| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.992 | 0.002 | 0.992 | Toll-Like receptor agonist | 0.989 0.003 CHEMBL3706465 0.971 0.003 CHEMBL3706466 0.988 0.003 CHEMBL3706467 0.954 0.004 CHEMBL3706471 0.985 0.003 CHEMBL3706468 0.986 0.003 CHEMBL3706479 0.957 0.004 CHEMBL3706472 0.96 0.004 CHEMBL3706474 | ||
| 0.992 | 0.002 | 0.992 | Toll-Like receptor 7 agonist | 0.989 0.003 CHEMBL3706465 0.97 0.003 CHEMBL3706466 0.988 0.003 CHEMBL3706467 0.952 0.004 CHEMBL3706471 0.985 0.003 CHEMBL3706468 0.986 0.003 CHEMBL3706479 0.955 0.004 CHEMBL3706472 0.959 0.004 CHEMBL3706474 | ||
| 0.931 | 0.003 | 0.931 | Spasmolytic | 0.819 0.004 CHEMBL3706465 0.222 0.104 CHEMBL3706466 0.826 0.004 CHEMBL3706467 0.332 0.058 CHEMBL3706471 0.827 0.004 CHEMBL3706468 0.908 0.003 CHEMBL3706479 0.351 0.052 CHEMBL3706472 0.791 0.004 CHEMBL3706474 0.197 0.122 CHEMBL1222314 | ||
| 0.905 | 0.003 | 0.948 | Bronchodilator | 0.948 0.003 CHEMBL3706465 0.32 0.008 CHEMBL3706466 0.787 0.003 CHEMBL3706467 0.415 0.005 CHEMBL3706471 0.765 0.004 CHEMBL3706468 0.794 0.003 CHEMBL3706479 0.446 0.005 CHEMBL3706472 0.6 0.004 CHEMBL3706474 0.086 0.079 CHEMBL3706478 | CHEMBL3706465 | |
| 0.902 | 0.002 | 0.902 | Cholinergic antagonist | 0.58 0.004 CHEMBL3706465 0.283 0.016 CHEMBL3706466 0.814 0.002 CHEMBL3706467 0.597 0.004 CHEMBL3706471 0.896 0.002 CHEMBL3706468 0.869 0.002 CHEMBL3706479 0.441 0.006 CHEMBL3706472 0.703 0.003 CHEMBL3706474 0.104 0.091 CHEMBL3706475 0.163 0.046 CHEMBL3706478 0.102 0.093 CHEMBL1222314 | ||
| 0.89 | 0.002 | 0.89 | Acetylcholine antagonist | 0.564 0.004 CHEMBL3706465 0.27 0.017 CHEMBL3706466 0.803 0.003 CHEMBL3706467 0.584 0.004 CHEMBL3706471 0.885 0.002 CHEMBL3706468 0.859 0.002 CHEMBL3706479 0.427 0.006 CHEMBL3706472 0.687 0.003 CHEMBL3706474 0.101 0.091 CHEMBL3706475 0.155 0.047 CHEMBL3706478 0.098 0.095 CHEMBL1222314 | ||
| 0.879 | 0.001 | 0.884 | Acetylcholine muscarinic antagonist | 0.488 0.004 CHEMBL3706465 0.312 0.008 CHEMBL3706466 0.797 0.002 CHEMBL3706467 0.558 0.003 CHEMBL3706471 0.884 0.001 CHEMBL3706468 0.848 0.002 CHEMBL3706479 0.386 0.005 CHEMBL3706472 0.649 0.003 CHEMBL3706474 0.132 0.056 CHEMBL3706475 0.194 0.026 CHEMBL3706478 0.131 0.057 CHEMBL1222314 | CHEMBL3706468 | |
| 0.778 | 0.002 | 0.818 | Acetylcholine M1 receptor antagonist | 0.508 0.004 CHEMBL3706465 0.265 0.022 CHEMBL3706466 0.651 0.003 CHEMBL3706467 0.524 0.004 CHEMBL3706471 0.818 0.002 CHEMBL3706468 0.729 0.003 CHEMBL3706479 0.488 0.004 CHEMBL3706472 0.461 0.004 CHEMBL3706474 0.187 0.048 CHEMBL3706475 0.116 0.115 CHEMBL1222314 | CHEMBL3706468 | |
| 0.773 | 0.001 | 0.773 | Acetylcholine M3 receptor antagonist | 0.367 0.003 CHEMBL3706465 0.261 0.005 CHEMBL3706466 0.648 0.002 CHEMBL3706467 0.282 0.004 CHEMBL3706471 0.768 0.001 CHEMBL3706468 0.744 0.001 CHEMBL3706479 0.105 0.017 CHEMBL3706472 0.517 0.002 CHEMBL3706474 0.072 0.03 CHEMBL3706475 0.169 0.009 CHEMBL3706478 0.084 0.024 CHEMBL1222314 | ||
| 0.681 | 0.002 | 0.705 | Acetylcholine M2 receptor antagonist | 0.3 0.004 CHEMBL3706465 0.091 0.024 CHEMBL3706466 0.5 0.003 CHEMBL3706467 0.139 0.013 CHEMBL3706471 0.705 0.002 CHEMBL3706468 0.611 0.003 CHEMBL3706479 0.097 0.022 CHEMBL3706472 0.311 0.004 CHEMBL3706474 | CHEMBL3706468 | |
| 0.456 | 0.02 | 0.458 | Cardiotonic | 0.458 0.02 CHEMBL3706465 0.179 0.14 CHEMBL3706466 0.207 0.112 CHEMBL3706467 0.213 0.107 CHEMBL3706468 0.347 0.04 CHEMBL3706479 | CHEMBL3706465 | |
| 0.436 | 0.003 | 0.452 | Acetylcholine M4 receptor antagonist | 0.25 0.005 CHEMBL3706465 0.075 0.052 CHEMBL3706466 0.253 0.005 CHEMBL3706467 0.452 0.003 CHEMBL3706468 0.363 0.004 CHEMBL3706479 0.216 0.005 CHEMBL3706474 | CHEMBL3706468 | |
| 0.354 | 0.006 | 0.541 | Expectorant | 0.218 0.017 CHEMBL3706465 0.315 0.008 CHEMBL3706466 0.283 0.01 CHEMBL3706467 0.541 0.003 CHEMBL3706471 0.311 0.008 CHEMBL3706468 0.319 0.007 CHEMBL3706479 0.373 0.005 CHEMBL3706472 0.24 0.014 CHEMBL3706474 0.205 0.019 CHEMBL3706475 0.322 0.007 CHEMBL3706478 0.476 0.004 CHEMBL1222314 | CHEMBL3706471 | |
| 0.306 | 0.004 | 0.45 | Mucolytic | 0.197 0.014 CHEMBL3706465 0.315 0.004 CHEMBL3706466 0.251 0.006 CHEMBL3706467 0.389 0.003 CHEMBL3706471 0.268 0.005 CHEMBL3706468 0.276 0.005 CHEMBL3706479 0.262 0.005 CHEMBL3706472 0.221 0.01 CHEMBL3706474 0.211 0.011 CHEMBL3706475 0.312 0.004 CHEMBL3706478 0.45 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.329 | 0.074 | 0.482 | Cholesterol antagonist | 0.477 0.036 CHEMBL3706465 0.482 0.035 CHEMBL3706466 0.185 0.179 CHEMBL3706467 0.22 0.148 CHEMBL3706468 0.296 0.094 CHEMBL3706479 0.262 0.116 CHEMBL3706474 0.365 0.059 CHEMBL3706475 0.434 0.043 CHEMBL3706478 0.471 0.037 CHEMBL1222314 | CHEMBL3706466 | |
| 0.251 | 0.009 | 0.393 | Acetylcholine nicotinic antagonist | 0.393 0.005 CHEMBL3706465 0.115 0.032 CHEMBL3706467 0.102 0.038 CHEMBL3706468 0.205 0.012 CHEMBL3706479 0.251 0.009 CHEMBL3706474 | CHEMBL3706465 | |
| 0.224 | 0.004 | 0.249 | Acetylcholine M5 receptor antagonist | 0.192 0.005 CHEMBL3706465 0.054 0.052 CHEMBL3706466 0.134 0.01 CHEMBL3706467 0.249 0.004 CHEMBL3706468 0.192 0.005 CHEMBL3706479 0.076 0.026 CHEMBL3706474 | CHEMBL3706468 | |
| 0.215 | 0.004 | 0.215 | Acetylcholine M3 receptor agonist | 0.177 0.008 CHEMBL3706465 0.17 0.01 CHEMBL3706466 0.208 0.004 CHEMBL3706467 0.144 0.023 CHEMBL3706471 0.203 0.004 CHEMBL3706468 0.191 0.005 CHEMBL3706479 0.14 0.024 CHEMBL3706472 0.175 0.009 CHEMBL3706474 | ||
| 0.221 | 0.038 | 0.244 | Cytidine deaminase inhibitor | 0.236 0.033 CHEMBL3706465 0.164 0.066 CHEMBL3706466 0.183 0.055 CHEMBL3706479 0.244 0.031 CHEMBL3706474 0.118 0.103 CHEMBL3706478 0.23 0.035 CHEMBL1222314 | CHEMBL3706474 | |
| 0.165 | 0.011 | 0.165 | Adrenaline agonist | 0.072 0.069 CHEMBL3706465 0.136 0.019 CHEMBL3706466 0.077 0.062 CHEMBL3706467 0.076 0.063 CHEMBL3706468 0.094 0.042 CHEMBL3706479 0.093 0.042 CHEMBL3706478 0.104 0.034 CHEMBL1222314 | ||
| 0.121 | 0.004 | 0.121 | Beta 2 adrenoreceptor agonist | 0.072 0.016 CHEMBL3706465 0.085 0.007 CHEMBL3706466 0.084 0.007 CHEMBL3706467 0.06 0.051 CHEMBL3706471 0.086 0.006 CHEMBL3706468 0.09 0.005 CHEMBL3706479 0.066 0.027 CHEMBL3706474 0.06 0.049 CHEMBL3706475 0.073 0.015 CHEMBL3706478 0.073 0.015 CHEMBL1222314 | ||
| 0.147 | 0.051 | 0.188 | Ca2+-transporting ATPase inhibitor | 0.188 0.005 CHEMBL3706465 0.162 0.021 CHEMBL3706466 0.13 0.12 CHEMBL3706467 0.133 0.103 CHEMBL3706468 0.142 0.065 CHEMBL3706479 0.147 0.049 CHEMBL3706474 0.179 0.008 CHEMBL3706475 0.165 0.018 CHEMBL3706478 0.174 0.01 CHEMBL1222314 | CHEMBL3706465 | |
| 0.197 | 0.107 | 0.528 | Vasodilator | 0.528 0.01 CHEMBL3706465 0.221 0.089 CHEMBL3706479 0.166 0.136 CHEMBL3706472 0.304 0.046 CHEMBL3706474 | CHEMBL3706465 | |
| 0.205 | 0.142 | 0.425 | 5 Hydroxytryptamine uptake stimulant | 0.425 0.01 CHEMBL3706465 0.273 0.062 CHEMBL3706466 0.189 0.176 CHEMBL3706479 0.257 0.074 CHEMBL3706474 0.297 0.046 CHEMBL3706475 0.248 0.083 CHEMBL3706478 0.318 0.037 CHEMBL1222314 | CHEMBL3706465 | |
| 0.104 | 0.044 | 0.13 | Acetylcholine agonist | 0.13 0.033 CHEMBL3706465 0.09 0.055 CHEMBL3706479 | CHEMBL3706465 | |
| 0.119 | 0.062 | 0.178 | Microtubule formation inhibitor | 0.159 0.033 CHEMBL3706465 0.144 0.041 CHEMBL3706466 0.108 0.078 CHEMBL3706479 0.122 0.059 CHEMBL3706474 0.163 0.031 CHEMBL3706475 0.163 0.031 CHEMBL3706478 0.178 0.026 CHEMBL1222314 | CHEMBL1222314 | |
| 0.135 | 0.08 | 0.302 | Cell wall synthesis inhibitor | 0.183 0.038 CHEMBL3706465 0.208 0.027 CHEMBL3706466 0.124 0.094 CHEMBL3706474 0.16 0.056 CHEMBL3706475 0.302 0.01 CHEMBL3706478 0.261 0.014 CHEMBL1222314 | CHEMBL3706478 | |
| 0.062 | 0.007 | 0.062 | Beta adrenoreceptor agonist | 0.057 0.01 CHEMBL3706466 0.045 0.033 CHEMBL3706467 0.045 0.032 CHEMBL3706468 0.048 0.023 CHEMBL3706479 0.048 0.021 CHEMBL3706478 0.051 0.015 CHEMBL1222314 | ||
| 0.149 | 0.111 | 0.893 | Hepatoprotectant | 0.216 0.056 CHEMBL3706465 0.149 0.111 CHEMBL3706466 0.158 0.101 CHEMBL3706467 0.47 0.008 CHEMBL3706471 0.561 0.005 CHEMBL3706468 0.135 0.126 CHEMBL3706479 0.501 0.007 CHEMBL3706472 0.893 0.002 CHEMBL3706475 0.14 0.121 CHEMBL3706478 | CHEMBL3706475 | |
| 0.057 | 0.024 | 0.182 | Nicotinic receptor alpha4 subunit antagonist | 0.182 0.004 CHEMBL3706465 0.053 0.028 CHEMBL3706479 0.091 0.01 CHEMBL3706474 | CHEMBL3706465 | |
| 0.058 | 0.026 | 0.11 | Glucose-6-phosphate translocase inhibitor | 0.087 0.009 CHEMBL3706466 0.05 0.039 CHEMBL3706468 0.055 0.03 CHEMBL3706479 0.063 0.021 CHEMBL3706474 0.073 0.014 CHEMBL3706475 0.076 0.013 CHEMBL3706478 0.11 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.06 | 0.034 | 0.075 | Acetylcholine muscarinic agonist | 0.075 0.024 CHEMBL3706465 0.049 0.044 CHEMBL3706479 | CHEMBL3706465 | |
| 0.06 | 0.038 | 0.101 | Dopamine uptake inhibitor | 0.101 0.018 CHEMBL3706465 0.098 0.019 CHEMBL3706474 | CHEMBL3706465 | |
| 0.049 | 0.033 | 0.112 | Dopamine transporter inhibitor | 0.112 0.009 CHEMBL3706465 0.043 0.04 CHEMBL3706479 0.092 0.014 CHEMBL3706474 | CHEMBL3706465 | |
| 0.036 | 0.02 | 0.05 | Tubulin agonist | 0.046 0.01 CHEMBL3706465 0.034 0.025 CHEMBL3706466 0.032 0.028 CHEMBL3706467 0.036 0.02 CHEMBL3706468 0.035 0.022 CHEMBL3706479 0.036 0.02 CHEMBL3706474 0.05 0.008 CHEMBL3706475 0.032 0.03 CHEMBL3706478 0.036 0.021 CHEMBL1222314 | CHEMBL3706475 | |
| 0.045 | 0.034 | 0.052 | Microtubule stabilization | 0.052 0.025 CHEMBL3706465 0.041 0.039 CHEMBL3706468 0.043 0.038 CHEMBL3706479 0.045 0.034 CHEMBL3706474 | CHEMBL3706465 | |
| 0.074 | 0.073 | 0.216 | Antineoplastic alkaloid | 0.216 0.01 CHEMBL3706465 | CHEMBL3706465 | |
| 0.042 | 0.058 | 0.073 | Acetylcholine M2 receptor agonist | 0.073 0.017 CHEMBL3706465 0.053 0.038 CHEMBL3706474 | CHEMBL3706465 | |
| 0.023 | 0.041 | 0.036 | 1,3-Beta-glucan synthase inhibitor | 0.036 0.005 CHEMBL3706465 | CHEMBL3706465 | |
| 0.074 | 0.094 | 0.118 | ATPase (Vacuolar H+) inhibitor | 0.118 0.021 CHEMBL3706465 0.082 0.074 CHEMBL3706475 0.107 0.031 CHEMBL3706478 | CHEMBL3706465 | |
| 0.037 | 0.058 | 0.124 | Beta 2 adrenoreceptor antagonist | 0.124 0.006 CHEMBL3706466 0.072 0.015 CHEMBL3706478 0.065 0.02 CHEMBL1222314 | CHEMBL3706466 | |
| 0.091 | 0.115 | 0.528 | Alpha-N-acetylglucosaminidase inhibitor | 0.476 0.006 CHEMBL3706465 0.374 0.01 CHEMBL3706466 0.528 0.005 CHEMBL3706475 0.404 0.009 CHEMBL3706478 0.506 0.005 CHEMBL1222314 | CHEMBL3706475 | |
| 0.125 | 0.151 | 0.145 | Lipocortins synthesis antagonist | 0.145 0.113 CHEMBL3706465 0.138 0.125 CHEMBL3706466 | CHEMBL3706465 | |
| 0.049 | 0.077 | 0.064 | Lipocortins synthesis agonist | 0.06 0.035 CHEMBL3706465 0.059 0.039 CHEMBL3706479 0.064 0.029 CHEMBL3706475 | CHEMBL3706475 | |
| 0.034 | 0.068 | 0.07 | Protein 50S ribosomal subunit inhibitor | 0.07 0.024 CHEMBL3706465 0.064 0.028 CHEMBL3706475 | CHEMBL3706465 | |
| 0.039 | 0.078 | 0.108 | Nicotinic receptor alpha7 subunit antagonist | 0.108 0.011 CHEMBL3706465 0.09 0.014 CHEMBL3706474 | CHEMBL3706465 | |
| 0.113 | 0.153 | 0.204 | Interferon gamma antagonist | 0.204 0.039 CHEMBL3706465 0.15 0.077 CHEMBL3706466 0.184 0.048 CHEMBL3706475 0.157 0.07 CHEMBL3706478 0.184 0.048 CHEMBL1222314 | CHEMBL3706465 | |
| 0.015 | 0.057 | 0.036 | Bradykinin B2 receptor agonist | 0.036 0.014 CHEMBL3706466 0.027 0.022 CHEMBL3706471 0.034 0.015 CHEMBL3706478 0.034 0.015 CHEMBL1222314 | CHEMBL3706466 | |
| 0.059 | 0.102 | 0.29 | Antiadrenergic | 0.29 0.014 CHEMBL3706466 | CHEMBL3706466 | |
| 0.01 | 0.055 | 0.017 | Adenosine A3 receptor agonist | 0.017 0.012 CHEMBL3706465 | CHEMBL3706465 | |
| 0.072 | 0.117 | 0.144 | Anabolic | 0.142 0.023 CHEMBL3706465 0.109 0.051 CHEMBL3706466 0.144 0.021 CHEMBL3706475 0.123 0.036 CHEMBL3706478 0.117 0.043 CHEMBL1222314 | CHEMBL3706475 | |
| 0.111 | 0.157 | 0.213 | Platelet adhesion inhibitor | 0.213 0.064 CHEMBL3706465 0.148 0.108 CHEMBL3706474 | CHEMBL3706465 | |
| 0.076 | 0.122 | 0.139 | Alpha 2d adrenoreceptor antagonist | 0.122 0.022 CHEMBL3706466 0.091 0.068 CHEMBL3706474 0.099 0.049 CHEMBL3706475 0.125 0.019 CHEMBL3706478 0.139 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.054 | 0.105 | 0.29 | Adrenaline antagonist | 0.29 0.014 CHEMBL3706466 | CHEMBL3706466 | |
| 0.01 | 0.062 | 0.035 | RNA-directed RNA polymerase stimulant | 0.035 0.018 CHEMBL3706465 0.032 0.02 CHEMBL3706475 | CHEMBL3706465 | |
| 0.107 | 0.161 | 0.499 | Psychostimulant | 0.499 0.011 CHEMBL3706465 0.134 0.132 CHEMBL3706474 | CHEMBL3706465 | |
| 0.022 | 0.078 | 0.059 | Opioid kappa receptor agonist | 0.059 0.019 CHEMBL3706465 | CHEMBL3706465 | |
| 0.004 | 0.062 | 0.01 | Calcineurin inhibitor | 0.01 0.009 CHEMBL3706465 | CHEMBL3706465 | |
| 0.052 | 0.113 | 0.161 | Glycine receptor agonist | 0.161 0.005 CHEMBL3706465 0.069 0.057 CHEMBL3706466 0.089 0.029 CHEMBL3706475 0.079 0.04 CHEMBL1222314 | CHEMBL3706465 | |
| 0.099 | 0.162 | 0.213 | Arachidonic acid antagonist | 0.209 0.025 CHEMBL3706465 0.2 0.033 CHEMBL3706466 0.213 0.022 CHEMBL3706475 0.19 0.043 CHEMBL3706478 0.195 0.038 CHEMBL1222314 | CHEMBL3706475 | |
| 0.054 | 0.119 | 0.126 | Glycine receptor antagonist | 0.126 0.015 CHEMBL3706465 0.079 0.058 CHEMBL3706466 0.116 0.02 CHEMBL3706475 0.098 0.034 CHEMBL1222314 | CHEMBL3706465 | |
| 0.04 | 0.108 | 0.12 | Beta adrenoreceptor antagonist | 0.12 0.01 CHEMBL3706466 0.062 0.051 CHEMBL3706475 0.099 0.017 CHEMBL3706478 0.07 0.038 CHEMBL1222314 | CHEMBL3706466 | |
| 0.008 | 0.077 | 0.021 | Telomerase stimulant | 0.019 0.008 CHEMBL3706465 0.021 0.006 CHEMBL3706475 | CHEMBL3706475 | |
| 0.012 | 0.082 | 0.186 | Prostaglandin agonist | 0.049 0.01 CHEMBL3706466 0.038 0.015 CHEMBL3706475 0.173 0.004 CHEMBL3706478 0.186 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.03 | 0.105 | 0.096 | Glucose-6-phosphate isomerase inhibitor | 0.072 0.011 CHEMBL3706465 0.082 0.008 CHEMBL3706466 0.096 0.005 CHEMBL3706475 0.08 0.009 CHEMBL3706478 0.072 0.011 CHEMBL1222314 | CHEMBL3706475 | |
| 0.034 | 0.111 | 0.135 | Antineoplastic antibiotic | 0.135 0.034 CHEMBL3706465 0.088 0.052 CHEMBL3706479 | CHEMBL3706465 | |
| 0.032 | 0.11 | 0.096 | Squalene epoxidase inhibitor | 0.066 0.016 CHEMBL3706466 0.075 0.012 CHEMBL3706475 0.058 0.023 CHEMBL3706478 0.096 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.03 | 0.112 | 0.093 | Acetylcholine M5 receptor agonist | 0.093 0.024 CHEMBL3706465 0.08 0.034 CHEMBL3706474 0.063 0.051 CHEMBL3706475 | CHEMBL3706465 | |
| 0.099 | 0.181 | 0.149 | Nitric oxide antagonist | 0.149 0.096 CHEMBL3706465 | CHEMBL3706465 | |
| 0.005 | 0.088 | 0.013 | Purine nucleoside phosphorylase inhibitor | 0.011 0.01 CHEMBL3706466 0.012 0.007 CHEMBL3706475 0.011 0.009 CHEMBL3706478 0.013 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.096 | 0.034 | Prostaglandin F2 alpha agonist | 0.023 0.015 CHEMBL3706465 0.025 0.012 CHEMBL3706475 0.034 0.007 CHEMBL3706478 0.029 0.009 CHEMBL1222314 | CHEMBL3706478 | |
| 0.041 | 0.13 | 0.083 | Analgesic, opioid | 0.083 0.044 CHEMBL3706465 | CHEMBL3706465 | |
| 0.021 | 0.111 | 0.046 | Antibiotic Aminoglycoside-like | 0.037 0.024 CHEMBL3706465 0.046 0.016 CHEMBL3706475 | CHEMBL3706475 | |
| 0.111 | 0.201 | 0.525 | Immunostimulant | 0.35 0.064 CHEMBL3706465 0.448 0.037 CHEMBL3706471 0.525 0.026 CHEMBL3706472 0.248 0.097 CHEMBL3706475 | CHEMBL3706472 | |
| 0.03 | 0.12 | 0.169 | Phosphofructokinase-1 inhibitor | 0.147 0.019 CHEMBL3706465 0.156 0.017 CHEMBL3706466 0.169 0.015 CHEMBL3706475 0.141 0.02 CHEMBL3706478 0.16 0.016 CHEMBL1222314 | CHEMBL3706475 | |
| 0.009 | 0.1 | 0.079 | Sodium/glucose cotransporter 2 inhibitor | 0.029 0.014 CHEMBL3706465 0.079 0.004 CHEMBL3706475 0.025 0.021 CHEMBL3706478 0.027 0.017 CHEMBL1222314 | CHEMBL3706475 | |
| 0.128 | 0.219 | 0.314 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.169 0.109 CHEMBL3706465 0.261 0.038 CHEMBL3706466 0.297 0.024 CHEMBL3706475 0.278 0.031 CHEMBL3706478 0.314 0.02 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.095 | 0.13 | Prostaglandin EP4 agonist | 0.027 0.008 CHEMBL3706466 0.091 0.004 CHEMBL3706478 0.13 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.019 | 0.113 | 0.076 | Membrane dipeptidase inhibitor | 0.059 0.011 CHEMBL3706466 0.036 0.033 CHEMBL3706475 0.076 0.006 CHEMBL3706478 0.065 0.008 CHEMBL1222314 | CHEMBL3706478 | |
| 0.058 | 0.152 | 0.144 | Anesthetic local | 0.144 0.052 CHEMBL3706465 | CHEMBL3706465 | |
| 0.013 | 0.108 | 0.061 | Dopamine D5 antagonist | 0.061 0.019 CHEMBL3706465 | CHEMBL3706465 | |
| 0.061 | 0.157 | 0.146 | Adenylate cyclase inhibitor | 0.146 0.048 CHEMBL3706465 0.113 0.073 CHEMBL3706466 0.12 0.067 CHEMBL3706475 0.142 0.05 CHEMBL3706478 0.134 0.057 CHEMBL1222314 | CHEMBL3706465 | |
| 0.049 | 0.147 | 0.126 | Opioid kappa receptor antagonist | 0.126 0.022 CHEMBL3706465 | CHEMBL3706465 | |
| 0.035 | 0.135 | 0.105 | Na+ K+ transporting ATPase inhibitor | 0.105 0.027 CHEMBL3706465 0.067 0.063 CHEMBL3706466 0.101 0.03 CHEMBL3706475 0.083 0.048 CHEMBL3706478 0.07 0.06 CHEMBL1222314 | CHEMBL3706465 | |
| 0.005 | 0.106 | 0.163 | Prostaglandin E2 agonist | 0.035 0.009 CHEMBL3706466 0.026 0.013 CHEMBL3706475 0.145 0.003 CHEMBL3706478 0.163 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.034 | 0.137 | 0.102 | Glucosylceramidase inhibitor | 0.08 0.015 CHEMBL3706465 0.102 0.008 CHEMBL3706475 0.068 0.023 CHEMBL3706478 0.073 0.02 CHEMBL1222314 | CHEMBL3706475 | |
| 0.087 | 0.191 | 0.189 | DNA repair enzyme inhibitor | 0.132 0.052 CHEMBL3706466 0.134 0.049 CHEMBL3706474 0.123 0.066 CHEMBL3706475 0.136 0.047 CHEMBL3706478 0.189 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.026 | 0.13 | 0.055 | Integrin alpha1beta1 antagonist | 0.055 0.005 CHEMBL3706466 0.052 0.006 CHEMBL3706478 0.053 0.006 CHEMBL1222314 | CHEMBL3706466 | |
| 0.003 | 0.112 | 0.02 | Glutamate (mGluR6) agonist | 0.013 0.007 CHEMBL3706466 0.012 0.009 CHEMBL3706475 0.013 0.008 CHEMBL3706478 0.02 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.118 | 0.025 | Adenosine kinase inhibitor | 0.025 0.013 CHEMBL3706465 | CHEMBL3706465 | |
| 0.024 | 0.139 | 0.074 | 5 Hydroxytryptamine 3 antagonist | 0.074 0.027 CHEMBL3706465 0.053 0.045 CHEMBL3706474 | CHEMBL3706465 | |
| 0.028 | 0.145 | 0.187 | Neuronal nicotinic receptor antagonist | 0.187 0.009 CHEMBL3706465 0.089 0.029 CHEMBL3706474 | CHEMBL3706465 | |
| 0.005 | 0.127 | 0.013 | Integrin alphaLbeta2 antagonist | 0.013 0.009 CHEMBL1222314 | CHEMBL1222314 | |
| 0.024 | 0.147 | 0.147 | Carbamoyl phosphate synthetase inhibitor | 0.115 0.017 CHEMBL3706465 0.127 0.014 CHEMBL3706466 0.147 0.012 CHEMBL3706475 0.115 0.017 CHEMBL3706478 0.099 0.021 CHEMBL1222314 | CHEMBL3706475 | |
| 0 | 0.123 | 0.004 | Human herpesvirus 2 protease inhibitor | 0.004 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.133 | 0.082 | LFA antagonist | 0.026 0.023 CHEMBL3706466 0.028 0.019 CHEMBL3706478 0.082 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.133 | 0.274 | Prostaglandin D2 agonist | 0.031 0.021 CHEMBL3706466 0.054 0.006 CHEMBL3706478 0.274 0.002 CHEMBL1222314 | CHEMBL1222314 | |
| 0.024 | 0.152 | 0.33 | Glucagon-like peptide 1 receptor antagonist | 0.088 0.005 CHEMBL3706466 0.093 0.005 CHEMBL3706478 0.33 0.002 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.133 | 0.075 | Prostaglandin EP2 agonist | 0.023 0.015 CHEMBL3706466 0.02 0.018 CHEMBL3706475 0.066 0.004 CHEMBL3706478 0.075 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.039 | 0.168 | 0.166 | Glutamate dehydrogenase inhibitor | 0.1 0.031 CHEMBL3706465 0.141 0.017 CHEMBL3706466 0.141 0.017 CHEMBL3706475 0.128 0.02 CHEMBL3706478 0.166 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.092 | 0.223 | 0.157 | P-glycoprotein inhibitor | 0.146 0.124 CHEMBL3706465 0.157 0.106 CHEMBL3706479 | CHEMBL3706479 | |
| 0.073 | 0.206 | 0.196 | Protein kinase stimulant | 0.196 0.043 CHEMBL3706465 0.111 0.104 CHEMBL3706475 | CHEMBL3706465 | |
| 0.051 | 0.186 | 0.134 | Cholesterol synthesis inhibitor | 0.119 0.066 CHEMBL3706465 0.122 0.063 CHEMBL3706466 0.129 0.057 CHEMBL3706475 0.134 0.054 CHEMBL3706478 0.111 0.074 CHEMBL1222314 | CHEMBL3706478 | |
| 0.006 | 0.143 | 0.017 | Purinergic P2Y1 agonist | 0.017 0.008 CHEMBL3706465 0.017 0.009 CHEMBL3706475 | CHEMBL3706475 | |
| 0.02 | 0.158 | 0.075 | Glutamate (mGluR8) agonist | 0.036 0.031 CHEMBL3706465 0.057 0.008 CHEMBL3706466 0.047 0.014 CHEMBL3706475 0.055 0.009 CHEMBL3706478 0.075 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.06 | 0.198 | 0.094 | Toll-Like receptor 4 antagonist | 0.094 0.081 CHEMBL3706465 0.09 0.088 CHEMBL3706472 | CHEMBL3706465 | |
| 0.022 | 0.163 | 0.358 | Carnitine palmitoyltransferase 1B inhibitor | 0.048 0.032 CHEMBL3706466 0.358 0.002 CHEMBL3706474 0.062 0.016 CHEMBL1222314 | CHEMBL3706474 | |
| 0.023 | 0.164 | 0.062 | Kainate receptor agonist | 0.045 0.021 CHEMBL3706465 0.056 0.009 CHEMBL3706466 0.052 0.012 CHEMBL3706475 0.051 0.012 CHEMBL3706478 0.062 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.135 | 0.276 | 0.361 | Antithrombotic | 0.277 0.105 CHEMBL3706465 0.209 0.166 CHEMBL3706466 0.253 0.124 CHEMBL3706471 0.297 0.09 CHEMBL3706472 0.202 0.175 CHEMBL3706474 0.32 0.076 CHEMBL3706475 0.282 0.101 CHEMBL3706478 0.361 0.061 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.167 | 0.045 | HCV polyprotein inhibitor | 0.045 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.041 | 0.192 | 0.111 | Glutamate (mGluR6) antagonist | 0.074 0.032 CHEMBL3706465 0.095 0.013 CHEMBL3706466 0.086 0.018 CHEMBL3706475 0.096 0.012 CHEMBL3706478 0.111 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.078 | 0.229 | 0.345 | Anesthetic general | 0.286 0.037 CHEMBL3706465 0.296 0.034 CHEMBL3706466 0.245 0.052 CHEMBL3706475 0.332 0.027 CHEMBL3706478 0.345 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.117 | 0.272 | 0.273 | Transcription factor NF kappa B inhibitor | 0.223 0.148 CHEMBL3706465 0.24 0.135 CHEMBL3706466 0.199 0.17 CHEMBL3706475 0.229 0.143 CHEMBL3706478 0.273 0.111 CHEMBL1222314 | CHEMBL1222314 | |
| 0.185 | 0.344 | 0.652 | Caspase 9 stimulant | 0.652 0.029 CHEMBL3706465 0.35 0.146 CHEMBL3706475 0.261 0.239 CHEMBL3706478 | CHEMBL3706465 | |
| 0.003 | 0.162 | 0.021 | Integrin beta2 antagonist | 0.021 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.039 | 0.2 | 0.111 | Exportin-1 inhibitor | 0.091 0.014 CHEMBL3706466 0.081 0.024 CHEMBL3706475 0.111 0.005 CHEMBL3706478 0.099 0.009 CHEMBL1222314 | CHEMBL3706478 | |
| 0.004 | 0.166 | 0.026 | Estrogen receptor beta agonist | 0.026 0.025 CHEMBL3706465 | CHEMBL3706465 | |
| 0.023 | 0.186 | 0.099 | Androgen agonist | 0.099 0.015 CHEMBL3706465 | CHEMBL3706465 | |
| 0.009 | 0.172 | 0.059 | Fumarate hydratase inhibitor | 0.033 0.025 CHEMBL3706465 0.057 0.011 CHEMBL3706466 0.059 0.011 CHEMBL3706475 0.05 0.013 CHEMBL3706478 0.059 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.167 | 0.025 | Ileal bile acid transport inhibitor | 0.025 0.006 CHEMBL3706478 | CHEMBL3706478 | |
| 0.002 | 0.166 | 0.022 | Thromboxane agonist | 0.01 0.008 CHEMBL3706475 0.014 0.005 CHEMBL3706478 0.022 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.175 | 0.059 | Sodium/glucose cotransporter inhibitor | 0.026 0.018 CHEMBL3706465 0.059 0.004 CHEMBL3706475 | CHEMBL3706475 | |
| 0.02 | 0.188 | 0.094 | Alpha-mannosidase inhibitor | 0.094 0.007 CHEMBL3706465 0.087 0.009 CHEMBL3706475 0.059 0.028 CHEMBL3706478 | CHEMBL3706465 | |
| 0.021 | 0.191 | 0.151 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.075 0.004 CHEMBL3706466 0.056 0.01 CHEMBL3706475 0.069 0.005 CHEMBL3706478 0.151 0.002 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.179 | 0.033 | HMG CoA reductase inhibitor | 0.033 0.026 CHEMBL3706465 | CHEMBL3706465 | |
| 0.008 | 0.181 | 0.056 | Estradiol 17 beta-dehydrogenase 2 inhibitor | 0.046 0.018 CHEMBL3706478 0.056 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.061 | 0.235 | 0.336 | Angiogenesis stimulant | 0.227 0.081 CHEMBL3706465 0.304 0.048 CHEMBL3706471 0.336 0.037 CHEMBL3706472 | CHEMBL3706472 | |
| 0.05 | 0.224 | 0.333 | Electrolyte absorption antagonist | 0.223 0.006 CHEMBL3706466 0.119 0.037 CHEMBL3706475 0.212 0.007 CHEMBL3706478 0.333 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.184 | 0.028 | Vanilloid 2 agonist | 0.028 0.013 CHEMBL3706465 0.027 0.014 CHEMBL3706475 0.026 0.017 CHEMBL1222314 | CHEMBL3706465 | |
| 0.122 | 0.299 | 0.333 | Peptidyltransferase inhibitor | 0.28 0.033 CHEMBL3706465 0.167 0.152 CHEMBL3706467 0.252 0.049 CHEMBL3706471 0.195 0.106 CHEMBL3706468 0.282 0.032 CHEMBL3706472 0.333 0.015 CHEMBL3706475 0.259 0.045 CHEMBL3706478 | CHEMBL3706475 | |
| 0.045 | 0.223 | 0.23 | Triose-phosphate isomerase inhibitor | 0.12 0.032 CHEMBL3706465 0.191 0.012 CHEMBL3706466 0.19 0.012 CHEMBL3706475 0.199 0.011 CHEMBL3706478 0.23 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.189 | 0.108 | Nicotinic acid receptor 2 antagonist | 0.049 0.004 CHEMBL3706466 0.044 0.004 CHEMBL3706478 0.108 0.002 CHEMBL1222314 | CHEMBL1222314 | |
| 0.062 | 0.244 | 0.209 | Cholinergic | 0.209 0.042 CHEMBL3706465 | CHEMBL3706465 | |
| 0.009 | 0.194 | 0.037 | Retinoid X gamma receptor antagonist | 0.028 0.016 CHEMBL3706466 0.026 0.022 CHEMBL3706478 0.037 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.191 | 0.026 | Isoleucine-tRNA ligase inhibitor | 0.026 0.009 CHEMBL3706475 0.021 0.019 CHEMBL1222314 | CHEMBL3706475 | |
| 0.076 | 0.261 | 0.269 | Growth hormone agonist | 0.212 0.054 CHEMBL3706471 0.269 0.039 CHEMBL3706472 | CHEMBL3706472 | |
| 0.003 | 0.188 | 0.014 | Adenosine A2a receptor agonist | 0.014 0.012 CHEMBL3706475 | CHEMBL3706475 | |
| 0.01 | 0.199 | 0.036 | Nicotinic receptor beta4 subunit antagonist | 0.036 0.028 CHEMBL3706465 | CHEMBL3706465 | |
| 0.058 | 0.248 | 0.126 | Acetylcholine release stimulant | 0.115 0.056 CHEMBL3706474 0.103 0.081 CHEMBL3706478 0.126 0.04 CHEMBL1222314 | CHEMBL1222314 | |
| 0.078 | 0.268 | 0.186 | Adenylate cyclase stimulant | 0.163 0.043 CHEMBL3706465 0.156 0.054 CHEMBL3706466 0.186 0.021 CHEMBL3706475 0.173 0.032 CHEMBL3706478 0.144 0.074 CHEMBL1222314 | CHEMBL3706475 | |
| 0.004 | 0.195 | 0.016 | Adenosine A2 receptor agonist | 0.016 0.012 CHEMBL3706475 | CHEMBL3706475 | |
| 0.034 | 0.228 | 0.087 | Opioid antagonist | 0.087 0.06 CHEMBL3706465 | CHEMBL3706465 | |
| 0.116 | 0.31 | 0.389 | Vasodilator, peripheral | 0.239 0.136 CHEMBL3706465 0.23 0.144 CHEMBL3706466 0.233 0.141 CHEMBL3706474 0.249 0.127 CHEMBL3706475 0.389 0.059 CHEMBL3706478 0.326 0.085 CHEMBL1222314 | CHEMBL3706478 | |
| 0.007 | 0.203 | 0.047 | Acetylcholine M1 receptor agonist | 0.047 0.027 CHEMBL3706465 | CHEMBL3706465 | |
| 0.008 | 0.204 | 0.04 | Carnitine palmitoyltransferase inhibitor | 0.04 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.206 | 0.041 | Retinoid X beta receptor antagonist | 0.027 0.006 CHEMBL3706466 0.024 0.008 CHEMBL3706478 0.041 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.205 | 0.025 | Antibiotic Anthracycline-like | 0.022 0.008 CHEMBL3706465 0.025 0.005 CHEMBL3706475 | CHEMBL3706475 | |
| 0.005 | 0.205 | 0.031 | Acetylcholine M4 receptor agonist | 0.031 0.021 CHEMBL3706465 | CHEMBL3706465 | |
| 0.012 | 0.213 | 0.051 | Collagenase inhibitor | 0.051 0.03 CHEMBL3706466 | CHEMBL3706466 | |
| 0.003 | 0.204 | 0.022 | Carbonic anhydrase VIII inhibitor | 0.017 0.012 CHEMBL3706466 0.016 0.013 CHEMBL3706478 0.022 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.204 | 0.022 | Carbonic anhydrase X inhibitor | 0.017 0.012 CHEMBL3706466 0.016 0.013 CHEMBL3706478 0.022 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.069 | 0.271 | 0.197 | Antimitotic | 0.197 0.086 CHEMBL3706465 0.146 0.125 CHEMBL3706474 | CHEMBL3706465 | |
| 0.025 | 0.227 | 0.078 | Androgen antagonist | 0.078 0.067 CHEMBL3706465 | CHEMBL3706465 | |
| 0.009 | 0.215 | 0.07 | Guanylate cyclase inhibitor | 0.046 0.025 CHEMBL3706465 0.044 0.028 CHEMBL3706466 0.066 0.007 CHEMBL3706475 0.045 0.026 CHEMBL3706478 0.07 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.229 | 0.117 | Nicotinic alpha4beta2 receptor antagonist | 0.117 0.019 CHEMBL3706465 0.087 0.043 CHEMBL3706474 | CHEMBL3706465 | |
| 0.129 | 0.337 | 0.425 | Antibacterial | 0.347 0.104 CHEMBL3706465 0.274 0.155 CHEMBL3706475 0.389 0.082 CHEMBL3706478 0.425 0.066 CHEMBL1222314 | CHEMBL1222314 | |
| 0.039 | 0.248 | 0.253 | UDP-glucose 4-epimerase inhibitor | 0.18 0.021 CHEMBL3706465 0.106 0.054 CHEMBL3706466 0.253 0.013 CHEMBL3706475 0.114 0.047 CHEMBL3706478 0.204 0.018 CHEMBL1222314 | CHEMBL3706475 | |
| 0.013 | 0.222 | 0.078 | Mannosidase inhibitor | 0.078 0.009 CHEMBL3706465 0.077 0.009 CHEMBL3706475 0.049 0.027 CHEMBL3706478 | CHEMBL3706465 | |
| 0.005 | 0.215 | 0.132 | Retinoid X gamma receptor agonist | 0.021 0.019 CHEMBL3706466 0.132 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.019 | 0.23 | 0.131 | Aconitate hydratase inhibitor | 0.104 0.008 CHEMBL3706466 0.066 0.021 CHEMBL3706475 0.093 0.01 CHEMBL3706478 0.131 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.217 | 0.154 | Retinoid X beta receptor agonist | 0.154 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.227 | 0.107 | Argininosuccinate synthase inhibitor | 0.069 0.031 CHEMBL3706465 0.09 0.022 CHEMBL3706466 0.097 0.02 CHEMBL3706475 0.077 0.027 CHEMBL3706478 0.107 0.018 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.234 | 0.131 | Dopamine beta hydroxylase inhibitor | 0.082 0.005 CHEMBL3706466 0.059 0.017 CHEMBL3706475 0.085 0.005 CHEMBL3706478 0.131 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.22 | 0.1 | HCV NS5B polymerase inhibitor | 0.1 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.221 | 0.158 | Carnitine palmitoyltransferase 1A inhibitor | 0.158 0.003 CHEMBL3706474 | CHEMBL3706474 | |
| 0.047 | 0.267 | 0.078 | Thioredoxin reductase inhibitor | 0.078 0.068 CHEMBL3706478 | CHEMBL3706478 | |
| 0.037 | 0.257 | 0.432 | GABA C receptor agonist | 0.148 0.035 CHEMBL3706465 0.307 0.009 CHEMBL3706466 0.225 0.016 CHEMBL3706475 0.27 0.012 CHEMBL3706478 0.432 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.23 | 0.1 | GABA uptake inhibitor | 0.067 0.008 CHEMBL3706466 0.049 0.016 CHEMBL3706478 0.1 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.225 | 0.01 | Purinergic P2Y2 agonist | 0.01 0.008 CHEMBL3706475 | CHEMBL3706475 | |
| 0.007 | 0.23 | 0.036 | Carnitine palmitoyltransferase 1 inhibitor | 0.036 0.02 CHEMBL1222314 | CHEMBL1222314 | |
| 0.085 | 0.309 | 0.19 | ATPase inhibitor | 0.19 0.046 CHEMBL3706465 0.153 0.096 CHEMBL3706466 0.151 0.1 CHEMBL3706475 0.175 0.063 CHEMBL3706478 0.156 0.091 CHEMBL1222314 | CHEMBL3706465 | |
| 0.16 | 0.384 | 0.688 | 5 Hydroxytryptamine release inhibitor | 0.558 0.018 CHEMBL3706466 0.426 0.063 CHEMBL3706475 0.626 0.008 CHEMBL3706478 0.688 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.237 | 0.045 | Macrophage elastase inhibitor | 0.045 0.029 CHEMBL3706478 | CHEMBL3706478 | |
| 0.009 | 0.237 | 0.162 | Carbonic anhydrase VB inhibitor | 0.084 0.021 CHEMBL3706466 0.093 0.018 CHEMBL3706478 0.162 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.246 | 0.158 | NMDA receptor glycine site agonist | 0.13 0.006 CHEMBL3706466 0.111 0.012 CHEMBL3706478 0.158 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.051 | 0.284 | 0.186 | Hematopoietic | 0.086 0.058 CHEMBL3706466 0.096 0.041 CHEMBL3706471 0.087 0.056 CHEMBL3706472 0.089 0.052 CHEMBL3706478 0.186 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.098 | 0.331 | 0.313 | DNA synthesis inhibitor | 0.313 0.039 CHEMBL3706465 0.199 0.125 CHEMBL3706466 0.291 0.047 CHEMBL3706475 0.192 0.135 CHEMBL3706478 0.222 0.092 CHEMBL1222314 | CHEMBL3706465 | |
| 0.053 | 0.289 | 0.158 | Glutamate release inhibitor | 0.088 0.067 CHEMBL3706465 0.11 0.03 CHEMBL3706466 0.112 0.028 CHEMBL3706475 0.131 0.016 CHEMBL3706478 0.158 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.24 | 0.074 | Retinoic acid beta receptor antagonist | 0.074 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.029 | 0.267 | 0.173 | Ornithine decarboxylase inhibitor | 0.104 0.04 CHEMBL3706466 0.078 0.07 CHEMBL3706475 0.123 0.024 CHEMBL3706478 0.173 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.071 | 0.31 | 0.124 | Vanilloid 1 agonist | 0.124 0.078 CHEMBL3706466 0.113 0.107 CHEMBL3706475 0.112 0.108 CHEMBL3706478 0.118 0.091 CHEMBL1222314 | CHEMBL3706466 | |
| 0.039 | 0.28 | 0.206 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.114 0.042 CHEMBL3706465 0.132 0.033 CHEMBL3706466 0.163 0.023 CHEMBL3706475 0.137 0.031 CHEMBL3706478 0.206 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.065 | 0.309 | 0.539 | Platelet antagonist | 0.201 0.1 CHEMBL3706465 0.402 0.027 CHEMBL3706471 0.248 0.073 CHEMBL3706468 0.439 0.021 CHEMBL3706472 0.539 0.01 CHEMBL3706475 | CHEMBL3706475 | |
| 0.013 | 0.258 | 0.052 | Nicotinic receptor alpha3 subunit antagonist | 0.052 0.023 CHEMBL3706465 | CHEMBL3706465 | |
| 0.126 | 0.371 | 0.351 | Interleukin 2 agonist | 0.351 0.045 CHEMBL3706465 0.234 0.137 CHEMBL3706471 0.275 0.093 CHEMBL3706472 0.197 0.194 CHEMBL3706475 0.3 0.074 CHEMBL3706478 | CHEMBL3706465 | |
| 0.003 | 0.249 | 0.029 | Prostaglandin H2 antagonist | 0.027 0.016 CHEMBL3706466 0.029 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.034 | 0.28 | 0.154 | Cystathionine beta-synthase inhibitor | 0.136 0.047 CHEMBL3706465 0.12 0.058 CHEMBL3706466 0.143 0.044 CHEMBL3706475 0.121 0.058 CHEMBL3706478 0.154 0.039 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.264 | 0.084 | Adenylate cyclase 1 inhibitor | 0.084 0.007 CHEMBL3706475 0.043 0.037 CHEMBL1222314 | CHEMBL3706475 | |
| 0.007 | 0.258 | 0.186 | Retinoic acid beta receptor agonist | 0.186 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.257 | 0.077 | Retinoic acid alpha receptor antagonist | 0.077 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.265 | 0.142 | Acyl-CoA dehydrogenase inhibitor | 0.073 0.025 CHEMBL3706465 0.081 0.022 CHEMBL3706466 0.142 0.01 CHEMBL3706475 0.085 0.02 CHEMBL3706478 0.13 0.011 CHEMBL1222314 | CHEMBL3706475 | |
| 0.003 | 0.258 | 0.016 | Thromboxane A2 agonist | 0.015 0.012 CHEMBL3706465 0.016 0.009 CHEMBL3706475 | CHEMBL3706475 | |
| 0.04 | 0.295 | 0.189 | NADH dehydrogenase inhibitor | 0.133 0.023 CHEMBL3706465 0.125 0.026 CHEMBL3706466 0.189 0.011 CHEMBL3706475 0.132 0.023 CHEMBL3706478 0.175 0.013 CHEMBL1222314 | CHEMBL3706475 | |
| 0.008 | 0.264 | 0.077 | Ornithine carbamoyltransferase inhibitor | 0.06 0.031 CHEMBL3706466 0.067 0.027 CHEMBL3706475 0.062 0.03 CHEMBL3706478 0.077 0.023 CHEMBL1222314 | CHEMBL1222314 | |
| 0.046 | 0.304 | 0.34 | Pyruvate kinase inhibitor | 0.223 0.07 CHEMBL3706466 0.145 0.12 CHEMBL3706474 0.241 0.064 CHEMBL3706478 0.34 0.037 CHEMBL1222314 | CHEMBL1222314 | |
| 0.115 | 0.374 | 0.232 | Apoptosis antagonist | 0.232 0.146 CHEMBL3706465 0.194 0.188 CHEMBL3706471 0.201 0.178 CHEMBL3706472 | CHEMBL3706465 | |
| 0.008 | 0.267 | 0.031 | Protein 30S ribosomal subunit inhibitor | 0.031 0.012 CHEMBL3706475 | CHEMBL3706475 | |
| 0.025 | 0.286 | 0.081 | Factor III inhibitor | 0.081 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.107 | 0.368 | 0.383 | Sodium/bile acid cotransporter inhibitor | 0.311 0.069 CHEMBL3706465 0.359 0.035 CHEMBL3706471 0.383 0.023 CHEMBL3706472 0.275 0.103 CHEMBL3706478 | CHEMBL3706472 | |
| 0.021 | 0.283 | 0.178 | NMDA receptor agonist | 0.131 0.011 CHEMBL3706466 0.127 0.012 CHEMBL3706478 0.178 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.273 | 0.033 | Carboxypeptidase B inhibitor | 0.033 0.022 CHEMBL3706478 0.031 0.026 CHEMBL1222314 | CHEMBL3706478 | |
| 0.006 | 0.269 | 0.111 | Retinoic acid receptor agonist | 0.111 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.032 | 0.295 | 0.184 | Alkylator | 0.184 0.031 CHEMBL3706465 | CHEMBL3706465 | |
| 0.021 | 0.284 | 0.154 | Carbonic anhydrase XIII inhibitor | 0.088 0.045 CHEMBL3706466 0.105 0.036 CHEMBL3706478 0.154 0.021 CHEMBL1222314 | CHEMBL1222314 | |
| 0.031 | 0.296 | 0.063 | Caspase 9 inhibitor | 0.062 0.042 CHEMBL3706466 0.063 0.042 CHEMBL1222314 | CHEMBL1222314 | |
| 0.116 | 0.381 | 0.288 | Tyrosine 3 hydroxylase inhibitor | 0.25 0.068 CHEMBL3706465 0.288 0.039 CHEMBL3706466 0.24 0.079 CHEMBL3706475 0.247 0.071 CHEMBL3706478 0.257 0.061 CHEMBL1222314 | CHEMBL3706466 | |
| 0.02 | 0.286 | 0.122 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.081 0.05 CHEMBL3706466 0.07 0.061 CHEMBL3706475 0.073 0.058 CHEMBL3706478 0.122 0.028 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.276 | 0.023 | Methylmalonyl-CoA mutase inhibitor | 0.023 0.005 CHEMBL3706475 0.017 0.016 CHEMBL3706478 0.019 0.01 CHEMBL1222314 | CHEMBL3706475 | |
| 0.021 | 0.289 | 0.092 | Topoisomerase II beta inhibitor | 0.051 0.031 CHEMBL3706466 0.057 0.025 CHEMBL3706478 0.092 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.025 | 0.294 | 0.29 | Macrophage migration inhibitory factor inhibitor | 0.14 0.018 CHEMBL3706466 0.076 0.057 CHEMBL3706475 0.14 0.018 CHEMBL3706478 0.29 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.069 | 0.339 | 0.138 | Pregnane X receptor agonist | 0.135 0.086 CHEMBL3706465 0.138 0.079 CHEMBL3706466 0.13 0.099 CHEMBL3706475 0.135 0.087 CHEMBL3706478 0.126 0.113 CHEMBL1222314 | CHEMBL3706466 | |
| 0.02 | 0.29 | 0.076 | Acetylcholine nicotinic agonist | 0.076 0.063 CHEMBL3706465 | CHEMBL3706465 | |
| 0.004 | 0.282 | 0.071 | Retinoic acid receptor antagonist | 0.071 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.283 | 0.104 | Retinoid X receptor agonist | 0.045 0.02 CHEMBL3706466 0.036 0.024 CHEMBL3706478 0.104 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.054 | 0.332 | 0.133 | Folate antagonist | 0.133 0.03 CHEMBL3706466 0.1 0.065 CHEMBL3706471 0.116 0.042 CHEMBL3706478 0.129 0.032 CHEMBL1222314 | CHEMBL3706466 | |
| 0.003 | 0.282 | 0.064 | Retinoic acid receptor gamma antagonist | 0.064 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.016 | 0.298 | 0.104 | Leukotriene synthesis inhibitor | 0.066 0.048 CHEMBL3706466 0.078 0.039 CHEMBL3706478 0.104 0.024 CHEMBL1222314 | CHEMBL1222314 | |
| 0.048 | 0.332 | 0.218 | Adenylate kinase inhibitor | 0.124 0.04 CHEMBL3706465 0.164 0.022 CHEMBL3706466 0.215 0.013 CHEMBL3706475 0.198 0.015 CHEMBL3706478 0.218 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.299 | 0.037 | Glutamate (mGluR3) agonist | 0.037 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.301 | 0.065 | Retinoid X alpha receptor antagonist | 0.042 0.013 CHEMBL3706466 0.037 0.019 CHEMBL3706478 0.065 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.016 | 0.305 | 0.057 | Angiotensin-converting enzyme inhibitor | 0.054 0.039 CHEMBL3706471 0.057 0.035 CHEMBL3706472 | CHEMBL3706472 | |
| 0.016 | 0.306 | 0.137 | Carbonic anhydrase VA inhibitor | 0.089 0.031 CHEMBL3706466 0.094 0.028 CHEMBL3706478 0.137 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.035 | 0.331 | 0.091 | Vanilloid 4 agonist | 0.073 0.057 CHEMBL3706466 0.091 0.025 CHEMBL3706475 0.069 0.067 CHEMBL3706478 0.075 0.052 CHEMBL1222314 | CHEMBL3706475 | |
| 0.017 | 0.316 | 0.157 | CYP2A6 inhibitor | 0.11 0.031 CHEMBL3706466 0.093 0.039 CHEMBL3706475 0.107 0.032 CHEMBL3706478 0.157 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.312 | 0.063 | Prolyl endopeptidase inhibitor | 0.063 0.021 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.313 | 0.032 | Hedgehog signaling activator | 0.032 0.009 CHEMBL3706465 0.031 0.012 CHEMBL3706475 | CHEMBL3706465 | |
| 0.013 | 0.314 | 0.075 | Retinoid X receptor antagonist | 0.047 0.015 CHEMBL3706466 0.041 0.021 CHEMBL3706478 0.075 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.081 | 0.382 | 0.378 | Hypoxia-inducible factor 1 alpha inhibitor | 0.378 0.036 CHEMBL3706466 0.288 0.071 CHEMBL3706478 0.298 0.067 CHEMBL1222314 | CHEMBL3706466 | |
| 0.033 | 0.338 | 0.075 | Transcription factor RelA inhibitor | 0.063 0.044 CHEMBL3706466 0.075 0.023 CHEMBL3706475 0.074 0.024 CHEMBL1222314 | CHEMBL3706475 | |
| 0.007 | 0.313 | 0.04 | Liver X receptor antagonist | 0.04 0.014 CHEMBL3706466 | CHEMBL3706466 | |
| 0.011 | 0.318 | 0.198 | Alcohol oxidase inhibitor | 0.1 0.018 CHEMBL3706465 0.108 0.016 CHEMBL3706466 0.174 0.008 CHEMBL3706475 0.116 0.015 CHEMBL3706478 0.198 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.323 | 0.15 | Glutamate decarboxylase inhibitor | 0.109 0.025 CHEMBL3706466 0.09 0.036 CHEMBL3706475 0.15 0.013 CHEMBL3706478 0.15 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.319 | 0.104 | HIV-1 integrase (3'-Processing) inhibitor | 0.104 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.317 | 0.05 | Oxytocin agonist | 0.04 0.031 CHEMBL3706475 0.05 0.024 CHEMBL1222314 | CHEMBL1222314 | |
| 0.016 | 0.326 | 0.041 | Glutamate (mGluR8) antagonist | 0.041 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.317 | 0.05 | Endothelial nitric-oxide synthase inhibitor | 0.038 0.014 CHEMBL3706466 0.05 0.009 CHEMBL3706478 0.048 0.01 CHEMBL1222314 | CHEMBL3706478 | |
| 0.007 | 0.321 | 0.473 | Prostaglandin EP2 antagonist | 0.091 0.022 CHEMBL3706466 0.189 0.007 CHEMBL3706478 0.473 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.028 | 0.342 | 0.125 | Sphingomyelinase inhibitor | 0.125 0.038 CHEMBL3706465 | CHEMBL3706465 | |
| 0.012 | 0.327 | 0.173 | Biliverdin reductase inhibitor | 0.053 0.048 CHEMBL3706465 0.111 0.016 CHEMBL3706466 0.129 0.012 CHEMBL3706475 0.114 0.015 CHEMBL3706478 0.173 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.338 | 0.054 | Nicotinic alpha3beta2 receptor antagonist | 0.054 0.035 CHEMBL3706465 | CHEMBL3706465 | |
| 0.006 | 0.325 | 0.125 | Retinoid X alpha receptor agonist | 0.043 0.018 CHEMBL3706466 0.034 0.025 CHEMBL3706478 0.125 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.325 | 0.048 | Farnesoid X receptor agonist | 0.036 0.029 CHEMBL3706465 0.048 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.326 | 0.116 | Endothelin A receptor antagonist | 0.116 0.004 CHEMBL3706478 0.043 0.007 CHEMBL1222314 | CHEMBL3706478 | |
| 0.004 | 0.326 | 0.036 | Estradiol 17 beta-dehydrogenase inhibitor | 0.036 0.035 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.336 | 0.148 | Carbonic anhydrase V inhibitor | 0.081 0.035 CHEMBL3706466 0.098 0.028 CHEMBL3706478 0.148 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.335 | 0.076 | Selectin antagonist | 0.058 0.051 CHEMBL3706472 0.076 0.039 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.336 | 0.093 | HIV-1 integrase (Strand Transfer) inhibitor | 0.093 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.039 | 0.37 | 0.197 | DOPA decarboxylase inhibitor | 0.16 0.017 CHEMBL3706466 0.149 0.022 CHEMBL3706475 0.149 0.022 CHEMBL3706478 0.197 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.341 | 0.056 | 5 Hydroxytryptamine 4 antagonist | 0.056 0.028 CHEMBL3706465 | CHEMBL3706465 | |
| 0.003 | 0.337 | 0.026 | Hexokinase stimulant | 0.026 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.348 | 0.089 | Histidine decarboxylase inhibitor | 0.08 0.042 CHEMBL3706465 0.069 0.052 CHEMBL3706466 0.076 0.045 CHEMBL3706475 0.089 0.037 CHEMBL1222314 | CHEMBL1222314 | |
| 0.056 | 0.393 | 0.271 | Succinate dehydrogenase inhibitor | 0.159 0.097 CHEMBL3706465 0.235 0.028 CHEMBL3706466 0.192 0.056 CHEMBL3706475 0.229 0.031 CHEMBL3706478 0.271 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.069 | 0.407 | 0.329 | Immunosuppressant | 0.329 0.098 CHEMBL3706465 0.2 0.197 CHEMBL1222314 | CHEMBL3706465 | |
| 0.012 | 0.35 | 0.123 | Catalase inhibitor | 0.078 0.048 CHEMBL3706466 0.123 0.032 CHEMBL3706478 0.091 0.042 CHEMBL1222314 | CHEMBL3706478 | |
| 0.017 | 0.356 | 0.102 | Aminopeptidase I inhibitor | 0.088 0.035 CHEMBL3706466 0.086 0.037 CHEMBL3706475 0.092 0.033 CHEMBL3706478 0.102 0.027 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.346 | 0.079 | Phosphorylase inhibitor | 0.053 0.028 CHEMBL3706478 0.079 0.017 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.349 | 0.044 | Dopamine D5 agonist | 0.044 0.022 CHEMBL3706475 | CHEMBL3706475 | |
| 0.011 | 0.355 | 0.067 | Adenosine deaminase inhibitor | 0.059 0.022 CHEMBL3706475 0.067 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.352 | 0.06 | Retinoic acid gamma receptor agonist | 0.06 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.083 | 0.432 | 0.33 | RNA-directed DNA polymerase inhibitor | 0.22 0.074 CHEMBL3706465 0.187 0.12 CHEMBL3706466 0.33 0.027 CHEMBL3706475 0.174 0.144 CHEMBL3706478 0.226 0.068 CHEMBL1222314 | CHEMBL3706475 | |
| 0.018 | 0.367 | 0.063 | Transcription factor AP-1 inhibitor | 0.063 0.039 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.357 | 0.055 | Glutamate (mGluR3) antagonist | 0.034 0.029 CHEMBL3706466 0.033 0.032 CHEMBL3706478 0.055 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.024 | 0.373 | 0.216 | Nitric-oxide synthase inhibitor | 0.15 0.022 CHEMBL3706466 0.163 0.018 CHEMBL3706478 0.216 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.361 | 0.07 | Leukotriene B4 antagonist | 0.049 0.047 CHEMBL3706466 0.07 0.019 CHEMBL3706478 0.053 0.039 CHEMBL1222314 | CHEMBL3706478 | |
| 0.023 | 0.376 | 0.16 | Creatine kinase inhibitor | 0.16 0.02 CHEMBL3706465 0.096 0.064 CHEMBL3706466 0.154 0.022 CHEMBL3706475 0.093 0.068 CHEMBL3706478 0.144 0.026 CHEMBL1222314 | CHEMBL3706465 | |
| 0.003 | 0.358 | 0.083 | Endothelin B receptor antagonist | 0.083 0.004 CHEMBL3706478 0.018 0.014 CHEMBL1222314 | CHEMBL3706478 | |
| 0.007 | 0.362 | 0.112 | RNA-directed RNA polymerase inhibitor | 0.112 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.073 | 0.428 | 0.245 | Growth factor agonist | 0.17 0.101 CHEMBL3706466 0.224 0.044 CHEMBL3706478 0.245 0.034 CHEMBL1222314 | CHEMBL1222314 | |
| 0.06 | 0.416 | 0.196 | Phospholipase C inhibitor | 0.196 0.047 CHEMBL3706465 0.138 0.134 CHEMBL3706466 0.177 0.064 CHEMBL3706475 0.159 0.089 CHEMBL1222314 | CHEMBL3706465 | |
| 0.05 | 0.407 | 0.13 | Antipruritic | 0.13 0.122 CHEMBL3706465 0.13 0.123 CHEMBL3706478 | CHEMBL3706478 | |
| 0.004 | 0.362 | 0.139 | Endothelin receptor antagonist | 0.139 0.004 CHEMBL3706478 0.051 0.01 CHEMBL1222314 | CHEMBL3706478 | |
| 0.024 | 0.383 | 0.069 | DNA helicase inhibitor | 0.069 0.018 CHEMBL3706466 0.066 0.021 CHEMBL3706478 0.059 0.03 CHEMBL1222314 | CHEMBL3706466 | |
| 0.012 | 0.373 | 0.188 | Phenylalanine 4-hydroxylase inhibitor | 0.115 0.02 CHEMBL3706466 0.096 0.028 CHEMBL3706475 0.188 0.008 CHEMBL3706478 0.12 0.018 CHEMBL1222314 | CHEMBL3706478 | |
| 0.053 | 0.413 | 0.17 | Melanin inhibitor | 0.125 0.124 CHEMBL3706466 0.17 0.06 CHEMBL3706475 0.142 0.093 CHEMBL3706478 0.133 0.109 CHEMBL1222314 | CHEMBL3706475 | |
| 0.013 | 0.376 | 0.043 | Thymidine kinase inhibitor | 0.043 0.025 CHEMBL3706465 0.04 0.03 CHEMBL3706475 | CHEMBL3706465 | |
| 0.003 | 0.366 | 0.064 | Methionyl aminopeptidase 2 inhibitor | 0.064 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.371 | 0.061 | ICAM 1 antagonist | 0.025 0.011 CHEMBL3706466 0.025 0.011 CHEMBL3706478 0.061 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.375 | 0.122 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.069 0.027 CHEMBL3706465 0.059 0.035 CHEMBL3706466 0.122 0.011 CHEMBL3706475 0.064 0.031 CHEMBL3706478 0.063 0.031 CHEMBL1222314 | CHEMBL3706475 | |
| 0.052 | 0.418 | 0.163 | NOS3 expression enhancer | 0.119 0.117 CHEMBL3706478 0.163 0.061 CHEMBL1222314 | CHEMBL1222314 | |
| 0.037 | 0.404 | 0.139 | Photosensitizer | 0.111 0.07 CHEMBL3706466 0.127 0.049 CHEMBL3706475 0.139 0.039 CHEMBL3706478 0.128 0.049 CHEMBL1222314 | CHEMBL3706478 | |
| 0.004 | 0.372 | 0.215 | TRPM8 blocker | 0.05 0.016 CHEMBL3706466 0.035 0.03 CHEMBL3706478 0.215 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.071 | 0.442 | 0.233 | Gastrin inhibitor | 0.233 0.1 CHEMBL3706465 0.188 0.167 CHEMBL3706466 0.198 0.152 CHEMBL3706475 0.214 0.128 CHEMBL3706478 0.217 0.123 CHEMBL1222314 | CHEMBL3706465 | |
| 0.004 | 0.376 | 0.039 | Prostaglandin EP3 antagonist | 0.033 0.018 CHEMBL3706478 0.039 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.386 | 0.096 | Thromboxane synthase inhibitor | 0.055 0.037 CHEMBL3706466 0.055 0.036 CHEMBL3706478 0.096 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.026 | 0.404 | 0.09 | Estrogen receptor beta antagonist | 0.09 0.084 CHEMBL3706465 | CHEMBL3706465 | |
| 0.023 | 0.402 | 0.114 | Prolactin inhibitor | 0.114 0.043 CHEMBL3706465 | CHEMBL3706465 | |
| 0.005 | 0.384 | 0.027 | Lysophosphatidic acid 1 receptor antagonist | 0.02 0.017 CHEMBL3706478 0.027 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.017 | 0.4 | 0.038 | Glucose-6-phosphate dehydrogenase inhibitor | 0.038 0.026 CHEMBL3706465 | CHEMBL3706465 | |
| 0.01 | 0.392 | 0.072 | Glutamate (mGluR4) agonist | 0.043 0.014 CHEMBL3706466 0.036 0.02 CHEMBL3706478 0.072 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.394 | 0.037 | Toll-Like receptor 2 agonist | 0.037 0.032 CHEMBL3706472 | CHEMBL3706472 | |
| 0.013 | 0.401 | 0.138 | Inducible nitric-oxide synthase inhibitor | 0.11 0.03 CHEMBL3706466 0.128 0.022 CHEMBL3706478 0.138 0.019 CHEMBL1222314 | CHEMBL1222314 | |
| 0.091 | 0.479 | 0.169 | Heat shock protein 70 antagonist | 0.133 0.107 CHEMBL3706465 0.143 0.064 CHEMBL3706466 0.153 0.04 CHEMBL3706475 0.136 0.09 CHEMBL3706478 0.169 0.019 CHEMBL1222314 | CHEMBL1222314 | |
| 0.04 | 0.435 | 0.091 | Estrogen-related receptor beta agonist | 0.085 0.053 CHEMBL3706465 0.091 0.038 CHEMBL3706475 0.079 0.071 CHEMBL1222314 | CHEMBL3706475 | |
| 0.034 | 0.434 | 0.259 | Insulin sensitizer | 0.182 0.093 CHEMBL3706466 0.259 0.03 CHEMBL3706478 0.201 0.072 CHEMBL1222314 | CHEMBL3706478 | |
| 0.007 | 0.408 | 0.057 | Nerve growth factor antagonist | 0.057 0.012 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.411 | 0.045 | Complement factor 1s inhibitor | 0.029 0.01 CHEMBL3706466 0.027 0.014 CHEMBL3706478 0.045 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.414 | 0.088 | Sphingosine kinase 2 inhibitor | 0.088 0.011 CHEMBL3706465 0.083 0.014 CHEMBL3706475 | CHEMBL3706465 | |
| 0.043 | 0.449 | 0.216 | Insulin secretagoues | 0.216 0.029 CHEMBL3706478 | CHEMBL3706478 | |
| 0.01 | 0.416 | 0.278 | Protein-tyrosine phosphatase 1B inhibitor | 0.278 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.023 | 0.429 | 0.138 | AMP-activated protein kinase stimulant | 0.138 0.036 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.42 | 0.043 | Vanilloid 3 antagonist | 0.043 0.017 CHEMBL3706475 | CHEMBL3706475 | |
| 0.017 | 0.424 | 0.076 | Interferon agonist | 0.076 0.059 CHEMBL3706475 | CHEMBL3706475 | |
| 0.027 | 0.44 | 0.099 | Bile acid receptor antagonist | 0.09 0.075 CHEMBL3706465 0.089 0.076 CHEMBL3706478 0.099 0.051 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.42 | 0.05 | HIV-1 protease inhibitor | 0.05 0.021 CHEMBL3706475 | CHEMBL3706475 | |
| 0.001 | 0.416 | 0.027 | Angiotensin AT1B receptor antagonist | 0.022 0.005 CHEMBL3706466 0.015 0.008 CHEMBL3706478 0.027 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.022 | 0.439 | 0.143 | Interleukin 1 beta converting enzyme inhibitor | 0.134 0.025 CHEMBL3706466 0.142 0.021 CHEMBL3706478 0.143 0.02 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.439 | 0.407 | Protein-tyrosine phosphatase inhibitor | 0.36 0.011 CHEMBL3706474 0.137 0.093 CHEMBL3706478 0.407 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.425 | 0.084 | Leukotriene antagonist | 0.084 0.029 CHEMBL3706478 0.078 0.034 CHEMBL1222314 | CHEMBL3706478 | |
| 0.004 | 0.423 | 0.12 | Prostaglandin EP4 antagonist | 0.039 0.011 CHEMBL3706478 0.12 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.425 | 0.067 | NMDA 2A receptor antagonist | 0.046 0.041 CHEMBL3706466 0.053 0.035 CHEMBL3706478 0.067 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.435 | 0.116 | Glutamate (mGluR group III) agonist | 0.052 0.022 CHEMBL3706466 0.056 0.02 CHEMBL3706478 0.116 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.025 | 0.448 | 0.146 | Bone formation stimulant | 0.146 0.062 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.44 | 0.068 | Glutamate (mGluR7) antagonist | 0.068 0.047 CHEMBL3706465 0.067 0.048 CHEMBL1222314 | CHEMBL3706465 | |
| 0.002 | 0.427 | 0.015 | Human herpes virus 5 capsid protein P40 inhibitor | 0.015 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.429 | 0.179 | Urate transporter 1 inhibitor | 0.072 0.01 CHEMBL3706466 0.089 0.006 CHEMBL3706478 0.179 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.435 | 0.027 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.027 0.016 CHEMBL3706465 0.025 0.023 CHEMBL3706475 | CHEMBL3706465 | |
| 0.011 | 0.438 | 0.043 | AICAR transformylase inhibitor | 0.041 0.036 CHEMBL3706466 0.043 0.032 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.437 | 0.125 | Monophenol monooxygenase inhibitor | 0.106 0.072 CHEMBL3706478 0.125 0.058 CHEMBL1222314 | CHEMBL1222314 | |
| 0.03 | 0.458 | 0.101 | Estrogen antagonist | 0.101 0.097 CHEMBL3706465 0.1 0.098 CHEMBL3706475 | CHEMBL3706465 | |
| 0.043 | 0.475 | 0.4 | Lipoxygenase inhibitor | 0.38 0.043 CHEMBL3706466 0.19 0.15 CHEMBL3706475 0.22 0.122 CHEMBL3706478 0.4 0.037 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.455 | 0.323 | Ferrochelatase inhibitor | 0.217 0.019 CHEMBL3706466 0.152 0.037 CHEMBL3706475 0.323 0.006 CHEMBL3706478 0.297 0.008 CHEMBL1222314 | CHEMBL3706478 | |
| 0.008 | 0.445 | 0.084 | Retinoic acid alpha receptor agonist | 0.084 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.457 | 0.149 | Aminopeptidase B inhibitor | 0.118 0.053 CHEMBL3706466 0.092 0.071 CHEMBL3706472 0.093 0.07 CHEMBL3706475 0.117 0.054 CHEMBL3706478 0.149 0.038 CHEMBL1222314 | CHEMBL1222314 | |
| 0.069 | 0.508 | 0.377 | 5 Hydroxytryptamine release stimulant | 0.377 0.051 CHEMBL3706465 0.218 0.107 CHEMBL3706475 | CHEMBL3706465 | |
| 0.002 | 0.441 | 0.026 | Nicotinic acid receptor 1 antagonist | 0.026 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.001 | 0.441 | 0.044 | Kainate receptor 1 antagonist | 0.044 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.002 | 0.443 | 0.029 | Uridine phosphorylase inhibitor | 0.029 0.019 CHEMBL3706475 | CHEMBL3706475 | |
| 0.026 | 0.471 | 0.263 | Antibacterial (Helicobacter pylori) | 0.134 0.063 CHEMBL3706466 0.119 0.083 CHEMBL3706475 0.263 0.01 CHEMBL3706478 0.192 0.024 CHEMBL1222314 | CHEMBL3706478 | |
| 0.017 | 0.463 | 0.102 | Purinergic P2X1 antagonist | 0.061 0.041 CHEMBL3706466 0.098 0.017 CHEMBL3706475 0.074 0.029 CHEMBL3706478 0.102 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.066 | 0.513 | 0.306 | Vasodilator, coronary | 0.306 0.082 CHEMBL3706465 0.199 0.183 CHEMBL3706475 | CHEMBL3706465 | |
| 0.035 | 0.483 | 0.375 | Aldehyde oxidase inhibitor | 0.246 0.084 CHEMBL3706465 0.246 0.084 CHEMBL3706466 0.326 0.06 CHEMBL3706475 0.223 0.093 CHEMBL3706478 0.375 0.051 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.453 | 0.038 | Phosphoglycerate kinase inhibitor | 0.038 0.021 CHEMBL3706475 0.032 0.028 CHEMBL1222314 | CHEMBL3706475 | |
| 0.004 | 0.454 | 0.046 | Peroxisome proliferator-activated receptor alpha agonist | 0.046 0.036 CHEMBL3706478 0.043 0.038 CHEMBL1222314 | CHEMBL3706478 | |
| 0.018 | 0.469 | 0.059 | Ryanodine receptor antagonist | 0.059 0.04 CHEMBL3706475 0.058 0.044 CHEMBL1222314 | CHEMBL3706475 | |
| 0.013 | 0.469 | 0.092 | Phospholipase D inhibitor | 0.092 0.021 CHEMBL3706465 | CHEMBL3706465 | |
| 0.074 | 0.53 | 0.274 | Calcium channel activator | 0.253 0.143 CHEMBL3706465 0.236 0.164 CHEMBL3706466 0.274 0.12 CHEMBL3706475 0.247 0.151 CHEMBL3706478 0.257 0.139 CHEMBL1222314 | CHEMBL3706475 | |
| 0.011 | 0.47 | 0.077 | Protein kinase C beta inhibitor | 0.069 0.05 CHEMBL3706478 0.077 0.035 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.477 | 0.089 | Cathepsin G inhibitor | 0.089 0.038 CHEMBL3706478 0.068 0.056 CHEMBL1222314 | CHEMBL3706478 | |
| 0.055 | 0.518 | 0.129 | Sphingosine 1-phosphate receptor 2 agonist | 0.129 0.043 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.472 | 0.044 | VCAM-1 antagonist | 0.039 0.031 CHEMBL3706466 0.038 0.031 CHEMBL3706478 0.044 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.473 | 0.044 | VCAM antagonist | 0.038 0.031 CHEMBL3706466 0.038 0.031 CHEMBL3706478 0.044 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.474 | 0.147 | 5-Lipoxygenase inhibitor | 0.102 0.062 CHEMBL3706466 0.147 0.039 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.469 | 0.05 | NMDA receptor subunit 3A antagonist | 0.035 0.029 CHEMBL3706478 0.05 0.02 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.474 | 0.042 | Ceramide glucosyltransferase inhibitor | 0.042 0.014 CHEMBL3706465 | CHEMBL3706465 | |
| 0.001 | 0.471 | 0.027 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.027 0.02 CHEMBL3706475 | CHEMBL3706475 | |
| 0.029 | 0.501 | 0.176 | Free radical scavenger | 0.176 0.118 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.476 | 0.033 | Peroxisome proliferator-activated receptor delta agonist | 0.033 0.023 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.479 | 0.083 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.083 0.023 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.478 | 0.059 | Geranyltranstransferase inhibitor | 0.045 0.029 CHEMBL3706475 0.059 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.484 | 0.069 | Glucagon-like peptide 1 agonist | 0.069 0.042 CHEMBL3706471 0.064 0.046 CHEMBL3706472 0.066 0.044 CHEMBL1222314 | CHEMBL3706471 | |
| 0.016 | 0.495 | 0.065 | Interferon inducer | 0.065 0.042 CHEMBL3706475 | CHEMBL3706475 | |
| 0.035 | 0.518 | 0.1 | 3C-Like protease (SARS coronavirus) inhibitor | 0.1 0.033 CHEMBL1222314 | CHEMBL1222314 | |
| 0.018 | 0.503 | 0.081 | Glutathione S-transferase inhibitor | 0.075 0.07 CHEMBL3706466 0.077 0.066 CHEMBL3706478 0.081 0.059 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.491 | 0.021 | Glutamate (mGluR1a) agonist | 0.021 0.018 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.494 | 0.057 | Angiotensin AT2 receptor antagonist | 0.057 0.009 CHEMBL3706466 0.048 0.01 CHEMBL3706478 0.022 0.015 CHEMBL1222314 | CHEMBL3706466 | |
| 0.007 | 0.498 | 0.1 | AMPA 4 receptor antagonist | 0.04 0.027 CHEMBL3706466 0.04 0.027 CHEMBL3706478 0.1 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.499 | 0.046 | Lysophosphatidic acid 3 receptor antagonist | 0.046 0.042 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.507 | 0.141 | Caspase 7 inhibitor | 0.101 0.027 CHEMBL3706466 0.109 0.021 CHEMBL3706478 0.141 0.009 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.503 | 0.073 | Sphingosine kinase inhibitor | 0.07 0.025 CHEMBL3706465 0.073 0.022 CHEMBL3706475 | CHEMBL3706475 | |
| 0.003 | 0.498 | 0.027 | Beta 1 adrenoreceptor agonist | 0.027 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.506 | 0.033 | Liver X receptor beta antagonist | 0.033 0.017 CHEMBL3706466 | CHEMBL3706466 | |
| 0.005 | 0.507 | 0.036 | Lysophosphatidic acid 2 receptor antagonist | 0.027 0.026 CHEMBL3706466 0.036 0.015 CHEMBL3706478 0.029 0.023 CHEMBL1222314 | CHEMBL3706478 | |
| 0.019 | 0.522 | 0.075 | Carbonic anhydrase VI inhibitor | 0.075 0.064 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.528 | 0.056 | Adenine nucleotide translocase inhibitor | 0.053 0.047 CHEMBL3706472 0.056 0.037 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.528 | 0.107 | HIV-1 integrase (Overall Integration) inhibitor | 0.087 0.068 CHEMBL3706466 0.107 0.048 CHEMBL3706478 0.091 0.063 CHEMBL1222314 | CHEMBL3706478 | |
| 0.058 | 0.57 | 0.268 | Analgesic | 0.268 0.167 CHEMBL3706465 | CHEMBL3706465 | |
| 0.008 | 0.522 | 0.036 | Tryptophan 5 hydroxylase inhibitor | 0.036 0.024 CHEMBL3706478 0.036 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.018 | 0.532 | 0.099 | Keratolytic | 0.069 0.068 CHEMBL3706466 0.075 0.056 CHEMBL3706475 0.07 0.066 CHEMBL3706478 0.099 0.031 CHEMBL1222314 | CHEMBL1222314 | |
| 0.029 | 0.544 | 0.368 | Non-steroidal antiinflammatory agent | 0.189 0.08 CHEMBL3706466 0.219 0.058 CHEMBL3706478 0.368 0.017 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.524 | 0.087 | CDC25B inhibitor | 0.058 0.053 CHEMBL3706478 0.087 0.023 CHEMBL1222314 | CHEMBL1222314 | |
| 0.001 | 0.517 | 0.027 | Thrombopoietin agonist | 0.027 0.003 CHEMBL1222314 | CHEMBL1222314 | |
| 0.035 | 0.552 | 0.232 | Hexokinase inhibitor | 0.173 0.055 CHEMBL3706466 0.167 0.061 CHEMBL3706475 0.144 0.086 CHEMBL3706478 0.232 0.021 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.522 | 0.037 | Purinergic P2Y15 antagonist | 0.034 0.012 CHEMBL3706465 0.037 0.009 CHEMBL3706475 | CHEMBL3706475 | |
| 0.025 | 0.546 | 0.242 | DNA methyltransferase I inhibitor | 0.148 0.106 CHEMBL3706466 0.134 0.125 CHEMBL3706478 0.242 0.05 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.53 | 0.048 | Purinergic P2Y14 antagonist | 0.048 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.031 | 0.557 | 0.119 | Transcription factor NF kappa B stimulant | 0.087 0.056 CHEMBL3706472 0.119 0.026 CHEMBL3706475 | CHEMBL3706475 | |
| 0.036 | 0.561 | 0.376 | 3C-like protease (Human coronavirus) inhibitor | 0.205 0.049 CHEMBL3706466 0.151 0.1 CHEMBL3706475 0.186 0.06 CHEMBL3706478 0.376 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.025 | 0.552 | 0.106 | Electron transport complex I inhibitor | 0.106 0.069 CHEMBL3706478 | CHEMBL3706478 | |
| 0.023 | 0.552 | 0.235 | Aldehyde dehydrogenase inhibitor | 0.146 0.05 CHEMBL3706466 0.115 0.076 CHEMBL3706475 0.143 0.052 CHEMBL3706478 0.235 0.021 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.537 | 0.215 | Porphobilinogen synthase inhibitor | 0.135 0.024 CHEMBL3706466 0.08 0.047 CHEMBL3706475 0.111 0.031 CHEMBL3706478 0.215 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.026 | 0.556 | 0.125 | Carbonic anhydrase XV inhibitor | 0.125 0.043 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.54 | 0.196 | HIV-1 integrase inhibitor | 0.196 0.005 CHEMBL3706478 | CHEMBL3706478 | |
| 0.002 | 0.533 | 0.04 | Kynurenine 3 monooxygenase inhibitor | 0.029 0.016 CHEMBL3706478 0.04 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.539 | 0.087 | Protein kinase C zeta inhibitor | 0.087 0.072 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.536 | 0.049 | NMDA receptor subunit 3B antagonist | 0.049 0.026 CHEMBL1222314 | CHEMBL1222314 | |
| 0.034 | 0.567 | 0.211 | Cyclic AMP phosphodiesterase inhibitor | 0.211 0.086 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.547 | 0.149 | Mediator release inhibitor | 0.098 0.072 CHEMBL3706478 0.149 0.029 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.548 | 0.132 | GABA C receptor antagonist | 0.11 0.064 CHEMBL3706465 0.1 0.078 CHEMBL3706466 0.109 0.065 CHEMBL3706475 0.132 0.042 CHEMBL1222314 | CHEMBL1222314 | |
| 0.034 | 0.568 | 0.249 | Interleukin agonist | 0.249 0.08 CHEMBL3706465 0.2 0.121 CHEMBL3706475 0.198 0.123 CHEMBL3706478 0.171 0.148 CHEMBL1222314 | CHEMBL3706465 | |
| 0.003 | 0.538 | 0.032 | Free fatty acid receptor 1 antagonist | 0.032 0.026 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.54 | 0.046 | GABA B receptor antagonist | 0.046 0.024 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.545 | 0.125 | Neuraminidase (influenza) inhibitor | 0.125 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.542 | 0.041 | Carbonic anhydrase VII inhibitor | 0.041 0.039 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.545 | 0.095 | Protein kinase (CK2) beta inhibitor | 0.095 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.074 | 0.613 | 0.236 | Nitric-oxide synthase stimulant | 0.205 0.08 CHEMBL3706465 0.236 0.044 CHEMBL3706475 0.207 0.078 CHEMBL3706478 0.181 0.126 CHEMBL1222314 | CHEMBL3706475 | |
| 0.01 | 0.548 | 0.212 | M17 leucyl aminopeptidase inhibitor | 0.212 0.029 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.546 | 0.101 | Peroxisome proliferator-activated receptor gamma agonist | 0.101 0.027 CHEMBL3706478 | CHEMBL3706478 | |
| 0.022 | 0.563 | 0.113 | Carbonic anhydrase III inhibitor | 0.094 0.07 CHEMBL3706475 0.093 0.07 CHEMBL3706478 0.113 0.05 CHEMBL1222314 | CHEMBL1222314 | |
| 0.02 | 0.562 | 0.099 | Thioredoxin inhibitor | 0.099 0.049 CHEMBL3706475 | CHEMBL3706475 | |
| 0.003 | 0.547 | 0.133 | Prostaglandin EP1 antagonist | 0.133 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.552 | 0.045 | Potassium channel (ATP-sensitive) activator | 0.045 0.041 CHEMBL3706475 | CHEMBL3706475 | |
| 0.007 | 0.553 | 0.073 | Plasminogen activator inhibitor antagonist | 0.073 0.018 CHEMBL1222314 | CHEMBL1222314 | |
| 0.025 | 0.57 | 0.116 | Lanosterol 14 alpha demethylase inhibitor | 0.087 0.077 CHEMBL3706465 0.116 0.035 CHEMBL3706475 0.105 0.049 CHEMBL3706478 | CHEMBL3706475 | |
| 0.014 | 0.56 | 0.08 | Dihydroorotate oxidase inhibitor | 0.051 0.047 CHEMBL3706478 0.08 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.557 | 0.139 | GABA aminotransferase inhibitor | 0.068 0.065 CHEMBL3706466 0.139 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.556 | 0.047 | Potassium channel (Inward rectifier) activator | 0.047 0.042 CHEMBL3706475 | CHEMBL3706475 | |
| 0.009 | 0.558 | 0.069 | Carbonic anhydrase stimulant | 0.069 0.033 CHEMBL3706478 | CHEMBL3706478 | |
| 0.003 | 0.554 | 0.087 | Fructose-1,6-bisphosphatase inhibitor | 0.042 0.035 CHEMBL3706466 0.087 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.032 | 0.584 | 0.519 | 15-Lipoxygenase inhibitor | 0.22 0.192 CHEMBL3706478 0.519 0.036 CHEMBL1222314 | CHEMBL1222314 | |
| 0.035 | 0.587 | 0.193 | Tumour necrosis factor antagonist | 0.193 0.058 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.558 | 0.025 | Glutamate (mGluR1) agonist | 0.025 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.567 | 0.162 | Phospholipase A2 inhibitor | 0.135 0.093 CHEMBL3706478 0.162 0.064 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.558 | 0.025 | Angiotensin AT1A receptor antagonist | 0.025 0.01 CHEMBL3706466 0.024 0.011 CHEMBL1222314 | CHEMBL3706466 | |
| 0.016 | 0.575 | 0.052 | CD45 antagonist | 0.052 0.031 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.566 | 0.093 | Neuraminidase inhibitor | 0.093 0.018 CHEMBL1222314 | CHEMBL1222314 | |
| 0.002 | 0.567 | 0.027 | Fructose-1,6-bisphosphatase 1 inhibitor | 0.027 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.016 | 0.583 | 0.127 | GABA C receptor rho-1 antagonist | 0.09 0.079 CHEMBL3706475 0.127 0.034 CHEMBL1222314 | CHEMBL1222314 | |
| 0.046 | 0.615 | 0.188 | Neurotensin receptor agonist | 0.17 0.063 CHEMBL3706466 0.159 0.08 CHEMBL3706478 0.188 0.042 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.582 | 0.106 | Gastric antisecretory | 0.106 0.058 CHEMBL3706478 | CHEMBL3706478 | |
| 0.023 | 0.593 | 0.212 | DNA methylase inhibitor | 0.212 0.071 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.584 | 0.178 | Caspase 3 inhibitor | 0.138 0.038 CHEMBL3706466 0.139 0.037 CHEMBL3706478 0.178 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.591 | 0.089 | mTOR complex 2 inhibitor | 0.089 0.049 CHEMBL3706465 | CHEMBL3706465 | |
| 0.021 | 0.592 | 0.088 | Granulocyte macrophage colony stimulating factor agonist | 0.088 0.056 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.58 | 0.092 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.092 0.02 CHEMBL3706475 0.073 0.052 CHEMBL1222314 | CHEMBL3706475 | |
| 0.017 | 0.591 | 0.234 | Xanthine oxidase inhibitor | 0.234 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.025 | 0.605 | 0.357 | Peroxidase inhibitor | 0.217 0.055 CHEMBL3706466 0.233 0.051 CHEMBL3706475 0.357 0.027 CHEMBL3706478 0.239 0.05 CHEMBL1222314 | CHEMBL3706478 | |
| 0.005 | 0.586 | 0.049 | Sphingosine kinase 1 inhibitor | 0.038 0.035 CHEMBL3706465 0.049 0.018 CHEMBL3706475 | CHEMBL3706475 | |
| 0.01 | 0.592 | 0.043 | Glutamate (mGluR group III) antagonist | 0.043 0.033 CHEMBL1222314 | CHEMBL1222314 | |
| 0.034 | 0.616 | 0.179 | Neurotrophic factor enhancer | 0.179 0.099 CHEMBL3706465 0.162 0.12 CHEMBL3706475 | CHEMBL3706465 | |
| 0.015 | 0.6 | 0.1 | Factor XII inhibitor | 0.1 0.038 CHEMBL1222314 | CHEMBL1222314 | |
| 0.002 | 0.589 | 0.033 | Methionyl aminopeptidase 1 inhibitor | 0.033 0.02 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.595 | 0.061 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.05 0.042 CHEMBL3706475 0.061 0.028 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.601 | 0.114 | Acetylcholinesterase inhibitor | 0.114 0.083 CHEMBL3706465 | CHEMBL3706465 | |
| 0.02 | 0.61 | 0.189 | Sphingosine 1-phosphate receptor 4 antagonist | 0.138 0.045 CHEMBL3706466 0.126 0.062 CHEMBL3706478 0.189 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.604 | 0.079 | Histamine H2 receptor antagonist | 0.079 0.067 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.601 | 0.113 | Urease inhibitor | 0.113 0.052 CHEMBL3706478 0.092 0.076 CHEMBL1222314 | CHEMBL3706478 | |
| 0.019 | 0.613 | 0.058 | Immunoglobulin Fc receptor antagonist | 0.053 0.047 CHEMBL3706475 0.058 0.029 CHEMBL1222314 | CHEMBL1222314 | |
| 0.022 | 0.618 | 0.184 | Hemostatic | 0.184 0.04 CHEMBL1222314 | CHEMBL1222314 | |
| 0.019 | 0.617 | 0.079 | MAP kinase kinase 7 inhibitor | 0.079 0.049 CHEMBL3706465 0.079 0.049 CHEMBL3706475 | CHEMBL3706475 | |
| 0.028 | 0.628 | 0.376 | DNA damaging | 0.376 0.034 CHEMBL3706475 | CHEMBL3706475 | |
| 0.008 | 0.609 | 0.088 | Peroxisome proliferator-activated receptor gamma antagonist | 0.068 0.06 CHEMBL3706466 0.088 0.024 CHEMBL3706478 0.076 0.04 CHEMBL1222314 | CHEMBL3706478 | |
| 0.002 | 0.609 | 0.071 | Kainate receptor antagonist | 0.071 0.012 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.622 | 0.272 | Hypolipemic | 0.272 0.058 CHEMBL3706478 | CHEMBL3706478 | |
| 0.014 | 0.621 | 0.097 | Beta glucuronidase inhibitor | 0.097 0.075 CHEMBL3706475 0.093 0.082 CHEMBL1222314 | CHEMBL3706475 | |
| 0.011 | 0.619 | 0.042 | Cathepsin F inhibitor | 0.042 0.027 CHEMBL1222314 | CHEMBL1222314 | |
| 0.021 | 0.631 | 0.127 | Amylase inhibitor | 0.105 0.092 CHEMBL3706465 0.127 0.076 CHEMBL3706475 | CHEMBL3706475 | |
| 0.011 | 0.621 | 0.078 | Histamine N-methyltransferase inhibitor | 0.078 0.07 CHEMBL3706465 | CHEMBL3706465 | |
| 0.037 | 0.65 | 0.468 | Histamine release inhibitor | 0.221 0.179 CHEMBL3706466 0.267 0.143 CHEMBL3706475 0.333 0.108 CHEMBL3706478 0.468 0.041 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.632 | 0.18 | Mannose-6-phosphate isomerase inhibitor | 0.124 0.093 CHEMBL3706466 0.178 0.044 CHEMBL3706475 0.122 0.098 CHEMBL3706478 0.18 0.042 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.632 | 0.369 | Aminoacyl-tRNA synthetase inhibitor | 0.369 0.004 CHEMBL3706478 | CHEMBL3706478 | |
| 0.002 | 0.623 | 0.019 | CC chemokine 9 receptor antagonist | 0.019 0.009 CHEMBL1222314 | CHEMBL1222314 | |
| 0.031 | 0.652 | 0.173 | CF transmembrane conductance regulator agonist | 0.173 0.043 CHEMBL3706475 0.139 0.097 CHEMBL1222314 | CHEMBL3706475 | |
| 0.012 | 0.633 | 0.091 | GABA B receptor agonist | 0.082 0.037 CHEMBL3706466 0.079 0.045 CHEMBL3706475 0.09 0.026 CHEMBL3706478 0.091 0.025 CHEMBL1222314 | CHEMBL1222314 | |
| 0.044 | 0.666 | 0.258 | Apoptosis agonist | 0.258 0.206 CHEMBL3706465 | CHEMBL3706465 | |
| 0.005 | 0.631 | 0.055 | Beta 1 adrenoreceptor antagonist | 0.053 0.042 CHEMBL3706475 0.055 0.04 CHEMBL3706478 0.051 0.045 CHEMBL1222314 | CHEMBL3706478 | |
| 0.003 | 0.633 | 0.064 | Angiotensin AT1 receptor antagonist | 0.05 0.018 CHEMBL3706466 0.051 0.016 CHEMBL3706478 0.064 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.635 | 0.06 | Angiotensin II receptor antagonist | 0.036 0.02 CHEMBL3706466 0.038 0.017 CHEMBL3706478 0.06 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.648 | 0.111 | Potassium channel (Ca-activated) activator | 0.111 0.047 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.651 | 0.41 | Alpha-glucosidase inhibitor | 0.41 0.11 CHEMBL1222314 | CHEMBL1222314 | |
| 0.032 | 0.671 | 0.265 | Superoxide dismutase inhibitor | 0.191 0.128 CHEMBL3706466 0.227 0.091 CHEMBL3706475 0.182 0.139 CHEMBL3706478 0.265 0.066 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.645 | 0.118 | Nicotinic acid receptor agonist | 0.118 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.649 | 0.085 | Sphingosine 1-phosphate receptor 4 agonist | 0.062 0.052 CHEMBL3706466 0.082 0.035 CHEMBL3706478 0.085 0.034 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.652 | 0.078 | NMDA receptor antagonist | 0.078 0.068 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.654 | 0.078 | Dihydroorotase inhibitor | 0.078 0.009 CHEMBL1222314 | CHEMBL1222314 | |
| 0.023 | 0.672 | 0.086 | D-Ala-D-Ala ligase inhibitor | 0.086 0.052 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.654 | 0.284 | Protein kinase (CK2) inhibitor | 0.284 0.008 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.665 | 0.36 | Thioredoxin glutathione reductase inhibitor | 0.36 0.073 CHEMBL1222314 | CHEMBL1222314 | |
| 0.017 | 0.669 | 0.115 | TRPA1 agonist | 0.115 0.064 CHEMBL1222314 | CHEMBL1222314 | |
| 0.002 | 0.654 | 0.048 | Kainate receptor 2 antagonist | 0.048 0.017 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.656 | 0.052 | Trypsin I inhibitor | 0.052 0.011 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.662 | 0.09 | Sirtuin 1 inhibitor | 0.09 0.028 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.668 | 0.215 | MAP kinase kinase 2 inhibitor | 0.215 0.072 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.67 | 0.057 | Potassium channel intermediate-conductance Ca-activated blocker | 0.057 0.049 CHEMBL1222314 | CHEMBL1222314 | |
| 0.001 | 0.664 | 0.014 | Egl nine homolog 3 inhibitor | 0.014 0.006 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.676 | 0.332 | Beta lactamase inhibitor | 0.332 0.122 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.674 | 0.107 | Glutamate (mGluR1) antagonist | 0.107 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.679 | 0.064 | Collagenase 3 inhibitor | 0.064 0.036 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.685 | 0.11 | Topoisomerase II inhibitor | 0.11 0.077 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.681 | 0.1 | Xanthine dehydrogenase inhibitor | 0.1 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.686 | 0.226 | Alcohol dehydrogenase inhibitor | 0.226 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.695 | 0.188 | 5 Hydroxytryptamine 1E antagonist | 0.188 0.145 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.686 | 0.058 | Glutamate (mGluR1a) antagonist | 0.058 0.016 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.687 | 0.256 | Protein kinase (CK2) alpha inhibitor | 0.256 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.016 | 0.7 | 0.189 | Interleukin 1 antagonist | 0.189 0.038 CHEMBL1222314 | CHEMBL1222314 | |
| 0.071 | 0.757 | 0.165 | 5 Hydroxytryptamine 3E antagonist | 0.165 0.154 CHEMBL3706475 0.165 0.152 CHEMBL1222314 | CHEMBL1222314 | |
| 0.038 | 0.725 | 0.334 | GABA C receptor rho-3 antagonist | 0.224 0.18 CHEMBL3706465 0.228 0.176 CHEMBL3706466 0.325 0.1 CHEMBL3706475 0.334 0.095 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.694 | 0.089 | Stem cell growth factor agonist | 0.089 0.056 CHEMBL1222314 | CHEMBL1222314 | |
| 0.029 | 0.718 | 0.37 | Hypoglycemic | 0.37 0.033 CHEMBL3706478 0.281 0.06 CHEMBL1222314 | CHEMBL3706478 | |
| 0.005 | 0.694 | 0.086 | Potassium channel (Voltage-sensitive) activator | 0.086 0.075 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.693 | 0.039 | Stearoyl-CoA desaturase inhibitor | 0.039 0.038 CHEMBL3706478 | CHEMBL3706478 | |
| 0.003 | 0.697 | 0.02 | Kainate receptor 5 antagonist | 0.02 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.703 | 0.147 | Sphingosine 1-phosphate receptor 2 antagonist | 0.132 0.069 CHEMBL3706466 0.114 0.112 CHEMBL3706475 0.119 0.099 CHEMBL3706478 0.147 0.044 CHEMBL1222314 | CHEMBL1222314 | |
| 0.019 | 0.717 | 0.148 | GABA C receptor rho-2 antagonist | 0.148 0.076 CHEMBL1222314 | CHEMBL1222314 | |
| 0.001 | 0.702 | 0.015 | Egl nine homolog 1 inhibitor | 0.015 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.709 | 0.106 | Dihydroorotate dehydrogenase inhibitor | 0.106 0.01 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.718 | 0.301 | 12-Lipoxygenase inhibitor | 0.193 0.16 CHEMBL3706466 0.199 0.153 CHEMBL3706478 0.301 0.079 CHEMBL1222314 | CHEMBL1222314 | |
| 0.002 | 0.711 | 0.032 | Sirtuin 2 inhibitor | 0.032 0.023 CHEMBL1222314 | CHEMBL1222314 | |
| 0.013 | 0.722 | 0.141 | Factor IXa inhibitor | 0.141 0.004 CHEMBL3706478 | CHEMBL3706478 | |
| 0.008 | 0.72 | 0.044 | Glutamate (mGluR4) antagonist | 0.044 0.03 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.719 | 0.251 | Aryl hydrocarbon receptor agonist | 0.251 0.078 CHEMBL1222314 | CHEMBL1222314 | |
| 0.008 | 0.723 | 0.29 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.157 0.134 CHEMBL3706466 0.29 0.067 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.72 | 0.019 | Calcium-sensing receptor antagonist | 0.019 0.009 CHEMBL3706478 | CHEMBL3706478 | |
| 0.006 | 0.726 | 0.07 | Histone deacetylase SIRT3 inhibitor | 0.07 0.028 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.729 | 0.109 | Nicotinic acid receptor 2 agonist | 0.109 0.005 CHEMBL1222314 | CHEMBL1222314 | |
| 0.014 | 0.74 | 0.174 | Sphingosine 1-phosphate receptor 5 antagonist | 0.146 0.069 CHEMBL3706466 0.174 0.029 CHEMBL1222314 | CHEMBL1222314 | |
| 0.023 | 0.751 | 0.111 | ABCA1 expression enhancer | 0.111 0.038 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.735 | 0.194 | Prostaglandin antagonist | 0.046 0.044 CHEMBL3706478 0.194 0.007 CHEMBL1222314 | CHEMBL1222314 | |
| 0.012 | 0.75 | 0.229 | Transcription factor STAT3 inhibitor | 0.229 0.102 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.749 | 0.405 | Dual specificity phosphatase 3 inhibitor | 0.405 0.013 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.754 | 0.538 | Cyclooxygenase 1 inhibitor | 0.538 0.005 CHEMBL3706475 0.164 0.05 CHEMBL1222314 | CHEMBL3706475 | |
| 0.005 | 0.761 | 0.475 | Prostaglandin dehydrogenase inhibitor | 0.475 0.047 CHEMBL1222314 | CHEMBL1222314 | |
| 0.022 | 0.78 | 0.926 | Immunomodulator | 0.283 0.092 CHEMBL3706471 0.565 0.015 CHEMBL3706468 0.597 0.012 CHEMBL3706472 0.926 0.003 CHEMBL3706475 | CHEMBL3706475 | |
| 0.008 | 0.768 | 0.079 | Trypsin inhibitor | 0.079 0.027 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.771 | 0.501 | DNA polymerase beta inhibitor | 0.501 0.087 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.773 | 0.487 | DNA directed DNA polymerase inhibitor | 0.313 0.155 CHEMBL3706478 0.487 0.086 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.776 | 0.177 | Polo-like kinase-3 inhibitor | 0.177 0.059 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.777 | 0.147 | Thiol protease inhibitor | 0.147 0.072 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.783 | 0.16 | Focal adhesion kinase 2 inhibitor | 0.16 0.115 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.785 | 0.169 | Heat shock protein 90 alpha antagonist | 0.169 0.071 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.786 | 0.053 | Purinergic P2Y2 antagonist | 0.053 0.009 CHEMBL1222314 | CHEMBL1222314 | |
| 0.007 | 0.786 | 0.301 | I kappa B kinase epsilon inhibitor | 0.301 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.792 | 0.194 | Thyroid hormone beta antagonist | 0.194 0.16 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.787 | 0.133 | GABA receptor agonist | 0.133 0.046 CHEMBL1222314 | CHEMBL1222314 | |
| 0.011 | 0.793 | 0.207 | Thyroid hormone antagonist | 0.207 0.156 CHEMBL1222314 | CHEMBL1222314 | |
| 0.018 | 0.802 | 0.249 | MAP kinase 1 inhibitor | 0.249 0.235 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.789 | 0.31 | Mcl-1 antagonist | 0.31 0.021 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.796 | 0.376 | Dual specificity phosphatase inhibitor | 0.208 0.051 CHEMBL3706478 0.376 0.017 CHEMBL1222314 | CHEMBL1222314 | |
| 0.015 | 0.802 | 0.415 | Transcription factor inhibitor | 0.259 0.18 CHEMBL3706466 0.415 0.104 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.792 | 0.02 | Factor IX inhibitor | 0.02 0.012 CHEMBL3706478 | CHEMBL3706478 | |
| 0.009 | 0.797 | 0.391 | Thrombolytic | 0.282 0.027 CHEMBL3706471 0.31 0.022 CHEMBL3706472 0.391 0.012 CHEMBL3706475 | CHEMBL3706475 | |
| 0.053 | 0.842 | 0.352 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.305 0.206 CHEMBL3706475 0.352 0.149 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.797 | 0.274 | Cyclooxygenase inhibitor | 0.2 0.042 CHEMBL3706466 0.274 0.022 CHEMBL3706475 0.168 0.058 CHEMBL1222314 | CHEMBL3706475 | |
| 0.016 | 0.809 | 0.18 | Histone acetyltransferase inhibitor | 0.18 0.099 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.809 | 0.394 | Streptokinase A inhibitor | 0.394 0.049 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.805 | 0.071 | Sphingosine 1-phosphate receptor 1 antagonist | 0.071 0.018 CHEMBL3706478 0.056 0.037 CHEMBL1222314 | CHEMBL3706478 | |
| 0.006 | 0.81 | 0.468 | Uric acid excretion stimulant | 0.091 0.063 CHEMBL3706478 0.468 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.017 | 0.825 | 0.224 | Insulysin inhibitor | 0.224 0.124 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.822 | 0.067 | Nicotinic acid receptor 1 agonist | 0.067 0.014 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.821 | 0.137 | CDC-like kinase 4 inhibitor | 0.137 0.112 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.826 | 0.086 | Sphingosine 1-phosphate receptor antagonist | 0.086 0.035 CHEMBL3706478 0.074 0.059 CHEMBL1222314 | CHEMBL3706478 | |
| 0.005 | 0.833 | 0.319 | Anticoagulant | 0.198 0.054 CHEMBL3706471 0.202 0.052 CHEMBL3706472 0.319 0.025 CHEMBL3706475 | CHEMBL3706475 | |
| 0.007 | 0.851 | 0.146 | Amyloid beta precursor protein antagonist | 0.146 0.106 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.848 | 0.249 | Calpain inhibitor | 0.249 0.066 CHEMBL1222314 | CHEMBL1222314 | |
| 0.004 | 0.85 | 0.276 | Prostaglandin E2 antagonist | 0.276 0.004 CHEMBL1222314 | CHEMBL1222314 | |
| 0.001 | 0.853 | 0.062 | AMPA receptor antagonist | 0.062 0.024 CHEMBL1222314 | CHEMBL1222314 | |
| 0.027 | 0.885 | 0.113 | Factor V inhibitor | 0.106 0.057 CHEMBL3706471 0.113 0.046 CHEMBL3706472 | CHEMBL3706472 | |
| 0.004 | 0.866 | 0.103 | Cyclooxygenase 2 inhibitor | 0.103 0.101 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.865 | 0.255 | Calpain 2 inhibitor | 0.218 0.173 CHEMBL3706478 0.255 0.146 CHEMBL1222314 | CHEMBL1222314 | |
| 0.003 | 0.867 | 0.039 | AMPA 2 receptor antagonist | 0.039 0.015 CHEMBL1222314 | CHEMBL1222314 | |
| 0.006 | 0.874 | 0.198 | Transcription factor STAT inhibitor | 0.198 0.142 CHEMBL1222314 | CHEMBL1222314 | |
| 0.009 | 0.881 | 0.581 | Cyclophilin D inhibitor | 0.378 0.103 CHEMBL3706474 0.581 0.031 CHEMBL3706475 0.42 0.08 CHEMBL3706478 0.355 0.118 CHEMBL1222314 | CHEMBL3706475 | |
| 0.051 | 0.926 | 0.39 | Calcium channel L-type activator | 0.39 0.088 CHEMBL3706478 | CHEMBL3706478 | |
| 0.004 | 0.881 | 0.123 | HIV-1 reverse transcriptase inhibitor | 0.123 0.021 CHEMBL3706475 | CHEMBL3706475 | |
| 0.004 | 0.896 | 0.26 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.26 0.063 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.897 | 0.223 | Death-associated protein kinase 3 inhibitor | 0.223 0.063 CHEMBL1222314 | CHEMBL1222314 | |
| 0.01 | 0.907 | 0.044 | Parathyroid hormone antagonist | 0.044 0.035 CHEMBL3706465 | CHEMBL3706465 | |
| 0.004 | 0.904 | 0.235 | Dyrk kinase inhibitor | 0.235 0.079 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.908 | 0.181 | Interleukin antagonist | 0.179 0.097 CHEMBL3706471 0.181 0.096 CHEMBL3706472 | CHEMBL3706472 | |
| 0.009 | 0.914 | 0.151 | Histone deacetylase SIRT1 inhibitor | 0.151 0.06 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.924 | 0.216 | DNA directed RNA polymerase inhibitor | 0.216 0.012 CHEMBL3706475 | CHEMBL3706475 | |
| 0.004 | 0.937 | 0.118 | Glutamate receptor antagonist | 0.118 0.075 CHEMBL1222314 | CHEMBL1222314 | |
| 0.005 | 0.94 | 0.239 | Antiobesity | 0.239 0.167 CHEMBL3706474 | CHEMBL3706474 | |
| 0.004 | 0.943 | 0.115 | DNA gyrase inhibitor | 0.115 0.014 CHEMBL1222314 | CHEMBL1222314 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |