Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6890.0120.689Antiobesity

0.646 0.015 CHEMBL3526890

0.231 0.176 CHEMBL3526548

0.317 0.105 CHEMBL3526891

0.238 0.169 CHEMBL3527277

0.37 0.078 CHEMBL3527211

0.278 0.133 CHEMBL3527278

0.417 0.059 CHEMBL3526547

0.6570.0020.657Cannabinoid CB1 receptor antagonist

0.455 0.003 CHEMBL3526890

0.143 0.008 CHEMBL3526891

0.187 0.005 CHEMBL3527277

0.101 0.016 CHEMBL3527278

0.292 0.004 CHEMBL3526547

0.6320.0030.632Cannabinoid receptor antagonist

0.399 0.004 CHEMBL3526890

0.14 0.016 CHEMBL3526891

0.152 0.014 CHEMBL3527277

0.086 0.036 CHEMBL3527278

0.278 0.005 CHEMBL3526547

0.4060.0550.406MAP kinase kinase 6 inhibitor

0.372 0.076 CHEMBL3526890

0.229 0.22 CHEMBL3526548

0.278 0.158 CHEMBL3526891

0.284 0.151 CHEMBL3527277

0.249 0.191 CHEMBL3527278

0.386 0.067 CHEMBL3526547

0.3710.1080.562Cyclophilin D inhibitor

0.301 0.162 CHEMBL3526890

0.521 0.044 CHEMBL3526548

0.245 0.218 CHEMBL3526891

0.562 0.035 CHEMBL3527211

CHEMBL3527211
0.2590.0180.359Ribosomal protein S6 kinase inhibitor

0.359 0.006 CHEMBL3526890

0.125 0.085 CHEMBL3526548

0.277 0.015 CHEMBL3526891

0.238 0.024 CHEMBL3527277

0.142 0.071 CHEMBL3527211

0.347 0.007 CHEMBL3527278

0.296 0.012 CHEMBL3526547

CHEMBL3526890
0.2420.0050.565Protein kinase B gamma inhibitor

0.565 0.003 CHEMBL3526890

0.123 0.024 CHEMBL3526548

0.28 0.005 CHEMBL3526891

0.191 0.009 CHEMBL3527277

0.083 0.044 CHEMBL3527211

0.145 0.017 CHEMBL3527278

0.195 0.008 CHEMBL3526547

CHEMBL3526890
0.2240.0040.332Phosphodiesterase II inhibitor

0.273 0.004 CHEMBL3526890

0.133 0.006 CHEMBL3526548

0.261 0.004 CHEMBL3526891

0.217 0.004 CHEMBL3527277

0.106 0.01 CHEMBL3527211

0.294 0.003 CHEMBL3527278

0.332 0.003 CHEMBL3526547

CHEMBL3526547
0.2120.0040.321Phosphodiesterase 2A inhibitor

0.262 0.004 CHEMBL3526890

0.124 0.006 CHEMBL3526548

0.249 0.004 CHEMBL3526891

0.206 0.004 CHEMBL3527277

0.097 0.009 CHEMBL3527211

0.283 0.003 CHEMBL3527278

0.321 0.003 CHEMBL3526547

CHEMBL3526547
0.20.0050.445Protein kinase B alpha inhibitor

0.445 0.003 CHEMBL3526890

0.135 0.013 CHEMBL3526548

0.257 0.004 CHEMBL3526891

0.189 0.005 CHEMBL3527277

0.104 0.028 CHEMBL3527211

0.162 0.006 CHEMBL3527278

0.193 0.005 CHEMBL3526547

CHEMBL3526890
0.2490.0670.431HERG channel blocker

0.431 0.023 CHEMBL3526890

CHEMBL3526890
0.1810.0050.414Protein kinase B beta inhibitor

0.414 0.003 CHEMBL3526890

0.108 0.021 CHEMBL3526548

0.287 0.004 CHEMBL3526891

0.178 0.005 CHEMBL3527277

0.094 0.03 CHEMBL3527211

0.127 0.013 CHEMBL3527278

0.154 0.007 CHEMBL3526547

CHEMBL3526890
0.3080.1350.461Analgesic

0.274 0.163 CHEMBL3526890

0.461 0.061 CHEMBL3526891

CHEMBL3526891
0.2270.0610.247MAP kinase kinase 3 inhibitor

0.247 0.034 CHEMBL3526890

0.19 0.155 CHEMBL3526548

0.218 0.077 CHEMBL3527277

0.192 0.148 CHEMBL3526547

CHEMBL3526890
0.3280.1770.442Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.344 0.157 CHEMBL3526890

0.354 0.146 CHEMBL3526891

0.373 0.126 CHEMBL3527278

0.442 0.067 CHEMBL3526547

CHEMBL3526547
0.2010.0620.314LIM domain kinase 1 inhibitor

0.314 0.018 CHEMBL3526890

0.176 0.076 CHEMBL3526891

0.139 0.11 CHEMBL3526547

CHEMBL3526890
0.140.0040.14Corticotropin releasing factor 2 receptor antagonist

0.107 0.005 CHEMBL3526890

0.066 0.034 CHEMBL3526891

0.071 0.027 CHEMBL3527277

0.082 0.016 CHEMBL3527278

0.128 0.004 CHEMBL3526547

0.2290.0970.25Ca2+/calmodulin-dependent kinase IV inhibitor

0.25 0.065 CHEMBL3526890

0.227 0.102 CHEMBL3526548

0.219 0.118 CHEMBL3526891

0.216 0.124 CHEMBL3527277

0.208 0.144 CHEMBL3527278

0.246 0.071 CHEMBL3526547

CHEMBL3526890
0.2090.080.289ErbB-1 antagonist

0.214 0.076 CHEMBL3526890

0.209 0.08 CHEMBL3526891

0.17 0.132 CHEMBL3527277

0.22 0.07 CHEMBL3527278

0.289 0.036 CHEMBL3526547

CHEMBL3526547
0.1460.0270.221Multidrug resistance-associated protein 1 inhibitor

0.166 0.019 CHEMBL3526890

0.096 0.086 CHEMBL3526548

0.161 0.021 CHEMBL3526891

0.13 0.038 CHEMBL3527277

0.122 0.046 CHEMBL3527211

0.186 0.014 CHEMBL3527278

0.221 0.007 CHEMBL3526547

CHEMBL3526547
0.1240.0180.171Phosphodiesterase XI inhibitor

0.14 0.013 CHEMBL3526890

0.102 0.03 CHEMBL3526891

0.109 0.025 CHEMBL3527277

0.126 0.018 CHEMBL3527278

0.171 0.007 CHEMBL3526547

CHEMBL3526547
0.1240.0180.171Phosphodiesterase 11A inhibitor

0.14 0.013 CHEMBL3526890

0.102 0.03 CHEMBL3526891

0.109 0.025 CHEMBL3527277

0.126 0.018 CHEMBL3527278

0.171 0.007 CHEMBL3526547

CHEMBL3526547
0.1990.0970.368Potassium channel (Voltage-sensitive) blocker

0.368 0.033 CHEMBL3526890

CHEMBL3526890
0.1550.0530.161MAP kinase kinase 4 inhibitor

0.154 0.054 CHEMBL3526890

0.133 0.104 CHEMBL3526548

0.147 0.067 CHEMBL3526891

0.136 0.096 CHEMBL3527277

0.133 0.105 CHEMBL3527278

0.161 0.044 CHEMBL3526547

CHEMBL3526547
0.0990.0040.248LIM domain kinase 2 inhibitor

0.248 0.002 CHEMBL3526890

0.04 0.01 CHEMBL3526548

0.132 0.004 CHEMBL3526891

0.085 0.004 CHEMBL3527277

0.035 0.014 CHEMBL3527211

0.041 0.009 CHEMBL3527278

0.056 0.005 CHEMBL3526547

CHEMBL3526890
0.1950.110.217MAP-kinase-activated kinase 5 inhibitor

0.217 0.085 CHEMBL3526890

0.167 0.154 CHEMBL3527277

0.206 0.096 CHEMBL3526547

CHEMBL3526890
0.1410.0570.18MAP kinase kinase inhibitor

0.125 0.069 CHEMBL3526890

0.18 0.036 CHEMBL3527277

0.107 0.087 CHEMBL3526547

CHEMBL3527277
0.10.0250.387Benzodiazepine agonist

0.114 0.019 CHEMBL3526890

0.087 0.034 CHEMBL3526891

0.067 0.056 CHEMBL3527277

0.137 0.01 CHEMBL3527278

0.387 0.003 CHEMBL3526547

CHEMBL3526547
0.1090.040.23Protein kinase A inhibitor

0.23 0.01 CHEMBL3526890

0.098 0.047 CHEMBL3526891

0.081 0.059 CHEMBL3527277

CHEMBL3526890
0.0930.0260.226Protein kinase C alpha inhibitor

0.226 0.005 CHEMBL3526890

0.106 0.02 CHEMBL3526548

0.167 0.008 CHEMBL3526891

0.076 0.037 CHEMBL3527277

0.075 0.038 CHEMBL3527211

CHEMBL3526890
0.140.0840.237MAP kinase 3 inhibitor

0.144 0.078 CHEMBL3526890

0.13 0.107 CHEMBL3526891

0.202 0.023 CHEMBL3527277

0.237 0.011 CHEMBL3527278

0.162 0.051 CHEMBL3526547

CHEMBL3527278
0.1660.110.429Anticonvulsant

0.158 0.12 CHEMBL3526890

0.159 0.118 CHEMBL3526548

0.429 0.019 CHEMBL3526891

0.162 0.115 CHEMBL3527278

0.364 0.027 CHEMBL3526547

CHEMBL3526891
0.170.1150.281Potassium channel blocker

0.281 0.053 CHEMBL3526890

0.166 0.119 CHEMBL3526547

CHEMBL3526890
0.0810.0280.081Cannabinoid CB1 receptor agonist
0.1010.0560.129Protein kinase C mu inhibitor

0.129 0.037 CHEMBL3526890

0.085 0.073 CHEMBL3526891

CHEMBL3526890
0.1130.0740.175Transcription factor STAT6 inhibitor

0.13 0.044 CHEMBL3526890

0.109 0.083 CHEMBL3526548

0.164 0.015 CHEMBL3527277

0.107 0.088 CHEMBL3527211

0.175 0.011 CHEMBL3527278

0.141 0.031 CHEMBL3526547

CHEMBL3527278
0.2010.1630.391Immunomodulator

0.289 0.088 CHEMBL3526890

0.319 0.072 CHEMBL3526548

0.308 0.078 CHEMBL3526891

0.391 0.047 CHEMBL3527211

CHEMBL3527211
0.1580.1210.161MAP kinase kinase 5 inhibitor

0.161 0.111 CHEMBL3526890

CHEMBL3526890
0.0590.0210.242Phosphodiesterase X inhibitor

0.078 0.014 CHEMBL3526890

0.07 0.016 CHEMBL3526891

0.046 0.03 CHEMBL3527277

0.114 0.009 CHEMBL3527278

0.242 0.004 CHEMBL3526547

CHEMBL3526547
0.0590.0210.242Phosphodiesterase 10A inhibitor

0.078 0.014 CHEMBL3526890

0.07 0.016 CHEMBL3526891

0.046 0.03 CHEMBL3527277

0.114 0.009 CHEMBL3527278

0.242 0.004 CHEMBL3526547

CHEMBL3526547
0.0710.0340.098Phosphodiesterase VII inhibitor

0.08 0.026 CHEMBL3526890

0.075 0.03 CHEMBL3526891

0.061 0.045 CHEMBL3527278

0.098 0.013 CHEMBL3526547

CHEMBL3526547
0.120.0820.434Phosphodiesterase inhibitor

0.155 0.055 CHEMBL3526890

0.141 0.064 CHEMBL3526891

0.137 0.067 CHEMBL3527277

0.258 0.021 CHEMBL3527278

0.434 0.005 CHEMBL3526547

CHEMBL3526547
0.130.0980.282Heat shock protein 90 antagonist

0.127 0.101 CHEMBL3526890

0.175 0.052 CHEMBL3527277

0.282 0.013 CHEMBL3527278

0.174 0.053 CHEMBL3526547

CHEMBL3527278
0.0640.0360.064Bombesin 1 receptor agonist
0.0970.070.189Hedgehog signaling inhibitor

0.109 0.051 CHEMBL3526890

0.094 0.075 CHEMBL3526891

0.109 0.052 CHEMBL3527278

0.189 0.013 CHEMBL3526547

CHEMBL3526547
0.0480.0230.056Dipeptidyl peptidase IV inhibitor

0.056 0.015 CHEMBL3526890

CHEMBL3526890
0.0950.070.139Check point kinase 2 inhibitor

0.139 0.036 CHEMBL3526890

0.089 0.075 CHEMBL3527277

0.106 0.06 CHEMBL3527278

CHEMBL3526890
0.0820.0580.095Transforming growth factor beta 3 antagonist

0.093 0.033 CHEMBL3526890

0.078 0.07 CHEMBL3526891

0.078 0.072 CHEMBL3527277

0.078 0.072 CHEMBL3527278

0.095 0.03 CHEMBL3526547

CHEMBL3526547
0.0620.0390.128Phosphatidylinositol kinase inhibitor

0.088 0.025 CHEMBL3526890

0.052 0.051 CHEMBL3526891

0.052 0.051 CHEMBL3527278

0.128 0.015 CHEMBL3526547

CHEMBL3526547
0.0770.0550.11MAP kinase kinase 7 inhibitor

0.089 0.026 CHEMBL3526890

0.084 0.035 CHEMBL3526891

0.11 0.006 CHEMBL3526547

CHEMBL3526547
0.1550.1370.181Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.181 0.107 CHEMBL3526890

CHEMBL3526890
0.0440.0270.085GHS receptor agonist

0.085 0.006 CHEMBL3526890

CHEMBL3526890
0.0520.0380.085Dipeptidyl peptidase inhibitor

0.085 0.012 CHEMBL3526890

CHEMBL3526890
0.1450.1340.205EphB2 antagonist

0.189 0.095 CHEMBL3526890

0.148 0.131 CHEMBL3526891

0.146 0.134 CHEMBL3527278

0.205 0.085 CHEMBL3526547

CHEMBL3526547
0.0540.0430.115Phosphatidylinositol 3-kinase delta inhibitor

0.086 0.023 CHEMBL3526890

0.052 0.045 CHEMBL3526891

0.049 0.047 CHEMBL3527278

0.115 0.017 CHEMBL3526547

CHEMBL3526547
0.0720.0660.148Platelet growth factor antagonist

0.071 0.067 CHEMBL3526890

0.071 0.067 CHEMBL3527277

0.148 0.02 CHEMBL3526547

CHEMBL3526547
0.010.0050.028Corticotropin releasing factor antagonist

0.01 0.005 CHEMBL3527278

0.028 0.003 CHEMBL3526547

CHEMBL3526547
0.1830.1790.183Ca2+/calmodulin-dependent kinase II alpha inhibitor
0.0480.0450.059Phosphodiesterase 7A inhibitor

0.051 0.039 CHEMBL3526890

0.059 0.023 CHEMBL3526547

CHEMBL3526547
0.0460.0540.0565 Hydroxytryptamine 3 antagonist

0.056 0.041 CHEMBL3526890

0.056 0.04 CHEMBL3526547

CHEMBL3526547
0.0130.0240.017Adenosine A3 receptor agonist

0.017 0.012 CHEMBL3526548

0.017 0.012 CHEMBL3527211

CHEMBL3527211
0.0160.0270.021Corticotropin releasing factor 1 receptor antagonist

0.021 0.017 CHEMBL3526547

CHEMBL3526547
0.0230.0350.027Purinergic P2Y15 antagonist

0.027 0.024 CHEMBL3526890

0.027 0.023 CHEMBL3527277

CHEMBL3527277
0.0940.1080.124Epidermal growth factor receptor kinase inhibitor

0.104 0.092 CHEMBL3526890

0.118 0.074 CHEMBL3527278

0.124 0.069 CHEMBL3526547

CHEMBL3526547
0.0250.0410.046Phosphoglycerate kinase inhibitor

0.046 0.016 CHEMBL3526548

CHEMBL3526548
0.0370.0530.084Phosphatidylinositol 3-kinase alpha inhibitor

0.051 0.036 CHEMBL3526890

0.084 0.02 CHEMBL3526547

CHEMBL3526547
0.0150.0320.034Adenosine A1 receptor agonist

0.034 0.01 CHEMBL3526548

0.031 0.011 CHEMBL3527211

CHEMBL3526548
0.0250.0450.033Potassium channel (Inward rectifier) 1 blocker

0.033 0.014 CHEMBL3526547

CHEMBL3526547
0.040.0610.128Adenosine A1 receptor antagonist

0.102 0.023 CHEMBL3526548

0.128 0.018 CHEMBL3526547

CHEMBL3526547
0.0630.0870.176Phosphodiesterase 3A inhibitor

0.074 0.065 CHEMBL3526890

0.085 0.048 CHEMBL3527278

0.176 0.011 CHEMBL3526547

CHEMBL3526547
0.0380.0630.053Histamine H4 receptor antagonist

0.053 0.026 CHEMBL3526547

CHEMBL3526547
0.0110.040.21Adenosine kinase inhibitor

0.023 0.014 CHEMBL3526890

0.21 0.002 CHEMBL3526548

0.026 0.012 CHEMBL3526891

0.03 0.01 CHEMBL3527211

0.04 0.007 CHEMBL3527278

0.037 0.008 CHEMBL3526547

CHEMBL3526548
0.0810.1130.126mTOR complex 1 inhibitor

0.126 0.023 CHEMBL3526547

CHEMBL3526547
0.0280.060.053Nicotinic acid receptor 1 agonist

0.053 0.019 CHEMBL3526891

0.049 0.021 CHEMBL3526547

CHEMBL3526891
0.0570.090.093Adenosine A3 receptor antagonist

0.093 0.03 CHEMBL3526548

0.074 0.052 CHEMBL3526547

CHEMBL3526548
0.0310.0640.138Phosphodiesterase 4A inhibitor

0.046 0.037 CHEMBL3527277

0.048 0.036 CHEMBL3527278

0.138 0.011 CHEMBL3526547

CHEMBL3526547
0.0090.0430.013Adenosine A2b receptor agonist

0.013 0.012 CHEMBL3526548

CHEMBL3526548
0.110.1520.275Death-associated protein kinase 1 inhibitor

0.123 0.104 CHEMBL3527277

0.275 0.004 CHEMBL3527278

0.126 0.092 CHEMBL3526547

CHEMBL3527278
0.070.1120.105Phosphodiesterase 7B inhibitor

0.091 0.068 CHEMBL3526890

0.102 0.054 CHEMBL3526891

0.105 0.051 CHEMBL3526547

CHEMBL3526547
0.1540.1970.1975 Hydroxytryptamine 3E antagonist

0.197 0.068 CHEMBL3526547

CHEMBL3526547
0.0430.0860.0685 Hydroxytryptamine 3A antagonist

0.068 0.044 CHEMBL3526547

CHEMBL3526547
0.0660.110.104Aminoacyl-tRNA synthetase inhibitor

0.104 0.041 CHEMBL3526548

0.085 0.067 CHEMBL3526891

0.085 0.068 CHEMBL3527211

CHEMBL3526548
0.1510.1980.231RNA-directed DNA polymerase inhibitor

0.231 0.063 CHEMBL3526548

0.192 0.113 CHEMBL3526891

0.222 0.072 CHEMBL3527211

0.207 0.09 CHEMBL3526547

CHEMBL3526548
0.0110.0590.023Purinergic P2X agonist

0.023 0.022 CHEMBL3526548

CHEMBL3526548
0.0160.0640.097Potassium channel small-conductance Ca-activated activator

0.029 0.025 CHEMBL3526890

0.097 0.004 CHEMBL3527278

0.042 0.014 CHEMBL3526547

CHEMBL3527278
0.0540.1040.07Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.07 0.068 CHEMBL3526890

0.07 0.069 CHEMBL3526547

CHEMBL3526547
0.1560.210.378Hypoxia-inducible factor 1 alpha inhibitor

0.184 0.173 CHEMBL3526891

0.235 0.114 CHEMBL3527211

0.261 0.091 CHEMBL3527278

0.378 0.036 CHEMBL3526547

CHEMBL3526547
0.0750.1290.115Protein-tyrosine kinase Lyn inhibitor

0.106 0.096 CHEMBL3526890

0.115 0.089 CHEMBL3526547

CHEMBL3526547
0.0330.0910.074Adenosine A2a receptor antagonist

0.074 0.034 CHEMBL3526547

CHEMBL3526547
0.0360.0950.076Adenosine A2 receptor antagonist

0.076 0.036 CHEMBL3526547

CHEMBL3526547
0.0290.090.066mTOR inhibitor

0.066 0.024 CHEMBL3526547

CHEMBL3526547
0.0550.1160.086ErbB-3 antagonist

0.086 0.053 CHEMBL3526547

CHEMBL3526547
0.1250.1880.151Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.151 0.132 CHEMBL3526547

CHEMBL3526547
0.110.1730.148CF transmembrane conductance regulator agonist

0.135 0.106 CHEMBL3526890

0.148 0.08 CHEMBL3527211

0.144 0.088 CHEMBL3526547

CHEMBL3527211
0.1020.1680.152Clk dual-specificity kinase inhibitor

0.152 0.112 CHEMBL3526547

CHEMBL3526547
0.030.10.061Phosphatidylinositol 3-kinase gamma inhibitor

0.061 0.031 CHEMBL3526547

CHEMBL3526547
0.0940.1650.147CDC-like kinase 4 inhibitor

0.147 0.103 CHEMBL3526547

CHEMBL3526547
0.0720.1430.389Glutamate receptor antagonist

0.107 0.089 CHEMBL3526890

0.389 0.005 CHEMBL3526891

0.113 0.082 CHEMBL3527278

CHEMBL3526891
0.040.1120.196Phosphodiesterase 4D inhibitor

0.07 0.055 CHEMBL3527278

0.196 0.011 CHEMBL3526547

CHEMBL3526547
0.0380.1110.061Phosphodiesterase 1B inhibitor

0.061 0.041 CHEMBL3526547

CHEMBL3526547
0.0640.150.101RET inhibitor

0.101 0.096 CHEMBL3527278

CHEMBL3527278
0.0570.1470.097Phosphodiesterase I inhibitor

0.097 0.048 CHEMBL3526547

CHEMBL3526547
0.0420.1330.113Platelet activating factor beta antagonist

0.113 0.054 CHEMBL3526547

CHEMBL3526547
0.0360.1310.109Cyclin B3 inhibitor

0.109 0.025 CHEMBL3527278

0.064 0.051 CHEMBL3526547

CHEMBL3527278
0.0250.1220.046Diacylglycerol O-acyltransferase inhibitor

0.046 0.042 CHEMBL3526547

CHEMBL3526547
0.030.1270.063Toll-Like receptor 7 antagonist

0.063 0.052 CHEMBL3526890

CHEMBL3526890
0.0450.1420.075Histamine N-methyltransferase inhibitor

0.075 0.073 CHEMBL3526547

CHEMBL3526547
0.020.1210.044Tryptophan 5 hydroxylase inhibitor

0.044 0.01 CHEMBL3526891

CHEMBL3526891
0.0540.160.096c-Src kinase inhibitor

0.096 0.093 CHEMBL3526547

CHEMBL3526547
0.0250.1320.048Benzodiazepine antagonist

0.048 0.03 CHEMBL3526547

CHEMBL3526547
0.0510.160.093Ephrin antagonist

0.093 0.069 CHEMBL3526547

CHEMBL3526547
0.0340.1460.0745 Hydroxytryptamine 3 agonist

0.074 0.032 CHEMBL3526890

0.058 0.052 CHEMBL3526891

0.059 0.049 CHEMBL3526547

CHEMBL3526890
0.0250.1370.049Pim-2 kinase inhibitor

0.049 0.047 CHEMBL3526890

CHEMBL3526890
0.0340.1460.118Rho-associated kinase inhibitor

0.118 0.027 CHEMBL3526890

CHEMBL3526890
0.070.1880.193CDK3/cyclin E inhibitor

0.193 0.008 CHEMBL3526548

0.129 0.044 CHEMBL3527278

CHEMBL3526548
0.0230.1420.22GABA receptor antagonist

0.22 0.005 CHEMBL3526547

CHEMBL3526547
0.0220.1420.111Phosphodiesterase 4C inhibitor

0.111 0.012 CHEMBL3526547

CHEMBL3526547
0.0260.1520.061Cyclin B1 inhibitor

0.061 0.042 CHEMBL3527278

CHEMBL3527278
0.0620.1920.093T cell inhibitor

0.093 0.033 CHEMBL3526547

CHEMBL3526547
0.0540.1880.094mTOR complex 2 inhibitor

0.077 0.076 CHEMBL3526890

0.094 0.04 CHEMBL3526547

CHEMBL3526547
0.0350.170.23Glutamate (mGluR) antagonist

0.073 0.057 CHEMBL3526890

0.23 0.008 CHEMBL3526891

CHEMBL3526891
0.0230.160.051Cyclin B inhibitor

0.051 0.045 CHEMBL3527278

CHEMBL3527278
0.0230.1620.072Potassium channel small-conductance Ca-activated blocker

0.072 0.012 CHEMBL3526547

CHEMBL3526547
0.0340.1750.133Rho-associated kinase II inhibitor

0.133 0.021 CHEMBL3526890

CHEMBL3526890
0.0210.1640.227GABA A receptor antagonist

0.227 0.005 CHEMBL3526547

CHEMBL3526547
0.0430.1870.121Glycogen synthase kinase-3 beta inhibitor

0.121 0.06 CHEMBL3527278

CHEMBL3527278
0.0210.170.104Purinergic P2X2 antagonist

0.104 0.028 CHEMBL3527278

CHEMBL3527278
0.1460.2970.355GABA C receptor rho-3 antagonist

0.211 0.194 CHEMBL3527278

0.355 0.083 CHEMBL3526547

CHEMBL3526547
0.0790.2340.165Heat shock protein 90 alpha antagonist

0.165 0.073 CHEMBL3527278

CHEMBL3527278
0.0240.1810.087Phosphodiesterase III inhibitor

0.087 0.03 CHEMBL3526547

CHEMBL3526547
0.0420.2020.133Glycogen synthase kinase-3 inhibitor

0.133 0.053 CHEMBL3527278

CHEMBL3527278
0.0460.2120.1375 Hydroxytryptamine 3A agonist

0.137 0.043 CHEMBL3526547

CHEMBL3526547
0.030.2010.077Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.077 0.075 CHEMBL3527278

CHEMBL3527278
0.0470.2270.143NADH dehydrogenase inhibitor

0.093 0.052 CHEMBL3526548

0.105 0.039 CHEMBL3526891

0.143 0.019 CHEMBL3527211

0.093 0.053 CHEMBL3526547

CHEMBL3527211
0.0180.20.052EphB4 antagonist

0.052 0.047 CHEMBL3526547

CHEMBL3526547
0.0780.2610.35Aldehyde oxidase inhibitor

0.188 0.111 CHEMBL3526891

0.35 0.055 CHEMBL3526547

CHEMBL3526547
0.1190.3090.256Peptidyltransferase inhibitor

0.184 0.122 CHEMBL3526548

0.256 0.047 CHEMBL3527211

CHEMBL3527211
0.0350.2260.097Platelet activating factor antagonist

0.097 0.081 CHEMBL3526547

CHEMBL3526547
0.0430.2360.218GABA receptor agonist

0.218 0.014 CHEMBL3526547

CHEMBL3526547
0.1060.3020.214Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.205 0.068 CHEMBL3526548

0.159 0.128 CHEMBL3527211

0.214 0.061 CHEMBL3526547

CHEMBL3526547
0.080.2790.268Antipruritic

0.164 0.079 CHEMBL3526890

0.268 0.02 CHEMBL3526891

CHEMBL3526891
0.0210.2220.083Phosphodiesterase 5A inhibitor

0.083 0.037 CHEMBL3526547

CHEMBL3526547
0.0050.2070.023Aggrecanase 2 inhibitor

0.023 0.014 CHEMBL3526891

CHEMBL3526891
0.0070.210.028Protocollagen prolyl hydroxylase inhibitor

0.028 0.018 CHEMBL3526547

CHEMBL3526547
0.0190.2330.082Phosphodiesterase V inhibitor

0.082 0.039 CHEMBL3526547

CHEMBL3526547
0.020.2420.094CDK2/cyclin E2 inhibitor

0.064 0.057 CHEMBL3526548

0.094 0.03 CHEMBL3527278

CHEMBL3527278
0.0680.2970.152Death-associated protein kinase 3 inhibitor

0.152 0.12 CHEMBL3527278

CHEMBL3527278
0.0910.3210.362Death-associated protein kinase 2 inhibitor

0.362 0.004 CHEMBL3527278

CHEMBL3527278
0.0270.2650.071Acetylcholine M3 receptor agonist

0.071 0.07 CHEMBL3527278

CHEMBL3527278
0.0520.2920.127Interleukin 12 antagonist

0.127 0.023 CHEMBL3526547

CHEMBL3526547
0.0830.3270.29Cyclic AMP phosphodiesterase inhibitor

0.29 0.046 CHEMBL3526548

0.228 0.075 CHEMBL3527278

0.226 0.077 CHEMBL3526547

CHEMBL3526548
0.0080.2550.025Protein 30S ribosomal subunit inhibitor

0.025 0.015 CHEMBL3527211

CHEMBL3527211
0.0160.2650.056Antibiotic Aminoglycoside-like

0.04 0.021 CHEMBL3526548

0.056 0.01 CHEMBL3527211

CHEMBL3527211
0.0150.270.095Phosphodiesterase 4B inhibitor

0.095 0.027 CHEMBL3526547

CHEMBL3526547
0.0370.2950.112Toll-Like receptor 9 antagonist

0.112 0.095 CHEMBL3526547

CHEMBL3526547
0.0340.2940.111Protein kinase C gamma inhibitor

0.111 0.062 CHEMBL3526890

CHEMBL3526890
0.0340.2940.075MAP kinase kinase 8 inhibitor

0.075 0.039 CHEMBL3527278

CHEMBL3527278
0.0310.2910.119GABA A receptor agonist

0.119 0.024 CHEMBL3526547

CHEMBL3526547
0.1510.4140.557Antiinflammatory

0.391 0.144 CHEMBL3526548

0.557 0.066 CHEMBL3527211

CHEMBL3527211
0.0160.2850.091Glutamate (mGluR8) antagonist

0.042 0.015 CHEMBL3526890

0.091 0.003 CHEMBL3526891

CHEMBL3526891
0.0370.3130.106Sodium channel blocker

0.106 0.104 CHEMBL3526890

CHEMBL3526890
0.0530.3340.163Aurora-C kinase inhibitor

0.163 0.038 CHEMBL3527278

CHEMBL3527278
0.0310.3160.078Phosphodiesterase VI inhibitor

0.078 0.044 CHEMBL3526547

CHEMBL3526547
0.0540.3520.264Interleukin agonist

0.264 0.069 CHEMBL3527211

CHEMBL3527211
0.0050.3030.178Glutamate (mGluR2) agonist

0.028 0.027 CHEMBL3526890

0.178 0.004 CHEMBL3526891

CHEMBL3526891
0.0970.3970.207Toll-Like receptor 7 agonist

0.207 0.193 CHEMBL3526890

CHEMBL3526890
0.0080.3110.207Glutamate (mGluR group II) agonist

0.032 0.027 CHEMBL3526890

0.207 0.004 CHEMBL3526891

CHEMBL3526891
0.0610.3640.132DNA repair enzyme inhibitor

0.132 0.051 CHEMBL3527211

CHEMBL3527211
0.0140.3190.145Phosphodiesterase IV inhibitor

0.076 0.066 CHEMBL3527278

0.145 0.024 CHEMBL3526547

CHEMBL3526547
0.0980.4040.136Heat shock protein 70 antagonist

0.129 0.126 CHEMBL3526891

0.136 0.093 CHEMBL3526547

CHEMBL3526547
0.0140.3230.052Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.052 0.045 CHEMBL3527211

CHEMBL3527211
0.0460.3560.093Adenylate kinase inhibitor

0.093 0.081 CHEMBL3526891

CHEMBL3526891
0.0930.4070.202Toll-Like receptor agonist

0.202 0.199 CHEMBL3526890

CHEMBL3526890
0.0650.3910.177Focal adhesion kinase 2 inhibitor

0.177 0.091 CHEMBL3526547

CHEMBL3526547
0.0190.350.039Glucagon-like peptide 1 receptor antagonist

0.039 0.028 CHEMBL3526891

CHEMBL3526891
0.0840.4160.214Nootropic

0.214 0.141 CHEMBL3526890

CHEMBL3526890
0.0170.3540.118MAP kinase kinase 10 inhibitor

0.118 0.015 CHEMBL3527278

CHEMBL3527278
0.0210.360.091Glucosylceramidase inhibitor

0.091 0.011 CHEMBL3526548

CHEMBL3526548
0.0560.3960.155Pregnane X receptor agonist

0.155 0.045 CHEMBL3526547

CHEMBL3526547
0.0110.3580.093NMDA receptor antagonist

0.093 0.051 CHEMBL3526891

CHEMBL3526891
0.0210.370.15Ca(v)2.2 blocker

0.15 0.029 CHEMBL3527278

CHEMBL3527278
0.0480.3980.192Hexokinase inhibitor

0.142 0.088 CHEMBL3526891

0.192 0.04 CHEMBL3527211

0.155 0.073 CHEMBL3526547

CHEMBL3527211
0.010.3630.043Adenosine deaminase inhibitor

0.043 0.037 CHEMBL3527211

CHEMBL3527211
0.0120.3720.068MAP kinase 10 inhibitor

0.068 0.067 CHEMBL3527278

CHEMBL3527278
0.0430.4090.206Prostaglandin dehydrogenase inhibitor

0.206 0.152 CHEMBL3526547

CHEMBL3526547
0.0130.380.127Acid-sensing ion channel blocker

0.127 0.003 CHEMBL3527278

CHEMBL3527278
0.0040.3730.051Glutamate (mGluR group II) antagonist

0.051 0.015 CHEMBL3526891

CHEMBL3526891
0.0030.3750.029Glutamate (mGluR2) antagonist

0.029 0.022 CHEMBL3526891

CHEMBL3526891
0.0330.4160.096Lanosterol 14 alpha demethylase inhibitor

0.096 0.062 CHEMBL3527278

CHEMBL3527278
0.0240.4180.157Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.157 0.125 CHEMBL3527278

CHEMBL3527278
0.0240.4190.151Dyrk kinase inhibitor

0.151 0.135 CHEMBL3527278

CHEMBL3527278
0.0070.4090.334Glutamate (mGluR) agonist

0.334 0.005 CHEMBL3526891

CHEMBL3526891
0.0050.4230.053Opioid kappa receptor agonist

0.053 0.022 CHEMBL3526891

CHEMBL3526891
0.0290.4630.114DNA polymerase I inhibitor

0.114 0.073 CHEMBL3526548

0.114 0.073 CHEMBL3527211

CHEMBL3527211
0.0260.4790.154Acetylcholine M1 receptor antagonist

0.154 0.07 CHEMBL3527278

CHEMBL3527278
0.0410.4940.393DNA synthesis inhibitor

0.393 0.022 CHEMBL3526548

0.294 0.046 CHEMBL3526891

0.281 0.05 CHEMBL3527211

CHEMBL3526548
0.0060.4740.0835 Hydroxytryptamine 1F antagonist

0.083 0.041 CHEMBL3527278

CHEMBL3527278
0.0050.4850.066Glutamate (mGluR3) antagonist

0.066 0.007 CHEMBL3526891

CHEMBL3526891
0.0210.5020.063Glutamate (mGluR6) antagonist

0.063 0.057 CHEMBL3526891

CHEMBL3526891
0.0690.5530.238Calcium channel activator

0.238 0.162 CHEMBL3526547

CHEMBL3526547
0.010.4950.052Protein 50S ribosomal subunit inhibitor

0.052 0.038 CHEMBL3527211

CHEMBL3527211
0.0330.5230.139Platelet adhesion inhibitor

0.139 0.119 CHEMBL3527211

CHEMBL3527211
0.0130.5190.045Glutamate (mGluR4) antagonist

0.045 0.028 CHEMBL3526891

CHEMBL3526891
0.0050.5160.068Phosphofructokinase-1 inhibitor

0.068 0.05 CHEMBL3527211

CHEMBL3527211
0.0790.5990.356Interleukin 2 agonist

0.245 0.125 CHEMBL3526548

0.356 0.043 CHEMBL3527211

CHEMBL3527211
0.0380.5760.281Immunosuppressant

0.231 0.165 CHEMBL3526548

0.263 0.138 CHEMBL3526891

0.281 0.127 CHEMBL3527211

CHEMBL3527211
0.0030.5490.043Phosphorylase inhibitor

0.043 0.035 CHEMBL3526548

CHEMBL3526548
0.0050.5970.172Selectin antagonist

0.085 0.034 CHEMBL3526548

0.172 0.015 CHEMBL3527211

CHEMBL3527211
0.0140.6230.326Immunostimulant

0.2 0.12 CHEMBL3526548

0.326 0.071 CHEMBL3527211

CHEMBL3527211
0.0090.6250.092Topoisomerase I inhibitor

0.092 0.078 CHEMBL3527211

CHEMBL3527211
0.0030.6210.032Dipeptidyl peptidase I inhibitor

0.032 0.02 CHEMBL3526890

CHEMBL3526890
0.0040.6340.022Histone deacetylase 6 inhibitor

0.022 0.021 CHEMBL3527277

CHEMBL3527277
0.0080.6520.04Glutamate (mGluR group III) antagonist

0.04 0.038 CHEMBL3526891

CHEMBL3526891
0.0220.7060.397Antibacterial

0.397 0.078 CHEMBL3527211

CHEMBL3527211
0.0040.6980.026Histone deacetylase class II inhibitor

0.026 0.023 CHEMBL3527277

CHEMBL3527277
0.010.7090.17Free radical scavenger

0.17 0.124 CHEMBL3527211

CHEMBL3527211
0.040.7610.196Lipocortins synthesis antagonist

0.196 0.059 CHEMBL3527278

CHEMBL3527278
0.0050.730.052Alpha-mannosidase inhibitor

0.052 0.04 CHEMBL3527211

CHEMBL3527211
0.0030.7480.041Mannosidase inhibitor

0.041 0.038 CHEMBL3527211

CHEMBL3527211
0.0230.7850.086Transcription factor NF kappa B stimulant

0.086 0.058 CHEMBL3527211

CHEMBL3527211
0.0110.7740.409Angiogenesis stimulant

0.409 0.02 CHEMBL3527211

CHEMBL3527211
0.0270.8150.123NOS3 expression enhancer

0.123 0.109 CHEMBL3527211

CHEMBL3527211
0.0070.7970.194Antioxidant

0.194 0.119 CHEMBL3527211

CHEMBL3527211
0.0150.8090.1Toll-Like receptor 4 antagonist

0.1 0.069 CHEMBL3527211

CHEMBL3527211
0.0030.8030.116Antineoplastic antibiotic

0.116 0.04 CHEMBL3527211

CHEMBL3527211
0.020.8390.186Hepatoprotectant

0.186 0.074 CHEMBL3527211

CHEMBL3527211
0.0120.8750.198Hypoglycemic

0.198 0.115 CHEMBL3527211

CHEMBL3527211
0.020.8930.241Apoptosis antagonist

0.241 0.137 CHEMBL3527211

CHEMBL3527211
0.0050.9010.137Nitric oxide antagonist

0.137 0.109 CHEMBL3527211

CHEMBL3527211
0.0080.9130.245Apoptosis agonist

0.245 0.22 CHEMBL3527211

CHEMBL3527211
Ext Pa Pi Pmax Activity Other Results ID Pa_max