| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.963 | 0.004 | 0.965 | Apoptosis agonist | 0.963 0.004 CHEMBL3542195 0.944 0.004 CHEMBL3542275 0.965 0.004 CHEMBL3542345 0.96 0.004 CHEMBL3542255 0.96 0.004 CHEMBL3542317 0.954 0.004 CHEMBL3542274 | CHEMBL3542345 | |
| 0.947 | 0.003 | 0.977 | Transcription factor NF kappa B inhibitor | 0.936 0.004 CHEMBL3542195 0.977 0.002 CHEMBL3542275 0.847 0.01 CHEMBL3542345 0.812 0.012 CHEMBL3542255 0.817 0.012 CHEMBL3542317 0.897 0.006 CHEMBL3542274 | CHEMBL3542275 | |
| 0.944 | 0.005 | 0.945 | Antiinflammatory | 0.942 0.005 CHEMBL3542195 0.945 0.005 CHEMBL3542275 0.932 0.005 CHEMBL3542345 0.927 0.005 CHEMBL3542255 0.922 0.005 CHEMBL3542317 0.925 0.005 CHEMBL3542274 | CHEMBL3542275 | |
| 0.89 | 0.002 | 0.891 | Angiogenesis stimulant | 0.891 0.002 CHEMBL3542195 0.715 0.004 CHEMBL3542275 0.881 0.002 CHEMBL3542345 0.866 0.003 CHEMBL3542255 0.868 0.003 CHEMBL3542317 0.862 0.003 CHEMBL3542274 | CHEMBL3542195 | |
| 0.875 | 0.003 | 0.88 | Nitric oxide antagonist | 0.875 0.003 CHEMBL3542195 0.88 0.003 CHEMBL3542275 0.859 0.004 CHEMBL3542345 0.872 0.003 CHEMBL3542255 0.848 0.004 CHEMBL3542317 0.831 0.004 CHEMBL3542274 | CHEMBL3542275 | |
| 0.816 | 0.003 | 0.816 | Hepatoprotectant | 0.813 0.003 CHEMBL3542195 0.8 0.003 CHEMBL3542275 0.8 0.003 CHEMBL3542345 0.755 0.003 CHEMBL3542255 0.754 0.003 CHEMBL3542317 0.773 0.003 CHEMBL3542274 | ||
| 0.817 | 0.009 | 0.919 | Caspase 9 stimulant | 0.823 0.008 CHEMBL3542195 0.919 0.002 CHEMBL3542275 0.663 0.028 CHEMBL3542345 0.516 0.054 CHEMBL3542255 0.363 0.136 CHEMBL3542317 0.564 0.042 CHEMBL3542274 | CHEMBL3542275 | |
| 0.799 | 0.004 | 0.799 | Apoptosis antagonist | 0.793 0.004 CHEMBL3542195 0.786 0.004 CHEMBL3542275 0.759 0.004 CHEMBL3542345 0.724 0.004 CHEMBL3542255 0.738 0.004 CHEMBL3542317 0.735 0.004 CHEMBL3542274 | ||
| 0.763 | 0.009 | 0.841 | Cyclophilin D inhibitor | 0.732 0.011 CHEMBL3542195 0.841 0.005 CHEMBL3542275 0.613 0.025 CHEMBL3542345 0.53 0.042 CHEMBL3542255 0.576 0.032 CHEMBL3542317 0.624 0.023 CHEMBL3542274 | CHEMBL3542275 | |
| 0.713 | 0.008 | 0.713 | Antibacterial | 0.679 0.01 CHEMBL3542195 0.665 0.012 CHEMBL3542275 0.408 0.073 CHEMBL3542345 0.409 0.073 CHEMBL3542255 0.335 0.111 CHEMBL3542317 0.489 0.044 CHEMBL3542274 | ||
| 0.669 | 0.01 | 0.828 | Immunostimulant | 0.623 0.014 CHEMBL3542195 0.828 0.004 CHEMBL3542275 0.425 0.043 CHEMBL3542345 0.382 0.055 CHEMBL3542255 0.339 0.068 CHEMBL3542317 0.424 0.043 CHEMBL3542274 | CHEMBL3542275 | |
| 0.654 | 0.005 | 0.654 | Tumour necrosis factor alpha release inhibitor | 0.645 0.005 CHEMBL3542195 0.507 0.013 CHEMBL3542275 0.572 0.009 CHEMBL3542345 0.48 0.016 CHEMBL3542255 0.496 0.014 CHEMBL3542317 0.525 0.012 CHEMBL3542274 | ||
| 0.646 | 0.006 | 0.726 | Hypoglycemic | 0.606 0.008 CHEMBL3542195 0.726 0.005 CHEMBL3542275 0.44 0.022 CHEMBL3542345 0.362 0.035 CHEMBL3542255 0.296 0.054 CHEMBL3542317 0.488 0.016 CHEMBL3542274 | CHEMBL3542275 | |
| 0.6 | 0.013 | 0.6 | Immunosuppressant | 0.583 0.015 CHEMBL3542195 0.558 0.019 CHEMBL3542275 0.53 0.025 CHEMBL3542345 0.505 0.032 CHEMBL3542255 0.534 0.024 CHEMBL3542317 0.512 0.03 CHEMBL3542274 | ||
| 0.593 | 0.012 | 0.593 | Immunomodulator | 0.55 0.017 CHEMBL3542195 0.352 0.059 CHEMBL3542275 0.421 0.038 CHEMBL3542345 0.339 0.064 CHEMBL3542255 0.339 0.063 CHEMBL3542317 0.351 0.059 CHEMBL3542274 | ||
| 0.587 | 0.012 | 0.732 | Antioxidant | 0.549 0.015 CHEMBL3542195 0.732 0.005 CHEMBL3542275 0.332 0.051 CHEMBL3542345 0.292 0.065 CHEMBL3542255 0.282 0.069 CHEMBL3542317 0.358 0.044 CHEMBL3542274 | CHEMBL3542275 | |
| 0.57 | 0.003 | 0.72 | Interferon gamma antagonist | 0.564 0.003 CHEMBL3542195 0.72 0.001 CHEMBL3542275 0.47 0.007 CHEMBL3542345 0.493 0.006 CHEMBL3542255 0.496 0.006 CHEMBL3542317 0.534 0.004 CHEMBL3542274 | CHEMBL3542275 | |
| 0.569 | 0.023 | 0.716 | Cholesterol antagonist | 0.448 0.041 CHEMBL3542195 0.716 0.007 CHEMBL3542275 0.242 0.131 CHEMBL3542274 | CHEMBL3542275 | |
| 0.542 | 0.015 | 0.68 | Caspase 3 stimulant | 0.522 0.017 CHEMBL3542195 0.68 0.006 CHEMBL3542275 0.45 0.029 CHEMBL3542345 0.371 0.053 CHEMBL3542255 0.419 0.039 CHEMBL3542317 0.458 0.027 CHEMBL3542274 | CHEMBL3542275 | |
| 0.52 | 0.004 | 0.52 | Cell adhesion inhibitor | 0.499 0.004 CHEMBL3542195 0.24 0.016 CHEMBL3542275 0.37 0.006 CHEMBL3542345 0.324 0.009 CHEMBL3542255 0.33 0.008 CHEMBL3542317 0.342 0.008 CHEMBL3542274 | ||
| 0.464 | 0.016 | 0.464 | DNA synthesis inhibitor | 0.439 0.018 CHEMBL3542195 0.353 0.03 CHEMBL3542275 0.254 0.064 CHEMBL3542345 0.254 0.064 CHEMBL3542255 0.223 0.091 CHEMBL3542317 0.296 0.045 CHEMBL3542274 | ||
| 0.441 | 0.004 | 0.836 | AMP-activated protein kinase stimulant | 0.343 0.004 CHEMBL3542195 0.836 0.001 CHEMBL3542275 0.216 0.009 CHEMBL3542345 0.155 0.025 CHEMBL3542255 0.104 0.066 CHEMBL3542317 0.336 0.004 CHEMBL3542274 | CHEMBL3542275 | |
| 0.438 | 0.003 | 0.447 | Beta amyloid protein antagonist | 0.447 0.003 CHEMBL3542195 0.234 0.01 CHEMBL3542275 0.324 0.005 CHEMBL3542345 0.224 0.011 CHEMBL3542255 0.177 0.025 CHEMBL3542317 0.264 0.008 CHEMBL3542274 | CHEMBL3542195 | |
| 0.448 | 0.038 | 0.845 | Antithrombotic | 0.366 0.059 CHEMBL3542195 0.845 0.004 CHEMBL3542275 | CHEMBL3542275 | |
| 0.427 | 0.025 | 0.53 | Free radical scavenger | 0.382 0.032 CHEMBL3542195 0.53 0.013 CHEMBL3542275 0.167 0.127 CHEMBL3542345 0.197 0.1 CHEMBL3542274 | CHEMBL3542275 | |
| 0.384 | 0.013 | 0.56 | Melanin inhibitor | 0.369 0.014 CHEMBL3542195 0.56 0.005 CHEMBL3542275 0.167 0.062 CHEMBL3542345 0.164 0.065 CHEMBL3542255 0.155 0.075 CHEMBL3542317 0.184 0.049 CHEMBL3542274 | CHEMBL3542275 | |
| 0.394 | 0.047 | 0.876 | 5 Hydroxytryptamine release stimulant | 0.268 0.081 CHEMBL3542195 0.876 0.002 CHEMBL3542275 | CHEMBL3542275 | |
| 0.36 | 0.041 | 0.433 | Interleukin 2 agonist | 0.335 0.052 CHEMBL3542195 0.433 0.019 CHEMBL3542275 0.197 0.194 CHEMBL3542345 0.22 0.157 CHEMBL3542255 0.219 0.158 CHEMBL3542274 | CHEMBL3542275 | |
| 0.325 | 0.008 | 0.332 | Antineoplastic antibiotic | 0.332 0.008 CHEMBL3542195 0.309 0.009 CHEMBL3542275 0.169 0.027 CHEMBL3542345 0.174 0.026 CHEMBL3542255 0.177 0.025 CHEMBL3542317 0.163 0.028 CHEMBL3542274 | CHEMBL3542195 | |
| 0.32 | 0.005 | 0.35 | Selectin antagonist | 0.268 0.007 CHEMBL3542195 0.35 0.004 CHEMBL3542275 | CHEMBL3542275 | |
| 0.325 | 0.017 | 0.428 | Lipocortins synthesis antagonist | 0.343 0.014 CHEMBL3542195 0.296 0.022 CHEMBL3542275 0.414 0.008 CHEMBL3542345 0.428 0.007 CHEMBL3542255 0.378 0.01 CHEMBL3542317 0.415 0.008 CHEMBL3542274 | CHEMBL3542255 | |
| 0.304 | 0.004 | 0.371 | Transcription factor NF kappa B stimulant | 0.288 0.004 CHEMBL3542195 0.371 0.003 CHEMBL3542275 0.236 0.006 CHEMBL3542345 0.197 0.009 CHEMBL3542255 0.179 0.011 CHEMBL3542317 0.259 0.005 CHEMBL3542274 | CHEMBL3542275 | |
| 0.312 | 0.017 | 0.474 | Protein-tyrosine phosphatase inhibitor | 0.328 0.015 CHEMBL3542195 0.439 0.006 CHEMBL3542275 0.449 0.006 CHEMBL3542345 0.424 0.007 CHEMBL3542255 0.346 0.013 CHEMBL3542317 0.474 0.005 CHEMBL3542274 | CHEMBL3542274 | |
| 0.312 | 0.02 | 0.327 | Peptidyltransferase inhibitor | 0.327 0.017 CHEMBL3542195 0.325 0.017 CHEMBL3542275 | CHEMBL3542195 | |
| 0.301 | 0.034 | 0.424 | Platelet adhesion inhibitor | 0.245 0.051 CHEMBL3542195 0.424 0.009 CHEMBL3542275 0.132 0.129 CHEMBL3542274 | CHEMBL3542275 | |
| 0.278 | 0.013 | 0.451 | Protein-tyrosine phosphatase 1B inhibitor | 0.299 0.011 CHEMBL3542195 0.451 0.005 CHEMBL3542275 0.422 0.005 CHEMBL3542345 0.389 0.005 CHEMBL3542255 0.321 0.009 CHEMBL3542317 0.448 0.005 CHEMBL3542274 | CHEMBL3542275 | |
| 0.261 | 0.021 | 0.387 | Interleukin 6 antagonist | 0.282 0.018 CHEMBL3542195 0.387 0.008 CHEMBL3542275 0.156 0.08 CHEMBL3542345 0.143 0.101 CHEMBL3542274 | CHEMBL3542275 | |
| 0.251 | 0.013 | 0.628 | Expectorant | 0.247 0.013 CHEMBL3542195 0.628 0.003 CHEMBL3542275 0.093 0.077 CHEMBL3542345 0.143 0.038 CHEMBL3542274 | CHEMBL3542275 | |
| 0.284 | 0.054 | 0.316 | Hypolipemic | 0.281 0.055 CHEMBL3542195 0.316 0.044 CHEMBL3542275 0.29 0.052 CHEMBL3542345 0.171 0.117 CHEMBL3542255 0.29 0.052 CHEMBL3542274 | CHEMBL3542275 | |
| 0.249 | 0.02 | 0.55 | Insulin secretagoues | 0.222 0.026 CHEMBL3542195 0.55 0.004 CHEMBL3542275 0.15 0.075 CHEMBL3542345 0.201 0.035 CHEMBL3542274 | CHEMBL3542275 | |
| 0.25 | 0.026 | 0.431 | Protein kinase stimulant | 0.253 0.026 CHEMBL3542195 0.431 0.006 CHEMBL3542275 0.119 0.093 CHEMBL3542345 0.108 0.107 CHEMBL3542255 0.159 0.062 CHEMBL3542274 | CHEMBL3542275 | |
| 0.225 | 0.021 | 0.29 | DNA polymerase I inhibitor | 0.211 0.025 CHEMBL3542195 0.29 0.012 CHEMBL3542275 0.252 0.017 CHEMBL3542345 0.194 0.03 CHEMBL3542255 0.179 0.035 CHEMBL3542317 0.253 0.016 CHEMBL3542274 | CHEMBL3542275 | |
| 0.205 | 0.002 | 0.374 | Na+ K+ transporting ATPase inhibitor | 0.202 0.002 CHEMBL3542195 0.374 0.001 CHEMBL3542275 0.142 0.008 CHEMBL3542345 0.143 0.007 CHEMBL3542255 0.118 0.018 CHEMBL3542317 0.136 0.009 CHEMBL3542274 | CHEMBL3542275 | |
| 0.219 | 0.035 | 0.427 | Lipid peroxidase inhibitor | 0.201 0.041 CHEMBL3542195 0.427 0.008 CHEMBL3542275 0.122 0.091 CHEMBL3542345 0.109 0.106 CHEMBL3542317 0.142 0.074 CHEMBL3542274 | CHEMBL3542275 | |
| 0.159 | 0.013 | 0.202 | CC chemokine 6 receptor antagonist | 0.161 0.012 CHEMBL3542195 0.202 0.004 CHEMBL3542275 0.152 0.02 CHEMBL3542345 0.141 0.037 CHEMBL3542255 0.151 0.021 CHEMBL3542317 0.154 0.017 CHEMBL3542274 | CHEMBL3542275 | |
| 0.172 | 0.034 | 0.196 | Topoisomerase I inhibitor | 0.153 0.04 CHEMBL3542195 0.196 0.027 CHEMBL3542275 | CHEMBL3542275 | |
| 0.145 | 0.012 | 0.2 | Estrogen agonist | 0.163 0.01 CHEMBL3542195 0.144 0.012 CHEMBL3542275 0.2 0.008 CHEMBL3542345 0.19 0.009 CHEMBL3542255 0.159 0.01 CHEMBL3542317 0.145 0.012 CHEMBL3542274 | CHEMBL3542345 | |
| 0.118 | 0.01 | 0.12 | Protein 50S ribosomal subunit inhibitor | 0.12 0.009 CHEMBL3542195 0.111 0.011 CHEMBL3542275 | CHEMBL3542195 | |
| 0.273 | 0.174 | 0.839 | Alpha-glucosidase inhibitor | 0.233 0.198 CHEMBL3542195 0.839 0.013 CHEMBL3542275 | CHEMBL3542275 | |
| 0.1 | 0.007 | 0.138 | Heme oxygenase stimulant | 0.105 0.006 CHEMBL3542195 0.122 0.004 CHEMBL3542275 0.128 0.004 CHEMBL3542345 0.127 0.004 CHEMBL3542255 0.125 0.004 CHEMBL3542317 0.138 0.003 CHEMBL3542274 | CHEMBL3542274 | |
| 0.122 | 0.029 | 0.216 | Topoisomerase II alpha inhibitor | 0.133 0.027 CHEMBL3542195 0.216 0.013 CHEMBL3542275 | CHEMBL3542275 | |
| 0.143 | 0.055 | 0.52 | Cyclooxygenase 3 inhibitor | 0.148 0.05 CHEMBL3542195 0.52 0.003 CHEMBL3542275 | CHEMBL3542275 | |
| 0.094 | 0.009 | 0.264 | Mineralocorticoid receptor antagonist | 0.113 0.007 CHEMBL3542195 0.236 0.004 CHEMBL3542345 0.264 0.004 CHEMBL3542255 0.244 0.004 CHEMBL3542317 0.206 0.004 CHEMBL3542274 | CHEMBL3542255 | |
| 0.156 | 0.073 | 0.318 | Diuretic | 0.22 0.037 CHEMBL3542195 0.318 0.02 CHEMBL3542275 0.177 0.055 CHEMBL3542345 0.179 0.054 CHEMBL3542255 0.308 0.021 CHEMBL3542274 | CHEMBL3542275 | |
| 0.188 | 0.108 | 0.219 | Antiamyloidogenic | 0.219 0.087 CHEMBL3542195 | CHEMBL3542195 | |
| 0.134 | 0.056 | 0.136 | Alkylator | 0.136 0.055 CHEMBL3542195 0.099 0.089 CHEMBL3542275 | CHEMBL3542195 | |
| 0.104 | 0.029 | 0.147 | Glycine receptor antagonist | 0.112 0.023 CHEMBL3542195 0.147 0.008 CHEMBL3542275 | CHEMBL3542275 | |
| 0.079 | 0.004 | 0.082 | Antibiotic Aminoglycoside-like | 0.068 0.006 CHEMBL3542195 0.082 0.004 CHEMBL3542275 | CHEMBL3542275 | |
| 0.228 | 0.153 | 0.36 | Sodium/bile acid cotransporter inhibitor | 0.261 0.116 CHEMBL3542195 0.316 0.065 CHEMBL3542275 0.354 0.037 CHEMBL3542345 0.35 0.039 CHEMBL3542255 0.236 0.144 CHEMBL3542317 0.36 0.034 CHEMBL3542274 | CHEMBL3542274 | |
| 0.126 | 0.06 | 0.298 | Cholesterol synthesis inhibitor | 0.179 0.032 CHEMBL3542195 0.22 0.022 CHEMBL3542275 0.275 0.014 CHEMBL3542345 0.263 0.016 CHEMBL3542255 0.156 0.041 CHEMBL3542317 0.298 0.012 CHEMBL3542274 | CHEMBL3542274 | |
| 0.079 | 0.014 | 0.1 | Lipocortins synthesis agonist | 0.081 0.013 CHEMBL3542195 0.087 0.01 CHEMBL3542275 0.086 0.01 CHEMBL3542345 0.09 0.009 CHEMBL3542255 0.1 0.005 CHEMBL3542317 0.084 0.011 CHEMBL3542274 | CHEMBL3542317 | |
| 0.134 | 0.072 | 0.609 | Amylase inhibitor | 0.609 0.004 CHEMBL3542275 | CHEMBL3542275 | |
| 0.145 | 0.085 | 0.22 | Thrombolytic | 0.14 0.089 CHEMBL3542195 0.22 0.043 CHEMBL3542275 | CHEMBL3542275 | |
| 0.121 | 0.066 | 0.237 | Topoisomerase II inhibitor | 0.123 0.064 CHEMBL3542195 0.237 0.026 CHEMBL3542275 | CHEMBL3542275 | |
| 0.138 | 0.084 | 0.189 | Adenylate cyclase stimulant | 0.123 0.119 CHEMBL3542195 0.189 0.019 CHEMBL3542275 0.159 0.049 CHEMBL3542345 0.15 0.063 CHEMBL3542255 0.143 0.075 CHEMBL3542274 | CHEMBL3542275 | |
| 0.06 | 0.006 | 0.063 | Protein 30S ribosomal subunit inhibitor | 0.043 0.009 CHEMBL3542195 0.063 0.005 CHEMBL3542275 | CHEMBL3542275 | |
| 0.049 | 0.001 | 0.079 | Telomerase stimulant | 0.046 0.001 CHEMBL3542195 0.079 0.001 CHEMBL3542275 0.03 0.003 CHEMBL3542345 0.029 0.003 CHEMBL3542255 0.021 0.007 CHEMBL3542317 0.026 0.004 CHEMBL3542274 | CHEMBL3542275 | |
| 0.106 | 0.06 | 0.112 | Toll-Like receptor 4 antagonist | 0.091 0.088 CHEMBL3542195 0.112 0.052 CHEMBL3542275 | CHEMBL3542275 | |
| 0.072 | 0.03 | 0.096 | Nitric oxide donor | 0.075 0.027 CHEMBL3542195 0.096 0.01 CHEMBL3542275 0.066 0.038 CHEMBL3542345 0.068 0.036 CHEMBL3542317 0.073 0.029 CHEMBL3542274 | CHEMBL3542275 | |
| 0.045 | 0.005 | 0.136 | Progesterone agonist | 0.06 0.004 CHEMBL3542195 0.121 0.003 CHEMBL3542345 0.136 0.003 CHEMBL3542255 0.116 0.003 CHEMBL3542317 0.098 0.004 CHEMBL3542274 | CHEMBL3542255 | |
| 0.16 | 0.124 | 0.231 | Neurotrophic factor enhancer | 0.166 0.115 CHEMBL3542195 0.231 0.05 CHEMBL3542275 0.152 0.135 CHEMBL3542255 0.153 0.133 CHEMBL3542274 | CHEMBL3542275 | |
| 0.166 | 0.136 | 0.35 | Vasodilator | 0.17 0.132 CHEMBL3542195 0.35 0.033 CHEMBL3542275 | CHEMBL3542275 | |
| 0.052 | 0.025 | 0.063 | Microtubule stabilization | 0.054 0.023 CHEMBL3542195 0.057 0.019 CHEMBL3542275 0.063 0.012 CHEMBL3542345 0.054 0.023 CHEMBL3542255 0.055 0.021 CHEMBL3542317 0.062 0.013 CHEMBL3542274 | CHEMBL3542345 | |
| 0.058 | 0.031 | 0.096 | Acetyl-CoA transferase inhibitor | 0.062 0.029 CHEMBL3542195 0.06 0.03 CHEMBL3542275 0.096 0.014 CHEMBL3542345 0.048 0.045 CHEMBL3542317 0.076 0.022 CHEMBL3542274 | CHEMBL3542345 | |
| 0.059 | 0.033 | 0.088 | Acetyl-CoA transferase 2 inhibitor | 0.064 0.024 CHEMBL3542195 0.068 0.019 CHEMBL3542275 0.088 0.008 CHEMBL3542345 0.063 0.025 CHEMBL3542317 0.085 0.009 CHEMBL3542274 | CHEMBL3542345 | |
| 0.063 | 0.037 | 0.191 | Androgen agonist | 0.093 0.018 CHEMBL3542195 0.083 0.022 CHEMBL3542275 0.191 0.005 CHEMBL3542345 0.164 0.006 CHEMBL3542255 0.183 0.005 CHEMBL3542317 0.166 0.006 CHEMBL3542274 | CHEMBL3542345 | |
| 0.088 | 0.066 | 0.119 | Glutamate release inhibitor | 0.119 0.023 CHEMBL3542275 | CHEMBL3542275 | |
| 0.038 | 0.017 | 0.079 | RNA-directed RNA polymerase stimulant | 0.042 0.016 CHEMBL3542195 0.079 0.008 CHEMBL3542275 0.064 0.01 CHEMBL3542345 0.068 0.01 CHEMBL3542255 0.036 0.018 CHEMBL3542317 0.059 0.011 CHEMBL3542274 | CHEMBL3542275 | |
| 0.054 | 0.037 | 0.058 | Alpha-mannosidase inhibitor | 0.05 0.044 CHEMBL3542195 0.058 0.029 CHEMBL3542275 | CHEMBL3542275 | |
| 0.024 | 0.011 | 0.039 | Corticosteroid-like | 0.025 0.01 CHEMBL3542195 0.031 0.006 CHEMBL3542275 0.028 0.008 CHEMBL3542345 0.03 0.007 CHEMBL3542255 0.039 0.004 CHEMBL3542317 0.027 0.009 CHEMBL3542274 | CHEMBL3542317 | |
| 0.029 | 0.018 | 0.032 | 1,3-Beta-glucan synthase inhibitor | 0.029 0.018 CHEMBL3542195 0.032 0.011 CHEMBL3542275 | CHEMBL3542275 | |
| 0.122 | 0.112 | 0.183 | NOS3 expression enhancer | 0.183 0.048 CHEMBL3542275 | CHEMBL3542275 | |
| 0.027 | 0.019 | 0.242 | 11-Beta-hydroxysteroid dehydrogenase 2 inhibitor | 0.035 0.013 CHEMBL3542195 0.242 0.003 CHEMBL3542275 0.084 0.005 CHEMBL3542345 0.088 0.005 CHEMBL3542255 0.154 0.004 CHEMBL3542274 | CHEMBL3542275 | |
| 0.016 | 0.009 | 0.016 | Antibiotic Macrolide-like | 0.016 0.008 CHEMBL3542195 0.015 0.009 CHEMBL3542275 | ||
| 0.04 | 0.037 | 0.669 | Phosphorylase inhibitor | 0.669 0.002 CHEMBL3542275 0.092 0.014 CHEMBL3542274 | CHEMBL3542275 | |
| 0.06 | 0.057 | 0.073 | Phosphofructokinase-1 inhibitor | 0.073 0.045 CHEMBL3542275 | CHEMBL3542275 | |
| 0.156 | 0.163 | 0.233 | DNA damaging | 0.233 0.091 CHEMBL3542275 | CHEMBL3542275 | |
| 0.05 | 0.073 | 0.112 | Lipase inhibitor | 0.112 0.021 CHEMBL3542275 | CHEMBL3542275 | |
| 0.005 | 0.029 | 0.039 | Glucocorticoid agonist | 0.039 0.005 CHEMBL3542317 | CHEMBL3542317 | |
| 0.126 | 0.156 | 0.284 | P-glycoprotein inhibitor | 0.284 0.032 CHEMBL3542275 0.141 0.131 CHEMBL3542274 | CHEMBL3542275 | |
| 0.012 | 0.047 | 0.024 | Adenosine A1 receptor agonist | 0.024 0.017 CHEMBL3542275 | CHEMBL3542275 | |
| 0.028 | 0.072 | 0.042 | Glucose-6-phosphate dehydrogenase inhibitor | 0.035 0.032 CHEMBL3542275 0.039 0.023 CHEMBL3542345 0.042 0.018 CHEMBL3542255 0.037 0.026 CHEMBL3542274 | CHEMBL3542255 | |
| 0.081 | 0.129 | 0.11 | Microtubule formation inhibitor | 0.101 0.088 CHEMBL3542195 0.101 0.09 CHEMBL3542275 0.11 0.073 CHEMBL3542345 0.103 0.086 CHEMBL3542317 0.11 0.074 CHEMBL3542274 | CHEMBL3542274 | |
| 0.05 | 0.111 | 0.071 | CDC25A inhibitor | 0.07 0.057 CHEMBL3542275 0.071 0.055 CHEMBL3542255 0.067 0.063 CHEMBL3542274 | CHEMBL3542255 | |
| 0.023 | 0.084 | 0.047 | Tubulin agonist | 0.047 0.009 CHEMBL3542345 0.045 0.011 CHEMBL3542274 | CHEMBL3542345 | |
| 0.033 | 0.113 | 0.051 | Heparanase inhibitor | 0.051 0.043 CHEMBL3542275 | CHEMBL3542275 | |
| 0.009 | 0.089 | 0.033 | Purinergic P2X agonist | 0.033 0.016 CHEMBL3542275 | CHEMBL3542275 | |
| 0.018 | 0.102 | 0.084 | 11-Beta-hydroxysteroid dehydrogenase 1 inhibitor | 0.044 0.036 CHEMBL3542275 0.076 0.017 CHEMBL3542345 0.061 0.023 CHEMBL3542255 0.084 0.015 CHEMBL3542274 | CHEMBL3542274 | |
| 0.062 | 0.147 | 0.157 | Anabolic | 0.119 0.041 CHEMBL3542275 0.136 0.027 CHEMBL3542345 0.157 0.014 CHEMBL3542255 0.143 0.022 CHEMBL3542317 0.137 0.026 CHEMBL3542274 | CHEMBL3542255 | |
| 0.011 | 0.102 | 0.037 | Glucocorticoid antagonist | 0.037 0.02 CHEMBL3542255 0.03 0.024 CHEMBL3542317 | CHEMBL3542255 | |
| 0.005 | 0.098 | 0.058 | Estrogen receptor alpha agonist | 0.058 0.015 CHEMBL3542275 | CHEMBL3542275 | |
| 0.005 | 0.108 | 0.046 | Estrogen receptor beta agonist | 0.046 0.02 CHEMBL3542275 | CHEMBL3542275 | |
| 0.008 | 0.112 | 0.022 | Retinoid X gamma receptor agonist | 0.022 0.017 CHEMBL3542274 | CHEMBL3542274 | |
| 0.04 | 0.16 | 0.139 | Monophenol monooxygenase inhibitor | 0.139 0.052 CHEMBL3542275 | CHEMBL3542275 | |
| 0.084 | 0.213 | 0.158 | Anesthetic general | 0.158 0.105 CHEMBL3542275 | CHEMBL3542275 | |
| 0.045 | 0.176 | 0.096 | Protease inhibitor | 0.096 0.069 CHEMBL3542275 0.093 0.071 CHEMBL3542274 | CHEMBL3542275 | |
| 0.094 | 0.232 | 0.264 | Non-steroidal antiinflammatory agent | 0.264 0.037 CHEMBL3542275 | CHEMBL3542275 | |
| 0.083 | 0.227 | 0.111 | Vanilloid 1 agonist | 0.111 0.11 CHEMBL3542275 | CHEMBL3542275 | |
| 0.013 | 0.168 | 0.038 | Opioid kappa receptor agonist | 0.038 0.037 CHEMBL3542255 | CHEMBL3542255 | |
| 0.119 | 0.276 | 0.264 | Gastrin inhibitor | 0.264 0.064 CHEMBL3542275 0.208 0.136 CHEMBL3542274 | CHEMBL3542275 | |
| 0.047 | 0.249 | 0.121 | Adenylate cyclase inhibitor | 0.121 0.067 CHEMBL3542275 | CHEMBL3542275 | |
| 0.054 | 0.258 | 0.104 | Estrogen antagonist | 0.104 0.088 CHEMBL3542275 | CHEMBL3542275 | |
| 0.096 | 0.333 | 0.512 | Hypoxia-inducible factor 1 alpha inhibitor | 0.512 0.014 CHEMBL3542275 0.218 0.131 CHEMBL3542274 | CHEMBL3542275 | |
| 0.035 | 0.282 | 0.128 | Uric acid excretion stimulant | 0.128 0.034 CHEMBL3542275 | CHEMBL3542275 | |
| 0.091 | 0.345 | 0.42 | Transcription factor STAT3 inhibitor | 0.42 0.015 CHEMBL3542275 | CHEMBL3542275 | |
| 0.098 | 0.363 | 0.431 | Vasodilator, peripheral | 0.431 0.046 CHEMBL3542275 | CHEMBL3542275 | |
| 0.057 | 0.334 | 0.217 | Interleukin agonist | 0.217 0.105 CHEMBL3542275 | CHEMBL3542275 | |
| 0.05 | 0.333 | 0.206 | Arachidonic acid antagonist | 0.188 0.045 CHEMBL3542345 0.206 0.027 CHEMBL3542255 0.179 0.054 CHEMBL3542317 0.186 0.047 CHEMBL3542274 | CHEMBL3542255 | |
| 0.033 | 0.326 | 0.128 | Beta glucuronidase inhibitor | 0.128 0.039 CHEMBL3542275 | CHEMBL3542275 | |
| 0.016 | 0.354 | 0.175 | Aldosterone antagonist | 0.076 0.012 CHEMBL3542345 0.175 0.004 CHEMBL3542255 0.065 0.016 CHEMBL3542317 0.074 0.013 CHEMBL3542274 | CHEMBL3542255 | |
| 0.062 | 0.407 | 0.202 | Phospholipase C inhibitor | 0.202 0.043 CHEMBL3542275 0.159 0.09 CHEMBL3542345 0.196 0.047 CHEMBL3542274 | CHEMBL3542275 | |
| 0.03 | 0.382 | 0.138 | Xanthine oxidase inhibitor | 0.138 0.039 CHEMBL3542275 | CHEMBL3542275 | |
| 0.039 | 0.397 | 0.234 | Insulin sensitizer | 0.234 0.044 CHEMBL3542275 0.161 0.118 CHEMBL3542274 | CHEMBL3542275 | |
| 0.08 | 0.458 | 0.273 | Vasodilator, coronary | 0.273 0.112 CHEMBL3542275 | CHEMBL3542275 | |
| 0.027 | 0.422 | 0.086 | Antineoplastic alkaloid | 0.086 0.058 CHEMBL3542317 | CHEMBL3542317 | |
| 0.036 | 0.44 | 0.135 | Farnesoid X receptor antagonist | 0.118 0.108 CHEMBL3542275 0.133 0.077 CHEMBL3542255 0.135 0.074 CHEMBL3542317 0.122 0.098 CHEMBL3542274 | CHEMBL3542317 | |
| 0.07 | 0.482 | 0.313 | Histamine release inhibitor | 0.313 0.117 CHEMBL3542275 | CHEMBL3542275 | |
| 0.025 | 0.472 | 0.101 | Bile acid receptor antagonist | 0.092 0.068 CHEMBL3542345 0.101 0.048 CHEMBL3542274 | CHEMBL3542274 | |
| 0.051 | 0.501 | 0.353 | Transcription factor STAT inhibitor | 0.353 0.033 CHEMBL3542275 | CHEMBL3542275 | |
| 0.024 | 0.59 | 0.099 | Interleukin 1b antagonist | 0.099 0.082 CHEMBL3542275 | CHEMBL3542275 | |
| 0.002 | 0.612 | 0.057 | Farnesoid X receptor agonist | 0.041 0.023 CHEMBL3542345 0.045 0.019 CHEMBL3542255 0.057 0.011 CHEMBL3542274 | CHEMBL3542274 | |
| 0.006 | 0.659 | 0.088 | Androgen antagonist | 0.083 0.063 CHEMBL3542345 0.088 0.057 CHEMBL3542255 | CHEMBL3542255 | |
| 0.004 | 0.727 | 0.082 | Inducible nitric-oxide synthase inhibitor | 0.082 0.058 CHEMBL3542275 | CHEMBL3542275 | |
| 0.006 | 0.846 | 0.126 | Pregnane X receptor agonist | 0.126 0.111 CHEMBL3542255 | CHEMBL3542255 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |