| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.995 | 0 | 0.995 | Dihydrofolate reductase inhibitor | 0.762 0.001 CHEMBL3544676 0.975 0.001 CHEMBL3544661 | ||
| 0.862 | 0.001 | 0.862 | Folate antagonist | 0.841 0.001 CHEMBL3544676 0.724 0.001 CHEMBL3544661 | ||
| 0.645 | 0.002 | 0.645 | Antimetabolite | 0.257 0.007 CHEMBL3544676 0.48 0.003 CHEMBL3544661 | ||
| 0.628 | 0 | 0.628 | AICAR transformylase inhibitor | 0.256 0.001 CHEMBL3544676 0.444 0 CHEMBL3544661 | ||
| 0.57 | 0.009 | 0.593 | DNA synthesis inhibitor | 0.593 0.008 CHEMBL3544676 0.502 0.013 CHEMBL3544661 | CHEMBL3544676 | |
| 0.571 | 0.014 | 0.635 | Immunomodulator | 0.51 0.022 CHEMBL3544676 0.635 0.009 CHEMBL3544661 | CHEMBL3544661 | |
| 0.55 | 0.001 | 0.55 | Thymidylate synthase inhibitor | 0.216 0.002 CHEMBL3544676 0.504 0.001 CHEMBL3544661 | ||
| 0.4 | 0.049 | 0.4 | Immunostimulant | 0.193 0.125 CHEMBL3544676 0.377 0.057 CHEMBL3544661 | ||
| 0.392 | 0.064 | 0.392 | Toll-Like receptor agonist | 0.367 0.074 CHEMBL3544676 0.241 0.157 CHEMBL3544661 | ||
| 0.363 | 0.076 | 0.363 | Toll-Like receptor 7 agonist | 0.346 0.084 CHEMBL3544676 0.214 0.184 CHEMBL3544661 | ||
| 0.275 | 0.036 | 0.275 | DNA methylase inhibitor | 0.242 0.053 CHEMBL3544676 0.272 0.038 CHEMBL3544661 | ||
| 0.211 | 0.002 | 0.228 | Dihydropteroate synthase inhibitor | 0.228 0.002 CHEMBL3544676 0.162 0.003 CHEMBL3544661 | CHEMBL3544676 | |
| 0.287 | 0.083 | 0.291 | Interleukin 2 agonist | 0.291 0.08 CHEMBL3544661 | CHEMBL3544661 | |
| 0.198 | 0.023 | 0.295 | Interleukin 4 antagonist | 0.295 0.009 CHEMBL3544676 0.195 0.024 CHEMBL3544661 | CHEMBL3544676 | |
| 0.248 | 0.08 | 0.248 | Interleukin agonist | 0.231 0.093 CHEMBL3544661 | ||
| 0.209 | 0.048 | 0.209 | Thrombolytic | 0.207 0.049 CHEMBL3544661 | ||
| 0.193 | 0.037 | 0.193 | Catenin beta inhibitor | 0.186 0.045 CHEMBL3544661 | ||
| 0.179 | 0.033 | 0.179 | Alkylator | 0.124 0.065 CHEMBL3544676 0.095 0.094 CHEMBL3544661 | ||
| 0.225 | 0.082 | 0.225 | Angiogenesis stimulant | 0.201 0.094 CHEMBL3544661 | ||
| 0.185 | 0.051 | 0.185 | Diuretic | 0.152 0.076 CHEMBL3544676 0.127 0.097 CHEMBL3544661 | ||
| 0.146 | 0.017 | 0.148 | Glutamate dehydrogenase inhibitor | 0.135 0.019 CHEMBL3544676 0.148 0.016 CHEMBL3544661 | CHEMBL3544661 | |
| 0.153 | 0.029 | 0.173 | DNA repair enzyme inhibitor | 0.173 0.016 CHEMBL3544676 0.11 0.096 CHEMBL3544661 | CHEMBL3544676 | |
| 0.134 | 0.016 | 0.182 | Purinergic P2X2 antagonist | 0.182 0.006 CHEMBL3544676 0.1 0.03 CHEMBL3544661 | CHEMBL3544676 | |
| 0.152 | 0.048 | 0.195 | DNA polymerase I inhibitor | 0.195 0.03 CHEMBL3544676 0.128 0.062 CHEMBL3544661 | CHEMBL3544676 | |
| 0.201 | 0.1 | 0.201 | Platelet antagonist | 0.2 0.1 CHEMBL3544661 | ||
| 0.115 | 0.019 | 0.153 | Interferon agonist | 0.112 0.021 CHEMBL3544676 0.153 0.01 CHEMBL3544661 | CHEMBL3544661 | |
| 0.169 | 0.074 | 0.169 | Growth hormone agonist | 0.149 0.088 CHEMBL3544661 | ||
| 0.141 | 0.052 | 0.141 | Cell adhesion inhibitor | 0.109 0.075 CHEMBL3544661 | ||
| 0.107 | 0.029 | 0.107 | Hematopoietic | 0.091 0.047 CHEMBL3544661 | ||
| 0.154 | 0.077 | 0.154 | Anticoagulant | 0.143 0.087 CHEMBL3544661 | ||
| 0.165 | 0.09 | 0.184 | DNA methyltransferase I inhibitor | 0.145 0.109 CHEMBL3544676 0.184 0.077 CHEMBL3544661 | CHEMBL3544661 | |
| 0.106 | 0.039 | 0.106 | Aminoacyl-tRNA synthetase inhibitor | 0.101 0.044 CHEMBL3544676 0.098 0.047 CHEMBL3544661 | ||
| 0.109 | 0.047 | 0.109 | Nitric-oxide synthase inhibitor | 0.101 0.058 CHEMBL3544676 | ||
| 0.107 | 0.049 | 0.107 | Interleukin 1 beta converting enzyme inhibitor | 0.093 0.067 CHEMBL3544661 | ||
| 0.11 | 0.062 | 0.11 | Nav1.4 sodium channel blocker | 0.095 0.085 CHEMBL3544661 | ||
| 0.074 | 0.029 | 0.092 | Interferon inducer | 0.079 0.025 CHEMBL3544676 0.092 0.016 CHEMBL3544661 | CHEMBL3544661 | |
| 0.064 | 0.02 | 0.064 | Complement C3a chemotactic receptor antagonist | 0.061 0.021 CHEMBL3544661 | ||
| 0.156 | 0.114 | 0.156 | Interleukin antagonist | 0.14 0.125 CHEMBL3544661 | ||
| 0.091 | 0.053 | 0.127 | Interleukin 5 antagonist | 0.127 0.019 CHEMBL3544676 0.081 0.072 CHEMBL3544661 | CHEMBL3544676 | |
| 0.058 | 0.021 | 0.058 | Farnesyltransferase inhibitor | |||
| 0.067 | 0.032 | 0.067 | Ribonucleotide reductase inhibitor | |||
| 0.056 | 0.025 | 0.086 | Adenosine deaminase inhibitor | 0.086 0.008 CHEMBL3544676 | CHEMBL3544676 | |
| 0.061 | 0.033 | 0.061 | Ribonucleoside-diphosphate reductase inhibitor | |||
| 0.061 | 0.036 | 0.077 | Argininosuccinate synthase inhibitor | 0.077 0.027 CHEMBL3544676 0.06 0.037 CHEMBL3544661 | CHEMBL3544676 | |
| 0.142 | 0.117 | 0.204 | Lipocortins synthesis antagonist | 0.204 0.054 CHEMBL3544676 0.141 0.119 CHEMBL3544661 | CHEMBL3544676 | |
| 0.202 | 0.177 | 0.202 | Apoptosis antagonist | |||
| 0.026 | 0.002 | 0.029 | Phosphoribosylglycinamide formyltransferase inhibitor | 0.008 0.004 CHEMBL3544676 0.029 0.002 CHEMBL3544661 | CHEMBL3544661 | |
| 0.069 | 0.047 | 0.155 | Phenylalanine 4-hydroxylase inhibitor | 0.155 0.011 CHEMBL3544676 0.086 0.033 CHEMBL3544661 | CHEMBL3544676 | |
| 0.062 | 0.041 | 0.069 | Carbamoyl phosphate synthetase inhibitor | 0.069 0.035 CHEMBL3544661 | CHEMBL3544661 | |
| 0.169 | 0.149 | 0.169 | Peptidyltransferase inhibitor | 0.169 0.148 CHEMBL3544661 | ||
| 0.058 | 0.043 | 0.058 | CXC chemokine 4 receptor antagonist | 0.055 0.046 CHEMBL3544676 | ||
| 0.02 | 0.006 | 0.024 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.024 0.004 CHEMBL3544676 0.018 0.01 CHEMBL3544661 | CHEMBL3544676 | |
| 0.095 | 0.081 | 0.095 | Factor V inhibitor | 0.095 0.082 CHEMBL3544661 | ||
| 0.02 | 0.007 | 0.02 | Tryptophan hydroxylase 1 inhibitor | 0.019 0.008 CHEMBL3544661 | ||
| 0.031 | 0.021 | 0.031 | Endothelial nitric-oxide synthase inhibitor | |||
| 0.022 | 0.014 | 0.022 | Geranylgeranyltransferase I inhibitor | |||
| 0.058 | 0.051 | 0.058 | Caspase 9 inhibitor | |||
| 0.078 | 0.071 | 0.081 | Factor XII inhibitor | 0.081 0.064 CHEMBL3544661 | CHEMBL3544661 | |
| 0.041 | 0.035 | 0.074 | Guanylate cyclase stimulant | 0.074 0.01 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.01 | 0.015 | N-Acetylated alpha-linked acidic dipeptidase inhibitor | 0.013 0.012 CHEMBL3544661 | ||
| 0.034 | 0.03 | 0.034 | Tryptophan 5 hydroxylase inhibitor | |||
| 0.185 | 0.182 | 0.185 | Insulysin inhibitor | |||
| 0.055 | 0.052 | 0.055 | Glucagon-like peptide 1 agonist | |||
| 0.036 | 0.034 | 0.036 | Integrin alpha1beta1 antagonist | |||
| 0.03 | 0.031 | 0.038 | RNA-directed RNA polymerase inhibitor | 0.038 0.02 CHEMBL3544676 | CHEMBL3544676 | |
| 0.011 | 0.019 | 0.014 | S-adenosyl-L-homocysteine hydrolase inhibitor | 0.014 0.012 CHEMBL3544676 | CHEMBL3544676 | |
| 0.06 | 0.068 | 0.084 | CXC chemokine receptor antagonist | 0.084 0.034 CHEMBL3544676 | CHEMBL3544676 | |
| 0.011 | 0.019 | 0.014 | Adenosine A2b receptor agonist | 0.014 0.012 CHEMBL3544676 | CHEMBL3544676 | |
| 0.115 | 0.125 | 0.134 | Hemostatic | 0.134 0.09 CHEMBL3544661 | CHEMBL3544661 | |
| 0.081 | 0.094 | 0.238 | Electrolyte absorption antagonist | 0.238 0.005 CHEMBL3544676 | CHEMBL3544676 | |
| 0.192 | 0.211 | 0.386 | Histamine release inhibitor | 0.386 0.083 CHEMBL3544676 | CHEMBL3544676 | |
| 0.036 | 0.057 | 0.06 | Ornithine carbamoyltransferase inhibitor | 0.06 0.031 CHEMBL3544676 | CHEMBL3544676 | |
| 0.095 | 0.125 | 0.113 | Transcription factor STAT6 inhibitor | 0.113 0.074 CHEMBL3544676 | CHEMBL3544676 | |
| 0.012 | 0.044 | 0.018 | Guanylate cyclase 1 stimulant | 0.018 0.015 CHEMBL3544676 | CHEMBL3544676 | |
| 0.078 | 0.125 | 0.136 | Adenylate kinase inhibitor | 0.136 0.032 CHEMBL3544676 | CHEMBL3544676 | |
| 0.037 | 0.088 | 0.049 | Antiviral (Hepatitis D) | 0.049 0.038 CHEMBL3544676 | CHEMBL3544676 | |
| 0.038 | 0.09 | 0.055 | Cyclin H inhibitor | 0.055 0.046 CHEMBL3544676 | CHEMBL3544676 | |
| 0.03 | 0.092 | 0.06 | Tyrosine-protein kinase EMT inhibitor | 0.06 0.038 CHEMBL3544676 | CHEMBL3544676 | |
| 0.036 | 0.098 | 0.06 | Phosphofructokinase-1 inhibitor | 0.06 0.056 CHEMBL3544676 | CHEMBL3544676 | |
| 0.032 | 0.096 | 0.073 | CDK1/cyclin B inhibitor | 0.073 0.037 CHEMBL3544676 | CHEMBL3544676 | |
| 0.032 | 0.1 | 0.061 | Cyclin B inhibitor | 0.061 0.031 CHEMBL3544676 | CHEMBL3544676 | |
| 0.052 | 0.121 | 0.069 | Phosphodiesterase VIII inhibitor | 0.069 0.056 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.086 | 0.054 | Phosphoglycerate kinase inhibitor | 0.054 0.013 CHEMBL3544676 | CHEMBL3544676 | |
| 0.045 | 0.118 | 0.074 | I kappa B kinase 1 inhibitor | 0.074 0.042 CHEMBL3544676 | CHEMBL3544676 | |
| 0.112 | 0.186 | 0.158 | MAP kinase kinase 4 inhibitor | 0.158 0.048 CHEMBL3544676 | CHEMBL3544676 | |
| 0.066 | 0.142 | 0.081 | Transforming growth factor beta 3 antagonist | 0.081 0.061 CHEMBL3544676 | CHEMBL3544676 | |
| 0.167 | 0.246 | 0.186 | MAP kinase kinase 3 inhibitor | 0.186 0.168 CHEMBL3544676 | CHEMBL3544676 | |
| 0.026 | 0.109 | 0.061 | Cyclin B2 inhibitor | 0.061 0.031 CHEMBL3544676 | CHEMBL3544676 | |
| 0.032 | 0.116 | 0.069 | Cyclin B1 inhibitor | 0.069 0.033 CHEMBL3544676 | CHEMBL3544676 | |
| 0.059 | 0.145 | 0.092 | MAP kinase kinase 7 inhibitor | 0.092 0.021 CHEMBL3544676 | CHEMBL3544676 | |
| 0.056 | 0.158 | 0.127 | GABA C receptor agonist | 0.127 0.045 CHEMBL3544676 | CHEMBL3544676 | |
| 0.073 | 0.179 | 0.169 | CDC-like kinase 1 inhibitor | 0.169 0.055 CHEMBL3544676 | CHEMBL3544676 | |
| 0.123 | 0.236 | 0.229 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.229 0.053 CHEMBL3544676 | CHEMBL3544676 | |
| 0.042 | 0.168 | 0.073 | AXL receptor tyrosine kinase inhibitor | 0.073 0.072 CHEMBL3544676 | CHEMBL3544676 | |
| 0.054 | 0.182 | 0.128 | Phosphodiesterase 7B inhibitor | 0.128 0.032 CHEMBL3544676 | CHEMBL3544676 | |
| 0.095 | 0.225 | 0.135 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.135 0.13 CHEMBL3544676 | CHEMBL3544676 | |
| 0.062 | 0.192 | 0.091 | mTOR complex 1 inhibitor | 0.091 0.083 CHEMBL3544676 | CHEMBL3544676 | |
| 0.071 | 0.205 | 0.208 | CDC-like kinase 4 inhibitor | 0.208 0.064 CHEMBL3544676 | CHEMBL3544676 | |
| 0.04 | 0.174 | 0.089 | Adenosine A3 receptor antagonist | 0.089 0.033 CHEMBL3544676 | CHEMBL3544676 | |
| 0.074 | 0.209 | 0.227 | Clk dual-specificity kinase inhibitor | 0.227 0.065 CHEMBL3544676 | CHEMBL3544676 | |
| 0.017 | 0.16 | 0.038 | Glutamate (mGluR1a) antagonist | 0.038 0.032 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.166 | 0.094 | Adenosine A2a receptor antagonist | 0.094 0.026 CHEMBL3544676 | CHEMBL3544676 | |
| 0.06 | 0.211 | 0.102 | Glutamate release inhibitor | 0.102 0.039 CHEMBL3544676 | CHEMBL3544676 | |
| 0.037 | 0.188 | 0.08 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.08 0.037 CHEMBL3544676 | CHEMBL3544676 | |
| 0.032 | 0.184 | 0.089 | Cyclin-dependent kinase 1 inhibitor | 0.089 0.074 CHEMBL3544676 | CHEMBL3544676 | |
| 0.039 | 0.191 | 0.102 | Alcohol dehydrogenase inhibitor | 0.102 0.05 CHEMBL3544676 | CHEMBL3544676 | |
| 0.091 | 0.244 | 0.177 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.177 0.035 CHEMBL3544676 | CHEMBL3544676 | |
| 0.038 | 0.192 | 0.193 | Protein kinase (CK2) alpha inhibitor | 0.193 0.026 CHEMBL3544676 | CHEMBL3544676 | |
| 0.05 | 0.206 | 0.138 | Xanthine oxidase inhibitor | 0.138 0.039 CHEMBL3544676 | CHEMBL3544676 | |
| 0.036 | 0.192 | 0.143 | Histamine N-methyltransferase inhibitor | 0.143 0.017 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.173 | 0.08 | Adenosine A1 receptor antagonist | 0.08 0.028 CHEMBL3544676 | CHEMBL3544676 | |
| 0.125 | 0.291 | 0.201 | Vasodilator, coronary | 0.201 0.181 CHEMBL3544676 | CHEMBL3544676 | |
| 0.055 | 0.222 | 0.18 | CDC-like kinase 2 inhibitor | 0.18 0.077 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.2 | 0.082 | Adenosine A2 receptor antagonist | 0.082 0.034 CHEMBL3544676 | CHEMBL3544676 | |
| 0.114 | 0.311 | 0.281 | RNA-directed DNA polymerase inhibitor | 0.281 0.036 CHEMBL3544676 | CHEMBL3544676 | |
| 0.038 | 0.237 | 0.093 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.093 0.045 CHEMBL3544676 | CHEMBL3544676 | |
| 0.011 | 0.218 | 0.05 | Adenosine A2b receptor antagonist | 0.05 0.033 CHEMBL3544676 | CHEMBL3544676 | |
| 0.069 | 0.277 | 0.17 | Sigma receptor agonist | 0.17 0.073 CHEMBL3544676 | CHEMBL3544676 | |
| 0.059 | 0.27 | 0.235 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.235 0.074 CHEMBL3544676 | CHEMBL3544676 | |
| 0.004 | 0.216 | 0.019 | Adenosine kinase inhibitor | 0.019 0.017 CHEMBL3544676 | CHEMBL3544676 | |
| 0.017 | 0.246 | 0.057 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.057 0.038 CHEMBL3544676 | CHEMBL3544676 | |
| 0.055 | 0.292 | 0.225 | Dyrk kinase inhibitor | 0.225 0.084 CHEMBL3544676 | CHEMBL3544676 | |
| 0.015 | 0.253 | 0.087 | Biliverdin reductase inhibitor | 0.087 0.023 CHEMBL3544676 | CHEMBL3544676 | |
| 0.114 | 0.367 | 0.28 | Antibacterial | 0.28 0.151 CHEMBL3544676 | CHEMBL3544676 | |
| 0.062 | 0.316 | 0.147 | Death-associated protein kinase 3 inhibitor | 0.147 0.127 CHEMBL3544676 | CHEMBL3544676 | |
| 0.041 | 0.299 | 0.085 | mTOR complex 2 inhibitor | 0.085 0.057 CHEMBL3544676 | CHEMBL3544676 | |
| 0.094 | 0.353 | 0.209 | Cholesterol antagonist | 0.209 0.157 CHEMBL3544676 | CHEMBL3544676 | |
| 0.02 | 0.28 | 0.157 | Protein kinase (CK2) inhibitor | 0.157 0.03 CHEMBL3544676 | CHEMBL3544676 | |
| 0.101 | 0.368 | 0.129 | Heat shock protein 70 antagonist | 0.129 0.128 CHEMBL3544676 | CHEMBL3544676 | |
| 0.01 | 0.311 | 0.059 | Acyl-CoA dehydrogenase inhibitor | 0.059 0.034 CHEMBL3544676 | CHEMBL3544676 | |
| 0.038 | 0.344 | 0.158 | LIM domain kinase 1 inhibitor | 0.158 0.09 CHEMBL3544676 | CHEMBL3544676 | |
| 0.076 | 0.396 | 0.149 | Histone acetyltransferase inhibitor | 0.149 0.141 CHEMBL3544676 | CHEMBL3544676 | |
| 0.034 | 0.373 | 0.108 | NADH dehydrogenase inhibitor | 0.108 0.036 CHEMBL3544676 | CHEMBL3544676 | |
| 0.041 | 0.383 | 0.165 | Heat shock protein 90 antagonist | 0.165 0.06 CHEMBL3544676 | CHEMBL3544676 | |
| 0.008 | 0.37 | 0.073 | Xanthine dehydrogenase inhibitor | 0.073 0.029 CHEMBL3544676 | CHEMBL3544676 | |
| 0.038 | 0.406 | 0.193 | Heat shock protein 90 alpha antagonist | 0.193 0.053 CHEMBL3544676 | CHEMBL3544676 | |
| 0.027 | 0.435 | 0.081 | Phosphodiesterase I inhibitor | 0.081 0.076 CHEMBL3544676 | CHEMBL3544676 | |
| 0.021 | 0.437 | 0.098 | Ferrochelatase inhibitor | 0.098 0.073 CHEMBL3544676 | CHEMBL3544676 | |
| 0.082 | 0.575 | 0.27 | 5 Hydroxytryptamine release inhibitor | 0.27 0.201 CHEMBL3544676 | CHEMBL3544676 | |
| 0.02 | 0.515 | 0.225 | I kappa B kinase epsilon inhibitor | 0.225 0.052 CHEMBL3544676 | CHEMBL3544676 | |
| 0.04 | 0.562 | 0.221 | Hypoxia-inducible factor 1 alpha inhibitor | 0.221 0.128 CHEMBL3544676 | CHEMBL3544676 | |
| 0.104 | 0.648 | 0.283 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.283 0.236 CHEMBL3544676 | CHEMBL3544676 | |
| 0.028 | 0.661 | 0.126 | Hexokinase inhibitor | 0.126 0.109 CHEMBL3544676 | CHEMBL3544676 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |