.128 0.045 CHEMBL3527224 0.128 0.045 CHEMBL3527010 0.117 0.055 CHEMBL3527226 0.113 0.06 CHEMBL3527068 | ||
| 0.092 | 0.009 | 0.092 | Epithelial sodium channel blocker | 0.079 0.013 CHEMBL3527225 0.071 0.017 CHEMBL3527224 0.061 0.027 CHEMBL3527010 0.079 0.013 CHEMBL3527226 0.076 0.014 CHEMBL3527068 | ||
| 0.084 | 0.005 | 0.084 | Factor XI inhibitor | 0.05 0.01 CHEMBL3527225 0.052 0.009 CHEMBL3527224 0.04 0.016 CHEMBL1710849 0.047 0.011 CHEMBL3527010 0.05 0.01 CHEMBL3527226 0.056 0.008 CHEMBL3527068 | ||
| 0.083 | 0.004 | 0.083 | Phenylethanolamine N methyltransferase inhibitor | 0.071 0.005 CHEMBL3527225 0.057 0.009 CHEMBL3527224 0.049 0.016 CHEMBL1710849 0.06 0.008 CHEMBL3527010 0.071 0.005 CHEMBL3527226 0.072 0.005 CHEMBL3527068 | ||
| 0.091 | 0.012 | 0.091 | Potassium channel intermediate-conductance Ca-activated blocker | |||
| 0.104 | 0.028 | 0.156 | Glutamate decarboxylase inhibitor | 0.135 0.016 CHEMBL3527225 0.11 0.024 CHEMBL3527224 0.084 0.04 CHEMBL1710849 0.15 0.013 CHEMBL3527010 0.135 0.016 CHEMBL3527226 0.156 0.012 CHEMBL3527068 | CHEMBL3527068 | |
| 0.08 | 0.005 | 0.08 | Acid-sensing ion channel blocker | 0.067 0.007 CHEMBL3527225 0.065 0.008 CHEMBL3527224 0.048 0.018 CHEMBL1710849 0.067 0.007 CHEMBL3527010 0.067 0.007 CHEMBL3527226 0.067 0.007 CHEMBL3527068 | ||
| 0.117 | 0.042 | 0.119 | Factor V inhibitor | 0.103 0.063 CHEMBL3527225 0.104 0.061 CHEMBL3527224 0.119 0.04 CHEMBL1710849 0.104 0.061 CHEMBL3527010 0.103 0.063 CHEMBL3527226 0.105 0.059 CHEMBL3527068 | CHEMBL1710849 | |
| 0.079 | 0.005 | 0.079 | Endothelial nitric-oxide synthase inhibitor | 0.029 0.024 CHEMBL3527225 0.035 0.017 CHEMBL3527224 0.032 0.02 CHEMBL3527010 0.029 0.024 CHEMBL3527226 0.031 0.021 CHEMBL3527068 | ||
| 0.223 | 0.151 | 0.251 | Vasodilator, peripheral | 0.227 0.147 CHEMBL3527225 0.23 0.144 CHEMBL3527224 0.227 0.147 CHEMBL3527226 0.251 0.126 CHEMBL3527068 | CHEMBL3527068 | |
| 0.131 | 0.059 | 0.131 | 5 Hydroxytryptamine antagonist | |||
| 0.197 | 0.125 | 0.197 | Neuropeptide Y2 antagonist | 0.184 0.151 CHEMBL3527225 0.184 0.151 CHEMBL3527226 | ||
| 0.115 | 0.045 | 0.115 | GABA C receptor rho-1 antagonist | 0.1 0.063 CHEMBL3527225 0.107 0.053 CHEMBL3527224 0.107 0.053 CHEMBL3527010 0.1 0.063 CHEMBL3527226 0.089 0.08 CHEMBL3527068 | ||
| 0.089 | 0.023 | 0.093 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.068 0.065 CHEMBL3527224 0.093 0.019 CHEMBL1710849 0.068 0.065 CHEMBL3527010 0.07 0.06 CHEMBL3527068 | CHEMBL1710849 | |
| 0.164 | 0.099 | 0.179 | Anesthetic general | 0.169 0.096 CHEMBL3527225 0.16 0.103 CHEMBL3527010 0.169 0.096 CHEMBL3527226 0.179 0.087 CHEMBL3527068 | CHEMBL3527068 | |
| 0.13 | 0.065 | 0.13 | Glutamate receptor antagonist | 0.122 0.072 CHEMBL3527225 0.103 0.093 CHEMBL3527224 0.119 0.075 CHEMBL1710849 0.122 0.072 CHEMBL3527226 0.102 0.094 CHEMBL3527068 | ||
| 0.069 | 0.005 | 0.069 | Lysine carboxypeptidase inhibitor | 0.058 0.006 CHEMBL3527225 0.052 0.007 CHEMBL3527224 0.046 0.009 CHEMBL1710849 0.052 0.007 CHEMBL3527010 0.058 0.006 CHEMBL3527226 0.058 0.006 CHEMBL3527068 | ||
| 0.082 | 0.023 | 0.082 | 5 Hydroxytryptamine 3 antagonist | |||
| 0.067 | 0.01 | 0.067 | Nicotinamide phosphoribosyltransferase inhibitor | |||
| 0.113 | 0.057 | 0.119 | Electron transport complex I inhibitor | 0.115 0.054 CHEMBL3527225 0.111 0.06 CHEMBL3527224 0.112 0.06 CHEMBL3527010 0.115 0.054 CHEMBL3527226 0.119 0.048 CHEMBL3527068 | CHEMBL3527068 | |
| 0.112 | 0.057 | 0.112 | Aminopeptidase B inhibitor | 0.097 0.067 CHEMBL3527225 0.096 0.068 CHEMBL3527224 0.098 0.066 CHEMBL1710849 0.096 0.068 CHEMBL3527010 0.097 0.067 CHEMBL3527226 0.096 0.068 CHEMBL3527068 | ||
| 0.105 | 0.05 | 0.14 | Prolactin inhibitor | 0.136 0.029 CHEMBL3527225 0.14 0.027 CHEMBL3527224 0.135 0.029 CHEMBL3527010 0.136 0.029 CHEMBL3527226 0.123 0.036 CHEMBL3527068 | CHEMBL3527224 | |
| 0.064 | 0.009 | 0.064 | Guanylate cyclase inhibitor | 0.053 0.018 CHEMBL3527225 0.044 0.028 CHEMBL3527224 0.043 0.029 CHEMBL1710849 0.057 0.014 CHEMBL3527010 0.053 0.018 CHEMBL3527226 0.051 0.02 CHEMBL3527068 | ||
| 0.101 | 0.047 | 0.101 | Alpha 2 adrenoreceptor antagonist | 0.087 0.058 CHEMBL3527225 0.088 0.057 CHEMBL3527224 0.087 0.058 CHEMBL3527010 0.087 0.058 CHEMBL3527226 0.1 0.048 CHEMBL3527068 | ||
| 0.062 | 0.008 | 0.062 | Nerve growth factor antagonist | 0.047 0.022 CHEMBL3527225 0.039 0.038 CHEMBL3527224 0.042 0.031 CHEMBL3527010 0.047 0.022 CHEMBL3527226 0.056 0.012 CHEMBL3527068 | ||
| 0.056 | 0.005 | 0.056 | Bradykinin B2 receptor antagonist | 0.042 0.014 CHEMBL3527225 0.04 0.016 CHEMBL3527224 0.052 0.006 CHEMBL1710849 0.037 0.018 CHEMBL3527010 0.042 0.014 CHEMBL3527226 0.042 0.014 CHEMBL3527068 | ||
| 0.123 | 0.071 | 0.123 | Cathepsin H inhibitor | 0.109 0.09 CHEMBL1710849 | ||
| 0.076 | 0.026 | 0.076 | 5 Hydroxytryptamine 5A antagonist | 0.061 0.043 CHEMBL3527225 0.069 0.033 CHEMBL3527224 0.061 0.042 CHEMBL3527010 0.061 0.043 CHEMBL3527226 0.056 0.052 CHEMBL3527068 | ||
| 0.111 | 0.06 | 0.111 | Ferrochelatase inhibitor | 0.094 0.078 CHEMBL1710849 | ||
| 0.093 | 0.043 | 0.139 | Opioid kappa receptor antagonist | 0.139 0.019 CHEMBL3527225 0.074 0.067 CHEMBL3527224 0.085 0.052 CHEMBL3527010 0.139 0.019 CHEMBL3527226 0.104 0.031 CHEMBL3527068 | CHEMBL3527226 | |
| 0.058 | 0.009 | 0.058 | Histamine H1 receptor agonist | |||
| 0.103 | 0.056 | 0.186 | Creatine kinase inhibitor | 0.186 0.013 CHEMBL3527225 0.15 0.024 CHEMBL3527224 0.121 0.041 CHEMBL1710849 0.174 0.016 CHEMBL3527010 0.186 0.013 CHEMBL3527226 0.168 0.017 CHEMBL3527068 | CHEMBL3527226 | |
| 0.088 | 0.042 | 0.088 | Nicotinic alpha4beta2 receptor antagonist | |||
| 0.071 | 0.025 | 0.229 | NMDA 2B receptor antagonist | 0.106 0.014 CHEMBL3527225 0.05 0.043 CHEMBL3527224 0.229 0.005 CHEMBL1710849 0.106 0.014 CHEMBL3527226 0.078 0.022 CHEMBL3527068 | CHEMBL1710849 | |
| 0.069 | 0.024 | 0.094 | Opioid agonist | 0.094 0.015 CHEMBL3527225 0.054 0.035 CHEMBL3527224 0.057 0.032 CHEMBL1710849 0.055 0.034 CHEMBL3527010 0.094 0.015 CHEMBL3527226 0.071 0.023 CHEMBL3527068 | CHEMBL3527226 | |
| 0.071 | 0.026 | 0.071 | Corticotropin releasing factor 2 receptor antagonist | |||
| 0.068 | 0.023 | 0.077 | Bcl-xL inhibitor | 0.065 0.028 CHEMBL3527225 0.065 0.028 CHEMBL3527226 0.077 0.013 CHEMBL3527068 | CHEMBL3527068 | |
| 0.107 | 0.063 | 0.161 | DOPA decarboxylase inhibitor | 0.161 0.016 CHEMBL3527225 0.152 0.02 CHEMBL3527224 0.147 0.023 CHEMBL3527010 0.161 0.016 CHEMBL3527226 0.16 0.017 CHEMBL3527068 | CHEMBL3527226 | |
| 0.06 | 0.018 | 0.131 | Factor III inhibitor | 0.065 0.013 CHEMBL3527225 0.054 0.025 CHEMBL3527224 0.047 0.044 CHEMBL1710849 0.131 0.004 CHEMBL3527010 0.065 0.013 CHEMBL3527226 0.064 0.014 CHEMBL3527068 | CHEMBL3527010 | |
| 0.135 | 0.094 | 0.141 | Ca2+-transporting ATPase inhibitor | 0.13 0.118 CHEMBL3527225 0.135 0.093 CHEMBL3527224 0.141 0.069 CHEMBL1710849 0.133 0.105 CHEMBL3527010 0.13 0.118 CHEMBL3527226 0.135 0.093 CHEMBL3527068 | CHEMBL1710849 | |
| 0.094 | 0.053 | 0.147 | Opioid antagonist | 0.147 0.027 CHEMBL3527225 0.082 0.067 CHEMBL3527224 0.098 0.049 CHEMBL3527010 0.147 0.027 CHEMBL3527226 0.109 0.042 CHEMBL3527068 | CHEMBL3527226 | |
| 0.065 | 0.024 | 0.065 | 5 Hydroxytryptamine 7 agonist | 0.063 0.027 CHEMBL3527225 0.063 0.027 CHEMBL3527226 0.051 0.05 CHEMBL3527068 | ||
| 0.092 | 0.051 | 0.092 | 5 Hydroxytryptamine 2A antagonist | |||
| 0.069 | 0.029 | 0.096 | Protein kinase C eta inhibitor | 0.078 0.024 CHEMBL3527225 0.06 0.034 CHEMBL3527224 0.096 0.018 CHEMBL1710849 0.067 0.03 CHEMBL3527010 0.078 0.024 CHEMBL3527226 0.071 0.028 CHEMBL3527068 | CHEMBL1710849 | |
| 0.133 | 0.094 | 0.136 | Neuropeptide Y1 antagonist | 0.136 0.088 CHEMBL3527225 0.136 0.088 CHEMBL3527226 | CHEMBL3527226 | |
| 0.088 | 0.049 | 0.088 | Histamine H2 receptor antagonist | |||
| 0.095 | 0.057 | 0.12 | Adrenaline antagonist | 0.086 0.063 CHEMBL3527225 0.12 0.043 CHEMBL3527224 0.088 0.062 CHEMBL3527010 0.086 0.063 CHEMBL3527226 0.095 0.057 CHEMBL3527068 | CHEMBL3527224 | |
| 0.209 | 0.172 | 0.209 | Ca(v)3.3 blocker | |||
| 0.051 | 0.015 | 0.051 | Membrane dipeptidase inhibitor | 0.036 0.032 CHEMBL3527225 0.036 0.034 CHEMBL3527224 0.04 0.027 CHEMBL1710849 0.038 0.03 CHEMBL3527010 0.036 0.032 CHEMBL3527226 0.043 0.023 CHEMBL3527068 | ||
| 0.095 | 0.06 | 0.095 | Alpha adrenoreceptor antagonist | 0.076 0.075 CHEMBL3527225 0.076 0.075 CHEMBL3527226 0.08 0.072 CHEMBL3527068 | ||
| 0.071 | 0.036 | 0.071 | Acetylcholine M2 receptor antagonist | 0.055 0.049 CHEMBL3527225 0.055 0.049 CHEMBL3527226 | ||
| 0.05 | 0.015 | 0.05 | Bradykinin antagonist | |||
| 0.059 | 0.027 | 0.059 | Dipeptidyl peptidase inhibitor | |||
| 0.056 | 0.023 | 0.056 | Histamine H3 receptor antagonist | |||
| 0.073 | 0.043 | 0.073 | Alpha adrenoreceptor agonist | 0.063 0.052 CHEMBL3527225 0.063 0.052 CHEMBL3527224 0.063 0.052 CHEMBL3527226 0.067 0.048 CHEMBL3527068 | ||
| 0.047 | 0.017 | 0.059 | Arginase inhibitor | 0.051 0.015 CHEMBL3527225 0.041 0.021 CHEMBL3527224 0.036 0.026 CHEMBL1710849 0.042 0.021 CHEMBL3527010 0.051 0.015 CHEMBL3527226 0.059 0.011 CHEMBL3527068 | CHEMBL3527068 | |
| 0.047 | 0.017 | 0.047 | Vascular adhesion protein 1 inhibitor | |||
| 0.04 | 0.011 | 0.042 | Protein kinase C beta II inhibitor | 0.039 0.012 CHEMBL3527225 0.036 0.015 CHEMBL3527224 0.042 0.01 CHEMBL1710849 0.035 0.017 CHEMBL3527010 0.039 0.012 CHEMBL3527226 0.037 0.015 CHEMBL3527068 | CHEMBL1710849 | |
| 0.073 | 0.045 | 0.073 | CXC chemokine receptor antagonist | |||
| 0.036 | 0.008 | 0.044 | Estrogen-related receptor gamma antagonist | 0.044 0.004 CHEMBL3527225 0.042 0.004 CHEMBL3527224 0.033 0.01 CHEMBL1710849 0.042 0.004 CHEMBL3527010 0.044 0.004 CHEMBL3527226 0.039 0.005 CHEMBL3527068 | CHEMBL3527226 | |
| 0.217 | 0.189 | 0.217 | Calcium channel activator | |||
| 0.09 | 0.062 | 0.09 | Glutamate release inhibitor | 0.088 0.066 CHEMBL3527224 | ||
| 0.109 | 0.082 | 0.186 | MAO inhibitor | 0.173 0.05 CHEMBL3527225 0.186 0.045 CHEMBL3527224 0.174 0.05 CHEMBL3527010 0.173 0.05 CHEMBL3527226 0.138 0.066 CHEMBL3527068 | CHEMBL3527224 | |
| 0.113 | 0.085 | 0.213 | Alpha-N-acetylglucosaminidase inhibitor | 0.213 0.03 CHEMBL1710849 0.113 0.085 CHEMBL3527068 | CHEMBL1710849 | |
| 0.082 | 0.055 | 0.082 | Histamine H1 receptor antagonist | |||
| 0.072 | 0.046 | 0.072 | 5 Hydroxytryptamine agonist | |||
| 0.061 | 0.035 | 0.061 | 5 Hydroxytryptamine 6 antagonist | |||
| 0.049 | 0.022 | 0.049 | Dipeptidyl peptidase IV inhibitor | |||
| 0.039 | 0.014 | 0.039 | Carboxypeptidase B inhibitor | 0.034 0.022 CHEMBL3527225 0.034 0.02 CHEMBL3527224 0.033 0.023 CHEMBL1710849 0.034 0.021 CHEMBL3527010 0.034 0.022 CHEMBL3527226 0.035 0.019 CHEMBL3527068 | ||
| 0.046 | 0.021 | 0.087 | NMDA receptor subunit 3A antagonist | 0.087 0.01 CHEMBL3527225 0.061 0.016 CHEMBL3527224 0.079 0.012 CHEMBL3527010 0.087 0.01 CHEMBL3527226 0.06 0.017 CHEMBL3527068 | CHEMBL3527226 | |
| 0.056 | 0.032 | 0.056 | Histamine agonist | |||
| 0.06 | 0.036 | 0.097 | Argininosuccinate synthase inhibitor | 0.049 0.048 CHEMBL3527224 0.097 0.02 CHEMBL1710849 0.049 0.048 CHEMBL3527010 0.058 0.038 CHEMBL3527068 | CHEMBL1710849 | |
| 0.06 | 0.038 | 0.064 | Neuropeptide agonist | 0.055 0.04 CHEMBL3527225 0.064 0.037 CHEMBL1710849 0.055 0.04 CHEMBL3527226 0.046 0.045 CHEMBL3527068 | CHEMBL1710849 | |
| 0.129 | 0.107 | 0.129 | GABA C receptor rho-2 antagonist | 0.122 0.121 CHEMBL3527225 0.129 0.108 CHEMBL3527224 0.129 0.108 CHEMBL3527010 0.122 0.121 CHEMBL3527226 | ||
| 0.029 | 0.009 | 0.029 | Integrin beta5 antagonist | 0.02 0.015 CHEMBL3527225 0.019 0.017 CHEMBL3527224 0.025 0.011 CHEMBL1710849 0.02 0.015 CHEMBL3527010 0.02 0.015 CHEMBL3527226 0.023 0.012 CHEMBL3527068 | ||
| 0.143 | 0.123 | 0.167 | Psychostimulant | 0.159 0.108 CHEMBL3527224 0.167 0.102 CHEMBL1710849 0.145 0.12 CHEMBL3527010 | CHEMBL1710849 | |
| 0.047 | 0.027 | 0.073 | Dopamine D5 antagonist | 0.062 0.018 CHEMBL3527225 0.064 0.017 CHEMBL3527224 0.063 0.018 CHEMBL3527010 0.062 0.018 CHEMBL3527226 0.073 0.014 CHEMBL3527068 | CHEMBL3527068 | |
| 0.039 | 0.02 | 0.053 | Opioid delta receptor agonist | 0.053 0.012 CHEMBL3527225 0.035 0.024 CHEMBL3527224 0.035 0.025 CHEMBL3527010 0.053 0.012 CHEMBL3527226 0.04 0.019 CHEMBL3527068 | CHEMBL3527226 | |
| 0.036 | 0.017 | 0.039 | Protein kinase C beta I inhibitor | 0.036 0.017 CHEMBL3527225 0.034 0.021 CHEMBL3527224 0.039 0.01 CHEMBL1710849 0.034 0.02 CHEMBL3527010 0.036 0.017 CHEMBL3527226 0.034 0.023 CHEMBL3527068 | CHEMBL1710849 | |
| 0.045 | 0.027 | 0.045 | Histamine H2 receptor agonist | |||
| 0.041 | 0.022 | 0.041 | Diamine oxidase inhibitor | |||
| 0.036 | 0.018 | 0.036 | Dipeptidyl peptidase II inhibitor | |||
| 0.071 | 0.056 | 0.079 | Alpha 2a adrenoreceptor antagonist | 0.068 0.06 CHEMBL3527225 0.069 0.058 CHEMBL3527224 0.067 0.061 CHEMBL3527010 0.068 0.06 CHEMBL3527226 0.079 0.049 CHEMBL3527068 | CHEMBL3527068 | |
| 0.175 | 0.16 | 0.225 | DNA synthesis inhibitor | 0.192 0.136 CHEMBL3527225 0.207 0.113 CHEMBL3527224 0.225 0.088 CHEMBL1710849 0.19 0.138 CHEMBL3527010 0.192 0.136 CHEMBL3527226 0.197 0.127 CHEMBL3527068 | CHEMBL1710849 | |
| 0.062 | 0.047 | 0.062 | Glucagon-like peptide 1 agonist | 0.062 0.047 CHEMBL3527225 0.062 0.047 CHEMBL3527226 | ||
| 0.069 | 0.055 | 0.079 | Aminopeptidase I inhibitor | 0.079 0.043 CHEMBL1710849 | CHEMBL1710849 | |
| 0.047 | 0.033 | 0.047 | Melanocortin antagonist | |||
| 0.024 | 0.01 | 0.024 | Melatonin 3 antagonist | |||
| 0.099 | 0.085 | 0.148 | Adenylate cyclase inhibitor | 0.126 0.062 CHEMBL3527225 0.107 0.078 CHEMBL3527224 0.099 0.085 CHEMBL1710849 0.126 0.062 CHEMBL3527226 0.148 0.046 CHEMBL3527068 | CHEMBL3527068 | |
| 0.08 | 0.068 | 0.08 | mTOR complex 2 inhibitor | |||
| 0.058 | 0.045 | 0.067 | Ryanodine receptor antagonist | 0.067 0.022 CHEMBL3527225 0.058 0.044 CHEMBL3527224 0.062 0.033 CHEMBL1710849 0.058 0.044 CHEMBL3527010 0.067 0.022 CHEMBL3527226 0.066 0.023 CHEMBL3527068 | CHEMBL3527226 | |
| 0.21 | 0.197 | 0.21 | Antiobesity | |||
| 0.023 | 0.011 | 0.023 | Imidazoline I1 receptor antagonist | |||
| 0.045 | 0.033 | 0.045 | Farnesyltransferase inhibitor | |||
| 0.038 | 0.027 | 0.038 | Melanocortin 1 antagonist | |||
| 0.039 | 0.028 | 0.039 | AMPA 4 receptor antagonist | |||
| 0.029 | 0.018 | 0.029 | 5 Hydroxytryptamine 6 agonist | |||
| 0.043 | 0.032 | 0.081 | NMDA receptor subunit 3B antagonist | 0.081 0.013 CHEMBL3527225 0.052 0.024 CHEMBL3527224 0.063 0.018 CHEMBL3527010 0.081 0.013 CHEMBL3527226 0.054 0.022 CHEMBL3527068 | CHEMBL3527226 | |
| 0.075 | 0.065 | 0.075 | Glycine receptor antagonist | 0.073 0.07 CHEMBL1710849 | ||
| 0.044 | 0.035 | 0.077 | Opioid mu receptor agonist | 0.077 0.018 CHEMBL3527225 0.077 0.018 CHEMBL3527226 0.05 0.029 CHEMBL3527068 | CHEMBL3527226 | |
| 0.043 | 0.035 | 0.095 | Mannosidase inhibitor | 0.095 0.006 CHEMBL1710849 0.042 0.037 CHEMBL3527068 | CHEMBL1710849 | |
| 0.018 | 0.011 | 0.023 | Sodium/hydrogen exchanger inhibitor | 0.023 0.006 CHEMBL1710849 | CHEMBL1710849 | |
| 0.02 | 0.013 | 0.02 | Integrin beta3 antagonist | |||
| 0.07 | 0.063 | 0.07 | Potassium channel (Tandem pore domain) blocker | |||
| 0.049 | 0.042 | 0.049 | Protein kinase C epsilon inhibitor | |||
| 0.093 | 0.087 | 0.106 | Nav1.4 sodium channel blocker | 0.106 0.068 CHEMBL3527225 0.096 0.082 CHEMBL3527010 0.106 0.068 CHEMBL3527226 | CHEMBL3527226 | |
| 0.037 | 0.031 | 0.037 | 5 Hydroxytryptamine 2B agonist | |||
| 0.121 | 0.116 | 0.121 | Thiol protease inhibitor | |||
| 0.047 | 0.043 | 0.067 | Factor IXa inhibitor | 0.047 0.041 CHEMBL3527225 0.067 0.022 CHEMBL1710849 0.047 0.041 CHEMBL3527226 | CHEMBL1710849 | |
| 0.042 | 0.039 | 0.042 | Glycine transporter inhibitor | |||
| 0.066 | 0.063 | 0.067 | Glycine receptor agonist | 0.067 0.061 CHEMBL1710849 | CHEMBL1710849 | |
| 0.122 | 0.119 | 0.122 | Sphingosine 1-phosphate receptor 5 antagonist | |||
| 0.037 | 0.035 | 0.049 | Oxytocin agonist | 0.049 0.025 CHEMBL3527225 0.039 0.033 CHEMBL3527224 0.04 0.032 CHEMBL3527010 0.049 0.025 CHEMBL3527226 0.042 0.029 CHEMBL3527068 | CHEMBL3527226 | |
| 0.059 | 0.057 | 0.081 | Neuraminidase (influenza) inhibitor | 0.071 0.033 CHEMBL3527225 0.068 0.038 CHEMBL3527224 0.08 0.025 CHEMBL1710849 0.068 0.037 CHEMBL3527010 0.071 0.033 CHEMBL3527226 0.081 0.024 CHEMBL3527068 | CHEMBL3527068 | |
| 0.01 | 0.009 | 0.01 | Melatonin 5 antagonist | |||
| 0.114 | 0.113 | 0.118 | Diuretic | 0.118 0.107 CHEMBL3527068 | CHEMBL3527068 | |
| 0.054 | 0.053 | 0.054 | 5 Hydroxytryptamine 2A agonist | |||
| 0.023 | 0.022 | 0.023 | Melanocortin 5 antagonist | |||
| 0.048 | 0.049 | 0.049 | Alpha 1L adrenoreceptor antagonist | 0.049 0.047 CHEMBL3527225 0.049 0.047 CHEMBL3527226 0.049 0.047 CHEMBL3527068 | CHEMBL3527068 | |
| 0.051 | 0.053 | 0.067 | Acetylcholine M3 receptor antagonist | 0.054 0.048 CHEMBL3527225 0.067 0.034 CHEMBL1710849 0.054 0.048 CHEMBL3527226 | CHEMBL1710849 | |
| 0.136 | 0.138 | 0.168 | Phospholipase C inhibitor | 0.157 0.093 CHEMBL3527225 0.14 0.128 CHEMBL3527224 0.168 0.076 CHEMBL1710849 0.144 0.119 CHEMBL3527010 0.157 0.093 CHEMBL3527226 0.161 0.087 CHEMBL3527068 | CHEMBL1710849 | |
| 0.051 | 0.053 | 0.116 | Opioid delta receptor antagonist | 0.116 0.027 CHEMBL3527225 0.116 0.027 CHEMBL3527226 0.072 0.039 CHEMBL3527068 | CHEMBL3527226 | |
| 0.047 | 0.05 | 0.086 | Alpha-mannosidase inhibitor | 0.086 0.009 CHEMBL1710849 | CHEMBL1710849 | |
| 0.012 | 0.016 | 0.014 | NMDA receptor phencyclidine site antagonist | 0.014 0.012 CHEMBL3527225 0.014 0.012 CHEMBL3527226 | CHEMBL3527226 | |
| 0.076 | 0.082 | 0.086 | CC chemokine 5 receptor agonist | 0.086 0.047 CHEMBL3527225 0.086 0.047 CHEMBL3527226 0.077 0.074 CHEMBL3527068 | CHEMBL3527226 | |
| 0.043 | 0.049 | 0.049 | Dopamine beta hydroxylase inhibitor | 0.046 0.04 CHEMBL3527225 0.046 0.04 CHEMBL3527226 0.049 0.032 CHEMBL3527068 | CHEMBL3527068 | |
| 0.049 | 0.056 | 0.084 | Carbamoyl phosphate synthetase inhibitor | 0.084 0.027 CHEMBL1710849 0.053 0.052 CHEMBL3527068 | CHEMBL1710849 | |
| 0.109 | 0.117 | 0.136 | Cell wall synthesis inhibitor | 0.118 0.103 CHEMBL3527225 0.118 0.103 CHEMBL3527224 0.125 0.093 CHEMBL1710849 0.118 0.103 CHEMBL3527226 0.136 0.08 CHEMBL3527068 | CHEMBL3527068 | |
| 0.059 | 0.068 | 0.07 | Telomerase inhibitor | 0.07 0.052 CHEMBL3527068 | CHEMBL3527068 | |
| 0.04 | 0.05 | 0.062 | Ornithine carbamoyltransferase inhibitor | 0.062 0.03 CHEMBL1710849 | CHEMBL1710849 | |
| 0.052 | 0.064 | 0.106 | Opioid mu receptor antagonist | 0.106 0.029 CHEMBL3527225 0.106 0.029 CHEMBL3527226 0.069 0.046 CHEMBL3527068 | CHEMBL3527226 | |
| 0.184 | 0.197 | 0.225 | Vasodilator, coronary | 0.225 0.159 CHEMBL3527010 0.21 0.173 CHEMBL3527068 | CHEMBL3527010 | |
| 0.081 | 0.095 | 0.107 | Anabolic | 0.107 0.053 CHEMBL3527225 0.087 0.085 CHEMBL1710849 0.097 0.067 CHEMBL3527010 0.107 0.053 CHEMBL3527226 0.103 0.058 CHEMBL3527068 | CHEMBL3527226 | |
| 0.05 | 0.065 | 0.085 | Dopamine D1 antagonist | 0.082 0.032 CHEMBL3527225 0.079 0.033 CHEMBL3527224 0.085 0.03 CHEMBL3527010 0.082 0.032 CHEMBL3527226 0.084 0.031 CHEMBL3527068 | CHEMBL3527010 | |
| 0.069 | 0.085 | 0.094 | MAP kinase kinase 7 inhibitor | 0.094 0.019 CHEMBL3527225 0.083 0.039 CHEMBL3527224 0.075 0.064 CHEMBL1710849 0.083 0.039 CHEMBL3527010 0.094 0.019 CHEMBL3527226 0.084 0.036 CHEMBL3527068 | CHEMBL3527226 | |
| 0.056 | 0.076 | 0.068 | Prolactin release inhibitor | 0.068 0.026 CHEMBL3527224 0.059 0.056 CHEMBL3527010 | CHEMBL3527224 | |
| 0.031 | 0.054 | 0.106 | Acetyl-CoA carboxylase inhibitor | 0.106 0.004 CHEMBL1710849 | CHEMBL1710849 | |
| 0.077 | 0.1 | 0.115 | Expectorant | 0.099 0.07 CHEMBL3527225 0.097 0.072 CHEMBL3527224 0.098 0.071 CHEMBL1710849 0.087 0.086 CHEMBL3527010 0.099 0.07 CHEMBL3527226 0.115 0.054 CHEMBL3527068 | CHEMBL3527068 | |
| 0.073 | 0.097 | 0.082 | Granulocyte macrophage colony stimulating factor agonist | 0.082 0.07 CHEMBL3527068 | CHEMBL3527068 | |
| 0.133 | 0.157 | 0.161 | Insulin sensitizer | 0.157 0.124 CHEMBL3527225 0.157 0.124 CHEMBL3527226 0.161 0.118 CHEMBL3527068 | CHEMBL3527068 | |
| 0.05 | 0.074 | 0.075 | Phenylalanine 4-hydroxylase inhibitor | 0.07 0.046 CHEMBL3527225 0.07 0.046 CHEMBL3527224 0.075 0.042 CHEMBL1710849 0.07 0.046 CHEMBL3527010 0.07 0.046 CHEMBL3527226 0.075 0.041 CHEMBL3527068 | CHEMBL3527068 | |
| 0.1 | 0.126 | 0.255 | Peroxidase inhibitor | 0.255 0.046 CHEMBL3527225 0.233 0.051 CHEMBL3527224 0.125 0.095 CHEMBL1710849 0.233 0.051 CHEMBL3527010 0.255 0.046 CHEMBL3527226 0.251 0.047 CHEMBL3527068 | CHEMBL3527226 | |
| 0.042 | 0.069 | 0.074 | Neuraminidase inhibitor | 0.06 0.043 CHEMBL3527225 0.055 0.05 CHEMBL3527224 0.068 0.035 CHEMBL1710849 0.058 0.046 CHEMBL3527010 0.06 0.043 CHEMBL3527226 0.074 0.03 CHEMBL3527068 | CHEMBL3527068 | |
| 0.015 | 0.043 | 0.047 | Dopamine D1 agonist | 0.024 0.014 CHEMBL3527225 0.047 0.005 CHEMBL3527224 0.033 0.008 CHEMBL3527010 0.024 0.014 CHEMBL3527226 0.034 0.007 CHEMBL3527068 | CHEMBL3527224 | |
| 0.067 | 0.097 | 0.124 | MAO A inhibitor | 0.11 0.058 CHEMBL3527225 0.117 0.054 CHEMBL3527224 0.124 0.05 CHEMBL3527010 0.11 0.058 CHEMBL3527226 0.087 0.073 CHEMBL3527068 | CHEMBL3527010 | |
| 0.017 | 0.048 | 0.027 | Bradykinin B2 receptor agonist | 0.027 0.021 CHEMBL1710849 | CHEMBL1710849 | |
| 0.081 | 0.114 | 0.122 | Adenylate kinase inhibitor | 0.122 0.042 CHEMBL1710849 | CHEMBL1710849 | |
| 0.032 | 0.066 | 0.041 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.041 0.031 CHEMBL3527068 | CHEMBL3527068 | |
| 0.024 | 0.059 | 0.096 | Dopamine D2 agonist | 0.044 0.031 CHEMBL3527225 0.096 0.011 CHEMBL3527224 0.06 0.021 CHEMBL3527010 0.044 0.031 CHEMBL3527226 0.054 0.024 CHEMBL3527068 | CHEMBL3527224 | |
| 0.036 | 0.071 | 0.065 | Alcohol oxidase inhibitor | 0.055 0.039 CHEMBL3527225 0.065 0.032 CHEMBL1710849 0.055 0.039 CHEMBL3527226 | CHEMBL1710849 | |
| 0.026 | 0.062 | 0.042 | Opioid kappa receptor agonist | 0.042 0.031 CHEMBL3527225 0.042 0.031 CHEMBL3527226 | CHEMBL3527226 | |
| 0.127 | 0.163 | 0.161 | Succinate dehydrogenase inhibitor | 0.139 0.134 CHEMBL3527225 0.139 0.134 CHEMBL3527226 0.161 0.093 CHEMBL3527068 | CHEMBL3527068 | |
| 0.01 | 0.048 | 0.077 | Acetyl-CoA carboxylase 2 inhibitor | 0.077 0.004 CHEMBL1710849 | CHEMBL1710849 | |
| 0.031 | 0.07 | 0.043 | Neuraminidase (Influenza A) inhibitor | 0.043 0.036 CHEMBL1710849 | CHEMBL1710849 | |
| 0.106 | 0.147 | 0.129 | Growth hormone agonist | 0.125 0.113 CHEMBL3527225 0.123 0.116 CHEMBL3527224 0.129 0.109 CHEMBL1710849 0.123 0.116 CHEMBL3527010 0.125 0.113 CHEMBL3527226 | CHEMBL1710849 | |
| 0.03 | 0.078 | 0.052 | Protein 50S ribosomal subunit inhibitor | 0.052 0.038 CHEMBL1710849 | CHEMBL1710849 | |
| 0.051 | 0.1 | 0.073 | Glutamate dehydrogenase inhibitor | 0.073 0.052 CHEMBL1710849 | CHEMBL1710849 | |
| 0.092 | 0.142 | 0.128 | Protein kinase stimulant | 0.124 0.088 CHEMBL3527225 0.124 0.088 CHEMBL3527226 0.128 0.085 CHEMBL3527068 | CHEMBL3527068 | |
| 0.036 | 0.087 | 0.067 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.067 0.028 CHEMBL1710849 | CHEMBL1710849 | |
| 0.039 | 0.091 | 0.074 | Glucosylceramidase inhibitor | 0.074 0.019 CHEMBL1710849 | CHEMBL1710849 | |
| 0.035 | 0.087 | 0.059 | Biliverdin reductase inhibitor | 0.059 0.041 CHEMBL1710849 | CHEMBL1710849 | |
| 0.075 | 0.128 | 0.104 | Mucolytic | 0.101 0.076 CHEMBL3527224 0.093 0.088 CHEMBL1710849 0.104 0.073 CHEMBL3527068 | CHEMBL3527068 | |
| 0.031 | 0.084 | 0.052 | Acyl-CoA dehydrogenase inhibitor | 0.052 0.041 CHEMBL1710849 | CHEMBL1710849 | |
| 0.09 | 0.144 | 0.109 | Transcription factor STAT6 inhibitor | 0.109 0.083 CHEMBL3527224 | CHEMBL3527224 | |
| 0.098 | 0.158 | 0.121 | Vanilloid 1 agonist | 0.113 0.105 CHEMBL3527224 0.121 0.086 CHEMBL3527068 | CHEMBL3527068 | |
| 0.063 | 0.124 | 0.091 | Triose-phosphate isomerase inhibitor | 0.091 0.059 CHEMBL1710849 | CHEMBL1710849 | |
| 0.185 | 0.248 | 0.315 | Antibacterial | 0.24 0.187 CHEMBL3527225 0.288 0.144 CHEMBL3527224 0.293 0.14 CHEMBL1710849 0.315 0.124 CHEMBL3527010 0.24 0.187 CHEMBL3527226 0.275 0.155 CHEMBL3527068 | CHEMBL3527010 | |
| 0.063 | 0.127 | 0.098 | NADH dehydrogenase inhibitor | 0.098 0.046 CHEMBL1710849 | CHEMBL1710849 | |
| 0.034 | 0.103 | 0.067 | Phosphofructokinase-1 inhibitor | 0.067 0.05 CHEMBL1710849 | CHEMBL1710849 | |
| 0.052 | 0.122 | 0.072 | Keratolytic | 0.072 0.061 CHEMBL3527225 0.072 0.061 CHEMBL3527010 0.072 0.061 CHEMBL3527226 0.071 0.064 CHEMBL3527068 | CHEMBL3527226 | |
| 0.143 | 0.217 | 0.183 | RNA-directed DNA polymerase inhibitor | 0.183 0.127 CHEMBL3527224 0.171 0.15 CHEMBL1710849 0.181 0.13 CHEMBL3527068 | CHEMBL3527224 | |
| 0.148 | 0.226 | 0.182 | Gastrin inhibitor | 0.182 0.176 CHEMBL1710849 | CHEMBL1710849 | |
| 0.115 | 0.195 | 0.209 | Immunostimulant | 0.209 0.115 CHEMBL1710849 0.169 0.14 CHEMBL3527010 | CHEMBL1710849 | |
| 0.032 | 0.117 | 0.119 | Dopamine agonist | 0.119 0.02 CHEMBL3527224 0.083 0.035 CHEMBL3527010 0.069 0.045 CHEMBL3527068 | CHEMBL3527224 | |
| 0.021 | 0.117 | 0.033 | Antibiotic Aminoglycoside-like | 0.033 0.03 CHEMBL1710849 | CHEMBL1710849 | |
| 0.062 | 0.163 | 0.08 | Estrogen-related receptor beta agonist | 0.08 0.068 CHEMBL3527225 0.08 0.068 CHEMBL3527226 | CHEMBL3527226 | |
| 0.11 | 0.215 | 0.162 | Spasmolytic | 0.162 0.152 CHEMBL1710849 | CHEMBL1710849 | |
| 0.054 | 0.162 | 0.093 | UDP-glucose 4-epimerase inhibitor | 0.093 0.069 CHEMBL1710849 | CHEMBL1710849 | |
| 0.056 | 0.166 | 0.117 | Cystathionine beta-synthase inhibitor | 0.117 0.06 CHEMBL3527225 0.106 0.07 CHEMBL3527224 0.106 0.07 CHEMBL3527010 0.117 0.06 CHEMBL3527226 0.109 0.067 CHEMBL3527068 | CHEMBL3527226 | |
| 0.036 | 0.145 | 0.055 | Heat shock protein 90 beta antagonist | 0.054 0.052 CHEMBL3527224 0.055 0.049 CHEMBL3527068 | CHEMBL3527068 | |
| 0.093 | 0.208 | 0.14 | Melanin inhibitor | 0.14 0.097 CHEMBL3527225 0.128 0.119 CHEMBL3527224 0.132 0.111 CHEMBL3527010 0.14 0.097 CHEMBL3527226 0.136 0.103 CHEMBL3527068 | CHEMBL3527226 | |
| 0.091 | 0.207 | 0.163 | Interleukin antagonist | 0.163 0.109 CHEMBL3527225 0.137 0.128 CHEMBL3527224 0.163 0.109 CHEMBL3527226 | CHEMBL3527226 | |
| 0.05 | 0.168 | 0.081 | Estrogen receptor alpha antagonist | 0.081 0.047 CHEMBL3527225 0.081 0.047 CHEMBL3527226 | CHEMBL3527226 | |
| 0.136 | 0.261 | 0.176 | Nitric-oxide synthase stimulant | 0.168 0.158 CHEMBL1710849 0.176 0.138 CHEMBL3527068 | CHEMBL3527068 | |
| 0.163 | 0.304 | 0.199 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.199 0.17 CHEMBL3527224 | CHEMBL3527224 | |
| 0.187 | 0.341 | 0.264 | Caspase 9 stimulant | 0.264 0.236 CHEMBL3527225 0.258 0.244 CHEMBL3527010 0.264 0.236 CHEMBL3527226 0.263 0.238 CHEMBL3527068 | CHEMBL3527226 | |
| 0.124 | 0.289 | 0.228 | Peptidyltransferase inhibitor | 0.167 0.154 CHEMBL3527225 0.185 0.12 CHEMBL3527224 0.228 0.068 CHEMBL1710849 0.185 0.12 CHEMBL3527010 0.167 0.154 CHEMBL3527226 0.186 0.119 CHEMBL3527068 | CHEMBL1710849 | |
| 0.082 | 0.279 | 0.113 | Papain-like protease (SARS coronavirus) inhibitor | 0.113 0.101 CHEMBL3527225 0.113 0.101 CHEMBL3527226 | CHEMBL3527226 | |
| 0.135 | 0.443 | 0.253 | Calcium channel L-type activator | 0.253 0.202 CHEMBL3527225 0.253 0.202 CHEMBL3527226 | CHEMBL3527226 | |
| 0.073 | 0.394 | 0.218 | Hypoglycemic | 0.165 0.155 CHEMBL1710849 0.218 0.097 CHEMBL3527010 | CHEMBL3527010 | |
| 0.025 | 0.415 | 0.127 | Estrogen receptor beta antagonist | 0.127 0.026 CHEMBL3527225 0.099 0.066 CHEMBL3527224 0.1 0.065 CHEMBL3527010 0.127 0.026 CHEMBL3527226 0.098 0.069 CHEMBL3527068 | CHEMBL3527226 | |
| 0.017 | 0.409 | 0.069 | HIV-1 integrase inhibitor | 0.069 0.049 CHEMBL3527068 | CHEMBL3527068 | |
| 0.02 | 0.439 | 0.412 | Ca(v)3.2 blocker | 0.412 0.002 CHEMBL1710849 | CHEMBL1710849 | |
| 0.032 | 0.453 | 0.144 | Amyloid beta aggregation inhibitor | 0.144 0.113 CHEMBL3527068 | CHEMBL3527068 | |
| 0.029 | 0.463 | 0.137 | Estrogen antagonist | 0.137 0.031 CHEMBL3527225 0.105 0.087 CHEMBL3527224 0.107 0.082 CHEMBL3527010 0.137 0.031 CHEMBL3527226 0.107 0.081 CHEMBL3527068 | CHEMBL3527226 | |
| 0.028 | 0.495 | 0.062 | Heme oxygenase stimulant | 0.062 0.039 CHEMBL3527224 | CHEMBL3527224 | |
| 0.062 | 0.553 | 0.224 | Sodium/bile acid cotransporter inhibitor | 0.224 0.157 CHEMBL3527225 0.224 0.157 CHEMBL3527226 | CHEMBL3527226 | |
| 0.008 | 0.571 | 0.031 | Estrogen-related receptor beta antagonist | 0.031 0.026 CHEMBL3527225 0.031 0.026 CHEMBL3527226 | CHEMBL3527226 | |
| 0.016 | 0.674 | 0.158 | Nitric oxide antagonist | 0.158 0.089 CHEMBL1710849 | CHEMBL1710849 | |
| 0.009 | 0.777 | 0.174 | Antioxidant | 0.174 0.138 CHEMBL3527068 | CHEMBL3527068 | |
| 0.025 | 0.795 | 0.291 | Antiinflammatory | 0.291 0.223 CHEMBL1710849 | CHEMBL1710849 | |
| 0.007 | 0.786 | 0.179 | Free radical scavenger | 0.153 0.141 CHEMBL3527010 0.179 0.115 CHEMBL3527068 | CHEMBL3527068 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |