| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.95 | 0.001 | 0.95 | Peroxisome proliferator-activated receptor gamma antagonist | 0.924 0.001 CHEMBL3526971 0.84 0.001 CHEMBL3526634 0.311 0.003 CHEMBL4525745 0.884 0.001 CHEMBL3526633 0.322 0.003 CHEMBL3526795 0.806 0.001 CHEMBL3526627 0.754 0.001 CHEMBL3526722 0.794 0.001 CHEMBL3526723 | ||
| 0.915 | 0.002 | 0.92 | Peroxisome proliferator-activated receptor gamma agonist | 0.92 0.002 CHEMBL3526971 0.805 0.002 CHEMBL3526634 0.317 0.004 CHEMBL4525745 0.898 0.002 CHEMBL3526633 0.755 0.002 CHEMBL3526795 0.866 0.002 CHEMBL3526627 0.873 0.002 CHEMBL3526722 0.811 0.002 CHEMBL3526723 | CHEMBL3526971 | |
| 0.901 | 0.005 | 0.927 | Cyclophilin D inhibitor | 0.911 0.005 CHEMBL3526971 0.917 0.004 CHEMBL3526634 0.518 0.045 CHEMBL4525745 0.895 0.005 CHEMBL3526633 0.913 0.004 CHEMBL3526795 0.882 0.005 CHEMBL3526627 0.894 0.005 CHEMBL3526722 0.927 0.004 CHEMBL3526723 | CHEMBL3526723 | |
| 0.85 | 0.001 | 0.85 | Peroxisome proliferator-activated receptor alpha agonist | 0.772 0.001 CHEMBL3526971 0.665 0.002 CHEMBL3526634 0.194 0.004 CHEMBL4525745 0.752 0.001 CHEMBL3526633 0.288 0.003 CHEMBL3526795 0.792 0.001 CHEMBL3526627 0.707 0.001 CHEMBL3526722 0.586 0.002 CHEMBL3526723 | ||
| 0.765 | 0.004 | 0.798 | Hypoglycemic | 0.786 0.004 CHEMBL3526971 0.684 0.005 CHEMBL3526634 0.376 0.032 CHEMBL4525745 0.764 0.004 CHEMBL3526633 0.798 0.004 CHEMBL3526795 0.71 0.005 CHEMBL3526627 0.726 0.005 CHEMBL3526722 0.708 0.005 CHEMBL3526723 | CHEMBL3526795 | |
| 0.717 | 0.005 | 0.745 | Hypolipemic | 0.732 0.004 CHEMBL3526971 0.733 0.004 CHEMBL3526634 0.387 0.028 CHEMBL4525745 0.704 0.005 CHEMBL3526633 0.661 0.005 CHEMBL3526795 0.659 0.005 CHEMBL3526627 0.675 0.005 CHEMBL3526722 0.745 0.004 CHEMBL3526723 | CHEMBL3526723 | |
| 0.705 | 0.002 | 0.741 | Insulin sensitizer | 0.741 0.002 CHEMBL3526971 0.63 0.003 CHEMBL3526634 0.273 0.023 CHEMBL4525745 0.697 0.003 CHEMBL3526633 0.462 0.004 CHEMBL3526795 0.494 0.004 CHEMBL3526627 0.522 0.004 CHEMBL3526722 0.669 0.003 CHEMBL3526723 | CHEMBL3526971 | |
| 0.694 | 0.001 | 0.694 | Peroxisome proliferator-activated receptor alpha antagonist | 0.669 0.001 CHEMBL3526971 0.272 0.002 CHEMBL3526634 0.072 0.006 CHEMBL4525745 0.556 0.001 CHEMBL3526633 0.113 0.004 CHEMBL3526795 0.6 0.001 CHEMBL3526627 0.568 0.001 CHEMBL3526722 0.26 0.002 CHEMBL3526723 | ||
| 0.687 | 0.012 | 0.708 | Antiobesity | 0.708 0.01 CHEMBL3526971 0.614 0.019 CHEMBL3526634 0.386 0.071 CHEMBL4525745 0.657 0.014 CHEMBL3526633 0.619 0.018 CHEMBL3526795 0.562 0.026 CHEMBL3526627 0.588 0.022 CHEMBL3526722 0.64 0.016 CHEMBL3526723 | CHEMBL3526971 | |
| 0.312 | 0.084 | 0.508 | Cholesterol antagonist | 0.361 0.06 CHEMBL3526971 0.274 0.109 CHEMBL3526634 0.335 0.071 CHEMBL4525745 0.335 0.071 CHEMBL3526633 0.508 0.031 CHEMBL3526795 0.344 0.067 CHEMBL3526627 0.409 0.047 CHEMBL3526722 0.32 0.079 CHEMBL3526723 | CHEMBL3526795 | |
| 0.304 | 0.076 | 0.377 | Sodium/bile acid cotransporter inhibitor | 0.325 0.058 CHEMBL3526971 0.315 0.066 CHEMBL3526634 0.377 0.025 CHEMBL4525745 0.323 0.059 CHEMBL3526633 0.288 0.091 CHEMBL3526627 0.312 0.069 CHEMBL3526722 0.334 0.051 CHEMBL3526723 | CHEMBL4525745 | |
| 0.258 | 0.045 | 0.333 | Peptidyltransferase inhibitor | 0.277 0.034 CHEMBL3526971 0.291 0.028 CHEMBL3526634 0.305 0.023 CHEMBL4525745 0.266 0.04 CHEMBL3526633 0.333 0.015 CHEMBL3526795 0.246 0.053 CHEMBL3526627 0.266 0.041 CHEMBL3526722 0.307 0.022 CHEMBL3526723 | CHEMBL3526795 | |
| 0.216 | 0.029 | 0.248 | Insulin secretagoues | 0.226 0.025 CHEMBL3526971 0.122 0.108 CHEMBL3526634 0.122 0.108 CHEMBL4525745 0.211 0.03 CHEMBL3526633 0.248 0.02 CHEMBL3526795 0.187 0.043 CHEMBL3526627 0.196 0.038 CHEMBL3526722 0.13 0.097 CHEMBL3526723 | CHEMBL3526795 | |
| 0.21 | 0.023 | 0.333 | Chelator | 0.267 0.014 CHEMBL3526971 0.183 0.028 CHEMBL3526634 0.333 0.009 CHEMBL4525745 0.246 0.017 CHEMBL3526633 0.112 0.061 CHEMBL3526795 0.191 0.026 CHEMBL3526627 0.25 0.016 CHEMBL3526722 0.244 0.017 CHEMBL3526723 | CHEMBL4525745 | |
| 0.216 | 0.041 | 0.245 | Protein-tyrosine phosphatase inhibitor | 0.245 0.032 CHEMBL3526971 0.23 0.037 CHEMBL3526633 0.199 0.047 CHEMBL3526795 0.195 0.049 CHEMBL3526627 0.224 0.038 CHEMBL3526722 0.129 0.103 CHEMBL3526723 | CHEMBL3526971 | |
| 0.195 | 0.034 | 0.265 | Acetylcholinesterase inhibitor | 0.183 0.039 CHEMBL3526971 0.148 0.056 CHEMBL3526634 0.265 0.018 CHEMBL4525745 0.193 0.035 CHEMBL3526633 0.111 0.088 CHEMBL3526795 0.186 0.038 CHEMBL3526627 0.174 0.042 CHEMBL3526722 0.138 0.063 CHEMBL3526723 | CHEMBL4525745 | |
| 0.173 | 0.037 | 0.198 | Protein-tyrosine phosphatase 1B inhibitor | 0.198 0.03 CHEMBL3526971 0.186 0.033 CHEMBL3526633 0.183 0.034 CHEMBL3526795 0.149 0.046 CHEMBL3526627 0.174 0.037 CHEMBL3526722 | CHEMBL3526971 | |
| 0.139 | 0.005 | 0.265 | Peroxisome proliferator-activated receptor delta antagonist | 0.145 0.005 CHEMBL3526971 0.034 0.022 CHEMBL3526634 0.114 0.005 CHEMBL3526633 0.044 0.012 CHEMBL3526795 0.261 0.004 CHEMBL3526627 0.265 0.004 CHEMBL3526722 0.034 0.022 CHEMBL3526723 | CHEMBL3526722 | |
| 0.174 | 0.06 | 0.223 | Cholinergic | 0.161 0.068 CHEMBL3526971 0.119 0.109 CHEMBL3526634 0.223 0.037 CHEMBL4525745 0.168 0.064 CHEMBL3526633 0.164 0.067 CHEMBL3526627 0.151 0.076 CHEMBL3526722 | CHEMBL4525745 | |
| 0.223 | 0.119 | 0.28 | Lipoxygenase inhibitor | 0.266 0.09 CHEMBL3526971 0.28 0.081 CHEMBL3526633 0.184 0.158 CHEMBL3526627 0.219 0.122 CHEMBL3526722 | CHEMBL3526633 | |
| 0.141 | 0.038 | 0.27 | Butyrylcholinesterase inhibitor | 0.132 0.041 CHEMBL3526971 0.11 0.054 CHEMBL3526634 0.27 0.013 CHEMBL4525745 0.135 0.04 CHEMBL3526633 0.128 0.043 CHEMBL3526627 0.12 0.047 CHEMBL3526722 0.103 0.059 CHEMBL3526723 | CHEMBL4525745 | |
| 0.11 | 0.009 | 0.11 | Phosphodiesterase VIII inhibitor | 0.109 0.01 CHEMBL3526971 0.108 0.01 CHEMBL3526634 0.106 0.011 CHEMBL3526633 0.09 0.022 CHEMBL3526795 0.078 0.038 CHEMBL3526627 0.075 0.043 CHEMBL3526722 0.107 0.011 CHEMBL3526723 | ||
| 0.081 | 0.007 | 0.081 | Peroxisome proliferator-activated receptor delta agonist | 0.051 0.012 CHEMBL3526971 0.048 0.013 CHEMBL3526633 0.053 0.012 CHEMBL3526627 0.037 0.02 CHEMBL3526722 | ||
| 0.098 | 0.034 | 0.098 | Phosphodiesterase 11A inhibitor | 0.081 0.057 CHEMBL3526971 0.086 0.049 CHEMBL3526634 0.09 0.042 CHEMBL3526633 0.085 0.05 CHEMBL3526627 | ||
| 0.098 | 0.034 | 0.098 | Phosphodiesterase XI inhibitor | 0.081 0.057 CHEMBL3526971 0.086 0.049 CHEMBL3526634 0.09 0.042 CHEMBL3526633 0.085 0.05 CHEMBL3526627 | ||
| 0.066 | 0.004 | 0.238 | Thiazolidinedione | 0.065 0.004 CHEMBL3526971 0.237 0.001 CHEMBL3526634 0.063 0.004 CHEMBL3526633 0.046 0.006 CHEMBL3526795 0.054 0.005 CHEMBL3526627 0.052 0.005 CHEMBL3526722 0.238 0.001 CHEMBL3526723 | CHEMBL3526723 | |
| 0.186 | 0.126 | 0.472 | Antioxidant | 0.237 0.091 CHEMBL3526971 0.162 0.151 CHEMBL3526634 0.164 0.148 CHEMBL4525745 0.247 0.086 CHEMBL3526633 0.472 0.024 CHEMBL3526795 0.203 0.111 CHEMBL3526627 0.254 0.081 CHEMBL3526722 0.207 0.109 CHEMBL3526723 | CHEMBL3526795 | |
| 0.153 | 0.106 | 0.271 | Amyloid beta aggregation inhibitor | 0.177 0.09 CHEMBL3526971 0.271 0.052 CHEMBL4525745 0.2 0.078 CHEMBL3526633 0.171 0.094 CHEMBL3526795 0.14 0.116 CHEMBL3526627 0.162 0.1 CHEMBL3526722 | CHEMBL4525745 | |
| 0.057 | 0.025 | 0.071 | Antiviral (Hepatitis D) | 0.054 0.029 CHEMBL3526971 0.057 0.025 CHEMBL3526634 0.071 0.013 CHEMBL4525745 0.055 0.029 CHEMBL3526633 0.06 0.022 CHEMBL3526627 0.057 0.026 CHEMBL3526722 0.054 0.029 CHEMBL3526723 | CHEMBL4525745 | |
| 0.202 | 0.176 | 0.32 | Apoptosis antagonist | 0.222 0.154 CHEMBL3526971 0.281 0.099 CHEMBL4525745 0.228 0.149 CHEMBL3526633 0.32 0.073 CHEMBL3526795 0.279 0.101 CHEMBL3526627 0.295 0.089 CHEMBL3526722 0.2 0.18 CHEMBL3526723 | CHEMBL3526795 | |
| 0.068 | 0.047 | 0.089 | Potassium channel large-conductance Ca-activated activator | 0.079 0.036 CHEMBL3526971 0.062 0.056 CHEMBL4525745 0.075 0.039 CHEMBL3526633 0.089 0.029 CHEMBL3526795 0.066 0.049 CHEMBL3526722 0.064 0.052 CHEMBL3526723 | CHEMBL3526795 | |
| 0.088 | 0.076 | 0.102 | Interleukin 12 antagonist | 0.101 0.051 CHEMBL3526971 0.1 0.054 CHEMBL3526633 0.096 0.06 CHEMBL3526795 0.089 0.075 CHEMBL3526627 0.102 0.051 CHEMBL3526722 | CHEMBL3526722 | |
| 0.039 | 0.03 | 0.04 | Integrin alpha5beta1 antagonist | 0.04 0.029 CHEMBL3526971 0.038 0.033 CHEMBL3526633 0.037 0.035 CHEMBL3526627 0.037 0.034 CHEMBL3526722 | CHEMBL3526971 | |
| 0.015 | 0.009 | 0.016 | Integrin beta6 antagonist | 0.016 0.006 CHEMBL3526971 0.015 0.008 CHEMBL3526633 0.014 0.01 CHEMBL3526627 0.016 0.007 CHEMBL3526722 | CHEMBL3526722 | |
| 0.017 | 0.017 | 0.019 | Integrin alphaVbeta1 antagonist | 0.019 0.014 CHEMBL3526971 0.018 0.015 CHEMBL3526722 | CHEMBL3526971 | |
| 0.026 | 0.041 | 0.035 | Integrin antagonist | 0.035 0.034 CHEMBL4525745 | CHEMBL4525745 | |
| 0.032 | 0.051 | 0.042 | Acetyl-CoA carboxylase inhibitor | 0.042 0.028 CHEMBL4525745 | CHEMBL4525745 | |
| 0.07 | 0.094 | 0.089 | 5-Lipoxygenase inhibitor | 0.089 0.073 CHEMBL3526971 0.089 0.072 CHEMBL3526633 | CHEMBL3526633 | |
| 0.065 | 0.09 | 0.089 | MAO B inhibitor | 0.089 0.067 CHEMBL3526971 0.081 0.074 CHEMBL3526633 0.08 0.076 CHEMBL3526722 | CHEMBL3526971 | |
| 0.084 | 0.11 | 0.108 | MAO inhibitor | 0.108 0.083 CHEMBL3526971 0.102 0.089 CHEMBL3526633 0.099 0.092 CHEMBL3526722 | CHEMBL3526971 | |
| 0.169 | 0.202 | 0.228 | Tyrosine 3 hydroxylase inhibitor | 0.218 0.106 CHEMBL3526971 0.228 0.093 CHEMBL4525745 0.198 0.14 CHEMBL3526633 | CHEMBL4525745 | |
| 0.134 | 0.169 | 0.39 | Free radical scavenger | 0.178 0.117 CHEMBL3526971 0.156 0.138 CHEMBL4525745 0.193 0.103 CHEMBL3526633 0.39 0.031 CHEMBL3526795 0.151 0.144 CHEMBL3526627 0.197 0.1 CHEMBL3526722 0.189 0.107 CHEMBL3526723 | CHEMBL3526795 | |
| 0.214 | 0.251 | 0.393 | Calcium channel L-type activator | 0.266 0.188 CHEMBL3526971 0.355 0.113 CHEMBL3526634 0.235 0.222 CHEMBL4525745 0.257 0.197 CHEMBL3526633 0.292 0.164 CHEMBL3526627 0.342 0.123 CHEMBL3526722 0.393 0.086 CHEMBL3526723 | CHEMBL3526723 | |
| 0.006 | 0.052 | 0.019 | Ileal bile acid transport inhibitor | 0.019 0.01 CHEMBL4525745 | CHEMBL4525745 | |
| 0.099 | 0.148 | 0.179 | Phospholipase A2 inhibitor | 0.12 0.118 CHEMBL3526971 0.179 0.055 CHEMBL4525745 | CHEMBL4525745 | |
| 0.013 | 0.064 | 0.032 | Prostacyclin antagonist | 0.032 0.024 CHEMBL3526627 0.029 0.027 CHEMBL3526722 | CHEMBL3526627 | |
| 0.026 | 0.082 | 0.147 | Aldose reductase inhibitor | 0.124 0.014 CHEMBL3526634 0.147 0.011 CHEMBL3526723 | CHEMBL3526723 | |
| 0.04 | 0.099 | 0.054 | DNA helicase inhibitor | 0.054 0.038 CHEMBL4525745 | CHEMBL4525745 | |
| 0.098 | 0.157 | 0.189 | Vanilloid 1 agonist | 0.189 0.015 CHEMBL4525745 | CHEMBL4525745 | |
| 0.007 | 0.072 | 0.029 | Thyroid hormone alpha antagonist | 0.02 0.007 CHEMBL3526627 0.029 0.005 CHEMBL3526722 | CHEMBL3526722 | |
| 0.015 | 0.088 | 0.043 | Vitamin D receptor antagonist | 0.04 0.005 CHEMBL3526627 0.043 0.005 CHEMBL3526722 | CHEMBL3526722 | |
| 0.056 | 0.133 | 0.084 | Protease inhibitor | 0.084 0.081 CHEMBL4525745 | CHEMBL4525745 | |
| 0.026 | 0.105 | 0.044 | Microtubule stabilization | 0.044 0.035 CHEMBL3526795 | CHEMBL3526795 | |
| 0.004 | 0.083 | 0.021 | Integrin alpha4beta1 antagonist | 0.021 0.009 CHEMBL4525745 | CHEMBL4525745 | |
| 0.115 | 0.195 | 0.361 | Antiamyloidogenic | 0.361 0.036 CHEMBL4525745 0.154 0.142 CHEMBL3526633 0.319 0.046 CHEMBL3526795 | CHEMBL4525745 | |
| 0.063 | 0.152 | 0.099 | Vanilloid agonist | 0.099 0.035 CHEMBL4525745 | CHEMBL4525745 | |
| 0.073 | 0.162 | 0.186 | Cyclooxygenase 3 inhibitor | 0.174 0.031 CHEMBL4525745 0.186 0.025 CHEMBL3526795 | CHEMBL3526795 | |
| 0.012 | 0.11 | 0.025 | Calcium-sensing receptor agonist | 0.025 0.022 CHEMBL4525745 | CHEMBL4525745 | |
| 0.094 | 0.193 | 0.118 | Papain-like protease (SARS coronavirus) inhibitor | 0.118 0.086 CHEMBL4525745 | CHEMBL4525745 | |
| 0.052 | 0.152 | 0.166 | Sphingomyelinase inhibitor | 0.166 0.018 CHEMBL4525745 | CHEMBL4525745 | |
| 0.162 | 0.266 | 0.377 | Interleukin 2 agonist | 0.201 0.188 CHEMBL3526971 0.197 0.194 CHEMBL3526634 0.202 0.186 CHEMBL4525745 0.377 0.035 CHEMBL3526795 0.201 0.188 CHEMBL3526627 0.237 0.134 CHEMBL3526722 0.233 0.139 CHEMBL3526723 | CHEMBL3526795 | |
| 0.079 | 0.186 | 0.406 | Angiogenesis stimulant | 0.183 0.104 CHEMBL4525745 0.406 0.021 CHEMBL3526795 0.137 0.131 CHEMBL3526722 | CHEMBL3526795 | |
| 0.073 | 0.188 | 0.097 | Factor V inhibitor | 0.097 0.077 CHEMBL4525745 | CHEMBL4525745 | |
| 0.09 | 0.206 | 0.26 | Nitric oxide antagonist | 0.26 0.049 CHEMBL3526795 | CHEMBL3526795 | |
| 0.067 | 0.192 | 0.13 | Electron transport complex I inhibitor | 0.13 0.035 CHEMBL3526634 0.113 0.058 CHEMBL3526723 | CHEMBL3526634 | |
| 0.038 | 0.167 | 0.059 | Caspase 9 inhibitor | 0.059 0.049 CHEMBL4525745 | CHEMBL4525745 | |
| 0.069 | 0.199 | 0.116 | Cell adhesion inhibitor | 0.097 0.096 CHEMBL4525745 0.116 0.068 CHEMBL3526795 | CHEMBL3526795 | |
| 0.025 | 0.171 | 0.07 | Catalase inhibitor | 0.07 0.055 CHEMBL4525745 | CHEMBL4525745 | |
| 0.058 | 0.205 | 0.098 | Microtubule formation inhibitor | 0.098 0.094 CHEMBL4525745 0.098 0.095 CHEMBL3526795 | CHEMBL3526795 | |
| 0.09 | 0.243 | 0.173 | Platelet antagonist | 0.153 0.142 CHEMBL4525745 0.173 0.123 CHEMBL3526795 | CHEMBL3526795 | |
| 0.052 | 0.211 | 0.095 | Transcription factor NF kappa B stimulant | 0.095 0.044 CHEMBL3526795 | CHEMBL3526795 | |
| 0.018 | 0.181 | 0.049 | Antibiotic Aminoglycoside-like | 0.049 0.014 CHEMBL3526795 | CHEMBL3526795 | |
| 0.079 | 0.247 | 0.123 | Growth hormone agonist | 0.123 0.116 CHEMBL4525745 | CHEMBL4525745 | |
| 0.063 | 0.232 | 0.113 | Folate antagonist | 0.113 0.046 CHEMBL4525745 | CHEMBL4525745 | |
| 0.018 | 0.192 | 0.06 | Protein 50S ribosomal subunit inhibitor | 0.06 0.031 CHEMBL3526795 | CHEMBL3526795 | |
| 0.017 | 0.197 | 0.046 | Lysophosphatidic acid 3 receptor antagonist | 0.046 0.043 CHEMBL4525745 | CHEMBL4525745 | |
| 0.019 | 0.201 | 0.052 | Alpha-mannosidase inhibitor | 0.052 0.04 CHEMBL4525745 | CHEMBL4525745 | |
| 0.1 | 0.284 | 0.13 | CC chemokine 6 receptor antagonist | 0.13 0.071 CHEMBL3526795 | CHEMBL3526795 | |
| 0.054 | 0.243 | 0.086 | Estrogen-related receptor beta agonist | 0.086 0.048 CHEMBL4525745 | CHEMBL4525745 | |
| 0.032 | 0.228 | 0.06 | Adenine nucleotide translocase inhibitor | 0.06 0.028 CHEMBL3526795 | CHEMBL3526795 | |
| 0.046 | 0.248 | 0.179 | Lipid peroxidase inhibitor | 0.179 0.051 CHEMBL3526795 | CHEMBL3526795 | |
| 0.064 | 0.271 | 0.135 | Amyloid beta precursor protein antagonist | 0.135 0.119 CHEMBL4525745 | CHEMBL4525745 | |
| 0.008 | 0.229 | 0.024 | Protein 30S ribosomal subunit inhibitor | 0.024 0.017 CHEMBL3526795 | CHEMBL3526795 | |
| 0.025 | 0.247 | 0.078 | Metalloproteinase-2 inhibitor | 0.078 0.054 CHEMBL4525745 | CHEMBL4525745 | |
| 0.015 | 0.247 | 0.051 | Matrix metalloproteinase (membrane-type) inhibitor | 0.051 0.045 CHEMBL4525745 | CHEMBL4525745 | |
| 0.067 | 0.299 | 0.251 | Platelet adhesion inhibitor | 0.251 0.049 CHEMBL3526795 | CHEMBL3526795 | |
| 0.049 | 0.288 | 0.123 | Estrogen antagonist | 0.101 0.097 CHEMBL3526971 0.123 0.049 CHEMBL3526722 | CHEMBL3526722 | |
| 0.016 | 0.261 | 0.067 | Matrix metalloproteinase inhibitor | 0.067 0.046 CHEMBL4525745 | CHEMBL4525745 | |
| 0.022 | 0.282 | 0.074 | Metalloproteinase-9 inhibitor | 0.074 0.049 CHEMBL4525745 | CHEMBL4525745 | |
| 0.02 | 0.282 | 0.051 | Glucose-6-phosphate translocase inhibitor | 0.051 0.037 CHEMBL3526795 | CHEMBL3526795 | |
| 0.01 | 0.279 | 0.084 | Antineoplastic antibiotic | 0.084 0.055 CHEMBL3526795 | CHEMBL3526795 | |
| 0.035 | 0.312 | 0.144 | Thrombolytic | 0.119 0.112 CHEMBL4525745 0.144 0.087 CHEMBL3526795 | CHEMBL3526795 | |
| 0.061 | 0.338 | 0.227 | Hepatoprotectant | 0.227 0.051 CHEMBL3526795 | CHEMBL3526795 | |
| 0.029 | 0.307 | 0.131 | Bronchodilator | 0.131 0.039 CHEMBL3526634 0.123 0.043 CHEMBL3526723 | CHEMBL3526634 | |
| 0.046 | 0.327 | 0.094 | Glutamate (mGluR7) agonist | 0.094 0.074 CHEMBL4525745 | CHEMBL4525745 | |
| 0.035 | 0.323 | 0.131 | Caspase 3 inhibitor | 0.131 0.045 CHEMBL4525745 | CHEMBL4525745 | |
| 0.012 | 0.305 | 0.192 | Selectin antagonist | 0.192 0.012 CHEMBL3526795 | CHEMBL3526795 | |
| 0.031 | 0.327 | 0.126 | Interleukin 1 beta converting enzyme inhibitor | 0.126 0.031 CHEMBL4525745 | CHEMBL4525745 | |
| 0.033 | 0.335 | 0.107 | Estrogen receptor beta antagonist | 0.107 0.052 CHEMBL3526722 | CHEMBL3526722 | |
| 0.021 | 0.336 | 0.153 | Topoisomerase I inhibitor | 0.153 0.04 CHEMBL3526795 | CHEMBL3526795 | |
| 0.038 | 0.364 | 0.129 | Anticoagulant | 0.129 0.101 CHEMBL4525745 | CHEMBL4525745 | |
| 0.008 | 0.346 | 0.066 | Glycine transporter 2 inhibitor | 0.066 0.022 CHEMBL4525745 | CHEMBL4525745 | |
| 0.053 | 0.397 | 0.251 | Tumour necrosis factor alpha release inhibitor | 0.251 0.075 CHEMBL3526795 | CHEMBL3526795 | |
| 0.022 | 0.366 | 0.111 | Alkylator | 0.111 0.077 CHEMBL4525745 0.104 0.084 CHEMBL3526795 | CHEMBL4525745 | |
| 0.009 | 0.393 | 0.038 | Ceramide glucosyltransferase inhibitor | 0.038 0.019 CHEMBL4525745 | CHEMBL4525745 | |
| 0.033 | 0.423 | 0.104 | Toll-Like receptor 4 antagonist | 0.104 0.063 CHEMBL3526795 | CHEMBL3526795 | |
| 0.062 | 0.466 | 0.239 | Antithrombotic | 0.239 0.135 CHEMBL3526795 | CHEMBL3526795 | |
| 0.015 | 0.45 | 0.079 | Topoisomerase II alpha inhibitor | 0.079 0.054 CHEMBL3526795 | CHEMBL3526795 | |
| 0.049 | 0.501 | 0.338 | Immunosuppressant | 0.338 0.093 CHEMBL3526795 | CHEMBL3526795 | |
| 0.023 | 0.513 | 0.296 | Immunostimulant | 0.174 0.136 CHEMBL4525745 0.296 0.079 CHEMBL3526795 | CHEMBL3526795 | |
| 0.034 | 0.557 | 0.181 | Interleukin agonist | 0.181 0.139 CHEMBL4525745 | CHEMBL4525745 | |
| 0.06 | 0.6 | 0.391 | Apoptosis agonist | 0.391 0.118 CHEMBL3526795 | CHEMBL3526795 | |
| 0.05 | 0.593 | 0.146 | Neurotensin receptor agonist | 0.146 0.113 CHEMBL4525745 | CHEMBL4525745 | |
| 0.017 | 0.673 | 0.258 | Transcription factor NF kappa B inhibitor | 0.258 0.122 CHEMBL3526795 | CHEMBL3526795 | |
| 0.031 | 0.76 | 0.406 | Antiinflammatory | 0.406 0.136 CHEMBL3526795 | CHEMBL3526795 | |
| 0.008 | 0.833 | 0.332 | Antibacterial | 0.332 0.113 CHEMBL3526795 | CHEMBL3526795 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |