| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.981 | 0.003 | 0.986 | Cyclophilin D inhibitor | 0.972 0.004 CHEMBL4525781 0.968 0.004 CHEMBL3527604 0.973 0.004 CHEMBL3526185 0.986 0.003 CHEMBL3527603 0.972 0.004 CHEMBL4525782 | CHEMBL3527603 | |
| 0.948 | 0 | 0.995 | Sodium/glucose cotransporter inhibitor | 0.539 0.001 CHEMBL4525781 0.995 0 CHEMBL3527604 0.995 0 CHEMBL3526185 0.829 0 CHEMBL3527603 0.539 0.001 CHEMBL4525782 | CHEMBL3526185 | |
| 0.951 | 0.004 | 0.96 | Antiobesity | 0.952 0.004 CHEMBL4525781 0.887 0.005 CHEMBL3527604 0.907 0.004 CHEMBL3526185 0.96 0.004 CHEMBL3527603 0.952 0.004 CHEMBL4525782 | CHEMBL3527603 | |
| 0.938 | 0 | 0.989 | Sodium/glucose cotransporter 2 inhibitor | 0.487 0 CHEMBL4525781 0.989 0 CHEMBL3527604 0.989 0 CHEMBL3526185 0.791 0 CHEMBL3527603 0.487 0 CHEMBL4525782 | CHEMBL3526185 | |
| 0.929 | 0.003 | 0.937 | Hypoglycemic | 0.904 0.003 CHEMBL4525781 0.91 0.003 CHEMBL3527604 0.924 0.003 CHEMBL3526185 0.937 0.003 CHEMBL3527603 0.904 0.003 CHEMBL4525782 | CHEMBL3527603 | |
| 0.549 | 0.025 | 0.74 | Cholesterol antagonist | 0.619 0.016 CHEMBL4525781 0.74 0.005 CHEMBL3527604 0.736 0.006 CHEMBL3526185 0.465 0.038 CHEMBL3527603 0.619 0.016 CHEMBL4525782 | CHEMBL3527604 | |
| 0.352 | 0.048 | 0.352 | Calcium channel activator | 0.311 0.081 CHEMBL3527603 | ||
| 0.297 | 0.087 | 0.428 | Apoptosis antagonist | 0.281 0.099 CHEMBL4525781 0.428 0.031 CHEMBL3527604 0.424 0.032 CHEMBL3526185 0.324 0.07 CHEMBL3527603 0.281 0.099 CHEMBL4525782 | CHEMBL3527604 | |
| 0.247 | 0.04 | 0.315 | Neurotrophic factor enhancer | 0.161 0.122 CHEMBL4525781 0.237 0.047 CHEMBL3527604 0.198 0.079 CHEMBL3526185 0.315 0.014 CHEMBL3527603 0.161 0.122 CHEMBL4525782 | CHEMBL3527603 | |
| 0.328 | 0.134 | 0.393 | Calcium channel L-type activator | 0.235 0.222 CHEMBL3527604 0.393 0.086 CHEMBL3527603 | CHEMBL3527603 | |
| 0.243 | 0.053 | 0.377 | Nitric oxide antagonist | 0.243 0.054 CHEMBL4525781 0.377 0.028 CHEMBL3527604 0.375 0.028 CHEMBL3526185 0.294 0.042 CHEMBL3527603 0.243 0.054 CHEMBL4525782 | CHEMBL3527604 | |
| 0.253 | 0.082 | 0.474 | Antioxidant | 0.228 0.096 CHEMBL4525781 0.454 0.026 CHEMBL3527604 0.474 0.023 CHEMBL3526185 0.324 0.054 CHEMBL3527603 0.228 0.096 CHEMBL4525782 | CHEMBL3526185 | |
| 0.217 | 0.056 | 0.379 | Hepatoprotectant | 0.207 0.061 CHEMBL4525781 0.379 0.015 CHEMBL3527604 0.375 0.016 CHEMBL3526185 0.241 0.046 CHEMBL3527603 0.207 0.061 CHEMBL4525782 | CHEMBL3527604 | |
| 0.258 | 0.122 | 0.601 | Transcription factor NF kappa B inhibitor | 0.234 0.139 CHEMBL4525781 0.601 0.031 CHEMBL3527604 0.585 0.033 CHEMBL3526185 0.281 0.106 CHEMBL3527603 0.234 0.139 CHEMBL4525782 | CHEMBL3527604 | |
| 0.176 | 0.052 | 0.269 | Protein kinase stimulant | 0.269 0.022 CHEMBL3527604 0.211 0.038 CHEMBL3526185 0.24 0.029 CHEMBL3527603 | CHEMBL3527604 | |
| 0.28 | 0.187 | 0.503 | Apoptosis agonist | 0.503 0.073 CHEMBL3527604 0.502 0.074 CHEMBL3526185 0.334 0.149 CHEMBL3527603 | CHEMBL3527604 | |
| 0.193 | 0.102 | 0.199 | Nitric-oxide synthase stimulant | 0.181 0.126 CHEMBL4525781 0.199 0.091 CHEMBL3527604 0.172 0.147 CHEMBL3526185 0.175 0.14 CHEMBL3527603 0.181 0.126 CHEMBL4525782 | CHEMBL3527604 | |
| 0.198 | 0.126 | 0.328 | DNA synthesis inhibitor | 0.19 0.139 CHEMBL4525781 0.328 0.035 CHEMBL3527604 0.272 0.055 CHEMBL3526185 0.244 0.07 CHEMBL3527603 0.19 0.139 CHEMBL4525782 | CHEMBL3527604 | |
| 0.157 | 0.089 | 0.277 | ATPase inhibitor | 0.277 0.009 CHEMBL3527604 0.226 0.021 CHEMBL3526185 0.165 0.077 CHEMBL3527603 | CHEMBL3527604 | |
| 0.136 | 0.09 | 0.141 | Ca2+-transporting ATPase inhibitor | 0.131 0.112 CHEMBL4525781 0.141 0.07 CHEMBL3527604 0.133 0.106 CHEMBL3526185 0.134 0.098 CHEMBL3527603 0.131 0.112 CHEMBL4525782 | CHEMBL3527604 | |
| 0.056 | 0.013 | 0.146 | Squalene synthetase inhibitor | 0.146 0.004 CHEMBL4525781 0.07 0.01 CHEMBL3527604 0.062 0.011 CHEMBL3526185 0.057 0.013 CHEMBL3527603 0.146 0.004 CHEMBL4525782 | CHEMBL4525782 | |
| 0.168 | 0.125 | 0.398 | Free radical scavenger | 0.393 0.03 CHEMBL3527604 0.398 0.029 CHEMBL3526185 0.243 0.071 CHEMBL3527603 | CHEMBL3526185 | |
| 0.135 | 0.104 | 0.182 | Melanin inhibitor | 0.179 0.052 CHEMBL3527604 0.155 0.075 CHEMBL3526185 0.182 0.05 CHEMBL3527603 | CHEMBL3527603 | |
| 0.136 | 0.106 | 0.162 | Arachidonic acid antagonist | 0.162 0.074 CHEMBL4525781 0.141 0.099 CHEMBL3527603 0.162 0.074 CHEMBL4525782 | CHEMBL4525782 | |
| 0.087 | 0.058 | 0.105 | Antineoplastic alkaloid | 0.105 0.044 CHEMBL3527603 | CHEMBL3527603 | |
| 0.081 | 0.057 | 0.181 | Antineoplastic antibiotic | 0.079 0.058 CHEMBL4525781 0.175 0.026 CHEMBL3527604 0.181 0.024 CHEMBL3526185 0.107 0.043 CHEMBL3527603 0.079 0.058 CHEMBL4525782 | CHEMBL3526185 | |
| 0.089 | 0.067 | 0.089 | ABCA1 expression enhancer | 0.083 0.079 CHEMBL3527603 | ||
| 0.224 | 0.202 | 0.612 | Antibacterial | 0.601 0.019 CHEMBL3527604 0.612 0.018 CHEMBL3526185 0.323 0.119 CHEMBL3527603 | CHEMBL3526185 | |
| 0.059 | 0.039 | 0.065 | Lipocortins synthesis agonist | 0.059 0.037 CHEMBL4525781 0.065 0.027 CHEMBL3527604 0.064 0.029 CHEMBL3526185 0.059 0.037 CHEMBL3527603 0.059 0.037 CHEMBL4525782 | CHEMBL3527604 | |
| 0.203 | 0.184 | 0.329 | Interleukin 2 agonist | 0.329 0.056 CHEMBL3527604 0.315 0.064 CHEMBL3526185 0.243 0.127 CHEMBL3527603 | CHEMBL3527604 | |
| 0.09 | 0.072 | 0.11 | Lanosterol 14 alpha demethylase inhibitor | 0.11 0.041 CHEMBL3527603 | CHEMBL3527603 | |
| 0.108 | 0.092 | 0.252 | Cyclooxygenase 3 inhibitor | 0.252 0.009 CHEMBL3527604 0.214 0.014 CHEMBL3526185 0.122 0.075 CHEMBL3527603 | CHEMBL3527604 | |
| 0.031 | 0.014 | 0.033 | 1,3-Beta-glucan synthase inhibitor | 0.029 0.017 CHEMBL4525781 0.029 0.017 CHEMBL3527604 0.032 0.011 CHEMBL3526185 0.033 0.009 CHEMBL3527603 0.029 0.017 CHEMBL4525782 | CHEMBL3527603 | |
| 0.092 | 0.085 | 0.144 | Toll-Like receptor 4 antagonist | 0.144 0.024 CHEMBL3527604 0.136 0.03 CHEMBL3526185 | CHEMBL3527604 | |
| 0.086 | 0.08 | 0.135 | UDP-glucose 4-epimerase inhibitor | 0.135 0.035 CHEMBL3527604 0.108 0.053 CHEMBL3526185 0.087 0.077 CHEMBL3527603 | CHEMBL3527604 | |
| 0.079 | 0.082 | 0.107 | ATPase (Vacuolar H+) inhibitor | 0.107 0.031 CHEMBL3527604 0.102 0.037 CHEMBL3526185 | CHEMBL3527604 | |
| 0.031 | 0.036 | 0.068 | Antibiotic Aminoglycoside-like | 0.064 0.007 CHEMBL3527604 0.068 0.006 CHEMBL3526185 0.033 0.031 CHEMBL3527603 | CHEMBL3526185 | |
| 0.121 | 0.131 | 0.174 | Interferon gamma antagonist | 0.174 0.054 CHEMBL3527604 0.15 0.078 CHEMBL3526185 0.146 0.083 CHEMBL3527603 | CHEMBL3527604 | |
| 0.123 | 0.141 | 0.464 | Angiogenesis stimulant | 0.464 0.014 CHEMBL3527604 0.439 0.016 CHEMBL3526185 0.15 0.122 CHEMBL3527603 | CHEMBL3527604 | |
| 0.073 | 0.09 | 0.118 | 5-Lipoxygenase inhibitor | 0.118 0.051 CHEMBL4525781 0.083 0.078 CHEMBL3527603 0.118 0.051 CHEMBL4525782 | CHEMBL4525782 | |
| 0.181 | 0.2 | 0.34 | Vasodilator, coronary | 0.224 0.16 CHEMBL4525781 0.34 0.06 CHEMBL3527604 0.28 0.105 CHEMBL3526185 0.224 0.16 CHEMBL4525782 | CHEMBL3527604 | |
| 0.072 | 0.094 | 0.104 | Triose-phosphate isomerase inhibitor | 0.104 0.044 CHEMBL3527604 0.085 0.068 CHEMBL3526185 0.087 0.064 CHEMBL3527603 | CHEMBL3527604 | |
| 0.092 | 0.127 | 0.201 | Lipid peroxidase inhibitor | 0.201 0.041 CHEMBL3527604 0.197 0.043 CHEMBL3526185 0.12 0.094 CHEMBL3527603 | CHEMBL3527604 | |
| 0.078 | 0.114 | 0.189 | AMP-activated protein kinase stimulant | 0.189 0.013 CHEMBL3527604 0.169 0.018 CHEMBL3526185 0.099 0.072 CHEMBL3527603 | CHEMBL3527604 | |
| 0.08 | 0.121 | 0.249 | Amylase inhibitor | 0.249 0.028 CHEMBL3527604 0.245 0.029 CHEMBL3526185 0.102 0.095 CHEMBL3527603 | CHEMBL3527604 | |
| 0.103 | 0.145 | 0.193 | Insulin secretagoues | 0.191 0.041 CHEMBL3527604 0.193 0.04 CHEMBL3526185 | CHEMBL3526185 | |
| 0.035 | 0.085 | 0.287 | Selectin antagonist | 0.264 0.008 CHEMBL3527604 0.287 0.006 CHEMBL3526185 | CHEMBL3526185 | |
| 0.029 | 0.081 | 0.089 | Protein 50S ribosomal subunit inhibitor | 0.089 0.016 CHEMBL3527604 0.088 0.016 CHEMBL3526185 | CHEMBL3527604 | |
| 0.113 | 0.165 | 0.145 | CC chemokine 6 receptor antagonist | 0.145 0.03 CHEMBL3527604 0.141 0.038 CHEMBL3526185 0.124 0.096 CHEMBL3527603 | CHEMBL3527604 | |
| 0.077 | 0.137 | 0.103 | Microtubule formation inhibitor | 0.103 0.085 CHEMBL3527604 | CHEMBL3527604 | |
| 0.064 | 0.125 | 0.12 | Transcription factor NF kappa B stimulant | 0.113 0.029 CHEMBL3527604 0.12 0.025 CHEMBL3526185 | CHEMBL3526185 | |
| 0.116 | 0.181 | 0.221 | Hypolipemic | 0.221 0.082 CHEMBL4525781 0.216 0.084 CHEMBL3527604 0.196 0.097 CHEMBL3526185 0.221 0.082 CHEMBL4525782 | CHEMBL4525782 | |
| 0.012 | 0.086 | 0.035 | Protein 30S ribosomal subunit inhibitor | 0.03 0.013 CHEMBL3527604 0.035 0.011 CHEMBL3526185 | CHEMBL3526185 | |
| 0.167 | 0.251 | 0.45 | Histamine release inhibitor | 0.206 0.195 CHEMBL4525781 0.45 0.05 CHEMBL3527604 0.442 0.054 CHEMBL3526185 0.206 0.195 CHEMBL4525782 | CHEMBL3527604 | |
| 0.092 | 0.192 | 0.306 | Platelet adhesion inhibitor | 0.306 0.032 CHEMBL3527604 0.305 0.032 CHEMBL3526185 | CHEMBL3527604 | |
| 0.156 | 0.258 | 0.406 | Alpha-glucosidase inhibitor | 0.406 0.112 CHEMBL3527604 0.326 0.147 CHEMBL3526185 | CHEMBL3527604 | |
| 0.111 | 0.216 | 0.138 | Phospholipase C inhibitor | 0.138 0.134 CHEMBL3527603 | CHEMBL3527603 | |
| 0.143 | 0.266 | 0.388 | Immunosuppressant | 0.38 0.072 CHEMBL3527604 0.388 0.068 CHEMBL3526185 | CHEMBL3526185 | |
| 0.198 | 0.324 | 0.274 | Caspase 9 stimulant | 0.274 0.223 CHEMBL3527604 | CHEMBL3527604 | |
| 0.052 | 0.181 | 0.118 | Cystathionine beta-synthase inhibitor | 0.118 0.06 CHEMBL3527603 | CHEMBL3527603 | |
| 0.036 | 0.166 | 0.054 | Adenine nucleotide translocase inhibitor | 0.054 0.041 CHEMBL3527604 0.052 0.049 CHEMBL3526185 | CHEMBL3527604 | |
| 0.016 | 0.15 | 0.027 | Toll-Like receptor 4 agonist | 0.027 0.016 CHEMBL3527604 0.026 0.019 CHEMBL3526185 | CHEMBL3527604 | |
| 0.025 | 0.189 | 0.052 | Glucose-6-phosphate translocase inhibitor | 0.052 0.035 CHEMBL3527604 0.048 0.043 CHEMBL3526185 | CHEMBL3527604 | |
| 0.122 | 0.299 | 0.326 | Peptidyltransferase inhibitor | 0.326 0.017 CHEMBL3527604 0.317 0.019 CHEMBL3526185 | CHEMBL3527604 | |
| 0.038 | 0.222 | 0.134 | Expectorant | 0.134 0.042 CHEMBL3527604 0.102 0.067 CHEMBL3526185 | CHEMBL3527604 | |
| 0.03 | 0.228 | 0.12 | Topoisomerase I inhibitor | 0.12 0.055 CHEMBL3527604 0.1 0.07 CHEMBL3526185 | CHEMBL3527604 | |
| 0.056 | 0.262 | 0.165 | Cell adhesion inhibitor | 0.155 0.043 CHEMBL3527604 0.165 0.038 CHEMBL3526185 | CHEMBL3526185 | |
| 0.168 | 0.384 | 0.59 | Antiinflammatory | 0.286 0.228 CHEMBL4525781 0.59 0.056 CHEMBL3527604 0.558 0.066 CHEMBL3526185 0.286 0.228 CHEMBL4525782 | CHEMBL3527604 | |
| 0.022 | 0.245 | 0.067 | Heparanase inhibitor | 0.067 0.014 CHEMBL3527604 0.067 0.014 CHEMBL3526185 | CHEMBL3526185 | |
| 0.088 | 0.312 | 0.159 | Cyclic AMP phosphodiesterase inhibitor | 0.159 0.137 CHEMBL3527604 | CHEMBL3527604 | |
| 0.121 | 0.365 | 0.203 | Caspase 3 stimulant | 0.203 0.164 CHEMBL3527604 0.201 0.167 CHEMBL3526185 | CHEMBL3527604 | |
| 0.06 | 0.325 | 0.17 | Spasmolytic | 0.17 0.145 CHEMBL4525781 0.17 0.145 CHEMBL4525782 | CHEMBL4525782 | |
| 0.048 | 0.329 | 0.169 | Cell wall synthesis inhibitor | 0.147 0.068 CHEMBL3527604 0.169 0.048 CHEMBL3526185 | CHEMBL3526185 | |
| 0.088 | 0.376 | 0.402 | Antithrombotic | 0.402 0.049 CHEMBL3527604 0.384 0.053 CHEMBL3526185 | CHEMBL3527604 | |
| 0.059 | 0.349 | 0.14 | Interleukin 6 antagonist | 0.14 0.106 CHEMBL3527604 | CHEMBL3527604 | |
| 0.06 | 0.353 | 0.122 | NOS3 expression enhancer | 0.122 0.111 CHEMBL3527604 | CHEMBL3527604 | |
| 0.033 | 0.332 | 0.091 | Beta glucuronidase inhibitor | 0.091 0.085 CHEMBL3527604 | CHEMBL3527604 | |
| 0.053 | 0.353 | 0.177 | Platelet antagonist | 0.177 0.12 CHEMBL3527604 0.153 0.141 CHEMBL3526185 | CHEMBL3527604 | |
| 0.032 | 0.339 | 0.19 | Thrombolytic | 0.187 0.058 CHEMBL4525781 0.19 0.057 CHEMBL3527604 0.166 0.07 CHEMBL3526185 0.187 0.058 CHEMBL4525782 | CHEMBL3527604 | |
| 0.057 | 0.382 | 0.142 | Non-steroidal antiinflammatory agent | 0.142 0.127 CHEMBL3527604 | CHEMBL3527604 | |
| 0.049 | 0.383 | 0.172 | Interleukin agonist | 0.172 0.147 CHEMBL3527604 | CHEMBL3527604 | |
| 0.011 | 0.355 | 0.068 | Dopamine transporter inhibitor | 0.068 0.021 CHEMBL4525781 0.068 0.021 CHEMBL4525782 | CHEMBL4525782 | |
| 0.053 | 0.42 | 0.121 | DNA repair enzyme inhibitor | 0.121 0.071 CHEMBL3527604 | CHEMBL3527604 | |
| 0.037 | 0.413 | 0.254 | Immunostimulant | 0.254 0.095 CHEMBL3527604 0.25 0.096 CHEMBL3526185 | CHEMBL3527604 | |
| 0.018 | 0.426 | 0.057 | Factor IXa inhibitor | 0.048 0.04 CHEMBL3527604 0.057 0.029 CHEMBL3526185 | CHEMBL3526185 | |
| 0.041 | 0.458 | 0.162 | Vasodilator | 0.162 0.14 CHEMBL3527604 | CHEMBL3527604 | |
| 0.017 | 0.453 | 0.12 | Topoisomerase II inhibitor | 0.12 0.067 CHEMBL3527604 0.113 0.073 CHEMBL3526185 | CHEMBL3527604 | |
| 0.014 | 0.456 | 0.066 | Topoisomerase II alpha inhibitor | 0.066 0.065 CHEMBL3527604 | CHEMBL3527604 | |
| 0.007 | 0.538 | 0.135 | Check point kinase 2 inhibitor | 0.135 0.038 CHEMBL4525781 0.135 0.038 CHEMBL4525782 | CHEMBL4525782 | |
| 0.027 | 0.603 | 0.182 | Tumour necrosis factor alpha release inhibitor | 0.182 0.125 CHEMBL3527604 0.158 0.148 CHEMBL3526185 | CHEMBL3527604 | |
| 0.023 | 0.607 | 0.132 | Hemostatic | 0.132 0.092 CHEMBL3527604 | CHEMBL3527604 | |
| 0.02 | 0.985 | 0.229 | MAP kinase kinase 3 inhibitor | 0.229 0.058 CHEMBL4525781 0.229 0.058 CHEMBL4525782 | CHEMBL4525782 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |