| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.754 | 0.026 | 0.754 | DNA directed DNA polymerase inhibitor | 0.569 0.064 CHEMBL222744 0.616 0.051 CHEMBL1256485 | ||
| 0.697 | 0 | 0.697 | Purine nucleoside phosphorylase inhibitor | 0.159 0.001 CHEMBL222744 0.407 0.001 CHEMBL1256485 | ||
| 0.677 | 0.003 | 0.68 | RNA-directed DNA polymerase inhibitor | 0.587 0.006 CHEMBL222744 0.68 0.003 CHEMBL1256485 | CHEMBL1256485 | |
| 0.678 | 0.006 | 0.814 | Immunomodulator | 0.814 0.004 CHEMBL222744 0.639 0.008 CHEMBL1256485 | CHEMBL222744 | |
| 0.656 | 0.001 | 0.656 | Thymidine kinase inhibitor | 0.268 0.002 CHEMBL222744 0.303 0.002 CHEMBL1256485 | ||
| 0.62 | 0.007 | 0.62 | DNA synthesis inhibitor | 0.592 0.008 CHEMBL222744 0.59 0.008 CHEMBL1256485 | ||
| 0.502 | 0.004 | 0.521 | DNA polymerase I inhibitor | 0.348 0.008 CHEMBL222744 0.521 0.004 CHEMBL1256485 | CHEMBL1256485 | |
| 0.484 | 0.031 | 0.581 | Vasodilator, peripheral | 0.269 0.114 CHEMBL222744 0.581 0.018 CHEMBL1256485 | CHEMBL1256485 | |
| 0.461 | 0.035 | 0.513 | Immunostimulant | 0.513 0.027 CHEMBL222744 0.5 0.029 CHEMBL1256485 | CHEMBL222744 | |
| 0.379 | 0.001 | 0.379 | Adenosine deaminase inhibitor | 0.127 0.003 CHEMBL222744 0.266 0.002 CHEMBL1256485 | ||
| 0.43 | 0.053 | 0.43 | Immunosuppressant | 0.279 0.129 CHEMBL222744 0.402 0.062 CHEMBL1256485 | ||
| 0.364 | 0.005 | 0.375 | DNA directed RNA polymerase inhibitor | 0.375 0.005 CHEMBL222744 0.292 0.007 CHEMBL1256485 | CHEMBL222744 | |
| 0.34 | 0.009 | 0.34 | Interleukin 1 antagonist | 0.326 0.009 CHEMBL222744 0.28 0.013 CHEMBL1256485 | ||
| 0.31 | 0.005 | 0.332 | Antimetabolite | 0.28 0.006 CHEMBL222744 0.332 0.005 CHEMBL1256485 | CHEMBL1256485 | |
| 0.295 | 0.013 | 0.295 | Nitric-oxide synthase stimulant | 0.252 0.031 CHEMBL222744 0.265 0.024 CHEMBL1256485 | ||
| 0.372 | 0.09 | 0.372 | Histamine release inhibitor | 0.243 0.161 CHEMBL222744 0.233 0.169 CHEMBL1256485 | ||
| 0.286 | 0.005 | 0.374 | HIV-1 reverse transcriptase inhibitor | 0.374 0.004 CHEMBL222744 0.214 0.009 CHEMBL1256485 | CHEMBL222744 | |
| 0.292 | 0.014 | 0.292 | Adenylate cyclase inhibitor | 0.187 0.028 CHEMBL222744 0.186 0.028 CHEMBL1256485 | ||
| 0.292 | 0.016 | 0.292 | Interleukin 6 antagonist | 0.274 0.019 CHEMBL222744 0.242 0.025 CHEMBL1256485 | ||
| 0.272 | 0.004 | 0.272 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.206 0.006 CHEMBL222744 0.261 0.005 CHEMBL1256485 | ||
| 0.26 | 0.004 | 0.261 | Folate antagonist | 0.253 0.005 CHEMBL222744 0.261 0.004 CHEMBL1256485 | CHEMBL1256485 | |
| 0.243 | 0 | 0.243 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.15 0.001 CHEMBL222744 0.231 0 CHEMBL1256485 | ||
| 0.244 | 0.006 | 0.244 | Phosphodiesterase 7B inhibitor | 0.197 0.01 CHEMBL222744 0.217 0.009 CHEMBL1256485 | ||
| 0.233 | 0.001 | 0.233 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.075 0.003 CHEMBL222744 0.101 0.002 CHEMBL1256485 | ||
| 0.268 | 0.055 | 0.515 | Interleukin antagonist | 0.515 0.019 CHEMBL222744 0.236 0.067 CHEMBL1256485 | CHEMBL222744 | |
| 0.215 | 0.02 | 0.215 | MAP kinase kinase 5 inhibitor | 0.179 0.064 CHEMBL1256485 | ||
| 0.204 | 0.012 | 0.206 | Interleukin 8 antagonist | 0.17 0.023 CHEMBL222744 0.206 0.011 CHEMBL1256485 | CHEMBL1256485 | |
| 0.201 | 0.01 | 0.218 | NADH dehydrogenase inhibitor | 0.138 0.021 CHEMBL222744 0.218 0.009 CHEMBL1256485 | CHEMBL1256485 | |
| 0.197 | 0.009 | 0.201 | DNA repair enzyme inhibitor | 0.172 0.016 CHEMBL222744 0.201 0.009 CHEMBL1256485 | CHEMBL1256485 | |
| 0.188 | 0.012 | 0.26 | Phosphofructokinase-1 inhibitor | 0.14 0.02 CHEMBL222744 0.26 0.007 CHEMBL1256485 | CHEMBL1256485 | |
| 0.175 | 0.013 | 0.175 | Adenosine A2 receptor antagonist | 0.078 0.036 CHEMBL222744 0.12 0.022 CHEMBL1256485 | ||
| 0.233 | 0.072 | 0.233 | Cyclic AMP phosphodiesterase inhibitor | 0.151 0.15 CHEMBL1256485 | ||
| 0.169 | 0.009 | 0.188 | Phenylalanine 4-hydroxylase inhibitor | 0.188 0.008 CHEMBL222744 0.15 0.012 CHEMBL1256485 | CHEMBL222744 | |
| 0.24 | 0.087 | 0.265 | Interleukin agonist | 0.265 0.068 CHEMBL1256485 | CHEMBL1256485 | |
| 0.159 | 0.013 | 0.159 | CDK1/cyclin B inhibitor | 0.088 0.03 CHEMBL222744 0.09 0.029 CHEMBL1256485 | ||
| 0.153 | 0.009 | 0.189 | Ornithine carbamoyltransferase inhibitor | 0.084 0.02 CHEMBL222744 0.189 0.007 CHEMBL1256485 | CHEMBL1256485 | |
| 0.151 | 0.011 | 0.223 | Argininosuccinate synthase inhibitor | 0.093 0.021 CHEMBL222744 0.223 0.006 CHEMBL1256485 | CHEMBL1256485 | |
| 0.154 | 0.015 | 0.234 | Glutamate dehydrogenase inhibitor | 0.104 0.029 CHEMBL222744 0.234 0.008 CHEMBL1256485 | CHEMBL1256485 | |
| 0.147 | 0.014 | 0.147 | Cyclin B3 inhibitor | 0.069 0.046 CHEMBL222744 0.079 0.039 CHEMBL1256485 | ||
| 0.148 | 0.017 | 0.148 | MAP kinase kinase 1 inhibitor | 0.099 0.058 CHEMBL222744 | ||
| 0.169 | 0.038 | 0.169 | Alkylator | 0.133 0.057 CHEMBL222744 0.14 0.052 CHEMBL1256485 | ||
| 0.139 | 0.012 | 0.237 | Interferon agonist | 0.237 0.005 CHEMBL222744 0.107 0.024 CHEMBL1256485 | CHEMBL222744 | |
| 0.139 | 0.013 | 0.163 | Carbamoyl phosphate synthetase inhibitor | 0.097 0.021 CHEMBL222744 0.163 0.01 CHEMBL1256485 | CHEMBL1256485 | |
| 0.176 | 0.056 | 0.25 | Diuretic | 0.25 0.03 CHEMBL1256485 | CHEMBL1256485 | |
| 0.15 | 0.034 | 0.218 | Xanthine oxidase inhibitor | 0.168 0.028 CHEMBL222744 0.218 0.016 CHEMBL1256485 | CHEMBL1256485 | |
| 0.129 | 0.018 | 0.129 | Adenosine A1 receptor antagonist | 0.088 0.026 CHEMBL222744 0.114 0.02 CHEMBL1256485 | ||
| 0.132 | 0.022 | 0.132 | Phosphodiesterase I inhibitor | 0.094 0.053 CHEMBL222744 0.12 0.027 CHEMBL1256485 | ||
| 0.15 | 0.041 | 0.15 | Cyclin-dependent kinase 1 inhibitor | |||
| 0.162 | 0.053 | 0.27 | Cytokine production inhibitor | 0.27 0.02 CHEMBL222744 0.169 0.049 CHEMBL1256485 | CHEMBL222744 | |
| 0.166 | 0.058 | 0.166 | CDC-like kinase 1 inhibitor | 0.128 0.088 CHEMBL1256485 | ||
| 0.115 | 0.008 | 0.173 | Interferon inducer | 0.173 0.004 CHEMBL222744 0.09 0.017 CHEMBL1256485 | CHEMBL222744 | |
| 0.176 | 0.071 | 0.176 | Tumour necrosis factor antagonist | 0.17 0.076 CHEMBL222744 0.143 0.11 CHEMBL1256485 | ||
| 0.154 | 0.049 | 0.154 | MAP kinase kinase inhibitor | |||
| 0.141 | 0.041 | 0.141 | GABA receptor agonist | |||
| 0.107 | 0.009 | 0.109 | Adenosine A2b receptor antagonist | 0.061 0.024 CHEMBL222744 0.109 0.009 CHEMBL1256485 | CHEMBL1256485 | |
| 0.201 | 0.108 | 0.208 | Tumour necrosis factor alpha release inhibitor | 0.163 0.141 CHEMBL222744 0.208 0.102 CHEMBL1256485 | CHEMBL1256485 | |
| 0.106 | 0.017 | 0.162 | Biliverdin reductase inhibitor | 0.065 0.035 CHEMBL222744 0.162 0.008 CHEMBL1256485 | CHEMBL1256485 | |
| 0.112 | 0.024 | 0.112 | CDK1/cyclin B1 inhibitor | 0.064 0.055 CHEMBL1256485 | ||
| 0.11 | 0.023 | 0.11 | mTOR complex 2 inhibitor | 0.089 0.048 CHEMBL222744 0.078 0.074 CHEMBL1256485 | ||
| 0.093 | 0.007 | 0.093 | Phosphoglycerate kinase inhibitor | 0.048 0.015 CHEMBL222744 0.072 0.009 CHEMBL1256485 | ||
| 0.091 | 0.005 | 0.116 | Thymidylate synthase inhibitor | 0.116 0.004 CHEMBL222744 0.092 0.005 CHEMBL1256485 | CHEMBL222744 | |
| 0.194 | 0.108 | 0.194 | Peptidyltransferase inhibitor | 0.18 0.129 CHEMBL222744 0.18 0.129 CHEMBL1256485 | ||
| 0.141 | 0.055 | 0.141 | Death-associated protein kinase 1 inhibitor | 0.135 0.069 CHEMBL1256485 | ||
| 0.111 | 0.025 | 0.111 | Myeloperoxidase inhibitor | 0.096 0.04 CHEMBL222744 0.105 0.03 CHEMBL1256485 | ||
| 0.178 | 0.096 | 0.185 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.185 0.086 CHEMBL1256485 | CHEMBL1256485 | |
| 0.142 | 0.071 | 0.142 | Ribosomal protein S6 kinase inhibitor | |||
| 0.117 | 0.047 | 0.117 | CDC-like kinase 3 inhibitor | |||
| 0.08 | 0.011 | 0.08 | Nicotinic acid receptor 1 agonist | 0.069 0.013 CHEMBL1256485 | ||
| 0.208 | 0.142 | 0.272 | Hypoxia-inducible factor 1 alpha inhibitor | 0.272 0.082 CHEMBL1256485 | CHEMBL1256485 | |
| 0.084 | 0.019 | 0.084 | Cyclin B1 inhibitor | 0.058 0.047 CHEMBL1256485 | ||
| 0.093 | 0.027 | 0.093 | Adenosine A2a receptor antagonist | 0.055 0.049 CHEMBL1256485 | ||
| 0.073 | 0.009 | 0.1 | AICAR transformylase inhibitor | 0.047 0.027 CHEMBL222744 0.1 0.005 CHEMBL1256485 | CHEMBL1256485 | |
| 0.245 | 0.181 | 0.261 | Antibacterial | 0.261 0.166 CHEMBL1256485 | CHEMBL1256485 | |
| 0.121 | 0.057 | 0.121 | Cyclin-dependent kinase 5 inhibitor | |||
| 0.078 | 0.016 | 0.078 | Cyclin B2 inhibitor | 0.055 0.039 CHEMBL1256485 | ||
| 0.077 | 0.017 | 0.077 | Cyclin B inhibitor | 0.054 0.04 CHEMBL1256485 | ||
| 0.176 | 0.122 | 0.176 | ErbB-1 antagonist | |||
| 0.086 | 0.032 | 0.086 | MAP kinase kinase 7 inhibitor | 0.074 0.067 CHEMBL1256485 | ||
| 0.078 | 0.025 | 0.104 | Xanthine dehydrogenase inhibitor | 0.104 0.014 CHEMBL222744 0.066 0.034 CHEMBL1256485 | CHEMBL222744 | |
| 0.103 | 0.05 | 0.103 | CDK/cyclin complex inhibitor | |||
| 0.087 | 0.035 | 0.087 | Phosphodiesterase V inhibitor | 0.065 0.057 CHEMBL222744 0.072 0.049 CHEMBL1256485 | ||
| 0.087 | 0.035 | 0.088 | Adenosine A3 receptor antagonist | 0.088 0.034 CHEMBL222744 0.082 0.04 CHEMBL1256485 | CHEMBL222744 | |
| 0.104 | 0.054 | 0.104 | mTOR complex 1 inhibitor | |||
| 0.111 | 0.061 | 0.138 | Nav1.4 sodium channel blocker | 0.098 0.079 CHEMBL222744 0.138 0.04 CHEMBL1256485 | CHEMBL1256485 | |
| 0.103 | 0.054 | 0.167 | Electrolyte absorption antagonist | 0.167 0.014 CHEMBL1256485 | CHEMBL1256485 | |
| 0.047 | 0.002 | 0.047 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.036 0.002 CHEMBL222744 0.043 0.002 CHEMBL1256485 | ||
| 0.112 | 0.067 | 0.112 | CDK3/cyclin E inhibitor | |||
| 0.082 | 0.038 | 0.082 | Phosphodiesterase 5A inhibitor | 0.062 0.059 CHEMBL222744 0.067 0.053 CHEMBL1256485 | ||
| 0.14 | 0.096 | 0.14 | Polo-like kinase-3 inhibitor | |||
| 0.047 | 0.004 | 0.047 | DNA polymerase III inhibitor | 0.046 0.004 CHEMBL222744 0.038 0.005 CHEMBL1256485 | ||
| 0.055 | 0.014 | 0.064 | Dihydropteroate synthase inhibitor | 0.054 0.014 CHEMBL222744 0.064 0.01 CHEMBL1256485 | CHEMBL1256485 | |
| 0.051 | 0.013 | 0.087 | Fumarate hydratase inhibitor | 0.035 0.023 CHEMBL222744 0.087 0.006 CHEMBL1256485 | CHEMBL1256485 | |
| 0.056 | 0.018 | 0.056 | CDK5/p25 inhibitor | |||
| 0.133 | 0.099 | 0.133 | MAP kinase 3 inhibitor | |||
| 0.036 | 0.004 | 0.036 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.021 0.013 CHEMBL222744 0.029 0.005 CHEMBL1256485 | ||
| 0.041 | 0.011 | 0.068 | Uridine phosphorylase inhibitor | 0.068 0.004 CHEMBL222744 | CHEMBL222744 | |
| 0.099 | 0.07 | 0.128 | Adenylate kinase inhibitor | 0.128 0.037 CHEMBL1256485 | CHEMBL1256485 | |
| 0.055 | 0.028 | 0.055 | Antiviral (Hepatitis D) | 0.053 0.032 CHEMBL1256485 | ||
| 0.215 | 0.189 | 0.225 | GABA C receptor rho-3 antagonist | 0.225 0.179 CHEMBL1256485 | CHEMBL1256485 | |
| 0.049 | 0.024 | 0.049 | Phosphodiesterase 6C inhibitor | 0.049 0.024 CHEMBL222744 | ||
| 0.057 | 0.035 | 0.158 | Phosphodiesterase II inhibitor | 0.158 0.005 CHEMBL222744 | CHEMBL222744 | |
| 0.038 | 0.018 | 0.04 | Purinergic P2Y2 antagonist | 0.04 0.016 CHEMBL222744 0.038 0.017 CHEMBL1256485 | CHEMBL222744 | |
| 0.063 | 0.043 | 0.063 | Phosphodiesterase VII inhibitor | |||
| 0.085 | 0.067 | 0.085 | Aminoacyl-tRNA synthetase inhibitor | |||
| 0.104 | 0.086 | 0.104 | Cyclin-dependent kinase inhibitor | |||
| 0.02 | 0.002 | 0.02 | DNA polymerase III subunit alpha inhibitor | 0.015 0.002 CHEMBL222744 0.015 0.002 CHEMBL1256485 | ||
| 0.094 | 0.077 | 0.121 | Mediator release inhibitor | 0.121 0.047 CHEMBL1256485 | CHEMBL1256485 | |
| 0.059 | 0.042 | 0.059 | Heat shock protein 90 beta antagonist | |||
| 0.05 | 0.034 | 0.149 | Phosphodiesterase 2A inhibitor | 0.149 0.005 CHEMBL222744 | CHEMBL222744 | |
| 0.118 | 0.103 | 0.163 | Cell wall synthesis inhibitor | 0.163 0.053 CHEMBL1256485 | CHEMBL1256485 | |
| 0.165 | 0.151 | 0.165 | DNA damaging | 0.161 0.156 CHEMBL222744 | ||
| 0.017 | 0.004 | 0.017 | DNA polymerase III polC-type inhibitor | 0.016 0.005 CHEMBL222744 0.014 0.008 CHEMBL1256485 | ||
| 0.146 | 0.134 | 0.146 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | |||
| 0.023 | 0.014 | 0.023 | Adenosine kinase inhibitor | |||
| 0.083 | 0.076 | 0.083 | Polo-like kinase-1 inhibitor | |||
| 0.011 | 0.003 | 0.012 | Phosphoribosylglycinamide formyltransferase inhibitor | 0.011 0.003 CHEMBL222744 0.012 0.003 CHEMBL1256485 | CHEMBL1256485 | |
| 0.064 | 0.057 | 0.064 | CDK2/cyclin E2 inhibitor | |||
| 0.041 | 0.035 | 0.419 | Phosphodiesterase 3B inhibitor | 0.419 0.003 CHEMBL222744 | CHEMBL222744 | |
| 0.077 | 0.07 | 0.077 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | |||
| 0.047 | 0.042 | 0.047 | Factor IXa inhibitor | |||
| 0.025 | 0.021 | 0.025 | Thymidine phosphorylase inhibitor | 0.024 0.022 CHEMBL222744 | ||
| 0.084 | 0.08 | 0.336 | Bronchodilator | 0.336 0.007 CHEMBL222744 | CHEMBL222744 | |
| 0.016 | 0.012 | 0.016 | Adenosine A2 receptor agonist | |||
| 0.028 | 0.025 | 0.028 | Phosphodiesterase 6B inhibitor | |||
| 0.037 | 0.034 | 0.037 | Glutamate (mGluR1a) antagonist | |||
| 0.085 | 0.083 | 0.085 | Cyclin-dependent kinase 9 inhibitor | |||
| 0.045 | 0.049 | 0.061 | Acyl-CoA dehydrogenase inhibitor | 0.061 0.032 CHEMBL1256485 | CHEMBL1256485 | |
| 0.074 | 0.094 | 0.082 | T cell inhibitor | 0.082 0.058 CHEMBL1256485 | CHEMBL1256485 | |
| 0.016 | 0.039 | 0.023 | Toll-Like receptor 8 agonist | 0.023 0.008 CHEMBL222744 | CHEMBL222744 | |
| 0.077 | 0.1 | 0.121 | GABA C receptor agonist | 0.121 0.049 CHEMBL1256485 | CHEMBL1256485 | |
| 0.023 | 0.063 | 0.041 | RNA-directed RNA polymerase inhibitor | 0.041 0.018 CHEMBL1256485 | CHEMBL1256485 | |
| 0.023 | 0.09 | 0.034 | Tryptophan 5 hydroxylase inhibitor | 0.034 0.03 CHEMBL1256485 | CHEMBL1256485 | |
| 0.033 | 0.11 | 0.35 | Phosphodiesterase III inhibitor | 0.35 0.004 CHEMBL222744 | CHEMBL222744 | |
| 0.067 | 0.15 | 0.113 | Mucolytic | 0.113 0.061 CHEMBL1256485 | CHEMBL1256485 | |
| 0.046 | 0.136 | 0.075 | Phosphodiesterase 3A inhibitor | 0.075 0.063 CHEMBL222744 | CHEMBL222744 | |
| 0.048 | 0.175 | 0.093 | Expectorant | 0.093 0.077 CHEMBL1256485 | CHEMBL1256485 | |
| 0.062 | 0.191 | 0.173 | Phosphodiesterase inhibitor | 0.173 0.045 CHEMBL222744 | CHEMBL222744 | |
| 0.048 | 0.178 | 0.129 | Glycogen synthase kinase-3 inhibitor | 0.129 0.055 CHEMBL222744 | CHEMBL222744 | |
| 0.128 | 0.273 | 0.417 | Angiogenesis inhibitor | 0.417 0.048 CHEMBL222744 | CHEMBL222744 | |
| 0.04 | 0.2 | 0.131 | Glycogen synthase kinase-3 beta inhibitor | 0.131 0.054 CHEMBL222744 | CHEMBL222744 | |
| 0.062 | 0.24 | 0.716 | Interleukin 4 antagonist | 0.716 0.003 CHEMBL222744 | CHEMBL222744 | |
| 0.079 | 0.306 | 0.14 | Succinate dehydrogenase inhibitor | 0.14 0.132 CHEMBL1256485 | CHEMBL1256485 | |
| 0.043 | 0.3 | 0.24 | Interleukin 5 antagonist | 0.24 0.005 CHEMBL222744 | CHEMBL222744 | |
| 0.005 | 0.296 | 0.024 | Purinergic P2Y12 antagonist | 0.024 0.015 CHEMBL222744 | CHEMBL222744 | |
| 0.005 | 0.363 | 0.039 | Prostacyclin antagonist | 0.039 0.019 CHEMBL1256485 | CHEMBL1256485 | |
| 0.044 | 0.414 | 0.172 | Platelet aggregation inhibitor | 0.172 0.104 CHEMBL1256485 | CHEMBL1256485 | |
| 0.061 | 0.513 | 0.332 | Toll-Like receptor agonist | 0.332 0.092 CHEMBL222744 | CHEMBL222744 | |
| 0.056 | 0.539 | 0.312 | Toll-Like receptor 7 agonist | 0.312 0.103 CHEMBL222744 | CHEMBL222744 | |
| 0.002 | 0.588 | 0.036 | Prostacyclin agonist | 0.036 0.005 CHEMBL1256485 | CHEMBL1256485 | |
| 0.016 | 0.632 | 0.208 | Platelet antagonist | 0.208 0.095 CHEMBL1256485 | CHEMBL1256485 | |
| 0.002 | 0.848 | 0.039 | Prostaglandin D2 agonist | 0.039 0.013 CHEMBL1256485 | CHEMBL1256485 | |
| 0.015 | 0.929 | 0.062 | Heme oxygenase stimulant | 0.062 0.04 CHEMBL222744 | CHEMBL222744 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |