| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.981 | 0 | 0.995 | Angiotensin AT1 receptor antagonist | 0.145 0.002 CHEMBL4525751 0.639 0.001 CHEMBL4525752 0.988 0 CHEMBL308493 0.782 0 CHEMBL4525754 0.67 0.001 CHEMBL4525753 0.995 0 CHEMBL907 | CHEMBL907 | |
| 0.976 | 0 | 0.992 | Angiotensin II receptor antagonist | 0.174 0.002 CHEMBL4525751 0.849 0 CHEMBL4525752 0.984 0 CHEMBL308493 0.786 0 CHEMBL4525754 0.87 0 CHEMBL4525753 0.992 0 CHEMBL907 | CHEMBL907 | |
| 0.805 | 0.001 | 0.986 | Angiotensin AT2 receptor antagonist | 0.276 0.002 CHEMBL4525751 0.413 0.002 CHEMBL4525752 0.986 0.001 CHEMBL308493 0.622 0.001 CHEMBL4525754 0.34 0.002 CHEMBL4525753 0.962 0.001 CHEMBL907 | CHEMBL308493 | |
| 0.718 | 0.005 | 0.72 | Cardiotonic | 0.32 0.049 CHEMBL4525751 0.631 0.006 CHEMBL4525752 0.481 0.017 CHEMBL308493 0.72 0.005 CHEMBL4525754 0.636 0.006 CHEMBL4525753 0.396 0.03 CHEMBL907 | CHEMBL4525754 | |
| 0.689 | 0.001 | 0.959 | Angiotensin AT1A receptor antagonist | 0.195 0.002 CHEMBL4525751 0.292 0.002 CHEMBL4525752 0.959 0.001 CHEMBL308493 0.413 0.002 CHEMBL4525754 0.261 0.002 CHEMBL4525753 0.937 0.001 CHEMBL907 | CHEMBL308493 | |
| 0.609 | 0.003 | 0.609 | NADPH oxidase inhibitor | 0.133 0.068 CHEMBL4525751 0.31 0.011 CHEMBL4525752 0.287 0.014 CHEMBL308493 0.328 0.009 CHEMBL4525754 0.155 0.051 CHEMBL4525753 0.571 0.004 CHEMBL907 | ||
| 0.558 | 0.001 | 0.993 | Angiotensin AT1B receptor antagonist | 0.062 0.002 CHEMBL4525751 0.121 0.002 CHEMBL4525752 0.961 0 CHEMBL308493 0.142 0.001 CHEMBL4525754 0.116 0.002 CHEMBL4525753 0.993 0 CHEMBL907 | CHEMBL907 | |
| 0.521 | 0.022 | 0.577 | Histamine release inhibitor | 0.305 0.121 CHEMBL4525751 0.45 0.05 CHEMBL4525752 0.285 0.132 CHEMBL308493 0.534 0.019 CHEMBL4525754 0.268 0.142 CHEMBL4525753 0.577 0.012 CHEMBL907 | CHEMBL907 | |
| 0.497 | 0.033 | 0.706 | 5 Hydroxytryptamine release inhibitor | 0.462 0.046 CHEMBL4525752 0.437 0.058 CHEMBL308493 0.409 0.072 CHEMBL4525754 0.43 0.061 CHEMBL4525753 0.706 0.004 CHEMBL907 | CHEMBL907 | |
| 0.477 | 0.037 | 0.525 | Calcium channel L-type activator | 0.388 0.089 CHEMBL4525751 0.525 0.019 CHEMBL4525752 0.462 0.045 CHEMBL4525754 | CHEMBL4525752 | |
| 0.424 | 0.013 | 0.424 | Growth hormone agonist | 0.155 0.083 CHEMBL4525751 0.323 0.028 CHEMBL4525752 0.159 0.08 CHEMBL308493 0.397 0.016 CHEMBL4525754 0.301 0.032 CHEMBL4525753 0.185 0.065 CHEMBL907 | ||
| 0.34 | 0.13 | 0.422 | Cyclophilin D inhibitor | 0.398 0.092 CHEMBL4525751 0.252 0.211 CHEMBL4525752 0.422 0.079 CHEMBL4525754 | CHEMBL4525754 | |
| 0.219 | 0.01 | 0.329 | Uric acid excretion stimulant | 0.154 0.022 CHEMBL4525751 0.144 0.025 CHEMBL4525752 0.095 0.058 CHEMBL308493 0.17 0.018 CHEMBL4525754 0.138 0.028 CHEMBL4525753 0.329 0.005 CHEMBL907 | CHEMBL907 | |
| 0.214 | 0.011 | 0.418 | Alcohol dehydrogenase inhibitor | 0.104 0.048 CHEMBL4525752 0.229 0.009 CHEMBL308493 0.243 0.008 CHEMBL4525754 0.117 0.037 CHEMBL4525753 0.418 0.004 CHEMBL907 | CHEMBL907 | |
| 0.189 | 0.009 | 0.203 | Phosphodiesterase 3A inhibitor | 0.123 0.021 CHEMBL4525752 0.203 0.008 CHEMBL308493 0.143 0.017 CHEMBL4525754 0.079 0.057 CHEMBL4525753 0.201 0.008 CHEMBL907 | CHEMBL308493 | |
| 0.178 | 0.019 | 0.178 | Mediator release inhibitor | 0.151 0.028 CHEMBL4525752 0.136 0.035 CHEMBL4525754 | ||
| 0.153 | 0.012 | 0.173 | Peroxisome proliferator-activated receptor gamma agonist | 0.074 0.045 CHEMBL4525751 0.095 0.031 CHEMBL4525752 0.135 0.016 CHEMBL308493 0.154 0.012 CHEMBL4525754 0.067 0.052 CHEMBL4525753 0.173 0.009 CHEMBL907 | CHEMBL907 | |
| 0.234 | 0.099 | 0.234 | Gastrin inhibitor | |||
| 0.18 | 0.054 | 0.18 | Diuretic | 0.124 0.1 CHEMBL4525754 | ||
| 0.119 | 0.004 | 0.119 | Urate transporter 1 inhibitor | 0.044 0.022 CHEMBL4525752 0.054 0.017 CHEMBL4525754 0.037 0.029 CHEMBL4525753 0.089 0.006 CHEMBL907 | ||
| 0.198 | 0.102 | 0.198 | Platelet antagonist | 0.172 0.124 CHEMBL4525751 0.162 0.133 CHEMBL4525752 0.165 0.13 CHEMBL4525754 | ||
| 0.128 | 0.043 | 0.148 | Xanthine oxidase inhibitor | 0.107 0.055 CHEMBL4525752 0.118 0.048 CHEMBL4525754 0.148 0.035 CHEMBL4525753 0.085 0.081 CHEMBL907 | CHEMBL4525753 | |
| 0.082 | 0.008 | 0.186 | Nicotinic acid receptor 2 agonist | 0.046 0.016 CHEMBL4525752 0.117 0.005 CHEMBL308493 0.045 0.017 CHEMBL4525754 0.057 0.012 CHEMBL4525753 0.186 0.004 CHEMBL907 | CHEMBL907 | |
| 0.109 | 0.047 | 0.394 | Phosphodiesterase 7B inhibitor | 0.394 0.003 CHEMBL308493 0.085 0.077 CHEMBL4525754 0.389 0.003 CHEMBL907 | CHEMBL308493 | |
| 0.089 | 0.031 | 0.146 | Sphingosine 1-phosphate receptor 4 agonist | 0.146 0.009 CHEMBL308493 0.096 0.027 CHEMBL907 | CHEMBL308493 | |
| 0.056 | 0.012 | 0.122 | Nicotinic acid receptor agonist | 0.052 0.014 CHEMBL308493 0.122 0.004 CHEMBL907 | CHEMBL907 | |
| 0.055 | 0.012 | 0.055 | Acid-sensing ion channel blocker | 0.053 0.013 CHEMBL4525752 0.052 0.015 CHEMBL4525754 0.052 0.015 CHEMBL4525753 | ||
| 0.045 | 0.011 | 0.192 | Leukotriene D4 antagonist | 0.025 0.019 CHEMBL4525752 0.159 0.004 CHEMBL308493 0.026 0.018 CHEMBL4525754 0.192 0.004 CHEMBL907 | CHEMBL907 | |
| 0.13 | 0.096 | 0.203 | Hemostatic | 0.203 0.031 CHEMBL907 | CHEMBL907 | |
| 0.073 | 0.042 | 0.073 | Leukotriene synthesis inhibitor | 0.063 0.052 CHEMBL4525752 | ||
| 0.067 | 0.036 | 0.111 | Prostaglandin F2 alpha antagonist | 0.059 0.049 CHEMBL4525752 0.111 0.008 CHEMBL4525754 0.066 0.037 CHEMBL907 | CHEMBL4525754 | |
| 0.096 | 0.069 | 0.143 | Bronchodilator | 0.143 0.034 CHEMBL4525752 0.106 0.057 CHEMBL4525754 | CHEMBL4525752 | |
| 0.07 | 0.044 | 0.07 | Potassium channel large-conductance Ca-activated activator | 0.064 0.052 CHEMBL4525754 | ||
| 0.066 | 0.044 | 0.115 | Leukotriene antagonist | 0.058 0.054 CHEMBL4525752 0.115 0.016 CHEMBL907 | CHEMBL907 | |
| 0.198 | 0.178 | 0.226 | Vasodilator, peripheral | 0.226 0.148 CHEMBL4525754 | CHEMBL4525754 | |
| 0.045 | 0.029 | 0.045 | Phosphodiesterase 3B inhibitor | 0.041 0.035 CHEMBL4525754 | ||
| 0.035 | 0.021 | 0.035 | Growth hormone releasing factor agonist | 0.032 0.024 CHEMBL4525754 | ||
| 0.068 | 0.057 | 0.071 | Phosphodiesterase VIII inhibitor | 0.071 0.051 CHEMBL308493 0.067 0.061 CHEMBL907 | CHEMBL308493 | |
| 0.052 | 0.041 | 0.06 | Maillard reaction inhibitor | 0.06 0.035 CHEMBL4525752 0.048 0.045 CHEMBL4525753 | CHEMBL4525752 | |
| 0.06 | 0.052 | 0.06 | Phosphodiesterase III inhibitor | 0.057 0.055 CHEMBL4525754 0.06 0.052 CHEMBL907 | ||
| 0.026 | 0.019 | 0.045 | Nicotinic acid receptor 2 antagonist | 0.045 0.004 CHEMBL907 | CHEMBL907 | |
| 0.022 | 0.017 | 0.029 | Bombesin agonist | 0.021 0.018 CHEMBL308493 0.029 0.009 CHEMBL907 | CHEMBL907 | |
| 0.018 | 0.014 | 0.025 | Bombesin 3 receptor agonist | 0.018 0.015 CHEMBL308493 0.025 0.008 CHEMBL907 | CHEMBL907 | |
| 0.052 | 0.055 | 0.078 | Leukotriene C antagonist | 0.054 0.048 CHEMBL308493 0.078 0.009 CHEMBL907 | CHEMBL907 | |
| 0.035 | 0.038 | 0.052 | Factor XIa inhibitor | 0.052 0.017 CHEMBL907 | CHEMBL907 | |
| 0.055 | 0.059 | 0.078 | Nitric oxide donor | 0.078 0.024 CHEMBL4525751 0.064 0.041 CHEMBL4525754 | CHEMBL4525751 | |
| 0.042 | 0.049 | 0.115 | Prostaglandin antagonist | 0.055 0.035 CHEMBL4525754 0.115 0.014 CHEMBL907 | CHEMBL907 | |
| 0.025 | 0.042 | 0.162 | Glutamate (mGluR group II) agonist | 0.13 0.005 CHEMBL308493 0.162 0.004 CHEMBL907 | CHEMBL907 | |
| 0.021 | 0.041 | 0.152 | Glutamate (mGluR2) agonist | 0.123 0.005 CHEMBL308493 0.152 0.004 CHEMBL907 | CHEMBL907 | |
| 0.106 | 0.127 | 0.146 | Thrombolytic | 0.146 0.085 CHEMBL4525751 | CHEMBL4525751 | |
| 0.033 | 0.056 | 0.054 | Leukotriene C4 antagonist | 0.054 0.008 CHEMBL907 | CHEMBL907 | |
| 0.029 | 0.06 | 0.041 | Adenosine deaminase inhibitor | 0.041 0.039 CHEMBL4525754 | CHEMBL4525754 | |
| 0.015 | 0.052 | 0.042 | Endothelin receptor antagonist | 0.042 0.012 CHEMBL907 | CHEMBL907 | |
| 0.01 | 0.053 | 0.022 | Endothelin A receptor antagonist | 0.022 0.014 CHEMBL907 | CHEMBL907 | |
| 0.026 | 0.075 | 0.036 | Nicotinic acid receptor 1 agonist | 0.036 0.035 CHEMBL907 | CHEMBL907 | |
| 0.038 | 0.088 | 0.063 | Sphingosine kinase 2 inhibitor | 0.055 0.038 CHEMBL308493 0.063 0.028 CHEMBL907 | CHEMBL907 | |
| 0.04 | 0.093 | 0.051 | Sphingosine 1-phosphate receptor 5 agonist | 0.051 0.043 CHEMBL907 | CHEMBL907 | |
| 0.011 | 0.067 | 0.026 | Leukotriene B4 receptor 1 antagonist | 0.026 0.021 CHEMBL907 | CHEMBL907 | |
| 0.023 | 0.081 | 0.061 | Oleamide hydrolase inhibitor | 0.061 0.02 CHEMBL308493 0.049 0.028 CHEMBL907 | CHEMBL308493 | |
| 0.036 | 0.094 | 0.052 | Autotaxin inhibitor | 0.052 0.037 CHEMBL907 | CHEMBL907 | |
| 0.008 | 0.068 | 0.019 | Nicotinic acid receptor 1 antagonist | 0.019 0.01 CHEMBL907 | CHEMBL907 | |
| 0.015 | 0.077 | 0.029 | CXC chemokine 3 receptor antagonist | 0.029 0.025 CHEMBL907 | CHEMBL907 | |
| 0.128 | 0.199 | 0.17 | Cyclic AMP phosphodiesterase inhibitor | 0.17 0.122 CHEMBL4525754 | CHEMBL4525754 | |
| 0.03 | 0.113 | 0.053 | Leukotriene B4 antagonist | 0.053 0.039 CHEMBL907 | CHEMBL907 | |
| 0.018 | 0.102 | 0.087 | Glutamate (mGluR group II) antagonist | 0.087 0.005 CHEMBL907 | CHEMBL907 | |
| 0.032 | 0.125 | 0.108 | Bombesin 3 receptor antagonist | 0.105 0.01 CHEMBL308493 0.108 0.01 CHEMBL907 | CHEMBL907 | |
| 0.004 | 0.102 | 0.039 | Kainate receptor 1 antagonist | 0.039 0.007 CHEMBL907 | CHEMBL907 | |
| 0.016 | 0.119 | 0.077 | AMPA receptor antagonist | 0.047 0.034 CHEMBL308493 0.077 0.018 CHEMBL907 | CHEMBL907 | |
| 0.059 | 0.166 | 0.111 | DNA polymerase I inhibitor | 0.111 0.076 CHEMBL4525751 | CHEMBL4525751 | |
| 0.05 | 0.159 | 0.088 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.088 0.051 CHEMBL907 | CHEMBL907 | |
| 0.008 | 0.122 | 0.023 | Leukotriene B4 receptor 2 antagonist | 0.023 0.014 CHEMBL907 | CHEMBL907 | |
| 0.025 | 0.142 | 0.069 | Phosphodiesterase VII inhibitor | 0.069 0.036 CHEMBL907 | CHEMBL907 | |
| 0.012 | 0.135 | 0.031 | Carnitine palmitoyltransferase 1 inhibitor | 0.031 0.03 CHEMBL907 | CHEMBL907 | |
| 0.017 | 0.144 | 0.061 | Prostaglandin E2 antagonist | 0.061 0.028 CHEMBL907 | CHEMBL907 | |
| 0.024 | 0.157 | 0.042 | Glucagon-like peptide 1 receptor antagonist | 0.042 0.023 CHEMBL907 | CHEMBL907 | |
| 0.027 | 0.162 | 0.048 | Factor IXa inhibitor | 0.048 0.04 CHEMBL4525752 | CHEMBL4525752 | |
| 0.025 | 0.166 | 0.054 | Glutamate (mGluR group III) antagonist | 0.054 0.017 CHEMBL907 | CHEMBL907 | |
| 0.014 | 0.165 | 0.054 | Prostaglandin EP2 antagonist | 0.054 0.046 CHEMBL4525754 | CHEMBL4525754 | |
| 0.148 | 0.302 | 0.331 | Interleukin 2 agonist | 0.331 0.055 CHEMBL4525751 | CHEMBL4525751 | |
| 0.007 | 0.17 | 0.062 | Glutamate (mGluR2) antagonist | 0.062 0.006 CHEMBL907 | CHEMBL907 | |
| 0.018 | 0.182 | 0.075 | Phosphodiesterase 4C inhibitor | 0.075 0.024 CHEMBL308493 0.073 0.025 CHEMBL907 | CHEMBL308493 | |
| 0.007 | 0.195 | 0.051 | Kainate receptor antagonist | 0.051 0.02 CHEMBL907 | CHEMBL907 | |
| 0.019 | 0.226 | 0.084 | Phosphodiesterase 4D inhibitor | 0.075 0.051 CHEMBL308493 0.084 0.045 CHEMBL907 | CHEMBL907 | |
| 0.028 | 0.237 | 0.066 | Phosphodiesterase 1A inhibitor | 0.062 0.036 CHEMBL308493 0.066 0.03 CHEMBL907 | CHEMBL907 | |
| 0.014 | 0.232 | 0.096 | Glutamate (mGluR) agonist | 0.063 0.042 CHEMBL308493 0.096 0.024 CHEMBL907 | CHEMBL907 | |
| 0.007 | 0.238 | 0.089 | AMPA 2 receptor antagonist | 0.058 0.009 CHEMBL308493 0.089 0.006 CHEMBL907 | CHEMBL907 | |
| 0.031 | 0.278 | 0.058 | Phosphodiesterase 1C inhibitor | 0.058 0.053 CHEMBL907 | CHEMBL907 | |
| 0.014 | 0.273 | 0.152 | Selectin antagonist | 0.152 0.018 CHEMBL4525751 | CHEMBL4525751 | |
| 0.054 | 0.332 | 0.149 | Hypolipemic | 0.149 0.137 CHEMBL4525754 | CHEMBL4525754 | |
| 0.013 | 0.295 | 0.153 | Glutamate receptor agonist | 0.153 0.017 CHEMBL907 | CHEMBL907 | |
| 0.004 | 0.293 | 0.028 | Kainate receptor 5 antagonist | 0.018 0.017 CHEMBL308493 0.028 0.01 CHEMBL907 | CHEMBL907 | |
| 0.066 | 0.355 | 0.274 | Antioxidant | 0.274 0.072 CHEMBL4525751 | CHEMBL4525751 | |
| 0.059 | 0.356 | 0.22 | Hepatoprotectant | 0.22 0.054 CHEMBL4525751 | CHEMBL4525751 | |
| 0.011 | 0.326 | 0.085 | AMPA 4 receptor antagonist | 0.085 0.006 CHEMBL907 | CHEMBL907 | |
| 0.015 | 0.331 | 0.044 | Antibiotic Aminoglycoside-like | 0.044 0.017 CHEMBL4525751 | CHEMBL4525751 | |
| 0.004 | 0.324 | 0.032 | HMG CoA reductase inhibitor | 0.032 0.03 CHEMBL4525754 | CHEMBL4525754 | |
| 0.021 | 0.344 | 0.054 | Carbonic anhydrase II stimulant | 0.051 0.037 CHEMBL308493 0.054 0.031 CHEMBL907 | CHEMBL907 | |
| 0.072 | 0.398 | 0.271 | Hypoglycemic | 0.271 0.065 CHEMBL4525751 | CHEMBL4525751 | |
| 0.009 | 0.336 | 0.037 | Carbonic anhydrase I stimulant | 0.037 0.027 CHEMBL907 | CHEMBL907 | |
| 0.022 | 0.354 | 0.158 | Glutamate receptor antagonist | 0.158 0.046 CHEMBL907 | CHEMBL907 | |
| 0.024 | 0.364 | 0.072 | Peroxisome proliferator-activated receptor gamma antagonist | 0.072 0.047 CHEMBL907 | CHEMBL907 | |
| 0.017 | 0.361 | 0.064 | Glutamate (mGluR4) antagonist | 0.041 0.034 CHEMBL308493 0.064 0.012 CHEMBL907 | CHEMBL907 | |
| 0.033 | 0.42 | 0.121 | Electron transport complex I inhibitor | 0.121 0.046 CHEMBL4525752 0.116 0.052 CHEMBL4525753 | CHEMBL4525752 | |
| 0.004 | 0.406 | 0.035 | AMPA 3 receptor antagonist | 0.035 0.017 CHEMBL907 | CHEMBL907 | |
| 0.004 | 0.41 | 0.039 | Kainate receptor 4 antagonist | 0.032 0.013 CHEMBL308493 0.039 0.01 CHEMBL907 | CHEMBL907 | |
| 0.004 | 0.436 | 0.017 | Kainate receptor 3 antagonist | 0.017 0.012 CHEMBL907 | CHEMBL907 | |
| 0.029 | 0.469 | 0.255 | Immunostimulant | 0.255 0.094 CHEMBL4525751 | CHEMBL4525751 | |
| 0.003 | 0.511 | 0.035 | Kainate receptor 2 antagonist | 0.035 0.025 CHEMBL907 | CHEMBL907 | |
| 0.004 | 0.517 | 0.086 | NMDA receptor subunit 3B antagonist | 0.086 0.013 CHEMBL907 | CHEMBL907 | |
| 0.003 | 0.522 | 0.067 | NMDA receptor subunit 3A antagonist | 0.067 0.015 CHEMBL907 | CHEMBL907 | |
| 0.005 | 0.533 | 0.053 | Fibroblast growth factor 4 antagonist | 0.053 0.048 CHEMBL308493 | CHEMBL308493 | |
| 0.04 | 0.569 | 0.195 | Antithrombotic | 0.195 0.183 CHEMBL4525751 | CHEMBL4525751 | |
| 0.011 | 0.576 | 0.292 | Topoisomerase I inhibitor | 0.292 0.012 CHEMBL4525751 | CHEMBL4525751 | |
| 0.016 | 0.583 | 0.202 | I kappa B kinase epsilon inhibitor | 0.202 0.069 CHEMBL907 | CHEMBL907 | |
| 0.017 | 0.61 | 0.335 | Angiogenesis stimulant | 0.335 0.037 CHEMBL4525751 | CHEMBL4525751 | |
| 0.052 | 0.651 | 0.261 | Catenin beta inhibitor | 0.227 0.017 CHEMBL308493 0.261 0.009 CHEMBL907 | CHEMBL907 | |
| 0.022 | 0.621 | 0.145 | Nitric oxide antagonist | 0.145 0.1 CHEMBL4525751 | CHEMBL4525751 | |
| 0.015 | 0.625 | 0.203 | Free radical scavenger | 0.203 0.095 CHEMBL4525751 | CHEMBL4525751 | |
| 0.03 | 0.65 | 0.225 | Immunosuppressant | 0.225 0.171 CHEMBL4525751 | CHEMBL4525751 | |
| 0.02 | 0.717 | 0.293 | Antibacterial | 0.293 0.141 CHEMBL4525751 | CHEMBL4525751 | |
| 0.06 | 0.818 | 0.246 | Peptidyltransferase inhibitor | 0.246 0.054 CHEMBL4525751 | CHEMBL4525751 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |