| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.851 | 0.003 | 0.851 | Vasodilator, coronary | 0.457 0.022 CHEMBL1573 0.451 0.023 CHEMBL3544724 0.48 0.018 CHEMBL3544725 0.333 0.064 CHEMBL3544726 | ||
| 0.85 | 0.003 | 0.85 | Vasodilator, peripheral | 0.578 0.018 CHEMBL1573 0.606 0.015 CHEMBL3544724 0.634 0.012 CHEMBL3544725 0.226 0.148 CHEMBL3544726 | ||
| 0.808 | 0.001 | 0.808 | Calcium channel activator | 0.621 0.002 CHEMBL1573 0.594 0.002 CHEMBL3544724 0.602 0.002 CHEMBL3544725 0.636 0.002 CHEMBL3544726 | ||
| 0.801 | 0.003 | 0.801 | Calcium channel blocker | 0.578 0.004 CHEMBL1573 0.499 0.004 CHEMBL3544724 0.441 0.004 CHEMBL3544725 0.32 0.008 CHEMBL3544726 | ||
| 0.763 | 0.001 | 0.763 | Calcium antagonist | 0.342 0.004 CHEMBL1573 0.29 0.005 CHEMBL3544724 0.279 0.005 CHEMBL3544725 0.193 0.014 CHEMBL3544726 | ||
| 0.751 | 0.004 | 0.751 | Vasodilator | 0.447 0.016 CHEMBL1573 0.412 0.021 CHEMBL3544724 0.413 0.021 CHEMBL3544725 0.309 0.045 CHEMBL3544726 | ||
| 0.74 | 0.002 | 0.748 | Calcium channel L-type activator | 0.739 0.002 CHEMBL1573 0.72 0.002 CHEMBL3544724 0.748 0.002 CHEMBL3544725 0.691 0.003 CHEMBL3544726 | CHEMBL3544725 | |
| 0.717 | 0.002 | 0.717 | TRPA1 agonist | 0.177 0.017 CHEMBL1573 0.172 0.019 CHEMBL3544724 0.115 0.064 CHEMBL3544725 0.117 0.062 CHEMBL3544726 | ||
| 0.664 | 0.002 | 0.664 | Calcium channel L-type blocker | 0.463 0.003 CHEMBL1573 0.46 0.003 CHEMBL3544724 0.44 0.003 CHEMBL3544725 0.2 0.005 CHEMBL3544726 | ||
| 0.657 | 0.003 | 0.657 | Calcium channel (voltage-sensitive) blocker | 0.402 0.004 CHEMBL1573 0.327 0.005 CHEMBL3544724 0.254 0.01 CHEMBL3544725 0.125 0.051 CHEMBL3544726 | ||
| 0.592 | 0.008 | 0.592 | Cardiotonic | 0.195 0.124 CHEMBL1573 0.182 0.137 CHEMBL3544724 0.219 0.103 CHEMBL3544725 0.299 0.057 CHEMBL3544726 | ||
| 0.389 | 0.005 | 0.389 | Alpha 2b adrenoreceptor antagonist | 0.229 0.018 CHEMBL1573 0.133 0.049 CHEMBL3544724 | ||
| 0.458 | 0.098 | 0.56 | DNA polymerase beta inhibitor | 0.56 0.069 CHEMBL1573 0.548 0.073 CHEMBL3544724 0.36 0.135 CHEMBL3544725 0.306 0.162 CHEMBL3544726 | CHEMBL1573 | |
| 0.35 | 0.026 | 0.356 | Cyclic AMP phosphodiesterase inhibitor | 0.232 0.073 CHEMBL1573 0.247 0.065 CHEMBL3544724 0.356 0.024 CHEMBL3544725 | CHEMBL3544725 | |
| 0.309 | 0.006 | 0.309 | Adenylate kinase inhibitor | 0.166 0.021 CHEMBL1573 0.232 0.011 CHEMBL3544724 0.182 0.018 CHEMBL3544725 | ||
| 0.353 | 0.052 | 0.353 | Spasmolytic | |||
| 0.313 | 0.02 | 0.313 | Diuretic | |||
| 0.339 | 0.049 | 0.339 | Hypoxia-inducible factor 1 alpha inhibitor | 0.27 0.083 CHEMBL1573 0.279 0.077 CHEMBL3544724 0.328 0.053 CHEMBL3544725 0.181 0.177 CHEMBL3544726 | ||
| 0.316 | 0.032 | 0.316 | Platelet aggregation inhibitor | |||
| 0.288 | 0.007 | 0.288 | Alpha 2c adrenoreceptor antagonist | 0.182 0.022 CHEMBL1573 0.116 0.052 CHEMBL3544724 0.129 0.043 CHEMBL3544725 | ||
| 0.394 | 0.118 | 0.498 | DNA directed DNA polymerase inhibitor | 0.497 0.083 CHEMBL1573 0.498 0.083 CHEMBL3544724 0.359 0.134 CHEMBL3544725 0.233 0.202 CHEMBL3544726 | CHEMBL3544724 | |
| 0.278 | 0.003 | 0.278 | Aldosterone antagonist | 0.048 0.032 CHEMBL1573 | ||
| 0.27 | 0.005 | 0.27 | CF transmembrane conductance regulator agonist | 0.152 0.072 CHEMBL1573 0.132 0.113 CHEMBL3544724 | ||
| 0.269 | 0.007 | 0.269 | Neuropeptide Y1 antagonist | 0.257 0.008 CHEMBL1573 0.233 0.01 CHEMBL3544724 0.209 0.015 CHEMBL3544725 0.133 0.095 CHEMBL3544726 | ||
| 0.295 | 0.033 | 0.295 | 5 Hydroxytryptamine 1E antagonist | 0.234 0.092 CHEMBL1573 | ||
| 0.288 | 0.031 | 0.288 | P-glycoprotein inhibitor | 0.199 0.064 CHEMBL1573 0.177 0.082 CHEMBL3544724 0.157 0.106 CHEMBL3544725 | ||
| 0.361 | 0.125 | 0.437 | Transcription factor inhibitor | 0.437 0.095 CHEMBL1573 0.369 0.122 CHEMBL3544724 0.259 0.18 CHEMBL3544725 0.298 0.156 CHEMBL3544726 | CHEMBL1573 | |
| 0.312 | 0.095 | 0.375 | Thioredoxin glutathione reductase inhibitor | 0.375 0.067 CHEMBL1573 0.323 0.089 CHEMBL3544724 0.198 0.174 CHEMBL3544725 0.217 0.158 CHEMBL3544726 | CHEMBL1573 | |
| 0.29 | 0.081 | 0.306 | Interleukin 2 agonist | 0.257 0.111 CHEMBL1573 0.286 0.084 CHEMBL3544724 0.306 0.069 CHEMBL3544725 | CHEMBL3544725 | |
| 0.276 | 0.069 | 0.621 | Aryl hydrocarbon receptor agonist | 0.621 0.013 CHEMBL1573 0.521 0.022 CHEMBL3544724 0.31 0.058 CHEMBL3544725 0.219 0.092 CHEMBL3544726 | CHEMBL1573 | |
| 0.199 | 0.004 | 0.199 | Glycine receptor antagonist | 0.078 0.06 CHEMBL1573 | ||
| 0.215 | 0.023 | 0.307 | Mannose-6-phosphate isomerase inhibitor | 0.292 0.006 CHEMBL1573 0.307 0.005 CHEMBL3544724 0.262 0.01 CHEMBL3544725 0.192 0.035 CHEMBL3544726 | CHEMBL3544724 | |
| 0.343 | 0.151 | 0.492 | Caspase 9 stimulant | 0.492 0.063 CHEMBL1573 0.414 0.103 CHEMBL3544724 0.356 0.141 CHEMBL3544725 | CHEMBL1573 | |
| 0.284 | 0.104 | 0.317 | Transcription factor NF kappa B inhibitor | 0.264 0.118 CHEMBL1573 0.285 0.103 CHEMBL3544724 0.317 0.087 CHEMBL3544725 0.2 0.169 CHEMBL3544726 | CHEMBL3544725 | |
| 0.188 | 0.015 | 0.188 | Androgen antagonist | 0.1 0.047 CHEMBL1573 0.085 0.06 CHEMBL3544724 | ||
| 0.187 | 0.016 | 0.187 | Alpha 1b adrenoreceptor antagonist | |||
| 0.176 | 0.012 | 0.176 | Alpha 1d adrenoreceptor antagonist | |||
| 0.212 | 0.05 | 0.212 | Amyloid beta precursor protein antagonist | 0.146 0.106 CHEMBL1573 0.173 0.078 CHEMBL3544724 | ||
| 0.177 | 0.017 | 0.177 | Alpha 2a adrenoreceptor antagonist | |||
| 0.198 | 0.042 | 0.203 | Interleukin 6 antagonist | 0.203 0.039 CHEMBL1573 0.167 0.067 CHEMBL3544724 0.171 0.063 CHEMBL3544726 | CHEMBL1573 | |
| 0.222 | 0.072 | 0.222 | RNA-directed DNA polymerase inhibitor | 0.214 0.081 CHEMBL1573 0.221 0.073 CHEMBL3544724 0.216 0.078 CHEMBL3544725 0.168 0.157 CHEMBL3544726 | ||
| 0.264 | 0.115 | 0.264 | Apoptosis antagonist | 0.207 0.171 CHEMBL3544724 0.228 0.149 CHEMBL3544725 0.241 0.137 CHEMBL3544726 | ||
| 0.184 | 0.039 | 0.241 | GABA C receptor rho-2 antagonist | 0.241 0.014 CHEMBL1573 0.199 0.029 CHEMBL3544724 0.137 0.093 CHEMBL3544725 0.192 0.033 CHEMBL3544726 | CHEMBL1573 | |
| 0.164 | 0.019 | 0.164 | Beta glucuronidase inhibitor | 0.121 0.045 CHEMBL1573 0.119 0.047 CHEMBL3544724 | ||
| 0.204 | 0.068 | 0.273 | Non-steroidal antiinflammatory agent | 0.239 0.047 CHEMBL1573 0.273 0.035 CHEMBL3544724 0.229 0.052 CHEMBL3544725 0.246 0.044 CHEMBL3544726 | CHEMBL3544724 | |
| 0.137 | 0.005 | 0.137 | Mineralocorticoid receptor antagonist | |||
| 0.268 | 0.137 | 0.286 | Calpain 2 inhibitor | 0.286 0.123 CHEMBL1573 0.204 0.184 CHEMBL3544724 | CHEMBL1573 | |
| 0.219 | 0.089 | 0.219 | Platelet antagonist | |||
| 0.183 | 0.055 | 0.301 | Cytidine deaminase inhibitor | 0.301 0.019 CHEMBL1573 0.29 0.021 CHEMBL3544724 0.246 0.03 CHEMBL3544725 0.121 0.099 CHEMBL3544726 | CHEMBL1573 | |
| 0.225 | 0.098 | 0.252 | Interleukin agonist | 0.223 0.1 CHEMBL1573 0.252 0.077 CHEMBL3544724 0.229 0.095 CHEMBL3544725 | CHEMBL3544724 | |
| 0.148 | 0.022 | 0.21 | DOPA decarboxylase inhibitor | 0.178 0.011 CHEMBL1573 0.21 0.005 CHEMBL3544724 0.158 0.017 CHEMBL3544725 0.101 0.073 CHEMBL3544726 | CHEMBL3544724 | |
| 0.135 | 0.014 | 0.135 | Adenosine A3 receptor antagonist | 0.074 0.052 CHEMBL1573 | ||
| 0.182 | 0.068 | 0.314 | Sigma receptor agonist | 0.314 0.036 CHEMBL1573 0.273 0.044 CHEMBL3544724 0.138 0.094 CHEMBL3544725 0.209 0.059 CHEMBL3544726 | CHEMBL1573 | |
| 0.156 | 0.046 | 0.156 | Farnesoid X receptor antagonist | |||
| 0.279 | 0.17 | 0.462 | Alpha-glucosidase inhibitor | 0.462 0.092 CHEMBL1573 0.445 0.098 CHEMBL3544724 0.367 0.128 CHEMBL3544725 0.301 0.159 CHEMBL3544726 | CHEMBL1573 | |
| 0.24 | 0.134 | 0.24 | Antithrombotic | 0.193 0.186 CHEMBL3544724 | ||
| 0.144 | 0.039 | 0.171 | Sphingosine 1-phosphate receptor 4 antagonist | 0.17 0.019 CHEMBL1573 0.171 0.019 CHEMBL3544724 0.138 0.045 CHEMBL3544725 | CHEMBL3544724 | |
| 0.159 | 0.057 | 0.169 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.135 0.103 CHEMBL1573 0.169 0.044 CHEMBL3544724 0.138 0.097 CHEMBL3544725 | CHEMBL3544724 | |
| 0.126 | 0.024 | 0.126 | Interleukin 12 antagonist | 0.123 0.026 CHEMBL1573 0.112 0.037 CHEMBL3544724 0.1 0.054 CHEMBL3544725 0.102 0.05 CHEMBL3544726 | ||
| 0.196 | 0.095 | 0.196 | Nitric-oxide synthase stimulant | 0.193 0.101 CHEMBL1573 0.168 0.158 CHEMBL3544724 | ||
| 0.252 | 0.156 | 0.311 | Beta lactamase inhibitor | 0.311 0.13 CHEMBL1573 0.238 0.163 CHEMBL3544724 | CHEMBL1573 | |
| 0.149 | 0.052 | 0.189 | M18 aspartyl aminopeptidase inhibitor | 0.186 0.038 CHEMBL1573 0.189 0.037 CHEMBL3544724 0.113 0.077 CHEMBL3544725 | CHEMBL3544724 | |
| 0.143 | 0.049 | 0.143 | Platelet activating factor antagonist | |||
| 0.168 | 0.076 | 0.194 | 3C-like protease (Human coronavirus) inhibitor | 0.194 0.055 CHEMBL1573 0.165 0.08 CHEMBL3544724 | CHEMBL1573 | |
| 0.194 | 0.104 | 0.394 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.39 0.04 CHEMBL1573 0.394 0.039 CHEMBL3544724 0.175 0.117 CHEMBL3544725 | CHEMBL3544724 | |
| 0.165 | 0.077 | 0.328 | Mcl-1 antagonist | 0.265 0.031 CHEMBL1573 0.328 0.019 CHEMBL3544724 0.244 0.038 CHEMBL3544725 0.173 0.071 CHEMBL3544726 | CHEMBL3544724 | |
| 0.169 | 0.081 | 0.238 | Succinate dehydrogenase inhibitor | 0.188 0.059 CHEMBL1573 0.238 0.027 CHEMBL3544724 0.183 0.064 CHEMBL3544725 | CHEMBL3544724 | |
| 0.123 | 0.035 | 0.123 | Alpha 2 adrenoreceptor antagonist | |||
| 0.18 | 0.093 | 0.238 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.212 0.063 CHEMBL1573 0.238 0.048 CHEMBL3544724 0.225 0.055 CHEMBL3544725 0.18 0.093 CHEMBL3544726 | CHEMBL3544724 | |
| 0.147 | 0.059 | 0.147 | Pregnane X receptor agonist | |||
| 0.244 | 0.159 | 0.387 | GABA C receptor rho-3 antagonist | 0.387 0.067 CHEMBL1573 0.262 0.144 CHEMBL3544724 | CHEMBL1573 | |
| 0.161 | 0.077 | 0.161 | Neurotensin receptor agonist | 0.138 0.135 CHEMBL1573 0.138 0.133 CHEMBL3544724 | ||
| 0.092 | 0.011 | 0.092 | Potassium channel intermediate-conductance Ca-activated blocker | 0.079 0.018 CHEMBL1573 0.059 0.044 CHEMBL3544724 0.067 0.031 CHEMBL3544726 | ||
| 0.097 | 0.017 | 0.097 | Calcium channel T-type blocker | |||
| 0.215 | 0.135 | 0.379 | 12-Lipoxygenase inhibitor | 0.379 0.046 CHEMBL1573 0.379 0.045 CHEMBL3544724 0.278 0.093 CHEMBL3544725 0.305 0.077 CHEMBL3544726 | CHEMBL3544724 | |
| 0.128 | 0.048 | 0.136 | Photosensitizer | 0.134 0.042 CHEMBL1573 0.136 0.041 CHEMBL3544724 0.112 0.068 CHEMBL3544725 0.114 0.066 CHEMBL3544726 | CHEMBL3544724 | |
| 0.133 | 0.057 | 0.233 | Alkylator | 0.208 0.024 CHEMBL1573 0.198 0.027 CHEMBL3544724 0.169 0.037 CHEMBL3544725 0.233 0.019 CHEMBL3544726 | CHEMBL3544726 | |
| 0.163 | 0.088 | 0.163 | Lipocortins synthesis antagonist | 0.161 0.091 CHEMBL3544724 | ||
| 0.108 | 0.034 | 0.108 | Bile acid receptor antagonist | |||
| 0.115 | 0.042 | 0.149 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.096 0.058 CHEMBL1573 0.149 0.027 CHEMBL3544724 0.123 0.037 CHEMBL3544725 | CHEMBL3544724 | |
| 0.166 | 0.098 | 0.199 | Anesthetic general | 0.199 0.075 CHEMBL1573 0.199 0.075 CHEMBL3544724 | CHEMBL3544724 | |
| 0.116 | 0.048 | 0.121 | Toll-Like receptor 4 antagonist | 0.121 0.043 CHEMBL1573 0.11 0.055 CHEMBL3544724 0.105 0.061 CHEMBL3544725 | CHEMBL1573 | |
| 0.107 | 0.041 | 0.107 | Alpha 1 adrenoreceptor antagonist | |||
| 0.078 | 0.013 | 0.078 | Thromboxane synthase inhibitor | 0.055 0.036 CHEMBL1573 0.07 0.018 CHEMBL3544724 0.062 0.025 CHEMBL3544725 | ||
| 0.188 | 0.124 | 0.188 | Antioxidant | 0.163 0.15 CHEMBL3544724 | ||
| 0.074 | 0.01 | 0.074 | Potassium channel (Inward rectifier) activator | 0.056 0.026 CHEMBL3544726 | ||
| 0.1 | 0.036 | 0.1 | Alpha 1a adrenoreceptor antagonist | |||
| 0.106 | 0.043 | 0.106 | ABCA1 expression enhancer | |||
| 0.139 | 0.077 | 0.141 | Heat shock protein 70 antagonist | 0.135 0.097 CHEMBL1573 0.141 0.07 CHEMBL3544724 | CHEMBL3544724 | |
| 0.071 | 0.009 | 0.071 | Potassium channel (ATP-sensitive) activator | 0.053 0.025 CHEMBL3544726 | ||
| 0.074 | 0.015 | 0.074 | Nicotinic alpha3beta2 receptor antagonist | 0.057 0.031 CHEMBL1573 | ||
| 0.079 | 0.024 | 0.101 | Glutamate (mGluR1) antagonist | 0.101 0.016 CHEMBL1573 0.09 0.019 CHEMBL3544724 0.089 0.019 CHEMBL3544725 | CHEMBL1573 | |
| 0.113 | 0.058 | 0.152 | Multidrug resistance-associated protein 1 inhibitor | 0.152 0.024 CHEMBL1573 0.143 0.029 CHEMBL3544724 0.109 0.064 CHEMBL3544725 0.103 0.074 CHEMBL3544726 | CHEMBL1573 | |
| 0.091 | 0.036 | 0.226 | Histidine decarboxylase inhibitor | 0.119 0.026 CHEMBL1573 0.226 0.01 CHEMBL3544724 0.199 0.013 CHEMBL3544725 | CHEMBL3544724 | |
| 0.233 | 0.18 | 0.324 | 15-Lipoxygenase inhibitor | 0.324 0.115 CHEMBL1573 0.283 0.142 CHEMBL3544724 | CHEMBL1573 | |
| 0.141 | 0.092 | 0.163 | Interferon gamma antagonist | 0.138 0.095 CHEMBL1573 0.163 0.063 CHEMBL3544724 0.148 0.08 CHEMBL3544725 | CHEMBL3544724 | |
| 0.103 | 0.054 | 0.103 | Antiadrenergic | |||
| 0.082 | 0.034 | 0.082 | Phosphodiesterase III inhibitor | |||
| 0.092 | 0.045 | 0.092 | Neuropeptide Y antagonist | |||
| 0.1 | 0.053 | 0.1 | Adrenaline antagonist | |||
| 0.074 | 0.028 | 0.074 | Nitric oxide donor | |||
| 0.05 | 0.007 | 0.05 | Transforming growth factor beta 2 antagonist | |||
| 0.057 | 0.015 | 0.073 | Glutamate (mGluR group III) antagonist | 0.049 0.022 CHEMBL1573 0.073 0.009 CHEMBL3544724 0.041 0.036 CHEMBL3544725 | CHEMBL3544724 | |
| 0.097 | 0.058 | 0.097 | Alpha adrenoreceptor antagonist | |||
| 0.201 | 0.164 | 0.37 | Cholesterol antagonist | 0.277 0.106 CHEMBL1573 0.37 0.057 CHEMBL3544724 0.338 0.069 CHEMBL3544725 | CHEMBL3544724 | |
| 0.071 | 0.036 | 0.071 | Beta adrenoreceptor antagonist | |||
| 0.147 | 0.113 | 0.147 | Hepatoprotectant | |||
| 0.048 | 0.013 | 0.062 | Glutamate (mGluR8) agonist | 0.048 0.013 CHEMBL1573 0.062 0.006 CHEMBL3544724 0.048 0.013 CHEMBL3544725 | CHEMBL3544724 | |
| 0.068 | 0.034 | 0.153 | Biliverdin reductase inhibitor | 0.09 0.022 CHEMBL1573 0.153 0.009 CHEMBL3544724 0.103 0.018 CHEMBL3544725 | CHEMBL3544724 | |
| 0.095 | 0.062 | 0.095 | Pim-1 kinase inhibitor | |||
| 0.076 | 0.044 | 0.076 | Potassium channel (Tandem pore domain) blocker | |||
| 0.09 | 0.06 | 0.09 | Potassium channel activator | |||
| 0.129 | 0.102 | 0.146 | Phospholipase A2 inhibitor | 0.146 0.079 CHEMBL3544724 | CHEMBL3544724 | |
| 0.047 | 0.024 | 0.064 | Glutamate (mGluR4) antagonist | 0.044 0.03 CHEMBL1573 0.064 0.012 CHEMBL3544724 | CHEMBL3544724 | |
| 0.063 | 0.04 | 0.063 | TRPA1 antagonist | |||
| 0.114 | 0.094 | 0.193 | Interleukin 4 antagonist | 0.171 0.034 CHEMBL1573 0.193 0.025 CHEMBL3544724 0.165 0.038 CHEMBL3544725 0.118 0.089 CHEMBL3544726 | CHEMBL3544724 | |
| 0.104 | 0.084 | 0.104 | Microtubule formation inhibitor | |||
| 0.031 | 0.012 | 0.031 | NMDA receptor glycine site antagonist | 0.029 0.013 CHEMBL3544724 | ||
| 0.084 | 0.065 | 0.097 | Granulocyte macrophage colony stimulating factor agonist | 0.097 0.04 CHEMBL1573 0.082 0.069 CHEMBL3544724 0.08 0.075 CHEMBL3544725 | CHEMBL1573 | |
| 0.056 | 0.039 | 0.056 | Beta 1 adrenoreceptor antagonist | |||
| 0.092 | 0.075 | 0.148 | GABA C receptor rho-1 antagonist | 0.128 0.034 CHEMBL1573 0.148 0.022 CHEMBL3544724 0.089 0.08 CHEMBL3544725 | CHEMBL3544724 | |
| 0.061 | 0.045 | 0.08 | NMDA receptor agonist | 0.08 0.029 CHEMBL3544724 | CHEMBL3544724 | |
| 0.171 | 0.155 | 0.276 | Superoxide dismutase inhibitor | 0.222 0.096 CHEMBL1573 0.276 0.06 CHEMBL3544724 0.165 0.163 CHEMBL3544725 | CHEMBL3544724 | |
| 0.104 | 0.088 | 0.107 | Calcium channel N-type blocker | 0.107 0.083 CHEMBL1573 | CHEMBL1573 | |
| 0.079 | 0.063 | 0.082 | Glutathione S-transferase inhibitor | 0.079 0.063 CHEMBL1573 0.082 0.059 CHEMBL3544724 | CHEMBL3544724 | |
| 0.06 | 0.045 | 0.074 | NMDA receptor glycine site agonist | 0.074 0.033 CHEMBL3544724 | CHEMBL3544724 | |
| 0.14 | 0.125 | 0.14 | Psychostimulant | |||
| 0.089 | 0.075 | 0.144 | UDP-glucose 4-epimerase inhibitor | 0.103 0.057 CHEMBL1573 0.142 0.031 CHEMBL3544724 0.144 0.031 CHEMBL3544725 | CHEMBL3544725 | |
| 0.072 | 0.059 | 0.136 | GABA aminotransferase inhibitor | 0.097 0.029 CHEMBL1573 0.136 0.011 CHEMBL3544724 0.094 0.032 CHEMBL3544725 | CHEMBL3544724 | |
| 0.036 | 0.024 | 0.036 | Progesterone antagonist | |||
| 0.08 | 0.07 | 0.08 | 3C-Like protease (SARS coronavirus) inhibitor | 0.08 0.07 CHEMBL3544724 | ||
| 0.064 | 0.054 | 0.073 | Glutamate (mGluR6) antagonist | 0.073 0.034 CHEMBL3544724 | CHEMBL3544724 | |
| 0.166 | 0.158 | 0.352 | Streptokinase A inhibitor | 0.352 0.061 CHEMBL1573 0.337 0.066 CHEMBL3544724 0.196 0.135 CHEMBL3544725 | CHEMBL1573 | |
| 0.025 | 0.017 | 0.036 | Kainate receptor 4 antagonist | 0.026 0.016 CHEMBL1573 0.036 0.011 CHEMBL3544724 | CHEMBL3544724 | |
| 0.089 | 0.083 | 0.089 | Mediator release inhibitor | |||
| 0.068 | 0.063 | 0.132 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.095 0.04 CHEMBL1573 0.114 0.031 CHEMBL3544724 0.132 0.025 CHEMBL3544725 | CHEMBL3544725 | |
| 0.047 | 0.043 | 0.047 | Sodium/calcium exchanger inhibitor | |||
| 0.04 | 0.036 | 0.062 | GABA B receptor antagonist | 0.062 0.011 CHEMBL1573 0.054 0.016 CHEMBL3544724 | CHEMBL1573 | |
| 0.038 | 0.036 | 0.039 | Kainate receptor agonist | 0.039 0.033 CHEMBL3544724 | CHEMBL3544724 | |
| 0.092 | 0.09 | 0.106 | Factor V inhibitor | 0.098 0.074 CHEMBL1573 0.106 0.056 CHEMBL3544724 0.096 0.079 CHEMBL3544725 | CHEMBL3544724 | |
| 0.015 | 0.015 | 0.02 | Kainate receptor 3 antagonist | 0.02 0.009 CHEMBL3544724 | CHEMBL3544724 | |
| 0.052 | 0.053 | 0.061 | Androgen agonist | 0.061 0.039 CHEMBL1573 | CHEMBL1573 | |
| 0.045 | 0.047 | 0.091 | CD45 antagonist | 0.059 0.023 CHEMBL1573 0.091 0.01 CHEMBL3544724 0.057 0.025 CHEMBL3544725 | CHEMBL3544724 | |
| 0.062 | 0.065 | 0.207 | Porphobilinogen synthase inhibitor | 0.111 0.031 CHEMBL1573 0.207 0.011 CHEMBL3544724 0.163 0.018 CHEMBL3544725 | CHEMBL3544724 | |
| 0.023 | 0.026 | 0.06 | NMDA 2D receptor antagonist | 0.03 0.016 CHEMBL1573 0.06 0.005 CHEMBL3544724 0.037 0.011 CHEMBL3544725 | CHEMBL3544724 | |
| 0.077 | 0.082 | 0.143 | Triose-phosphate isomerase inhibitor | 0.097 0.051 CHEMBL1573 0.143 0.022 CHEMBL3544724 0.136 0.025 CHEMBL3544725 | CHEMBL3544724 | |
| 0.074 | 0.08 | 0.095 | Thioredoxin reductase inhibitor | 0.095 0.033 CHEMBL1573 0.094 0.035 CHEMBL3544724 0.088 0.044 CHEMBL3544725 0.077 0.071 CHEMBL3544726 | CHEMBL1573 | |
| 0.09 | 0.096 | 0.112 | GABA C receptor antagonist | 0.101 0.076 CHEMBL1573 0.112 0.061 CHEMBL3544724 | CHEMBL3544724 | |
| 0.048 | 0.056 | 0.057 | Dihydroorotate oxidase inhibitor | 0.057 0.034 CHEMBL3544724 | CHEMBL3544724 | |
| 0.143 | 0.152 | 0.294 | Histone acetyltransferase inhibitor | 0.294 0.015 CHEMBL1573 0.288 0.016 CHEMBL3544724 0.204 0.063 CHEMBL3544725 0.202 0.067 CHEMBL3544726 | CHEMBL1573 | |
| 0.014 | 0.024 | 0.035 | Kainate receptor 5 antagonist | 0.035 0.008 CHEMBL3544724 | CHEMBL3544724 | |
| 0.057 | 0.067 | 0.077 | Transcription factor RelA inhibitor | 0.077 0.02 CHEMBL1573 0.065 0.041 CHEMBL3544724 0.064 0.043 CHEMBL3544726 | CHEMBL1573 | |
| 0.026 | 0.038 | 0.044 | Catechol O-methyltransferase inhibitor | 0.041 0.013 CHEMBL1573 0.041 0.013 CHEMBL3544724 0.044 0.011 CHEMBL3544725 | CHEMBL3544725 | |
| 0.036 | 0.049 | 0.053 | AICAR transformylase inhibitor | 0.046 0.027 CHEMBL1573 0.053 0.019 CHEMBL3544724 | CHEMBL3544724 | |
| 0.096 | 0.109 | 0.181 | M17 leucyl aminopeptidase inhibitor | 0.13 0.069 CHEMBL1573 0.181 0.04 CHEMBL3544724 0.12 0.078 CHEMBL3544725 | CHEMBL3544724 | |
| 0.043 | 0.057 | 0.146 | Alcohol oxidase inhibitor | 0.067 0.03 CHEMBL1573 0.146 0.01 CHEMBL3544724 0.065 0.032 CHEMBL3544725 | CHEMBL3544724 | |
| 0.075 | 0.09 | 0.249 | Breast cancer-resistant protein inhibitor | 0.249 0.009 CHEMBL1573 0.193 0.015 CHEMBL3544724 0.136 0.03 CHEMBL3544725 0.216 0.012 CHEMBL3544726 | CHEMBL1573 | |
| 0.067 | 0.082 | 0.07 | GABA B receptor agonist | 0.07 0.069 CHEMBL3544724 | CHEMBL3544724 | |
| 0.1 | 0.116 | 0.171 | Alkaline phosphatase inhibitor | 0.163 0.052 CHEMBL1573 0.171 0.047 CHEMBL3544724 0.134 0.072 CHEMBL3544725 | CHEMBL3544724 | |
| 0.167 | 0.184 | 0.199 | Transcription factor STAT3 inhibitor | 0.185 0.156 CHEMBL1573 0.199 0.135 CHEMBL3544724 | CHEMBL3544724 | |
| 0.172 | 0.191 | 0.201 | Gastrin inhibitor | 0.201 0.147 CHEMBL3544724 0.182 0.176 CHEMBL3544725 | CHEMBL3544724 | |
| 0.204 | 0.224 | 0.362 | Antibacterial | 0.248 0.179 CHEMBL1573 0.355 0.099 CHEMBL3544724 0.362 0.095 CHEMBL3544725 | CHEMBL3544725 | |
| 0.126 | 0.146 | 0.135 | Ca2+-transporting ATPase inhibitor | 0.135 0.096 CHEMBL3544724 | CHEMBL3544724 | |
| 0.256 | 0.277 | 0.312 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.306 0.205 CHEMBL1573 0.312 0.197 CHEMBL3544724 | CHEMBL3544724 | |
| 0.164 | 0.188 | 0.396 | Prostaglandin dehydrogenase inhibitor | 0.396 0.068 CHEMBL1573 0.346 0.084 CHEMBL3544724 0.178 0.174 CHEMBL3544725 0.265 0.119 CHEMBL3544726 | CHEMBL1573 | |
| 0.072 | 0.097 | 0.099 | D-Ala-D-Ala ligase inhibitor | 0.086 0.052 CHEMBL1573 0.099 0.03 CHEMBL3544724 | CHEMBL3544724 | |
| 0.094 | 0.12 | 0.104 | Cathepsin H inhibitor | 0.103 0.101 CHEMBL1573 0.104 0.1 CHEMBL3544724 | CHEMBL3544724 | |
| 0.082 | 0.109 | 0.133 | Interleukin 1b antagonist | 0.133 0.053 CHEMBL1573 0.122 0.061 CHEMBL3544724 | CHEMBL1573 | |
| 0.024 | 0.051 | 0.048 | Kainate receptor antagonist | 0.048 0.023 CHEMBL3544724 | CHEMBL3544724 | |
| 0.137 | 0.165 | 0.151 | Free radical scavenger | 0.151 0.144 CHEMBL3544724 | CHEMBL3544724 | |
| 0.024 | 0.054 | 0.043 | Purinergic P2Y2 antagonist | 0.034 0.023 CHEMBL3544724 0.043 0.014 CHEMBL3544725 | CHEMBL3544725 | |
| 0.005 | 0.035 | 0.014 | Angiotensin AT1B receptor antagonist | 0.014 0.01 CHEMBL3544724 0.014 0.009 CHEMBL3544725 | CHEMBL3544725 | |
| 0.117 | 0.149 | 0.267 | DNA methyltransferase I inhibitor | 0.198 0.07 CHEMBL1573 0.267 0.039 CHEMBL3544724 0.185 0.077 CHEMBL3544725 | CHEMBL3544724 | |
| 0.051 | 0.084 | 0.071 | Interferon inducer | 0.071 0.034 CHEMBL1573 0.069 0.036 CHEMBL3544724 0.064 0.045 CHEMBL3544725 | CHEMBL1573 | |
| 0.072 | 0.105 | 0.084 | Thioredoxin inhibitor | 0.084 0.073 CHEMBL1573 | CHEMBL1573 | |
| 0.157 | 0.19 | 0.218 | DNA synthesis inhibitor | 0.218 0.097 CHEMBL3544724 0.212 0.106 CHEMBL3544725 | CHEMBL3544724 | |
| 0.049 | 0.084 | 0.058 | Ryanodine receptor antagonist | 0.057 0.046 CHEMBL1573 0.058 0.045 CHEMBL3544724 | CHEMBL3544724 | |
| 0.05 | 0.085 | 0.072 | Bcl-xL inhibitor | 0.06 0.04 CHEMBL1573 0.061 0.037 CHEMBL3544724 0.072 0.018 CHEMBL3544725 | CHEMBL3544725 | |
| 0.057 | 0.096 | 0.069 | MDM2 inhibitor | 0.063 0.061 CHEMBL1573 0.069 0.042 CHEMBL3544724 | CHEMBL3544724 | |
| 0.068 | 0.108 | 0.079 | Transcription factor NF kappa B stimulant | 0.079 0.073 CHEMBL3544725 | CHEMBL3544725 | |
| 0.03 | 0.076 | 0.103 | Dihydroorotate dehydrogenase inhibitor | 0.055 0.033 CHEMBL1573 0.103 0.01 CHEMBL3544724 0.062 0.027 CHEMBL3544725 | CHEMBL3544724 | |
| 0.034 | 0.08 | 0.057 | Argininosuccinate synthase inhibitor | 0.057 0.039 CHEMBL3544724 | CHEMBL3544724 | |
| 0.026 | 0.074 | 0.044 | NMDA receptor subunit 3B antagonist | 0.044 0.031 CHEMBL3544724 | CHEMBL3544724 | |
| 0.067 | 0.115 | 0.102 | Interleukin 5 antagonist | 0.092 0.052 CHEMBL1573 0.102 0.039 CHEMBL3544724 0.091 0.053 CHEMBL3544725 | CHEMBL3544724 | |
| 0.072 | 0.121 | 0.155 | Xanthine oxidase inhibitor | 0.091 0.069 CHEMBL1573 0.155 0.033 CHEMBL3544724 0.111 0.052 CHEMBL3544725 | CHEMBL3544724 | |
| 0.011 | 0.061 | 0.042 | Kynurenine 3 monooxygenase inhibitor | 0.023 0.022 CHEMBL1573 0.042 0.009 CHEMBL3544724 | CHEMBL3544724 | |
| 0.028 | 0.078 | 0.057 | Nerve growth factor antagonist | 0.051 0.017 CHEMBL1573 0.057 0.011 CHEMBL3544724 | CHEMBL3544724 | |
| 0.019 | 0.07 | 0.038 | NMDA receptor subunit 3A antagonist | 0.038 0.027 CHEMBL3544724 | CHEMBL3544724 | |
| 0.072 | 0.124 | 0.288 | Anesthetic local | 0.288 0.014 CHEMBL1573 0.233 0.024 CHEMBL3544724 0.164 0.043 CHEMBL3544725 | CHEMBL1573 | |
| 0.012 | 0.065 | 0.04 | AMPA 2 receptor antagonist | 0.028 0.022 CHEMBL1573 0.04 0.014 CHEMBL3544724 0.03 0.02 CHEMBL3544725 | CHEMBL3544724 | |
| 0.018 | 0.072 | 0.031 | Complement factor 1r inhibitor | 0.031 0.01 CHEMBL3544726 | CHEMBL3544726 | |
| 0.055 | 0.112 | 0.082 | Interferon agonist | 0.082 0.05 CHEMBL1573 0.081 0.051 CHEMBL3544724 0.074 0.063 CHEMBL3544725 | CHEMBL1573 | |
| 0.218 | 0.276 | 0.371 | 5 Hydroxytryptamine release inhibitor | 0.29 0.176 CHEMBL1573 0.371 0.098 CHEMBL3544724 0.243 0.238 CHEMBL3544725 | CHEMBL3544724 | |
| 0.1 | 0.162 | 0.128 | NOS3 expression enhancer | 0.128 0.101 CHEMBL3544724 | CHEMBL3544724 | |
| 0.065 | 0.129 | 0.135 | Ferrochelatase inhibitor | 0.135 0.045 CHEMBL3544724 | CHEMBL3544724 | |
| 0.042 | 0.106 | 0.082 | Na+ K+ transporting ATPase inhibitor | 0.082 0.049 CHEMBL1573 0.077 0.053 CHEMBL3544724 0.069 0.061 CHEMBL3544725 | CHEMBL1573 | |
| 0.098 | 0.164 | 0.277 | Dual specificity phosphatase 3 inhibitor | 0.219 0.051 CHEMBL1573 0.277 0.033 CHEMBL3544724 0.245 0.042 CHEMBL3544725 0.138 0.108 CHEMBL3544726 | CHEMBL3544724 | |
| 0.021 | 0.091 | 0.06 | Angiotensin AT1 receptor antagonist | 0.052 0.014 CHEMBL1573 0.059 0.007 CHEMBL3544724 0.06 0.006 CHEMBL3544725 | CHEMBL3544725 | |
| 0.039 | 0.11 | 0.108 | Purinergic P2X1 antagonist | 0.073 0.03 CHEMBL1573 0.108 0.014 CHEMBL3544724 0.081 0.025 CHEMBL3544725 | CHEMBL3544724 | |
| 0.029 | 0.101 | 0.059 | DNA gyrase subunit A inhibitor | 0.042 0.03 CHEMBL3544724 0.059 0.01 CHEMBL3544726 | CHEMBL3544726 | |
| 0.047 | 0.12 | 0.078 | Glutamate dehydrogenase inhibitor | 0.078 0.047 CHEMBL3544724 | CHEMBL3544724 | |
| 0.042 | 0.117 | 0.077 | Bcl2 antagonist | 0.077 0.034 CHEMBL1573 0.074 0.038 CHEMBL3544724 0.076 0.036 CHEMBL3544725 | CHEMBL1573 | |
| 0.028 | 0.103 | 0.056 | GABA A receptor antagonist | 0.056 0.034 CHEMBL1573 | CHEMBL1573 | |
| 0.033 | 0.109 | 0.077 | Phosphofructokinase-1 inhibitor | 0.077 0.043 CHEMBL3544724 0.073 0.046 CHEMBL3544725 | CHEMBL3544724 | |
| 0.014 | 0.092 | 0.03 | Fumarate hydratase inhibitor | 0.03 0.029 CHEMBL3544724 | CHEMBL3544724 | |
| 0.023 | 0.102 | 0.046 | Carbonic anhydrase XIV inhibitor | 0.046 0.038 CHEMBL3544724 | CHEMBL3544724 | |
| 0.038 | 0.118 | 0.092 | Carbonic anhydrase XIII inhibitor | 0.092 0.042 CHEMBL3544724 0.069 0.059 CHEMBL3544725 | CHEMBL3544724 | |
| 0.063 | 0.144 | 0.114 | Carbonic anhydrase III inhibitor | 0.114 0.048 CHEMBL3544724 0.091 0.073 CHEMBL3544725 | CHEMBL3544724 | |
| 0.034 | 0.116 | 0.071 | Sphingosine 1-phosphate receptor 4 agonist | 0.071 0.044 CHEMBL1573 0.065 0.049 CHEMBL3544724 0.068 0.046 CHEMBL3544725 | CHEMBL1573 | |
| 0.08 | 0.162 | 0.213 | Toll-Like receptor antagonist | 0.213 0.026 CHEMBL1573 0.123 0.08 CHEMBL3544724 0.114 0.095 CHEMBL3544725 | CHEMBL1573 | |
| 0.018 | 0.101 | 0.051 | Angiotensin II receptor antagonist | 0.039 0.015 CHEMBL1573 0.05 0.007 CHEMBL3544724 0.051 0.006 CHEMBL3544725 | CHEMBL3544725 | |
| 0.05 | 0.134 | 0.07 | Keratolytic | 0.07 0.066 CHEMBL3544724 | CHEMBL3544724 | |
| 0.137 | 0.221 | 0.278 | Thyroid hormone beta antagonist | 0.278 0.1 CHEMBL1573 0.214 0.143 CHEMBL3544724 | CHEMBL1573 | |
| 0.096 | 0.182 | 0.144 | Heat shock protein 90 alpha antagonist | 0.144 0.093 CHEMBL1573 0.134 0.106 CHEMBL3544724 | CHEMBL1573 | |
| 0.077 | 0.163 | 0.167 | Toll-Like receptor 9 antagonist | 0.167 0.053 CHEMBL1573 | CHEMBL1573 | |
| 0.137 | 0.225 | 0.287 | Thyroid hormone antagonist | 0.287 0.1 CHEMBL1573 0.232 0.136 CHEMBL3544724 | CHEMBL1573 | |
| 0.027 | 0.115 | 0.053 | GABA receptor antagonist | 0.053 0.04 CHEMBL1573 0.048 0.047 CHEMBL3544726 | CHEMBL1573 | |
| 0.018 | 0.108 | 0.091 | AMPA receptor antagonist | 0.06 0.025 CHEMBL1573 0.091 0.014 CHEMBL3544724 0.052 0.029 CHEMBL3544725 | CHEMBL3544724 | |
| 0.097 | 0.19 | 0.233 | Dual specificity phosphatase inhibitor | 0.177 0.069 CHEMBL1573 0.233 0.042 CHEMBL3544724 0.198 0.056 CHEMBL3544725 | CHEMBL3544724 | |
| 0.008 | 0.101 | 0.029 | Methionyl aminopeptidase 2 inhibitor | 0.029 0.014 CHEMBL3544724 | CHEMBL3544724 | |
| 0.009 | 0.103 | 0.029 | AMPA 3 receptor antagonist | 0.029 0.021 CHEMBL3544724 | CHEMBL3544724 | |
| 0.089 | 0.184 | 0.206 | Hexokinase inhibitor | 0.157 0.071 CHEMBL1573 0.206 0.032 CHEMBL3544724 0.171 0.057 CHEMBL3544725 | CHEMBL3544724 | |
| 0.031 | 0.125 | 0.057 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.057 0.043 CHEMBL3544724 | CHEMBL3544724 | |
| 0.026 | 0.121 | 0.041 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.041 0.031 CHEMBL3544724 | CHEMBL3544724 | |
| 0.048 | 0.145 | 0.078 | Calcium channel P-type blocker | 0.078 0.017 CHEMBL1573 0.069 0.031 CHEMBL3544724 | CHEMBL1573 | |
| 0.056 | 0.156 | 0.089 | GABA C receptor agonist | 0.089 0.08 CHEMBL3544724 | CHEMBL3544724 | |
| 0.047 | 0.148 | 0.082 | Aminopeptidase B inhibitor | 0.082 0.08 CHEMBL3544724 | CHEMBL3544724 | |
| 0.078 | 0.18 | 0.204 | Interleukin 1 antagonist | 0.204 0.031 CHEMBL1573 0.182 0.041 CHEMBL3544724 0.121 0.087 CHEMBL3544725 0.184 0.04 CHEMBL3544726 | CHEMBL1573 | |
| 0.027 | 0.129 | 0.056 | Aconitate hydratase inhibitor | 0.056 0.031 CHEMBL3544724 | CHEMBL3544724 | |
| 0.189 | 0.291 | 0.43 | Apoptosis agonist | 0.326 0.155 CHEMBL1573 0.313 0.163 CHEMBL3544724 0.31 0.165 CHEMBL3544725 0.43 0.1 CHEMBL3544726 | CHEMBL3544726 | |
| 0.121 | 0.224 | 0.383 | DNA damaging | 0.356 0.039 CHEMBL1573 0.292 0.06 CHEMBL3544724 0.271 0.07 CHEMBL3544725 0.383 0.032 CHEMBL3544726 | CHEMBL3544726 | |
| 0.042 | 0.145 | 0.086 | Ornithine decarboxylase inhibitor | 0.086 0.06 CHEMBL3544724 | CHEMBL3544724 | |
| 0.064 | 0.167 | 0.109 | Carbonic anhydrase XV inhibitor | 0.109 0.057 CHEMBL3544724 0.096 0.072 CHEMBL3544725 | CHEMBL3544724 | |
| 0.024 | 0.129 | 0.053 | Elastase inhibitor | 0.053 0.037 CHEMBL3544726 | CHEMBL3544726 | |
| 0.029 | 0.135 | 0.069 | Benzodiazepine inverse agonist | 0.069 0.01 CHEMBL3544725 | CHEMBL3544725 | |
| 0.012 | 0.118 | 0.043 | Urate transporter 1 inhibitor | 0.043 0.023 CHEMBL3544724 | CHEMBL3544724 | |
| 0.027 | 0.145 | 0.073 | Prostaglandin-E synthase inhibitor | 0.073 0.045 CHEMBL3544724 | CHEMBL3544724 | |
| 0.029 | 0.147 | 0.072 | Catalase inhibitor | 0.072 0.053 CHEMBL3544724 | CHEMBL3544724 | |
| 0.108 | 0.227 | 0.147 | Phospholipase C inhibitor | 0.147 0.112 CHEMBL3544724 | CHEMBL3544724 | |
| 0.018 | 0.137 | 0.079 | Xanthine dehydrogenase inhibitor | 0.079 0.025 CHEMBL3544724 0.055 0.042 CHEMBL3544725 | CHEMBL3544724 | |
| 0.154 | 0.277 | 0.369 | Histamine release inhibitor | 0.222 0.179 CHEMBL1573 0.369 0.091 CHEMBL3544724 0.336 0.106 CHEMBL3544725 | CHEMBL3544724 | |
| 0.148 | 0.272 | 0.293 | Sodium/bile acid cotransporter inhibitor | 0.207 0.179 CHEMBL1573 0.293 0.085 CHEMBL3544724 0.24 0.139 CHEMBL3544725 | CHEMBL3544724 | |
| 0.09 | 0.219 | 0.212 | DNA methylase inhibitor | 0.154 0.114 CHEMBL1573 0.212 0.072 CHEMBL3544724 0.142 0.125 CHEMBL3544725 | CHEMBL3544724 | |
| 0.047 | 0.179 | 0.105 | Creatine kinase inhibitor | 0.105 0.054 CHEMBL3544724 | CHEMBL3544724 | |
| 0.004 | 0.136 | 0.021 | Angiotensin AT1A receptor antagonist | 0.021 0.016 CHEMBL3544725 | CHEMBL3544725 | |
| 0.036 | 0.17 | 0.069 | Adenine nucleotide translocase inhibitor | 0.069 0.016 CHEMBL3544724 0.067 0.019 CHEMBL3544725 | CHEMBL3544724 | |
| 0.061 | 0.195 | 0.127 | Alpha-N-acetylglucosaminidase inhibitor | 0.127 0.071 CHEMBL3544724 0.122 0.075 CHEMBL3544725 | CHEMBL3544724 | |
| 0.065 | 0.199 | 0.104 | Aldehyde dehydrogenase inhibitor | 0.104 0.091 CHEMBL3544724 | CHEMBL3544724 | |
| 0.052 | 0.191 | 0.221 | Glutamate receptor antagonist | 0.21 0.023 CHEMBL1573 0.221 0.02 CHEMBL3544724 0.183 0.032 CHEMBL3544725 | CHEMBL3544724 | |
| 0.065 | 0.206 | 0.139 | NADPH oxidase inhibitor | 0.13 0.071 CHEMBL1573 0.139 0.063 CHEMBL3544724 | CHEMBL3544724 | |
| 0.035 | 0.179 | 0.122 | Potassium channel (Ca-activated) activator | 0.078 0.077 CHEMBL1573 0.122 0.04 CHEMBL3544724 | CHEMBL3544724 | |
| 0.025 | 0.172 | 0.082 | HIV-1 integrase (3'-Processing) inhibitor | 0.082 0.033 CHEMBL3544724 0.058 0.05 CHEMBL3544725 | CHEMBL3544724 | |
| 0.053 | 0.201 | 0.094 | Protein kinase C gamma inhibitor | 0.094 0.088 CHEMBL3544724 | CHEMBL3544724 | |
| 0.016 | 0.164 | 0.045 | Retinoic acid alpha receptor agonist | 0.045 0.019 CHEMBL3544724 0.037 0.03 CHEMBL3544725 | CHEMBL3544724 | |
| 0.036 | 0.185 | 0.094 | Phosphodiesterase 3A inhibitor | 0.094 0.038 CHEMBL3544726 | CHEMBL3544726 | |
| 0.073 | 0.225 | 0.334 | Pyruvate kinase inhibitor | 0.334 0.039 CHEMBL1573 0.327 0.041 CHEMBL3544724 0.152 0.113 CHEMBL3544725 0.264 0.057 CHEMBL3544726 | CHEMBL1573 | |
| 0.055 | 0.208 | 0.104 | Caspase 3 inhibitor | 0.104 0.085 CHEMBL3544724 | CHEMBL3544724 | |
| 0.028 | 0.183 | 0.085 | Glutamate decarboxylase inhibitor | 0.085 0.039 CHEMBL3544724 | CHEMBL3544724 | |
| 0.08 | 0.236 | 0.107 | DNA repair enzyme inhibitor | 0.107 0.104 CHEMBL1573 | CHEMBL1573 | |
| 0.01 | 0.17 | 0.048 | Retinoid X alpha receptor agonist | 0.048 0.015 CHEMBL3544724 | CHEMBL3544724 | |
| 0.048 | 0.216 | 0.079 | NADH dehydrogenase inhibitor | 0.079 0.077 CHEMBL3544724 | CHEMBL3544724 | |
| 0.17 | 0.341 | 0.272 | MAP kinase 1 inhibitor | 0.272 0.21 CHEMBL1573 | CHEMBL1573 | |
| 0.033 | 0.206 | 0.074 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.074 0.05 CHEMBL1573 | CHEMBL1573 | |
| 0.015 | 0.188 | 0.068 | Neuraminidase inhibitor | 0.068 0.035 CHEMBL3544724 0.057 0.047 CHEMBL3544725 | CHEMBL3544724 | |
| 0.041 | 0.215 | 0.118 | Antineoplastic alkaloid | 0.118 0.039 CHEMBL3544726 | CHEMBL3544726 | |
| 0.045 | 0.219 | 0.11 | Tubulin antagonist | 0.11 0.091 CHEMBL3544726 | CHEMBL3544726 | |
| 0.03 | 0.21 | 0.097 | Glutamate (mGluR group I) antagonist | 0.097 0.027 CHEMBL1573 0.066 0.053 CHEMBL3544724 0.062 0.061 CHEMBL3544725 | CHEMBL1573 | |
| 0.042 | 0.222 | 0.106 | Cholesterol synthesis inhibitor | 0.106 0.08 CHEMBL3544724 | CHEMBL3544724 | |
| 0.007 | 0.187 | 0.041 | Retinoid X receptor agonist | 0.041 0.022 CHEMBL3544724 | CHEMBL3544724 | |
| 0.102 | 0.284 | 0.165 | Catenin beta inhibitor | 0.139 0.133 CHEMBL1573 0.164 0.076 CHEMBL3544724 0.165 0.074 CHEMBL3544726 | CHEMBL3544726 | |
| 0.039 | 0.225 | 0.1 | DNA intercalator | 0.1 0.074 CHEMBL3544726 | CHEMBL3544726 | |
| 0.032 | 0.22 | 0.07 | Macrophage migration inhibitory factor inhibitor | 0.07 0.067 CHEMBL3544724 | CHEMBL3544724 | |
| 0.038 | 0.233 | 0.151 | Glycogen synthase kinase-3 alpha inhibitor | 0.151 0.066 CHEMBL1573 0.151 0.066 CHEMBL3544724 | CHEMBL3544724 | |
| 0.025 | 0.231 | 0.09 | Monophenol monooxygenase inhibitor | 0.09 0.083 CHEMBL3544724 | CHEMBL3544724 | |
| 0.097 | 0.314 | 0.136 | CC chemokine 6 receptor antagonist | 0.12 0.116 CHEMBL1573 0.136 0.051 CHEMBL3544724 0.128 0.079 CHEMBL3544725 | CHEMBL3544724 | |
| 0.02 | 0.241 | 0.065 | Neuraminidase (influenza) inhibitor | 0.065 0.043 CHEMBL3544724 0.059 0.055 CHEMBL3544725 | CHEMBL3544724 | |
| 0.091 | 0.312 | 0.24 | Lipoxygenase inhibitor | 0.22 0.121 CHEMBL1573 0.24 0.106 CHEMBL3544724 | CHEMBL3544724 | |
| 0.031 | 0.253 | 0.065 | Potassium channel large-conductance Ca-activated activator | 0.065 0.05 CHEMBL3544724 | CHEMBL3544724 | |
| 0.047 | 0.272 | 0.172 | Protein-tyrosine phosphatase inhibitor | 0.16 0.069 CHEMBL3544724 0.172 0.061 CHEMBL3544725 | CHEMBL3544725 | |
| 0.024 | 0.275 | 0.107 | Glutamate (mGluR) antagonist | 0.107 0.031 CHEMBL1573 0.081 0.048 CHEMBL3544724 0.081 0.048 CHEMBL3544725 | CHEMBL1573 | |
| 0.018 | 0.274 | 0.058 | CDC25B inhibitor | 0.058 0.053 CHEMBL3544724 | CHEMBL3544724 | |
| 0.046 | 0.305 | 0.129 | Antibacterial (Helicobacter pylori) | 0.11 0.098 CHEMBL1573 0.129 0.069 CHEMBL3544725 | CHEMBL3544725 | |
| 0.115 | 0.383 | 0.239 | Caspase 3 stimulant | 0.239 0.123 CHEMBL3544726 | CHEMBL3544726 | |
| 0.025 | 0.293 | 0.087 | Alcohol dehydrogenase inhibitor | 0.087 0.068 CHEMBL3544724 | CHEMBL3544724 | |
| 0.012 | 0.313 | 0.053 | Potassium channel (Inward rectifier) blocker | 0.053 0.03 CHEMBL3544726 | CHEMBL3544726 | |
| 0.042 | 0.346 | 0.129 | Cytokine production inhibitor | 0.114 0.096 CHEMBL1573 0.129 0.081 CHEMBL3544726 | CHEMBL3544726 | |
| 0.005 | 0.332 | 0.045 | Potassium channel (Inward rectifier) 1 blocker | 0.045 0.005 CHEMBL3544726 | CHEMBL3544726 | |
| 0.046 | 0.402 | 0.223 | Platelet adhesion inhibitor | 0.163 0.093 CHEMBL1573 0.165 0.091 CHEMBL3544724 0.153 0.103 CHEMBL3544725 0.223 0.06 CHEMBL3544726 | CHEMBL3544726 | |
| 0.021 | 0.399 | 0.131 | Topoisomerase II inhibitor | 0.131 0.059 CHEMBL3544726 | CHEMBL3544726 | |
| 0.024 | 0.419 | 0.096 | Uric acid excretion stimulant | 0.096 0.057 CHEMBL3544724 | CHEMBL3544724 | |
| 0.012 | 0.445 | 0.109 | 5-Lipoxygenase inhibitor | 0.096 0.067 CHEMBL1573 0.109 0.057 CHEMBL3544724 | CHEMBL3544724 | |
| 0.019 | 0.469 | 0.084 | ATPase (Vacuolar H+) inhibitor | 0.084 0.07 CHEMBL3544726 | CHEMBL3544726 | |
| 0.015 | 0.472 | 0.187 | Topoisomerase I inhibitor | 0.187 0.03 CHEMBL3544726 | CHEMBL3544726 | |
| 0.02 | 0.515 | 0.081 | Viral attachment inhibitor | 0.081 0.047 CHEMBL1573 | CHEMBL1573 | |
| 0.012 | 0.554 | 0.109 | Topoisomerase II alpha inhibitor | 0.109 0.034 CHEMBL3544726 | CHEMBL3544726 | |
| 0.013 | 0.633 | 0.181 | Potassium channel blocker | 0.181 0.106 CHEMBL3544726 | CHEMBL3544726 | |
| 0.03 | 0.65 | 0.206 | Immunosuppressant | 0.206 0.191 CHEMBL3544724 | CHEMBL3544724 | |
| 0.012 | 0.633 | 0.062 | Autotaxin inhibitor | 0.062 0.027 CHEMBL3544725 | CHEMBL3544725 | |
| 0.03 | 0.708 | 0.297 | Hypoglycemic | 0.179 0.135 CHEMBL3544724 0.297 0.054 CHEMBL3544725 | CHEMBL3544725 | |
| 0.005 | 0.691 | 0.074 | HIV-1 integrase inhibitor | 0.074 0.044 CHEMBL3544724 0.066 0.055 CHEMBL3544725 | CHEMBL3544724 | |
| 0.003 | 0.744 | 0.055 | Potassium channel subfamily K member 3 blocker | 0.055 0.011 CHEMBL3544726 | CHEMBL3544726 | |
| 0.005 | 0.921 | 0.289 | Cyclophilin D inhibitor | 0.289 0.173 CHEMBL3544725 | CHEMBL3544725 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |