| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.899 | 0.003 | 0.9 | Caspase 9 stimulant | 0.896 0.003 CHEMBL3527009 0.9 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.85 | 0.011 | 0.85 | Apoptosis agonist | 0.84 0.012 CHEMBL3527009 0.838 0.012 CHEMBL442289 | ||
| 0.804 | 0.004 | 0.852 | Free radical scavenger | 0.847 0.004 CHEMBL3527009 0.852 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.782 | 0.004 | 0.782 | Caspase 3 stimulant | 0.712 0.005 CHEMBL3527009 0.712 0.005 CHEMBL442289 | ||
| 0.759 | 0.003 | 0.759 | Breast cancer-resistant protein inhibitor | 0.681 0.004 CHEMBL3527009 0.68 0.004 CHEMBL442289 | ||
| 0.759 | 0.005 | 0.846 | Antioxidant | 0.837 0.004 CHEMBL3527009 0.846 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.7 | 0.002 | 0.929 | Cystathionine beta-synthase inhibitor | 0.915 0.001 CHEMBL3527009 0.929 0.001 CHEMBL442289 | CHEMBL442289 | |
| 0.677 | 0.01 | 0.845 | Aryl hydrocarbon receptor agonist | 0.841 0.005 CHEMBL3527009 0.845 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.643 | 0.004 | 0.702 | GABA C receptor rho-3 antagonist | 0.688 0.003 CHEMBL3527009 0.702 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.64 | 0.004 | 0.64 | P-glycoprotein inhibitor | 0.611 0.005 CHEMBL3527009 0.599 0.005 CHEMBL442289 | ||
| 0.627 | 0.007 | 0.7 | Amyloid beta aggregation inhibitor | 0.692 0.005 CHEMBL3527009 0.7 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.618 | 0.004 | 0.799 | Peroxidase inhibitor | 0.781 0.002 CHEMBL3527009 0.799 0.002 CHEMBL442289 | CHEMBL442289 | |
| 0.617 | 0.009 | 0.617 | 5 Hydroxytryptamine release inhibitor | 0.573 0.015 CHEMBL3527009 0.583 0.013 CHEMBL442289 | ||
| 0.62 | 0.012 | 0.843 | 12-Lipoxygenase inhibitor | 0.829 0.004 CHEMBL3527009 0.843 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.621 | 0.016 | 0.804 | Aldehyde oxidase inhibitor | 0.77 0.005 CHEMBL3527009 0.804 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.607 | 0.009 | 0.668 | Histamine release inhibitor | 0.66 0.006 CHEMBL3527009 0.668 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.596 | 0.007 | 0.677 | Superoxide dismutase inhibitor | 0.668 0.005 CHEMBL3527009 0.677 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.592 | 0.004 | 0.693 | NADPH oxidase inhibitor | 0.68 0.003 CHEMBL3527009 0.693 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.608 | 0.052 | 0.789 | Alpha-glucosidase inhibitor | 0.764 0.023 CHEMBL3527009 0.789 0.019 CHEMBL442289 | CHEMBL442289 | |
| 0.582 | 0.033 | 0.69 | Transcription factor NF kappa B inhibitor | 0.673 0.024 CHEMBL3527009 0.69 0.022 CHEMBL442289 | CHEMBL442289 | |
| 0.549 | 0.006 | 0.679 | MAO inhibitor | 0.646 0.005 CHEMBL3527009 0.679 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.542 | 0.011 | 0.542 | Vasodilator, coronary | 0.492 0.017 CHEMBL3527009 0.488 0.017 CHEMBL442289 | ||
| 0.561 | 0.03 | 0.838 | 15-Lipoxygenase inhibitor | 0.822 0.005 CHEMBL3527009 0.838 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.532 | 0.005 | 0.687 | MAO A inhibitor | 0.647 0.004 CHEMBL3527009 0.687 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.585 | 0.058 | 0.653 | Antiinflammatory | 0.653 0.04 CHEMBL3527009 0.649 0.041 CHEMBL442289 | CHEMBL3527009 | |
| 0.529 | 0.012 | 0.529 | Tumour necrosis factor alpha release inhibitor | 0.502 0.014 CHEMBL3527009 0.492 0.015 CHEMBL442289 | ||
| 0.515 | 0.017 | 0.72 | Lipoxygenase inhibitor | 0.705 0.005 CHEMBL3527009 0.72 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.505 | 0.012 | 0.505 | Vasodilator | 0.483 0.013 CHEMBL3527009 0.484 0.013 CHEMBL442289 | ||
| 0.498 | 0.014 | 0.498 | DNA damaging | 0.448 0.02 CHEMBL3527009 0.449 0.019 CHEMBL442289 | ||
| 0.485 | 0.004 | 0.667 | Xanthine oxidase inhibitor | 0.621 0.003 CHEMBL3527009 0.667 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.474 | 0.005 | 0.474 | Acetylcholinesterase inhibitor | 0.436 0.005 CHEMBL3527009 0.428 0.005 CHEMBL442289 | ||
| 0.49 | 0.022 | 0.584 | Apoptosis antagonist | 0.583 0.012 CHEMBL3527009 0.584 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.477 | 0.018 | 0.528 | Nitric oxide antagonist | 0.522 0.014 CHEMBL3527009 0.528 0.014 CHEMBL442289 | CHEMBL442289 | |
| 0.474 | 0.018 | 0.541 | Hypoglycemic | 0.536 0.013 CHEMBL3527009 0.541 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.45 | 0.009 | 0.695 | Monophenol monooxygenase inhibitor | 0.657 0.004 CHEMBL3527009 0.695 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.444 | 0.005 | 0.553 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.542 0.003 CHEMBL3527009 0.553 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.442 | 0.005 | 0.675 | Interleukin 4 antagonist | 0.666 0.003 CHEMBL3527009 0.675 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.446 | 0.01 | 0.453 | Tubulin antagonist | 0.453 0.009 CHEMBL3527009 0.437 0.01 CHEMBL442289 | CHEMBL3527009 | |
| 0.451 | 0.02 | 0.656 | Hypoxia-inducible factor 1 alpha inhibitor | 0.642 0.005 CHEMBL3527009 0.656 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.426 | 0.004 | 0.591 | Carbonic anhydrase XIII inhibitor | 0.528 0.003 CHEMBL3527009 0.591 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.432 | 0.015 | 0.524 | RNA-directed DNA polymerase inhibitor | 0.524 0.009 CHEMBL3527009 0.523 0.009 CHEMBL442289 | CHEMBL3527009 | |
| 0.464 | 0.05 | 0.56 | Prostaglandin dehydrogenase inhibitor | 0.56 0.031 CHEMBL3527009 0.551 0.032 CHEMBL442289 | CHEMBL3527009 | |
| 0.442 | 0.032 | 0.466 | Spasmolytic | 0.451 0.031 CHEMBL3527009 0.466 0.028 CHEMBL442289 | CHEMBL442289 | |
| 0.42 | 0.011 | 0.549 | Melanin inhibitor | 0.52 0.006 CHEMBL3527009 0.549 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.411 | 0.005 | 0.461 | Topoisomerase II alpha inhibitor | 0.45 0.004 CHEMBL3527009 0.461 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.414 | 0.009 | 0.684 | Amylase inhibitor | 0.653 0.003 CHEMBL3527009 0.684 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.429 | 0.024 | 0.512 | Antiamyloidogenic | 0.492 0.017 CHEMBL3527009 0.512 0.015 CHEMBL442289 | CHEMBL442289 | |
| 0.413 | 0.012 | 0.425 | 5 Hydroxytryptamine uptake stimulant | 0.425 0.01 CHEMBL3527009 0.395 0.015 CHEMBL442289 | CHEMBL3527009 | |
| 0.41 | 0.012 | 0.438 | Hepatoprotectant | 0.435 0.01 CHEMBL3527009 0.438 0.01 CHEMBL442289 | CHEMBL442289 | |
| 0.4 | 0.005 | 0.406 | Alkaline phosphatase inhibitor | 0.4 0.005 CHEMBL3527009 0.406 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.399 | 0.008 | 0.621 | NOS3 expression enhancer | 0.599 0.004 CHEMBL3527009 0.621 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.4 | 0.01 | 0.513 | Topoisomerase II inhibitor | 0.493 0.007 CHEMBL3527009 0.513 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.393 | 0.004 | 0.455 | Nitric-oxide synthase stimulant | 0.448 0.003 CHEMBL3527009 0.455 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.397 | 0.008 | 0.436 | Protein kinase stimulant | 0.42 0.007 CHEMBL3527009 0.436 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.387 | 0.01 | 0.387 | Cholinergic | 0.342 0.014 CHEMBL3527009 0.331 0.015 CHEMBL442289 | ||
| 0.372 | 0.003 | 0.372 | Multidrug resistance-associated protein 1 inhibitor | 0.351 0.003 CHEMBL3527009 0.349 0.003 CHEMBL442289 | ||
| 0.378 | 0.017 | 0.493 | Dual specificity phosphatase inhibitor | 0.493 0.006 CHEMBL3527009 0.482 0.007 CHEMBL442289 | CHEMBL3527009 | |
| 0.358 | 0.004 | 0.438 | GABA C receptor rho-2 antagonist | 0.414 0.003 CHEMBL3527009 0.438 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.377 | 0.025 | 0.568 | Pyruvate kinase inhibitor | 0.556 0.005 CHEMBL3527009 0.568 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.36 | 0.009 | 0.398 | Tumour necrosis factor antagonist | 0.398 0.006 CHEMBL3527009 0.386 0.007 CHEMBL442289 | CHEMBL3527009 | |
| 0.361 | 0.011 | 0.407 | Protein-tyrosine phosphatase inhibitor | 0.407 0.008 CHEMBL3527009 0.405 0.008 CHEMBL442289 | CHEMBL3527009 | |
| 0.358 | 0.009 | 0.358 | Cytokine production inhibitor | 0.269 0.02 CHEMBL3527009 0.261 0.021 CHEMBL442289 | ||
| 0.352 | 0.004 | 0.352 | Aldose reductase inhibitor | 0.337 0.004 CHEMBL3527009 0.344 0.004 CHEMBL442289 | ||
| 0.347 | 0.004 | 0.622 | Creatine kinase inhibitor | 0.584 0.002 CHEMBL3527009 0.622 0.001 CHEMBL442289 | CHEMBL442289 | |
| 0.351 | 0.009 | 0.474 | MAO B inhibitor | 0.443 0.006 CHEMBL3527009 0.474 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.349 | 0.013 | 0.505 | Lipid peroxidase inhibitor | 0.499 0.005 CHEMBL3527009 0.505 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.348 | 0.014 | 0.442 | DNA methyltransferase I inhibitor | 0.437 0.006 CHEMBL3527009 0.442 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.353 | 0.02 | 0.492 | Dual specificity phosphatase 3 inhibitor | 0.492 0.007 CHEMBL3527009 0.482 0.008 CHEMBL442289 | CHEMBL3527009 | |
| 0.329 | 0.004 | 0.588 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.535 0.002 CHEMBL3527009 0.588 0.002 CHEMBL442289 | CHEMBL442289 | |
| 0.328 | 0.004 | 0.328 | Histone deacetylase stimulant | 0.305 0.004 CHEMBL3527009 0.326 0.004 CHEMBL442289 | ||
| 0.328 | 0.004 | 0.328 | Histone deacetylase SIRT1 stimulant | 0.305 0.004 CHEMBL3527009 0.326 0.004 CHEMBL442289 | ||
| 0.341 | 0.034 | 0.341 | Antimitotic | 0.321 0.039 CHEMBL3527009 0.312 0.041 CHEMBL442289 | ||
| 0.311 | 0.01 | 0.311 | Butyrylcholinesterase inhibitor | 0.263 0.013 CHEMBL3527009 0.259 0.014 CHEMBL442289 | ||
| 0.323 | 0.022 | 0.401 | DNA methylase inhibitor | 0.398 0.011 CHEMBL3527009 0.401 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.305 | 0.006 | 0.338 | Telomerase inhibitor | 0.338 0.005 CHEMBL3527009 0.32 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.343 | 0.052 | 0.555 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.555 0.014 CHEMBL3527009 0.526 0.017 CHEMBL442289 | CHEMBL3527009 | |
| 0.292 | 0.006 | 0.639 | Carbonic anhydrase III inhibitor | 0.6 0.003 CHEMBL3527009 0.639 0.002 CHEMBL442289 | CHEMBL442289 | |
| 0.3 | 0.017 | 0.327 | Amyloid beta precursor protein antagonist | 0.327 0.012 CHEMBL3527009 0.327 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.288 | 0.009 | 0.389 | Carbonic anhydrase XV inhibitor | 0.366 0.005 CHEMBL3527009 0.389 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.391 | 0.123 | 0.479 | DNA polymerase beta inhibitor | 0.479 0.092 CHEMBL3527009 0.475 0.093 CHEMBL442289 | CHEMBL3527009 | |
| 0.279 | 0.013 | 0.364 | 5-Lipoxygenase inhibitor | 0.364 0.006 CHEMBL3527009 0.36 0.007 CHEMBL442289 | CHEMBL3527009 | |
| 0.312 | 0.049 | 0.424 | Transcription factor STAT inhibitor | 0.421 0.015 CHEMBL3527009 0.424 0.015 CHEMBL442289 | CHEMBL442289 | |
| 0.359 | 0.097 | 0.47 | Antibacterial | 0.467 0.051 CHEMBL3527009 0.47 0.05 CHEMBL442289 | CHEMBL442289 | |
| 0.273 | 0.013 | 0.301 | Protein-tyrosine phosphatase 1B inhibitor | 0.299 0.011 CHEMBL3527009 0.301 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.294 | 0.036 | 0.308 | Platelet adhesion inhibitor | 0.308 0.032 CHEMBL3527009 0.308 0.031 CHEMBL442289 | CHEMBL442289 | |
| 0.255 | 0.004 | 0.394 | Xanthine dehydrogenase inhibitor | 0.372 0.003 CHEMBL3527009 0.394 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.258 | 0.008 | 0.258 | Cyclooxygenase 3 inhibitor | 0.238 0.01 CHEMBL3527009 0.243 0.009 CHEMBL442289 | ||
| 0.256 | 0.008 | 0.562 | Carbonic anhydrase VI inhibitor | 0.511 0.003 CHEMBL3527009 0.562 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.287 | 0.054 | 0.37 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.338 0.038 CHEMBL3527009 0.37 0.031 CHEMBL442289 | CHEMBL442289 | |
| 0.301 | 0.07 | 0.317 | 5 Hydroxytryptamine release stimulant | 0.297 0.071 CHEMBL3527009 0.317 0.065 CHEMBL442289 | CHEMBL442289 | |
| 0.231 | 0.004 | 0.231 | Protease activated receptor antagonist | 0.124 0.008 CHEMBL3527009 0.118 0.009 CHEMBL442289 | ||
| 0.234 | 0.009 | 0.303 | Beta glucuronidase inhibitor | 0.269 0.007 CHEMBL3527009 0.303 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.251 | 0.027 | 0.251 | 3C-like protease (Human coronavirus) inhibitor | 0.168 0.076 CHEMBL3527009 0.162 0.084 CHEMBL442289 | ||
| 0.23 | 0.006 | 0.269 | Electron transport complex I inhibitor | 0.269 0.005 CHEMBL3527009 0.234 0.006 CHEMBL442289 | CHEMBL3527009 | |
| 0.226 | 0.009 | 0.251 | Photosensitizer | 0.249 0.006 CHEMBL3527009 0.251 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.218 | 0.004 | 0.295 | Carbonic anhydrase VII inhibitor | 0.271 0.004 CHEMBL3527009 0.295 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.22 | 0.007 | 0.22 | T cell inhibitor | 0.169 0.009 CHEMBL3527009 0.151 0.01 CHEMBL442289 | ||
| 0.253 | 0.042 | 0.413 | Non-steroidal antiinflammatory agent | 0.413 0.012 CHEMBL3527009 0.403 0.013 CHEMBL442289 | CHEMBL3527009 | |
| 0.238 | 0.029 | 0.25 | Cyclooxygenase inhibitor | 0.25 0.026 CHEMBL3527009 0.245 0.027 CHEMBL442289 | CHEMBL3527009 | |
| 0.299 | 0.093 | 0.299 | Calcium channel activator | 0.235 0.166 CHEMBL3527009 0.228 0.175 CHEMBL442289 | ||
| 0.345 | 0.14 | 0.462 | DNA directed DNA polymerase inhibitor | 0.462 0.094 CHEMBL3527009 0.456 0.095 CHEMBL442289 | CHEMBL3527009 | |
| 0.232 | 0.029 | 0.26 | Succinate dehydrogenase inhibitor | 0.26 0.019 CHEMBL3527009 0.243 0.025 CHEMBL442289 | CHEMBL3527009 | |
| 0.211 | 0.016 | 0.255 | CF transmembrane conductance regulator agonist | 0.244 0.007 CHEMBL3527009 0.255 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.199 | 0.005 | 0.199 | Interleukin 5 antagonist | 0.141 0.013 CHEMBL3527009 0.144 0.013 CHEMBL442289 | ||
| 0.201 | 0.008 | 0.24 | GABA C receptor rho-1 antagonist | 0.233 0.005 CHEMBL3527009 0.24 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.22 | 0.028 | 0.252 | Cyclooxygenase 1 inhibitor | 0.25 0.021 CHEMBL3527009 0.252 0.021 CHEMBL442289 | CHEMBL442289 | |
| 0.233 | 0.045 | 0.254 | Insulin sensitizer | 0.254 0.032 CHEMBL3527009 0.252 0.033 CHEMBL442289 | CHEMBL3527009 | |
| 0.256 | 0.069 | 0.332 | Dyrk kinase inhibitor | 0.304 0.051 CHEMBL3527009 0.332 0.042 CHEMBL442289 | CHEMBL442289 | |
| 0.219 | 0.036 | 0.438 | Proto-oncogene tyrosine-protein kinase Yes inhibitor | 0.416 0.006 CHEMBL3527009 0.438 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.195 | 0.014 | 0.271 | Uric acid excretion stimulant | 0.271 0.005 CHEMBL3527009 0.267 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.207 | 0.027 | 0.208 | Mannose-6-phosphate isomerase inhibitor | 0.208 0.026 CHEMBL3527009 0.188 0.037 CHEMBL442289 | CHEMBL3527009 | |
| 0.297 | 0.117 | 0.347 | Immunosuppressant | 0.347 0.089 CHEMBL3527009 0.34 0.092 CHEMBL442289 | CHEMBL3527009 | |
| 0.208 | 0.029 | 0.21 | Cyclooxygenase 2 inhibitor | 0.21 0.028 CHEMBL3527009 0.205 0.029 CHEMBL442289 | CHEMBL3527009 | |
| 0.209 | 0.031 | 0.388 | M18 aspartyl aminopeptidase inhibitor | 0.384 0.005 CHEMBL3527009 0.388 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.27 | 0.092 | 0.408 | Streptokinase A inhibitor | 0.408 0.045 CHEMBL3527009 0.403 0.046 CHEMBL442289 | CHEMBL3527009 | |
| 0.183 | 0.007 | 0.26 | Myeloperoxidase inhibitor | 0.25 0.004 CHEMBL3527009 0.26 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.19 | 0.014 | 0.19 | Phosphodiesterase IV inhibitor | 0.108 0.039 CHEMBL3527009 0.103 0.043 CHEMBL442289 | ||
| 0.179 | 0.004 | 0.338 | D-Ala-D-Ala ligase inhibitor | 0.331 0.002 CHEMBL3527009 0.338 0.002 CHEMBL442289 | CHEMBL442289 | |
| 0.182 | 0.008 | 0.236 | Cyclin B3 inhibitor | 0.236 0.004 CHEMBL3527009 0.235 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.203 | 0.031 | 0.246 | Hemostatic | 0.245 0.023 CHEMBL3527009 0.246 0.022 CHEMBL442289 | CHEMBL442289 | |
| 0.244 | 0.073 | 0.365 | Angiogenesis stimulant | 0.36 0.03 CHEMBL3527009 0.365 0.029 CHEMBL442289 | CHEMBL442289 | |
| 0.186 | 0.015 | 0.186 | Nav1.5 sodium channel blocker | 0.124 0.05 CHEMBL3527009 0.123 0.051 CHEMBL442289 | ||
| 0.202 | 0.035 | 0.226 | Bone formation stimulant | 0.207 0.034 CHEMBL3527009 0.226 0.03 CHEMBL442289 | CHEMBL442289 | |
| 0.237 | 0.071 | 0.237 | Cyclic AMP phosphodiesterase inhibitor | 0.233 0.073 CHEMBL3527009 0.233 0.073 CHEMBL442289 | ||
| 0.171 | 0.006 | 0.171 | Thioredoxin reductase inhibitor | 0.161 0.008 CHEMBL3527009 0.158 0.008 CHEMBL442289 | ||
| 0.177 | 0.013 | 0.262 | Heat shock protein 70 antagonist | 0.249 0.004 CHEMBL3527009 0.262 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.314 | 0.15 | 0.383 | Cyclophilin D inhibitor | 0.383 0.101 CHEMBL3527009 0.378 0.103 CHEMBL442289 | CHEMBL3527009 | |
| 0.232 | 0.069 | 0.32 | Interleukin antagonist | 0.278 0.053 CHEMBL3527009 0.32 0.044 CHEMBL442289 | CHEMBL442289 | |
| 0.272 | 0.11 | 0.312 | Antithrombotic | 0.312 0.081 CHEMBL3527009 0.309 0.082 CHEMBL442289 | CHEMBL3527009 | |
| 0.175 | 0.014 | 0.175 | Phosphodiesterase 4D inhibitor | 0.16 0.017 CHEMBL3527009 0.159 0.017 CHEMBL442289 | ||
| 0.198 | 0.039 | 0.313 | Heat shock protein 90 antagonist | 0.3 0.01 CHEMBL3527009 0.313 0.009 CHEMBL442289 | CHEMBL442289 | |
| 0.168 | 0.01 | 0.192 | Beta tubulin antagonist | 0.192 0.008 CHEMBL3527009 0.192 0.008 CHEMBL442289 | CHEMBL442289 | |
| 0.168 | 0.01 | 0.226 | CDC25A inhibitor | 0.226 0.005 CHEMBL3527009 0.219 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.172 | 0.017 | 0.173 | DNA repair enzyme inhibitor | 0.173 0.016 CHEMBL3527009 0.169 0.018 CHEMBL442289 | CHEMBL3527009 | |
| 0.17 | 0.017 | 0.262 | AMP-activated protein kinase stimulant | 0.261 0.006 CHEMBL3527009 0.262 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.152 | 0.004 | 0.152 | Potassium channel Kv1.3 blocker | 0.09 0.01 CHEMBL3527009 0.078 0.013 CHEMBL442289 | ||
| 0.152 | 0.007 | 0.383 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.333 0.003 CHEMBL3527009 0.383 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.163 | 0.019 | 0.163 | Calcium antagonist | 0.097 0.05 CHEMBL3527009 0.077 0.066 CHEMBL442289 | ||
| 0.153 | 0.013 | 0.257 | Aromatase inhibitor | 0.233 0.007 CHEMBL3527009 0.257 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.159 | 0.019 | 0.199 | Urease inhibitor | 0.188 0.012 CHEMBL3527009 0.199 0.01 CHEMBL442289 | CHEMBL442289 | |
| 0.16 | 0.021 | 0.171 | Sphingomyelinase inhibitor | 0.171 0.017 CHEMBL3527009 0.154 0.023 CHEMBL442289 | CHEMBL3527009 | |
| 0.254 | 0.116 | 0.291 | Thyroid hormone beta antagonist | 0.291 0.093 CHEMBL3527009 0.272 0.104 CHEMBL442289 | CHEMBL3527009 | |
| 0.234 | 0.097 | 0.261 | Transcription factor STAT3 inhibitor | 0.261 0.075 CHEMBL3527009 0.257 0.078 CHEMBL442289 | CHEMBL3527009 | |
| 0.156 | 0.019 | 0.233 | Transcription factor STAT6 inhibitor | 0.222 0.005 CHEMBL3527009 0.233 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.162 | 0.025 | 0.18 | Papain-like protease (SARS coronavirus) inhibitor | 0.169 0.021 CHEMBL3527009 0.18 0.016 CHEMBL442289 | CHEMBL442289 | |
| 0.146 | 0.01 | 0.215 | Alpha tubulin antagonist | 0.214 0.005 CHEMBL3527009 0.215 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.255 | 0.12 | 0.303 | Thyroid hormone antagonist | 0.303 0.092 CHEMBL3527009 0.282 0.103 CHEMBL442289 | CHEMBL3527009 | |
| 0.153 | 0.02 | 0.222 | DOPA decarboxylase inhibitor | 0.212 0.005 CHEMBL3527009 0.222 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.227 | 0.094 | 0.274 | Tyrosine 3 hydroxylase inhibitor | 0.26 0.059 CHEMBL3527009 0.274 0.048 CHEMBL442289 | CHEMBL442289 | |
| 0.15 | 0.017 | 0.163 | Thioredoxin inhibitor | 0.159 0.014 CHEMBL3527009 0.163 0.013 CHEMBL442289 | CHEMBL442289 | |
| 0.148 | 0.016 | 0.351 | Macrophage migration inhibitory factor inhibitor | 0.309 0.004 CHEMBL3527009 0.351 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.135 | 0.004 | 0.135 | Glutamate (mGluR7) antagonist | 0.115 0.005 CHEMBL3527009 0.114 0.005 CHEMBL442289 | ||
| 0.157 | 0.026 | 0.203 | GABA C receptor antagonist | 0.202 0.012 CHEMBL3527009 0.203 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.169 | 0.038 | 0.292 | Aldehyde dehydrogenase inhibitor | 0.262 0.016 CHEMBL3527009 0.292 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.146 | 0.015 | 0.225 | Carbonic anhydrase V inhibitor | 0.212 0.006 CHEMBL3527009 0.225 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.135 | 0.006 | 0.182 | Aryl hydrocarbon receptor antagonist | 0.179 0.004 CHEMBL3527009 0.182 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.149 | 0.02 | 0.22 | Protein kinase C zeta inhibitor | 0.197 0.011 CHEMBL3527009 0.22 0.009 CHEMBL442289 | CHEMBL442289 | |
| 0.144 | 0.014 | 0.287 | HIV-1 integrase (3'-Processing) inhibitor | 0.287 0.005 CHEMBL3527009 0.286 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.142 | 0.013 | 0.288 | HIV-1 integrase (Strand Transfer) inhibitor | 0.288 0.005 CHEMBL3527009 0.283 0.005 CHEMBL442289 | CHEMBL3527009 | |
| 0.198 | 0.072 | 0.198 | Histone acetyltransferase inhibitor | 0.174 0.108 CHEMBL3527009 0.167 0.117 CHEMBL442289 | ||
| 0.143 | 0.017 | 0.407 | Estrogen receptor beta antagonist | 0.317 0.005 CHEMBL3527009 0.407 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.161 | 0.036 | 0.296 | Protein kinase (CK2) alpha inhibitor | 0.291 0.012 CHEMBL3527009 0.296 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.148 | 0.024 | 0.371 | Estrogen antagonist | 0.283 0.007 CHEMBL3527009 0.371 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.137 | 0.014 | 0.199 | Carbonic anhydrase VA inhibitor | 0.188 0.005 CHEMBL3527009 0.199 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.163 | 0.04 | 0.198 | Alkylator | 0.197 0.027 CHEMBL3527009 0.198 0.027 CHEMBL442289 | CHEMBL442289 | |
| 0.173 | 0.054 | 0.238 | Insulin secretagoues | 0.238 0.022 CHEMBL3527009 0.235 0.023 CHEMBL442289 | CHEMBL3527009 | |
| 0.155 | 0.037 | 0.155 | Beta amyloid protein antagonist | |||
| 0.117 | 0.004 | 0.119 | Transcription factor RelA inhibitor | 0.116 0.004 CHEMBL3527009 0.119 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.152 | 0.04 | 0.248 | Topoisomerase I inhibitor | 0.231 0.02 CHEMBL3527009 0.248 0.017 CHEMBL442289 | CHEMBL442289 | |
| 0.129 | 0.023 | 0.129 | CYP2A6 inhibitor | 0.085 0.045 CHEMBL3527009 0.082 0.047 CHEMBL442289 | ||
| 0.114 | 0.008 | 0.226 | Fatty acid synthase inhibitor | 0.214 0.004 CHEMBL3527009 0.226 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.173 | 0.068 | 0.322 | Heat shock protein 90 alpha antagonist | 0.307 0.013 CHEMBL3527009 0.322 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.15 | 0.046 | 0.151 | Antibacterial (Helicobacter pylori) | 0.151 0.045 CHEMBL3527009 0.15 0.046 CHEMBL442289 | CHEMBL3527009 | |
| 0.127 | 0.023 | 0.151 | Interleukin 12 antagonist | 0.139 0.016 CHEMBL3527009 0.151 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.121 | 0.017 | 0.137 | Lipase inhibitor | 0.135 0.013 CHEMBL3527009 0.137 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.12 | 0.018 | 0.262 | Estrogen receptor alpha antagonist | 0.22 0.007 CHEMBL3527009 0.262 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.124 | 0.025 | 0.298 | Histidine decarboxylase inhibitor | 0.273 0.008 CHEMBL3527009 0.298 0.006 CHEMBL442289 | CHEMBL442289 | |
| 0.139 | 0.04 | 0.389 | Chelator | 0.389 0.006 CHEMBL3527009 0.383 0.006 CHEMBL442289 | CHEMBL3527009 | |
| 0.105 | 0.009 | 0.105 | CD45 antagonist | 0.101 0.009 CHEMBL3527009 0.095 0.01 CHEMBL442289 | ||
| 0.166 | 0.069 | 0.166 | Interleukin 6 antagonist | 0.134 0.117 CHEMBL3527009 0.132 0.121 CHEMBL442289 | ||
| 0.114 | 0.02 | 0.114 | Granulocyte macrophage colony stimulating factor agonist | 0.104 0.03 CHEMBL3527009 0.097 0.04 CHEMBL442289 | ||
| 0.168 | 0.075 | 0.272 | Mcl-1 antagonist | 0.272 0.029 CHEMBL3527009 0.268 0.03 CHEMBL442289 | CHEMBL3527009 | |
| 0.185 | 0.092 | 0.258 | Neurotrophic factor enhancer | 0.248 0.039 CHEMBL3527009 0.258 0.034 CHEMBL442289 | CHEMBL442289 | |
| 0.124 | 0.032 | 0.301 | Alcohol dehydrogenase inhibitor | 0.269 0.006 CHEMBL3527009 0.301 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.181 | 0.089 | 0.181 | I kappa B kinase epsilon inhibitor | 0.165 0.104 CHEMBL3527009 0.163 0.106 CHEMBL442289 | ||
| 0.096 | 0.005 | 0.096 | GABA B receptor antagonist | 0.073 0.008 CHEMBL3527009 0.075 0.007 CHEMBL442289 | ||
| 0.144 | 0.057 | 0.197 | Toll-Like receptor 2 antagonist | 0.19 0.029 CHEMBL3527009 0.197 0.025 CHEMBL442289 | CHEMBL442289 | |
| 0.183 | 0.097 | 0.183 | 5 Hydroxytryptamine 3E antagonist | |||
| 0.207 | 0.123 | 0.207 | 5 Hydroxytryptamine 1E antagonist | 0.194 0.138 CHEMBL3527009 0.203 0.128 CHEMBL442289 | ||
| 0.126 | 0.042 | 0.141 | Mediator release inhibitor | 0.134 0.037 CHEMBL3527009 0.141 0.033 CHEMBL442289 | CHEMBL442289 | |
| 0.122 | 0.038 | 0.178 | Antineoplastic antibiotic | 0.178 0.025 CHEMBL3527009 0.176 0.025 CHEMBL442289 | CHEMBL3527009 | |
| 0.088 | 0.005 | 0.088 | Ryanodine receptor antagonist | 0.085 0.006 CHEMBL3527009 0.084 0.007 CHEMBL442289 | ||
| 0.16 | 0.08 | 0.177 | Neurotensin receptor agonist | 0.169 0.064 CHEMBL3527009 0.177 0.053 CHEMBL442289 | CHEMBL442289 | |
| 0.158 | 0.079 | 0.175 | Arachidonic acid antagonist | 0.175 0.059 CHEMBL3527009 0.164 0.073 CHEMBL442289 | CHEMBL3527009 | |
| 0.096 | 0.017 | 0.152 | CDC25B inhibitor | 0.152 0.006 CHEMBL3527009 0.15 0.006 CHEMBL442289 | CHEMBL3527009 | |
| 0.105 | 0.028 | 0.105 | mTOR complex 2 inhibitor | 0.091 0.045 CHEMBL3527009 0.087 0.052 CHEMBL442289 | ||
| 0.12 | 0.043 | 0.142 | Toll-Like receptor 4 antagonist | 0.136 0.03 CHEMBL3527009 0.142 0.026 CHEMBL442289 | CHEMBL442289 | |
| 0.103 | 0.026 | 0.103 | Phosphodiesterase V inhibitor | |||
| 0.102 | 0.029 | 0.158 | Keratolytic | 0.14 0.016 CHEMBL3527009 0.158 0.013 CHEMBL442289 | CHEMBL442289 | |
| 0.141 | 0.069 | 0.142 | Ca2+-transporting ATPase inhibitor | 0.142 0.066 CHEMBL3527009 0.138 0.082 CHEMBL442289 | CHEMBL3527009 | |
| 0.222 | 0.152 | 0.285 | Vasodilator, peripheral | 0.285 0.105 CHEMBL3527009 0.274 0.111 CHEMBL442289 | CHEMBL3527009 | |
| 0.139 | 0.07 | 0.139 | Toll-Like receptor 9 antagonist | |||
| 0.08 | 0.011 | 0.08 | Glucose-6-phosphate translocase inhibitor | 0.071 0.015 CHEMBL3527009 0.073 0.014 CHEMBL442289 | ||
| 0.097 | 0.028 | 0.097 | Phosphodiesterase 5A inhibitor | |||
| 0.081 | 0.016 | 0.15 | Carbonic anhydrase XIV inhibitor | 0.131 0.006 CHEMBL3527009 0.15 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.144 | 0.081 | 0.15 | Phospholipase A2 inhibitor | 0.15 0.074 CHEMBL3527009 0.149 0.075 CHEMBL442289 | CHEMBL3527009 | |
| 0.092 | 0.031 | 0.092 | Adenosine A3 receptor antagonist | 0.091 0.031 CHEMBL3527009 0.087 0.035 CHEMBL442289 | ||
| 0.089 | 0.029 | 0.089 | Phosphodiesterase VI inhibitor | 0.081 0.04 CHEMBL3527009 0.08 0.041 CHEMBL442289 | ||
| 0.079 | 0.019 | 0.079 | Cyclin D1 inhibitor | 0.076 0.022 CHEMBL3527009 0.075 0.023 CHEMBL442289 | ||
| 0.073 | 0.015 | 0.279 | Estradiol 17 beta-dehydrogenase inhibitor | 0.238 0.004 CHEMBL3527009 0.279 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.083 | 0.024 | 0.113 | Carbonic anhydrase XII inhibitor | 0.104 0.019 CHEMBL3527009 0.113 0.017 CHEMBL442289 | CHEMBL442289 | |
| 0.111 | 0.055 | 0.205 | Protein kinase (CK2) inhibitor | 0.205 0.018 CHEMBL3527009 0.204 0.018 CHEMBL442289 | CHEMBL3527009 | |
| 0.099 | 0.044 | 0.099 | Glutamate release inhibitor | |||
| 0.087 | 0.033 | 0.145 | HIV-1 integrase inhibitor | 0.145 0.009 CHEMBL3527009 0.142 0.01 CHEMBL442289 | CHEMBL3527009 | |
| 0.076 | 0.024 | 0.271 | Estrogen agonist | 0.187 0.009 CHEMBL3527009 0.271 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.112 | 0.062 | 0.138 | Mucolytic | 0.138 0.04 CHEMBL3527009 0.135 0.042 CHEMBL442289 | CHEMBL3527009 | |
| 0.106 | 0.056 | 0.106 | Cyclin-dependent kinase 9 inhibitor | |||
| 0.097 | 0.048 | 0.105 | Ornithine decarboxylase inhibitor | 0.105 0.039 CHEMBL3527009 0.103 0.042 CHEMBL442289 | CHEMBL3527009 | |
| 0.108 | 0.06 | 0.141 | Expectorant | 0.141 0.039 CHEMBL3527009 0.138 0.04 CHEMBL442289 | CHEMBL3527009 | |
| 0.202 | 0.154 | 0.216 | Insulysin inhibitor | 0.206 0.148 CHEMBL3527009 0.216 0.134 CHEMBL442289 | CHEMBL442289 | |
| 0.24 | 0.194 | 0.272 | Transcription factor inhibitor | 0.272 0.172 CHEMBL3527009 0.265 0.176 CHEMBL442289 | CHEMBL3527009 | |
| 0.089 | 0.043 | 0.089 | Caspase 7 inhibitor | 0.085 0.051 CHEMBL3527009 0.081 0.06 CHEMBL442289 | ||
| 0.156 | 0.111 | 0.17 | Psychostimulant | 0.169 0.1 CHEMBL3527009 0.17 0.1 CHEMBL442289 | CHEMBL442289 | |
| 0.11 | 0.065 | 0.11 | Acetylcholine release stimulant | |||
| 0.115 | 0.07 | 0.16 | Cholesterol synthesis inhibitor | 0.154 0.042 CHEMBL3527009 0.16 0.04 CHEMBL442289 | CHEMBL442289 | |
| 0.074 | 0.03 | 0.113 | Neuraminidase inhibitor | 0.11 0.012 CHEMBL3527009 0.113 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.077 | 0.034 | 0.104 | Leukotriene antagonist | 0.104 0.02 CHEMBL3527009 0.098 0.023 CHEMBL442289 | CHEMBL3527009 | |
| 0.118 | 0.076 | 0.118 | Sphingosine 1-phosphate receptor 4 antagonist | |||
| 0.137 | 0.097 | 0.165 | Interferon gamma antagonist | 0.161 0.065 CHEMBL3527009 0.165 0.062 CHEMBL442289 | CHEMBL442289 | |
| 0.103 | 0.063 | 0.103 | Alpha 2c adrenoreceptor antagonist | |||
| 0.096 | 0.056 | 0.128 | ABCA1 expression enhancer | 0.128 0.025 CHEMBL3527009 0.127 0.026 CHEMBL442289 | CHEMBL3527009 | |
| 0.11 | 0.071 | 0.128 | TRPA1 agonist | 0.12 0.058 CHEMBL3527009 0.128 0.05 CHEMBL442289 | CHEMBL442289 | |
| 0.058 | 0.019 | 0.058 | Leukocyte elastase inhibitor | 0.04 0.034 CHEMBL3527009 | ||
| 0.088 | 0.05 | 0.088 | Inducible nitric-oxide synthase inhibitor | |||
| 0.26 | 0.222 | 0.26 | MAP kinase 1 inhibitor | 0.247 0.237 CHEMBL3527009 | ||
| 0.071 | 0.034 | 0.114 | Neuraminidase (influenza) inhibitor | 0.107 0.014 CHEMBL3527009 0.114 0.013 CHEMBL442289 | CHEMBL442289 | |
| 0.09 | 0.055 | 0.153 | Androgen antagonist | 0.144 0.024 CHEMBL3527009 0.153 0.022 CHEMBL442289 | CHEMBL442289 | |
| 0.064 | 0.032 | 0.088 | Carbonic anhydrase VB inhibitor | 0.079 0.023 CHEMBL3527009 0.088 0.019 CHEMBL442289 | CHEMBL442289 | |
| 0.054 | 0.024 | 0.054 | Cholesterol esterase inhibitor | 0.053 0.026 CHEMBL3527009 0.047 0.034 CHEMBL442289 | ||
| 0.052 | 0.023 | 0.052 | Benzodiazepine antagonist | |||
| 0.079 | 0.051 | 0.093 | Na+ K+ transporting ATPase inhibitor | 0.093 0.038 CHEMBL3527009 0.093 0.038 CHEMBL442289 | CHEMBL442289 | |
| 0.039 | 0.012 | 0.067 | Estrogen-related receptor beta antagonist | 0.055 0.005 CHEMBL3527009 0.067 0.004 CHEMBL442289 | CHEMBL442289 | |
| 0.145 | 0.119 | 0.145 | Anesthetic general | |||
| 0.102 | 0.078 | 0.102 | Interleukin 1b antagonist | |||
| 0.064 | 0.04 | 0.064 | Phosphodiesterase 1C inhibitor | |||
| 0.083 | 0.059 | 0.097 | 3C-Like protease (SARS coronavirus) inhibitor | 0.097 0.036 CHEMBL3527009 0.096 0.038 CHEMBL442289 | CHEMBL3527009 | |
| 0.043 | 0.02 | 0.068 | Arginase inhibitor | 0.066 0.009 CHEMBL3527009 0.068 0.008 CHEMBL442289 | CHEMBL442289 | |
| 0.105 | 0.082 | 0.105 | Microtubule formation inhibitor | 0.105 0.082 CHEMBL3527009 0.099 0.092 CHEMBL442289 | ||
| 0.057 | 0.036 | 0.09 | Cyclin B2 inhibitor | 0.088 0.012 CHEMBL3527009 0.09 0.011 CHEMBL442289 | CHEMBL442289 | |
| 0.164 | 0.143 | 0.196 | Immunostimulant | 0.186 0.129 CHEMBL3527009 0.196 0.123 CHEMBL442289 | CHEMBL442289 | |
| 0.103 | 0.083 | 0.141 | Proteasome inhibitor | 0.139 0.053 CHEMBL3527009 0.141 0.052 CHEMBL442289 | CHEMBL442289 | |
| 0.195 | 0.175 | 0.233 | Angiogenesis inhibitor | 0.233 0.136 CHEMBL3527009 0.23 0.138 CHEMBL442289 | CHEMBL3527009 | |
| 0.055 | 0.035 | 0.072 | Leukotriene B4 antagonist | 0.072 0.019 CHEMBL3527009 0.069 0.02 CHEMBL442289 | CHEMBL3527009 | |
| 0.032 | 0.012 | 0.032 | Dopamine autoreceptor agonist | |||
| 0.061 | 0.042 | 0.093 | Cyclin B1 inhibitor | 0.091 0.014 CHEMBL3527009 0.093 0.014 CHEMBL442289 | CHEMBL442289 | |
| 0.038 | 0.02 | 0.038 | ATM kinase inhibitor | |||
| 0.061 | 0.043 | 0.061 | Transcription factor AP-1 inhibitor | 0.06 0.045 CHEMBL3527009 0.059 0.047 CHEMBL442289 | ||
| 0.065 | 0.048 | 0.094 | Leukotriene synthesis inhibitor | 0.094 0.03 CHEMBL3527009 0.094 0.03 CHEMBL442289 | CHEMBL442289 | |
| 0.056 | 0.039 | 0.059 | Leukotriene C antagonist | 0.059 0.032 CHEMBL3527009 0.057 0.036 CHEMBL442289 | CHEMBL3527009 | |
| 0.093 | 0.076 | 0.093 | Glutamate (mGluR7) agonist | |||
| 0.095 | 0.079 | 0.137 | DNA intercalator | 0.136 0.049 CHEMBL3527009 0.137 0.049 CHEMBL442289 | CHEMBL442289 | |
| 0.125 | 0.111 | 0.169 | Hexokinase inhibitor | 0.166 0.061 CHEMBL3527009 0.169 0.058 CHEMBL442289 | CHEMBL442289 | |
| 0.085 | 0.071 | 0.175 | HIV-1 integrase (Overall Integration) inhibitor | 0.175 0.018 CHEMBL3527009 0.152 0.024 CHEMBL442289 | CHEMBL3527009 | |
| 0.083 | 0.07 | 0.083 | Phosphodiesterase I inhibitor | |||
| 0.039 | 0.025 | 0.039 | Vanilloid 3 antagonist | 0.036 0.035 CHEMBL3527009 | ||
| 0.062 | 0.049 | 0.062 | Calcium channel P-type blocker | |||
| 0.033 | 0.022 | 0.059 | Protein kinase (CK2) beta inhibitor | 0.057 0.005 CHEMBL3527009 0.059 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.039 | 0.029 | 0.078 | Dopamine D5 agonist | 0.072 0.008 CHEMBL3527009 0.078 0.007 CHEMBL442289 | CHEMBL442289 | |
| 0.025 | 0.014 | 0.135 | Estradiol 17 beta-dehydrogenase 1 inhibitor | 0.107 0.004 CHEMBL3527009 0.135 0.003 CHEMBL442289 | CHEMBL442289 | |
| 0.039 | 0.03 | 0.039 | DNA-dependent protein kinase inhibitor | |||
| 0.014 | 0.006 | 0.014 | Melatonin 2 antagonist | |||
| 0.117 | 0.11 | 0.157 | Farnesoid X receptor antagonist | 0.144 0.06 CHEMBL3527009 0.157 0.045 CHEMBL442289 | CHEMBL442289 | |
| 0.267 | 0.26 | 0.267 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | |||
| 0.022 | 0.015 | 0.024 | Estrone sulfatase inhibitor | 0.022 0.015 CHEMBL3527009 0.024 0.013 CHEMBL442289 | CHEMBL442289 | |
| 0.037 | 0.031 | 0.038 | Retinoic acid alpha receptor agonist | 0.038 0.029 CHEMBL3527009 | CHEMBL3527009 | |
| 0.032 | 0.026 | 0.032 | Melatonin receptor 1A agonist | |||
| 0.08 | 0.074 | 0.093 | NADH dehydrogenase inhibitor | 0.093 0.052 CHEMBL3527009 0.085 0.065 CHEMBL442289 | CHEMBL3527009 | |
| 0.031 | 0.026 | 0.052 | Catechol O-methyltransferase inhibitor | 0.052 0.008 CHEMBL3527009 0.05 0.009 CHEMBL442289 | CHEMBL3527009 | |
| 0.06 | 0.056 | 0.063 | Beta 3 adrenoreceptor antagonist | 0.061 0.054 CHEMBL3527009 0.063 0.047 CHEMBL442289 | CHEMBL442289 | |
| 0.041 | 0.038 | 0.041 | Fructose-1,6-bisphosphatase inhibitor | 0.041 0.038 CHEMBL3527009 0.04 0.039 CHEMBL442289 | ||
| 0.022 | 0.02 | 0.022 | Fructose-1,6-bisphosphatase 1 inhibitor | 0.022 0.019 CHEMBL3527009 0.022 0.02 CHEMBL442289 | ||
| 0.064 | 0.062 | 0.064 | Cathepsin G inhibitor | |||
| 0.048 | 0.047 | 0.048 | GABA receptor antagonist | |||
| 0.137 | 0.136 | 0.163 | Phospholipase C inhibitor | 0.158 0.091 CHEMBL3527009 0.163 0.082 CHEMBL442289 | CHEMBL442289 | |
| 0.073 | 0.074 | 0.113 | Glutathione S-transferase inhibitor | 0.113 0.027 CHEMBL3527009 0.108 0.03 CHEMBL442289 | CHEMBL3527009 | |
| 0.078 | 0.078 | 0.123 | Potassium channel (Ca-activated) activator | 0.123 0.039 CHEMBL3527009 0.118 0.042 CHEMBL442289 | CHEMBL3527009 | |
| 0.017 | 0.019 | 0.02 | Antibiotic Anthracycline-like | 0.02 0.01 CHEMBL3527009 0.02 0.012 CHEMBL442289 | CHEMBL442289 | |
| 0.026 | 0.03 | 0.136 | Estrogen receptor alpha agonist | 0.096 0.009 CHEMBL3527009 0.136 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.047 | 0.051 | 0.078 | Cyclin B inhibitor | 0.076 0.017 CHEMBL3527009 0.078 0.016 CHEMBL442289 | CHEMBL442289 | |
| 0.022 | 0.027 | 0.18 | Estrogen receptor beta agonist | 0.133 0.008 CHEMBL3527009 0.18 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.084 | 0.09 | 0.108 | Anabolic | 0.106 0.054 CHEMBL3527009 0.108 0.052 CHEMBL442289 | CHEMBL442289 | |
| 0.042 | 0.049 | 0.057 | Topoisomerase II beta inhibitor | 0.053 0.028 CHEMBL3527009 0.057 0.025 CHEMBL442289 | CHEMBL442289 | |
| 0.043 | 0.051 | 0.059 | Squalene epoxidase inhibitor | 0.059 0.021 CHEMBL3527009 0.059 0.021 CHEMBL442289 | CHEMBL442289 | |
| 0.026 | 0.034 | 0.046 | ATP citrate lysase inhibitor | 0.043 0.011 CHEMBL3527009 0.046 0.009 CHEMBL442289 | CHEMBL442289 | |
| 0.075 | 0.084 | 0.092 | Estrogen-related receptor beta agonist | 0.088 0.046 CHEMBL3527009 0.092 0.036 CHEMBL442289 | CHEMBL442289 | |
| 0.043 | 0.052 | 0.103 | Maillard reaction inhibitor | 0.103 0.015 CHEMBL3527009 0.101 0.016 CHEMBL442289 | CHEMBL3527009 | |
| 0.043 | 0.056 | 0.075 | Protein kinase C eta inhibitor | 0.061 0.034 CHEMBL3527009 0.075 0.026 CHEMBL442289 | CHEMBL442289 | |
| 0.046 | 0.061 | 0.059 | Carbonic anhydrase inhibitor | 0.055 0.05 CHEMBL3527009 0.059 0.047 CHEMBL442289 | CHEMBL442289 | |
| 0.076 | 0.091 | 0.084 | Bronchodilator | 0.084 0.081 CHEMBL442289 | CHEMBL442289 | |
| 0.117 | 0.133 | 0.136 | Adenylate cyclase stimulant | 0.136 0.089 CHEMBL3527009 0.135 0.09 CHEMBL442289 | CHEMBL3527009 | |
| 0.036 | 0.053 | 0.044 | Neuraminidase (Influenza A) inhibitor | 0.044 0.035 CHEMBL3527009 0.043 0.037 CHEMBL442289 | CHEMBL3527009 | |
| 0.023 | 0.04 | 0.035 | Estradiol 17 beta-dehydrogenase 3 inhibitor | 0.03 0.024 CHEMBL3527009 0.035 0.019 CHEMBL442289 | CHEMBL442289 | |
| 0.049 | 0.067 | 0.07 | Sphingosine kinase inhibitor | 0.07 0.024 CHEMBL3527009 0.07 0.025 CHEMBL442289 | CHEMBL442289 | |
| 0.022 | 0.043 | 0.11 | Estradiol 17 beta-dehydrogenase 2 inhibitor | 0.082 0.006 CHEMBL3527009 0.11 0.005 CHEMBL442289 | CHEMBL442289 | |
| 0.08 | 0.102 | 0.09 | Bile acid receptor antagonist | 0.088 0.079 CHEMBL3527009 0.09 0.073 CHEMBL442289 | CHEMBL442289 | |
| 0.04 | 0.062 | 0.069 | Alcohol oxidase inhibitor | 0.06 0.035 CHEMBL3527009 0.069 0.029 CHEMBL442289 | CHEMBL442289 | |
| 0.028 | 0.051 | 0.044 | Carbonic anhydrase IV inhibitor | 0.044 0.029 CHEMBL3527009 0.044 0.029 CHEMBL442289 | CHEMBL442289 | |
| 0.022 | 0.045 | 0.035 | Estrogen-related receptor alpha antagonist | 0.035 0.021 CHEMBL442289 | CHEMBL442289 | |
| 0.091 | 0.115 | 0.104 | Alpha-N-acetylglucosaminidase inhibitor | 0.104 0.096 CHEMBL3527009 | CHEMBL3527009 | |
| 0.033 | 0.061 | 0.041 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.041 0.03 CHEMBL3527009 | CHEMBL3527009 | |
| 0.074 | 0.102 | 0.089 | UDP-glucose 4-epimerase inhibitor | 0.089 0.075 CHEMBL3527009 | CHEMBL3527009 | |
| 0.029 | 0.059 | 0.056 | Adenosine deaminase inhibitor | 0.056 0.024 CHEMBL3527009 0.054 0.026 CHEMBL442289 | CHEMBL3527009 | |
| 0.104 | 0.135 | 0.118 | Vanilloid 1 agonist | 0.118 0.094 CHEMBL3527009 0.116 0.098 CHEMBL442289 | CHEMBL3527009 | |
| 0.052 | 0.084 | 0.085 | Potassium channel large-conductance Ca-activated activator | 0.085 0.032 CHEMBL3527009 0.081 0.035 CHEMBL442289 | CHEMBL3527009 | |
| 0.088 | 0.121 | 0.156 | Glycogen synthase kinase-3 alpha inhibitor | 0.15 0.067 CHEMBL3527009 0.156 0.063 CHEMBL442289 | CHEMBL442289 | |
| 0.044 | 0.08 | 0.064 | Dopamine D1 antagonist | 0.061 0.049 CHEMBL3527009 0.064 0.045 CHEMBL442289 | CHEMBL442289 | |
| 0.067 | 0.106 | 0.113 | Prolactin inhibitor | 0.102 0.053 CHEMBL3527009 0.113 0.043 CHEMBL442289 | CHEMBL442289 | |
| 0.049 | 0.092 | 0.071 | Glutamate decarboxylase inhibitor | 0.066 0.06 CHEMBL3527009 0.071 0.053 CHEMBL442289 | CHEMBL442289 | |
| 0.036 | 0.081 | 0.069 | CXC chemokine 1 receptor antagonist | 0.069 0.014 CHEMBL3527009 0.068 0.014 CHEMBL442289 | CHEMBL3527009 | |
| 0.042 | 0.091 | 0.055 | Purinergic P2X1 antagonist | 0.055 0.052 CHEMBL3527009 | CHEMBL3527009 | |
| 0.034 | 0.084 | 0.067 | Phosphatidylinositol 3-kinase gamma inhibitor | 0.062 0.03 CHEMBL3527009 0.067 0.026 CHEMBL442289 | CHEMBL442289 | |
| 0.042 | 0.102 | 0.095 | Heat shock protein 90 beta antagonist | 0.092 0.014 CHEMBL3527009 0.095 0.013 CHEMBL442289 | CHEMBL442289 | |
| 0.03 | 0.094 | 0.048 | DNA gyrase subunit A inhibitor | 0.048 0.02 CHEMBL3527009 0.047 0.021 CHEMBL442289 | CHEMBL3527009 | |
| 0.024 | 0.105 | 0.072 | CDK4/cyclin D1 inhibitor | 0.072 0.029 CHEMBL3527009 0.07 0.031 CHEMBL442289 | CHEMBL3527009 | |
| 0.113 | 0.194 | 0.135 | ATPase inhibitor | 0.135 0.131 CHEMBL3527009 0.135 0.13 CHEMBL442289 | CHEMBL442289 | |
| 0.029 | 0.12 | 0.055 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.049 0.045 CHEMBL3527009 0.055 0.036 CHEMBL442289 | CHEMBL442289 | |
| 0.019 | 0.118 | 0.046 | Phosphatidylinositol 3-kinase alpha inhibitor | 0.046 0.04 CHEMBL442289 | CHEMBL442289 | |
| 0.129 | 0.229 | 0.261 | MAP-kinase-activated kinase 5 inhibitor | 0.25 0.059 CHEMBL3527009 0.261 0.053 CHEMBL442289 | CHEMBL442289 | |
| 0.009 | 0.12 | 0.015 | Antibiotic Tetracycline-like | 0.015 0.013 CHEMBL3527009 | CHEMBL3527009 | |
| 0.132 | 0.246 | 0.187 | DNA synthesis inhibitor | 0.187 0.143 CHEMBL3527009 0.183 0.15 CHEMBL442289 | CHEMBL3527009 | |
| 0.008 | 0.127 | 0.022 | Dopamine D1 agonist | 0.022 0.018 CHEMBL3527009 0.022 0.017 CHEMBL442289 | CHEMBL442289 | |
| 0.046 | 0.17 | 0.086 | Pim-1 kinase inhibitor | 0.085 0.073 CHEMBL3527009 0.086 0.072 CHEMBL442289 | CHEMBL442289 | |
| 0.049 | 0.216 | 0.117 | DNA polymerase I inhibitor | 0.109 0.077 CHEMBL3527009 0.117 0.071 CHEMBL442289 | CHEMBL442289 | |
| 0.1 | 0.273 | 0.147 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.145 0.142 CHEMBL3527009 0.147 0.138 CHEMBL442289 | CHEMBL442289 | |
| 0.036 | 0.215 | 0.081 | CDK2/cyclin A inhibitor | 0.081 0.079 CHEMBL442289 | CHEMBL442289 | |
| 0.121 | 0.33 | 0.217 | Sodium/bile acid cotransporter inhibitor | 0.196 0.193 CHEMBL3527009 0.217 0.165 CHEMBL442289 | CHEMBL442289 | |
| 0.141 | 0.422 | 0.297 | Calcium channel L-type activator | 0.297 0.16 CHEMBL442289 | CHEMBL442289 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |