Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.3690.010.449NOS3 expression enhancer

0.421 0.007 CHEMBL3542206

0.309 0.016 CHEMBL3542205

0.449 0.006 CHEMBL3542260

CHEMBL3542260
0.320.0280.371Ca(v)3.3 blocker

0.371 0.009 CHEMBL3542206

0.293 0.048 CHEMBL3542219

0.287 0.054 CHEMBL3542262

0.288 0.054 CHEMBL3542205

0.366 0.01 CHEMBL3542260

CHEMBL3542206
0.3240.0960.346Toll-Like receptor agonist

0.346 0.084 CHEMBL3542206

0.271 0.13 CHEMBL3542205

0.319 0.099 CHEMBL3542260

CHEMBL3542206
0.320.0980.345Toll-Like receptor 7 agonist

0.345 0.084 CHEMBL3542206

0.267 0.133 CHEMBL3542205

0.312 0.102 CHEMBL3542260

CHEMBL3542206
0.1770.0290.183MAP3K9 inhibitor

0.183 0.024 CHEMBL3542206

0.138 0.079 CHEMBL3542219

0.182 0.025 CHEMBL3542262

0.164 0.042 CHEMBL3542205

0.158 0.049 CHEMBL3542260

CHEMBL3542206
0.1520.0080.152Bromodomain-containing protein 2 inhibitor

0.121 0.022 CHEMBL3542219

0.082 0.073 CHEMBL3542262

0.094 0.049 CHEMBL3542205

0.084 0.069 CHEMBL3542260

0.1690.0450.169Sodium channel blocker

0.16 0.051 CHEMBL3542206

0.109 0.099 CHEMBL3542219

0.148 0.059 CHEMBL3542205

0.112 0.094 CHEMBL3542260

0.1680.050.168Hemostatic

0.16 0.057 CHEMBL3542205

0.1830.0690.183Amyloid beta precursor protein antagonist

0.129 0.128 CHEMBL3542206

0.159 0.092 CHEMBL3542262

0.17 0.081 CHEMBL3542205

0.182 0.071 CHEMBL3542260

0.160.0510.16Neuropeptide Y1 antagonist
0.2750.180.305Calcium channel L-type activator

0.292 0.164 CHEMBL3542219

0.275 0.18 CHEMBL3542262

0.305 0.153 CHEMBL3542205

CHEMBL3542205
0.2740.1870.406Cyclophilin D inhibitor

0.272 0.188 CHEMBL3542206

0.406 0.087 CHEMBL3542205

CHEMBL3542205
0.1230.0460.142AMP-activated protein kinase stimulant

0.103 0.066 CHEMBL3542219

0.102 0.068 CHEMBL3542262

0.142 0.034 CHEMBL3542205

0.099 0.072 CHEMBL3542260

CHEMBL3542205
0.0820.0240.3225 Hydroxytryptamine 1 agonist

0.322 0.005 CHEMBL3542206

0.155 0.014 CHEMBL3542260

CHEMBL3542206
0.0980.0480.098Acetylcholine agonist

0.091 0.054 CHEMBL3542262

0.1850.1340.211Cardiotonic

0.211 0.109 CHEMBL3542219

0.178 0.142 CHEMBL3542262

0.209 0.111 CHEMBL3542205

CHEMBL3542219
0.0940.0450.199Histamine H1 receptor antagonist

0.199 0.015 CHEMBL3542206

0.105 0.039 CHEMBL3542260

CHEMBL3542206
0.0810.0370.081Amidase inhibitor

0.067 0.054 CHEMBL3542205

0.110.0690.147Protein kinase (CK2) alpha inhibitor

0.147 0.044 CHEMBL3542206

0.093 0.083 CHEMBL3542205

0.142 0.046 CHEMBL3542260

CHEMBL3542206
0.1640.1260.292Potassium channel (Voltage-sensitive) blocker

0.292 0.052 CHEMBL3542206

0.211 0.088 CHEMBL3542260

CHEMBL3542206
0.0590.0240.059Antiviral (Hepatitis D)

0.048 0.04 CHEMBL3542219

0.054 0.029 CHEMBL3542262

0.0940.060.18Antihistaminic

0.18 0.024 CHEMBL3542206

0.087 0.068 CHEMBL3542260

CHEMBL3542206
0.0580.0250.066Alpha 1L adrenoreceptor antagonist

0.066 0.015 CHEMBL3542206

0.053 0.034 CHEMBL3542219

0.053 0.034 CHEMBL3542262

0.052 0.037 CHEMBL3542205

0.059 0.023 CHEMBL3542260

CHEMBL3542206
0.0550.0230.055Oleamide hydrolase inhibitor
0.0350.0050.035Apolipoprotein B-100 inhibitor

0.02 0.011 CHEMBL3542260

0.1170.0880.152Sodium channel (voltage-gated) blocker

0.152 0.053 CHEMBL3542206

0.106 0.103 CHEMBL3542260

CHEMBL3542206
0.0850.0590.177Histamine antagonist

0.177 0.023 CHEMBL3542206

0.077 0.067 CHEMBL3542260

CHEMBL3542206
0.0570.0310.057Autotaxin inhibitor

0.048 0.044 CHEMBL3542262

0.053 0.035 CHEMBL3542205

0.05 0.04 CHEMBL3542260

0.040.0160.04Factor XI inhibitor

0.036 0.02 CHEMBL3542206

0.033 0.025 CHEMBL3542205

0.033 0.024 CHEMBL3542260

0.150.1290.179Anticonvulsant

0.179 0.1 CHEMBL3542219

CHEMBL3542219
0.0440.0240.044Factor XIa inhibitor

0.039 0.03 CHEMBL3542206

0.036 0.035 CHEMBL3542205

0.0480.030.1465 Hydroxytryptamine 1A agonist

0.146 0.011 CHEMBL3542206

0.092 0.017 CHEMBL3542260

CHEMBL3542206
0.0480.030.069Farnesyltransferase inhibitor

0.069 0.016 CHEMBL3542206

0.058 0.021 CHEMBL3542260

CHEMBL3542206
0.1050.0880.137Sphingosine 1-phosphate receptor 2 agonist

0.137 0.035 CHEMBL3542206

0.102 0.095 CHEMBL3542262

0.108 0.079 CHEMBL3542205

0.102 0.098 CHEMBL3542260

CHEMBL3542206
0.0780.0620.084Phosphodiesterase 11A inhibitor

0.084 0.05 CHEMBL3542206

CHEMBL3542206
0.0780.0620.084Phosphodiesterase XI inhibitor

0.084 0.05 CHEMBL3542206

CHEMBL3542206
0.0640.050.111Leukotriene synthesis inhibitor

0.111 0.02 CHEMBL3542206

0.06 0.055 CHEMBL3542205

0.094 0.03 CHEMBL3542260

CHEMBL3542206
0.0640.0510.2045 Hydroxytryptamine agonist

0.204 0.014 CHEMBL3542206

0.094 0.035 CHEMBL3542260

CHEMBL3542206
0.0410.0280.041Glutamate (mGluR1a) antagonist
0.0510.0390.198Melanin-concentrating hormone receptor 1 antagonist

0.089 0.017 CHEMBL3542206

0.198 0.005 CHEMBL3542260

CHEMBL3542260
0.0660.0550.066Glutamate (mGluR group I) antagonist

0.066 0.054 CHEMBL3542206

0.065 0.056 CHEMBL3542260

0.0810.0710.088Hematopoietic

0.082 0.068 CHEMBL3542219

0.087 0.056 CHEMBL3542262

0.088 0.052 CHEMBL3542205

CHEMBL3542205
0.0660.0570.091Secretase beta inhibitor

0.083 0.032 CHEMBL3542206

0.091 0.024 CHEMBL3542260

CHEMBL3542260
0.0850.0770.085Butyrylcholinesterase inhibitor
0.020.0130.02Apolipoprotein B inhibitor
0.2070.20.207Antiobesity
0.0530.050.182Cannabinoid CB1 receptor agonist

0.076 0.031 CHEMBL3542206

0.182 0.007 CHEMBL3542260

CHEMBL3542260
0.0350.0330.048Dopamine D3 agonist

0.048 0.021 CHEMBL3542206

CHEMBL3542206
0.0510.0510.098Protein kinase C theta inhibitor

0.098 0.008 CHEMBL3542206

0.063 0.032 CHEMBL3542260

CHEMBL3542206
0.0220.0230.0345 Hydroxytryptamine 1F agonist

0.033 0.01 CHEMBL3542206

0.034 0.01 CHEMBL3542260

CHEMBL3542260
0.0810.0840.094DNA directed RNA polymerase inhibitor

0.094 0.064 CHEMBL3542206

CHEMBL3542206
0.1810.1860.228Nootropic

0.228 0.127 CHEMBL3542206

0.218 0.136 CHEMBL3542219

0.198 0.161 CHEMBL3542260

CHEMBL3542206
0.0640.0690.15MAP-kinase-activated kinase 2 inhibitor

0.15 0.011 CHEMBL3542206

0.084 0.041 CHEMBL3542260

CHEMBL3542206
0.0390.0470.083Dipeptidyl peptidase IV inhibitor

0.083 0.007 CHEMBL3542206

0.048 0.023 CHEMBL3542260

CHEMBL3542206
0.0160.0240.023Geranylgeranyltransferase I inhibitor

0.023 0.013 CHEMBL3542206

0.019 0.017 CHEMBL3542260

CHEMBL3542206
0.0690.080.16MAP-kinase-activated kinase inhibitor

0.16 0.012 CHEMBL3542206

0.092 0.047 CHEMBL3542260

CHEMBL3542206
0.0080.020.015Egl nine homolog 2 inhibitor

0.015 0.005 CHEMBL3542206

0.012 0.008 CHEMBL3542260

CHEMBL3542206
0.0510.0650.126Toll-Like receptor 7 antagonist

0.126 0.01 CHEMBL3542206

0.095 0.025 CHEMBL3542260

CHEMBL3542206
0.0350.0510.042Glutamate (mGluR5) antagonist

0.042 0.039 CHEMBL3542206

CHEMBL3542206
0.2080.2270.381Analgesic

0.381 0.093 CHEMBL3542219

CHEMBL3542219
0.0260.0450.032Somatostatin 5 agonist

0.032 0.029 CHEMBL3542260

CHEMBL3542260
0.0370.0560.05Bromodomain-containing protein 3 inhibitor

0.05 0.033 CHEMBL3542219

CHEMBL3542219
0.0170.0380.0955 Hydroxytryptamine 1D agonist

0.095 0.004 CHEMBL3542206

0.042 0.013 CHEMBL3542260

CHEMBL3542206
0.0460.0680.086Dopamine agonist

0.086 0.034 CHEMBL3542206

CHEMBL3542206
0.1310.1530.181Cyclin-dependent kinase 3 inhibitor

0.147 0.104 CHEMBL3542262

0.147 0.103 CHEMBL3542205

0.181 0.048 CHEMBL3542260

CHEMBL3542260
0.0430.0670.087Dipeptidyl peptidase inhibitor

0.087 0.012 CHEMBL3542206

0.055 0.033 CHEMBL3542260

CHEMBL3542206
0.1730.1980.221Immunomodulator

0.221 0.14 CHEMBL3542262

CHEMBL3542262
0.0190.0450.035Plasma kallikrein inhibitor

0.035 0.023 CHEMBL3542206

CHEMBL3542206
0.0570.0830.071Glutamate (mGluR) antagonist

0.071 0.059 CHEMBL3542206

CHEMBL3542206
0.070.0980.107Protein kinase (CK2) inhibitor

0.107 0.058 CHEMBL3542206

0.096 0.068 CHEMBL3542260

CHEMBL3542206
0.0280.0580.072Chemokine receptor agonist

0.065 0.023 CHEMBL3542206

0.072 0.016 CHEMBL3542260

CHEMBL3542260
0.0270.060.032Protein kinase C beta I inhibitor

0.032 0.028 CHEMBL3542262

CHEMBL3542262
0.0650.1030.148Protein kinase C delta inhibitor

0.148 0.022 CHEMBL3542206

0.098 0.054 CHEMBL3542262

0.084 0.071 CHEMBL3542260

CHEMBL3542206
0.0370.0770.07Protein kinase C eta inhibitor

0.059 0.034 CHEMBL3542206

0.07 0.029 CHEMBL3542262

CHEMBL3542262
0.0070.0490.025CXC chemokine 4 receptor agonist

0.025 0.004 CHEMBL3542206

0.018 0.007 CHEMBL3542260

CHEMBL3542206
0.1740.2170.225MAP kinase kinase 3 inhibitor

0.225 0.064 CHEMBL3542206

0.211 0.094 CHEMBL3542262

0.195 0.137 CHEMBL3542260

CHEMBL3542206
0.0640.1090.089Caspase 7 inhibitor

0.089 0.044 CHEMBL3542260

CHEMBL3542260
0.0110.0560.039CXC chemokine receptor agonist

0.035 0.023 CHEMBL3542206

0.039 0.018 CHEMBL3542260

CHEMBL3542260
0.0150.0610.027Protocollagen prolyl hydroxylase inhibitor

0.027 0.02 CHEMBL3542206

CHEMBL3542206
0.080.1330.168Nav1.5 sodium channel blocker

0.168 0.019 CHEMBL3542206

0.112 0.065 CHEMBL3542260

CHEMBL3542206
0.0440.0990.062Phosphodiesterase 5A inhibitor

0.062 0.06 CHEMBL3542206

CHEMBL3542206
0.1180.1730.198Potassium channel blocker

0.198 0.094 CHEMBL3542206

0.158 0.127 CHEMBL3542260

CHEMBL3542206
0.0340.0950.067CXC chemokine 4 receptor antagonist

0.067 0.038 CHEMBL3542206

0.063 0.04 CHEMBL3542260

CHEMBL3542206
0.1120.1760.274HERG channel blocker

0.274 0.057 CHEMBL3542206

0.176 0.105 CHEMBL3542260

CHEMBL3542206
0.0290.0950.126Toll-Like receptor 8 antagonist

0.126 0.005 CHEMBL3542206

0.059 0.032 CHEMBL3542260

CHEMBL3542206
0.0310.1010.111Dopamine D3 antagonist

0.078 0.033 CHEMBL3542206

0.111 0.022 CHEMBL3542260

CHEMBL3542260
0.0330.1040.083Cyclin-dependent kinase 6 inhibitor

0.083 0.019 CHEMBL3542206

0.06 0.041 CHEMBL3542260

CHEMBL3542206
0.0410.1130.101Protein kinase C beta inhibitor

0.101 0.013 CHEMBL3542206

0.066 0.056 CHEMBL3542260

CHEMBL3542206
0.1140.1880.15Platelet aggregation inhibitor

0.15 0.128 CHEMBL3542262

CHEMBL3542262
0.1560.2330.257Vasodilator, peripheral

0.257 0.122 CHEMBL3542262

CHEMBL3542262
0.0570.1370.1965 Hydroxytryptamine antagonist

0.196 0.035 CHEMBL3542206

0.153 0.048 CHEMBL3542260

CHEMBL3542206
0.0580.1390.084Uric acid excretion stimulant

0.084 0.075 CHEMBL3542206

0.083 0.078 CHEMBL3542219

CHEMBL3542206
0.0320.1140.093Dopamine antagonist

0.093 0.042 CHEMBL3542206

0.09 0.042 CHEMBL3542260

CHEMBL3542206
0.060.1460.099DNA intercalator

0.099 0.074 CHEMBL3542262

CHEMBL3542262
0.0380.1260.086Nav1.7 sodium channel blocker

0.086 0.029 CHEMBL3542206

CHEMBL3542206
0.1080.2010.12CC chemokine 6 receptor antagonist

0.12 0.117 CHEMBL3542206

CHEMBL3542206
0.0220.120.06Dopamine D2 antagonist

0.06 0.05 CHEMBL3542206

0.058 0.051 CHEMBL3542260

CHEMBL3542206
0.0320.1330.07Cannabinoid receptor antagonist

0.07 0.05 CHEMBL3542260

CHEMBL3542260
0.0690.1770.132Cytokine production inhibitor

0.132 0.077 CHEMBL3542206

CHEMBL3542206
0.0570.1670.128GABA receptor agonist

0.128 0.05 CHEMBL3542206

CHEMBL3542206
0.0220.1330.084Protein kinase C epsilon inhibitor

0.084 0.018 CHEMBL3542206

CHEMBL3542206
0.0310.1430.085Glutamate receptor agonist

0.085 0.048 CHEMBL3542206

CHEMBL3542206
0.0270.140.0825 Hydroxytryptamine 1 antagonist

0.082 0.046 CHEMBL3542206

CHEMBL3542206
0.0450.1590.068Phosphodiesterase VIII inhibitor

0.068 0.059 CHEMBL3542206

CHEMBL3542206
0.0210.1390.314Raf kinase C inhibitor

0.314 0.005 CHEMBL3542219

CHEMBL3542219
0.0560.1740.081Transcription factor NF kappa B stimulant

0.081 0.068 CHEMBL3542219

CHEMBL3542219
0.0650.1830.143Glutamate (mGluR7) agonist

0.105 0.05 CHEMBL3542206

0.143 0.015 CHEMBL3542260

CHEMBL3542260
0.0870.2060.176Insulin secretagoues

0.176 0.051 CHEMBL3542205

CHEMBL3542205
0.0220.1420.101Cannabinoid receptor agonist

0.101 0.026 CHEMBL3542260

CHEMBL3542260
0.0330.1560.099Protein kinase C alpha inhibitor

0.099 0.023 CHEMBL3542206

CHEMBL3542206
0.0250.1530.0915 Hydroxytryptamine 1B antagonist

0.091 0.028 CHEMBL3542206

0.076 0.037 CHEMBL3542260

CHEMBL3542206
0.0390.1760.091MAP kinase kinase kinase inhibitor

0.091 0.075 CHEMBL3542206

CHEMBL3542206
0.0430.1830.085Potassium channel activator

0.085 0.067 CHEMBL3542219

CHEMBL3542219
0.0290.170.071CXC chemokine receptor antagonist

0.071 0.048 CHEMBL3542206

0.065 0.056 CHEMBL3542260

CHEMBL3542206
0.0240.1670.087Lysine-specific demethylase 1A inhibitor

0.087 0.01 CHEMBL3542206

CHEMBL3542206
0.0160.1590.085Dopamine D4 antagonist

0.085 0.031 CHEMBL3542206

CHEMBL3542206
0.0270.1730.065Check point kinase 1 inhibitor

0.065 0.051 CHEMBL3542206

CHEMBL3542206
0.0220.1710.05Nicotinic alpha7 receptor agonist

0.05 0.042 CHEMBL3542260

CHEMBL3542260
0.0960.2630.127MAP kinase kinase 4 inhibitor

0.127 0.124 CHEMBL3542262

CHEMBL3542262
0.0840.2570.158Platelet antagonist

0.158 0.136 CHEMBL3542262

CHEMBL3542262
0.0190.1920.0525 Hydroxytryptamine 3 antagonist

0.052 0.045 CHEMBL3542206

CHEMBL3542206
0.0370.210.085Pim-3 kinase inhibitor

0.085 0.067 CHEMBL3542206

CHEMBL3542206
0.0280.2260.078Analgesic, opioid

0.078 0.05 CHEMBL3542219

CHEMBL3542219
0.0080.2060.046AMPA receptor antagonist

0.046 0.035 CHEMBL3542206

CHEMBL3542206
0.0410.2540.141Protein kinase C gamma inhibitor

0.141 0.037 CHEMBL3542206

CHEMBL3542206
0.0490.2930.165Toll-Like receptor antagonist

0.165 0.046 CHEMBL3542206

0.11 0.101 CHEMBL3542260

CHEMBL3542206
0.0310.2790.082MAP kinase 9 inhibitor

0.082 0.081 CHEMBL3542206

CHEMBL3542206
0.0080.2570.077Cannabinoid CB2 receptor antagonist

0.077 0.021 CHEMBL3542260

CHEMBL3542260
0.0180.2690.123Neuraminidase (influenza) inhibitor

0.123 0.011 CHEMBL3542262

CHEMBL3542262
0.0120.2680.091Neuraminidase inhibitor

0.091 0.019 CHEMBL3542262

0.056 0.049 CHEMBL3542260

CHEMBL3542262
0.0210.3140.114Pim-1 kinase inhibitor

0.114 0.046 CHEMBL3542206

CHEMBL3542206
0.0310.3250.123Toll-Like receptor 9 antagonist

0.123 0.083 CHEMBL3542206

CHEMBL3542206
0.0090.3040.056Opioid agonist

0.056 0.034 CHEMBL3542219

CHEMBL3542219
0.0170.3460.15Acetyl-CoA transferase 2 inhibitor

0.15 0.003 CHEMBL3542219

CHEMBL3542219
0.0250.3760.154GABA C receptor antagonist

0.154 0.028 CHEMBL3542206

CHEMBL3542206
0.0060.360.021Protein 30S ribosomal subunit inhibitor

0.021 0.02 CHEMBL3542262

CHEMBL3542262
0.0050.3740.091Opioid kappa receptor agonist

0.091 0.01 CHEMBL3542219

CHEMBL3542219
0.0090.3820.078Acetyl-CoA transferase inhibitor

0.078 0.021 CHEMBL3542219

CHEMBL3542219
0.0110.3910.07CDC7 inhibitor

0.07 0.044 CHEMBL3542206

CHEMBL3542206
0.0130.40.051Antibiotic Aminoglycoside-like

0.051 0.013 CHEMBL3542262

CHEMBL3542262
0.0330.4290.145Death-associated protein kinase 3 inhibitor

0.145 0.13 CHEMBL3542206

CHEMBL3542206
0.0050.4130.119Antineoplastic antibiotic

0.119 0.039 CHEMBL3542219

CHEMBL3542219
0.0740.5010.209Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.209 0.147 CHEMBL3542206

CHEMBL3542206
0.0230.4570.097GABA C receptor rho-1 antagonist

0.097 0.067 CHEMBL3542206

CHEMBL3542206
0.0310.4710.157Cyclin-dependent kinase 8 inhibitor

0.157 0.073 CHEMBL3542206

CHEMBL3542206
0.1010.5420.255MAP kinase kinase 6 inhibitor

0.255 0.184 CHEMBL3542206

CHEMBL3542206
0.0680.5190.1645 Hydroxytryptamine release stimulant

0.164 0.16 CHEMBL3542206

CHEMBL3542206
0.0140.5160.088Nitric-oxide synthase inhibitor

0.088 0.081 CHEMBL3542206

CHEMBL3542206
Ext Pa Pi Pmax Activity Other Results ID Pa_max