| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.975 | 0.004 | 0.98 | Cyclophilin D inhibitor | 0.688 0.015 CHEMBL3526469 0.976 0.004 CHEMBL3526208 0.286 0.175 CHEMBL3526243 0.908 0.005 CHEMBL3526849 0.979 0.004 CHEMBL3526767 0.481 0.056 CHEMBL3526242 0.975 0.004 CHEMBL3526746 0.918 0.004 CHEMBL3542322 0.969 0.004 CHEMBL3526234 0.64 0.021 CHEMBL3527076 0.812 0.006 CHEMBL3527595 0.811 0.006 CHEMBL3526963 0.735 0.011 CHEMBL3527594 0.705 0.014 CHEMBL3526660 0.594 0.028 CHEMBL3526244 0.6 0.027 CHEMBL3526471 0.414 0.083 CHEMBL3526620 0.807 0.006 CHEMBL3526470 0.719 0.012 CHEMBL3526829 0.682 0.016 CHEMBL3526211 0.789 0.007 CHEMBL3526754 0.98 0.004 CHEMBL3526766 | CHEMBL3526766 | |
| 0.881 | 0.004 | 0.9 | Hypoglycemic | 0.72 0.005 CHEMBL3526469 0.887 0.003 CHEMBL3526208 0.353 0.037 CHEMBL3526243 0.747 0.004 CHEMBL3526849 0.874 0.004 CHEMBL3526767 0.58 0.009 CHEMBL3526242 0.9 0.003 CHEMBL3526746 0.767 0.004 CHEMBL3542322 0.788 0.004 CHEMBL3526234 0.537 0.012 CHEMBL3527076 0.695 0.005 CHEMBL3527595 0.596 0.008 CHEMBL3526963 0.197 0.116 CHEMBL3527594 0.294 0.055 CHEMBL3526660 0.523 0.013 CHEMBL3526244 0.503 0.015 CHEMBL3526471 0.496 0.015 CHEMBL3526620 0.709 0.005 CHEMBL3526470 0.331 0.043 CHEMBL3526829 0.447 0.021 CHEMBL3526211 0.579 0.009 CHEMBL3526754 0.881 0.004 CHEMBL3526766 | CHEMBL3526746 | |
| 0.802 | 0 | 0.885 | Thiazolidinedione | 0.164 0.001 CHEMBL3526469 0.724 0 CHEMBL3526208 0.055 0.005 CHEMBL3526243 0.219 0.001 CHEMBL3526849 0.885 0 CHEMBL3526767 0.057 0.004 CHEMBL3526242 0.327 0.001 CHEMBL3526746 0.224 0.001 CHEMBL3542322 0.481 0 CHEMBL3526234 0.054 0.005 CHEMBL3527076 0.038 0.009 CHEMBL3527595 0.045 0.007 CHEMBL3526963 0.048 0.005 CHEMBL3527594 0.048 0.005 CHEMBL3526660 0.056 0.004 CHEMBL3526244 0.058 0.004 CHEMBL3526471 0.045 0.007 CHEMBL3526620 0.059 0.004 CHEMBL3526470 0.053 0.005 CHEMBL3526829 0.053 0.005 CHEMBL3526211 0.046 0.006 CHEMBL3526754 0.859 0 CHEMBL3526766 | CHEMBL3526767 | |
| 0.75 | 0.002 | 0.75 | Peroxisome proliferator-activated receptor gamma agonist | 0.244 0.005 CHEMBL3526469 0.744 0.002 CHEMBL3526208 0.155 0.012 CHEMBL3526243 0.372 0.004 CHEMBL3526849 0.679 0.003 CHEMBL3526767 0.24 0.005 CHEMBL3526242 0.574 0.003 CHEMBL3526746 0.384 0.004 CHEMBL3542322 0.616 0.003 CHEMBL3526234 0.154 0.012 CHEMBL3527076 0.126 0.019 CHEMBL3527595 0.285 0.005 CHEMBL3526963 0.096 0.03 CHEMBL3527594 0.093 0.032 CHEMBL3526660 0.368 0.004 CHEMBL3526244 0.152 0.012 CHEMBL3526471 0.254 0.005 CHEMBL3526620 0.494 0.004 CHEMBL3526470 0.147 0.014 CHEMBL3526829 0.142 0.015 CHEMBL3526211 0.275 0.005 CHEMBL3526754 0.672 0.003 CHEMBL3526766 | ||
| 0.713 | 0.002 | 0.823 | Insulin sensitizer | 0.266 0.026 CHEMBL3526469 0.798 0.002 CHEMBL3526208 0.144 0.141 CHEMBL3526243 0.306 0.014 CHEMBL3526849 0.745 0.002 CHEMBL3526767 0.427 0.005 CHEMBL3526242 0.771 0.002 CHEMBL3526746 0.323 0.012 CHEMBL3542322 0.589 0.003 CHEMBL3526234 0.229 0.048 CHEMBL3527076 0.221 0.054 CHEMBL3527595 0.158 0.123 CHEMBL3526660 0.213 0.06 CHEMBL3526244 0.205 0.068 CHEMBL3526471 0.309 0.014 CHEMBL3526620 0.268 0.025 CHEMBL3526470 0.195 0.079 CHEMBL3526211 0.823 0.002 CHEMBL3526766 | CHEMBL3526766 | |
| 0.591 | 0.007 | 0.645 | Hypolipemic | 0.604 0.006 CHEMBL3526208 0.446 0.018 CHEMBL3526849 0.633 0.005 CHEMBL3526767 0.592 0.007 CHEMBL3526746 0.461 0.016 CHEMBL3542322 0.531 0.01 CHEMBL3526234 0.213 0.085 CHEMBL3527595 0.286 0.053 CHEMBL3526963 0.36 0.033 CHEMBL3526470 0.271 0.059 CHEMBL3526754 0.645 0.005 CHEMBL3526766 | CHEMBL3526766 | |
| 0.525 | 0.005 | 0.574 | Insulin secretagoues | 0.227 0.025 CHEMBL3526469 0.541 0.005 CHEMBL3526208 0.193 0.039 CHEMBL3526243 0.486 0.005 CHEMBL3526849 0.358 0.008 CHEMBL3526767 0.325 0.01 CHEMBL3526242 0.574 0.004 CHEMBL3526746 0.505 0.005 CHEMBL3542322 0.331 0.009 CHEMBL3526234 0.263 0.017 CHEMBL3527076 0.361 0.008 CHEMBL3527595 0.275 0.015 CHEMBL3526963 0.206 0.033 CHEMBL3526660 0.329 0.01 CHEMBL3526244 0.241 0.021 CHEMBL3526471 0.309 0.011 CHEMBL3526620 0.398 0.006 CHEMBL3526470 0.2 0.036 CHEMBL3526829 0.348 0.008 CHEMBL3526211 0.259 0.018 CHEMBL3526754 0.382 0.007 CHEMBL3526766 | CHEMBL3526746 | |
| 0.453 | 0.007 | 0.47 | Sodium/bile acid cotransporter inhibitor | 0.288 0.09 CHEMBL3526469 0.461 0.006 CHEMBL3526208 0.381 0.024 CHEMBL3526849 0.461 0.006 CHEMBL3526767 0.426 0.011 CHEMBL3526746 0.388 0.021 CHEMBL3542322 0.442 0.009 CHEMBL3526234 0.224 0.157 CHEMBL3526660 0.215 0.168 CHEMBL3526470 0.226 0.155 CHEMBL3526211 0.47 0.005 CHEMBL3526766 | CHEMBL3526766 | |
| 0.424 | 0.004 | 0.469 | Aldose reductase inhibitor | 0.085 0.022 CHEMBL3526469 0.457 0.004 CHEMBL3526208 0.178 0.008 CHEMBL3526849 0.439 0.004 CHEMBL3526767 0.374 0.004 CHEMBL3526746 0.198 0.007 CHEMBL3542322 0.402 0.004 CHEMBL3526234 0.469 0.003 CHEMBL3526766 | CHEMBL3526766 | |
| 0.45 | 0.053 | 0.481 | Prostaglandin dehydrogenase inhibitor | 0.481 0.046 CHEMBL3526208 0.412 0.064 CHEMBL3526767 0.445 0.055 CHEMBL3526766 | CHEMBL3526208 | |
| 0.378 | 0.013 | 0.426 | MAO inhibitor | 0.426 0.01 CHEMBL3526208 0.238 0.031 CHEMBL3526767 0.105 0.086 CHEMBL3526234 0.275 0.023 CHEMBL3526766 | CHEMBL3526208 | |
| 0.401 | 0.065 | 0.54 | Antiobesity | 0.421 0.058 CHEMBL3526208 0.414 0.06 CHEMBL3526767 0.456 0.048 CHEMBL3526746 0.54 0.029 CHEMBL3526234 0.219 0.188 CHEMBL3526660 0.435 0.054 CHEMBL3526766 | CHEMBL3526234 | |
| 0.271 | 0.015 | 0.32 | MAO B inhibitor | 0.32 0.011 CHEMBL3526208 0.172 0.031 CHEMBL3526767 0.206 0.023 CHEMBL3526766 | CHEMBL3526208 | |
| 0.249 | 0.003 | 0.307 | Free fatty acid receptor 1 agonist | 0.237 0.003 CHEMBL3526208 0.026 0.008 CHEMBL3526849 0.307 0.003 CHEMBL3526767 0.097 0.004 CHEMBL3526746 0.026 0.007 CHEMBL3542322 0.119 0.004 CHEMBL3526234 0.293 0.003 CHEMBL3526766 | CHEMBL3526767 | |
| 0.305 | 0.069 | 0.393 | Lipoxygenase inhibitor | 0.393 0.039 CHEMBL3526208 0.276 0.083 CHEMBL3526767 0.192 0.148 CHEMBL3527076 0.299 0.072 CHEMBL3526244 0.319 0.062 CHEMBL3526470 0.36 0.048 CHEMBL3526766 | CHEMBL3526208 | |
| 0.282 | 0.049 | 0.591 | Cyclic AMP phosphodiesterase inhibitor | 0.273 0.053 CHEMBL3526208 0.591 0.004 CHEMBL3526849 0.298 0.043 CHEMBL3526767 0.422 0.014 CHEMBL3526746 0.576 0.004 CHEMBL3542322 0.29 0.046 CHEMBL3526766 | CHEMBL3526849 | |
| 0.291 | 0.1 | 0.33 | Calcium channel activator | 0.232 0.169 CHEMBL3526208 0.238 0.162 CHEMBL3526849 0.33 0.064 CHEMBL3526767 0.276 0.117 CHEMBL3526766 | CHEMBL3526767 | |
| 0.198 | 0.011 | 0.216 | Phosphodiesterase I inhibitor | 0.095 0.051 CHEMBL3526469 0.153 0.017 CHEMBL3526208 0.092 0.056 CHEMBL3526849 0.216 0.009 CHEMBL3526767 0.081 0.074 CHEMBL3542322 0.171 0.014 CHEMBL3526766 | CHEMBL3526767 | |
| 0.194 | 0.01 | 0.238 | ABCA1 expression enhancer | 0.2 0.009 CHEMBL3526208 0.09 0.065 CHEMBL3526849 0.23 0.007 CHEMBL3526767 0.125 0.027 CHEMBL3526746 0.093 0.061 CHEMBL3542322 0.147 0.018 CHEMBL3526234 0.238 0.007 CHEMBL3526766 | CHEMBL3526766 | |
| 0.212 | 0.036 | 0.349 | NOS3 expression enhancer | 0.285 0.02 CHEMBL3526208 0.153 0.069 CHEMBL3526849 0.286 0.02 CHEMBL3526767 0.349 0.012 CHEMBL3526746 0.189 0.045 CHEMBL3542322 0.17 0.056 CHEMBL3526234 0.348 0.012 CHEMBL3526766 | CHEMBL3526746 | |
| 0.166 | 0.004 | 0.192 | Estrogen-related receptor alpha antagonist | 0.105 0.005 CHEMBL3526469 0.167 0.004 CHEMBL3526208 0.069 0.009 CHEMBL3526849 0.191 0.003 CHEMBL3526767 0.088 0.007 CHEMBL3526746 0.073 0.009 CHEMBL3542322 0.108 0.005 CHEMBL3526234 0.192 0.003 CHEMBL3526766 | CHEMBL3526766 | |
| 0.292 | 0.164 | 0.4 | Calcium channel L-type activator | 0.324 0.137 CHEMBL3526469 0.37 0.103 CHEMBL3526208 0.332 0.131 CHEMBL3526767 0.358 0.111 CHEMBL3526242 0.292 0.164 CHEMBL3527076 0.253 0.202 CHEMBL3526244 0.235 0.222 CHEMBL3526470 0.4 0.081 CHEMBL3526766 | CHEMBL3526766 | |
| 0.179 | 0.051 | 0.303 | Lipid peroxidase inhibitor | 0.113 0.101 CHEMBL3526469 0.228 0.032 CHEMBL3526208 0.13 0.084 CHEMBL3526849 0.191 0.045 CHEMBL3526767 0.303 0.018 CHEMBL3526746 0.153 0.066 CHEMBL3542322 0.181 0.05 CHEMBL3526234 0.126 0.088 CHEMBL3527595 0.134 0.08 CHEMBL3526963 0.113 0.101 CHEMBL3526754 0.246 0.028 CHEMBL3526766 | CHEMBL3526746 | |
| 0.144 | 0.021 | 0.232 | Telomerase inhibitor | 0.072 0.051 CHEMBL3526469 0.159 0.019 CHEMBL3526208 0.217 0.012 CHEMBL3526767 0.079 0.045 CHEMBL3526746 0.066 0.056 CHEMBL3526234 0.232 0.011 CHEMBL3526766 | CHEMBL3526766 | |
| 0.177 | 0.057 | 0.24 | Interleukin 6 antagonist | 0.189 0.048 CHEMBL3526208 0.174 0.06 CHEMBL3526767 0.24 0.025 CHEMBL3526746 0.131 0.124 CHEMBL3527595 0.188 0.049 CHEMBL3526766 | CHEMBL3526746 | |
| 0.132 | 0.02 | 0.387 | Adrenaline agonist | 0.219 0.005 CHEMBL3526208 0.277 0.004 CHEMBL3526767 0.387 0.003 CHEMBL3526766 | CHEMBL3526766 | |
| 0.121 | 0.01 | 0.199 | Phosphodiesterase 1B inhibitor | 0.09 0.017 CHEMBL3526208 0.199 0.005 CHEMBL3526767 0.151 0.007 CHEMBL3526766 | CHEMBL3526767 | |
| 0.111 | 0.013 | 0.135 | Maillard reaction inhibitor | 0.125 0.009 CHEMBL3526208 0.12 0.01 CHEMBL3526767 0.101 0.016 CHEMBL3526746 0.058 0.036 CHEMBL3526234 0.135 0.008 CHEMBL3526766 | CHEMBL3526766 | |
| 0.111 | 0.022 | 0.14 | Lipase inhibitor | 0.124 0.016 CHEMBL3526208 0.127 0.015 CHEMBL3526767 0.101 0.027 CHEMBL3526746 0.14 0.012 CHEMBL3526766 | CHEMBL3526766 | |
| 0.203 | 0.116 | 0.548 | Cardiotonic | 0.182 0.137 CHEMBL3526208 0.548 0.011 CHEMBL3526243 0.193 0.125 CHEMBL3526767 0.423 0.025 CHEMBL3527076 0.325 0.047 CHEMBL3527595 0.319 0.049 CHEMBL3526244 0.446 0.021 CHEMBL3526471 0.366 0.035 CHEMBL3526620 0.191 0.128 CHEMBL3526470 0.256 0.078 CHEMBL3526829 0.166 0.157 CHEMBL3526211 0.171 0.15 CHEMBL3526766 | CHEMBL3526243 | |
| 0.226 | 0.14 | 0.226 | Thyroid hormone antagonist | 0.207 0.156 CHEMBL3526208 0.191 0.17 CHEMBL3526767 | ||
| 0.1 | 0.015 | 0.122 | Peroxisome proliferator-activated receptor gamma antagonist | 0.101 0.015 CHEMBL3526208 0.12 0.01 CHEMBL3526767 0.066 0.065 CHEMBL3526234 0.07 0.054 CHEMBL3526244 0.109 0.012 CHEMBL3526470 0.122 0.009 CHEMBL3526766 | CHEMBL3526766 | |
| 0.088 | 0.015 | 0.143 | Peroxisome proliferator-activated receptor alpha agonist | 0.082 0.017 CHEMBL3526208 0.103 0.012 CHEMBL3526767 0.046 0.035 CHEMBL3526746 0.045 0.036 CHEMBL3526244 0.143 0.007 CHEMBL3526470 0.097 0.013 CHEMBL3526766 | CHEMBL3526470 | |
| 0.138 | 0.066 | 0.165 | Phosphodiesterase inhibitor | 0.165 0.049 CHEMBL3526767 0.104 0.101 CHEMBL3526766 | CHEMBL3526767 | |
| 0.183 | 0.129 | 0.478 | Antioxidant | 0.254 0.081 CHEMBL3526208 0.262 0.077 CHEMBL3526849 0.18 0.132 CHEMBL3526767 0.478 0.023 CHEMBL3526746 0.293 0.064 CHEMBL3542322 0.28 0.07 CHEMBL3526234 0.356 0.045 CHEMBL3527595 0.253 0.082 CHEMBL3526963 0.164 0.149 CHEMBL3527594 0.172 0.14 CHEMBL3526620 0.225 0.098 CHEMBL3526754 0.256 0.08 CHEMBL3526766 | CHEMBL3526746 | |
| 0.115 | 0.062 | 0.152 | Alpha 2b adrenoreceptor antagonist | 0.152 0.038 CHEMBL3526767 0.108 0.068 CHEMBL3526766 | CHEMBL3526767 | |
| 0.162 | 0.109 | 0.162 | MAP kinase kinase 5 inhibitor | 0.16 0.117 CHEMBL3526469 0.161 0.111 CHEMBL3526242 | ||
| 0.084 | 0.032 | 0.099 | Phosphodiesterase III inhibitor | 0.071 0.042 CHEMBL3526208 0.099 0.023 CHEMBL3526767 0.085 0.031 CHEMBL3526766 | CHEMBL3526767 | |
| 0.06 | 0.019 | 0.076 | Phosphodiesterase 3B inhibitor | 0.059 0.02 CHEMBL3526208 0.076 0.015 CHEMBL3526767 0.075 0.016 CHEMBL3526766 | CHEMBL3526767 | |
| 0.102 | 0.062 | 0.139 | Bronchodilator | 0.096 0.069 CHEMBL3526208 0.139 0.035 CHEMBL3526767 0.13 0.039 CHEMBL3526766 | CHEMBL3526767 | |
| 0.049 | 0.01 | 0.07 | Peroxisome proliferator-activated receptor delta antagonist | 0.052 0.009 CHEMBL3526208 0.064 0.007 CHEMBL3526767 0.037 0.018 CHEMBL3526746 0.033 0.024 CHEMBL3526234 0.07 0.007 CHEMBL3526766 | CHEMBL3526766 | |
| 0.03 | 0.012 | 0.11 | Thyroid hormone agonist | 0.064 0.004 CHEMBL3526208 0.051 0.004 CHEMBL3526767 0.064 0.004 CHEMBL3526234 0.11 0.002 CHEMBL3526766 | CHEMBL3526766 | |
| 0.197 | 0.183 | 0.367 | Apoptosis antagonist | 0.233 0.144 CHEMBL3526208 0.267 0.111 CHEMBL3526849 0.282 0.099 CHEMBL3526767 0.367 0.048 CHEMBL3526746 0.277 0.102 CHEMBL3542322 0.287 0.094 CHEMBL3527595 0.311 0.079 CHEMBL3526766 | CHEMBL3526746 | |
| 0.122 | 0.111 | 0.28 | Protein-tyrosine phosphatase inhibitor | 0.153 0.075 CHEMBL3526208 0.178 0.058 CHEMBL3526767 0.156 0.073 CHEMBL3526746 0.28 0.023 CHEMBL3526234 0.129 0.103 CHEMBL3526660 0.22 0.04 CHEMBL3526766 | CHEMBL3526234 | |
| 0.108 | 0.097 | 0.169 | Bone formation stimulant | 0.137 0.07 CHEMBL3526208 0.143 0.065 CHEMBL3526767 0.125 0.081 CHEMBL3526746 0.169 0.046 CHEMBL3526766 | CHEMBL3526766 | |
| 0.092 | 0.082 | 0.389 | AMP-activated protein kinase stimulant | 0.129 0.042 CHEMBL3526208 0.167 0.019 CHEMBL3526849 0.152 0.027 CHEMBL3526767 0.389 0.004 CHEMBL3526746 0.188 0.013 CHEMBL3542322 0.19 0.013 CHEMBL3526766 | CHEMBL3526746 | |
| 0.086 | 0.079 | 0.093 | Toll-Like receptor 3 antagonist | 0.093 0.062 CHEMBL3526767 0.085 0.081 CHEMBL3526242 | CHEMBL3526767 | |
| 0.049 | 0.047 | 0.075 | Phosphodiesterase 4C inhibitor | 0.075 0.023 CHEMBL3526767 0.066 0.029 CHEMBL3526211 | CHEMBL3526767 | |
| 0.05 | 0.048 | 0.058 | Bombesin 3 receptor antagonist | 0.052 0.043 CHEMBL3526208 0.055 0.038 CHEMBL3526767 0.058 0.034 CHEMBL3526766 | CHEMBL3526766 | |
| 0.018 | 0.019 | 0.03 | Aggrecanase 2 inhibitor | 0.022 0.015 CHEMBL3526208 0.025 0.012 CHEMBL3526767 0.03 0.01 CHEMBL3526766 | CHEMBL3526766 | |
| 0.042 | 0.044 | 0.104 | Beta adrenoreceptor agonist | 0.057 0.01 CHEMBL3526208 0.059 0.009 CHEMBL3526767 0.104 0.004 CHEMBL3526766 | CHEMBL3526766 | |
| 0.089 | 0.091 | 0.194 | Protein-tyrosine phosphatase 1B inhibitor | 0.117 0.065 CHEMBL3526208 0.157 0.043 CHEMBL3526767 0.135 0.053 CHEMBL3526746 0.182 0.034 CHEMBL3526234 0.194 0.031 CHEMBL3526766 | CHEMBL3526766 | |
| 0.087 | 0.091 | 0.121 | EphA2 antagonist | 0.107 0.068 CHEMBL3526243 0.115 0.059 CHEMBL3526767 0.121 0.054 CHEMBL3526242 0.12 0.054 CHEMBL3526471 0.094 0.083 CHEMBL3526620 0.101 0.074 CHEMBL3526470 0.091 0.086 CHEMBL3526211 | CHEMBL3526242 | |
| 0.013 | 0.02 | 0.027 | Peroxisome proliferator-activated receptor alpha antagonist | 0.022 0.015 CHEMBL3526767 0.023 0.014 CHEMBL3526470 0.027 0.012 CHEMBL3526766 | CHEMBL3526766 | |
| 0.005 | 0.014 | 0.056 | Thyroid hormone beta agonist | 0.016 0.004 CHEMBL3526208 0.012 0.004 CHEMBL3526767 0.056 0.002 CHEMBL3526766 | CHEMBL3526766 | |
| 0.038 | 0.048 | 0.066 | Alpha 1L adrenoreceptor agonist | 0.066 0.006 CHEMBL3526767 0.059 0.009 CHEMBL3526766 | CHEMBL3526767 | |
| 0.02 | 0.031 | 0.027 | Phosphodiesterase 9A inhibitor | 0.027 0.012 CHEMBL3526767 0.025 0.016 CHEMBL3526766 | CHEMBL3526767 | |
| 0.074 | 0.087 | 0.097 | MAO A inhibitor | 0.097 0.066 CHEMBL3526208 | CHEMBL3526208 | |
| 0.115 | 0.13 | 0.23 | Growth hormone agonist | 0.14 0.095 CHEMBL3526208 0.121 0.12 CHEMBL3526767 0.15 0.087 CHEMBL3526242 0.23 0.049 CHEMBL3527076 0.125 0.113 CHEMBL3527595 0.191 0.062 CHEMBL3526471 0.169 0.074 CHEMBL3526620 0.17 0.073 CHEMBL3526470 0.129 0.109 CHEMBL3526829 0.129 0.109 CHEMBL3526211 0.152 0.086 CHEMBL3526766 | CHEMBL3527076 | |
| 0.017 | 0.034 | 0.026 | Phosphodiesterase IX inhibitor | 0.026 0.013 CHEMBL3526767 0.023 0.017 CHEMBL3526766 | CHEMBL3526767 | |
| 0.12 | 0.152 | 0.327 | Hepatoprotectant | 0.137 0.124 CHEMBL3526208 0.279 0.036 CHEMBL3526849 0.327 0.023 CHEMBL3526746 0.286 0.034 CHEMBL3542322 0.16 0.1 CHEMBL3526234 0.295 0.031 CHEMBL3527595 0.177 0.082 CHEMBL3526963 0.152 0.108 CHEMBL3526244 0.318 0.025 CHEMBL3526620 0.173 0.086 CHEMBL3526754 0.138 0.123 CHEMBL3526766 | CHEMBL3526746 | |
| 0.014 | 0.047 | 0.034 | Beta 1 adrenoreceptor agonist | 0.023 0.015 CHEMBL3526208 0.021 0.018 CHEMBL3526767 0.034 0.006 CHEMBL3526766 | CHEMBL3526766 | |
| 0.04 | 0.074 | 0.053 | Autotaxin inhibitor | 0.053 0.036 CHEMBL3526234 | CHEMBL3526234 | |
| 0.004 | 0.044 | 0.027 | Beta 3 adrenoreceptor agonist | 0.027 0.004 CHEMBL3526766 | CHEMBL3526766 | |
| 0.052 | 0.099 | 0.082 | Beta 2 adrenoreceptor agonist | 0.066 0.027 CHEMBL3526208 0.064 0.034 CHEMBL3526767 0.082 0.008 CHEMBL3526766 | CHEMBL3526766 | |
| 0.146 | 0.194 | 0.251 | ErbB-1 antagonist | 0.177 0.12 CHEMBL3526242 0.162 0.149 CHEMBL3526471 0.251 0.051 CHEMBL3526211 | CHEMBL3526211 | |
| 0.189 | 0.238 | 0.227 | Transcription factor inhibitor | 0.227 0.204 CHEMBL3526767 | CHEMBL3526767 | |
| 0.042 | 0.106 | 0.085 | Phosphodiesterase 4D inhibitor | 0.085 0.044 CHEMBL3526767 0.075 0.051 CHEMBL3526211 | CHEMBL3526767 | |
| 0.024 | 0.09 | 0.046 | Phosphodiesterase 4A inhibitor | 0.046 0.038 CHEMBL3526211 | CHEMBL3526211 | |
| 0.05 | 0.121 | 0.076 | Adenosine A3 receptor antagonist | 0.076 0.049 CHEMBL3526849 0.072 0.055 CHEMBL3542322 | CHEMBL3526849 | |
| 0.035 | 0.107 | 0.066 | Collagenase 3 inhibitor | 0.066 0.035 CHEMBL3526244 | CHEMBL3526244 | |
| 0.029 | 0.104 | 0.078 | Alpha 1 adrenoreceptor agonist | 0.078 0.024 CHEMBL3526767 0.057 0.04 CHEMBL3526766 | CHEMBL3526767 | |
| 0.124 | 0.2 | 0.265 | Vasodilator | 0.259 0.064 CHEMBL3526849 0.249 0.069 CHEMBL3526746 0.265 0.062 CHEMBL3542322 0.18 0.122 CHEMBL3527595 0.222 0.088 CHEMBL3526620 | CHEMBL3542322 | |
| 0.011 | 0.1 | 0.032 | Peroxisome proliferator-activated receptor delta agonist | 0.032 0.025 CHEMBL3526470 | CHEMBL3526470 | |
| 0.151 | 0.241 | 0.226 | Calpain 2 inhibitor | 0.226 0.167 CHEMBL3526243 | CHEMBL3526243 | |
| 0.047 | 0.16 | 0.123 | 5-Lipoxygenase inhibitor | 0.123 0.049 CHEMBL3526244 0.121 0.049 CHEMBL3526470 | CHEMBL3526244 | |
| 0.082 | 0.203 | 0.179 | Pyruvate kinase inhibitor | 0.134 0.131 CHEMBL3526767 0.151 0.114 CHEMBL3526244 0.179 0.094 CHEMBL3526766 | CHEMBL3526766 | |
| 0.034 | 0.156 | 0.155 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.072 0.059 CHEMBL3526243 0.155 0.017 CHEMBL3526244 | CHEMBL3526244 | |
| 0.048 | 0.175 | 0.145 | Gastric antisecretory | 0.129 0.037 CHEMBL3526242 0.145 0.029 CHEMBL3527594 0.089 0.08 CHEMBL3526660 0.094 0.073 CHEMBL3526620 0.086 0.084 CHEMBL3526470 0.119 0.044 CHEMBL3526829 | CHEMBL3527594 | |
| 0.106 | 0.238 | 0.203 | Streptokinase A inhibitor | 0.203 0.131 CHEMBL3526766 | CHEMBL3526766 | |
| 0.061 | 0.203 | 0.086 | Alpha 2d adrenoreceptor antagonist | 0.086 0.081 CHEMBL3526767 | CHEMBL3526767 | |
| 0.024 | 0.169 | 0.171 | NMDA 2B receptor antagonist | 0.171 0.007 CHEMBL3526234 0.104 0.014 CHEMBL3527594 0.101 0.015 CHEMBL3526660 0.08 0.021 CHEMBL3526766 | CHEMBL3526234 | |
| 0.044 | 0.2 | 0.09 | DNA intercalator | 0.09 0.086 CHEMBL3526746 | CHEMBL3526746 | |
| 0.02 | 0.205 | 0.084 | Leukotriene antagonist | 0.058 0.054 CHEMBL3526242 0.074 0.036 CHEMBL3526244 0.084 0.029 CHEMBL3526470 | CHEMBL3526470 | |
| 0.119 | 0.306 | 0.429 | Immunomodulator | 0.403 0.043 CHEMBL3526849 0.2 0.164 CHEMBL3526242 0.359 0.057 CHEMBL3526746 0.429 0.036 CHEMBL3542322 0.324 0.07 CHEMBL3527595 0.229 0.133 CHEMBL3526963 0.284 0.092 CHEMBL3526620 0.212 0.15 CHEMBL3526754 | CHEMBL3542322 | |
| 0.045 | 0.233 | 0.095 | Xanthine oxidase inhibitor | 0.095 0.065 CHEMBL3526746 | CHEMBL3526746 | |
| 0.019 | 0.209 | 0.067 | H+/K+-transporting ATPase inhibitor | 0.067 0.02 CHEMBL3527594 0.054 0.032 CHEMBL3526829 | CHEMBL3527594 | |
| 0.031 | 0.223 | 0.083 | Epidermal growth factor antagonist | 0.083 0.061 CHEMBL3526211 | CHEMBL3526211 | |
| 0.018 | 0.214 | 0.063 | Beta 1 adrenoreceptor antagonist | 0.063 0.033 CHEMBL3526766 | CHEMBL3526766 | |
| 0.02 | 0.223 | 0.072 | Cytokine production stimulant | 0.058 0.015 CHEMBL3526242 0.053 0.023 CHEMBL3527076 0.072 0.006 CHEMBL3527595 0.054 0.021 CHEMBL3526471 0.049 0.03 CHEMBL3526470 0.06 0.013 CHEMBL3526211 | CHEMBL3527595 | |
| 0.065 | 0.271 | 0.216 | Dual specificity phosphatase inhibitor | 0.21 0.05 CHEMBL3526234 0.216 0.047 CHEMBL3526244 | CHEMBL3526244 | |
| 0.018 | 0.233 | 0.057 | Beta 2 adrenoreceptor antagonist | 0.057 0.027 CHEMBL3526766 | CHEMBL3526766 | |
| 0.012 | 0.231 | 0.1 | Adenosine A1 receptor antagonist | 0.079 0.029 CHEMBL3526849 0.1 0.023 CHEMBL3542322 | CHEMBL3542322 | |
| 0.04 | 0.264 | 0.078 | Falcipain 2 inhibitor | 0.078 0.072 CHEMBL3526243 0.076 0.075 CHEMBL3527595 | CHEMBL3526243 | |
| 0.04 | 0.266 | 0.101 | Epidermal growth factor receptor kinase inhibitor | 0.101 0.096 CHEMBL3526211 | CHEMBL3526211 | |
| 0.04 | 0.271 | 0.079 | Falcipain inhibitor | 0.079 0.075 CHEMBL3526243 0.078 0.077 CHEMBL3527595 | CHEMBL3526243 | |
| 0.036 | 0.267 | 0.109 | Tubulin antagonist | 0.104 0.097 CHEMBL3526470 0.109 0.092 CHEMBL3526211 | CHEMBL3526211 | |
| 0.033 | 0.285 | 0.106 | M17 leucyl aminopeptidase inhibitor | 0.106 0.093 CHEMBL3526244 | CHEMBL3526244 | |
| 0.036 | 0.291 | 0.121 | Cyclooxygenase 1 inhibitor | 0.121 0.079 CHEMBL3526470 | CHEMBL3526470 | |
| 0.005 | 0.264 | 0.242 | Cholecystokinin A agonist | 0.214 0.003 CHEMBL3526234 0.242 0.002 CHEMBL3527594 0.234 0.002 CHEMBL3526660 | CHEMBL3527594 | |
| 0.055 | 0.318 | 0.103 | Folate antagonist | 0.103 0.059 CHEMBL3526620 | CHEMBL3526620 | |
| 0.039 | 0.303 | 0.193 | Cytidine deaminase inhibitor | 0.193 0.051 CHEMBL3526849 0.155 0.072 CHEMBL3542322 | CHEMBL3526849 | |
| 0.037 | 0.3 | 0.109 | Estrogen receptor beta antagonist | 0.099 0.067 CHEMBL3526208 0.109 0.048 CHEMBL3526766 | CHEMBL3526766 | |
| 0.083 | 0.355 | 0.314 | Alpha-glucosidase inhibitor | 0.314 0.153 CHEMBL3526746 | CHEMBL3526746 | |
| 0.03 | 0.304 | 0.142 | Sphingomyelinase inhibitor | 0.142 0.028 CHEMBL3526242 | CHEMBL3526242 | |
| 0.046 | 0.326 | 0.28 | Dual specificity phosphatase 3 inhibitor | 0.133 0.113 CHEMBL3526243 0.201 0.06 CHEMBL3526234 0.128 0.118 CHEMBL3527594 0.134 0.112 CHEMBL3526660 0.28 0.033 CHEMBL3526244 | CHEMBL3526244 | |
| 0.038 | 0.318 | 0.076 | MAP kinase kinase 7 inhibitor | 0.076 0.058 CHEMBL3526766 | CHEMBL3526766 | |
| 0.057 | 0.352 | 0.346 | DNA methylase inhibitor | 0.345 0.018 CHEMBL3526849 0.319 0.023 CHEMBL3542322 0.157 0.111 CHEMBL3527595 0.236 0.056 CHEMBL3526244 0.346 0.017 CHEMBL3526620 0.184 0.09 CHEMBL3526470 0.14 0.127 CHEMBL3526754 | CHEMBL3526620 | |
| 0.004 | 0.305 | 0.308 | Cholecystokinin agonist | 0.256 0.003 CHEMBL3526234 0.308 0.003 CHEMBL3527594 0.297 0.003 CHEMBL3526660 | CHEMBL3527594 | |
| 0.034 | 0.338 | 0.09 | Thioredoxin inhibitor | 0.089 0.064 CHEMBL3527595 0.09 0.061 CHEMBL3526620 | CHEMBL3526620 | |
| 0.03 | 0.334 | 0.115 | ErbB-3 antagonist | 0.115 0.032 CHEMBL3526620 | CHEMBL3526620 | |
| 0.052 | 0.358 | 0.305 | DNA methyltransferase I inhibitor | 0.305 0.024 CHEMBL3526849 0.284 0.032 CHEMBL3542322 0.193 0.073 CHEMBL3526244 0.281 0.033 CHEMBL3526620 0.143 0.112 CHEMBL3526470 | CHEMBL3526849 | |
| 0.034 | 0.34 | 0.093 | Bile acid receptor antagonist | 0.087 0.083 CHEMBL3526242 0.093 0.066 CHEMBL3526244 0.089 0.077 CHEMBL3526470 | CHEMBL3526244 | |
| 0.078 | 0.393 | 0.217 | Hypoxia-inducible factor 1 alpha inhibitor | 0.217 0.132 CHEMBL3526849 0.213 0.137 CHEMBL3542322 | CHEMBL3526849 | |
| 0.056 | 0.377 | 0.268 | Hemostatic | 0.268 0.019 CHEMBL3526746 0.236 0.024 CHEMBL3526234 0.174 0.046 CHEMBL3527595 0.151 0.067 CHEMBL3526660 | CHEMBL3526746 | |
| 0.019 | 0.352 | 0.117 | ErbB-2 antagonist | 0.117 0.029 CHEMBL3526211 | CHEMBL3526211 | |
| 0.046 | 0.385 | 0.142 | Neuropeptide Y1 antagonist | 0.121 0.12 CHEMBL3526243 0.142 0.077 CHEMBL3526242 | CHEMBL3526242 | |
| 0.046 | 0.397 | 0.327 | Free radical scavenger | 0.15 0.145 CHEMBL3526849 0.327 0.045 CHEMBL3526746 0.177 0.117 CHEMBL3542322 0.297 0.053 CHEMBL3527595 0.187 0.109 CHEMBL3526963 0.16 0.133 CHEMBL3526754 | CHEMBL3526746 | |
| 0.047 | 0.402 | 0.299 | Beta lactamase inhibitor | 0.299 0.135 CHEMBL3526244 | CHEMBL3526244 | |
| 0.035 | 0.393 | 0.104 | Electron transport complex I inhibitor | 0.104 0.074 CHEMBL3526242 | CHEMBL3526242 | |
| 0.023 | 0.381 | 0.105 | Nitric-oxide synthase inhibitor | 0.105 0.052 CHEMBL3526620 | CHEMBL3526620 | |
| 0.005 | 0.368 | 0.025 | Sodium/glucose cotransporter inhibitor | 0.025 0.019 CHEMBL3526746 0.024 0.022 CHEMBL3527595 | CHEMBL3526746 | |
| 0.035 | 0.4 | 0.115 | Estrogen antagonist | 0.101 0.096 CHEMBL3526208 0.115 0.064 CHEMBL3526766 | CHEMBL3526766 | |
| 0.014 | 0.381 | 0.087 | Inducible nitric-oxide synthase inhibitor | 0.087 0.051 CHEMBL3526620 | CHEMBL3526620 | |
| 0.044 | 0.411 | 0.21 | Nitric oxide antagonist | 0.21 0.064 CHEMBL3526746 0.204 0.066 CHEMBL3527595 | CHEMBL3526746 | |
| 0.005 | 0.375 | 0.05 | Beta tubulin antagonist | 0.05 0.047 CHEMBL3526211 | CHEMBL3526211 | |
| 0.045 | 0.427 | 0.083 | Glutamate release inhibitor | 0.083 0.079 CHEMBL3526242 | CHEMBL3526242 | |
| 0.077 | 0.461 | 0.17 | RNA-directed DNA polymerase inhibitor | 0.168 0.156 CHEMBL3526242 0.17 0.152 CHEMBL3542322 | CHEMBL3542322 | |
| 0.03 | 0.423 | 0.099 | NADH dehydrogenase inhibitor | 0.088 0.059 CHEMBL3526849 0.099 0.045 CHEMBL3542322 | CHEMBL3542322 | |
| 0.008 | 0.415 | 0.063 | Phosphodiesterase VII inhibitor | 0.063 0.042 CHEMBL3526829 | CHEMBL3526829 | |
| 0.049 | 0.456 | 0.121 | DNA repair enzyme inhibitor | 0.121 0.071 CHEMBL3526849 0.112 0.089 CHEMBL3526746 0.116 0.08 CHEMBL3542322 0.108 0.101 CHEMBL3527595 | CHEMBL3526849 | |
| 0.02 | 0.435 | 0.08 | ATPase (Vacuolar H+) inhibitor | 0.08 0.078 CHEMBL3526746 0.08 0.079 CHEMBL3527595 | CHEMBL3527595 | |
| 0.024 | 0.446 | 0.061 | Adenine nucleotide translocase inhibitor | 0.057 0.034 CHEMBL3526849 0.061 0.027 CHEMBL3542322 0.053 0.045 CHEMBL3527594 0.053 0.045 CHEMBL3526660 | CHEMBL3542322 | |
| 0.012 | 0.444 | 0.061 | Epithelial sodium channel blocker | 0.061 0.027 CHEMBL3526242 | CHEMBL3526242 | |
| 0.1 | 0.541 | 0.258 | Caspase 9 stimulant | 0.258 0.243 CHEMBL3526242 | CHEMBL3526242 | |
| 0.019 | 0.46 | 0.064 | Vanilloid 2 antagonist | 0.064 0.019 CHEMBL3526243 0.061 0.021 CHEMBL3526244 | CHEMBL3526243 | |
| 0.034 | 0.475 | 0.079 | D-Ala-D-Ala ligase inhibitor | 0.079 0.072 CHEMBL3526470 | CHEMBL3526470 | |
| 0.029 | 0.474 | 0.175 | DNA polymerase I inhibitor | 0.16 0.044 CHEMBL3526849 0.175 0.037 CHEMBL3542322 | CHEMBL3542322 | |
| 0.014 | 0.465 | 0.057 | Heparanase inhibitor | 0.053 0.037 CHEMBL3526746 0.049 0.047 CHEMBL3527595 0.051 0.042 CHEMBL3526963 0.057 0.029 CHEMBL3526754 | CHEMBL3526754 | |
| 0.025 | 0.476 | 0.096 | Kallikrein 1 inhibitor | 0.096 0.013 CHEMBL3526242 | CHEMBL3526242 | |
| 0.06 | 0.512 | 0.283 | Histamine release inhibitor | 0.283 0.133 CHEMBL3527595 0.223 0.178 CHEMBL3526470 | CHEMBL3527595 | |
| 0.005 | 0.463 | 0.043 | AMPA receptor agonist | 0.033 0.028 CHEMBL3527076 0.032 0.031 CHEMBL3526471 0.043 0.014 CHEMBL3526620 0.036 0.023 CHEMBL3526470 0.032 0.031 CHEMBL3526211 | CHEMBL3526620 | |
| 0.036 | 0.498 | 0.136 | Histone deacetylase SIRT1 inhibitor | 0.136 0.074 CHEMBL3527076 0.111 0.103 CHEMBL3526471 | CHEMBL3527076 | |
| 0.033 | 0.496 | 0.184 | Aldehyde oxidase inhibitor | 0.184 0.114 CHEMBL3526244 | CHEMBL3526244 | |
| 0.077 | 0.542 | 0.334 | Apoptosis agonist | 0.248 0.217 CHEMBL3526469 0.334 0.149 CHEMBL3526746 0.248 0.216 CHEMBL3527595 | CHEMBL3526746 | |
| 0.012 | 0.478 | 0.236 | Alkylator | 0.095 0.094 CHEMBL3526242 0.151 0.046 CHEMBL3527595 0.176 0.034 CHEMBL3526963 0.236 0.018 CHEMBL3526620 0.171 0.037 CHEMBL3526754 | CHEMBL3526620 | |
| 0.014 | 0.481 | 0.062 | Glucose-6-phosphate translocase inhibitor | 0.062 0.022 CHEMBL3527595 | CHEMBL3527595 | |
| 0.011 | 0.479 | 0.241 | Expectorant | 0.118 0.052 CHEMBL3527595 0.166 0.029 CHEMBL3526244 0.241 0.014 CHEMBL3526620 | CHEMBL3526620 | |
| 0.014 | 0.483 | 0.162 | Topoisomerase I inhibitor | 0.146 0.043 CHEMBL3526849 0.162 0.037 CHEMBL3542322 0.088 0.082 CHEMBL3527595 | CHEMBL3542322 | |
| 0.039 | 0.511 | 0.095 | Interleukin 12 antagonist | 0.095 0.063 CHEMBL3527595 | CHEMBL3527595 | |
| 0.003 | 0.479 | 0.025 | Purinergic P2X agonist | 0.024 0.022 CHEMBL3526849 0.025 0.02 CHEMBL3542322 | CHEMBL3542322 | |
| 0.014 | 0.492 | 0.245 | Mucolytic | 0.095 0.085 CHEMBL3526243 0.182 0.018 CHEMBL3526244 0.245 0.007 CHEMBL3526620 0.103 0.073 CHEMBL3526470 | CHEMBL3526620 | |
| 0.027 | 0.513 | 0.152 | Interleukin antagonist | 0.138 0.128 CHEMBL3526243 0.152 0.116 CHEMBL3526766 | CHEMBL3526766 | |
| 0.012 | 0.504 | 0.081 | Thrombin inhibitor | 0.079 0.042 CHEMBL3526242 0.081 0.041 CHEMBL3527594 0.081 0.04 CHEMBL3526660 | CHEMBL3526660 | |
| 0.02 | 0.511 | 0.244 | Thrombolytic | 0.164 0.072 CHEMBL3526243 0.131 0.098 CHEMBL3526242 0.184 0.06 CHEMBL3526746 0.244 0.035 CHEMBL3527595 0.163 0.073 CHEMBL3526963 0.164 0.071 CHEMBL3527594 0.137 0.093 CHEMBL3526660 0.231 0.039 CHEMBL3526244 0.2 0.052 CHEMBL3526620 0.144 0.087 CHEMBL3526470 0.149 0.083 CHEMBL3526754 | CHEMBL3527595 | |
| 0.06 | 0.555 | 0.187 | Death-associated protein kinase 1 inhibitor | 0.187 0.01 CHEMBL3526243 0.179 0.014 CHEMBL3527076 0.126 0.093 CHEMBL3527595 0.134 0.071 CHEMBL3527594 0.134 0.071 CHEMBL3526660 0.186 0.011 CHEMBL3526471 0.171 0.018 CHEMBL3526829 0.171 0.018 CHEMBL3526211 | CHEMBL3526243 | |
| 0.022 | 0.518 | 0.084 | HIV-1 integrase (Overall Integration) inhibitor | 0.084 0.073 CHEMBL3526244 | CHEMBL3526244 | |
| 0.056 | 0.555 | 0.301 | Vasodilator, coronary | 0.301 0.086 CHEMBL3526243 0.277 0.108 CHEMBL3526849 0.27 0.115 CHEMBL3526242 0.244 0.141 CHEMBL3542322 0.272 0.113 CHEMBL3527595 0.295 0.092 CHEMBL3526244 | CHEMBL3526243 | |
| 0.004 | 0.515 | 0.075 | Antineoplastic antibiotic | 0.075 0.061 CHEMBL3527595 | CHEMBL3527595 | |
| 0.022 | 0.534 | 0.464 | Angiogenesis stimulant | 0.147 0.124 CHEMBL3526243 0.233 0.078 CHEMBL3526849 0.401 0.021 CHEMBL3526746 0.249 0.07 CHEMBL3542322 0.225 0.082 CHEMBL3526234 0.464 0.014 CHEMBL3527595 0.267 0.062 CHEMBL3526963 0.282 0.056 CHEMBL3527594 0.288 0.054 CHEMBL3526660 0.154 0.12 CHEMBL3526244 0.253 0.069 CHEMBL3526754 | CHEMBL3527595 | |
| 0.024 | 0.537 | 0.139 | Amylase inhibitor | 0.139 0.07 CHEMBL3527595 | CHEMBL3527595 | |
| 0.004 | 0.523 | 0.018 | Adenosine A3 receptor agonist | 0.017 0.012 CHEMBL3526849 0.018 0.011 CHEMBL3542322 | CHEMBL3542322 | |
| 0.017 | 0.547 | 0.14 | Histone deacetylase class III inhibitor | 0.098 0.092 CHEMBL3527076 0.126 0.065 CHEMBL3526620 0.14 0.052 CHEMBL3526470 | CHEMBL3526470 | |
| 0.022 | 0.559 | 0.145 | Antimitotic | 0.145 0.126 CHEMBL3526620 | CHEMBL3526620 | |
| 0.005 | 0.556 | 0.389 | Angiotensin-converting enzyme inhibitor | 0.389 0.003 CHEMBL3526243 0.123 0.006 CHEMBL3527076 0.078 0.015 CHEMBL3527595 0.05 0.047 CHEMBL3526963 0.214 0.004 CHEMBL3526244 0.106 0.008 CHEMBL3526471 0.179 0.004 CHEMBL3526620 0.074 0.017 CHEMBL3526470 0.053 0.042 CHEMBL3526829 0.05 0.047 CHEMBL3526211 | CHEMBL3526243 | |
| 0.027 | 0.596 | 0.427 | Tumour necrosis factor alpha release inhibitor | 0.331 0.043 CHEMBL3526243 0.157 0.15 CHEMBL3526746 0.287 0.058 CHEMBL3527076 0.427 0.023 CHEMBL3527595 0.169 0.135 CHEMBL3527594 0.215 0.096 CHEMBL3526660 0.332 0.043 CHEMBL3526471 0.243 0.078 CHEMBL3526829 0.294 0.056 CHEMBL3526211 | CHEMBL3527595 | |
| 0.066 | 0.637 | 0.186 | Tyrosine 3 hydroxylase inhibitor | 0.186 0.162 CHEMBL3527076 | CHEMBL3527076 | |
| 0.072 | 0.65 | 0.12 | CC chemokine 6 receptor antagonist | 0.12 0.116 CHEMBL3526746 | CHEMBL3526746 | |
| 0.036 | 0.619 | 0.566 | Antibacterial | 0.386 0.083 CHEMBL3526849 0.521 0.035 CHEMBL3526746 0.436 0.062 CHEMBL3542322 0.566 0.025 CHEMBL3527595 0.421 0.067 CHEMBL3526963 0.37 0.091 CHEMBL3526754 | CHEMBL3527595 | |
| 0.026 | 0.617 | 0.211 | Platelet adhesion inhibitor | 0.182 0.081 CHEMBL3526849 0.185 0.079 CHEMBL3526746 0.183 0.081 CHEMBL3542322 0.211 0.066 CHEMBL3527595 | CHEMBL3527595 | |
| 0.054 | 0.647 | 0.205 | 5 Hydroxytryptamine release stimulant | 0.205 0.117 CHEMBL3526242 | CHEMBL3526242 | |
| 0.005 | 0.602 | 0.069 | Metalloproteinase-9 inhibitor | 0.069 0.058 CHEMBL3526244 | CHEMBL3526244 | |
| 0.028 | 0.626 | 0.088 | Transcription factor NF kappa B stimulant | 0.079 0.071 CHEMBL3526746 0.088 0.054 CHEMBL3527595 | CHEMBL3527595 | |
| 0.003 | 0.601 | 0.153 | Cholecystokinin A antagonist | 0.11 0.007 CHEMBL3526234 0.153 0.005 CHEMBL3527594 0.145 0.005 CHEMBL3526660 | CHEMBL3527594 | |
| 0.003 | 0.602 | 0.093 | Cholecystokinin B antagonist | 0.056 0.009 CHEMBL3526234 0.093 0.005 CHEMBL3527594 0.079 0.005 CHEMBL3526660 | CHEMBL3527594 | |
| 0.009 | 0.61 | 0.455 | Cholecystokinin B agonist | 0.402 0.003 CHEMBL3526234 0.455 0.002 CHEMBL3527594 0.455 0.002 CHEMBL3526660 | CHEMBL3526660 | |
| 0.021 | 0.622 | 0.106 | Nav1.4 sodium channel blocker | 0.106 0.068 CHEMBL3527076 0.098 0.078 CHEMBL3527594 0.098 0.078 CHEMBL3526660 | CHEMBL3527076 | |
| 0.013 | 0.615 | 0.084 | Opioid antagonist | 0.084 0.063 CHEMBL3527076 | CHEMBL3527076 | |
| 0.004 | 0.61 | 0.014 | Adenosine A2b receptor agonist | 0.013 0.012 CHEMBL3526849 0.014 0.011 CHEMBL3542322 | CHEMBL3542322 | |
| 0.022 | 0.629 | 0.1 | Toll-Like receptor 4 antagonist | 0.091 0.086 CHEMBL3526746 0.1 0.07 CHEMBL3527595 | CHEMBL3527595 | |
| 0.022 | 0.64 | 0.124 | Cyclooxygenase 3 inhibitor | 0.124 0.073 CHEMBL3527595 | CHEMBL3527595 | |
| 0.003 | 0.625 | 0.123 | Cholecystokinin antagonist | 0.075 0.013 CHEMBL3526234 0.123 0.006 CHEMBL3527594 0.106 0.008 CHEMBL3526660 | CHEMBL3527594 | |
| 0.002 | 0.63 | 0.108 | Angiotensin-converting enzyme 2 inhibitor | 0.108 0.003 CHEMBL3526243 0.04 0.004 CHEMBL3526244 | CHEMBL3526243 | |
| 0.018 | 0.646 | 0.234 | DNA synthesis inhibitor | 0.216 0.1 CHEMBL3526849 0.234 0.078 CHEMBL3542322 0.183 0.149 CHEMBL3526963 | CHEMBL3542322 | |
| 0.01 | 0.638 | 0.054 | Antibiotic Aminoglycoside-like | 0.05 0.014 CHEMBL3526746 0.054 0.011 CHEMBL3527595 | CHEMBL3527595 | |
| 0.004 | 0.645 | 0.064 | Prostaglandin EP2 antagonist | 0.064 0.037 CHEMBL3526242 | CHEMBL3526242 | |
| 0.023 | 0.667 | 0.054 | Lipocortins synthesis agonist | 0.054 0.051 CHEMBL3527595 | CHEMBL3527595 | |
| 0.002 | 0.657 | 0.356 | Neutral endopeptidase inhibitor | 0.356 0.002 CHEMBL3526243 0.137 0.004 CHEMBL3527076 0.047 0.008 CHEMBL3527595 0.176 0.004 CHEMBL3526244 0.127 0.004 CHEMBL3526471 0.14 0.004 CHEMBL3526620 0.03 0.012 CHEMBL3526470 | CHEMBL3526243 | |
| 0.027 | 0.696 | 0.204 | Toll-Like receptor agonist | 0.204 0.196 CHEMBL3526242 | CHEMBL3526242 | |
| 0.004 | 0.672 | 0.038 | Kinesin-like protein 1 inhibitor | 0.038 0.024 CHEMBL3526620 | CHEMBL3526620 | |
| 0.004 | 0.672 | 0.038 | Kinesin antagonist | 0.038 0.024 CHEMBL3526620 | CHEMBL3526620 | |
| 0.011 | 0.687 | 0.058 | Trypsin inhibitor | 0.058 0.052 CHEMBL3526242 | CHEMBL3526242 | |
| 0.004 | 0.681 | 0.1 | Glutamate decarboxylase inhibitor | 0.08 0.044 CHEMBL3526244 0.1 0.03 CHEMBL3526620 | CHEMBL3526620 | |
| 0.004 | 0.691 | 0.04 | Macrophage elastase inhibitor | 0.04 0.033 CHEMBL3526244 | CHEMBL3526244 | |
| 0.059 | 0.748 | 0.325 | Interleukin 2 agonist | 0.301 0.073 CHEMBL3526746 0.325 0.058 CHEMBL3527595 0.23 0.143 CHEMBL3526963 0.227 0.147 CHEMBL3526620 0.206 0.178 CHEMBL3526754 | CHEMBL3527595 | |
| 0.003 | 0.694 | 0.028 | 1,3-Beta-glucan synthase inhibitor | 0.028 0.02 CHEMBL3527594 0.028 0.02 CHEMBL3526660 | CHEMBL3526660 | |
| 0.012 | 0.705 | 0.129 | Multidrug resistance-associated protein 1 inhibitor | 0.104 0.072 CHEMBL3526234 0.129 0.039 CHEMBL3527594 0.127 0.041 CHEMBL3526660 | CHEMBL3527594 | |
| 0.005 | 0.711 | 0.142 | Analgesic, opioid | 0.142 0.016 CHEMBL3527076 0.08 0.047 CHEMBL3527595 0.103 0.03 CHEMBL3526471 0.078 0.05 CHEMBL3526620 | CHEMBL3527076 | |
| 0.007 | 0.721 | 0.062 | Protein 50S ribosomal subunit inhibitor | 0.055 0.035 CHEMBL3526746 0.062 0.029 CHEMBL3527595 | CHEMBL3527595 | |
| 0.009 | 0.726 | 0.332 | Anticoagulant | 0.169 0.067 CHEMBL3526242 0.219 0.047 CHEMBL3526234 0.179 0.062 CHEMBL3527595 0.322 0.025 CHEMBL3527594 0.332 0.024 CHEMBL3526660 | CHEMBL3526660 | |
| 0.005 | 0.728 | 0.034 | p53 inhibitor | 0.034 0.026 CHEMBL3526211 | CHEMBL3526211 | |
| 0.013 | 0.74 | 0.145 | Cell wall synthesis inhibitor | 0.141 0.074 CHEMBL3527595 0.145 0.07 CHEMBL3526660 | CHEMBL3526660 | |
| 0.009 | 0.742 | 0.384 | Immunostimulant | 0.198 0.121 CHEMBL3526849 0.183 0.131 CHEMBL3526746 0.257 0.093 CHEMBL3542322 0.384 0.054 CHEMBL3527595 0.381 0.055 CHEMBL3526963 0.157 0.149 CHEMBL3527594 0.281 0.084 CHEMBL3526620 0.332 0.07 CHEMBL3526754 | CHEMBL3527595 | |
| 0.003 | 0.739 | 0.014 | S-adenosyl-L-homocysteine hydrolase inhibitor | 0.014 0.012 CHEMBL3526849 0.014 0.011 CHEMBL3542322 | CHEMBL3542322 | |
| 0.012 | 0.751 | 0.048 | Factor IXa inhibitor | 0.048 0.04 CHEMBL3527595 | CHEMBL3527595 | |
| 0.014 | 0.76 | 0.451 | Antithrombotic | 0.261 0.118 CHEMBL3526746 0.451 0.038 CHEMBL3527595 0.217 0.157 CHEMBL3527594 0.24 0.135 CHEMBL3526620 | CHEMBL3527595 | |
| 0.003 | 0.755 | 0.03 | Adenosine A1 receptor agonist | 0.03 0.012 CHEMBL3526849 0.03 0.011 CHEMBL3542322 | CHEMBL3542322 | |
| 0.007 | 0.762 | 0.091 | Aminoacyl-tRNA synthetase inhibitor | 0.086 0.065 CHEMBL3526849 0.091 0.057 CHEMBL3542322 | CHEMBL3542322 | |
| 0.004 | 0.763 | 0.141 | Endothelin-converting enzyme inhibitor | 0.141 0.01 CHEMBL3526243 0.106 0.014 CHEMBL3526244 | CHEMBL3526243 | |
| 0.004 | 0.768 | 0.23 | Selectin antagonist | 0.193 0.012 CHEMBL3526746 0.23 0.009 CHEMBL3527595 0.1 0.028 CHEMBL3526963 0.09 0.031 CHEMBL3526754 | CHEMBL3527595 | |
| 0.008 | 0.788 | 0.259 | Chelator | 0.183 0.028 CHEMBL3526244 0.259 0.015 CHEMBL3526620 | CHEMBL3526620 | |
| 0.023 | 0.804 | 0.435 | Antiinflammatory | 0.435 0.118 CHEMBL3526746 0.319 0.198 CHEMBL3527595 | CHEMBL3526746 | |
| 0.057 | 0.843 | 0.315 | Peptidyltransferase inhibitor | 0.274 0.036 CHEMBL3526849 0.284 0.031 CHEMBL3526746 0.287 0.03 CHEMBL3542322 0.315 0.02 CHEMBL3527595 0.219 0.077 CHEMBL3526963 0.204 0.094 CHEMBL3526754 | CHEMBL3527595 | |
| 0.006 | 0.801 | 0.087 | Protease inhibitor | 0.087 0.078 CHEMBL3526242 | CHEMBL3526242 | |
| 0.015 | 0.826 | 0.313 | Immunosuppressant | 0.238 0.158 CHEMBL3526746 0.313 0.107 CHEMBL3527595 0.231 0.165 CHEMBL3527594 0.239 0.157 CHEMBL3526829 | CHEMBL3527595 | |
| 0.004 | 0.828 | 0.104 | Aminopeptidase N inhibitor | 0.104 0.012 CHEMBL3526620 | CHEMBL3526620 | |
| 0.008 | 0.847 | 0.1 | Aminopeptidase B inhibitor | 0.1 0.065 CHEMBL3526620 | CHEMBL3526620 | |
| 0.005 | 0.85 | 0.134 | Aminopeptidase microsomal inhibitor | 0.134 0.01 CHEMBL3526620 | CHEMBL3526620 | |
| 0.011 | 0.86 | 0.345 | Analgesic | 0.345 0.111 CHEMBL3527076 0.293 0.147 CHEMBL3526471 0.27 0.165 CHEMBL3526620 | CHEMBL3527076 | |
| 0.003 | 0.854 | 0.046 | Collagenase inhibitor | 0.046 0.041 CHEMBL3526243 | CHEMBL3526243 | |
| 0.003 | 0.854 | 0.022 | Protein 30S ribosomal subunit inhibitor | 0.022 0.019 CHEMBL3527595 | CHEMBL3527595 | |
| 0.002 | 0.858 | 0.021 | Estrone sulfatase inhibitor | 0.021 0.016 CHEMBL3526234 0.02 0.017 CHEMBL3527594 0.02 0.016 CHEMBL3526660 | CHEMBL3526234 | |
| 0.007 | 0.872 | 0.099 | Cell adhesion inhibitor | 0.099 0.091 CHEMBL3527595 | CHEMBL3527595 | |
| 0.005 | 0.87 | 0.156 | Platelet antagonist | 0.156 0.138 CHEMBL3526620 | CHEMBL3526620 | |
| 0.003 | 0.907 | 0.181 | Diuretic | 0.181 0.053 CHEMBL3527594 0.115 0.11 CHEMBL3526660 | CHEMBL3527594 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |