| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.918 | 0.001 | 0.918 | Peroxisome proliferator-activated receptor alpha agonist | 0.854 0.001 CHEMBL254989 0.366 0.003 CHEMBL4525746 | ||
| 0.907 | 0.002 | 0.912 | Peroxisome proliferator-activated receptor gamma agonist | 0.912 0.002 CHEMBL254989 0.733 0.003 CHEMBL4525746 | CHEMBL254989 | |
| 0.887 | 0.002 | 0.911 | Insulin sensitizer | 0.911 0.002 CHEMBL254989 0.618 0.003 CHEMBL4525746 | CHEMBL254989 | |
| 0.875 | 0.005 | 0.897 | Cyclophilin D inhibitor | 0.888 0.005 CHEMBL254989 0.897 0.005 CHEMBL4525746 | CHEMBL4525746 | |
| 0.803 | 0.001 | 0.803 | Peroxisome proliferator-activated receptor gamma antagonist | 0.751 0.001 CHEMBL254989 0.204 0.004 CHEMBL4525746 | ||
| 0.777 | 0.004 | 0.809 | Hypoglycemic | 0.8 0.004 CHEMBL254989 0.809 0.004 CHEMBL4525746 | CHEMBL4525746 | |
| 0.757 | 0.001 | 0.757 | Peroxisome proliferator-activated receptor alpha antagonist | 0.729 0.001 CHEMBL254989 0.134 0.004 CHEMBL4525746 | ||
| 0.672 | 0.005 | 0.688 | Hypolipemic | 0.688 0.005 CHEMBL254989 0.619 0.006 CHEMBL4525746 | CHEMBL254989 | |
| 0.513 | 0.035 | 0.541 | Antiobesity | 0.541 0.029 CHEMBL254989 0.468 0.045 CHEMBL4525746 | CHEMBL254989 | |
| 0.326 | 0.057 | 0.345 | Sodium/bile acid cotransporter inhibitor | 0.345 0.043 CHEMBL254989 | CHEMBL254989 | |
| 0.281 | 0.013 | 0.346 | Chelator | 0.346 0.008 CHEMBL254989 0.141 0.039 CHEMBL4525746 | CHEMBL254989 | |
| 0.335 | 0.071 | 0.543 | Cholesterol antagonist | 0.394 0.051 CHEMBL254989 0.543 0.026 CHEMBL4525746 | CHEMBL4525746 | |
| 0.269 | 0.016 | 0.298 | Insulin secretagoues | 0.285 0.014 CHEMBL254989 0.298 0.013 CHEMBL4525746 | CHEMBL4525746 | |
| 0.238 | 0.034 | 0.268 | Protein-tyrosine phosphatase inhibitor | 0.268 0.026 CHEMBL254989 0.217 0.041 CHEMBL4525746 | CHEMBL254989 | |
| 0.252 | 0.05 | 0.332 | Peptidyltransferase inhibitor | 0.272 0.037 CHEMBL254989 0.332 0.015 CHEMBL4525746 | CHEMBL4525746 | |
| 0.218 | 0.028 | 0.218 | Acetylcholinesterase inhibitor | 0.206 0.031 CHEMBL254989 0.12 0.078 CHEMBL4525746 | ||
| 0.194 | 0.004 | 0.2 | Peroxisome proliferator-activated receptor delta antagonist | 0.2 0.004 CHEMBL254989 0.052 0.009 CHEMBL4525746 | CHEMBL254989 | |
| 0.205 | 0.028 | 0.227 | Protein-tyrosine phosphatase 1B inhibitor | 0.227 0.022 CHEMBL254989 0.208 0.027 CHEMBL4525746 | CHEMBL254989 | |
| 0.193 | 0.05 | 0.193 | Cholinergic | 0.179 0.057 CHEMBL254989 | ||
| 0.134 | 0.004 | 0.134 | Peroxisome proliferator-activated receptor delta agonist | 0.095 0.006 CHEMBL254989 | ||
| 0.154 | 0.032 | 0.154 | Butyrylcholinesterase inhibitor | 0.147 0.035 CHEMBL254989 | ||
| 0.197 | 0.079 | 0.224 | Amyloid beta aggregation inhibitor | 0.224 0.067 CHEMBL254989 0.207 0.074 CHEMBL4525746 | CHEMBL254989 | |
| 0.219 | 0.102 | 0.509 | Antioxidant | 0.271 0.073 CHEMBL254989 0.509 0.019 CHEMBL4525746 | CHEMBL4525746 | |
| 0.113 | 0.008 | 0.113 | Phosphodiesterase VIII inhibitor | 0.112 0.008 CHEMBL254989 0.093 0.019 CHEMBL4525746 | ||
| 0.115 | 0.018 | 0.133 | Potassium channel large-conductance Ca-activated activator | 0.133 0.014 CHEMBL254989 0.133 0.014 CHEMBL4525746 | CHEMBL4525746 | |
| 0.137 | 0.055 | 0.137 | Vanilloid 1 agonist | 0.131 0.064 CHEMBL254989 0.117 0.094 CHEMBL4525746 | ||
| 0.214 | 0.137 | 0.259 | Insulysin inhibitor | 0.259 0.088 CHEMBL254989 | CHEMBL254989 | |
| 0.119 | 0.051 | 0.151 | MAO B inhibitor | 0.151 0.037 CHEMBL254989 | CHEMBL254989 | |
| 0.071 | 0.003 | 0.071 | Thiazolidinedione | 0.069 0.003 CHEMBL254989 0.048 0.006 CHEMBL4525746 | ||
| 0.099 | 0.033 | 0.099 | Phosphodiesterase 11A inhibitor | 0.081 0.058 CHEMBL254989 | ||
| 0.099 | 0.033 | 0.099 | Phosphodiesterase XI inhibitor | 0.081 0.058 CHEMBL254989 | ||
| 0.156 | 0.093 | 0.168 | Catenin beta inhibitor | 0.168 0.069 CHEMBL254989 | CHEMBL254989 | |
| 0.11 | 0.048 | 0.144 | Potassium channel (Ca-activated) activator | 0.144 0.03 CHEMBL254989 0.083 0.072 CHEMBL4525746 | CHEMBL254989 | |
| 0.175 | 0.119 | 0.427 | Antiamyloidogenic | 0.175 0.119 CHEMBL254989 0.427 0.025 CHEMBL4525746 | CHEMBL4525746 | |
| 0.125 | 0.072 | 0.167 | MAO inhibitor | 0.167 0.053 CHEMBL254989 | CHEMBL254989 | |
| 0.196 | 0.145 | 0.234 | Lipoxygenase inhibitor | 0.234 0.111 CHEMBL254989 | CHEMBL254989 | |
| 0.099 | 0.055 | 0.113 | Interleukin 12 antagonist | 0.113 0.036 CHEMBL254989 0.105 0.046 CHEMBL4525746 | CHEMBL254989 | |
| 0.113 | 0.079 | 0.175 | Aldehyde dehydrogenase inhibitor | 0.175 0.035 CHEMBL254989 | CHEMBL254989 | |
| 0.198 | 0.164 | 0.198 | Thyroid hormone antagonist | 0.187 0.173 CHEMBL254989 | ||
| 0.074 | 0.044 | 0.083 | Amidase inhibitor | 0.083 0.035 CHEMBL254989 | CHEMBL254989 | |
| 0.158 | 0.135 | 0.422 | Free radical scavenger | 0.207 0.092 CHEMBL254989 0.422 0.025 CHEMBL4525746 | CHEMBL4525746 | |
| 0.127 | 0.105 | 0.143 | Phospholipase A2 inhibitor | 0.143 0.082 CHEMBL254989 | CHEMBL254989 | |
| 0.1 | 0.082 | 0.1 | Electron transport complex I inhibitor | |||
| 0.046 | 0.029 | 0.046 | Sphingosine 1-phosphate receptor agonist | 0.042 0.034 CHEMBL254989 | ||
| 0.041 | 0.028 | 0.042 | Integrin alpha5beta1 antagonist | 0.042 0.027 CHEMBL254989 | CHEMBL254989 | |
| 0.235 | 0.222 | 0.292 | Calcium channel L-type activator | 0.292 0.164 CHEMBL254989 | CHEMBL254989 | |
| 0.192 | 0.19 | 0.318 | Apoptosis antagonist | 0.211 0.166 CHEMBL254989 0.318 0.074 CHEMBL4525746 | CHEMBL4525746 | |
| 0.013 | 0.014 | 0.015 | Integrin beta6 antagonist | 0.015 0.009 CHEMBL254989 | CHEMBL254989 | |
| 0.025 | 0.03 | 0.027 | Liver X receptor alpha antagonist | 0.027 0.024 CHEMBL254989 | CHEMBL254989 | |
| 0.013 | 0.073 | 0.034 | Protein 30S ribosomal subunit inhibitor | 0.034 0.011 CHEMBL4525746 | CHEMBL4525746 | |
| 0.102 | 0.174 | 0.284 | Nitric oxide antagonist | 0.284 0.044 CHEMBL4525746 | CHEMBL4525746 | |
| 0.071 | 0.146 | 0.114 | Multidrug resistance-associated protein 1 inhibitor | 0.114 0.056 CHEMBL4525746 | CHEMBL4525746 | |
| 0.089 | 0.172 | 0.423 | Angiogenesis stimulant | 0.423 0.018 CHEMBL4525746 | CHEMBL4525746 | |
| 0.071 | 0.171 | 0.21 | Lipid peroxidase inhibitor | 0.21 0.038 CHEMBL4525746 | CHEMBL4525746 | |
| 0.069 | 0.178 | 0.179 | Cyclooxygenase 3 inhibitor | 0.179 0.028 CHEMBL4525746 | CHEMBL4525746 | |
| 0.074 | 0.184 | 0.128 | Interleukin 4 antagonist | 0.128 0.075 CHEMBL4525746 | CHEMBL4525746 | |
| 0.027 | 0.161 | 0.061 | Glucose-6-phosphate translocase inhibitor | 0.061 0.023 CHEMBL4525746 | CHEMBL4525746 | |
| 0.096 | 0.229 | 0.184 | Platelet antagonist | 0.184 0.114 CHEMBL4525746 | CHEMBL4525746 | |
| 0.068 | 0.204 | 0.118 | Cell adhesion inhibitor | 0.118 0.066 CHEMBL4525746 | CHEMBL4525746 | |
| 0.027 | 0.17 | 0.054 | Heparanase inhibitor | 0.054 0.035 CHEMBL4525746 | CHEMBL4525746 | |
| 0.082 | 0.228 | 0.292 | Platelet adhesion inhibitor | 0.292 0.036 CHEMBL4525746 | CHEMBL4525746 | |
| 0.035 | 0.185 | 0.064 | Adenine nucleotide translocase inhibitor | 0.064 0.022 CHEMBL4525746 | CHEMBL4525746 | |
| 0.039 | 0.226 | 0.084 | ATPase (Vacuolar H+) inhibitor | 0.084 0.07 CHEMBL4525746 | CHEMBL4525746 | |
| 0.055 | 0.248 | 0.108 | Estrogen antagonist | 0.108 0.078 CHEMBL254989 | CHEMBL254989 | |
| 0.025 | 0.23 | 0.108 | Monophenol monooxygenase inhibitor | 0.108 0.07 CHEMBL4525746 | CHEMBL4525746 | |
| 0.029 | 0.238 | 0.191 | Topoisomerase I inhibitor | 0.191 0.029 CHEMBL4525746 | CHEMBL4525746 | |
| 0.041 | 0.255 | 0.151 | Alkylator | 0.151 0.046 CHEMBL4525746 | CHEMBL4525746 | |
| 0.068 | 0.295 | 0.246 | Hepatoprotectant | 0.246 0.044 CHEMBL4525746 | CHEMBL4525746 | |
| 0.045 | 0.291 | 0.09 | Transcription factor NF kappa B stimulant | 0.09 0.051 CHEMBL4525746 | CHEMBL4525746 | |
| 0.045 | 0.291 | 0.122 | Toll-Like receptor 4 antagonist | 0.122 0.042 CHEMBL4525746 | CHEMBL4525746 | |
| 0.038 | 0.289 | 0.089 | Estrogen receptor beta antagonist | 0.089 0.085 CHEMBL254989 | CHEMBL254989 | |
| 0.013 | 0.279 | 0.208 | Selectin antagonist | 0.208 0.01 CHEMBL4525746 | CHEMBL4525746 | |
| 0.035 | 0.312 | 0.149 | Thrombolytic | 0.149 0.083 CHEMBL4525746 | CHEMBL4525746 | |
| 0.009 | 0.287 | 0.087 | Antineoplastic antibiotic | 0.087 0.053 CHEMBL4525746 | CHEMBL4525746 | |
| 0.015 | 0.318 | 0.047 | Antibiotic Aminoglycoside-like | 0.047 0.015 CHEMBL4525746 | CHEMBL4525746 | |
| 0.013 | 0.339 | 0.055 | Protein 50S ribosomal subunit inhibitor | 0.055 0.035 CHEMBL4525746 | CHEMBL4525746 | |
| 0.038 | 0.365 | 0.118 | Anticoagulant | 0.118 0.115 CHEMBL4525746 | CHEMBL4525746 | |
| 0.018 | 0.349 | 0.099 | Topoisomerase II alpha inhibitor | 0.099 0.04 CHEMBL4525746 | CHEMBL4525746 | |
| 0.103 | 0.463 | 0.354 | Interleukin 2 agonist | 0.354 0.044 CHEMBL4525746 | CHEMBL4525746 | |
| 0.067 | 0.448 | 0.249 | Antithrombotic | 0.249 0.127 CHEMBL4525746 | CHEMBL4525746 | |
| 0.054 | 0.47 | 0.357 | Immunosuppressant | 0.357 0.083 CHEMBL4525746 | CHEMBL4525746 | |
| 0.028 | 0.481 | 0.318 | Immunostimulant | 0.318 0.074 CHEMBL4525746 | CHEMBL4525746 | |
| 0.037 | 0.498 | 0.227 | Tumour necrosis factor alpha release inhibitor | 0.227 0.087 CHEMBL4525746 | CHEMBL4525746 | |
| 0.02 | 0.503 | 0.104 | Beta glucuronidase inhibitor | 0.104 0.064 CHEMBL4525746 | CHEMBL4525746 | |
| 0.07 | 0.561 | 0.416 | Apoptosis agonist | 0.416 0.106 CHEMBL4525746 | CHEMBL4525746 | |
| 0.012 | 0.545 | 0.105 | Topoisomerase II inhibitor | 0.105 0.081 CHEMBL4525746 | CHEMBL4525746 | |
| 0.029 | 0.584 | 0.306 | Transcription factor NF kappa B inhibitor | 0.306 0.091 CHEMBL4525746 | CHEMBL4525746 | |
| 0.043 | 0.711 | 0.456 | Antiinflammatory | 0.456 0.107 CHEMBL4525746 | CHEMBL4525746 | |
| 0.018 | 0.732 | 0.418 | Antibacterial | 0.418 0.069 CHEMBL4525746 | CHEMBL4525746 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |