Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8510.0030.851Vasodilator, coronary

0.457 0.022 CHEMBL1573

0.451 0.023 CHEMBL3544724

0.48 0.018 CHEMBL3544725

0.333 0.064 CHEMBL3544726

0.850.0030.85Vasodilator, peripheral

0.578 0.018 CHEMBL1573

0.606 0.015 CHEMBL3544724

0.634 0.012 CHEMBL3544725

0.226 0.148 CHEMBL3544726

0.8080.0010.808Calcium channel activator

0.621 0.002 CHEMBL1573

0.594 0.002 CHEMBL3544724

0.602 0.002 CHEMBL3544725

0.636 0.002 CHEMBL3544726

0.8010.0030.801Calcium channel blocker

0.578 0.004 CHEMBL1573

0.499 0.004 CHEMBL3544724

0.441 0.004 CHEMBL3544725

0.32 0.008 CHEMBL3544726

0.7630.0010.763Calcium antagonist

0.342 0.004 CHEMBL1573

0.29 0.005 CHEMBL3544724

0.279 0.005 CHEMBL3544725

0.193 0.014 CHEMBL3544726

0.7510.0040.751Vasodilator

0.447 0.016 CHEMBL1573

0.412 0.021 CHEMBL3544724

0.413 0.021 CHEMBL3544725

0.309 0.045 CHEMBL3544726

0.740.0020.748Calcium channel L-type activator

0.739 0.002 CHEMBL1573

0.72 0.002 CHEMBL3544724

0.748 0.002 CHEMBL3544725

0.691 0.003 CHEMBL3544726

CHEMBL3544725
0.7170.0020.717TRPA1 agonist

0.177 0.017 CHEMBL1573

0.172 0.019 CHEMBL3544724

0.115 0.064 CHEMBL3544725

0.117 0.062 CHEMBL3544726

0.6640.0020.664Calcium channel L-type blocker

0.463 0.003 CHEMBL1573

0.46 0.003 CHEMBL3544724

0.44 0.003 CHEMBL3544725

0.2 0.005 CHEMBL3544726

0.6570.0030.657Calcium channel (voltage-sensitive) blocker

0.402 0.004 CHEMBL1573

0.327 0.005 CHEMBL3544724

0.254 0.01 CHEMBL3544725

0.125 0.051 CHEMBL3544726

0.5920.0080.592Cardiotonic

0.195 0.124 CHEMBL1573

0.182 0.137 CHEMBL3544724

0.219 0.103 CHEMBL3544725

0.299 0.057 CHEMBL3544726

0.3890.0050.389Alpha 2b adrenoreceptor antagonist

0.229 0.018 CHEMBL1573

0.133 0.049 CHEMBL3544724

0.4580.0980.56DNA polymerase beta inhibitor

0.56 0.069 CHEMBL1573

0.548 0.073 CHEMBL3544724

0.36 0.135 CHEMBL3544725

0.306 0.162 CHEMBL3544726

CHEMBL1573
0.350.0260.356Cyclic AMP phosphodiesterase inhibitor

0.232 0.073 CHEMBL1573

0.247 0.065 CHEMBL3544724

0.356 0.024 CHEMBL3544725

CHEMBL3544725
0.3090.0060.309Adenylate kinase inhibitor

0.166 0.021 CHEMBL1573

0.232 0.011 CHEMBL3544724

0.182 0.018 CHEMBL3544725

0.3530.0520.353Spasmolytic
0.3130.020.313Diuretic
0.3390.0490.339Hypoxia-inducible factor 1 alpha inhibitor

0.27 0.083 CHEMBL1573

0.279 0.077 CHEMBL3544724

0.328 0.053 CHEMBL3544725

0.181 0.177 CHEMBL3544726

0.3160.0320.316Platelet aggregation inhibitor
0.2880.0070.288Alpha 2c adrenoreceptor antagonist

0.182 0.022 CHEMBL1573

0.116 0.052 CHEMBL3544724

0.129 0.043 CHEMBL3544725

0.3940.1180.498DNA directed DNA polymerase inhibitor

0.497 0.083 CHEMBL1573

0.498 0.083 CHEMBL3544724

0.359 0.134 CHEMBL3544725

0.233 0.202 CHEMBL3544726

CHEMBL3544724
0.2780.0030.278Aldosterone antagonist

0.048 0.032 CHEMBL1573

0.270.0050.27CF transmembrane conductance regulator agonist

0.152 0.072 CHEMBL1573

0.132 0.113 CHEMBL3544724

0.2690.0070.269Neuropeptide Y1 antagonist

0.257 0.008 CHEMBL1573

0.233 0.01 CHEMBL3544724

0.209 0.015 CHEMBL3544725

0.133 0.095 CHEMBL3544726

0.2950.0330.2955 Hydroxytryptamine 1E antagonist

0.234 0.092 CHEMBL1573

0.2880.0310.288P-glycoprotein inhibitor

0.199 0.064 CHEMBL1573

0.177 0.082 CHEMBL3544724

0.157 0.106 CHEMBL3544725

0.3610.1250.437Transcription factor inhibitor

0.437 0.095 CHEMBL1573

0.369 0.122 CHEMBL3544724

0.259 0.18 CHEMBL3544725

0.298 0.156 CHEMBL3544726

CHEMBL1573
0.3120.0950.375Thioredoxin glutathione reductase inhibitor

0.375 0.067 CHEMBL1573

0.323 0.089 CHEMBL3544724

0.198 0.174 CHEMBL3544725

0.217 0.158 CHEMBL3544726

CHEMBL1573
0.290.0810.306Interleukin 2 agonist

0.257 0.111 CHEMBL1573

0.286 0.084 CHEMBL3544724

0.306 0.069 CHEMBL3544725

CHEMBL3544725
0.2760.0690.621Aryl hydrocarbon receptor agonist

0.621 0.013 CHEMBL1573

0.521 0.022 CHEMBL3544724

0.31 0.058 CHEMBL3544725

0.219 0.092 CHEMBL3544726

CHEMBL1573
0.1990.0040.199Glycine receptor antagonist

0.078 0.06 CHEMBL1573

0.2150.0230.307Mannose-6-phosphate isomerase inhibitor

0.292 0.006 CHEMBL1573

0.307 0.005 CHEMBL3544724

0.262 0.01 CHEMBL3544725

0.192 0.035 CHEMBL3544726

CHEMBL3544724
0.3430.1510.492Caspase 9 stimulant

0.492 0.063 CHEMBL1573

0.414 0.103 CHEMBL3544724

0.356 0.141 CHEMBL3544725

CHEMBL1573
0.2840.1040.317Transcription factor NF kappa B inhibitor

0.264 0.118 CHEMBL1573

0.285 0.103 CHEMBL3544724

0.317 0.087 CHEMBL3544725

0.2 0.169 CHEMBL3544726

CHEMBL3544725
0.1880.0150.188Androgen antagonist

0.1 0.047 CHEMBL1573

0.085 0.06 CHEMBL3544724

0.1870.0160.187Alpha 1b adrenoreceptor antagonist
0.1760.0120.176Alpha 1d adrenoreceptor antagonist
0.2120.050.212Amyloid beta precursor protein antagonist

0.146 0.106 CHEMBL1573

0.173 0.078 CHEMBL3544724

0.1770.0170.177Alpha 2a adrenoreceptor antagonist
0.1980.0420.203Interleukin 6 antagonist

0.203 0.039 CHEMBL1573

0.167 0.067 CHEMBL3544724

0.171 0.063 CHEMBL3544726

CHEMBL1573
0.2220.0720.222RNA-directed DNA polymerase inhibitor

0.214 0.081 CHEMBL1573

0.221 0.073 CHEMBL3544724

0.216 0.078 CHEMBL3544725

0.168 0.157 CHEMBL3544726

0.2640.1150.264Apoptosis antagonist

0.207 0.171 CHEMBL3544724

0.228 0.149 CHEMBL3544725

0.241 0.137 CHEMBL3544726

0.1840.0390.241GABA C receptor rho-2 antagonist

0.241 0.014 CHEMBL1573

0.199 0.029 CHEMBL3544724

0.137 0.093 CHEMBL3544725

0.192 0.033 CHEMBL3544726

CHEMBL1573
0.1640.0190.164Beta glucuronidase inhibitor

0.121 0.045 CHEMBL1573

0.119 0.047 CHEMBL3544724

0.2040.0680.273Non-steroidal antiinflammatory agent

0.239 0.047 CHEMBL1573

0.273 0.035 CHEMBL3544724

0.229 0.052 CHEMBL3544725

0.246 0.044 CHEMBL3544726

CHEMBL3544724
0.1370.0050.137Mineralocorticoid receptor antagonist
0.2680.1370.286Calpain 2 inhibitor

0.286 0.123 CHEMBL1573

0.204 0.184 CHEMBL3544724

CHEMBL1573
0.2190.0890.219Platelet antagonist
0.1830.0550.301Cytidine deaminase inhibitor

0.301 0.019 CHEMBL1573

0.29 0.021 CHEMBL3544724

0.246 0.03 CHEMBL3544725

0.121 0.099 CHEMBL3544726

CHEMBL1573
0.2250.0980.252Interleukin agonist

0.223 0.1 CHEMBL1573

0.252 0.077 CHEMBL3544724

0.229 0.095 CHEMBL3544725

CHEMBL3544724
0.1480.0220.21DOPA decarboxylase inhibitor

0.178 0.011 CHEMBL1573

0.21 0.005 CHEMBL3544724

0.158 0.017 CHEMBL3544725

0.101 0.073 CHEMBL3544726

CHEMBL3544724
0.1350.0140.135Adenosine A3 receptor antagonist

0.074 0.052 CHEMBL1573

0.1820.0680.314Sigma receptor agonist

0.314 0.036 CHEMBL1573

0.273 0.044 CHEMBL3544724

0.138 0.094 CHEMBL3544725

0.209 0.059 CHEMBL3544726

CHEMBL1573
0.1560.0460.156Farnesoid X receptor antagonist
0.2790.170.462Alpha-glucosidase inhibitor

0.462 0.092 CHEMBL1573

0.445 0.098 CHEMBL3544724

0.367 0.128 CHEMBL3544725

0.301 0.159 CHEMBL3544726

CHEMBL1573
0.240.1340.24Antithrombotic

0.193 0.186 CHEMBL3544724

0.1440.0390.171Sphingosine 1-phosphate receptor 4 antagonist

0.17 0.019 CHEMBL1573

0.171 0.019 CHEMBL3544724

0.138 0.045 CHEMBL3544725

CHEMBL3544724
0.1590.0570.169Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.135 0.103 CHEMBL1573

0.169 0.044 CHEMBL3544724

0.138 0.097 CHEMBL3544725

CHEMBL3544724
0.1260.0240.126Interleukin 12 antagonist

0.123 0.026 CHEMBL1573

0.112 0.037 CHEMBL3544724

0.1 0.054 CHEMBL3544725

0.102 0.05 CHEMBL3544726

0.1960.0950.196Nitric-oxide synthase stimulant

0.193 0.101 CHEMBL1573

0.168 0.158 CHEMBL3544724

0.2520.1560.311Beta lactamase inhibitor

0.311 0.13 CHEMBL1573

0.238 0.163 CHEMBL3544724

CHEMBL1573
0.1490.0520.189M18 aspartyl aminopeptidase inhibitor

0.186 0.038 CHEMBL1573

0.189 0.037 CHEMBL3544724

0.113 0.077 CHEMBL3544725

CHEMBL3544724
0.1430.0490.143Platelet activating factor antagonist
0.1680.0760.1943C-like protease (Human coronavirus) inhibitor

0.194 0.055 CHEMBL1573

0.165 0.08 CHEMBL3544724

CHEMBL1573
0.1940.1040.394Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.39 0.04 CHEMBL1573

0.394 0.039 CHEMBL3544724

0.175 0.117 CHEMBL3544725

CHEMBL3544724
0.1650.0770.328Mcl-1 antagonist

0.265 0.031 CHEMBL1573

0.328 0.019 CHEMBL3544724

0.244 0.038 CHEMBL3544725

0.173 0.071 CHEMBL3544726

CHEMBL3544724
0.1690.0810.238Succinate dehydrogenase inhibitor

0.188 0.059 CHEMBL1573

0.238 0.027 CHEMBL3544724

0.183 0.064 CHEMBL3544725

CHEMBL3544724
0.1230.0350.123Alpha 2 adrenoreceptor antagonist
0.180.0930.238Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.212 0.063 CHEMBL1573

0.238 0.048 CHEMBL3544724

0.225 0.055 CHEMBL3544725

0.18 0.093 CHEMBL3544726

CHEMBL3544724
0.1470.0590.147Pregnane X receptor agonist
0.2440.1590.387GABA C receptor rho-3 antagonist

0.387 0.067 CHEMBL1573

0.262 0.144 CHEMBL3544724

CHEMBL1573
0.1610.0770.161Neurotensin receptor agonist

0.138 0.135 CHEMBL1573

0.138 0.133 CHEMBL3544724

0.0920.0110.092Potassium channel intermediate-conductance Ca-activated blocker

0.079 0.018 CHEMBL1573

0.059 0.044 CHEMBL3544724

0.067 0.031 CHEMBL3544726

0.0970.0170.097Calcium channel T-type blocker
0.2150.1350.37912-Lipoxygenase inhibitor

0.379 0.046 CHEMBL1573

0.379 0.045 CHEMBL3544724

0.278 0.093 CHEMBL3544725

0.305 0.077 CHEMBL3544726

CHEMBL3544724
0.1280.0480.136Photosensitizer

0.134 0.042 CHEMBL1573

0.136 0.041 CHEMBL3544724

0.112 0.068 CHEMBL3544725

0.114 0.066 CHEMBL3544726

CHEMBL3544724
0.1330.0570.233Alkylator

0.208 0.024 CHEMBL1573

0.198 0.027 CHEMBL3544724

0.169 0.037 CHEMBL3544725

0.233 0.019 CHEMBL3544726

CHEMBL3544726
0.1630.0880.163Lipocortins synthesis antagonist

0.161 0.091 CHEMBL3544724

0.1080.0340.108Bile acid receptor antagonist
0.1150.0420.149UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.096 0.058 CHEMBL1573

0.149 0.027 CHEMBL3544724

0.123 0.037 CHEMBL3544725

CHEMBL3544724
0.1660.0980.199Anesthetic general

0.199 0.075 CHEMBL1573

0.199 0.075 CHEMBL3544724

CHEMBL3544724
0.1160.0480.121Toll-Like receptor 4 antagonist

0.121 0.043 CHEMBL1573

0.11 0.055 CHEMBL3544724

0.105 0.061 CHEMBL3544725

CHEMBL1573
0.1070.0410.107Alpha 1 adrenoreceptor antagonist
0.0780.0130.078Thromboxane synthase inhibitor

0.055 0.036 CHEMBL1573

0.07 0.018 CHEMBL3544724

0.062 0.025 CHEMBL3544725

0.1880.1240.188Antioxidant

0.163 0.15 CHEMBL3544724

0.0740.010.074Potassium channel (Inward rectifier) activator

0.056 0.026 CHEMBL3544726

0.10.0360.1Alpha 1a adrenoreceptor antagonist
0.1060.0430.106ABCA1 expression enhancer
0.1390.0770.141Heat shock protein 70 antagonist

0.135 0.097 CHEMBL1573

0.141 0.07 CHEMBL3544724

CHEMBL3544724
0.0710.0090.071Potassium channel (ATP-sensitive) activator

0.053 0.025 CHEMBL3544726

0.0740.0150.074Nicotinic alpha3beta2 receptor antagonist

0.057 0.031 CHEMBL1573

0.0790.0240.101Glutamate (mGluR1) antagonist

0.101 0.016 CHEMBL1573

0.09 0.019 CHEMBL3544724

0.089 0.019 CHEMBL3544725

CHEMBL1573
0.1130.0580.152Multidrug resistance-associated protein 1 inhibitor

0.152 0.024 CHEMBL1573

0.143 0.029 CHEMBL3544724

0.109 0.064 CHEMBL3544725

0.103 0.074 CHEMBL3544726

CHEMBL1573
0.0910.0360.226Histidine decarboxylase inhibitor

0.119 0.026 CHEMBL1573

0.226 0.01 CHEMBL3544724

0.199 0.013 CHEMBL3544725

CHEMBL3544724
0.2330.180.32415-Lipoxygenase inhibitor

0.324 0.115 CHEMBL1573

0.283 0.142 CHEMBL3544724

CHEMBL1573
0.1410.0920.163Interferon gamma antagonist

0.138 0.095 CHEMBL1573

0.163 0.063 CHEMBL3544724

0.148 0.08 CHEMBL3544725

CHEMBL3544724
0.1030.0540.103Antiadrenergic
0.0820.0340.082Phosphodiesterase III inhibitor
0.0920.0450.092Neuropeptide Y antagonist
0.10.0530.1Adrenaline antagonist
0.0740.0280.074Nitric oxide donor
0.050.0070.05Transforming growth factor beta 2 antagonist
0.0570.0150.073Glutamate (mGluR group III) antagonist

0.049 0.022 CHEMBL1573

0.073 0.009 CHEMBL3544724

0.041 0.036 CHEMBL3544725

CHEMBL3544724
0.0970.0580.097Alpha adrenoreceptor antagonist
0.2010.1640.37Cholesterol antagonist

0.277 0.106 CHEMBL1573

0.37 0.057 CHEMBL3544724

0.338 0.069 CHEMBL3544725

CHEMBL3544724
0.0710.0360.071Beta adrenoreceptor antagonist
0.1470.1130.147Hepatoprotectant
0.0480.0130.062Glutamate (mGluR8) agonist

0.048 0.013 CHEMBL1573

0.062 0.006 CHEMBL3544724

0.048 0.013 CHEMBL3544725

CHEMBL3544724
0.0680.0340.153Biliverdin reductase inhibitor

0.09 0.022 CHEMBL1573

0.153 0.009 CHEMBL3544724

0.103 0.018 CHEMBL3544725

CHEMBL3544724
0.0950.0620.095Pim-1 kinase inhibitor
0.0760.0440.076Potassium channel (Tandem pore domain) blocker
0.090.060.09Potassium channel activator
0.1290.1020.146Phospholipase A2 inhibitor

0.146 0.079 CHEMBL3544724

CHEMBL3544724
0.0470.0240.064Glutamate (mGluR4) antagonist

0.044 0.03 CHEMBL1573

0.064 0.012 CHEMBL3544724

CHEMBL3544724
0.0630.040.063TRPA1 antagonist
0.1140.0940.193Interleukin 4 antagonist

0.171 0.034 CHEMBL1573

0.193 0.025 CHEMBL3544724

0.165 0.038 CHEMBL3544725

0.118 0.089 CHEMBL3544726

CHEMBL3544724
0.1040.0840.104Microtubule formation inhibitor
0.0310.0120.031NMDA receptor glycine site antagonist

0.029 0.013 CHEMBL3544724

0.0840.0650.097Granulocyte macrophage colony stimulating factor agonist

0.097 0.04 CHEMBL1573

0.082 0.069 CHEMBL3544724

0.08 0.075 CHEMBL3544725

CHEMBL1573
0.0560.0390.056Beta 1 adrenoreceptor antagonist
0.0920.0750.148GABA C receptor rho-1 antagonist

0.128 0.034 CHEMBL1573

0.148 0.022 CHEMBL3544724

0.089 0.08 CHEMBL3544725

CHEMBL3544724
0.0610.0450.08NMDA receptor agonist

0.08 0.029 CHEMBL3544724

CHEMBL3544724
0.1710.1550.276Superoxide dismutase inhibitor

0.222 0.096 CHEMBL1573

0.276 0.06 CHEMBL3544724

0.165 0.163 CHEMBL3544725

CHEMBL3544724
0.1040.0880.107Calcium channel N-type blocker

0.107 0.083 CHEMBL1573

CHEMBL1573
0.0790.0630.082Glutathione S-transferase inhibitor

0.079 0.063 CHEMBL1573

0.082 0.059 CHEMBL3544724

CHEMBL3544724
0.060.0450.074NMDA receptor glycine site agonist

0.074 0.033 CHEMBL3544724

CHEMBL3544724
0.140.1250.14Psychostimulant
0.0890.0750.144UDP-glucose 4-epimerase inhibitor

0.103 0.057 CHEMBL1573

0.142 0.031 CHEMBL3544724

0.144 0.031 CHEMBL3544725

CHEMBL3544725
0.0720.0590.136GABA aminotransferase inhibitor

0.097 0.029 CHEMBL1573

0.136 0.011 CHEMBL3544724

0.094 0.032 CHEMBL3544725

CHEMBL3544724
0.0360.0240.036Progesterone antagonist
0.080.070.083C-Like protease (SARS coronavirus) inhibitor

0.08 0.07 CHEMBL3544724

0.0640.0540.073Glutamate (mGluR6) antagonist

0.073 0.034 CHEMBL3544724

CHEMBL3544724
0.1660.1580.352Streptokinase A inhibitor

0.352 0.061 CHEMBL1573

0.337 0.066 CHEMBL3544724

0.196 0.135 CHEMBL3544725

CHEMBL1573
0.0250.0170.036Kainate receptor 4 antagonist

0.026 0.016 CHEMBL1573

0.036 0.011 CHEMBL3544724

CHEMBL3544724
0.0890.0830.089Mediator release inhibitor
0.0680.0630.132NAD(P)H dehydrogenase (quinone) inhibitor

0.095 0.04 CHEMBL1573

0.114 0.031 CHEMBL3544724

0.132 0.025 CHEMBL3544725

CHEMBL3544725
0.0470.0430.047Sodium/calcium exchanger inhibitor
0.040.0360.062GABA B receptor antagonist

0.062 0.011 CHEMBL1573

0.054 0.016 CHEMBL3544724

CHEMBL1573
0.0380.0360.039Kainate receptor agonist

0.039 0.033 CHEMBL3544724

CHEMBL3544724
0.0920.090.106Factor V inhibitor

0.098 0.074 CHEMBL1573

0.106 0.056 CHEMBL3544724

0.096 0.079 CHEMBL3544725

CHEMBL3544724
0.0150.0150.02Kainate receptor 3 antagonist

0.02 0.009 CHEMBL3544724

CHEMBL3544724
0.0520.0530.061Androgen agonist

0.061 0.039 CHEMBL1573

CHEMBL1573
0.0450.0470.091CD45 antagonist

0.059 0.023 CHEMBL1573

0.091 0.01 CHEMBL3544724

0.057 0.025 CHEMBL3544725

CHEMBL3544724
0.0620.0650.207Porphobilinogen synthase inhibitor

0.111 0.031 CHEMBL1573

0.207 0.011 CHEMBL3544724

0.163 0.018 CHEMBL3544725

CHEMBL3544724
0.0230.0260.06NMDA 2D receptor antagonist

0.03 0.016 CHEMBL1573

0.06 0.005 CHEMBL3544724

0.037 0.011 CHEMBL3544725

CHEMBL3544724
0.0770.0820.143Triose-phosphate isomerase inhibitor

0.097 0.051 CHEMBL1573

0.143 0.022 CHEMBL3544724

0.136 0.025 CHEMBL3544725

CHEMBL3544724
0.0740.080.095Thioredoxin reductase inhibitor

0.095 0.033 CHEMBL1573

0.094 0.035 CHEMBL3544724

0.088 0.044 CHEMBL3544725

0.077 0.071 CHEMBL3544726

CHEMBL1573
0.090.0960.112GABA C receptor antagonist

0.101 0.076 CHEMBL1573

0.112 0.061 CHEMBL3544724

CHEMBL3544724
0.0480.0560.057Dihydroorotate oxidase inhibitor

0.057 0.034 CHEMBL3544724

CHEMBL3544724
0.1430.1520.294Histone acetyltransferase inhibitor

0.294 0.015 CHEMBL1573

0.288 0.016 CHEMBL3544724

0.204 0.063 CHEMBL3544725

0.202 0.067 CHEMBL3544726

CHEMBL1573
0.0140.0240.035Kainate receptor 5 antagonist

0.035 0.008 CHEMBL3544724

CHEMBL3544724
0.0570.0670.077Transcription factor RelA inhibitor

0.077 0.02 CHEMBL1573

0.065 0.041 CHEMBL3544724

0.064 0.043 CHEMBL3544726

CHEMBL1573
0.0260.0380.044Catechol O-methyltransferase inhibitor

0.041 0.013 CHEMBL1573

0.041 0.013 CHEMBL3544724

0.044 0.011 CHEMBL3544725

CHEMBL3544725
0.0360.0490.053AICAR transformylase inhibitor

0.046 0.027 CHEMBL1573

0.053 0.019 CHEMBL3544724

CHEMBL3544724
0.0960.1090.181M17 leucyl aminopeptidase inhibitor

0.13 0.069 CHEMBL1573

0.181 0.04 CHEMBL3544724

0.12 0.078 CHEMBL3544725

CHEMBL3544724
0.0430.0570.146Alcohol oxidase inhibitor

0.067 0.03 CHEMBL1573

0.146 0.01 CHEMBL3544724

0.065 0.032 CHEMBL3544725

CHEMBL3544724
0.0750.090.249Breast cancer-resistant protein inhibitor

0.249 0.009 CHEMBL1573

0.193 0.015 CHEMBL3544724

0.136 0.03 CHEMBL3544725

0.216 0.012 CHEMBL3544726

CHEMBL1573
0.0670.0820.07GABA B receptor agonist

0.07 0.069 CHEMBL3544724

CHEMBL3544724
0.10.1160.171Alkaline phosphatase inhibitor

0.163 0.052 CHEMBL1573

0.171 0.047 CHEMBL3544724

0.134 0.072 CHEMBL3544725

CHEMBL3544724
0.1670.1840.199Transcription factor STAT3 inhibitor

0.185 0.156 CHEMBL1573

0.199 0.135 CHEMBL3544724

CHEMBL3544724
0.1720.1910.201Gastrin inhibitor

0.201 0.147 CHEMBL3544724

0.182 0.176 CHEMBL3544725

CHEMBL3544724
0.2040.2240.362Antibacterial

0.248 0.179 CHEMBL1573

0.355 0.099 CHEMBL3544724

0.362 0.095 CHEMBL3544725

CHEMBL3544725
0.1260.1460.135Ca2+-transporting ATPase inhibitor

0.135 0.096 CHEMBL3544724

CHEMBL3544724
0.2560.2770.312Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.306 0.205 CHEMBL1573

0.312 0.197 CHEMBL3544724

CHEMBL3544724
0.1640.1880.396Prostaglandin dehydrogenase inhibitor

0.396 0.068 CHEMBL1573

0.346 0.084 CHEMBL3544724

0.178 0.174 CHEMBL3544725

0.265 0.119 CHEMBL3544726

CHEMBL1573
0.0720.0970.099D-Ala-D-Ala ligase inhibitor

0.086 0.052 CHEMBL1573

0.099 0.03 CHEMBL3544724

CHEMBL3544724
0.0940.120.104Cathepsin H inhibitor

0.103 0.101 CHEMBL1573

0.104 0.1 CHEMBL3544724

CHEMBL3544724
0.0820.1090.133Interleukin 1b antagonist

0.133 0.053 CHEMBL1573

0.122 0.061 CHEMBL3544724

CHEMBL1573
0.0240.0510.048Kainate receptor antagonist

0.048 0.023 CHEMBL3544724

CHEMBL3544724
0.1370.1650.151Free radical scavenger

0.151 0.144 CHEMBL3544724

CHEMBL3544724
0.0240.0540.043Purinergic P2Y2 antagonist

0.034 0.023 CHEMBL3544724

0.043 0.014 CHEMBL3544725

CHEMBL3544725
0.0050.0350.014Angiotensin AT1B receptor antagonist

0.014 0.01 CHEMBL3544724

0.014 0.009 CHEMBL3544725

CHEMBL3544725
0.1170.1490.267DNA methyltransferase I inhibitor

0.198 0.07 CHEMBL1573

0.267 0.039 CHEMBL3544724

0.185 0.077 CHEMBL3544725

CHEMBL3544724
0.0510.0840.071Interferon inducer

0.071 0.034 CHEMBL1573

0.069 0.036 CHEMBL3544724

0.064 0.045 CHEMBL3544725

CHEMBL1573
0.0720.1050.084Thioredoxin inhibitor

0.084 0.073 CHEMBL1573

CHEMBL1573
0.1570.190.218DNA synthesis inhibitor

0.218 0.097 CHEMBL3544724

0.212 0.106 CHEMBL3544725

CHEMBL3544724
0.0490.0840.058Ryanodine receptor antagonist

0.057 0.046 CHEMBL1573

0.058 0.045 CHEMBL3544724

CHEMBL3544724
0.050.0850.072Bcl-xL inhibitor

0.06 0.04 CHEMBL1573

0.061 0.037 CHEMBL3544724

0.072 0.018 CHEMBL3544725

CHEMBL3544725
0.0570.0960.069MDM2 inhibitor

0.063 0.061 CHEMBL1573

0.069 0.042 CHEMBL3544724

CHEMBL3544724
0.0680.1080.079Transcription factor NF kappa B stimulant

0.079 0.073 CHEMBL3544725

CHEMBL3544725
0.030.0760.103Dihydroorotate dehydrogenase inhibitor

0.055 0.033 CHEMBL1573

0.103 0.01 CHEMBL3544724

0.062 0.027 CHEMBL3544725

CHEMBL3544724
0.0340.080.057Argininosuccinate synthase inhibitor

0.057 0.039 CHEMBL3544724

CHEMBL3544724
0.0260.0740.044NMDA receptor subunit 3B antagonist

0.044 0.031 CHEMBL3544724

CHEMBL3544724
0.0670.1150.102Interleukin 5 antagonist

0.092 0.052 CHEMBL1573

0.102 0.039 CHEMBL3544724

0.091 0.053 CHEMBL3544725

CHEMBL3544724
0.0720.1210.155Xanthine oxidase inhibitor

0.091 0.069 CHEMBL1573

0.155 0.033 CHEMBL3544724

0.111 0.052 CHEMBL3544725

CHEMBL3544724
0.0110.0610.042Kynurenine 3 monooxygenase inhibitor

0.023 0.022 CHEMBL1573

0.042 0.009 CHEMBL3544724

CHEMBL3544724
0.0280.0780.057Nerve growth factor antagonist

0.051 0.017 CHEMBL1573

0.057 0.011 CHEMBL3544724

CHEMBL3544724
0.0190.070.038NMDA receptor subunit 3A antagonist

0.038 0.027 CHEMBL3544724

CHEMBL3544724
0.0720.1240.288Anesthetic local

0.288 0.014 CHEMBL1573

0.233 0.024 CHEMBL3544724

0.164 0.043 CHEMBL3544725

CHEMBL1573
0.0120.0650.04AMPA 2 receptor antagonist

0.028 0.022 CHEMBL1573

0.04 0.014 CHEMBL3544724

0.03 0.02 CHEMBL3544725

CHEMBL3544724
0.0180.0720.031Complement factor 1r inhibitor

0.031 0.01 CHEMBL3544726

CHEMBL3544726
0.0550.1120.082Interferon agonist

0.082 0.05 CHEMBL1573

0.081 0.051 CHEMBL3544724

0.074 0.063 CHEMBL3544725

CHEMBL1573
0.2180.2760.3715 Hydroxytryptamine release inhibitor

0.29 0.176 CHEMBL1573

0.371 0.098 CHEMBL3544724

0.243 0.238 CHEMBL3544725

CHEMBL3544724
0.10.1620.128NOS3 expression enhancer

0.128 0.101 CHEMBL3544724

CHEMBL3544724
0.0650.1290.135Ferrochelatase inhibitor

0.135 0.045 CHEMBL3544724

CHEMBL3544724
0.0420.1060.082Na+ K+ transporting ATPase inhibitor

0.082 0.049 CHEMBL1573

0.077 0.053 CHEMBL3544724

0.069 0.061 CHEMBL3544725

CHEMBL1573
0.0980.1640.277Dual specificity phosphatase 3 inhibitor

0.219 0.051 CHEMBL1573

0.277 0.033 CHEMBL3544724

0.245 0.042 CHEMBL3544725

0.138 0.108 CHEMBL3544726

CHEMBL3544724
0.0210.0910.06Angiotensin AT1 receptor antagonist

0.052 0.014 CHEMBL1573

0.059 0.007 CHEMBL3544724

0.06 0.006 CHEMBL3544725

CHEMBL3544725
0.0390.110.108Purinergic P2X1 antagonist

0.073 0.03 CHEMBL1573

0.108 0.014 CHEMBL3544724

0.081 0.025 CHEMBL3544725

CHEMBL3544724
0.0290.1010.059DNA gyrase subunit A inhibitor

0.042 0.03 CHEMBL3544724

0.059 0.01 CHEMBL3544726

CHEMBL3544726
0.0470.120.078Glutamate dehydrogenase inhibitor

0.078 0.047 CHEMBL3544724

CHEMBL3544724
0.0420.1170.077Bcl2 antagonist

0.077 0.034 CHEMBL1573

0.074 0.038 CHEMBL3544724

0.076 0.036 CHEMBL3544725

CHEMBL1573
0.0280.1030.056GABA A receptor antagonist

0.056 0.034 CHEMBL1573

CHEMBL1573
0.0330.1090.077Phosphofructokinase-1 inhibitor

0.077 0.043 CHEMBL3544724

0.073 0.046 CHEMBL3544725

CHEMBL3544724
0.0140.0920.03Fumarate hydratase inhibitor

0.03 0.029 CHEMBL3544724

CHEMBL3544724
0.0230.1020.046Carbonic anhydrase XIV inhibitor

0.046 0.038 CHEMBL3544724

CHEMBL3544724
0.0380.1180.092Carbonic anhydrase XIII inhibitor

0.092 0.042 CHEMBL3544724

0.069 0.059 CHEMBL3544725

CHEMBL3544724
0.0630.1440.114Carbonic anhydrase III inhibitor

0.114 0.048 CHEMBL3544724

0.091 0.073 CHEMBL3544725

CHEMBL3544724
0.0340.1160.071Sphingosine 1-phosphate receptor 4 agonist

0.071 0.044 CHEMBL1573

0.065 0.049 CHEMBL3544724

0.068 0.046 CHEMBL3544725

CHEMBL1573
0.080.1620.213Toll-Like receptor antagonist

0.213 0.026 CHEMBL1573

0.123 0.08 CHEMBL3544724

0.114 0.095 CHEMBL3544725

CHEMBL1573
0.0180.1010.051Angiotensin II receptor antagonist

0.039 0.015 CHEMBL1573

0.05 0.007 CHEMBL3544724

0.051 0.006 CHEMBL3544725

CHEMBL3544725
0.050.1340.07Keratolytic

0.07 0.066 CHEMBL3544724

CHEMBL3544724
0.1370.2210.278Thyroid hormone beta antagonist

0.278 0.1 CHEMBL1573

0.214 0.143 CHEMBL3544724

CHEMBL1573
0.0960.1820.144Heat shock protein 90 alpha antagonist

0.144 0.093 CHEMBL1573

0.134 0.106 CHEMBL3544724

CHEMBL1573
0.0770.1630.167Toll-Like receptor 9 antagonist

0.167 0.053 CHEMBL1573

CHEMBL1573
0.1370.2250.287Thyroid hormone antagonist

0.287 0.1 CHEMBL1573

0.232 0.136 CHEMBL3544724

CHEMBL1573
0.0270.1150.053GABA receptor antagonist

0.053 0.04 CHEMBL1573

0.048 0.047 CHEMBL3544726

CHEMBL1573
0.0180.1080.091AMPA receptor antagonist

0.06 0.025 CHEMBL1573

0.091 0.014 CHEMBL3544724

0.052 0.029 CHEMBL3544725

CHEMBL3544724
0.0970.190.233Dual specificity phosphatase inhibitor

0.177 0.069 CHEMBL1573

0.233 0.042 CHEMBL3544724

0.198 0.056 CHEMBL3544725

CHEMBL3544724
0.0080.1010.029Methionyl aminopeptidase 2 inhibitor

0.029 0.014 CHEMBL3544724

CHEMBL3544724
0.0090.1030.029AMPA 3 receptor antagonist

0.029 0.021 CHEMBL3544724

CHEMBL3544724
0.0890.1840.206Hexokinase inhibitor

0.157 0.071 CHEMBL1573

0.206 0.032 CHEMBL3544724

0.171 0.057 CHEMBL3544725

CHEMBL3544724
0.0310.1250.0573-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.057 0.043 CHEMBL3544724

CHEMBL3544724
0.0260.1210.0413-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.041 0.031 CHEMBL3544724

CHEMBL3544724
0.0480.1450.078Calcium channel P-type blocker

0.078 0.017 CHEMBL1573

0.069 0.031 CHEMBL3544724

CHEMBL1573
0.0560.1560.089GABA C receptor agonist

0.089 0.08 CHEMBL3544724

CHEMBL3544724
0.0470.1480.082Aminopeptidase B inhibitor

0.082 0.08 CHEMBL3544724

CHEMBL3544724
0.0780.180.204Interleukin 1 antagonist

0.204 0.031 CHEMBL1573

0.182 0.041 CHEMBL3544724

0.121 0.087 CHEMBL3544725

0.184 0.04 CHEMBL3544726

CHEMBL1573
0.0270.1290.056Aconitate hydratase inhibitor

0.056 0.031 CHEMBL3544724

CHEMBL3544724
0.1890.2910.43Apoptosis agonist

0.326 0.155 CHEMBL1573

0.313 0.163 CHEMBL3544724

0.31 0.165 CHEMBL3544725

0.43 0.1 CHEMBL3544726

CHEMBL3544726
0.1210.2240.383DNA damaging

0.356 0.039 CHEMBL1573

0.292 0.06 CHEMBL3544724

0.271 0.07 CHEMBL3544725

0.383 0.032 CHEMBL3544726

CHEMBL3544726
0.0420.1450.086Ornithine decarboxylase inhibitor

0.086 0.06 CHEMBL3544724

CHEMBL3544724
0.0640.1670.109Carbonic anhydrase XV inhibitor

0.109 0.057 CHEMBL3544724

0.096 0.072 CHEMBL3544725

CHEMBL3544724
0.0240.1290.053Elastase inhibitor

0.053 0.037 CHEMBL3544726

CHEMBL3544726
0.0290.1350.069Benzodiazepine inverse agonist

0.069 0.01 CHEMBL3544725

CHEMBL3544725
0.0120.1180.043Urate transporter 1 inhibitor

0.043 0.023 CHEMBL3544724

CHEMBL3544724
0.0270.1450.073Prostaglandin-E synthase inhibitor

0.073 0.045 CHEMBL3544724

CHEMBL3544724
0.0290.1470.072Catalase inhibitor

0.072 0.053 CHEMBL3544724

CHEMBL3544724
0.1080.2270.147Phospholipase C inhibitor

0.147 0.112 CHEMBL3544724

CHEMBL3544724
0.0180.1370.079Xanthine dehydrogenase inhibitor

0.079 0.025 CHEMBL3544724

0.055 0.042 CHEMBL3544725

CHEMBL3544724
0.1540.2770.369Histamine release inhibitor

0.222 0.179 CHEMBL1573

0.369 0.091 CHEMBL3544724

0.336 0.106 CHEMBL3544725

CHEMBL3544724
0.1480.2720.293Sodium/bile acid cotransporter inhibitor

0.207 0.179 CHEMBL1573

0.293 0.085 CHEMBL3544724

0.24 0.139 CHEMBL3544725

CHEMBL3544724
0.090.2190.212DNA methylase inhibitor

0.154 0.114 CHEMBL1573

0.212 0.072 CHEMBL3544724

0.142 0.125 CHEMBL3544725

CHEMBL3544724
0.0470.1790.105Creatine kinase inhibitor

0.105 0.054 CHEMBL3544724

CHEMBL3544724
0.0040.1360.021Angiotensin AT1A receptor antagonist

0.021 0.016 CHEMBL3544725

CHEMBL3544725
0.0360.170.069Adenine nucleotide translocase inhibitor

0.069 0.016 CHEMBL3544724

0.067 0.019 CHEMBL3544725

CHEMBL3544724
0.0610.1950.127Alpha-N-acetylglucosaminidase inhibitor

0.127 0.071 CHEMBL3544724

0.122 0.075 CHEMBL3544725

CHEMBL3544724
0.0650.1990.104Aldehyde dehydrogenase inhibitor

0.104 0.091 CHEMBL3544724

CHEMBL3544724
0.0520.1910.221Glutamate receptor antagonist

0.21 0.023 CHEMBL1573

0.221 0.02 CHEMBL3544724

0.183 0.032 CHEMBL3544725

CHEMBL3544724
0.0650.2060.139NADPH oxidase inhibitor

0.13 0.071 CHEMBL1573

0.139 0.063 CHEMBL3544724

CHEMBL3544724
0.0350.1790.122Potassium channel (Ca-activated) activator

0.078 0.077 CHEMBL1573

0.122 0.04 CHEMBL3544724

CHEMBL3544724
0.0250.1720.082HIV-1 integrase (3'-Processing) inhibitor

0.082 0.033 CHEMBL3544724

0.058 0.05 CHEMBL3544725

CHEMBL3544724
0.0530.2010.094Protein kinase C gamma inhibitor

0.094 0.088 CHEMBL3544724

CHEMBL3544724
0.0160.1640.045Retinoic acid alpha receptor agonist

0.045 0.019 CHEMBL3544724

0.037 0.03 CHEMBL3544725

CHEMBL3544724
0.0360.1850.094Phosphodiesterase 3A inhibitor

0.094 0.038 CHEMBL3544726

CHEMBL3544726
0.0730.2250.334Pyruvate kinase inhibitor

0.334 0.039 CHEMBL1573

0.327 0.041 CHEMBL3544724

0.152 0.113 CHEMBL3544725

0.264 0.057 CHEMBL3544726

CHEMBL1573
0.0550.2080.104Caspase 3 inhibitor

0.104 0.085 CHEMBL3544724

CHEMBL3544724
0.0280.1830.085Glutamate decarboxylase inhibitor

0.085 0.039 CHEMBL3544724

CHEMBL3544724
0.080.2360.107DNA repair enzyme inhibitor

0.107 0.104 CHEMBL1573

CHEMBL1573
0.010.170.048Retinoid X alpha receptor agonist

0.048 0.015 CHEMBL3544724

CHEMBL3544724
0.0480.2160.079NADH dehydrogenase inhibitor

0.079 0.077 CHEMBL3544724

CHEMBL3544724
0.170.3410.272MAP kinase 1 inhibitor

0.272 0.21 CHEMBL1573

CHEMBL1573
0.0330.2060.074S-adenosyl-L-methionine decarboxylase inhibitor

0.074 0.05 CHEMBL1573

CHEMBL1573
0.0150.1880.068Neuraminidase inhibitor

0.068 0.035 CHEMBL3544724

0.057 0.047 CHEMBL3544725

CHEMBL3544724
0.0410.2150.118Antineoplastic alkaloid

0.118 0.039 CHEMBL3544726

CHEMBL3544726
0.0450.2190.11Tubulin antagonist

0.11 0.091 CHEMBL3544726

CHEMBL3544726
0.030.210.097Glutamate (mGluR group I) antagonist

0.097 0.027 CHEMBL1573

0.066 0.053 CHEMBL3544724

0.062 0.061 CHEMBL3544725

CHEMBL1573
0.0420.2220.106Cholesterol synthesis inhibitor

0.106 0.08 CHEMBL3544724

CHEMBL3544724
0.0070.1870.041Retinoid X receptor agonist

0.041 0.022 CHEMBL3544724

CHEMBL3544724
0.1020.2840.165Catenin beta inhibitor

0.139 0.133 CHEMBL1573

0.164 0.076 CHEMBL3544724

0.165 0.074 CHEMBL3544726

CHEMBL3544726
0.0390.2250.1DNA intercalator

0.1 0.074 CHEMBL3544726

CHEMBL3544726
0.0320.220.07Macrophage migration inhibitory factor inhibitor

0.07 0.067 CHEMBL3544724

CHEMBL3544724
0.0380.2330.151Glycogen synthase kinase-3 alpha inhibitor

0.151 0.066 CHEMBL1573

0.151 0.066 CHEMBL3544724

CHEMBL3544724
0.0250.2310.09Monophenol monooxygenase inhibitor

0.09 0.083 CHEMBL3544724

CHEMBL3544724
0.0970.3140.136CC chemokine 6 receptor antagonist

0.12 0.116 CHEMBL1573

0.136 0.051 CHEMBL3544724

0.128 0.079 CHEMBL3544725

CHEMBL3544724
0.020.2410.065Neuraminidase (influenza) inhibitor

0.065 0.043 CHEMBL3544724

0.059 0.055 CHEMBL3544725

CHEMBL3544724
0.0910.3120.24Lipoxygenase inhibitor

0.22 0.121 CHEMBL1573

0.24 0.106 CHEMBL3544724

CHEMBL3544724
0.0310.2530.065Potassium channel large-conductance Ca-activated activator

0.065 0.05 CHEMBL3544724

CHEMBL3544724
0.0470.2720.172Protein-tyrosine phosphatase inhibitor

0.16 0.069 CHEMBL3544724

0.172 0.061 CHEMBL3544725

CHEMBL3544725
0.0240.2750.107Glutamate (mGluR) antagonist

0.107 0.031 CHEMBL1573

0.081 0.048 CHEMBL3544724

0.081 0.048 CHEMBL3544725

CHEMBL1573
0.0180.2740.058CDC25B inhibitor

0.058 0.053 CHEMBL3544724

CHEMBL3544724
0.0460.3050.129Antibacterial (Helicobacter pylori)

0.11 0.098 CHEMBL1573

0.129 0.069 CHEMBL3544725

CHEMBL3544725
0.1150.3830.239Caspase 3 stimulant

0.239 0.123 CHEMBL3544726

CHEMBL3544726
0.0250.2930.087Alcohol dehydrogenase inhibitor

0.087 0.068 CHEMBL3544724

CHEMBL3544724
0.0120.3130.053Potassium channel (Inward rectifier) blocker

0.053 0.03 CHEMBL3544726

CHEMBL3544726
0.0420.3460.129Cytokine production inhibitor

0.114 0.096 CHEMBL1573

0.129 0.081 CHEMBL3544726

CHEMBL3544726
0.0050.3320.045Potassium channel (Inward rectifier) 1 blocker

0.045 0.005 CHEMBL3544726

CHEMBL3544726
0.0460.4020.223Platelet adhesion inhibitor

0.163 0.093 CHEMBL1573

0.165 0.091 CHEMBL3544724

0.153 0.103 CHEMBL3544725

0.223 0.06 CHEMBL3544726

CHEMBL3544726
0.0210.3990.131Topoisomerase II inhibitor

0.131 0.059 CHEMBL3544726

CHEMBL3544726
0.0240.4190.096Uric acid excretion stimulant

0.096 0.057 CHEMBL3544724

CHEMBL3544724
0.0120.4450.1095-Lipoxygenase inhibitor

0.096 0.067 CHEMBL1573

0.109 0.057 CHEMBL3544724

CHEMBL3544724
0.0190.4690.084ATPase (Vacuolar H+) inhibitor

0.084 0.07 CHEMBL3544726

CHEMBL3544726
0.0150.4720.187Topoisomerase I inhibitor

0.187 0.03 CHEMBL3544726

CHEMBL3544726
0.020.5150.081Viral attachment inhibitor

0.081 0.047 CHEMBL1573

CHEMBL1573
0.0120.5540.109Topoisomerase II alpha inhibitor

0.109 0.034 CHEMBL3544726

CHEMBL3544726
0.0130.6330.181Potassium channel blocker

0.181 0.106 CHEMBL3544726

CHEMBL3544726
0.030.650.206Immunosuppressant

0.206 0.191 CHEMBL3544724

CHEMBL3544724
0.0120.6330.062Autotaxin inhibitor

0.062 0.027 CHEMBL3544725

CHEMBL3544725
0.030.7080.297Hypoglycemic

0.179 0.135 CHEMBL3544724

0.297 0.054 CHEMBL3544725

CHEMBL3544725
0.0050.6910.074HIV-1 integrase inhibitor

0.074 0.044 CHEMBL3544724

0.066 0.055 CHEMBL3544725

CHEMBL3544724
0.0030.7440.055Potassium channel subfamily K member 3 blocker

0.055 0.011 CHEMBL3544726

CHEMBL3544726
0.0050.9210.289Cyclophilin D inhibitor

0.289 0.173 CHEMBL3544725

CHEMBL3544725
Ext Pa Pi Pmax Activity Other Results ID Pa_max