| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.975 | 0.002 | 0.975 | Vasodilator, coronary | 0.747 0.004 CHEMBL3544800 0.855 0.003 CHEMBL3544801 | ||
| 0.942 | 0.002 | 0.942 | Calcium channel blocker | 0.781 0.003 CHEMBL3544800 0.787 0.003 CHEMBL3544801 | ||
| 0.931 | 0.001 | 0.931 | Calcium antagonist | 0.578 0.002 CHEMBL3544800 0.617 0.002 CHEMBL3544801 | ||
| 0.89 | 0.002 | 0.89 | Calcium channel (voltage-sensitive) blocker | 0.651 0.003 CHEMBL3544800 0.603 0.003 CHEMBL3544801 | ||
| 0.866 | 0.001 | 0.866 | Calcium channel L-type blocker | 0.747 0.001 CHEMBL3544800 0.739 0.001 CHEMBL3544801 | ||
| 0.84 | 0.003 | 0.84 | Vasodilator, peripheral | 0.794 0.004 CHEMBL3544800 0.807 0.004 CHEMBL3544801 | ||
| 0.751 | 0.004 | 0.751 | Vasodilator | 0.717 0.004 CHEMBL3544800 0.741 0.004 CHEMBL3544801 | ||
| 0.709 | 0.002 | 0.714 | Calcium channel L-type activator | 0.677 0.003 CHEMBL3544800 0.714 0.002 CHEMBL3544801 | CHEMBL3544801 | |
| 0.706 | 0.001 | 0.706 | Calcium channel activator | 0.655 0.002 CHEMBL3544800 0.664 0.002 CHEMBL3544801 | ||
| 0.568 | 0.009 | 0.608 | Cardiotonic | 0.574 0.009 CHEMBL3544800 0.608 0.007 CHEMBL3544801 | CHEMBL3544801 | |
| 0.554 | 0.003 | 0.554 | TRPA1 agonist | 0.415 0.004 CHEMBL3544800 0.233 0.006 CHEMBL3544801 | ||
| 0.552 | 0.018 | 0.668 | Spasmolytic | 0.616 0.011 CHEMBL3544800 0.668 0.008 CHEMBL3544801 | CHEMBL3544801 | |
| 0.358 | 0.074 | 0.358 | Transcription factor NF kappa B inhibitor | 0.236 0.137 CHEMBL3544800 0.199 0.17 CHEMBL3544801 | ||
| 0.31 | 0.027 | 0.31 | P-glycoprotein inhibitor | 0.198 0.065 CHEMBL3544800 0.199 0.064 CHEMBL3544801 | ||
| 0.401 | 0.119 | 0.401 | DNA polymerase beta inhibitor | |||
| 0.3 | 0.022 | 0.3 | Diuretic | 0.209 0.041 CHEMBL3544800 0.128 0.097 CHEMBL3544801 | ||
| 0.307 | 0.034 | 0.313 | Platelet aggregation inhibitor | 0.283 0.04 CHEMBL3544800 0.313 0.033 CHEMBL3544801 | CHEMBL3544801 | |
| 0.276 | 0.006 | 0.276 | Neuropeptide Y1 antagonist | 0.161 0.05 CHEMBL3544800 0.142 0.077 CHEMBL3544801 | ||
| 0.387 | 0.121 | 0.387 | DNA directed DNA polymerase inhibitor | |||
| 0.286 | 0.037 | 0.286 | Anesthetic general | 0.173 0.092 CHEMBL3544800 | ||
| 0.318 | 0.08 | 0.318 | Cholesterol antagonist | 0.269 0.112 CHEMBL3544800 0.229 0.14 CHEMBL3544801 | ||
| 0.233 | 0.011 | 0.314 | Adenylate kinase inhibitor | 0.314 0.006 CHEMBL3544800 0.257 0.009 CHEMBL3544801 | CHEMBL3544800 | |
| 0.298 | 0.087 | 0.298 | Apoptosis antagonist | 0.217 0.159 CHEMBL3544800 0.232 0.145 CHEMBL3544801 | ||
| 0.343 | 0.133 | 0.343 | Transcription factor inhibitor | |||
| 0.264 | 0.066 | 0.264 | Platelet antagonist | 0.181 0.117 CHEMBL3544800 0.211 0.094 CHEMBL3544801 | ||
| 0.281 | 0.088 | 0.3 | Interleukin 2 agonist | 0.284 0.086 CHEMBL3544800 0.3 0.074 CHEMBL3544801 | CHEMBL3544801 | |
| 0.191 | 0.026 | 0.191 | Alpha 2b adrenoreceptor antagonist | |||
| 0.188 | 0.03 | 0.221 | CF transmembrane conductance regulator agonist | 0.221 0.013 CHEMBL3544800 0.196 0.024 CHEMBL3544801 | CHEMBL3544800 | |
| 0.16 | 0.005 | 0.171 | Aldosterone antagonist | 0.171 0.005 CHEMBL3544800 0.073 0.013 CHEMBL3544801 | CHEMBL3544800 | |
| 0.281 | 0.127 | 0.281 | Calpain 2 inhibitor | |||
| 0.224 | 0.078 | 0.248 | Cyclic AMP phosphodiesterase inhibitor | 0.226 0.076 CHEMBL3544800 0.248 0.065 CHEMBL3544801 | CHEMBL3544801 | |
| 0.261 | 0.127 | 0.261 | Thioredoxin glutathione reductase inhibitor | |||
| 0.192 | 0.063 | 0.194 | Amyloid beta precursor protein antagonist | 0.194 0.061 CHEMBL3544800 0.139 0.114 CHEMBL3544801 | CHEMBL3544800 | |
| 0.137 | 0.011 | 0.168 | Glycine receptor antagonist | 0.168 0.005 CHEMBL3544800 0.137 0.011 CHEMBL3544801 | CHEMBL3544800 | |
| 0.194 | 0.076 | 0.194 | Non-steroidal antiinflammatory agent | 0.178 0.089 CHEMBL3544800 0.143 0.125 CHEMBL3544801 | ||
| 0.123 | 0.01 | 0.123 | Calcium channel T-type blocker | |||
| 0.137 | 0.026 | 0.185 | Androgen antagonist | 0.185 0.015 CHEMBL3544800 0.165 0.019 CHEMBL3544801 | CHEMBL3544800 | |
| 0.118 | 0.019 | 0.118 | Adenosine A3 receptor antagonist | 0.076 0.048 CHEMBL3544800 0.079 0.044 CHEMBL3544801 | ||
| 0.148 | 0.054 | 0.175 | Farnesoid X receptor antagonist | 0.175 0.032 CHEMBL3544800 0.156 0.046 CHEMBL3544801 | CHEMBL3544800 | |
| 0.129 | 0.035 | 0.129 | Toll-Like receptor 4 antagonist | |||
| 0.134 | 0.04 | 0.134 | Alpha 2c adrenoreceptor antagonist | |||
| 0.143 | 0.052 | 0.143 | Anesthetic local | |||
| 0.22 | 0.129 | 0.22 | Hypoxia-inducible factor 1 alpha inhibitor | |||
| 0.169 | 0.081 | 0.244 | Lipocortins synthesis antagonist | 0.244 0.035 CHEMBL3544800 0.211 0.05 CHEMBL3544801 | CHEMBL3544800 | |
| 0.159 | 0.076 | 0.159 | Interleukin 6 antagonist | |||
| 0.154 | 0.07 | 0.154 | Phospholipase A2 inhibitor | 0.144 0.08 CHEMBL3544800 0.133 0.097 CHEMBL3544801 | ||
| 0.087 | 0.01 | 0.122 | Mineralocorticoid receptor antagonist | 0.122 0.006 CHEMBL3544800 0.113 0.007 CHEMBL3544801 | CHEMBL3544800 | |
| 0.164 | 0.095 | 0.164 | Hepatoprotectant | 0.145 0.115 CHEMBL3544800 0.162 0.097 CHEMBL3544801 | ||
| 0.141 | 0.073 | 0.141 | Mannose-6-phosphate isomerase inhibitor | 0.128 0.088 CHEMBL3544800 | ||
| 0.209 | 0.142 | 0.209 | 12-Lipoxygenase inhibitor | |||
| 0.078 | 0.013 | 0.078 | Thromboxane synthase inhibitor | 0.077 0.013 CHEMBL3544800 0.067 0.019 CHEMBL3544801 | ||
| 0.195 | 0.14 | 0.195 | Transcription factor STAT3 inhibitor | |||
| 0.119 | 0.064 | 0.119 | Calcium channel N-type blocker | |||
| 0.078 | 0.024 | 0.078 | Nitric oxide donor | 0.068 0.036 CHEMBL3544800 0.064 0.041 CHEMBL3544801 | ||
| 0.155 | 0.103 | 0.177 | Succinate dehydrogenase inhibitor | 0.177 0.072 CHEMBL3544800 | CHEMBL3544800 | |
| 0.185 | 0.134 | 0.377 | Interleukin agonist | 0.377 0.023 CHEMBL3544800 0.35 0.029 CHEMBL3544801 | CHEMBL3544800 | |
| 0.1 | 0.05 | 0.102 | Bile acid receptor antagonist | 0.102 0.045 CHEMBL3544800 0.089 0.075 CHEMBL3544801 | CHEMBL3544800 | |
| 0.222 | 0.172 | 0.222 | Beta lactamase inhibitor | |||
| 0.101 | 0.052 | 0.104 | Interleukin 12 antagonist | 0.104 0.048 CHEMBL3544800 0.092 0.068 CHEMBL3544801 | CHEMBL3544800 | |
| 0.053 | 0.006 | 0.053 | Transforming growth factor beta 2 antagonist | |||
| 0.138 | 0.092 | 0.138 | GABA C receptor rho-2 antagonist | |||
| 0.143 | 0.097 | 0.165 | Mcl-1 antagonist | 0.165 0.077 CHEMBL3544800 0.127 0.116 CHEMBL3544801 | CHEMBL3544800 | |
| 0.178 | 0.134 | 0.178 | Immunostimulant | |||
| 0.075 | 0.032 | 0.075 | Beta adrenoreceptor antagonist | |||
| 0.106 | 0.065 | 0.106 | DOPA decarboxylase inhibitor | |||
| 0.145 | 0.107 | 0.145 | Cyclin-dependent kinase 3 inhibitor | |||
| 0.089 | 0.053 | 0.089 | Granulocyte macrophage colony stimulating factor agonist | |||
| 0.102 | 0.066 | 0.102 | Beta glucuronidase inhibitor | 0.098 0.073 CHEMBL3544800 | ||
| 0.107 | 0.072 | 0.107 | Platelet activating factor antagonist | 0.1 0.079 CHEMBL3544801 | ||
| 0.064 | 0.032 | 0.064 | Beta 1 adrenoreceptor antagonist | |||
| 0.145 | 0.114 | 0.145 | Neurotensin receptor agonist | |||
| 0.107 | 0.077 | 0.107 | Photosensitizer | |||
| 0.171 | 0.141 | 0.194 | Antioxidant | 0.17 0.142 CHEMBL3544800 0.194 0.118 CHEMBL3544801 | CHEMBL3544801 | |
| 0.229 | 0.2 | 0.229 | Alpha-glucosidase inhibitor | |||
| 0.09 | 0.066 | 0.124 | ABCA1 expression enhancer | 0.124 0.028 CHEMBL3544800 0.103 0.047 CHEMBL3544801 | CHEMBL3544800 | |
| 0.1 | 0.078 | 0.1 | Multidrug resistance-associated protein 1 inhibitor | |||
| 0.053 | 0.031 | 0.053 | Potassium channel (Inward rectifier) activator | 0.052 0.031 CHEMBL3544800 | ||
| 0.05 | 0.03 | 0.05 | Potassium channel (ATP-sensitive) activator | 0.05 0.03 CHEMBL3544800 | ||
| 0.082 | 0.062 | 0.082 | 3C-Like protease (SARS coronavirus) inhibitor | 0.08 0.069 CHEMBL3544800 | ||
| 0.124 | 0.109 | 0.124 | Sigma receptor agonist | |||
| 0.087 | 0.076 | 0.087 | Sphingomyelinase inhibitor | |||
| 0.057 | 0.047 | 0.057 | Potassium channel intermediate-conductance Ca-activated blocker | |||
| 0.108 | 0.098 | 0.108 | Sphingosine 1-phosphate receptor 4 antagonist | |||
| 0.1 | 0.09 | 0.1 | Microtubule formation inhibitor | |||
| 0.05 | 0.043 | 0.05 | Nicotinic alpha3beta2 receptor antagonist | |||
| 0.042 | 0.035 | 0.053 | Glutamate (mGluR group III) antagonist | 0.053 0.018 CHEMBL3544800 | CHEMBL3544800 | |
| 0.063 | 0.058 | 0.076 | Glutamate (mGluR6) antagonist | 0.076 0.029 CHEMBL3544800 0.062 0.061 CHEMBL3544801 | CHEMBL3544800 | |
| 0.057 | 0.055 | 0.063 | Phosphodiesterase III inhibitor | 0.063 0.049 CHEMBL3544801 | CHEMBL3544801 | |
| 0.123 | 0.121 | 0.123 | Pregnane X receptor agonist | |||
| 0.124 | 0.124 | 0.196 | Interferon gamma antagonist | 0.196 0.042 CHEMBL3544800 0.175 0.053 CHEMBL3544801 | CHEMBL3544800 | |
| 0.165 | 0.176 | 0.19 | DNA synthesis inhibitor | 0.19 0.139 CHEMBL3544800 0.175 0.16 CHEMBL3544801 | CHEMBL3544800 | |
| 0.185 | 0.197 | 0.245 | Antithrombotic | 0.245 0.13 CHEMBL3544800 0.232 0.141 CHEMBL3544801 | CHEMBL3544800 | |
| 0.123 | 0.136 | 0.14 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.14 0.092 CHEMBL3544800 | CHEMBL3544800 | |
| 0.012 | 0.026 | 0.016 | Kainate receptor 3 antagonist | 0.016 0.014 CHEMBL3544800 | CHEMBL3544800 | |
| 0.016 | 0.03 | 0.025 | Kainate receptor 4 antagonist | 0.025 0.017 CHEMBL3544800 | CHEMBL3544800 | |
| 0.079 | 0.096 | 0.087 | Xanthine oxidase inhibitor | 0.087 0.076 CHEMBL3544800 | CHEMBL3544800 | |
| 0.035 | 0.057 | 0.041 | Glutamate (mGluR4) antagonist | 0.041 0.035 CHEMBL3544800 | CHEMBL3544800 | |
| 0.03 | 0.055 | 0.035 | Glutamate (mGluR8) agonist | 0.035 0.032 CHEMBL3544800 | CHEMBL3544800 | |
| 0.01 | 0.045 | 0.019 | Kainate receptor 5 antagonist | 0.019 0.016 CHEMBL3544800 | CHEMBL3544800 | |
| 0.061 | 0.097 | 0.094 | Antiadrenergic | 0.094 0.06 CHEMBL3544801 | CHEMBL3544801 | |
| 0.067 | 0.104 | 0.079 | Potassium channel activator | 0.079 0.078 CHEMBL3544800 | CHEMBL3544800 | |
| 0.153 | 0.19 | 0.167 | RNA-directed DNA polymerase inhibitor | 0.167 0.159 CHEMBL3544800 | CHEMBL3544800 | |
| 0.059 | 0.096 | 0.092 | Adrenaline antagonist | 0.092 0.058 CHEMBL3544801 | CHEMBL3544801 | |
| 0.041 | 0.101 | 0.064 | NMDA receptor agonist | 0.064 0.042 CHEMBL3544800 | CHEMBL3544800 | |
| 0.036 | 0.097 | 0.048 | CD45 antagonist | 0.048 0.04 CHEMBL3544800 | CHEMBL3544800 | |
| 0.081 | 0.141 | 0.106 | M17 leucyl aminopeptidase inhibitor | 0.106 0.094 CHEMBL3544800 | CHEMBL3544800 | |
| 0.032 | 0.098 | 0.055 | NMDA receptor glycine site agonist | 0.055 0.051 CHEMBL3544800 | CHEMBL3544800 | |
| 0.079 | 0.15 | 0.11 | Factor V inhibitor | 0.11 0.051 CHEMBL3544800 0.102 0.065 CHEMBL3544801 | CHEMBL3544800 | |
| 0.03 | 0.109 | 0.081 | Biliverdin reductase inhibitor | 0.081 0.026 CHEMBL3544800 0.054 0.048 CHEMBL3544801 | CHEMBL3544800 | |
| 0.021 | 0.103 | 0.044 | Glutamate (mGluR1a) antagonist | 0.044 0.025 CHEMBL3544801 | CHEMBL3544801 | |
| 0.023 | 0.111 | 0.051 | Glutamate (mGluR1) antagonist | 0.051 0.047 CHEMBL3544801 | CHEMBL3544801 | |
| 0.039 | 0.128 | 0.079 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.079 0.052 CHEMBL3544801 | CHEMBL3544801 | |
| 0.025 | 0.121 | 0.075 | Argininosuccinate synthase inhibitor | 0.075 0.028 CHEMBL3544800 0.051 0.045 CHEMBL3544801 | CHEMBL3544800 | |
| 0.038 | 0.141 | 0.052 | Adenine nucleotide translocase inhibitor | 0.052 0.05 CHEMBL3544800 | CHEMBL3544800 | |
| 0.055 | 0.16 | 0.105 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.105 0.049 CHEMBL3544800 0.092 0.062 CHEMBL3544801 | CHEMBL3544800 | |
| 0.054 | 0.16 | 0.109 | UDP-glucose 4-epimerase inhibitor | 0.109 0.052 CHEMBL3544800 0.104 0.057 CHEMBL3544801 | CHEMBL3544800 | |
| 0.052 | 0.16 | 0.076 | GABA B receptor agonist | 0.076 0.051 CHEMBL3544800 | CHEMBL3544800 | |
| 0.046 | 0.159 | 0.07 | Keratolytic | 0.07 0.066 CHEMBL3544800 | CHEMBL3544800 | |
| 0.133 | 0.249 | 0.182 | Peptidyltransferase inhibitor | 0.182 0.126 CHEMBL3544800 | CHEMBL3544800 | |
| 0.052 | 0.174 | 0.138 | Triose-phosphate isomerase inhibitor | 0.138 0.024 CHEMBL3544800 0.125 0.029 CHEMBL3544801 | CHEMBL3544800 | |
| 0.158 | 0.286 | 0.263 | Antibacterial | 0.263 0.165 CHEMBL3544800 0.243 0.184 CHEMBL3544801 | CHEMBL3544800 | |
| 0.12 | 0.274 | 0.203 | Gastrin inhibitor | 0.203 0.145 CHEMBL3544800 0.186 0.17 CHEMBL3544801 | CHEMBL3544800 | |
| 0.02 | 0.179 | 0.072 | Phosphofructokinase-1 inhibitor | 0.072 0.046 CHEMBL3544800 0.064 0.053 CHEMBL3544801 | CHEMBL3544800 | |
| 0.063 | 0.224 | 0.142 | Interleukin 1 antagonist | 0.142 0.064 CHEMBL3544800 | CHEMBL3544800 | |
| 0.035 | 0.202 | 0.07 | Glutamate dehydrogenase inhibitor | 0.07 0.056 CHEMBL3544800 | CHEMBL3544800 | |
| 0.141 | 0.308 | 0.247 | Histamine release inhibitor | 0.247 0.157 CHEMBL3544800 0.219 0.182 CHEMBL3544801 | CHEMBL3544800 | |
| 0.053 | 0.225 | 0.16 | Interleukin 1b antagonist | 0.16 0.033 CHEMBL3544800 0.129 0.055 CHEMBL3544801 | CHEMBL3544800 | |
| 0.023 | 0.207 | 0.067 | Porphobilinogen synthase inhibitor | 0.067 0.059 CHEMBL3544800 | CHEMBL3544800 | |
| 0.106 | 0.299 | 0.132 | Ca2+-transporting ATPase inhibitor | 0.132 0.109 CHEMBL3544800 | CHEMBL3544800 | |
| 0.041 | 0.243 | 0.09 | Anabolic | 0.09 0.078 CHEMBL3544800 | CHEMBL3544800 | |
| 0.07 | 0.284 | 0.263 | Platelet adhesion inhibitor | 0.263 0.045 CHEMBL3544800 0.237 0.054 CHEMBL3544801 | CHEMBL3544800 | |
| 0.009 | 0.882 | 0.245 | Cyclophilin D inhibitor | 0.245 0.218 CHEMBL3544801 | CHEMBL3544801 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |