| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.669 | 0.017 | 0.91 | Cyclophilin D inhibitor | 0.624 0.023 CHEMBL3526179 0.749 0.01 CHEMBL3526440 0.669 0.017 CHEMBL3526439 0.726 0.012 CHEMBL3526292 0.631 0.022 CHEMBL3526178 0.91 0.005 CHEMBL4525762 | CHEMBL4525762 | |
| 0.584 | 0.003 | 0.584 | Insulin sensitizer | 0.464 0.004 CHEMBL3526179 0.436 0.005 CHEMBL3526440 0.584 0.003 CHEMBL3526439 0.439 0.005 CHEMBL3526292 0.396 0.007 CHEMBL3526178 0.308 0.014 CHEMBL4525762 | ||
| 0.541 | 0.014 | 0.73 | Lipoxygenase inhibitor | 0.274 0.085 CHEMBL3526179 0.541 0.014 CHEMBL3526439 0.73 0.005 CHEMBL3526178 | CHEMBL3526178 | |
| 0.464 | 0.019 | 0.628 | Hypoglycemic | 0.471 0.018 CHEMBL3526179 0.58 0.009 CHEMBL3526440 0.464 0.019 CHEMBL3526439 0.542 0.012 CHEMBL3526292 0.372 0.033 CHEMBL3526178 0.628 0.007 CHEMBL4525762 | CHEMBL4525762 | |
| 0.39 | 0.051 | 0.64 | Cholesterol antagonist | 0.64 0.014 CHEMBL3526179 0.622 0.016 CHEMBL3526440 0.39 0.051 CHEMBL3526439 0.579 0.021 CHEMBL3526292 0.287 0.099 CHEMBL3526178 0.561 0.024 CHEMBL4525762 | CHEMBL3526179 | |
| 0.313 | 0.004 | 0.313 | Leukotriene antagonist | 0.161 0.009 CHEMBL3526179 0.213 0.005 CHEMBL3526440 0.313 0.004 CHEMBL3526439 0.14 0.012 CHEMBL3526292 0.201 0.005 CHEMBL3526178 0.165 0.008 CHEMBL4525762 | ||
| 0.343 | 0.044 | 0.42 | Sodium/bile acid cotransporter inhibitor | 0.42 0.012 CHEMBL3526179 0.269 0.108 CHEMBL3526440 0.343 0.044 CHEMBL3526439 0.261 0.116 CHEMBL3526292 0.356 0.036 CHEMBL3526178 0.316 0.065 CHEMBL4525762 | CHEMBL3526179 | |
| 0.343 | 0.091 | 0.704 | Antiobesity | 0.3 0.116 CHEMBL3526179 0.308 0.111 CHEMBL3526440 0.343 0.091 CHEMBL3526439 0.287 0.126 CHEMBL3526292 0.266 0.142 CHEMBL3526178 0.704 0.01 CHEMBL4525762 | CHEMBL4525762 | |
| 0.29 | 0.052 | 0.339 | Hypolipemic | 0.237 0.074 CHEMBL3526179 0.321 0.043 CHEMBL3526440 0.29 0.052 CHEMBL3526439 0.339 0.038 CHEMBL3526292 0.238 0.073 CHEMBL3526178 0.295 0.05 CHEMBL4525762 | CHEMBL3526292 | |
| 0.234 | 0.004 | 0.234 | Peroxisome proliferator-activated receptor alpha agonist | 0.065 0.024 CHEMBL3526179 0.066 0.024 CHEMBL3526440 0.234 0.004 CHEMBL3526439 0.139 0.007 CHEMBL3526178 0.055 0.028 CHEMBL4525762 | ||
| 0.318 | 0.099 | 0.421 | Toll-Like receptor 7 agonist | 0.421 0.052 CHEMBL3526179 0.318 0.099 CHEMBL3526439 | CHEMBL3526179 | |
| 0.313 | 0.103 | 0.419 | Toll-Like receptor agonist | 0.419 0.053 CHEMBL3526179 0.313 0.103 CHEMBL3526439 | CHEMBL3526179 | |
| 0.214 | 0.004 | 0.221 | Protease activated receptor antagonist | 0.126 0.008 CHEMBL3526440 0.214 0.004 CHEMBL3526439 0.123 0.008 CHEMBL3526292 0.221 0.004 CHEMBL3526178 0.133 0.006 CHEMBL4525762 | CHEMBL3526178 | |
| 0.2 | 0.007 | 0.2 | Peroxisome proliferator-activated receptor gamma agonist | 0.166 0.01 CHEMBL3526179 0.125 0.019 CHEMBL3526440 0.2 0.007 CHEMBL3526439 0.109 0.024 CHEMBL3526292 0.169 0.009 CHEMBL3526178 0.128 0.018 CHEMBL4525762 | ||
| 0.255 | 0.07 | 0.317 | Platelet antagonist | 0.315 0.048 CHEMBL3526179 0.278 0.061 CHEMBL3526440 0.255 0.07 CHEMBL3526439 0.268 0.065 CHEMBL3526292 0.235 0.079 CHEMBL3526178 0.317 0.047 CHEMBL4525762 | CHEMBL4525762 | |
| 0.184 | 0.028 | 0.269 | 5-Lipoxygenase inhibitor | 0.1 0.064 CHEMBL3526179 0.184 0.028 CHEMBL3526439 0.269 0.013 CHEMBL3526178 | CHEMBL3526178 | |
| 0.217 | 0.062 | 0.356 | Platelet adhesion inhibitor | 0.356 0.018 CHEMBL3526440 0.217 0.062 CHEMBL3526439 0.343 0.021 CHEMBL3526292 0.215 0.063 CHEMBL3526178 0.356 0.018 CHEMBL4525762 | CHEMBL4525762 | |
| 0.151 | 0.009 | 0.169 | Prostaglandin E2 antagonist | 0.169 0.007 CHEMBL3526179 0.046 0.04 CHEMBL3526440 0.151 0.009 CHEMBL3526439 0.047 0.039 CHEMBL3526292 0.152 0.009 CHEMBL3526178 0.068 0.024 CHEMBL4525762 | CHEMBL3526179 | |
| 0.128 | 0.008 | 0.128 | Peroxisome proliferator-activated receptor gamma antagonist | 0.086 0.026 CHEMBL3526179 0.128 0.008 CHEMBL3526439 0.096 0.018 CHEMBL3526178 | ||
| 0.156 | 0.046 | 0.282 | Farnesoid X receptor antagonist | 0.282 0.008 CHEMBL3526179 0.156 0.046 CHEMBL3526439 0.123 0.098 CHEMBL3526292 0.157 0.045 CHEMBL3526178 0.121 0.101 CHEMBL4525762 | CHEMBL3526179 | |
| 0.282 | 0.172 | 0.282 | DNA directed DNA polymerase inhibitor | 0.282 0.172 CHEMBL3526439 | ||
| 0.113 | 0.004 | 0.113 | Peroxisome proliferator-activated receptor alpha antagonist | 0.023 0.014 CHEMBL3526179 0.113 0.004 CHEMBL3526439 0.041 0.009 CHEMBL3526178 | ||
| 0.119 | 0.014 | 0.16 | Prostaglandin antagonist | 0.16 0.009 CHEMBL3526179 0.119 0.014 CHEMBL3526439 0.116 0.014 CHEMBL3526178 | CHEMBL3526179 | |
| 0.229 | 0.135 | 0.298 | Ca(v)3.3 blocker | 0.298 0.044 CHEMBL3526179 0.229 0.135 CHEMBL3526439 | CHEMBL3526179 | |
| 0.091 | 0.006 | 0.091 | Peroxisome proliferator-activated receptor delta agonist | 0.091 0.006 CHEMBL3526439 0.044 0.015 CHEMBL3526178 | ||
| 0.107 | 0.023 | 0.115 | Leukotriene synthesis inhibitor | 0.059 0.057 CHEMBL3526440 0.107 0.023 CHEMBL3526439 0.115 0.019 CHEMBL3526178 0.072 0.043 CHEMBL4525762 | CHEMBL3526178 | |
| 0.3 | 0.216 | 0.64 | Antiinflammatory | 0.443 0.114 CHEMBL3526179 0.634 0.045 CHEMBL3526440 0.3 0.216 CHEMBL3526439 0.64 0.043 CHEMBL3526292 0.61 0.051 CHEMBL4525762 | CHEMBL3526292 | |
| 0.087 | 0.008 | 0.108 | Guanylate cyclase stimulant | 0.108 0.005 CHEMBL3526179 0.087 0.008 CHEMBL3526439 0.089 0.007 CHEMBL3526178 0.043 0.031 CHEMBL4525762 | CHEMBL3526179 | |
| 0.149 | 0.076 | 0.199 | Insulin secretagoues | 0.158 0.066 CHEMBL3526179 0.178 0.05 CHEMBL3526440 0.149 0.076 CHEMBL3526439 0.156 0.068 CHEMBL3526292 0.122 0.108 CHEMBL3526178 0.199 0.036 CHEMBL4525762 | CHEMBL4525762 | |
| 0.171 | 0.106 | 0.24 | Platelet aggregation inhibitor | 0.24 0.056 CHEMBL3526179 0.171 0.106 CHEMBL3526439 | CHEMBL3526179 | |
| 0.114 | 0.054 | 0.153 | Mediator release inhibitor | 0.134 0.037 CHEMBL3526440 0.114 0.054 CHEMBL3526439 0.095 0.075 CHEMBL3526292 0.153 0.027 CHEMBL4525762 | CHEMBL4525762 | |
| 0.139 | 0.087 | 0.283 | Phospholipase A2 inhibitor | 0.283 0.016 CHEMBL3526179 0.139 0.087 CHEMBL3526439 0.122 0.113 CHEMBL3526178 | CHEMBL3526179 | |
| 0.099 | 0.054 | 0.139 | Uric acid excretion stimulant | 0.108 0.046 CHEMBL3526440 0.099 0.054 CHEMBL3526439 0.106 0.047 CHEMBL3526292 0.126 0.035 CHEMBL3526178 0.139 0.028 CHEMBL4525762 | CHEMBL4525762 | |
| 0.218 | 0.173 | 0.218 | Calpain 2 inhibitor | 0.218 0.173 CHEMBL3526439 | ||
| 0.052 | 0.011 | 0.094 | Plasma kallikrein inhibitor | 0.094 0.005 CHEMBL3526179 0.052 0.011 CHEMBL3526439 0.048 0.013 CHEMBL3526178 | CHEMBL3526179 | |
| 0.133 | 0.097 | 0.173 | Protein-tyrosine phosphatase inhibitor | 0.127 0.105 CHEMBL3526440 0.133 0.097 CHEMBL3526439 0.135 0.095 CHEMBL3526292 0.173 0.06 CHEMBL3526178 0.144 0.085 CHEMBL4525762 | CHEMBL3526178 | |
| 0.045 | 0.012 | 0.045 | Free fatty acid receptor 1 antagonist | 0.034 0.023 CHEMBL3526179 0.045 0.012 CHEMBL3526439 0.032 0.026 CHEMBL3526178 | ||
| 0.042 | 0.013 | 0.042 | Peroxisome proliferator-activated receptor delta antagonist | 0.042 0.013 CHEMBL3526179 0.042 0.013 CHEMBL3526439 0.038 0.017 CHEMBL3526178 | ||
| 0.038 | 0.011 | 0.112 | Prostaglandin EP4 antagonist | 0.112 0.004 CHEMBL3526179 0.038 0.011 CHEMBL3526439 | CHEMBL3526179 | |
| 0.053 | 0.028 | 0.086 | Kallikrein inhibitor | 0.086 0.013 CHEMBL3526179 0.053 0.028 CHEMBL3526439 0.049 0.031 CHEMBL3526178 | CHEMBL3526179 | |
| 0.031 | 0.006 | 0.031 | Free fatty acid receptor 1 agonist | 0.023 0.008 CHEMBL3526179 0.031 0.006 CHEMBL3526439 0.031 0.006 CHEMBL3526178 | ||
| 0.063 | 0.041 | 0.105 | Prostaglandin F2 alpha antagonist | 0.105 0.01 CHEMBL3526179 0.063 0.041 CHEMBL3526439 0.069 0.033 CHEMBL3526178 0.056 0.054 CHEMBL4525762 | CHEMBL3526179 | |
| 0.055 | 0.033 | 0.061 | Sphingosine 1-phosphate receptor 5 agonist | 0.061 0.025 CHEMBL3526179 0.055 0.033 CHEMBL3526439 0.055 0.033 CHEMBL3526178 | CHEMBL3526179 | |
| 0.046 | 0.025 | 0.056 | Sphingosine 1-phosphate receptor 1 agonist | 0.056 0.015 CHEMBL3526179 0.046 0.025 CHEMBL3526439 | CHEMBL3526179 | |
| 0.028 | 0.008 | 0.028 | Guanylate cyclase 1 stimulant | 0.028 0.008 CHEMBL3526179 0.028 0.008 CHEMBL3526439 0.028 0.008 CHEMBL3526178 | ||
| 0.029 | 0.01 | 0.035 | Prostaglandin EP1 antagonist | 0.019 0.015 CHEMBL3526179 0.029 0.01 CHEMBL3526439 0.035 0.009 CHEMBL3526178 | CHEMBL3526178 | |
| 0.035 | 0.017 | 0.035 | Prostaglandin agonist | 0.035 0.017 CHEMBL3526439 0.035 0.017 CHEMBL3526178 | ||
| 0.029 | 0.011 | 0.029 | Prostaglandin E2 agonist | 0.029 0.011 CHEMBL3526439 0.028 0.012 CHEMBL3526178 | ||
| 0.046 | 0.029 | 0.06 | Sphingosine 1-phosphate receptor agonist | 0.06 0.017 CHEMBL3526179 0.046 0.029 CHEMBL3526439 | CHEMBL3526179 | |
| 0.031 | 0.015 | 0.033 | Leukotriene D4 antagonist | 0.031 0.015 CHEMBL3526439 0.033 0.014 CHEMBL3526178 0.024 0.021 CHEMBL4525762 | CHEMBL3526178 | |
| 0.097 | 0.081 | 0.097 | GABA receptor agonist | 0.097 0.081 CHEMBL3526439 | ||
| 0.052 | 0.037 | 0.061 | Autotaxin inhibitor | 0.052 0.037 CHEMBL3526439 0.061 0.028 CHEMBL3526178 | CHEMBL3526178 | |
| 0.06 | 0.047 | 0.06 | Phosphodiesterase 1C inhibitor | 0.06 0.047 CHEMBL3526439 | ||
| 0.127 | 0.116 | 0.127 | Mcl-1 antagonist | 0.127 0.116 CHEMBL3526439 0.123 0.122 CHEMBL3526178 | ||
| 0.03 | 0.021 | 0.042 | Prostaglandin EP3 antagonist | 0.042 0.013 CHEMBL3526179 0.03 0.021 CHEMBL3526439 0.036 0.017 CHEMBL3526178 | CHEMBL3526179 | |
| 0.056 | 0.048 | 0.056 | Phosphodiesterase 1B inhibitor | 0.054 0.052 CHEMBL3526179 0.056 0.048 CHEMBL3526439 | ||
| 0.054 | 0.047 | 0.097 | Prostaglandin EP2 antagonist | 0.097 0.02 CHEMBL3526179 0.054 0.047 CHEMBL3526439 0.053 0.048 CHEMBL4525762 | CHEMBL3526179 | |
| 0.08 | 0.076 | 0.092 | Phosphodiesterase I inhibitor | 0.092 0.055 CHEMBL3526179 0.08 0.076 CHEMBL3526439 | CHEMBL3526179 | |
| 0.025 | 0.022 | 0.035 | Leukotriene B4 receptor 1 antagonist | 0.035 0.015 CHEMBL3526179 0.025 0.022 CHEMBL3526439 | CHEMBL3526179 | |
| 0.043 | 0.041 | 0.043 | Benzodiazepine inverse agonist | 0.043 0.041 CHEMBL3526439 | ||
| 0.018 | 0.019 | 0.028 | Prostaglandin EP2 agonist | 0.028 0.013 CHEMBL3526178 | CHEMBL3526178 | |
| 0.027 | 0.029 | 0.039 | Prostacyclin antagonist | 0.039 0.018 CHEMBL3526179 | CHEMBL3526179 | |
| 0.067 | 0.072 | 0.123 | Macrophage migration inhibitory factor inhibitor | 0.123 0.024 CHEMBL3526179 0.079 0.052 CHEMBL3526178 | CHEMBL3526179 | |
| 0.03 | 0.038 | 0.048 | AMPA receptor agonist | 0.038 0.02 CHEMBL3526179 0.048 0.01 CHEMBL3526178 | CHEMBL3526178 | |
| 0.011 | 0.023 | 0.013 | Integrin beta6 antagonist | 0.013 0.012 CHEMBL3526179 | CHEMBL3526179 | |
| 0.021 | 0.033 | 0.031 | Protocollagen prolyl hydroxylase inhibitor | 0.031 0.014 CHEMBL3526179 0.031 0.014 CHEMBL3526178 | CHEMBL3526178 | |
| 0.083 | 0.097 | 0.09 | EphA2 antagonist | 0.09 0.087 CHEMBL3526178 | CHEMBL3526178 | |
| 0.021 | 0.034 | 0.104 | Sodium/glucose cotransporter 2 inhibitor | 0.086 0.004 CHEMBL3526440 0.077 0.004 CHEMBL3526292 0.104 0.003 CHEMBL4525762 | CHEMBL4525762 | |
| 0.021 | 0.037 | 0.095 | Sodium/glucose cotransporter inhibitor | 0.074 0.004 CHEMBL3526440 0.06 0.004 CHEMBL3526292 0.095 0.003 CHEMBL4525762 | CHEMBL4525762 | |
| 0.05 | 0.072 | 0.058 | CDC25B inhibitor | 0.058 0.054 CHEMBL3526178 | CHEMBL3526178 | |
| 0.018 | 0.041 | 0.03 | Sphingosine 1-phosphate receptor 3 agonist | 0.03 0.027 CHEMBL3526179 | CHEMBL3526179 | |
| 0.011 | 0.035 | 0.02 | Thyroid hormone alpha agonist | 0.02 0.007 CHEMBL3526179 | CHEMBL3526179 | |
| 0.008 | 0.032 | 0.022 | Egl nine homolog 1 inhibitor | 0.015 0.009 CHEMBL3526179 0.022 0.005 CHEMBL3526178 | CHEMBL3526178 | |
| 0.203 | 0.234 | 0.381 | Analgesic | 0.381 0.093 CHEMBL3526179 | CHEMBL3526179 | |
| 0.024 | 0.059 | 0.047 | Urate transporter 1 inhibitor | 0.047 0.02 CHEMBL3526178 | CHEMBL3526178 | |
| 0.038 | 0.073 | 0.046 | Phosphodiesterase 6C inhibitor | 0.046 0.033 CHEMBL3526179 | CHEMBL3526179 | |
| 0.108 | 0.147 | 0.128 | Dual specificity phosphatase 3 inhibitor | 0.128 0.118 CHEMBL3526178 | CHEMBL3526178 | |
| 0.037 | 0.081 | 0.054 | Leukotriene B4 antagonist | 0.054 0.037 CHEMBL3526179 | CHEMBL3526179 | |
| 0.042 | 0.088 | 0.076 | Lipase inhibitor | 0.076 0.047 CHEMBL3526179 0.067 0.057 CHEMBL3526440 | CHEMBL3526179 | |
| 0.01 | 0.057 | 0.037 | Somatostatin 5 antagonist | 0.037 0.02 CHEMBL3526179 | CHEMBL3526179 | |
| 0.069 | 0.121 | 0.099 | Protein-tyrosine phosphatase 1B inhibitor | 0.099 0.079 CHEMBL3526178 0.094 0.085 CHEMBL4525762 | CHEMBL3526178 | |
| 0.021 | 0.074 | 0.04 | Angiotensin II receptor antagonist | 0.04 0.014 CHEMBL3526179 | CHEMBL3526179 | |
| 0.024 | 0.077 | 0.051 | Angiotensin AT1 receptor antagonist | 0.051 0.016 CHEMBL3526179 | CHEMBL3526179 | |
| 0.07 | 0.128 | 0.125 | Xanthine oxidase inhibitor | 0.091 0.07 CHEMBL3526440 0.125 0.045 CHEMBL3526292 0.087 0.077 CHEMBL3526178 0.098 0.062 CHEMBL4525762 | CHEMBL3526292 | |
| 0.003 | 0.065 | 0.044 | Thyroid hormone beta agonist | 0.044 0.003 CHEMBL3526179 | CHEMBL3526179 | |
| 0.015 | 0.079 | 0.089 | Thyroid hormone agonist | 0.089 0.003 CHEMBL3526179 | CHEMBL3526179 | |
| 0.068 | 0.133 | 0.136 | Bile acid receptor antagonist | 0.136 0.011 CHEMBL3526179 0.089 0.077 CHEMBL3526178 | CHEMBL3526179 | |
| 0.044 | 0.113 | 0.058 | Leukotriene C antagonist | 0.058 0.033 CHEMBL3526179 | CHEMBL3526179 | |
| 0.024 | 0.101 | 0.08 | Thromboxane antagonist | 0.08 0.02 CHEMBL3526179 | CHEMBL3526179 | |
| 0.097 | 0.173 | 0.193 | Growth hormone agonist | 0.193 0.062 CHEMBL3526179 | CHEMBL3526179 | |
| 0.055 | 0.133 | 0.104 | Bronchodilator | 0.104 0.06 CHEMBL3526179 | CHEMBL3526179 | |
| 0.028 | 0.108 | 0.037 | Leukotriene C4 antagonist | 0.037 0.033 CHEMBL3526179 | CHEMBL3526179 | |
| 0.016 | 0.107 | 0.045 | 1-Alkyl-2-acetylglycerophosphocholine esterase inhibitor | 0.045 0.012 CHEMBL3526179 | CHEMBL3526179 | |
| 0.06 | 0.161 | 0.085 | ABCA1 expression enhancer | 0.085 0.074 CHEMBL3526179 | CHEMBL3526179 | |
| 0.086 | 0.192 | 0.2 | Arachidonic acid antagonist | 0.2 0.033 CHEMBL3526179 | CHEMBL3526179 | |
| 0.159 | 0.266 | 0.469 | Histamine release inhibitor | 0.469 0.041 CHEMBL3526179 0.234 0.168 CHEMBL4525762 | CHEMBL3526179 | |
| 0.098 | 0.221 | 0.192 | Non-steroidal antiinflammatory agent | 0.138 0.134 CHEMBL3526179 0.192 0.078 CHEMBL3526440 0.139 0.132 CHEMBL3526292 0.153 0.111 CHEMBL4525762 | CHEMBL3526440 | |
| 0.029 | 0.156 | 0.066 | Thromboxane synthase inhibitor | 0.066 0.021 CHEMBL3526179 | CHEMBL3526179 | |
| 0.062 | 0.197 | 0.193 | Thrombolytic | 0.123 0.107 CHEMBL3526179 0.167 0.07 CHEMBL3526440 0.163 0.072 CHEMBL3526292 0.193 0.055 CHEMBL4525762 | CHEMBL4525762 | |
| 0.021 | 0.161 | 0.045 | Diacylglycerol O-acyltransferase inhibitor | 0.045 0.044 CHEMBL3526179 | CHEMBL3526179 | |
| 0.057 | 0.202 | 0.102 | Nav1.4 sodium channel blocker | 0.102 0.074 CHEMBL3526179 | CHEMBL3526179 | |
| 0.034 | 0.181 | 0.071 | Histone deacetylase SIRT1 stimulant | 0.071 0.053 CHEMBL3526292 | CHEMBL3526292 | |
| 0.034 | 0.181 | 0.071 | Histone deacetylase stimulant | 0.071 0.053 CHEMBL3526292 | CHEMBL3526292 | |
| 0.035 | 0.184 | 0.149 | Monophenol monooxygenase inhibitor | 0.131 0.055 CHEMBL3526179 0.149 0.047 CHEMBL3526440 0.115 0.065 CHEMBL4525762 | CHEMBL3526440 | |
| 0.051 | 0.206 | 0.115 | DNA polymerase I inhibitor | 0.115 0.072 CHEMBL3526179 0.095 0.092 CHEMBL4525762 | CHEMBL3526179 | |
| 0.102 | 0.259 | 0.136 | CC chemokine 6 receptor antagonist | 0.132 0.064 CHEMBL3526440 0.13 0.069 CHEMBL3526292 0.136 0.052 CHEMBL4525762 | CHEMBL4525762 | |
| 0.081 | 0.239 | 0.278 | Hepatoprotectant | 0.262 0.04 CHEMBL3526440 0.278 0.036 CHEMBL3526292 0.267 0.039 CHEMBL4525762 | CHEMBL3526292 | |
| 0.024 | 0.188 | 0.072 | Glutamate receptor agonist | 0.072 0.061 CHEMBL3526178 | CHEMBL3526178 | |
| 0.144 | 0.313 | 0.327 | Interleukin 2 agonist | 0.243 0.127 CHEMBL3526179 0.327 0.057 CHEMBL3526440 0.238 0.133 CHEMBL3526292 0.324 0.058 CHEMBL4525762 | CHEMBL3526440 | |
| 0.121 | 0.302 | 0.33 | Immunomodulator | 0.317 0.073 CHEMBL3526440 0.33 0.067 CHEMBL3526292 0.286 0.09 CHEMBL4525762 | CHEMBL3526292 | |
| 0.135 | 0.323 | 0.196 | Caspase 3 stimulant | 0.196 0.176 CHEMBL3526440 0.19 0.184 CHEMBL4525762 | CHEMBL3526440 | |
| 0.033 | 0.223 | 0.07 | Adenine nucleotide translocase inhibitor | 0.063 0.024 CHEMBL3526440 0.07 0.015 CHEMBL3526292 | CHEMBL3526292 | |
| 0.023 | 0.225 | 0.055 | Glucose-6-phosphate translocase inhibitor | 0.052 0.034 CHEMBL3526440 0.055 0.03 CHEMBL3526292 0.055 0.03 CHEMBL4525762 | CHEMBL4525762 | |
| 0.084 | 0.29 | 0.338 | Antioxidant | 0.189 0.124 CHEMBL3526179 0.338 0.05 CHEMBL3526440 0.309 0.058 CHEMBL3526292 0.314 0.057 CHEMBL4525762 | CHEMBL3526440 | |
| 0.036 | 0.253 | 0.181 | Cholesterol synthesis inhibitor | 0.181 0.032 CHEMBL3526179 | CHEMBL3526179 | |
| 0.124 | 0.343 | 0.286 | Apoptosis antagonist | 0.209 0.168 CHEMBL3526179 0.255 0.123 CHEMBL3526440 0.213 0.163 CHEMBL3526292 0.286 0.095 CHEMBL4525762 | CHEMBL4525762 | |
| 0.033 | 0.261 | 0.085 | Sphingosine 1-phosphate receptor antagonist | 0.085 0.037 CHEMBL3526179 | CHEMBL3526179 | |
| 0.038 | 0.267 | 0.115 | Interleukin 1 beta converting enzyme inhibitor | 0.115 0.04 CHEMBL3526179 | CHEMBL3526179 | |
| 0.042 | 0.272 | 0.162 | Lipid peroxidase inhibitor | 0.162 0.061 CHEMBL3526440 0.157 0.064 CHEMBL3526292 0.129 0.084 CHEMBL4525762 | CHEMBL3526440 | |
| 0.076 | 0.311 | 0.207 | Vasodilator | 0.177 0.125 CHEMBL3526179 0.207 0.099 CHEMBL3526440 0.181 0.121 CHEMBL3526292 | CHEMBL3526440 | |
| 0.067 | 0.302 | 0.127 | Sphingosine 1-phosphate receptor 2 antagonist | 0.127 0.08 CHEMBL3526179 | CHEMBL3526179 | |
| 0.112 | 0.353 | 0.218 | Insulysin inhibitor | 0.218 0.132 CHEMBL3526179 | CHEMBL3526179 | |
| 0.055 | 0.296 | 0.178 | Cell wall synthesis inhibitor | 0.156 0.06 CHEMBL3526440 0.178 0.041 CHEMBL4525762 | CHEMBL4525762 | |
| 0.029 | 0.27 | 0.105 | Myeloperoxidase inhibitor | 0.105 0.03 CHEMBL3526179 | CHEMBL3526179 | |
| 0.022 | 0.268 | 0.056 | Sphingosine 1-phosphate receptor 1 antagonist | 0.056 0.036 CHEMBL3526179 | CHEMBL3526179 | |
| 0.008 | 0.255 | 0.032 | Nicotinic acid receptor agonist | 0.032 0.03 CHEMBL3526179 | CHEMBL3526179 | |
| 0.081 | 0.333 | 0.142 | Lipocortins synthesis antagonist | 0.142 0.117 CHEMBL3526179 | CHEMBL3526179 | |
| 0.048 | 0.301 | 0.115 | Cell adhesion inhibitor | 0.115 0.069 CHEMBL4525762 | CHEMBL4525762 | |
| 0.017 | 0.271 | 0.152 | Phenylalanine 4-hydroxylase inhibitor | 0.152 0.011 CHEMBL3526179 | CHEMBL3526179 | |
| 0.09 | 0.353 | 0.159 | Catenin beta inhibitor | 0.159 0.086 CHEMBL3526179 | CHEMBL3526179 | |
| 0.095 | 0.358 | 0.394 | Antithrombotic | 0.294 0.092 CHEMBL3526179 0.323 0.075 CHEMBL3526440 0.394 0.051 CHEMBL3526292 0.383 0.054 CHEMBL4525762 | CHEMBL3526292 | |
| 0.017 | 0.284 | 0.149 | Porphobilinogen synthase inhibitor | 0.149 0.021 CHEMBL3526179 | CHEMBL3526179 | |
| 0.144 | 0.412 | 0.317 | Calcium channel L-type activator | 0.317 0.143 CHEMBL3526179 | CHEMBL3526179 | |
| 0.024 | 0.301 | 0.145 | Alcohol dehydrogenase inhibitor | 0.145 0.022 CHEMBL3526179 | CHEMBL3526179 | |
| 0.076 | 0.367 | 0.432 | Transcription factor NF kappa B inhibitor | 0.432 0.057 CHEMBL3526440 0.429 0.057 CHEMBL3526292 0.298 0.095 CHEMBL4525762 | CHEMBL3526440 | |
| 0.012 | 0.313 | 0.181 | Selectin antagonist | 0.171 0.015 CHEMBL3526440 0.141 0.019 CHEMBL3526292 0.181 0.013 CHEMBL4525762 | CHEMBL4525762 | |
| 0.04 | 0.343 | 0.143 | Toll-Like receptor 4 antagonist | 0.102 0.067 CHEMBL3526179 0.123 0.041 CHEMBL3526440 0.143 0.025 CHEMBL3526292 0.095 0.079 CHEMBL4525762 | CHEMBL3526292 | |
| 0.058 | 0.367 | 0.173 | Hemostatic | 0.158 0.059 CHEMBL3526440 0.152 0.065 CHEMBL3526292 0.173 0.046 CHEMBL4525762 | CHEMBL4525762 | |
| 0.041 | 0.352 | 0.094 | Transcription factor NF kappa B stimulant | 0.078 0.076 CHEMBL3526440 0.094 0.046 CHEMBL3526292 0.079 0.072 CHEMBL4525762 | CHEMBL3526292 | |
| 0.05 | 0.362 | 0.204 | Nitric oxide antagonist | 0.204 0.066 CHEMBL3526440 0.186 0.073 CHEMBL3526292 0.181 0.076 CHEMBL4525762 | CHEMBL3526440 | |
| 0.041 | 0.354 | 0.168 | Aldehyde dehydrogenase inhibitor | 0.168 0.038 CHEMBL3526179 | CHEMBL3526179 | |
| 0.04 | 0.355 | 0.375 | Angiogenesis stimulant | 0.351 0.032 CHEMBL3526440 0.324 0.04 CHEMBL3526292 0.375 0.026 CHEMBL4525762 | CHEMBL4525762 | |
| 0.131 | 0.45 | 0.402 | 5 Hydroxytryptamine release inhibitor | 0.402 0.077 CHEMBL3526179 | CHEMBL3526179 | |
| 0.072 | 0.397 | 0.386 | Immunosuppressant | 0.347 0.088 CHEMBL3526440 0.386 0.069 CHEMBL3526292 0.291 0.121 CHEMBL4525762 | CHEMBL3526292 | |
| 0.031 | 0.366 | 0.057 | Lipocortins synthesis agonist | 0.057 0.043 CHEMBL3526292 | CHEMBL3526292 | |
| 0.056 | 0.394 | 0.23 | Succinate dehydrogenase inhibitor | 0.23 0.03 CHEMBL3526179 | CHEMBL3526179 | |
| 0.052 | 0.391 | 0.251 | Antipruritic | 0.251 0.024 CHEMBL3526179 | CHEMBL3526179 | |
| 0.031 | 0.376 | 0.081 | Thioredoxin inhibitor | 0.081 0.079 CHEMBL3526292 | CHEMBL3526292 | |
| 0.028 | 0.395 | 0.09 | GABA B receptor agonist | 0.09 0.025 CHEMBL3526179 | CHEMBL3526179 | |
| 0.063 | 0.437 | 0.187 | Superoxide dismutase inhibitor | 0.187 0.132 CHEMBL3526179 | CHEMBL3526179 | |
| 0.034 | 0.412 | 0.115 | Estrogen antagonist | 0.115 0.065 CHEMBL3526179 | CHEMBL3526179 | |
| 0.099 | 0.477 | 0.422 | Apoptosis agonist | 0.422 0.103 CHEMBL3526440 0.412 0.108 CHEMBL3526292 0.27 0.195 CHEMBL4525762 | CHEMBL3526440 | |
| 0.051 | 0.433 | 0.116 | DNA repair enzyme inhibitor | 0.116 0.08 CHEMBL3526440 | CHEMBL3526440 | |
| 0.041 | 0.425 | 0.255 | Free radical scavenger | 0.15 0.145 CHEMBL3526179 0.255 0.066 CHEMBL3526440 0.247 0.07 CHEMBL3526292 0.238 0.074 CHEMBL4525762 | CHEMBL3526440 | |
| 0.03 | 0.421 | 0.123 | Amylase inhibitor | 0.123 0.079 CHEMBL3526179 | CHEMBL3526179 | |
| 0.031 | 0.43 | 0.109 | Toll-Like receptor 2 antagonist | 0.109 0.091 CHEMBL3526179 | CHEMBL3526179 | |
| 0.021 | 0.428 | 0.127 | Ferrochelatase inhibitor | 0.127 0.049 CHEMBL3526179 | CHEMBL3526179 | |
| 0.034 | 0.442 | 0.101 | Phosphodiesterase 6D inhibitor | 0.101 0.051 CHEMBL3526179 | CHEMBL3526179 | |
| 0.088 | 0.51 | 0.137 | Heat shock protein 70 antagonist | 0.137 0.088 CHEMBL3526179 | CHEMBL3526179 | |
| 0.057 | 0.491 | 0.127 | Sphingosine 1-phosphate receptor 5 antagonist | 0.127 0.108 CHEMBL3526179 | CHEMBL3526179 | |
| 0.038 | 0.475 | 0.091 | Adenylate kinase inhibitor | 0.091 0.085 CHEMBL3526179 | CHEMBL3526179 | |
| 0.038 | 0.476 | 0.11 | Interleukin 4 antagonist | 0.11 0.1 CHEMBL3526179 | CHEMBL3526179 | |
| 0.066 | 0.511 | 0.196 | Vasodilator, coronary | 0.196 0.186 CHEMBL3526179 | CHEMBL3526179 | |
| 0.084 | 0.531 | 0.327 | Tyrosine 3 hydroxylase inhibitor | 0.327 0.022 CHEMBL3526179 | CHEMBL3526179 | |
| 0.02 | 0.467 | 0.088 | Estrogen receptor beta antagonist | 0.088 0.087 CHEMBL3526179 | CHEMBL3526179 | |
| 0.041 | 0.495 | 0.136 | Melanin inhibitor | 0.136 0.102 CHEMBL3526179 | CHEMBL3526179 | |
| 0.059 | 0.516 | 0.538 | Antibacterial | 0.522 0.035 CHEMBL3526440 0.536 0.032 CHEMBL3526292 0.538 0.031 CHEMBL4525762 | CHEMBL4525762 | |
| 0.017 | 0.494 | 0.159 | Creatine kinase inhibitor | 0.159 0.021 CHEMBL3526179 | CHEMBL3526179 | |
| 0.011 | 0.49 | 0.066 | Aminopeptidase I inhibitor | 0.066 0.059 CHEMBL3526179 | CHEMBL3526179 | |
| 0.011 | 0.517 | 0.027 | Toll-Like receptor 4 agonist | 0.027 0.017 CHEMBL3526292 | CHEMBL3526292 | |
| 0.024 | 0.532 | 0.098 | DOPA decarboxylase inhibitor | 0.098 0.081 CHEMBL3526179 | CHEMBL3526179 | |
| 0.005 | 0.524 | 0.06 | Alcohol oxidase inhibitor | 0.06 0.035 CHEMBL3526179 | CHEMBL3526179 | |
| 0.026 | 0.546 | 0.22 | Alpha-glucosidase inhibitor | 0.22 0.206 CHEMBL3526440 0.216 0.209 CHEMBL3526292 | CHEMBL3526440 | |
| 0.053 | 0.574 | 0.149 | Neurotensin receptor agonist | 0.149 0.103 CHEMBL3526179 | CHEMBL3526179 | |
| 0.013 | 0.539 | 0.15 | Anesthetic general | 0.15 0.114 CHEMBL3526179 | CHEMBL3526179 | |
| 0.02 | 0.548 | 0.118 | Protein kinase stimulant | 0.118 0.094 CHEMBL3526179 | CHEMBL3526179 | |
| 0.007 | 0.55 | 0.072 | Glutamate decarboxylase inhibitor | 0.072 0.052 CHEMBL3526179 | CHEMBL3526179 | |
| 0.068 | 0.616 | 0.134 | Ca2+-transporting ATPase inhibitor | 0.134 0.1 CHEMBL3526179 | CHEMBL3526179 | |
| 0.038 | 0.593 | 0.151 | NOS3 expression enhancer | 0.151 0.071 CHEMBL3526292 | CHEMBL3526292 | |
| 0.011 | 0.567 | 0.046 | Antibiotic Aminoglycoside-like | 0.041 0.02 CHEMBL3526440 0.037 0.024 CHEMBL3526292 0.046 0.016 CHEMBL4525762 | CHEMBL4525762 | |
| 0.031 | 0.596 | 0.083 | Estrogen-related receptor beta agonist | 0.083 0.059 CHEMBL3526179 | CHEMBL3526179 | |
| 0.076 | 0.645 | 0.276 | Peptidyltransferase inhibitor | 0.237 0.061 CHEMBL3526440 0.208 0.089 CHEMBL3526292 0.276 0.035 CHEMBL4525762 | CHEMBL4525762 | |
| 0.012 | 0.583 | 0.104 | Cystathionine beta-synthase inhibitor | 0.104 0.073 CHEMBL3526179 | CHEMBL3526179 | |
| 0.031 | 0.603 | 0.177 | Interleukin agonist | 0.177 0.142 CHEMBL3526179 | CHEMBL3526179 | |
| 0.013 | 0.587 | 0.088 | GABA C receptor agonist | 0.088 0.081 CHEMBL3526179 | CHEMBL3526179 | |
| 0.048 | 0.661 | 0.267 | GABA C receptor rho-3 antagonist | 0.267 0.14 CHEMBL3526179 | CHEMBL3526179 | |
| 0.024 | 0.639 | 0.187 | Tumour necrosis factor alpha release inhibitor | 0.187 0.121 CHEMBL3526440 0.179 0.127 CHEMBL3526292 | CHEMBL3526440 | |
| 0.021 | 0.659 | 0.133 | Adenylate cyclase stimulant | 0.133 0.094 CHEMBL3526179 | CHEMBL3526179 | |
| 0.05 | 0.689 | 0.164 | 5 Hydroxytryptamine release stimulant | 0.164 0.161 CHEMBL3526179 | CHEMBL3526179 | |
| 0.017 | 0.694 | 0.201 | Aldehyde oxidase inhibitor | 0.201 0.104 CHEMBL3526179 | CHEMBL3526179 | |
| 0.011 | 0.706 | 0.161 | Spasmolytic | 0.161 0.153 CHEMBL3526179 | CHEMBL3526179 | |
| 0.056 | 0.759 | 0.169 | Nitric-oxide synthase stimulant | 0.169 0.155 CHEMBL3526179 | CHEMBL3526179 | |
| 0.007 | 0.762 | 0.05 | Protein 50S ribosomal subunit inhibitor | 0.046 0.044 CHEMBL3526440 0.05 0.04 CHEMBL3526292 0.05 0.04 CHEMBL4525762 | CHEMBL4525762 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |