Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8250.0040.848Aldehyde oxidase inhibitor

0.848 0.004 CHEMBL4525772

0.693 0.009 CHEMBL4525777

0.698 0.008 CHEMBL4525778

0.772 0.005 CHEMBL3526632

0.744 0.005 CHEMBL3526715

0.553 0.025 CHEMBL1688

0.393 0.048 CHEMBL3526874

0.733 0.006 CHEMBL845

0.499 0.033 CHEMBL4525779

0.508 0.032 CHEMBL4525780

0.361 0.053 CHEMBL3526631

CHEMBL4525772
0.6580.0040.658Dopamine D4 antagonist

0.349 0.005 CHEMBL4525772

0.403 0.005 CHEMBL4525777

0.397 0.005 CHEMBL4525778

0.466 0.004 CHEMBL3526632

0.395 0.005 CHEMBL3526715

0.263 0.009 CHEMBL1688

0.118 0.022 CHEMBL3526874

0.369 0.005 CHEMBL845

0.345 0.005 CHEMBL4525779

0.307 0.007 CHEMBL4525780

0.097 0.027 CHEMBL3526631

0.5720.0110.593GABA C receptor rho-3 antagonist

0.593 0.008 CHEMBL4525772

0.565 0.012 CHEMBL4525777

0.565 0.012 CHEMBL4525778

0.524 0.02 CHEMBL3526632

0.537 0.017 CHEMBL3526715

0.437 0.046 CHEMBL1688

0.501 0.026 CHEMBL3526874

0.547 0.015 CHEMBL845

0.305 0.112 CHEMBL4525779

0.305 0.112 CHEMBL4525780

0.531 0.018 CHEMBL3526631

CHEMBL4525772
0.5290.0020.5295 Hydroxytryptamine 3B antagonist

0.395 0.002 CHEMBL4525772

0.294 0.003 CHEMBL4525777

0.451 0.002 CHEMBL4525778

0.201 0.003 CHEMBL3526632

0.151 0.004 CHEMBL3526715

0.087 0.006 CHEMBL1688

0.036 0.025 CHEMBL3526874

0.311 0.003 CHEMBL845

0.103 0.005 CHEMBL4525779

0.116 0.004 CHEMBL4525780

0.5410.0180.551Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.471 0.048 CHEMBL4525772

0.535 0.02 CHEMBL4525777

0.502 0.033 CHEMBL4525778

0.445 0.065 CHEMBL3526632

0.431 0.075 CHEMBL3526715

0.441 0.068 CHEMBL1688

0.504 0.032 CHEMBL3526874

0.551 0.016 CHEMBL845

0.365 0.135 CHEMBL4525779

0.322 0.184 CHEMBL4525780

0.462 0.053 CHEMBL3526631

CHEMBL845
0.5080.0260.5185 Hydroxytryptamine release stimulant

0.357 0.055 CHEMBL4525772

0.461 0.034 CHEMBL4525777

0.366 0.053 CHEMBL4525778

0.307 0.068 CHEMBL3526632

0.44 0.038 CHEMBL3526715

0.214 0.11 CHEMBL1688

0.264 0.082 CHEMBL3526874

0.518 0.024 CHEMBL845

0.207 0.116 CHEMBL4525779

0.165 0.159 CHEMBL4525780

0.37 0.052 CHEMBL3526631

CHEMBL845
0.4820.0070.5265 Hydroxytryptamine 2 antagonist

0.317 0.015 CHEMBL4525772

0.278 0.018 CHEMBL4525777

0.392 0.01 CHEMBL4525778

0.349 0.013 CHEMBL3526632

0.221 0.026 CHEMBL3526715

0.526 0.005 CHEMBL1688

0.098 0.073 CHEMBL3526874

0.402 0.01 CHEMBL845

0.251 0.021 CHEMBL4525779

0.149 0.045 CHEMBL4525780

CHEMBL1688
0.4780.0080.4785 Hydroxytryptamine antagonist

0.297 0.019 CHEMBL4525772

0.341 0.015 CHEMBL4525777

0.358 0.014 CHEMBL4525778

0.266 0.023 CHEMBL3526632

0.184 0.038 CHEMBL3526715

0.41 0.011 CHEMBL1688

0.093 0.085 CHEMBL3526874

0.356 0.014 CHEMBL845

0.233 0.027 CHEMBL4525779

0.118 0.066 CHEMBL4525780

0.4810.0230.491MAP kinase kinase 6 inhibitor

0.426 0.044 CHEMBL4525772

0.47 0.027 CHEMBL4525777

0.435 0.04 CHEMBL4525778

0.438 0.039 CHEMBL3526632

0.414 0.05 CHEMBL3526715

0.395 0.062 CHEMBL1688

0.385 0.067 CHEMBL3526874

0.491 0.02 CHEMBL845

0.398 0.06 CHEMBL4525779

0.357 0.087 CHEMBL4525780

0.365 0.081 CHEMBL3526631

CHEMBL845
0.4560.0030.4565 Hydroxytryptamine 3 antagonist

0.419 0.003 CHEMBL4525772

0.283 0.004 CHEMBL4525777

0.368 0.004 CHEMBL4525778

0.161 0.008 CHEMBL3526632

0.121 0.013 CHEMBL3526715

0.269 0.004 CHEMBL1688

0.324 0.004 CHEMBL845

0.214 0.005 CHEMBL4525779

0.114 0.014 CHEMBL4525780

0.4590.0120.524Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.344 0.039 CHEMBL4525772

0.415 0.018 CHEMBL4525777

0.424 0.017 CHEMBL4525778

0.428 0.016 CHEMBL3526632

0.524 0.005 CHEMBL3526715

0.32 0.051 CHEMBL1688

0.366 0.03 CHEMBL3526874

0.453 0.013 CHEMBL845

0.249 0.107 CHEMBL3526422

0.241 0.115 CHEMBL3526420

0.248 0.108 CHEMBL3526421

0.284 0.076 CHEMBL3526423

0.343 0.039 CHEMBL4525779

0.351 0.036 CHEMBL4525780

0.455 0.012 CHEMBL3526631

CHEMBL3526715
0.4450.0040.4455 Hydroxytryptamine 1E antagonist

0.347 0.01 CHEMBL4525772

0.373 0.006 CHEMBL4525777

0.394 0.005 CHEMBL4525778

0.365 0.007 CHEMBL3526632

0.372 0.006 CHEMBL3526715

0.306 0.026 CHEMBL1688

0.342 0.012 CHEMBL3526874

0.37 0.007 CHEMBL845

0.293 0.034 CHEMBL4525779

0.308 0.025 CHEMBL4525780

0.317 0.02 CHEMBL3526631

0.4390.0020.439Histamine H4 receptor antagonist

0.343 0.002 CHEMBL4525772

0.274 0.003 CHEMBL4525777

0.273 0.003 CHEMBL4525778

0.121 0.004 CHEMBL3526632

0.106 0.005 CHEMBL3526715

0.1 0.005 CHEMBL1688

0.159 0.004 CHEMBL3526874

0.308 0.002 CHEMBL845

0.265 0.003 CHEMBL4525779

0.253 0.003 CHEMBL4525780

0.177 0.004 CHEMBL3526631

0.4410.0060.4485 Hydroxytryptamine 2A antagonist

0.279 0.013 CHEMBL4525772

0.243 0.015 CHEMBL4525777

0.354 0.009 CHEMBL4525778

0.285 0.012 CHEMBL3526632

0.176 0.023 CHEMBL3526715

0.448 0.005 CHEMBL1688

0.069 0.067 CHEMBL3526874

0.352 0.009 CHEMBL845

0.226 0.017 CHEMBL4525779

0.127 0.035 CHEMBL4525780

CHEMBL1688
0.4350.0070.4975 Hydroxytryptamine 2B antagonist

0.29 0.015 CHEMBL4525772

0.258 0.018 CHEMBL4525777

0.384 0.009 CHEMBL4525778

0.36 0.01 CHEMBL3526632

0.212 0.024 CHEMBL3526715

0.497 0.005 CHEMBL1688

0.364 0.01 CHEMBL845

0.156 0.038 CHEMBL4525779

0.134 0.049 CHEMBL4525780

CHEMBL1688
0.4310.0040.441Toll-Like receptor 9 antagonist

0.441 0.004 CHEMBL4525772

0.322 0.01 CHEMBL4525777

0.327 0.009 CHEMBL4525778

0.364 0.005 CHEMBL3526632

0.312 0.011 CHEMBL3526715

0.181 0.045 CHEMBL1688

0.38 0.005 CHEMBL3526874

0.359 0.006 CHEMBL845

0.376 0.005 CHEMBL4525779

0.268 0.017 CHEMBL4525780

0.258 0.019 CHEMBL3526631

CHEMBL4525772
0.4260.0040.636Dopamine D1 antagonist

0.285 0.006 CHEMBL4525772

0.234 0.009 CHEMBL4525777

0.256 0.008 CHEMBL4525778

0.636 0.003 CHEMBL3526632

0.468 0.004 CHEMBL3526715

0.504 0.003 CHEMBL1688

0.261 0.007 CHEMBL845

0.256 0.008 CHEMBL4525779

0.174 0.012 CHEMBL4525780

CHEMBL3526632
0.4190.0190.419Anticonvulsant

0.263 0.052 CHEMBL4525772

0.199 0.083 CHEMBL4525777

0.209 0.076 CHEMBL4525778

0.154 0.124 CHEMBL3526632

0.144 0.136 CHEMBL3526715

0.146 0.135 CHEMBL3526874

0.314 0.037 CHEMBL845

0.194 0.087 CHEMBL4525779

0.173 0.105 CHEMBL4525780

0.168 0.109 CHEMBL3526631

0.4040.0080.454Dopamine antagonist

0.223 0.017 CHEMBL4525772

0.185 0.02 CHEMBL4525777

0.183 0.021 CHEMBL4525778

0.454 0.006 CHEMBL3526632

0.274 0.013 CHEMBL3526715

0.425 0.007 CHEMBL1688

0.248 0.015 CHEMBL845

0.205 0.018 CHEMBL4525779

0.109 0.035 CHEMBL4525780

CHEMBL3526632
0.3840.0060.3845 Hydroxytryptamine 2C antagonist

0.229 0.014 CHEMBL4525772

0.226 0.014 CHEMBL4525777

0.335 0.008 CHEMBL4525778

0.265 0.011 CHEMBL3526632

0.164 0.023 CHEMBL3526715

0.186 0.019 CHEMBL1688

0.321 0.008 CHEMBL845

0.132 0.032 CHEMBL4525779

0.101 0.045 CHEMBL4525780

0.3840.0180.401ErbB-1 antagonist

0.397 0.016 CHEMBL4525772

0.308 0.031 CHEMBL4525777

0.343 0.024 CHEMBL4525778

0.401 0.016 CHEMBL3526632

0.325 0.027 CHEMBL3526715

0.246 0.053 CHEMBL1688

0.329 0.026 CHEMBL3526874

0.319 0.028 CHEMBL845

0.3 0.033 CHEMBL4525779

0.332 0.026 CHEMBL4525780

0.341 0.024 CHEMBL3526631

CHEMBL3526632
0.3820.0190.382Cyclic AMP phosphodiesterase inhibitor

0.289 0.046 CHEMBL4525772

0.283 0.049 CHEMBL4525777

0.27 0.054 CHEMBL4525778

0.311 0.037 CHEMBL3526632

0.347 0.026 CHEMBL3526715

0.159 0.137 CHEMBL1688

0.359 0.024 CHEMBL845

0.182 0.109 CHEMBL4525779

0.209 0.087 CHEMBL4525780

0.3630.0050.363Alpha 2b adrenoreceptor antagonist

0.233 0.017 CHEMBL4525772

0.241 0.016 CHEMBL4525777

0.267 0.012 CHEMBL4525778

0.278 0.011 CHEMBL3526632

0.226 0.018 CHEMBL3526715

0.313 0.008 CHEMBL1688

0.207 0.022 CHEMBL3526874

0.322 0.008 CHEMBL845

0.186 0.027 CHEMBL4525779

0.146 0.041 CHEMBL4525780

0.125 0.054 CHEMBL3526631

0.3610.0050.3615 Hydroxytryptamine 1F antagonist

0.223 0.009 CHEMBL4525772

0.192 0.011 CHEMBL4525777

0.241 0.008 CHEMBL4525778

0.184 0.012 CHEMBL3526632

0.186 0.011 CHEMBL3526715

0.095 0.034 CHEMBL1688

0.122 0.023 CHEMBL3526874

0.308 0.005 CHEMBL845

0.06 0.059 CHEMBL3526422

0.078 0.044 CHEMBL3526423

0.211 0.009 CHEMBL4525779

0.148 0.017 CHEMBL4525780

0.061 0.058 CHEMBL3526631

0.3550.0040.407Protein kinase C zeta inhibitor

0.214 0.01 CHEMBL4525772

0.263 0.007 CHEMBL4525777

0.288 0.005 CHEMBL4525778

0.407 0.004 CHEMBL3526632

0.269 0.006 CHEMBL3526715

0.111 0.039 CHEMBL1688

0.179 0.014 CHEMBL3526874

0.305 0.005 CHEMBL845

0.138 0.023 CHEMBL4525779

0.131 0.026 CHEMBL4525780

0.301 0.005 CHEMBL3526631

CHEMBL3526632
0.4170.0670.451Histamine release inhibitor

0.41 0.07 CHEMBL4525772

0.302 0.122 CHEMBL4525777

0.33 0.109 CHEMBL4525778

0.373 0.089 CHEMBL3526632

0.313 0.117 CHEMBL3526715

0.34 0.105 CHEMBL845

0.323 0.112 CHEMBL3526422

0.304 0.121 CHEMBL3526420

0.293 0.127 CHEMBL3526421

0.451 0.05 CHEMBL3526423

CHEMBL3526423
0.3510.0050.351Alpha 2a adrenoreceptor antagonist

0.215 0.012 CHEMBL4525772

0.19 0.015 CHEMBL4525777

0.302 0.007 CHEMBL4525778

0.271 0.008 CHEMBL3526632

0.215 0.012 CHEMBL3526715

0.229 0.011 CHEMBL1688

0.105 0.034 CHEMBL3526874

0.31 0.006 CHEMBL845

0.166 0.019 CHEMBL4525779

0.095 0.039 CHEMBL4525780

0.069 0.059 CHEMBL3526631

0.3340.0050.334Toll-Like receptor antagonist

0.308 0.006 CHEMBL4525772

0.226 0.022 CHEMBL4525777

0.235 0.019 CHEMBL4525778

0.261 0.013 CHEMBL3526632

0.239 0.018 CHEMBL3526715

0.303 0.007 CHEMBL3526874

0.293 0.008 CHEMBL845

0.267 0.011 CHEMBL4525779

0.199 0.031 CHEMBL4525780

0.273 0.01 CHEMBL3526631

0.3260.0040.326Alpha 1 adrenoreceptor agonist

0.16 0.009 CHEMBL4525772

0.168 0.008 CHEMBL4525777

0.302 0.004 CHEMBL4525778

0.226 0.005 CHEMBL3526632

0.192 0.007 CHEMBL3526715

0.055 0.043 CHEMBL1688

0.093 0.019 CHEMBL3526874

0.268 0.005 CHEMBL845

0.093 0.019 CHEMBL4525779

0.063 0.033 CHEMBL4525780

0.058 0.038 CHEMBL3526631

0.3170.0030.3275 Hydroxytryptamine 3 agonist

0.327 0.003 CHEMBL4525772

0.217 0.004 CHEMBL4525777

0.215 0.004 CHEMBL4525778

0.181 0.004 CHEMBL3526632

0.136 0.006 CHEMBL3526715

0.099 0.016 CHEMBL1688

0.247 0.003 CHEMBL845

0.121 0.008 CHEMBL4525779

0.097 0.016 CHEMBL4525780

0.076 0.03 CHEMBL3526631

CHEMBL4525772
0.3220.0090.373Dopamine D2 antagonist

0.167 0.02 CHEMBL4525772

0.139 0.024 CHEMBL4525777

0.134 0.025 CHEMBL4525778

0.357 0.008 CHEMBL3526632

0.216 0.015 CHEMBL3526715

0.373 0.008 CHEMBL1688

0.203 0.017 CHEMBL845

0.161 0.021 CHEMBL4525779

0.078 0.04 CHEMBL4525780

CHEMBL1688
0.3210.0140.401Alpha adrenoreceptor antagonist

0.206 0.027 CHEMBL4525772

0.153 0.037 CHEMBL4525777

0.264 0.019 CHEMBL4525778

0.234 0.022 CHEMBL3526632

0.163 0.034 CHEMBL3526715

0.401 0.009 CHEMBL1688

0.142 0.04 CHEMBL3526874

0.277 0.017 CHEMBL845

0.22 0.024 CHEMBL4525779

0.184 0.03 CHEMBL4525780

0.078 0.074 CHEMBL3526631

CHEMBL1688
0.3010.0040.315 Hydroxytryptamine 3A agonist

0.267 0.004 CHEMBL4525772

0.264 0.005 CHEMBL4525777

0.266 0.004 CHEMBL4525778

0.22 0.01 CHEMBL3526632

0.237 0.007 CHEMBL3526715

0.18 0.022 CHEMBL1688

0.116 0.059 CHEMBL3526874

0.31 0.003 CHEMBL845

0.149 0.036 CHEMBL4525779

0.151 0.035 CHEMBL4525780

0.209 0.013 CHEMBL3526631

CHEMBL845
0.2950.0120.323Ribosomal protein S6 kinase inhibitor

0.29 0.013 CHEMBL4525772

0.25 0.02 CHEMBL4525777

0.244 0.022 CHEMBL4525778

0.261 0.018 CHEMBL3526632

0.178 0.048 CHEMBL3526715

0.179 0.047 CHEMBL1688

0.174 0.05 CHEMBL3526874

0.323 0.009 CHEMBL845

0.209 0.033 CHEMBL4525779

0.161 0.057 CHEMBL4525780

0.217 0.031 CHEMBL3526631

CHEMBL845
0.3190.0380.322Psychostimulant

0.207 0.076 CHEMBL4525772

0.2 0.08 CHEMBL4525777

0.224 0.068 CHEMBL4525778

0.195 0.083 CHEMBL3526632

0.163 0.105 CHEMBL3526715

0.136 0.13 CHEMBL1688

0.322 0.037 CHEMBL3526874

0.31 0.04 CHEMBL845

0.159 0.109 CHEMBL3526422

0.192 0.085 CHEMBL3526420

0.172 0.099 CHEMBL3526421

0.191 0.085 CHEMBL3526631

CHEMBL3526874
0.280.0040.28Benzodiazepine agonist

0.215 0.004 CHEMBL4525772

0.204 0.004 CHEMBL4525777

0.194 0.005 CHEMBL4525778

0.124 0.014 CHEMBL3526632

0.104 0.023 CHEMBL3526715

0.137 0.01 CHEMBL1688

0.085 0.035 CHEMBL3526874

0.187 0.005 CHEMBL845

0.146 0.009 CHEMBL4525779

0.136 0.011 CHEMBL4525780

0.079 0.04 CHEMBL3526631

0.3050.0290.344Gastrin inhibitor

0.272 0.056 CHEMBL4525772

0.241 0.09 CHEMBL4525777

0.248 0.082 CHEMBL4525778

0.248 0.082 CHEMBL3526632

0.235 0.098 CHEMBL3526715

0.18 0.179 CHEMBL3526874

0.234 0.099 CHEMBL845

0.275 0.053 CHEMBL3526422

0.261 0.067 CHEMBL3526420

0.286 0.044 CHEMBL3526421

0.344 0.012 CHEMBL3526423

0.183 0.175 CHEMBL4525780

CHEMBL3526423
0.2990.0250.312Ca2+/calmodulin-dependent kinase IV inhibitor

0.259 0.055 CHEMBL4525772

0.282 0.035 CHEMBL4525777

0.274 0.041 CHEMBL4525778

0.258 0.056 CHEMBL3526632

0.264 0.05 CHEMBL3526715

0.237 0.083 CHEMBL1688

0.236 0.085 CHEMBL3526874

0.312 0.02 CHEMBL845

0.244 0.073 CHEMBL4525779

0.237 0.084 CHEMBL4525780

0.248 0.068 CHEMBL3526631

CHEMBL845
0.2730.0030.2735 Hydroxytryptamine 3A antagonist

0.241 0.003 CHEMBL4525772

0.176 0.004 CHEMBL4525777

0.243 0.003 CHEMBL4525778

0.122 0.009 CHEMBL3526632

0.094 0.02 CHEMBL3526715

0.085 0.026 CHEMBL1688

0.202 0.004 CHEMBL845

0.101 0.016 CHEMBL4525779

0.108 0.013 CHEMBL4525780

0.2820.0120.411Alpha 1 adrenoreceptor antagonist

0.185 0.023 CHEMBL4525772

0.142 0.031 CHEMBL4525777

0.177 0.024 CHEMBL4525778

0.205 0.02 CHEMBL3526632

0.137 0.032 CHEMBL3526715

0.411 0.006 CHEMBL1688

0.111 0.04 CHEMBL3526874

0.258 0.014 CHEMBL845

0.204 0.02 CHEMBL4525779

0.18 0.024 CHEMBL4525780

CHEMBL1688
0.270.0090.396Alpha 1b adrenoreceptor antagonist

0.168 0.019 CHEMBL4525772

0.147 0.022 CHEMBL4525777

0.197 0.015 CHEMBL4525778

0.197 0.015 CHEMBL3526632

0.136 0.025 CHEMBL3526715

0.396 0.005 CHEMBL1688

0.076 0.049 CHEMBL3526874

0.229 0.012 CHEMBL845

0.161 0.02 CHEMBL4525779

0.08 0.046 CHEMBL4525780

CHEMBL1688
0.2710.0110.271Alpha 1a adrenoreceptor antagonist

0.171 0.02 CHEMBL4525772

0.134 0.026 CHEMBL4525777

0.169 0.021 CHEMBL4525778

0.177 0.019 CHEMBL3526632

0.117 0.03 CHEMBL3526715

0.187 0.018 CHEMBL1688

0.101 0.036 CHEMBL3526874

0.256 0.012 CHEMBL845

0.18 0.019 CHEMBL4525779

0.078 0.046 CHEMBL4525780

0.2580.0050.319Platelet growth factor antagonist

0.319 0.005 CHEMBL4525772

0.199 0.009 CHEMBL4525777

0.187 0.011 CHEMBL4525778

0.227 0.007 CHEMBL3526632

0.182 0.011 CHEMBL3526715

0.138 0.023 CHEMBL1688

0.116 0.031 CHEMBL3526874

0.215 0.008 CHEMBL845

0.137 0.023 CHEMBL4525779

0.117 0.031 CHEMBL4525780

0.09 0.048 CHEMBL3526631

CHEMBL4525772
0.2790.0260.336LIM domain kinase 1 inhibitor

0.237 0.045 CHEMBL4525772

0.241 0.043 CHEMBL4525777

0.232 0.047 CHEMBL4525778

0.219 0.054 CHEMBL3526632

0.25 0.038 CHEMBL3526715

0.135 0.114 CHEMBL1688

0.259 0.034 CHEMBL3526874

0.274 0.028 CHEMBL845

0.194 0.066 CHEMBL4525779

0.336 0.014 CHEMBL3526631

CHEMBL3526631
0.2610.010.261Alpha 2 adrenoreceptor antagonist

0.177 0.021 CHEMBL4525772

0.145 0.029 CHEMBL4525777

0.238 0.013 CHEMBL4525778

0.195 0.018 CHEMBL3526632

0.159 0.025 CHEMBL3526715

0.153 0.026 CHEMBL1688

0.097 0.05 CHEMBL3526874

0.236 0.013 CHEMBL845

0.152 0.027 CHEMBL4525779

0.076 0.072 CHEMBL4525780

0.3080.0590.308Aryl hydrocarbon receptor agonist

0.261 0.074 CHEMBL4525772

0.251 0.078 CHEMBL4525777

0.251 0.078 CHEMBL4525778

0.182 0.112 CHEMBL3526632

0.227 0.089 CHEMBL3526715

0.164 0.125 CHEMBL1688

0.158 0.13 CHEMBL3526874

0.273 0.07 CHEMBL845

0.281 0.067 CHEMBL3526631

0.2880.0390.315MAP kinase kinase 2 inhibitor

0.254 0.052 CHEMBL4525772

0.213 0.074 CHEMBL4525777

0.235 0.061 CHEMBL4525778

0.248 0.055 CHEMBL3526632

0.315 0.03 CHEMBL3526715

0.215 0.073 CHEMBL3526874

0.262 0.049 CHEMBL845

0.138 0.132 CHEMBL4525780

0.306 0.033 CHEMBL3526631

CHEMBL3526715
0.2860.0380.29MAP-kinase-activated kinase 5 inhibitor

0.25 0.059 CHEMBL4525772

0.254 0.057 CHEMBL4525777

0.254 0.057 CHEMBL4525778

0.252 0.058 CHEMBL3526632

0.218 0.084 CHEMBL3526715

0.163 0.161 CHEMBL1688

0.264 0.051 CHEMBL3526874

0.29 0.036 CHEMBL845

0.229 0.074 CHEMBL4525779

0.201 0.102 CHEMBL4525780

0.221 0.081 CHEMBL3526631

CHEMBL845
0.2870.040.382Ca2+/calmodulin-dependent kinase II beta inhibitor

0.165 0.11 CHEMBL4525772

0.22 0.064 CHEMBL4525777

0.245 0.053 CHEMBL4525778

0.216 0.066 CHEMBL3526632

0.191 0.084 CHEMBL3526715

0.331 0.028 CHEMBL3526874

0.238 0.055 CHEMBL845

0.141 0.14 CHEMBL4525780

0.382 0.017 CHEMBL3526631

CHEMBL3526631
0.2470.0060.251Alpha adrenoreceptor agonist

0.137 0.019 CHEMBL4525772

0.233 0.006 CHEMBL4525777

0.247 0.006 CHEMBL4525778

0.185 0.01 CHEMBL3526632

0.173 0.012 CHEMBL3526715

0.115 0.023 CHEMBL3526874

0.251 0.005 CHEMBL845

0.076 0.041 CHEMBL4525779

0.069 0.047 CHEMBL3526631

CHEMBL845
0.2590.0190.259Activin receptor-like kinase 2 inhibitor

0.233 0.025 CHEMBL4525772

0.212 0.032 CHEMBL4525777

0.225 0.027 CHEMBL4525778

0.206 0.034 CHEMBL3526632

0.187 0.043 CHEMBL3526715

0.256 0.019 CHEMBL845

0.189 0.042 CHEMBL4525779

0.171 0.052 CHEMBL4525780

0.2860.0470.524Ca2+/calmodulin-dependent protein kinase inhibitor

0.156 0.107 CHEMBL4525772

0.203 0.073 CHEMBL4525777

0.224 0.065 CHEMBL4525778

0.239 0.06 CHEMBL3526632

0.317 0.038 CHEMBL3526715

0.415 0.015 CHEMBL3526874

0.296 0.044 CHEMBL845

0.151 0.11 CHEMBL4525779

0.14 0.122 CHEMBL4525780

0.524 0.007 CHEMBL3526631

CHEMBL3526631
0.2550.0160.282Platelet activating factor beta antagonist

0.28 0.013 CHEMBL4525772

0.213 0.022 CHEMBL4525777

0.156 0.036 CHEMBL4525778

0.209 0.023 CHEMBL3526632

0.187 0.027 CHEMBL3526715

0.282 0.013 CHEMBL1688

0.088 0.072 CHEMBL3526874

0.202 0.024 CHEMBL845

CHEMBL1688
0.3690.1310.456Caspase 9 stimulant

0.334 0.159 CHEMBL4525772

0.322 0.17 CHEMBL4525777

0.287 0.208 CHEMBL4525778

0.375 0.127 CHEMBL3526632

0.303 0.191 CHEMBL3526715

0.311 0.182 CHEMBL3526874

0.456 0.08 CHEMBL845

0.319 0.174 CHEMBL3526631

CHEMBL845
0.2580.0230.298Acetylcholine M1 receptor antagonist

0.235 0.029 CHEMBL4525772

0.154 0.07 CHEMBL4525777

0.17 0.059 CHEMBL4525778

0.209 0.039 CHEMBL3526632

0.19 0.047 CHEMBL3526715

0.298 0.015 CHEMBL1688

0.191 0.047 CHEMBL845

0.18 0.052 CHEMBL4525779

0.152 0.072 CHEMBL4525780

CHEMBL1688
0.2410.0080.241Dopamine D3 antagonist

0.156 0.014 CHEMBL4525772

0.12 0.02 CHEMBL4525777

0.118 0.02 CHEMBL4525778

0.183 0.012 CHEMBL3526632

0.156 0.014 CHEMBL3526715

0.124 0.019 CHEMBL1688

0.139 0.017 CHEMBL845

0.109 0.023 CHEMBL4525779

0.074 0.035 CHEMBL4525780

0.2770.0440.277EphB2 antagonist

0.237 0.064 CHEMBL4525772

0.237 0.064 CHEMBL4525777

0.228 0.069 CHEMBL4525778

0.257 0.053 CHEMBL3526632

0.238 0.064 CHEMBL3526715

0.18 0.102 CHEMBL3526874

0.24 0.062 CHEMBL845

0.217 0.077 CHEMBL3526631

0.2710.040.419Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.128 0.107 CHEMBL4525772

0.198 0.065 CHEMBL4525777

0.227 0.053 CHEMBL4525778

0.201 0.064 CHEMBL3526632

0.154 0.086 CHEMBL3526715

0.302 0.034 CHEMBL3526874

0.208 0.06 CHEMBL845

0.419 0.014 CHEMBL3526631

CHEMBL3526631
0.2410.010.336Histamine H1 receptor antagonist

0.244 0.01 CHEMBL4525772

0.138 0.027 CHEMBL4525777

0.232 0.011 CHEMBL4525778

0.119 0.032 CHEMBL3526632

0.083 0.055 CHEMBL3526715

0.336 0.005 CHEMBL1688

0.147 0.025 CHEMBL845

0.12 0.032 CHEMBL4525779

0.079 0.059 CHEMBL4525780

CHEMBL1688
0.2590.0330.262I kappa B kinase epsilon inhibitor

0.211 0.062 CHEMBL4525772

0.216 0.058 CHEMBL4525777

0.241 0.042 CHEMBL4525778

0.262 0.032 CHEMBL3526632

0.217 0.058 CHEMBL3526715

0.227 0.05 CHEMBL3526874

0.252 0.037 CHEMBL845

0.158 0.111 CHEMBL4525780

0.185 0.084 CHEMBL3526631

CHEMBL3526632
0.280.0550.349HERG channel blocker

0.349 0.038 CHEMBL4525772

0.149 0.132 CHEMBL4525777

0.193 0.095 CHEMBL4525778

0.273 0.057 CHEMBL845

0.241 0.07 CHEMBL4525779

0.2 0.091 CHEMBL4525780

CHEMBL4525772
0.2880.0720.423Hypoxia-inducible factor 1 alpha inhibitor

0.423 0.025 CHEMBL4525772

0.194 0.159 CHEMBL4525777

0.194 0.159 CHEMBL4525778

0.297 0.067 CHEMBL3526632

0.356 0.043 CHEMBL3526715

0.229 0.12 CHEMBL3526874

0.3 0.066 CHEMBL845

0.185 0.171 CHEMBL3526631

CHEMBL4525772
0.220.0050.29GABA A receptor antagonist

0.17 0.007 CHEMBL4525772

0.159 0.008 CHEMBL4525777

0.151 0.009 CHEMBL4525778

0.082 0.021 CHEMBL3526632

0.082 0.021 CHEMBL3526715

0.062 0.029 CHEMBL1688

0.29 0.004 CHEMBL845

0.078 0.023 CHEMBL4525779

0.07 0.026 CHEMBL4525780

CHEMBL845
0.2240.010.224Potassium channel (Ca-activated) activator

0.127 0.037 CHEMBL4525772

0.141 0.031 CHEMBL4525777

0.125 0.038 CHEMBL4525778

0.181 0.019 CHEMBL3526632

0.19 0.017 CHEMBL3526715

0.1 0.056 CHEMBL1688

0.215 0.012 CHEMBL3526874

0.199 0.015 CHEMBL845

0.125 0.038 CHEMBL4525779

0.13 0.035 CHEMBL4525780

0.17 0.022 CHEMBL3526631

0.2540.0420.265Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.208 0.066 CHEMBL4525772

0.194 0.078 CHEMBL4525777

0.208 0.066 CHEMBL4525778

0.225 0.054 CHEMBL3526632

0.265 0.038 CHEMBL3526715

0.214 0.062 CHEMBL3526874

0.242 0.046 CHEMBL845

0.2 0.073 CHEMBL4525779

0.158 0.121 CHEMBL4525780

0.23 0.052 CHEMBL3526631

CHEMBL3526715
0.2170.0050.295GABA receptor antagonist

0.16 0.008 CHEMBL4525772

0.154 0.009 CHEMBL4525777

0.144 0.01 CHEMBL4525778

0.079 0.022 CHEMBL3526632

0.078 0.022 CHEMBL3526715

0.06 0.032 CHEMBL1688

0.295 0.004 CHEMBL845

0.071 0.025 CHEMBL4525779

0.065 0.028 CHEMBL4525780

0.051 0.042 CHEMBL3526631

CHEMBL845
0.2140.0030.214Potassium channel small-conductance Ca-activated blocker

0.153 0.004 CHEMBL4525772

0.199 0.004 CHEMBL4525777

0.159 0.004 CHEMBL4525778

0.075 0.011 CHEMBL3526632

0.052 0.022 CHEMBL3526715

0.075 0.011 CHEMBL1688

0.144 0.004 CHEMBL3526874

0.151 0.004 CHEMBL845

0.102 0.006 CHEMBL4525779

0.056 0.02 CHEMBL4525780

0.086 0.009 CHEMBL3526631

0.30.0920.377Calcium channel activator

0.235 0.165 CHEMBL4525772

0.265 0.13 CHEMBL4525777

0.265 0.13 CHEMBL4525778

0.279 0.114 CHEMBL3526632

0.268 0.126 CHEMBL3526715

0.206 0.204 CHEMBL1688

0.257 0.139 CHEMBL3526874

0.377 0.034 CHEMBL845

0.24 0.159 CHEMBL3526631

CHEMBL845
0.210.0080.215 Hydroxytryptamine 1B antagonist

0.1 0.023 CHEMBL4525772

0.113 0.019 CHEMBL4525777

0.125 0.016 CHEMBL4525778

0.1 0.023 CHEMBL3526632

0.108 0.02 CHEMBL3526715

0.13 0.015 CHEMBL845

0.135 0.015 CHEMBL4525779

0.073 0.039 CHEMBL4525780

0.220.0230.36Death-associated protein kinase 2 inhibitor

0.21 0.028 CHEMBL4525777

0.21 0.028 CHEMBL4525778

0.195 0.038 CHEMBL3526632

0.211 0.027 CHEMBL3526715

0.198 0.036 CHEMBL1688

0.26 0.011 CHEMBL3526874

0.236 0.017 CHEMBL845

0.179 0.055 CHEMBL4525779

0.179 0.055 CHEMBL4525780

0.36 0.004 CHEMBL3526631

CHEMBL3526631
0.2540.0580.394Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.204 0.088 CHEMBL4525777

0.237 0.067 CHEMBL4525778

0.165 0.124 CHEMBL3526632

0.152 0.142 CHEMBL3526715

0.252 0.059 CHEMBL3526874

0.232 0.07 CHEMBL845

0.152 0.142 CHEMBL4525780

0.394 0.015 CHEMBL3526631

CHEMBL3526631
0.210.0150.428GABA receptor agonist

0.198 0.018 CHEMBL4525772

0.16 0.031 CHEMBL4525777

0.168 0.027 CHEMBL4525778

0.125 0.052 CHEMBL3526632

0.129 0.049 CHEMBL3526715

0.428 0.004 CHEMBL1688

0.187 0.021 CHEMBL845

0.092 0.087 CHEMBL4525779

0.121 0.056 CHEMBL4525780

CHEMBL1688
0.2060.0140.206Insulin receptor antagonist

0.148 0.028 CHEMBL4525772

0.145 0.029 CHEMBL4525777

0.179 0.019 CHEMBL4525778

0.17 0.022 CHEMBL3526632

0.111 0.049 CHEMBL3526715

0.097 0.066 CHEMBL3526874

0.139 0.032 CHEMBL845

0.09 0.077 CHEMBL4525779

0.09 0.076 CHEMBL4525780

0.105 0.055 CHEMBL3526631

0.2010.0120.266Protein kinase C mu inhibitor

0.19 0.014 CHEMBL4525772

0.161 0.021 CHEMBL4525777

0.176 0.017 CHEMBL4525778

0.168 0.019 CHEMBL3526632

0.163 0.021 CHEMBL3526715

0.103 0.054 CHEMBL1688

0.146 0.028 CHEMBL3526874

0.266 0.006 CHEMBL845

0.096 0.06 CHEMBL3526423

0.166 0.02 CHEMBL4525779

0.114 0.045 CHEMBL4525780

0.176 0.017 CHEMBL3526631

CHEMBL845
0.2540.0650.299Potassium channel blocker

0.299 0.047 CHEMBL4525772

0.186 0.102 CHEMBL3526874

0.24 0.071 CHEMBL845

0.22 0.08 CHEMBL4525779

CHEMBL4525772
0.1950.0060.313Acetylcholine M4 receptor antagonist

0.155 0.009 CHEMBL4525772

0.117 0.019 CHEMBL4525777

0.12 0.018 CHEMBL4525778

0.098 0.03 CHEMBL3526632

0.087 0.04 CHEMBL3526715

0.313 0.004 CHEMBL1688

0.141 0.012 CHEMBL845

0.12 0.018 CHEMBL4525779

0.112 0.021 CHEMBL4525780

CHEMBL1688
0.2050.0170.205Alpha 2c adrenoreceptor antagonist

0.148 0.033 CHEMBL4525772

0.128 0.044 CHEMBL4525777

0.137 0.039 CHEMBL4525778

0.168 0.025 CHEMBL3526632

0.134 0.04 CHEMBL3526715

0.165 0.026 CHEMBL1688

0.135 0.04 CHEMBL3526874

0.17 0.025 CHEMBL845

0.135 0.04 CHEMBL4525779

0.2040.0160.272Check point kinase 2 inhibitor

0.118 0.05 CHEMBL4525772

0.17 0.026 CHEMBL4525777

0.17 0.026 CHEMBL4525778

0.182 0.022 CHEMBL3526632

0.125 0.045 CHEMBL3526715

0.134 0.039 CHEMBL1688

0.185 0.021 CHEMBL3526874

0.272 0.008 CHEMBL845

0.122 0.047 CHEMBL4525779

0.13 0.042 CHEMBL4525780

0.265 0.008 CHEMBL3526631

CHEMBL845
0.2520.0660.291Tyrosine 3 hydroxylase inhibitor

0.199 0.137 CHEMBL4525772

0.203 0.129 CHEMBL4525777

0.181 0.174 CHEMBL4525778

0.272 0.05 CHEMBL3526632

0.291 0.038 CHEMBL3526715

0.206 0.125 CHEMBL1688

0.201 0.133 CHEMBL3526874

0.247 0.071 CHEMBL845

0.198 0.138 CHEMBL3526423

0.204 0.128 CHEMBL4525779

0.221 0.102 CHEMBL3526631

CHEMBL3526715
0.2070.0320.207NADPH oxidase inhibitor

0.112 0.094 CHEMBL4525772

0.12 0.083 CHEMBL4525777

0.135 0.067 CHEMBL4525778

0.193 0.037 CHEMBL3526632

0.151 0.054 CHEMBL3526715

0.19 0.038 CHEMBL845

0.1890.0170.212Protein kinase C gamma inhibitor

0.125 0.049 CHEMBL4525772

0.149 0.032 CHEMBL4525777

0.206 0.013 CHEMBL4525778

0.152 0.03 CHEMBL3526632

0.148 0.033 CHEMBL3526715

0.185 0.017 CHEMBL3526874

0.165 0.024 CHEMBL845

0.113 0.059 CHEMBL4525779

0.212 0.012 CHEMBL3526631

CHEMBL3526631
0.1920.0230.206Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.151 0.071 CHEMBL4525772

0.176 0.036 CHEMBL4525777

0.183 0.029 CHEMBL4525778

0.206 0.015 CHEMBL3526632

0.179 0.033 CHEMBL3526715

0.145 0.083 CHEMBL1688

0.152 0.069 CHEMBL3526874

0.178 0.034 CHEMBL845

0.151 0.07 CHEMBL4525779

0.158 0.058 CHEMBL4525780

0.145 0.081 CHEMBL3526631

CHEMBL3526632
0.1760.0120.176Alpha 1d adrenoreceptor antagonist

0.104 0.022 CHEMBL4525772

0.091 0.026 CHEMBL4525777

0.086 0.028 CHEMBL4525778

0.121 0.019 CHEMBL3526632

0.075 0.032 CHEMBL3526715

0.121 0.019 CHEMBL1688

0.075 0.033 CHEMBL3526874

0.155 0.014 CHEMBL845

0.068 0.035 CHEMBL4525779

0.1940.0330.213GABA C receptor rho-2 antagonist

0.208 0.025 CHEMBL4525772

0.194 0.032 CHEMBL4525777

0.194 0.032 CHEMBL4525778

0.166 0.055 CHEMBL3526632

0.168 0.053 CHEMBL3526715

0.132 0.102 CHEMBL1688

0.213 0.023 CHEMBL3526874

0.189 0.036 CHEMBL845

0.174 0.047 CHEMBL3526631

CHEMBL3526874
0.1760.0150.179Hedgehog signaling inhibitor

0.159 0.02 CHEMBL4525772

0.137 0.029 CHEMBL4525777

0.175 0.016 CHEMBL4525778

0.101 0.064 CHEMBL3526632

0.097 0.069 CHEMBL3526715

0.097 0.069 CHEMBL3526874

0.179 0.015 CHEMBL845

0.156 0.021 CHEMBL4525779

0.13 0.033 CHEMBL4525780

CHEMBL845
0.190.0290.23Glutamate receptor antagonist

0.151 0.05 CHEMBL4525772

0.144 0.055 CHEMBL4525777

0.161 0.044 CHEMBL4525778

0.141 0.057 CHEMBL3526632

0.102 0.094 CHEMBL3526715

0.174 0.036 CHEMBL3526874

0.218 0.021 CHEMBL845

0.15 0.051 CHEMBL4525779

0.141 0.057 CHEMBL4525780

0.23 0.019 CHEMBL3526631

CHEMBL3526631
0.1750.0150.175ALK inhibitor

0.124 0.028 CHEMBL4525772

0.118 0.031 CHEMBL4525777

0.138 0.022 CHEMBL4525778

0.157 0.018 CHEMBL3526632

0.149 0.02 CHEMBL3526715

0.172 0.015 CHEMBL845

0.097 0.043 CHEMBL4525779

0.111 0.035 CHEMBL4525780

0.3090.150.535Calcium channel L-type activator

0.262 0.193 CHEMBL4525777

0.262 0.193 CHEMBL4525778

0.42 0.068 CHEMBL3526632

0.375 0.099 CHEMBL3526715

0.288 0.168 CHEMBL1688

0.535 0.017 CHEMBL3526874

0.352 0.116 CHEMBL845

0.324 0.137 CHEMBL3526631

CHEMBL3526874
0.1640.0050.1645 Hydroxytryptamine 6 antagonist

0.123 0.01 CHEMBL4525772

0.152 0.006 CHEMBL4525777

0.129 0.009 CHEMBL4525778

0.077 0.025 CHEMBL3526632

0.079 0.024 CHEMBL3526715

0.05 0.049 CHEMBL1688

0.074 0.027 CHEMBL3526874

0.148 0.006 CHEMBL845

0.105 0.013 CHEMBL4525779

0.071 0.029 CHEMBL4525780

0.073 0.027 CHEMBL3526631

0.1780.020.181Pregnane X receptor agonist

0.181 0.018 CHEMBL4525772

0.157 0.041 CHEMBL4525777

0.167 0.03 CHEMBL4525778

0.136 0.083 CHEMBL3526632

0.131 0.097 CHEMBL3526715

0.127 0.107 CHEMBL1688

0.164 0.033 CHEMBL845

0.126 0.111 CHEMBL4525780

CHEMBL4525772
0.170.0160.175 Hydroxytryptamine 7 antagonist

0.137 0.019 CHEMBL4525772

0.069 0.038 CHEMBL4525777

0.077 0.033 CHEMBL4525778

0.084 0.029 CHEMBL3526632

0.067 0.04 CHEMBL3526715

0.151 0.018 CHEMBL845

0.064 0.042 CHEMBL4525779

0.1730.020.1735 Hydroxytryptamine 1 antagonist

0.097 0.038 CHEMBL4525772

0.081 0.047 CHEMBL4525777

0.086 0.044 CHEMBL4525778

0.089 0.042 CHEMBL3526632

0.079 0.048 CHEMBL3526715

0.063 0.06 CHEMBL1688

0.114 0.032 CHEMBL845

0.084 0.045 CHEMBL4525779

0.1570.0070.168Bromodomain-containing protein 2 inhibitor

0.168 0.005 CHEMBL4525772

0.136 0.014 CHEMBL4525777

0.146 0.01 CHEMBL4525778

0.089 0.057 CHEMBL3526632

0.083 0.07 CHEMBL3526715

0.115 0.027 CHEMBL3526874

0.144 0.011 CHEMBL845

0.123 0.021 CHEMBL4525779

0.132 0.016 CHEMBL4525780

0.106 0.034 CHEMBL3526631

CHEMBL4525772
0.1990.050.233Antipruritic

0.233 0.031 CHEMBL4525772

0.142 0.104 CHEMBL3526632

0.202 0.048 CHEMBL3526715

0.175 0.069 CHEMBL845

CHEMBL4525772
0.160.0120.185Cyclin B3 inhibitor

0.105 0.026 CHEMBL4525772

0.119 0.021 CHEMBL4525777

0.143 0.015 CHEMBL4525778

0.157 0.012 CHEMBL3526632

0.157 0.012 CHEMBL3526715

0.079 0.039 CHEMBL1688

0.096 0.03 CHEMBL3526874

0.185 0.008 CHEMBL845

0.081 0.038 CHEMBL4525779

0.091 0.032 CHEMBL4525780

0.121 0.021 CHEMBL3526631

CHEMBL845
0.1730.0260.203Antihistaminic

0.203 0.02 CHEMBL4525772

0.09 0.064 CHEMBL4525777

0.149 0.032 CHEMBL4525778

0.171 0.027 CHEMBL1688

0.105 0.051 CHEMBL845

0.094 0.06 CHEMBL4525779

CHEMBL4525772
0.2250.080.278Potassium channel (Voltage-sensitive) blocker

0.278 0.056 CHEMBL4525772

0.148 0.139 CHEMBL4525778

0.215 0.085 CHEMBL845

0.196 0.098 CHEMBL4525779

0.161 0.128 CHEMBL4525780

CHEMBL4525772
0.2380.0930.2585 Hydroxytryptamine uptake stimulant

0.254 0.077 CHEMBL4525772

0.196 0.159 CHEMBL4525777

0.196 0.159 CHEMBL4525778

0.211 0.132 CHEMBL3526632

0.258 0.073 CHEMBL3526715

0.223 0.113 CHEMBL845

0.218 0.12 CHEMBL3526631

CHEMBL3526715
0.1580.0190.1585 Hydroxytryptamine 1A antagonist

0.092 0.035 CHEMBL4525772

0.077 0.042 CHEMBL4525777

0.078 0.042 CHEMBL4525778

0.086 0.037 CHEMBL3526632

0.076 0.042 CHEMBL3526715

0.068 0.047 CHEMBL1688

0.118 0.026 CHEMBL845

0.1430.0050.143Histamine agonist

0.129 0.006 CHEMBL4525772

0.092 0.01 CHEMBL4525777

0.092 0.01 CHEMBL4525778

0.053 0.036 CHEMBL3526632

0.049 0.041 CHEMBL3526715

0.072 0.018 CHEMBL3526874

0.102 0.009 CHEMBL845

0.066 0.022 CHEMBL4525779

0.053 0.035 CHEMBL4525780

0.075 0.016 CHEMBL3526631

0.1630.0260.196Histamine antagonist

0.196 0.02 CHEMBL4525772

0.08 0.063 CHEMBL4525777

0.141 0.032 CHEMBL4525778

0.163 0.026 CHEMBL1688

0.095 0.051 CHEMBL845

0.086 0.058 CHEMBL4525779

CHEMBL4525772
0.1450.0080.192Acetylcholine M5 receptor antagonist

0.119 0.013 CHEMBL4525772

0.073 0.029 CHEMBL4525777

0.079 0.025 CHEMBL4525778

0.096 0.019 CHEMBL3526632

0.09 0.02 CHEMBL3526715

0.192 0.005 CHEMBL1688

0.094 0.019 CHEMBL845

0.07 0.031 CHEMBL4525779

0.058 0.045 CHEMBL4525780

CHEMBL1688
0.1380.0060.1915 Hydroxytryptamine 2A agonist

0.091 0.019 CHEMBL4525772

0.106 0.012 CHEMBL4525777

0.095 0.017 CHEMBL4525778

0.104 0.013 CHEMBL3526632

0.096 0.016 CHEMBL3526715

0.191 0.004 CHEMBL845

0.088 0.021 CHEMBL4525779

0.073 0.034 CHEMBL4525780

0.07 0.037 CHEMBL3526631

CHEMBL845
0.1980.0670.2275 Hydroxytryptamine 3E antagonist

0.186 0.09 CHEMBL4525772

0.197 0.068 CHEMBL4525777

0.197 0.068 CHEMBL4525778

0.227 0.03 CHEMBL3526874

0.201 0.061 CHEMBL845

0.213 0.044 CHEMBL3526631

CHEMBL3526874
0.20.070.2Focal adhesion kinase 2 inhibitor

0.171 0.099 CHEMBL4525772

0.153 0.127 CHEMBL4525777

0.16 0.115 CHEMBL4525778

0.166 0.106 CHEMBL3526632

0.158 0.118 CHEMBL3526874

0.2 0.069 CHEMBL845

0.1430.0130.1435 Hydroxytryptamine 1D antagonist

0.065 0.044 CHEMBL4525772

0.079 0.031 CHEMBL4525777

0.094 0.025 CHEMBL4525778

0.068 0.04 CHEMBL3526632

0.08 0.031 CHEMBL3526715

0.085 0.028 CHEMBL845

0.086 0.028 CHEMBL4525779

0.1490.020.149Acetylcholine M3 receptor agonist

0.102 0.044 CHEMBL4525772

0.112 0.039 CHEMBL4525777

0.122 0.034 CHEMBL4525778

0.11 0.04 CHEMBL3526632

0.091 0.051 CHEMBL3526715

0.078 0.062 CHEMBL1688

0.141 0.024 CHEMBL845

0.101 0.044 CHEMBL4525779

0.111 0.039 CHEMBL4525780

0.1410.0110.162Protein kinase B alpha inhibitor

0.156 0.008 CHEMBL4525772

0.122 0.017 CHEMBL4525777

0.099 0.03 CHEMBL4525778

0.095 0.033 CHEMBL3526632

0.082 0.039 CHEMBL3526715

0.074 0.044 CHEMBL1688

0.162 0.007 CHEMBL845

0.099 0.031 CHEMBL4525779

0.068 0.05 CHEMBL4525780

0.067 0.051 CHEMBL3526631

CHEMBL845
0.1810.0530.212Protein-tyrosine kinase Lyn inhibitor

0.153 0.064 CHEMBL4525772

0.121 0.084 CHEMBL4525777

0.129 0.078 CHEMBL4525778

0.117 0.088 CHEMBL3526632

0.118 0.087 CHEMBL1688

0.153 0.064 CHEMBL3526874

0.161 0.06 CHEMBL845

0.212 0.041 CHEMBL3526631

CHEMBL3526631
0.1330.0050.25 Hydroxytryptamine 2 agonist

0.089 0.012 CHEMBL4525772

0.08 0.015 CHEMBL4525777

0.074 0.017 CHEMBL4525778

0.09 0.012 CHEMBL3526632

0.066 0.022 CHEMBL3526715

0.066 0.022 CHEMBL3526874

0.2 0.004 CHEMBL845

0.067 0.021 CHEMBL4525779

0.06 0.027 CHEMBL4525780

0.069 0.02 CHEMBL3526631

CHEMBL845
0.1570.030.181Death-associated protein kinase 1 inhibitor

0.154 0.033 CHEMBL4525777

0.147 0.044 CHEMBL4525778

0.154 0.034 CHEMBL3526632

0.157 0.03 CHEMBL3526715

0.139 0.059 CHEMBL1688

0.181 0.013 CHEMBL845

CHEMBL845
0.1350.0080.153Toll-Like receptor 7 antagonist

0.097 0.023 CHEMBL4525772

0.105 0.018 CHEMBL4525777

0.108 0.016 CHEMBL4525778

0.096 0.024 CHEMBL3526632

0.092 0.027 CHEMBL3526715

0.096 0.024 CHEMBL3526874

0.153 0.005 CHEMBL845

0.148 0.006 CHEMBL4525779

0.118 0.012 CHEMBL4525780

CHEMBL845
0.1290.0020.129Histamine H4 receptor agonist

0.1 0.003 CHEMBL4525772

0.089 0.003 CHEMBL4525777

0.089 0.003 CHEMBL4525778

0.028 0.007 CHEMBL3526632

0.028 0.007 CHEMBL3526715

0.022 0.01 CHEMBL1688

0.047 0.005 CHEMBL3526874

0.087 0.003 CHEMBL845

0.039 0.005 CHEMBL4525779

0.039 0.005 CHEMBL4525780

0.044 0.005 CHEMBL3526631

0.1530.0270.2Activin receptor-like kinase 4 inhibitor

0.143 0.032 CHEMBL4525772

0.137 0.036 CHEMBL4525777

0.139 0.034 CHEMBL4525778

0.115 0.059 CHEMBL3526632

0.104 0.077 CHEMBL3526715

0.101 0.083 CHEMBL1688

0.2 0.014 CHEMBL845

0.103 0.08 CHEMBL4525779

0.105 0.076 CHEMBL4525780

CHEMBL845
0.1820.0560.3ATPase inhibitor

0.171 0.069 CHEMBL4525772

0.143 0.114 CHEMBL4525777

0.148 0.105 CHEMBL4525778

0.142 0.116 CHEMBL3526632

0.3 0.006 CHEMBL3526874

0.163 0.081 CHEMBL845

0.241 0.016 CHEMBL3526631

CHEMBL3526874
0.1290.0030.129Potassium channel small-conductance Ca-activated activator

0.122 0.003 CHEMBL4525772

0.117 0.004 CHEMBL4525777

0.094 0.004 CHEMBL4525778

0.03 0.023 CHEMBL3526632

0.029 0.024 CHEMBL3526715

0.053 0.01 CHEMBL1688

0.067 0.007 CHEMBL3526874

0.108 0.004 CHEMBL845

0.062 0.008 CHEMBL4525779

0.031 0.022 CHEMBL4525780

0.092 0.005 CHEMBL3526631

0.1930.0710.508CDC-like kinase 4 inhibitor

0.169 0.086 CHEMBL4525772

0.156 0.097 CHEMBL4525777

0.196 0.069 CHEMBL4525778

0.142 0.107 CHEMBL3526632

0.174 0.082 CHEMBL3526715

0.438 0.011 CHEMBL3526874

0.23 0.054 CHEMBL845

0.508 0.006 CHEMBL3526631

CHEMBL3526631
0.1770.0540.237Cyclin-dependent kinase 8 inhibitor

0.169 0.062 CHEMBL4525772

0.156 0.073 CHEMBL4525777

0.155 0.074 CHEMBL4525778

0.169 0.061 CHEMBL3526632

0.171 0.06 CHEMBL3526715

0.219 0.025 CHEMBL3526874

0.179 0.052 CHEMBL845

0.237 0.019 CHEMBL3526631

CHEMBL3526631
0.180.0580.386Polo-like kinase-3 inhibitor

0.153 0.081 CHEMBL4525772

0.137 0.1 CHEMBL4525777

0.16 0.073 CHEMBL4525778

0.156 0.078 CHEMBL3526632

0.386 0.004 CHEMBL1688

0.142 0.094 CHEMBL3526874

0.141 0.094 CHEMBL845

0.141 0.095 CHEMBL4525779

0.146 0.089 CHEMBL4525780

CHEMBL1688
0.1450.0240.195Protein kinase C delta inhibitor

0.123 0.035 CHEMBL4525772

0.117 0.039 CHEMBL4525777

0.113 0.042 CHEMBL4525778

0.117 0.039 CHEMBL3526632

0.113 0.042 CHEMBL3526715

0.195 0.009 CHEMBL1688

0.103 0.049 CHEMBL3526874

0.169 0.014 CHEMBL845

0.154 0.019 CHEMBL4525779

0.122 0.036 CHEMBL4525780

0.157 0.018 CHEMBL3526631

CHEMBL1688
0.1540.0340.154Polo-like kinase-4 inhibitor

0.12 0.056 CHEMBL4525772

0.105 0.072 CHEMBL4525777

0.133 0.047 CHEMBL4525778

0.123 0.054 CHEMBL3526632

0.112 0.064 CHEMBL3526715

0.114 0.062 CHEMBL845

0.1590.040.208Antibacterial (Helicobacter pylori)

0.132 0.064 CHEMBL4525772

0.136 0.06 CHEMBL4525777

0.121 0.079 CHEMBL4525778

0.124 0.076 CHEMBL3526632

0.112 0.094 CHEMBL3526874

0.149 0.047 CHEMBL845

0.125 0.074 CHEMBL3526422

0.208 0.02 CHEMBL3526423

CHEMBL3526423
0.1380.0190.19Protein kinase B gamma inhibitor

0.146 0.017 CHEMBL4525772

0.111 0.028 CHEMBL4525777

0.092 0.037 CHEMBL4525778

0.071 0.057 CHEMBL3526632

0.072 0.055 CHEMBL3526715

0.128 0.023 CHEMBL3526874

0.155 0.015 CHEMBL845

0.19 0.009 CHEMBL3526631

CHEMBL3526631
0.1270.010.1275 Hydroxytryptamine 5A antagonist

0.081 0.023 CHEMBL4525772

0.08 0.024 CHEMBL4525777

0.091 0.018 CHEMBL4525778

0.072 0.029 CHEMBL3526632

0.071 0.03 CHEMBL3526715

0.103 0.015 CHEMBL3526874

0.112 0.013 CHEMBL845

0.06 0.045 CHEMBL4525779

0.076 0.026 CHEMBL3526631

0.1610.0460.164MAP3K9 inhibitor

0.145 0.067 CHEMBL4525777

0.142 0.073 CHEMBL4525778

0.15 0.06 CHEMBL3526632

0.15 0.06 CHEMBL3526715

0.134 0.087 CHEMBL3526874

0.164 0.041 CHEMBL845

0.144 0.07 CHEMBL3526631

CHEMBL845
0.1560.0410.189Platelet activating factor antagonist

0.189 0.029 CHEMBL4525772

0.152 0.043 CHEMBL4525777

0.125 0.06 CHEMBL4525778

0.145 0.048 CHEMBL3526632

0.112 0.069 CHEMBL3526715

0.149 0.045 CHEMBL1688

0.12 0.063 CHEMBL845

CHEMBL4525772
0.1670.0530.202RET inhibitor

0.127 0.074 CHEMBL4525772

0.171 0.051 CHEMBL4525777

0.113 0.084 CHEMBL4525778

0.202 0.042 CHEMBL3526632

0.166 0.053 CHEMBL3526715

0.105 0.091 CHEMBL3526874

0.129 0.073 CHEMBL845

0.102 0.095 CHEMBL3526631

CHEMBL3526632
0.1570.0430.157Nav1.3 sodium channel blocker

0.147 0.05 CHEMBL4525772

0.101 0.097 CHEMBL4525777

0.106 0.09 CHEMBL4525778

0.102 0.096 CHEMBL3526715

0.141 0.054 CHEMBL3526874

0.107 0.09 CHEMBL845

0.1240.0110.1285 Hydroxytryptamine 5 antagonist

0.073 0.024 CHEMBL4525772

0.072 0.025 CHEMBL4525777

0.085 0.019 CHEMBL4525778

0.063 0.033 CHEMBL3526632

0.063 0.033 CHEMBL3526715

0.128 0.01 CHEMBL3526874

0.108 0.014 CHEMBL845

0.058 0.039 CHEMBL4525779

0.053 0.051 CHEMBL4525780

0.083 0.019 CHEMBL3526631

CHEMBL3526874
0.1350.0240.2575 Hydroxytryptamine agonist

0.068 0.048 CHEMBL4525772

0.062 0.053 CHEMBL4525777

0.082 0.041 CHEMBL4525778

0.061 0.054 CHEMBL3526632

0.257 0.01 CHEMBL845

0.068 0.048 CHEMBL4525779

CHEMBL845
0.1350.0270.135Insulin growth factor antagonist

0.123 0.032 CHEMBL4525772

0.094 0.051 CHEMBL4525777

0.108 0.041 CHEMBL4525778

0.119 0.034 CHEMBL3526632

0.095 0.05 CHEMBL3526715

0.113 0.038 CHEMBL845

0.1310.0240.328Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.094 0.039 CHEMBL4525777

0.099 0.036 CHEMBL4525778

0.122 0.026 CHEMBL3526632

0.104 0.033 CHEMBL3526715

0.073 0.056 CHEMBL1688

0.209 0.013 CHEMBL3526874

0.249 0.009 CHEMBL845

0.091 0.041 CHEMBL4525779

0.089 0.043 CHEMBL4525780

0.328 0.006 CHEMBL3526631

CHEMBL3526631
0.1930.0860.213Platelet aggregation inhibitor

0.213 0.073 CHEMBL4525772

0.168 0.109 CHEMBL4525777

0.185 0.093 CHEMBL3526632

0.145 0.134 CHEMBL3526715

0.211 0.074 CHEMBL1688

0.192 0.087 CHEMBL845

0.145 0.135 CHEMBL3526422

0.152 0.126 CHEMBL3526420

0.21 0.074 CHEMBL3526423

CHEMBL4525772
0.1620.0590.196Protein kinase (CK1) inhibitor

0.122 0.09 CHEMBL4525777

0.117 0.095 CHEMBL4525778

0.113 0.097 CHEMBL3526632

0.11 0.1 CHEMBL3526715

0.12 0.091 CHEMBL3526874

0.173 0.052 CHEMBL845

0.196 0.041 CHEMBL3526631

CHEMBL3526631
0.1290.0260.129Insulin like growth factor 1 antagonist

0.115 0.032 CHEMBL4525772

0.09 0.049 CHEMBL4525777

0.102 0.04 CHEMBL4525778

0.1 0.042 CHEMBL3526632

0.087 0.053 CHEMBL3526715

0.106 0.038 CHEMBL845

0.1610.0590.161Tyrosine-protein kinase receptor antagonist

0.121 0.086 CHEMBL4525772

0.111 0.095 CHEMBL4525777

0.113 0.093 CHEMBL4525778

0.108 0.099 CHEMBL3526715

0.147 0.065 CHEMBL845

0.1780.0770.196Tyrosine kinase inhibitor

0.192 0.072 CHEMBL4525772

0.168 0.081 CHEMBL4525778

0.196 0.07 CHEMBL3526632

0.133 0.099 CHEMBL3526715

0.146 0.091 CHEMBL1688

0.138 0.096 CHEMBL845

CHEMBL3526632
0.1650.0670.165Cyclin-dependent kinase 3 inhibitor

0.137 0.131 CHEMBL4525772

0.155 0.086 CHEMBL4525777

0.156 0.083 CHEMBL4525778

0.148 0.101 CHEMBL3526632

0.159 0.078 CHEMBL3526715

0.141 0.12 CHEMBL845

0.1290.0310.144Phosphodiesterase 7B inhibitor

0.143 0.024 CHEMBL4525772

0.115 0.041 CHEMBL4525777

0.105 0.051 CHEMBL4525778

0.086 0.076 CHEMBL3526632

0.101 0.055 CHEMBL3526715

0.099 0.057 CHEMBL1688

0.1 0.056 CHEMBL3526874

0.144 0.024 CHEMBL845

0.083 0.081 CHEMBL4525779

0.103 0.053 CHEMBL3526631

CHEMBL845
0.1250.0280.167Pim-3 kinase inhibitor

0.118 0.032 CHEMBL4525772

0.104 0.042 CHEMBL4525777

0.101 0.045 CHEMBL4525778

0.096 0.05 CHEMBL3526632

0.085 0.066 CHEMBL3526715

0.106 0.04 CHEMBL3526874

0.165 0.014 CHEMBL845

0.167 0.014 CHEMBL3526631

CHEMBL3526631
0.1990.1010.219RNA-directed DNA polymerase inhibitor

0.165 0.162 CHEMBL4525772

0.172 0.148 CHEMBL4525777

0.209 0.087 CHEMBL3526632

0.219 0.075 CHEMBL3526715

0.183 0.127 CHEMBL845

0.174 0.145 CHEMBL3526631

CHEMBL3526715
0.1340.0370.217Fibroblast growth factor 1 antagonist

0.143 0.034 CHEMBL4525772

0.115 0.047 CHEMBL4525777

0.104 0.054 CHEMBL4525778

0.106 0.053 CHEMBL3526632

0.09 0.066 CHEMBL3526715

0.217 0.013 CHEMBL1688

0.183 0.021 CHEMBL3526874

0.098 0.059 CHEMBL845

0.14 0.034 CHEMBL3526631

CHEMBL1688
0.1370.040.261Antiadrenergic

0.1 0.056 CHEMBL4525772

0.118 0.046 CHEMBL4525778

0.114 0.048 CHEMBL3526632

0.098 0.057 CHEMBL3526715

0.192 0.026 CHEMBL1688

0.077 0.074 CHEMBL3526874

0.16 0.033 CHEMBL845

0.093 0.06 CHEMBL4525779

0.261 0.016 CHEMBL4525780

CHEMBL4525780
0.1030.0060.117Corticotropin releasing factor 2 receptor antagonist

0.117 0.004 CHEMBL4525772

0.086 0.013 CHEMBL4525777

0.085 0.013 CHEMBL4525778

0.06 0.045 CHEMBL3526632

0.057 0.053 CHEMBL3526874

0.096 0.008 CHEMBL845

0.085 0.014 CHEMBL3526631

CHEMBL4525772
0.1140.0180.126Protein kinase B beta inhibitor

0.126 0.013 CHEMBL4525772

0.1 0.025 CHEMBL4525777

0.091 0.031 CHEMBL4525778

0.082 0.04 CHEMBL3526632

0.074 0.05 CHEMBL3526715

0.07 0.058 CHEMBL1688

0.124 0.014 CHEMBL845

0.074 0.051 CHEMBL4525779

0.071 0.055 CHEMBL3526631

CHEMBL4525772
0.1040.0090.152Dopamine D5 antagonist

0.081 0.012 CHEMBL4525772

0.057 0.021 CHEMBL4525777

0.066 0.016 CHEMBL4525778

0.152 0.006 CHEMBL3526632

0.087 0.011 CHEMBL3526715

0.079 0.012 CHEMBL1688

0.053 0.023 CHEMBL845

0.061 0.019 CHEMBL4525779

0.06 0.019 CHEMBL4525780

CHEMBL3526632
0.1810.0850.213Growth factor agonist

0.213 0.052 CHEMBL4525772

0.149 0.144 CHEMBL4525777

0.162 0.117 CHEMBL4525778

0.165 0.11 CHEMBL3526632

0.192 0.071 CHEMBL3526874

0.164 0.113 CHEMBL845

CHEMBL4525772
0.1210.0260.26I kappa B kinase inhibitor

0.095 0.043 CHEMBL4525772

0.084 0.055 CHEMBL4525777

0.082 0.058 CHEMBL4525778

0.123 0.025 CHEMBL3526632

0.109 0.032 CHEMBL3526715

0.173 0.011 CHEMBL3526874

0.142 0.018 CHEMBL845

0.085 0.054 CHEMBL4525779

0.26 0.005 CHEMBL3526631

CHEMBL3526631
0.1370.0430.209Interleukin 8 antagonist

0.105 0.085 CHEMBL4525772

0.101 0.094 CHEMBL4525777

0.124 0.056 CHEMBL4525778

0.143 0.038 CHEMBL3526632

0.121 0.06 CHEMBL3526715

0.178 0.02 CHEMBL3526874

0.141 0.041 CHEMBL845

0.209 0.01 CHEMBL3526631

CHEMBL3526631
0.1340.0390.259Adrenaline antagonist

0.098 0.055 CHEMBL4525772

0.115 0.046 CHEMBL4525778

0.112 0.047 CHEMBL3526632

0.095 0.056 CHEMBL3526715

0.19 0.025 CHEMBL1688

0.157 0.033 CHEMBL845

0.091 0.06 CHEMBL4525779

0.259 0.016 CHEMBL4525780

CHEMBL4525780
0.1070.0130.126Dopamine D4 agonist

0.126 0.011 CHEMBL4525772

0.063 0.026 CHEMBL4525777

0.063 0.025 CHEMBL4525778

0.054 0.031 CHEMBL3526632

0.048 0.037 CHEMBL3526715

0.071 0.022 CHEMBL845

0.049 0.036 CHEMBL4525780

CHEMBL4525772
0.1160.0220.148Phosphodiesterase 11A inhibitor

0.079 0.061 CHEMBL4525772

0.097 0.035 CHEMBL4525777

0.094 0.038 CHEMBL4525778

0.097 0.035 CHEMBL3526632

0.148 0.011 CHEMBL3526715

0.093 0.039 CHEMBL3526874

0.102 0.03 CHEMBL845

0.077 0.065 CHEMBL4525779

0.114 0.023 CHEMBL3526631

CHEMBL3526715
0.1160.0220.148Phosphodiesterase XI inhibitor

0.079 0.061 CHEMBL4525772

0.097 0.035 CHEMBL4525777

0.094 0.038 CHEMBL4525778

0.097 0.035 CHEMBL3526632

0.148 0.011 CHEMBL3526715

0.093 0.039 CHEMBL3526874

0.102 0.03 CHEMBL845

0.077 0.065 CHEMBL4525779

0.114 0.023 CHEMBL3526631

CHEMBL3526715
0.1280.0340.189Acetylcholine agonist

0.094 0.051 CHEMBL4525772

0.081 0.064 CHEMBL4525778

0.189 0.016 CHEMBL1688

0.08 0.066 CHEMBL3526874

0.106 0.043 CHEMBL845

CHEMBL1688
0.1190.0260.119Phosphodiesterase 6D inhibitor

0.096 0.06 CHEMBL4525772

0.092 0.069 CHEMBL4525777

0.099 0.054 CHEMBL4525778

0.108 0.039 CHEMBL3526632

0.101 0.05 CHEMBL3526715

0.089 0.078 CHEMBL845

0.1470.0540.201Tyrosine-protein kinase receptor FLT3 inhibitor

0.178 0.043 CHEMBL4525772

0.149 0.054 CHEMBL4525778

0.102 0.079 CHEMBL3526632

0.201 0.037 CHEMBL1688

0.122 0.067 CHEMBL3526874

0.124 0.066 CHEMBL845

0.11 0.074 CHEMBL3526631

CHEMBL1688
0.1330.040.137Transcription factor STAT6 inhibitor

0.125 0.052 CHEMBL4525772

0.111 0.077 CHEMBL4525777

0.119 0.062 CHEMBL4525778

0.137 0.035 CHEMBL3526632

0.125 0.051 CHEMBL3526715

0.132 0.041 CHEMBL845

0.105 0.093 CHEMBL3526631

CHEMBL3526632
0.1170.0240.169Glutamate release inhibitor

0.169 0.007 CHEMBL4525772

0.085 0.076 CHEMBL4525777

0.099 0.044 CHEMBL4525778

0.107 0.034 CHEMBL3526632

0.108 0.032 CHEMBL3526715

0.094 0.054 CHEMBL3526874

0.083 0.082 CHEMBL845

0.098 0.046 CHEMBL3526631

CHEMBL4525772
0.1790.0880.44Death-associated protein kinase 3 inhibitor

0.156 0.113 CHEMBL4525777

0.165 0.102 CHEMBL4525778

0.17 0.096 CHEMBL3526632

0.323 0.032 CHEMBL3526874

0.216 0.066 CHEMBL845

0.44 0.012 CHEMBL3526631

CHEMBL3526631
0.1810.090.48Clk dual-specificity kinase inhibitor

0.151 0.113 CHEMBL4525772

0.143 0.121 CHEMBL4525777

0.18 0.091 CHEMBL4525778

0.142 0.121 CHEMBL3526632

0.166 0.101 CHEMBL3526715

0.399 0.019 CHEMBL3526874

0.192 0.084 CHEMBL845

0.48 0.009 CHEMBL3526631

CHEMBL3526631
0.1290.0390.147Multidrug resistance-associated protein 1 inhibitor

0.147 0.026 CHEMBL4525772

0.112 0.059 CHEMBL4525777

0.102 0.075 CHEMBL3526632

0.111 0.061 CHEMBL3526715

0.108 0.065 CHEMBL845

0.107 0.067 CHEMBL4525779

CHEMBL4525772
0.1450.0560.15Protein kinase (CK1) delta inhibitor

0.109 0.083 CHEMBL4525777

0.106 0.086 CHEMBL4525778

0.098 0.095 CHEMBL3526632

0.101 0.091 CHEMBL3526715

0.138 0.061 CHEMBL845

0.15 0.053 CHEMBL3526631

CHEMBL3526631
0.0970.010.097Potassium channel (Ca-activated) blocker

0.072 0.025 CHEMBL4525772

0.089 0.013 CHEMBL4525777

0.082 0.017 CHEMBL4525778

0.069 0.028 CHEMBL3526632

0.061 0.039 CHEMBL1688

0.085 0.015 CHEMBL3526874

0.09 0.013 CHEMBL845

0.078 0.02 CHEMBL4525779

0.055 0.052 CHEMBL4525780

0.078 0.019 CHEMBL3526631

0.1480.0610.285Cyclin-dependent kinase 7 inhibitor

0.119 0.086 CHEMBL4525777

0.132 0.074 CHEMBL4525778

0.177 0.044 CHEMBL3526715

0.214 0.029 CHEMBL3526874

0.168 0.048 CHEMBL845

0.285 0.014 CHEMBL3526631

CHEMBL3526631
0.1010.0140.113Alpha 2 adrenoreceptor agonist

0.067 0.034 CHEMBL4525772

0.065 0.037 CHEMBL4525777

0.07 0.031 CHEMBL4525778

0.074 0.028 CHEMBL3526632

0.07 0.032 CHEMBL3526715

0.083 0.022 CHEMBL3526874

0.113 0.011 CHEMBL845

0.06 0.042 CHEMBL3526631

CHEMBL845
0.1150.0280.166MAP-kinase-activated kinase inhibitor

0.097 0.042 CHEMBL4525777

0.102 0.038 CHEMBL4525778

0.077 0.066 CHEMBL3526632

0.078 0.065 CHEMBL3526715

0.095 0.044 CHEMBL3526874

0.166 0.01 CHEMBL845

0.095 0.043 CHEMBL4525779

0.084 0.057 CHEMBL4525780

0.124 0.024 CHEMBL3526631

CHEMBL845
0.1330.0490.164Cyclin-dependent kinase 1 inhibitor

0.085 0.079 CHEMBL4525777

0.122 0.054 CHEMBL4525778

0.104 0.064 CHEMBL3526632

0.088 0.075 CHEMBL3526715

0.109 0.061 CHEMBL3526874

0.164 0.036 CHEMBL845

0.161 0.037 CHEMBL3526631

CHEMBL845
0.120.0360.227NMDA receptor antagonist

0.078 0.068 CHEMBL4525778

0.1 0.047 CHEMBL3526632

0.087 0.057 CHEMBL3526715

0.173 0.019 CHEMBL3526874

0.172 0.019 CHEMBL845

0.227 0.011 CHEMBL3526631

CHEMBL3526631
0.1020.0190.109Acetylcholine M5 receptor agonist

0.092 0.025 CHEMBL4525772

0.063 0.052 CHEMBL4525777

0.07 0.044 CHEMBL4525778

0.109 0.015 CHEMBL845

CHEMBL845
0.150.0670.263Glycogen synthase kinase-3 alpha inhibitor

0.103 0.101 CHEMBL4525777

0.123 0.082 CHEMBL4525778

0.175 0.05 CHEMBL3526632

0.131 0.078 CHEMBL3526715

0.168 0.054 CHEMBL3526874

0.17 0.053 CHEMBL845

0.263 0.023 CHEMBL3526631

CHEMBL3526631
0.0980.0150.149Pim-2 kinase inhibitor

0.091 0.017 CHEMBL4525772

0.066 0.026 CHEMBL4525777

0.065 0.027 CHEMBL4525778

0.057 0.034 CHEMBL3526632

0.078 0.021 CHEMBL3526874

0.131 0.009 CHEMBL845

0.149 0.007 CHEMBL3526631

CHEMBL3526631
0.0920.010.096MDM2 inhibitor

0.083 0.017 CHEMBL4525772

0.072 0.034 CHEMBL4525777

0.077 0.025 CHEMBL4525778

0.067 0.048 CHEMBL3526632

0.096 0.008 CHEMBL845

0.067 0.047 CHEMBL4525779

0.077 0.025 CHEMBL4525780

CHEMBL845
0.0970.0150.103Protein kinase C beta inhibitor

0.079 0.031 CHEMBL4525772

0.076 0.036 CHEMBL4525777

0.103 0.012 CHEMBL4525778

0.079 0.032 CHEMBL3526632

0.086 0.023 CHEMBL3526715

0.074 0.04 CHEMBL3526874

0.087 0.022 CHEMBL845

0.083 0.026 CHEMBL4525779

0.073 0.041 CHEMBL4525780

0.077 0.034 CHEMBL3526631

CHEMBL4525778
0.1480.0660.378Ca2+/calmodulin-dependent kinase II delta inhibitor

0.11 0.092 CHEMBL4525777

0.123 0.082 CHEMBL4525778

0.35 0.01 CHEMBL3526874

0.143 0.069 CHEMBL845

0.378 0.008 CHEMBL3526631

CHEMBL3526631
0.1430.0630.146Heat shock protein 70 antagonist

0.146 0.054 CHEMBL4525772

0.13 0.123 CHEMBL3526632

0.14 0.075 CHEMBL3526715

CHEMBL4525772
0.1440.0650.179Proto-oncogene tyrosine-protein kinase Yes inhibitor

0.15 0.061 CHEMBL4525772

0.102 0.099 CHEMBL4525778

0.117 0.085 CHEMBL3526632

0.118 0.083 CHEMBL3526715

0.179 0.048 CHEMBL1688

0.133 0.072 CHEMBL845

CHEMBL1688
0.1140.0360.124mTOR complex 1 inhibitor

0.114 0.036 CHEMBL4525772

0.106 0.049 CHEMBL4525777

0.094 0.075 CHEMBL4525778

0.1 0.062 CHEMBL3526632

0.095 0.075 CHEMBL3526715

0.11 0.042 CHEMBL845

0.11 0.043 CHEMBL4525779

0.124 0.025 CHEMBL4525780

CHEMBL4525780
0.10.0220.125Protein kinase C alpha inhibitor

0.079 0.034 CHEMBL4525772

0.079 0.034 CHEMBL4525777

0.092 0.026 CHEMBL4525778

0.07 0.044 CHEMBL3526632

0.086 0.029 CHEMBL3526715

0.061 0.059 CHEMBL3526874

0.125 0.015 CHEMBL845

0.079 0.035 CHEMBL4525779

0.061 0.059 CHEMBL4525780

0.081 0.033 CHEMBL3526631

CHEMBL845
0.1030.0270.153MAP-kinase-activated kinase 2 inhibitor

0.085 0.039 CHEMBL4525777

0.09 0.035 CHEMBL4525778

0.067 0.063 CHEMBL3526632

0.069 0.06 CHEMBL3526715

0.084 0.04 CHEMBL3526874

0.153 0.01 CHEMBL845

0.083 0.041 CHEMBL4525779

0.072 0.054 CHEMBL4525780

0.115 0.022 CHEMBL3526631

CHEMBL845
0.110.0340.121Phosphodiesterase I inhibitor

0.121 0.026 CHEMBL4525772

0.082 0.073 CHEMBL4525777

0.088 0.062 CHEMBL4525778

0.084 0.068 CHEMBL3526632

CHEMBL4525772
0.1330.0580.24Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.137 0.055 CHEMBL4525772

0.122 0.067 CHEMBL3526632

0.24 0.019 CHEMBL1688

0.115 0.073 CHEMBL845

CHEMBL1688
0.1330.0580.24Abl kinase inhibitor

0.136 0.055 CHEMBL4525772

0.121 0.068 CHEMBL3526632

0.24 0.019 CHEMBL1688

0.115 0.073 CHEMBL845

CHEMBL1688
0.080.0050.1875 Hydroxytryptamine 2B agonist

0.06 0.009 CHEMBL4525772

0.06 0.008 CHEMBL4525777

0.05 0.013 CHEMBL4525778

0.042 0.022 CHEMBL3526632

0.043 0.02 CHEMBL3526715

0.043 0.02 CHEMBL1688

0.187 0.003 CHEMBL845

0.054 0.011 CHEMBL3526631

CHEMBL845
0.0780.0040.078Histamine H1 receptor agonist

0.063 0.007 CHEMBL4525772

0.073 0.004 CHEMBL4525777

0.074 0.004 CHEMBL4525778

0.047 0.023 CHEMBL3526632

0.048 0.022 CHEMBL3526715

0.054 0.014 CHEMBL1688

0.064 0.006 CHEMBL3526874

0.075 0.004 CHEMBL845

0.044 0.029 CHEMBL4525779

0.045 0.028 CHEMBL4525780

0.063 0.007 CHEMBL3526631

0.1290.0560.129DNA repair enzyme inhibitor

0.126 0.062 CHEMBL4525772

0.126 0.061 CHEMBL3526632

0.114 0.086 CHEMBL3526715

0.118 0.076 CHEMBL845

0.1750.1040.218Neurotrophic factor enhancer

0.218 0.06 CHEMBL4525772

0.15 0.137 CHEMBL3526632

0.17 0.11 CHEMBL845

CHEMBL4525772
0.0750.0070.075Acetylcholine M4 receptor agonist

0.045 0.013 CHEMBL4525772

0.033 0.019 CHEMBL4525777

0.035 0.017 CHEMBL4525778

0.059 0.009 CHEMBL845

0.1270.060.185Aurora-B kinase inhibitor

0.094 0.09 CHEMBL4525772

0.101 0.081 CHEMBL4525778

0.099 0.084 CHEMBL3526632

0.108 0.074 CHEMBL3526715

0.146 0.048 CHEMBL3526874

0.122 0.063 CHEMBL845

0.185 0.035 CHEMBL3526631

CHEMBL3526631
0.240.1730.35115-Lipoxygenase inhibitor

0.225 0.187 CHEMBL4525772

0.217 0.195 CHEMBL4525777

0.235 0.177 CHEMBL3526632

0.351 0.099 CHEMBL3526715

0.239 0.174 CHEMBL3526874

0.316 0.121 CHEMBL3526631

CHEMBL3526715
0.1550.0890.183Neurotensin receptor agonist

0.163 0.074 CHEMBL4525772

0.142 0.122 CHEMBL4525777

0.157 0.085 CHEMBL3526632

0.142 0.124 CHEMBL3526715

0.183 0.047 CHEMBL845

0.15 0.1 CHEMBL3526422

0.154 0.093 CHEMBL3526420

0.151 0.099 CHEMBL3526421

0.156 0.088 CHEMBL3526423

CHEMBL845
0.0880.0220.094MAP kinase 7 inhibitor

0.094 0.013 CHEMBL4525772

0.079 0.049 CHEMBL4525777

0.085 0.03 CHEMBL4525778

0.085 0.029 CHEMBL3526632

0.077 0.057 CHEMBL3526715

CHEMBL4525772
0.0890.0260.123MAP kinase kinase 7 inhibitor

0.079 0.05 CHEMBL4525777

0.098 0.014 CHEMBL3526632

0.099 0.014 CHEMBL3526715

0.101 0.012 CHEMBL3526874

0.108 0.008 CHEMBL845

0.123 0.004 CHEMBL3526631

CHEMBL3526631
0.0970.0350.124Glycine receptor antagonist

0.08 0.056 CHEMBL3526874

0.124 0.016 CHEMBL845

0.079 0.057 CHEMBL3526631

CHEMBL845
0.080.0180.089Toll-Like receptor 8 antagonist

0.059 0.032 CHEMBL4525772

0.053 0.038 CHEMBL4525777

0.056 0.035 CHEMBL4525778

0.077 0.019 CHEMBL3526874

0.089 0.013 CHEMBL845

0.071 0.023 CHEMBL4525779

0.06 0.031 CHEMBL4525780

0.077 0.019 CHEMBL3526631

CHEMBL845
0.0830.0210.185Acetylcholine muscarinic agonist

0.063 0.032 CHEMBL4525772

0.185 0.007 CHEMBL1688

0.065 0.03 CHEMBL845

CHEMBL1688
0.1180.0570.133EphA2 antagonist

0.115 0.059 CHEMBL4525772

0.093 0.083 CHEMBL4525778

0.133 0.042 CHEMBL3526632

0.107 0.068 CHEMBL3526874

0.098 0.077 CHEMBL845

0.09 0.088 CHEMBL4525780

0.121 0.053 CHEMBL3526631

CHEMBL3526632
0.1170.0560.119Aurora-A kinase inhibitor

0.091 0.074 CHEMBL4525772

0.084 0.08 CHEMBL4525778

0.107 0.061 CHEMBL3526715

0.119 0.055 CHEMBL3526874

0.102 0.065 CHEMBL845

0.116 0.056 CHEMBL3526631

CHEMBL3526874
0.1750.1140.42Dyrk kinase inhibitor

0.23 0.081 CHEMBL3526632

0.238 0.078 CHEMBL3526715

0.274 0.062 CHEMBL3526874

0.172 0.116 CHEMBL845

0.42 0.023 CHEMBL3526631

CHEMBL3526631
0.0670.0070.067Protein kinase (CK1) epsilon inhibitor

0.042 0.022 CHEMBL4525772

0.049 0.014 CHEMBL4525777

0.047 0.015 CHEMBL4525778

0.042 0.022 CHEMBL3526632

0.061 0.008 CHEMBL845

0.036 0.035 CHEMBL4525779

0.0970.0370.111Janus tyrosine kinase 2 inhibitor

0.103 0.035 CHEMBL4525772

0.065 0.061 CHEMBL4525777

0.111 0.032 CHEMBL4525778

0.089 0.042 CHEMBL845

0.078 0.049 CHEMBL4525779

0.074 0.052 CHEMBL4525780

CHEMBL4525778
0.0770.0180.097Phosphodiesterase 1A inhibitor

0.097 0.01 CHEMBL4525772

0.059 0.043 CHEMBL4525777

0.065 0.031 CHEMBL4525778

0.056 0.052 CHEMBL3526874

0.057 0.048 CHEMBL845

CHEMBL4525772
0.1090.050.255Pim-1 kinase inhibitor

0.104 0.054 CHEMBL4525772

0.083 0.077 CHEMBL4525777

0.084 0.076 CHEMBL4525778

0.084 0.075 CHEMBL3526632

0.097 0.06 CHEMBL3526715

0.161 0.024 CHEMBL3526874

0.16 0.024 CHEMBL845

0.255 0.008 CHEMBL3526631

CHEMBL3526631
0.1020.0440.142Histamine N-methyltransferase inhibitor

0.137 0.019 CHEMBL4525772

0.098 0.048 CHEMBL4525777

0.098 0.048 CHEMBL4525778

0.111 0.037 CHEMBL3526874

0.116 0.033 CHEMBL845

0.142 0.017 CHEMBL3526631

CHEMBL3526631
0.0980.040.098GABA A receptor agonist

0.098 0.039 CHEMBL4525772

0.082 0.059 CHEMBL4525777

0.082 0.059 CHEMBL4525778

0.098 0.04 CHEMBL845

0.1270.0690.165Cyclin-dependent kinase inhibitor

0.105 0.085 CHEMBL4525778

0.099 0.091 CHEMBL3526632

0.099 0.091 CHEMBL3526715

0.103 0.087 CHEMBL3526874

0.165 0.049 CHEMBL845

0.139 0.062 CHEMBL3526631

CHEMBL845
0.0880.030.11Phosphodiesterase VI inhibitor

0.074 0.053 CHEMBL4525772

0.071 0.06 CHEMBL4525778

0.11 0.015 CHEMBL3526632

0.101 0.019 CHEMBL3526715

0.076 0.048 CHEMBL3526874

0.087 0.032 CHEMBL3526631

CHEMBL3526632
0.1330.0760.221Aurora-C kinase inhibitor

0.12 0.106 CHEMBL4525777

0.125 0.093 CHEMBL4525778

0.117 0.115 CHEMBL3526632

0.118 0.111 CHEMBL3526715

0.221 0.015 CHEMBL3526874

0.132 0.079 CHEMBL845

0.186 0.024 CHEMBL3526631

CHEMBL3526874
0.0670.0090.067Kainate receptor 2 antagonist

0.034 0.027 CHEMBL4525777

0.051 0.015 CHEMBL4525778

0.054 0.014 CHEMBL3526874

0.061 0.011 CHEMBL845

0.06 0.012 CHEMBL3526631

0.0720.0150.117NMDA receptor subunit 3B antagonist

0.039 0.037 CHEMBL4525772

0.044 0.03 CHEMBL4525778

0.116 0.009 CHEMBL3526632

0.062 0.018 CHEMBL3526715

0.069 0.016 CHEMBL3526874

0.117 0.009 CHEMBL845

0.078 0.014 CHEMBL3526631

CHEMBL845
0.0720.0160.0725 Hydroxytryptamine 4 antagonist

0.061 0.023 CHEMBL4525772

0.049 0.039 CHEMBL4525778

0.058 0.026 CHEMBL3526632

0.053 0.033 CHEMBL845

0.1430.0880.183Src kinase inhibitor

0.146 0.086 CHEMBL4525772

0.181 0.064 CHEMBL3526632

0.16 0.077 CHEMBL3526715

0.172 0.069 CHEMBL1688

0.168 0.072 CHEMBL3526874

0.116 0.112 CHEMBL845

0.183 0.063 CHEMBL3526631

CHEMBL3526631
0.1130.0580.169Granulocyte macrophage colony stimulating factor antagonist

0.112 0.059 CHEMBL4525772

0.096 0.076 CHEMBL4525778

0.169 0.03 CHEMBL1688

0.089 0.086 CHEMBL845

CHEMBL1688
0.0790.0240.139Protein kinase C eta inhibitor

0.054 0.039 CHEMBL4525772

0.05 0.043 CHEMBL4525777

0.056 0.037 CHEMBL4525778

0.068 0.03 CHEMBL3526632

0.069 0.029 CHEMBL3526715

0.114 0.014 CHEMBL3526874

0.056 0.037 CHEMBL845

0.139 0.009 CHEMBL3526631

CHEMBL3526631
0.0630.0080.063Acid-sensing ion channel blocker

0.055 0.012 CHEMBL4525772

0.046 0.02 CHEMBL4525777

0.053 0.014 CHEMBL4525778

0.049 0.018 CHEMBL3526632

0.051 0.015 CHEMBL3526715

0.037 0.033 CHEMBL1688

0.057 0.011 CHEMBL845

0.047 0.019 CHEMBL4525779

0.047 0.019 CHEMBL4525780

0.0880.0340.215Check point kinase 1 inhibitor

0.064 0.052 CHEMBL4525777

0.068 0.048 CHEMBL4525778

0.089 0.033 CHEMBL3526632

0.082 0.037 CHEMBL3526715

0.149 0.015 CHEMBL3526874

0.153 0.014 CHEMBL845

0.065 0.051 CHEMBL4525779

0.064 0.053 CHEMBL4525780

0.215 0.008 CHEMBL3526631

CHEMBL3526631
0.1530.0990.194Catenin beta inhibitor

0.142 0.126 CHEMBL4525772

0.152 0.101 CHEMBL3526632

0.164 0.076 CHEMBL3526715

0.192 0.039 CHEMBL3526874

0.171 0.065 CHEMBL845

0.162 0.08 CHEMBL3526422

0.167 0.071 CHEMBL3526420

0.161 0.083 CHEMBL3526421

0.166 0.073 CHEMBL3526423

0.142 0.125 CHEMBL4525779

0.194 0.037 CHEMBL3526631

CHEMBL3526631
0.0880.0340.117Phosphodiesterase V inhibitor

0.064 0.058 CHEMBL4525772

0.068 0.054 CHEMBL4525778

0.117 0.02 CHEMBL3526632

0.114 0.021 CHEMBL3526715

0.116 0.021 CHEMBL1688

0.089 0.033 CHEMBL3526874

0.071 0.051 CHEMBL845

0.105 0.026 CHEMBL3526631

CHEMBL3526632
0.0720.0180.0725 Hydroxytryptamine 7 agonist

0.064 0.025 CHEMBL4525772

0.058 0.034 CHEMBL4525777

0.056 0.038 CHEMBL4525778

0.055 0.041 CHEMBL3526715

0.062 0.029 CHEMBL845

0.0760.0220.076Cyclin D1 inhibitor

0.062 0.039 CHEMBL4525777

0.074 0.024 CHEMBL4525778

0.07 0.028 CHEMBL3526632

0.073 0.025 CHEMBL3526715

0.071 0.027 CHEMBL845

0.0620.0090.09Vascular adhesion protein 1 inhibitor

0.09 0.004 CHEMBL4525772

0.042 0.023 CHEMBL4525777

0.038 0.029 CHEMBL4525778

0.065 0.008 CHEMBL845

0.055 0.012 CHEMBL4525779

0.068 0.007 CHEMBL4525780

CHEMBL4525772
0.0730.0190.078AMPA receptor antagonist

0.078 0.018 CHEMBL4525778

0.044 0.038 CHEMBL3526874

0.067 0.022 CHEMBL845

0.044 0.038 CHEMBL4525780

0.078 0.018 CHEMBL3526631

CHEMBL3526631
0.0770.0240.081Cyclin-dependent kinase 6 inhibitor

0.081 0.021 CHEMBL4525772

0.059 0.042 CHEMBL4525777

0.059 0.042 CHEMBL4525778

0.055 0.048 CHEMBL3526715

0.077 0.025 CHEMBL845

0.056 0.046 CHEMBL4525779

CHEMBL4525772
0.090.0380.101Transforming growth factor beta 3 antagonist

0.101 0.023 CHEMBL4525772

0.086 0.047 CHEMBL4525777

0.083 0.054 CHEMBL4525778

0.079 0.069 CHEMBL3526632

0.085 0.05 CHEMBL3526715

0.092 0.035 CHEMBL1688

0.089 0.04 CHEMBL845

CHEMBL4525772
0.0630.0110.068Benzodiazepine antagonist

0.068 0.008 CHEMBL4525772

0.057 0.017 CHEMBL4525777

0.057 0.016 CHEMBL4525778

0.049 0.028 CHEMBL3526874

0.062 0.012 CHEMBL845

CHEMBL4525772
0.0620.0110.076GABA B receptor antagonist

0.05 0.019 CHEMBL4525777

0.054 0.016 CHEMBL4525778

0.04 0.036 CHEMBL3526632

0.076 0.007 CHEMBL845

0.043 0.029 CHEMBL4525779

0.067 0.009 CHEMBL3526631

CHEMBL845
0.0760.0250.149I kappa B kinase 2 inhibitor

0.062 0.044 CHEMBL4525772

0.07 0.033 CHEMBL3526632

0.073 0.029 CHEMBL3526715

0.099 0.013 CHEMBL3526874

0.092 0.016 CHEMBL845

0.057 0.053 CHEMBL4525779

0.149 0.005 CHEMBL3526631

CHEMBL3526631
0.1230.0720.182c-Src kinase inhibitor

0.135 0.064 CHEMBL4525772

0.098 0.091 CHEMBL4525777

0.182 0.041 CHEMBL3526632

0.123 0.072 CHEMBL3526715

0.106 0.085 CHEMBL3526874

0.127 0.07 CHEMBL3526631

CHEMBL3526632
0.0760.0250.113Phosphodiesterase 1B inhibitor

0.113 0.011 CHEMBL4525772

0.053 0.052 CHEMBL4525778

CHEMBL4525772
0.0690.0190.161Acetylcholine M1 receptor agonist

0.043 0.03 CHEMBL4525772

0.161 0.006 CHEMBL1688

0.049 0.026 CHEMBL845

CHEMBL1688
0.0850.0360.116Phosphodiesterase 5A inhibitor

0.065 0.055 CHEMBL4525772

0.064 0.057 CHEMBL4525778

0.116 0.02 CHEMBL3526632

0.112 0.021 CHEMBL3526715

0.114 0.021 CHEMBL1688

0.088 0.034 CHEMBL3526874

0.066 0.055 CHEMBL845

0.102 0.026 CHEMBL3526631

CHEMBL3526632
0.0820.0340.115Cyclin-dependent kinase 4 inhibitor

0.06 0.052 CHEMBL4525772

0.058 0.055 CHEMBL4525777

0.061 0.051 CHEMBL4525778

0.072 0.039 CHEMBL3526632

0.057 0.056 CHEMBL3526715

0.115 0.02 CHEMBL845

0.058 0.055 CHEMBL4525779

CHEMBL845
0.1380.0890.147MAP kinase 3 inhibitor

0.147 0.072 CHEMBL4525772

0.129 0.108 CHEMBL4525777

0.146 0.075 CHEMBL4525778

0.141 0.083 CHEMBL845

CHEMBL4525772
0.0960.0480.112Stem cell growth factor agonist

0.112 0.036 CHEMBL4525772

0.082 0.064 CHEMBL4525778

CHEMBL4525772
0.1140.0660.149Sphingosine 1-phosphate receptor 2 agonist

0.146 0.028 CHEMBL4525772

0.106 0.084 CHEMBL4525777

0.106 0.084 CHEMBL4525778

0.149 0.027 CHEMBL845

0.117 0.059 CHEMBL4525779

0.117 0.059 CHEMBL4525780

CHEMBL845
0.0920.0450.096mTOR complex 2 inhibitor

0.096 0.038 CHEMBL4525772

0.081 0.066 CHEMBL4525777

0.085 0.056 CHEMBL3526715

0.095 0.039 CHEMBL845

CHEMBL4525772
0.0810.0350.321I kappa B kinase 1 inhibitor

0.073 0.043 CHEMBL4525777

0.073 0.045 CHEMBL4525778

0.076 0.04 CHEMBL3526632

0.067 0.052 CHEMBL3526715

0.211 0.005 CHEMBL3526874

0.117 0.016 CHEMBL845

0.321 0.004 CHEMBL3526631

CHEMBL3526631
0.0640.0180.1855 Hydroxytryptamine 2C agonist

0.051 0.027 CHEMBL4525772

0.042 0.034 CHEMBL4525777

0.048 0.029 CHEMBL3526632

0.185 0.004 CHEMBL845

0.039 0.038 CHEMBL4525779

0.043 0.033 CHEMBL4525780

CHEMBL845
0.080.0350.125Phospholipase D inhibitor

0.065 0.064 CHEMBL4525777

0.107 0.011 CHEMBL3526874

0.125 0.005 CHEMBL845

0.071 0.052 CHEMBL3526631

CHEMBL845
0.1030.0590.18Cyclin-dependent kinase 9 inhibitor

0.094 0.07 CHEMBL4525778

0.087 0.079 CHEMBL3526715

0.131 0.04 CHEMBL3526874

0.111 0.052 CHEMBL845

0.18 0.027 CHEMBL3526631

CHEMBL3526631
0.0790.0360.144CDC7 inhibitor

0.066 0.048 CHEMBL4525777

0.069 0.045 CHEMBL4525778

0.087 0.031 CHEMBL3526874

0.105 0.021 CHEMBL845

0.144 0.011 CHEMBL3526631

CHEMBL3526631
0.1370.0940.167Hexokinase inhibitor

0.15 0.079 CHEMBL4525772

0.153 0.075 CHEMBL3526715

0.167 0.06 CHEMBL845

CHEMBL845
0.1280.0850.25Growth factor antagonist

0.164 0.061 CHEMBL4525772

0.25 0.035 CHEMBL4525778

0.144 0.074 CHEMBL3526632

0.108 0.105 CHEMBL1688

0.127 0.086 CHEMBL3526874

CHEMBL4525778
0.070.0280.075 Hydroxytryptamine 1 agonist
0.0910.0490.091Leucine-rich repeat kinase 2 inhibitor

0.083 0.055 CHEMBL4525772

0.074 0.065 CHEMBL4525778

0.072 0.066 CHEMBL845

0.0720.030.086Cyclin B1 inhibitor

0.055 0.05 CHEMBL4525777

0.064 0.038 CHEMBL4525778

0.068 0.034 CHEMBL3526632

0.07 0.032 CHEMBL3526715

0.086 0.017 CHEMBL845

CHEMBL845
0.0790.0380.087Dopamine agonist

0.087 0.033 CHEMBL3526632

0.078 0.038 CHEMBL3526715

CHEMBL3526632
0.1270.0860.414Protein kinase C nu inhibitor

0.117 0.096 CHEMBL3526632

0.274 0.03 CHEMBL3526874

0.156 0.067 CHEMBL845

0.414 0.009 CHEMBL3526631

CHEMBL3526631
0.1610.1210.4Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.22 0.081 CHEMBL3526632

0.229 0.077 CHEMBL3526715

0.254 0.066 CHEMBL3526874

0.159 0.123 CHEMBL845

0.4 0.025 CHEMBL3526631

CHEMBL3526631
0.1160.0750.138MAP kinase 12 inhibitor

0.108 0.087 CHEMBL4525777

0.103 0.093 CHEMBL4525778

0.113 0.079 CHEMBL3526874

0.138 0.051 CHEMBL845

0.133 0.055 CHEMBL3526631

CHEMBL845
0.1550.1150.325Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.208 0.071 CHEMBL3526874

0.209 0.07 CHEMBL845

0.325 0.022 CHEMBL3526631

CHEMBL3526631
0.0540.0140.069Nerve growth factor antagonist

0.069 0.005 CHEMBL4525772

0.052 0.016 CHEMBL4525777

0.043 0.03 CHEMBL4525778

0.04 0.037 CHEMBL3526715

0.045 0.026 CHEMBL845

CHEMBL4525772
0.1280.0890.308Protein kinase (CK1) gamma 1 inhibitor

0.11 0.109 CHEMBL4525777

0.115 0.104 CHEMBL4525778

0.174 0.053 CHEMBL3526874

0.131 0.086 CHEMBL845

0.308 0.019 CHEMBL3526631

CHEMBL3526631
0.1320.0930.279Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.116 0.111 CHEMBL4525778

0.122 0.105 CHEMBL3526632

0.195 0.045 CHEMBL3526715

0.172 0.058 CHEMBL3526874

0.136 0.088 CHEMBL845

0.279 0.02 CHEMBL3526631

CHEMBL3526631
0.0910.0520.191Protein kinase A inhibitor

0.071 0.07 CHEMBL4525777

0.159 0.022 CHEMBL3526874

0.122 0.033 CHEMBL845

0.191 0.015 CHEMBL3526631

CHEMBL3526631
0.1120.0740.112TRKA antagonist

0.107 0.081 CHEMBL845

0.0840.0460.09Nicotinic alpha4beta2 receptor antagonist

0.086 0.044 CHEMBL4525772

0.08 0.05 CHEMBL4525778

0.08 0.05 CHEMBL1688

0.09 0.04 CHEMBL845

CHEMBL845
0.1120.0750.153Acetylcholine muscarinic antagonist

0.106 0.084 CHEMBL4525772

0.114 0.074 CHEMBL3526632

0.153 0.042 CHEMBL1688

CHEMBL1688
0.0930.0560.133Polo-like kinase-1 inhibitor

0.092 0.058 CHEMBL4525772

0.089 0.063 CHEMBL4525777

0.083 0.076 CHEMBL4525778

0.093 0.055 CHEMBL3526632

0.133 0.024 CHEMBL1688

CHEMBL1688
0.1010.0660.114Urease inhibitor

0.103 0.064 CHEMBL3526632

0.114 0.051 CHEMBL845

0.092 0.076 CHEMBL3526631

CHEMBL845
0.1750.1390.373DNA damaging

0.179 0.135 CHEMBL4525772

0.182 0.132 CHEMBL4525778

0.178 0.137 CHEMBL3526632

0.176 0.138 CHEMBL3526715

0.33 0.047 CHEMBL3526874

0.179 0.135 CHEMBL845

0.373 0.034 CHEMBL3526631

CHEMBL3526631
0.0750.0390.086Tyk2 inhibitor

0.086 0.033 CHEMBL4525772

0.075 0.039 CHEMBL845

CHEMBL4525772
0.0830.0470.11Fibroblast growth factor 3 antagonist

0.09 0.04 CHEMBL4525772

0.071 0.064 CHEMBL4525778

0.11 0.027 CHEMBL3526874

0.087 0.043 CHEMBL3526631

CHEMBL3526874
0.0630.0290.076Cyclin B2 inhibitor

0.05 0.046 CHEMBL4525777

0.058 0.035 CHEMBL4525778

0.062 0.03 CHEMBL3526632

0.061 0.03 CHEMBL3526715

0.076 0.017 CHEMBL845

0.053 0.042 CHEMBL3526631

CHEMBL845
0.0870.0530.123Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.077 0.07 CHEMBL4525772

0.082 0.061 CHEMBL4525777

0.077 0.07 CHEMBL4525778

0.088 0.051 CHEMBL3526632

0.082 0.06 CHEMBL3526715

0.081 0.061 CHEMBL3526874

0.079 0.065 CHEMBL845

0.123 0.023 CHEMBL3526631

CHEMBL3526631
0.0830.050.113ErbB-4 antagonist

0.113 0.034 CHEMBL4525772

0.089 0.046 CHEMBL3526632

CHEMBL4525772
0.0420.0090.056Adenosine uptake inhibitor

0.056 0.004 CHEMBL4525772

0.035 0.023 CHEMBL3526632

0.034 0.027 CHEMBL3526715

CHEMBL4525772
0.1370.1040.169Protein kinase (CK1) gamma 3 inhibitor

0.127 0.117 CHEMBL4525778

0.135 0.108 CHEMBL845

0.169 0.07 CHEMBL3526631

CHEMBL3526631
0.060.0270.065 Hydroxytryptamine 1B agonist

0.053 0.037 CHEMBL4525778

0.049 0.044 CHEMBL4525779

0.0610.030.076Cyclin B inhibitor

0.054 0.04 CHEMBL4525778

0.058 0.034 CHEMBL3526632

0.058 0.034 CHEMBL3526715

0.076 0.018 CHEMBL845

CHEMBL845
0.0570.0260.057Potassium channel (Inward rectifier) blocker

0.052 0.031 CHEMBL4525772

0.05 0.034 CHEMBL845

0.049 0.035 CHEMBL4525779

0.0770.0470.077Polo-like kinase-2 inhibitor

0.066 0.057 CHEMBL4525778

0.068 0.055 CHEMBL4525779

0.067 0.056 CHEMBL4525780

0.1030.0730.17CDC-like kinase 3 inhibitor

0.096 0.088 CHEMBL4525777

0.097 0.087 CHEMBL4525778

0.096 0.089 CHEMBL3526632

0.138 0.025 CHEMBL3526874

0.17 0.012 CHEMBL3526631

CHEMBL3526631
0.050.0210.05Phosphodiesterase 6C inhibitor

0.044 0.04 CHEMBL4525772

0.047 0.03 CHEMBL4525778

0.047 0.029 CHEMBL3526632

0.049 0.024 CHEMBL3526715

0.0750.0480.183Telomerase inhibitor

0.102 0.032 CHEMBL4525772

0.072 0.05 CHEMBL1688

0.152 0.02 CHEMBL3526874

0.064 0.059 CHEMBL845

0.183 0.016 CHEMBL3526631

CHEMBL3526631
0.0630.0350.074Dopamine uptake inhibitor

0.074 0.028 CHEMBL4525772

CHEMBL4525772
0.1330.1050.153MAP kinase kinase 4 inhibitor

0.13 0.114 CHEMBL4525777

0.131 0.109 CHEMBL3526632

0.136 0.094 CHEMBL3526715

0.153 0.056 CHEMBL845

CHEMBL845
0.0990.0720.119AMP-activated protein kinase stimulant

0.09 0.085 CHEMBL3526632

0.098 0.073 CHEMBL3526874

0.111 0.057 CHEMBL845

0.119 0.05 CHEMBL3526631

CHEMBL3526631
0.0360.0090.0365 Hydroxytryptamine 1F agonist

0.03 0.013 CHEMBL4525778

0.023 0.021 CHEMBL3526715

0.0540.0270.056Bromodomain-containing protein 3 inhibitor

0.056 0.024 CHEMBL4525772

0.046 0.039 CHEMBL4525777

0.05 0.034 CHEMBL4525778

0.045 0.041 CHEMBL845

CHEMBL4525772
0.1140.0880.202Phosphodiesterase inhibitor

0.131 0.072 CHEMBL4525772

0.168 0.048 CHEMBL3526715

0.202 0.034 CHEMBL1688

0.118 0.084 CHEMBL845

CHEMBL1688
0.1040.0780.105Interleukin 2 antagonist

0.105 0.077 CHEMBL4525772

0.099 0.096 CHEMBL3526632

0.099 0.094 CHEMBL3526874

CHEMBL4525772
0.0360.010.0375 Hydroxytryptamine 6 agonist

0.031 0.015 CHEMBL4525772

0.031 0.016 CHEMBL4525777

0.034 0.012 CHEMBL4525778

0.037 0.009 CHEMBL845

CHEMBL845
0.0490.0240.121Poly(ADP-ribose) polymerase inhibitor

0.121 0.006 CHEMBL1688

0.065 0.015 CHEMBL845

CHEMBL1688
0.0640.0390.085NMDA 2C receptor antagonist

0.06 0.045 CHEMBL3526632

0.071 0.032 CHEMBL3526715

0.085 0.022 CHEMBL845

0.076 0.028 CHEMBL3526631

CHEMBL845
0.060.0370.077Protein kinase C theta inhibitor

0.054 0.047 CHEMBL4525778

0.062 0.034 CHEMBL3526715

0.065 0.029 CHEMBL1688

0.063 0.032 CHEMBL845

0.077 0.017 CHEMBL4525779

0.066 0.028 CHEMBL4525780

CHEMBL4525779
0.0740.0510.126Adenosine A3 receptor antagonist

0.072 0.055 CHEMBL4525772

0.126 0.016 CHEMBL3526874

0.118 0.019 CHEMBL3526631

CHEMBL3526874
0.0550.0330.06mTOR inhibitor

0.06 0.029 CHEMBL4525772

0.05 0.038 CHEMBL3526632

0.047 0.042 CHEMBL845

CHEMBL4525772
0.1080.0860.142MAP kinase kinase inhibitor

0.105 0.089 CHEMBL4525772

0.114 0.08 CHEMBL3526632

0.142 0.056 CHEMBL3526715

0.103 0.091 CHEMBL3526874

0.134 0.061 CHEMBL3526631

CHEMBL3526715
0.1330.1110.317Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.217 0.06 CHEMBL3526874

0.144 0.1 CHEMBL845

0.317 0.026 CHEMBL3526631

CHEMBL3526631
0.1780.1560.222DNA synthesis inhibitor

0.181 0.152 CHEMBL4525772

0.222 0.093 CHEMBL3526632

0.217 0.098 CHEMBL3526715

0.193 0.134 CHEMBL845

CHEMBL3526632
0.0530.0310.063Adenosine A2b receptor antagonist

0.05 0.034 CHEMBL3526874

0.044 0.042 CHEMBL845

0.063 0.022 CHEMBL3526631

CHEMBL3526631
0.0640.0430.0685 Hydroxytryptamine uptake inhibitor

0.061 0.046 CHEMBL4525772

0.062 0.045 CHEMBL3526874

0.068 0.04 CHEMBL845

CHEMBL845
0.130.1090.412CDC-like kinase 2 inhibitor

0.298 0.032 CHEMBL3526874

0.144 0.097 CHEMBL845

0.412 0.012 CHEMBL3526631

CHEMBL3526631
0.0440.0230.072NMDA receptor subunit 3A antagonist

0.055 0.018 CHEMBL3526632

0.034 0.031 CHEMBL3526715

0.046 0.021 CHEMBL3526874

0.072 0.014 CHEMBL845

0.052 0.019 CHEMBL3526631

CHEMBL845
0.0550.0340.065Nicotinic alpha3beta2 receptor antagonist

0.065 0.021 CHEMBL1688

0.051 0.041 CHEMBL845

CHEMBL1688
0.0560.0360.101Glucosylceramidase inhibitor

0.073 0.02 CHEMBL4525772

0.101 0.008 CHEMBL845

CHEMBL845
0.0620.0420.11Adrenaline uptake inhibitor

0.069 0.035 CHEMBL4525772

0.063 0.041 CHEMBL1688

0.11 0.016 CHEMBL3526874

0.066 0.038 CHEMBL845

CHEMBL3526874
0.0320.0120.034Kainate receptor 4 antagonist

0.026 0.016 CHEMBL4525778

0.034 0.011 CHEMBL845

0.026 0.016 CHEMBL3526631

CHEMBL845
0.10.0810.124MAP kinase 13 inhibitor

0.095 0.09 CHEMBL4525777

0.106 0.072 CHEMBL3526874

0.124 0.052 CHEMBL845

0.106 0.072 CHEMBL3526631

CHEMBL845
0.0640.0460.096Aryl hydrocarbon receptor antagonist

0.066 0.043 CHEMBL4525772

0.06 0.054 CHEMBL4525777

0.06 0.054 CHEMBL4525778

0.096 0.015 CHEMBL3526874

0.075 0.032 CHEMBL845

0.089 0.019 CHEMBL3526631

CHEMBL3526874
0.0340.0160.034Phosphodiesterase 6B inhibitor

0.029 0.024 CHEMBL4525778

0.031 0.021 CHEMBL3526632

0.032 0.019 CHEMBL3526715

0.0980.0810.169Glycogen synthase kinase-3 inhibitor

0.114 0.066 CHEMBL4525778

0.152 0.045 CHEMBL3526874

0.169 0.039 CHEMBL3526631

CHEMBL3526631
0.0980.0810.15Glycogen synthase kinase-3 beta inhibitor

0.117 0.063 CHEMBL4525778

0.142 0.047 CHEMBL3526874

0.093 0.087 CHEMBL845

0.15 0.043 CHEMBL3526631

CHEMBL3526631
0.1310.1150.138Ca2+-transporting ATPase inhibitor

0.138 0.081 CHEMBL4525772

0.131 0.115 CHEMBL3526715

CHEMBL4525772
0.070.0550.07MAP3K7 inhibitor

0.069 0.056 CHEMBL3526632

0.0310.0170.042Poly(ADP-ribose) polymerase 2 inhibitor

0.042 0.011 CHEMBL845

CHEMBL845
0.0390.0250.114Poly(ADP-ribose) polymerase 1 inhibitor

0.114 0.005 CHEMBL1688

0.053 0.016 CHEMBL845

CHEMBL1688
0.0470.0330.066CC chemokine 4 receptor antagonist

0.052 0.024 CHEMBL4525772

0.066 0.012 CHEMBL3526874

0.049 0.028 CHEMBL845

0.065 0.013 CHEMBL3526631

CHEMBL3526874
0.1120.0990.29Protein kinase (CK1) gamma inhibitor

0.111 0.101 CHEMBL3526715

0.176 0.054 CHEMBL3526874

0.121 0.089 CHEMBL845

0.29 0.02 CHEMBL3526631

CHEMBL3526631
0.0560.0430.056Adenosine A1 receptor antagonist

0.051 0.048 CHEMBL4525772

0.053 0.045 CHEMBL3526874

0.054 0.045 CHEMBL3526631

0.0420.0290.093Smo receptor antagonist

0.053 0.022 CHEMBL4525772

0.093 0.009 CHEMBL4525778

0.038 0.033 CHEMBL4525779

0.067 0.016 CHEMBL4525780

CHEMBL4525778
0.040.0270.046Cyclin D3 inhibitor

0.038 0.028 CHEMBL4525772

0.035 0.031 CHEMBL4525778

0.046 0.023 CHEMBL845

CHEMBL845
0.0390.0280.051AMPA 4 receptor antagonist

0.039 0.028 CHEMBL845

0.038 0.03 CHEMBL4525780

0.051 0.015 CHEMBL3526631

CHEMBL3526631
0.0480.0360.063Transforming growth factor beta 1 antagonist

0.056 0.029 CHEMBL4525772

0.048 0.036 CHEMBL3526874

0.063 0.024 CHEMBL845

CHEMBL845
0.0580.0480.063Enoyl-[acyl-carrier-protein] reductase inhibitor

0.057 0.05 CHEMBL4525772

0.063 0.038 CHEMBL3526632

CHEMBL3526632
0.0420.0320.068Alpha 1L adrenoreceptor agonist

0.068 0.005 CHEMBL845

CHEMBL845
0.1030.0930.151Epidermal growth factor receptor kinase inhibitor

0.122 0.071 CHEMBL4525772

0.132 0.062 CHEMBL3526632

0.151 0.048 CHEMBL3526874

0.145 0.051 CHEMBL3526631

CHEMBL3526874
0.0920.0830.15Beta glucuronidase inhibitor

0.095 0.077 CHEMBL3526632

0.097 0.074 CHEMBL3526715

0.15 0.025 CHEMBL845

CHEMBL845
0.0570.0480.068Cannabinoid CB1 receptor antagonist

0.065 0.039 CHEMBL4525772

0.068 0.036 CHEMBL845

CHEMBL845
0.0560.0470.062Cyclin A1 inhibitor

0.056 0.046 CHEMBL4525772

0.062 0.034 CHEMBL845

CHEMBL845
0.0340.0250.035Benzodiazepine receptor peripheral-type antagonist

0.032 0.031 CHEMBL4525772

0.035 0.021 CHEMBL845

CHEMBL845
0.0420.0340.072Phosphodiesterase X inhibitor

0.072 0.016 CHEMBL4525772

0.046 0.03 CHEMBL845

CHEMBL4525772
0.0420.0340.072Phosphodiesterase 10A inhibitor

0.072 0.016 CHEMBL4525772

0.046 0.03 CHEMBL845

CHEMBL4525772
0.0370.0280.044DNA gyrase subunit B inhibitor

0.044 0.018 CHEMBL4525772

0.039 0.024 CHEMBL845

CHEMBL4525772
0.0920.0830.238DNA intercalator

0.125 0.055 CHEMBL4525772

0.09 0.085 CHEMBL3526632

0.091 0.084 CHEMBL3526715

0.128 0.053 CHEMBL1688

0.238 0.018 CHEMBL3526874

0.221 0.021 CHEMBL3526631

CHEMBL3526874
0.1160.1080.149Sphingosine 1-phosphate receptor 2 antagonist

0.115 0.111 CHEMBL3526632

0.131 0.072 CHEMBL3526874

0.115 0.11 CHEMBL845

0.149 0.043 CHEMBL3526631

CHEMBL3526631
0.030.0230.037LIM domain kinase 2 inhibitor

0.032 0.019 CHEMBL4525772

0.029 0.025 CHEMBL845

0.037 0.012 CHEMBL4525779

CHEMBL4525779
0.0380.0310.068Kainate receptor antagonist

0.035 0.034 CHEMBL3526874

0.043 0.026 CHEMBL845

0.068 0.013 CHEMBL3526631

CHEMBL3526631
0.1360.1290.165Pyruvate kinase inhibitor

0.15 0.115 CHEMBL4525778

0.165 0.103 CHEMBL3526632

0.134 0.132 CHEMBL3526715

CHEMBL3526632
0.0830.0770.102Platelet activating factor alpha antagonist

0.086 0.073 CHEMBL4525772

0.09 0.069 CHEMBL4525777

0.102 0.058 CHEMBL3526632

0.081 0.079 CHEMBL3526715

CHEMBL3526632
0.0580.0520.065DNA gyrase inhibitor

0.065 0.042 CHEMBL4525772

0.062 0.046 CHEMBL845

CHEMBL4525772
0.1280.1230.191TRKC antagonist

0.191 0.073 CHEMBL3526715

CHEMBL3526715
0.010.0060.011CXC chemokine 3 receptor agonist

0.009 0.008 CHEMBL4525777

0.01 0.007 CHEMBL4525778

0.009 0.008 CHEMBL845

0.011 0.004 CHEMBL4525779

CHEMBL4525779
0.0310.0280.035ATR kinase inhibitor

0.032 0.026 CHEMBL4525772

0.035 0.019 CHEMBL845

CHEMBL845
0.0220.020.022Phosphodiesterase 6G inhibitor
0.0220.020.022Phosphodiesterase 6H inhibitor
0.0530.0510.07Acetylcholine M2 receptor antagonist

0.07 0.037 CHEMBL1688

CHEMBL1688
0.0190.0170.02Kainate receptor 5 antagonist

0.02 0.015 CHEMBL845

CHEMBL845
0.0190.0170.033Imidazoline I1 receptor antagonist

0.033 0.006 CHEMBL845

CHEMBL845
0.0980.0960.138Acetylcholine antagonist

0.138 0.057 CHEMBL1688

CHEMBL1688
0.0690.0670.081Vanilloid 4 agonist

0.081 0.038 CHEMBL4525772

CHEMBL4525772
0.040.0380.0415 Hydroxytryptamine 1A agonist

0.041 0.036 CHEMBL845

CHEMBL845
0.1010.10.111TRKB antagonist

0.111 0.085 CHEMBL4525772

CHEMBL4525772
0.0990.0970.148Cholinergic antagonist

0.148 0.053 CHEMBL1688

CHEMBL1688
0.0520.0510.052Calcium channel T-type blocker
0.0860.0850.136GABA C receptor rho-1 antagonist

0.1 0.062 CHEMBL4525772

0.102 0.059 CHEMBL3526874

0.114 0.046 CHEMBL845

0.136 0.028 CHEMBL3526631

CHEMBL3526631
0.0820.0810.213Protein kinase (CK2) inhibitor

0.093 0.07 CHEMBL4525772

0.086 0.077 CHEMBL3526632

0.136 0.04 CHEMBL3526874

0.096 0.067 CHEMBL845

0.213 0.016 CHEMBL3526631

CHEMBL3526631
0.0330.0320.041Somatostatin 4 agonist

0.034 0.031 CHEMBL3526874

0.041 0.021 CHEMBL845

0.037 0.026 CHEMBL3526631

CHEMBL845
0.0460.0450.073Melanin-concentrating hormone receptor 1 antagonist

0.073 0.023 CHEMBL3526874

CHEMBL3526874
0.050.0490.08EphB4 antagonist

0.065 0.033 CHEMBL4525772

0.058 0.04 CHEMBL3526632

0.08 0.023 CHEMBL1688

CHEMBL1688
0.0240.0240.082AMPA 1 receptor antagonist

0.032 0.019 CHEMBL3526874

0.034 0.018 CHEMBL845

0.028 0.021 CHEMBL3526422

0.082 0.007 CHEMBL3526631

CHEMBL3526631
0.060.0620.076Janus tyrosine kinase 3 inhibitor

0.076 0.047 CHEMBL4525772

0.074 0.049 CHEMBL4525778

CHEMBL4525772
0.0590.0610.061Potassium channel large-conductance Ca-activated activator

0.061 0.058 CHEMBL3526715

CHEMBL3526715
0.0420.0450.061Phosphatidylinositol 3-kinase alpha inhibitor

0.061 0.029 CHEMBL4525772

CHEMBL4525772
0.0310.0340.035Protein kinase C beta I inhibitor

0.035 0.017 CHEMBL4525778

CHEMBL4525778
0.0740.0760.089CDK/cyclin complex inhibitor

0.089 0.06 CHEMBL845

CHEMBL845
0.0160.0190.02Kainate receptor 1 antagonist

0.02 0.016 CHEMBL845

CHEMBL845
0.0470.0520.062CDK4/cyclin D1 inhibitor

0.062 0.037 CHEMBL845

CHEMBL845
0.050.0540.225Protein kinase C iota inhibitor

0.136 0.011 CHEMBL3526874

0.083 0.024 CHEMBL845

0.225 0.004 CHEMBL3526631

CHEMBL3526631
0.0290.0340.08Phosphoglycerate kinase inhibitor

0.05 0.014 CHEMBL4525772

0.054 0.013 CHEMBL3526632

0.08 0.008 CHEMBL3526631

CHEMBL3526631
0.0910.0960.197Protein kinase (CK1) gamma 2 inhibitor

0.097 0.087 CHEMBL3526715

0.131 0.058 CHEMBL3526874

0.104 0.08 CHEMBL845

0.197 0.033 CHEMBL3526631

CHEMBL3526631
0.0560.0620.079Phosphodiesterase 1C inhibitor

0.079 0.02 CHEMBL4525772

CHEMBL4525772
0.0470.0540.057Phosphodiesterase II inhibitor

0.057 0.035 CHEMBL4525772

0.055 0.039 CHEMBL3526715

CHEMBL4525772
0.0320.0380.035Dopamine D3 agonist

0.035 0.033 CHEMBL3526632

CHEMBL3526632
0.0710.0780.207Neuropeptide Y antagonist

0.129 0.027 CHEMBL3526874

0.088 0.049 CHEMBL845

0.207 0.014 CHEMBL3526631

CHEMBL3526631
0.0360.0440.043CF transmembrane conductance regulator antagonist

0.038 0.032 CHEMBL4525772

0.04 0.027 CHEMBL3526632

0.043 0.019 CHEMBL3526715

CHEMBL3526715
0.0380.0470.044Dopamine transporter inhibitor

0.044 0.038 CHEMBL4525772

CHEMBL4525772
0.0770.0870.166Vascular endothelial growth factor 1 antagonist

0.166 0.035 CHEMBL1688

0.089 0.074 CHEMBL3526874

0.094 0.07 CHEMBL3526631

CHEMBL1688
0.0170.0280.031NMDA receptor glycine site antagonist

0.024 0.018 CHEMBL845

0.031 0.012 CHEMBL3526631

CHEMBL3526631
0.0290.040.042Protein kinase (CK2) beta inhibitor

0.042 0.011 CHEMBL4525772

CHEMBL4525772
0.0470.0590.057CDK4/cyclin D inhibitor

0.057 0.043 CHEMBL845

CHEMBL845
0.0520.0640.092Fibroblast growth factor 2 antagonist

0.068 0.043 CHEMBL4525772

0.092 0.027 CHEMBL3526874

0.071 0.04 CHEMBL3526631

CHEMBL3526874
0.0470.0590.053Fatty acid synthase inhibitor

0.053 0.046 CHEMBL4525772

CHEMBL4525772
0.0310.0440.049Dopamine D2 agonist

0.049 0.028 CHEMBL3526632

0.043 0.032 CHEMBL3526715

CHEMBL3526632
0.0190.0330.028Cyclin E2 inhibitor

0.028 0.02 CHEMBL3526631

CHEMBL3526631
0.0250.0390.046Methionyl aminopeptidase 1 inhibitor

0.042 0.01 CHEMBL4525772

0.046 0.008 CHEMBL845

0.039 0.013 CHEMBL3526631

CHEMBL845
0.0170.0310.024Bombesin agonist

0.024 0.013 CHEMBL845

CHEMBL845
0.0820.0960.094Nav1.1 sodium channel blocker

0.094 0.074 CHEMBL4525778

CHEMBL4525778
0.0740.0880.105HIV-1 integrase (Overall Integration) inhibitor

0.105 0.05 CHEMBL845

0.104 0.051 CHEMBL3526631

CHEMBL845
0.0190.0340.023Phosphodiesterase 6A inhibitor

0.022 0.02 CHEMBL3526715

0.023 0.017 CHEMBL3526631

CHEMBL3526631
0.0370.0520.061Glutamate (mGluR5) agonist

0.061 0.017 CHEMBL4525772

CHEMBL4525772
0.0460.0620.065Phosphatidylinositol kinase inhibitor

0.065 0.037 CHEMBL4525772

CHEMBL4525772
0.070.0870.102Caspase 7 inhibitor

0.102 0.026 CHEMBL4525772

CHEMBL4525772
0.2340.2510.4145 Hydroxytryptamine release inhibitor

0.267 0.205 CHEMBL4525772

0.285 0.183 CHEMBL3526874

0.288 0.179 CHEMBL845

0.414 0.07 CHEMBL3526631

CHEMBL3526631
0.0540.0720.064Cannabinoid receptor antagonist

0.064 0.058 CHEMBL4525772

0.063 0.058 CHEMBL845

CHEMBL4525772
0.0920.1090.136Acetylcholine release stimulant

0.136 0.028 CHEMBL4525772

CHEMBL4525772
0.0650.0840.084Bcr-Abl kinase inhibitor

0.084 0.059 CHEMBL4525772

CHEMBL4525772
0.0130.0320.019Bombesin 3 receptor agonist

0.019 0.013 CHEMBL845

CHEMBL845
0.0180.0360.042AMPA 3 receptor antagonist

0.029 0.021 CHEMBL845

0.042 0.013 CHEMBL3526631

CHEMBL3526631
0.0530.0710.11NMDA 2 receptor antagonist

0.084 0.041 CHEMBL3526874

0.099 0.032 CHEMBL845

0.11 0.027 CHEMBL3526631

CHEMBL3526631
0.0110.030.015Nicotinic alpha4 receptor agonist

0.015 0.014 CHEMBL845

CHEMBL845
0.080.0990.128Ferrochelatase inhibitor

0.103 0.068 CHEMBL4525772

0.128 0.049 CHEMBL3526631

CHEMBL3526631
0.0260.0460.031CDK6/cyclin D3 inhibitor

0.031 0.03 CHEMBL845

CHEMBL845
0.0810.1010.123Vascular endothelial growth factor antagonist

0.123 0.067 CHEMBL3526874

0.094 0.088 CHEMBL3526631

CHEMBL3526874
0.10.1210.379Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.177 0.061 CHEMBL3526874

0.145 0.081 CHEMBL845

0.379 0.01 CHEMBL3526631

CHEMBL3526631
0.0150.0360.019Granulocyte colony stimulating factor receptor agonist

0.019 0.01 CHEMBL3526631

CHEMBL3526631
0.1270.1480.1633C-like protease (Human coronavirus) inhibitor

0.141 0.118 CHEMBL4525772

0.163 0.082 CHEMBL845

CHEMBL845
0.0380.0590.049Phosphodiesterase 2A inhibitor

0.049 0.035 CHEMBL4525772

CHEMBL4525772
0.0050.0280.009Corticotropin releasing factor antagonist

0.009 0.007 CHEMBL4525772

CHEMBL4525772
0.1220.1440.228Interleukin 6 antagonist

0.15 0.089 CHEMBL3526874

0.129 0.128 CHEMBL3526422

0.153 0.085 CHEMBL3526420

0.138 0.109 CHEMBL3526421

0.159 0.077 CHEMBL3526423

0.228 0.028 CHEMBL3526631

CHEMBL3526631
0.010.0330.041Cyclin T1 inhibitor

0.024 0.008 CHEMBL3526874

0.041 0.004 CHEMBL3526631

CHEMBL3526631
0.0310.0530.061Chemokine receptor agonist

0.046 0.038 CHEMBL845

0.061 0.026 CHEMBL4525779

CHEMBL4525779
0.0120.0360.019Adenosine kinase inhibitor

0.019 0.017 CHEMBL845

CHEMBL845
0.0510.0750.092Bcl2 antagonist

0.074 0.038 CHEMBL3526422

0.084 0.029 CHEMBL3526420

0.08 0.032 CHEMBL3526421

0.092 0.023 CHEMBL3526423

CHEMBL3526423
0.0810.1060.122Adenylate cyclase inhibitor

0.122 0.066 CHEMBL3526632

CHEMBL3526632
0.0430.0690.095NMDA receptor glycine site agonist

0.056 0.05 CHEMBL845

0.095 0.019 CHEMBL3526631

CHEMBL3526631
0.0160.0420.035CXC chemokine receptor agonist

0.035 0.023 CHEMBL4525779

CHEMBL4525779
0.0890.1150.17Lck kinase inhibitor

0.154 0.063 CHEMBL3526874

0.17 0.054 CHEMBL3526631

CHEMBL3526631
0.0550.0810.065Transforming growth factor antagonist

0.065 0.057 CHEMBL4525772

0.065 0.056 CHEMBL845

CHEMBL845
0.0250.0530.032Vanilloid 4 antagonist

0.032 0.024 CHEMBL4525772

CHEMBL4525772
0.0730.1010.132T cell inhibitor

0.081 0.062 CHEMBL4525772

0.122 0.014 CHEMBL3526874

0.132 0.012 CHEMBL3526631

CHEMBL3526631
0.0360.0640.047Phosphatidylinositol 3-kinase beta inhibitor

0.047 0.038 CHEMBL4525772

CHEMBL4525772
0.0990.1280.127Interleukin 1 antagonist

0.111 0.103 CHEMBL845

0.127 0.079 CHEMBL3526631

CHEMBL3526631
0.0280.0570.034Tryptophan 5 hydroxylase inhibitor

0.034 0.031 CHEMBL4525772

CHEMBL4525772
0.0250.0530.045Estrogen-related receptor beta antagonist

0.045 0.007 CHEMBL4525772

0.03 0.029 CHEMBL3526632

CHEMBL4525772
0.040.0680.076Fibroblast growth factor 4 antagonist

0.076 0.021 CHEMBL4525772

0.064 0.033 CHEMBL3526874

CHEMBL4525772
0.0970.1270.239CDC-like kinase 1 inhibitor

0.181 0.048 CHEMBL3526874

0.239 0.021 CHEMBL3526631

CHEMBL3526631
0.0690.10.109Vascular endothelial growth factor 2 antagonist

0.109 0.066 CHEMBL3526874

CHEMBL3526874
0.0250.0550.033Protein kinase C beta II inhibitor

0.033 0.021 CHEMBL4525778

CHEMBL4525778
0.0460.0770.112Heat shock protein 90 beta antagonist

0.054 0.051 CHEMBL4525772

0.112 0.008 CHEMBL3526632

0.071 0.027 CHEMBL3526715

CHEMBL3526632
0.0710.1020.233Ephrin antagonist

0.092 0.071 CHEMBL3526632

0.233 0.017 CHEMBL1688

0.086 0.077 CHEMBL3526874

0.084 0.079 CHEMBL3526631

CHEMBL1688
0.0760.1080.093Electrolyte absorption antagonist

0.093 0.068 CHEMBL4525772

CHEMBL4525772
0.0190.0520.024Complement factor 1r inhibitor

0.024 0.022 CHEMBL4525772

CHEMBL4525772
0.0740.1070.101MAP kinase kinase 1 inhibitor

0.101 0.055 CHEMBL3526715

CHEMBL3526715
0.070.1040.118MAP kinase kinase kinase inhibitor

0.085 0.081 CHEMBL3526874

0.118 0.052 CHEMBL3526631

CHEMBL3526631
0.0610.0950.092AXL receptor tyrosine kinase inhibitor

0.079 0.062 CHEMBL4525772

0.092 0.046 CHEMBL4525778

CHEMBL4525778
0.070.1050.087D-Ala-D-Ala ligase inhibitor

0.079 0.071 CHEMBL3526715

0.087 0.05 CHEMBL3526631

CHEMBL3526631
0.0750.1110.242Protein kinase (CK2) alpha inhibitor

0.148 0.043 CHEMBL3526874

0.242 0.017 CHEMBL3526631

CHEMBL3526631
0.0360.0740.161Glutamate (mGluR1) antagonist

0.109 0.014 CHEMBL3526874

0.161 0.005 CHEMBL3526631

CHEMBL3526631
0.0380.0760.049Nicotinic receptor alpha4 subunit antagonist

0.049 0.035 CHEMBL4525779

CHEMBL4525779
0.0260.0640.078Glutamate (mGluR1a) antagonist

0.054 0.018 CHEMBL3526874

0.078 0.009 CHEMBL3526631

CHEMBL3526631
0.0880.1280.16Cytokine production inhibitor

0.16 0.055 CHEMBL4525772

CHEMBL4525772
0.1690.2090.204Angiogenesis inhibitor

0.204 0.164 CHEMBL3526632

0.191 0.181 CHEMBL3526874

CHEMBL3526632
0.0740.1150.128Cyclin-dependent kinase 2 inhibitor

0.098 0.072 CHEMBL3526874

0.128 0.048 CHEMBL3526631

CHEMBL3526631
0.0080.0490.028Alpha 2a adrenoreceptor agonist

0.028 0.005 CHEMBL3526874

0.019 0.011 CHEMBL845

0.025 0.007 CHEMBL3526631

CHEMBL3526874
0.0740.1160.124Cystathionine beta-synthase inhibitor

0.107 0.069 CHEMBL4525772

0.119 0.059 CHEMBL3526632

0.124 0.055 CHEMBL3526715

CHEMBL3526715
0.0660.1080.116Topoisomerase I inhibitor

0.116 0.058 CHEMBL4525772

0.099 0.071 CHEMBL3526632

0.106 0.065 CHEMBL3526874

0.111 0.061 CHEMBL3526631

CHEMBL4525772
0.0350.0780.133Raf kinase C inhibitor

0.052 0.049 CHEMBL3526632

0.133 0.017 CHEMBL3526874

0.067 0.037 CHEMBL3526631

CHEMBL3526874
0.040.0830.082Phosphodiesterase III inhibitor

0.082 0.034 CHEMBL1688

CHEMBL1688
0.1080.1550.168Neuropeptide Y1 antagonist

0.127 0.107 CHEMBL4525772

0.156 0.057 CHEMBL3526874

0.168 0.041 CHEMBL3526631

CHEMBL3526631
0.0320.0790.054Neuropeptide Y5 antagonist

0.054 0.033 CHEMBL3526631

CHEMBL3526631
0.0310.0780.103Protein kinase C epsilon inhibitor

0.052 0.039 CHEMBL3526874

0.103 0.012 CHEMBL3526631

CHEMBL3526631
0.0270.0740.05Janus tyrosine kinase 1 inhibitor

0.05 0.046 CHEMBL4525778

CHEMBL4525778
0.0660.1140.095NADH dehydrogenase inhibitor

0.095 0.05 CHEMBL4525772

0.086 0.063 CHEMBL845

0.084 0.066 CHEMBL3526631

CHEMBL4525772
0.0590.1110.151Epidermal growth factor antagonist

0.075 0.073 CHEMBL4525772

0.151 0.023 CHEMBL4525778

0.08 0.065 CHEMBL3526632

0.089 0.054 CHEMBL3526874

0.089 0.054 CHEMBL3526631

CHEMBL4525778
0.0160.0680.035Somatostatin agonist

0.035 0.019 CHEMBL3526631

CHEMBL3526631
0.0470.1020.085Rho-associated kinase I inhibitor

0.068 0.059 CHEMBL845

0.085 0.042 CHEMBL3526631

CHEMBL3526631
0.0320.0870.06H+/K+-transporting ATPase inhibitor

0.06 0.025 CHEMBL3526874

0.053 0.032 CHEMBL3526631

CHEMBL3526874
0.0470.1040.065Nav1.8 sodium channel blocker

0.065 0.063 CHEMBL845

CHEMBL845
0.0640.1220.14Gastric antisecretory

0.14 0.031 CHEMBL3526874

CHEMBL3526874
0.0340.0940.045Heme oxygenase inhibitor

0.045 0.022 CHEMBL4525772

CHEMBL4525772
0.0410.1020.093NMDA receptor agonist

0.076 0.032 CHEMBL3526874

0.093 0.022 CHEMBL3526631

CHEMBL3526631
0.0440.1070.092CXC chemokine receptor antagonist

0.068 0.052 CHEMBL3526874

0.092 0.029 CHEMBL3526631

CHEMBL3526631
0.0460.1090.101Bcl-xL inhibitor

0.078 0.013 CHEMBL3526422

0.081 0.011 CHEMBL3526420

0.08 0.011 CHEMBL3526421

0.101 0.006 CHEMBL3526423

CHEMBL3526423
0.1120.1750.148Antimitotic

0.148 0.123 CHEMBL3526632

0.143 0.128 CHEMBL3526631

CHEMBL3526632
0.0210.0850.053NMDA 2A receptor antagonist

0.049 0.039 CHEMBL3526874

0.053 0.035 CHEMBL3526631

CHEMBL3526631
0.0220.0870.048Glutamate (mGluR group I) agonist

0.048 0.033 CHEMBL4525772

CHEMBL4525772
0.0320.0980.051Lysine-specific demethylase 1A inhibitor

0.051 0.042 CHEMBL4525772

CHEMBL4525772
0.0720.1380.134GABA C receptor antagonist

0.108 0.066 CHEMBL845

0.134 0.04 CHEMBL3526631

CHEMBL3526631
0.0620.1280.189Cyclin-dependent kinase 5 inhibitor

0.128 0.053 CHEMBL3526874

0.189 0.025 CHEMBL3526631

CHEMBL3526631
0.0550.1230.091Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.077 0.076 CHEMBL3526874

0.091 0.055 CHEMBL3526631

CHEMBL3526631
0.0380.1070.078Syk tyrosine kinase inhibitor

0.078 0.042 CHEMBL3526631

CHEMBL3526631
0.0260.0950.045Phenylethanolamine N methyltransferase inhibitor

0.045 0.021 CHEMBL845

CHEMBL845
0.0760.1460.13Vascular endothelial growth factor 3 antagonist

0.119 0.096 CHEMBL3526874

0.13 0.085 CHEMBL3526631

CHEMBL3526631
0.1570.230.197Vasodilator, coronary

0.197 0.185 CHEMBL3526874

CHEMBL3526874
0.0160.090.027MAP3K8 inhibitor

0.027 0.025 CHEMBL3526874

CHEMBL3526874
0.0140.090.086Kinesin-like protein 1 inhibitor

0.057 0.014 CHEMBL1688

0.086 0.009 CHEMBL3526631

CHEMBL3526631
0.0140.090.086Kinesin antagonist

0.057 0.014 CHEMBL1688

0.086 0.009 CHEMBL3526631

CHEMBL3526631
0.0110.0870.062Cholecystokinin antagonist

0.036 0.031 CHEMBL3526422

0.043 0.028 CHEMBL3526420

0.062 0.018 CHEMBL3526421

0.054 0.023 CHEMBL3526423

CHEMBL3526421
0.0760.1540.103Photosensitizer

0.103 0.082 CHEMBL3526631

CHEMBL3526631
0.1670.2460.184MAP kinase kinase 3 inhibitor

0.184 0.176 CHEMBL4525772

CHEMBL4525772
0.0490.1280.1Myeloperoxidase inhibitor

0.079 0.069 CHEMBL3526874

0.1 0.035 CHEMBL3526631

CHEMBL3526631
0.070.150.089Alpha 2d adrenoreceptor antagonist

0.089 0.072 CHEMBL845

CHEMBL845
0.1030.1840.146Sphingosine 1-phosphate receptor 5 antagonist

0.146 0.069 CHEMBL3526631

CHEMBL3526631
0.1480.2330.231Neuropeptide Y2 antagonist

0.179 0.162 CHEMBL3526874

0.231 0.075 CHEMBL3526631

CHEMBL3526631
0.0280.1130.057Purinergic P2X4 antagonist

0.057 0.017 CHEMBL845

CHEMBL845
0.0340.1190.059Epithelial sodium channel blocker

0.059 0.03 CHEMBL3526631

CHEMBL3526631
0.1030.1880.155Tumour necrosis factor antagonist

0.132 0.124 CHEMBL4525772

0.136 0.119 CHEMBL845

0.155 0.094 CHEMBL3526631

CHEMBL3526631
0.0490.1350.059Prolactin release inhibitor

0.059 0.057 CHEMBL4525779

CHEMBL4525779
0.0170.1050.046Cyclin E1 inhibitor

0.046 0.039 CHEMBL3526631

CHEMBL3526631
0.0080.0970.036Cholecystokinin A antagonist

0.036 0.027 CHEMBL3526421

0.034 0.029 CHEMBL3526423

CHEMBL3526421
0.0430.1330.07Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.07 0.068 CHEMBL3526632

CHEMBL3526632
0.0170.1080.034Glutamate (mGluR group II) antagonist

0.034 0.033 CHEMBL4525772

CHEMBL4525772
0.010.1020.043Endothelial nitric-oxide synthase inhibitor

0.037 0.015 CHEMBL3526874

0.043 0.012 CHEMBL3526631

CHEMBL3526631
0.060.1520.106DNA directed RNA polymerase inhibitor

0.106 0.05 CHEMBL4525779

0.083 0.08 CHEMBL4525780

CHEMBL4525779
0.0480.1420.105Butyrylcholinesterase inhibitor

0.098 0.064 CHEMBL4525772

0.105 0.058 CHEMBL3526874

CHEMBL3526874
0.030.1250.045Topoisomerase II beta inhibitor

0.045 0.042 CHEMBL3526874

CHEMBL3526874
0.0180.1150.054Cyclin E inhibitor

0.054 0.045 CHEMBL3526631

CHEMBL3526631
0.0810.1790.216Cholinergic

0.137 0.089 CHEMBL4525772

0.216 0.04 CHEMBL1688

0.123 0.104 CHEMBL3526874

CHEMBL1688
0.0170.1160.05Somatostatin 5 agonist

0.05 0.012 CHEMBL3526631

CHEMBL3526631
0.1280.2280.27Superoxide dismutase inhibitor

0.206 0.111 CHEMBL845

0.27 0.063 CHEMBL3526631

CHEMBL3526631
0.0520.1520.096Histamine H2 receptor antagonist

0.096 0.039 CHEMBL3526874

0.077 0.072 CHEMBL3526631

CHEMBL3526874
0.0360.140.085Sirtuin 1 inhibitor

0.078 0.037 CHEMBL3526422

0.077 0.038 CHEMBL3526420

0.083 0.033 CHEMBL3526421

0.085 0.031 CHEMBL3526423

CHEMBL3526423
0.0410.1450.064Beta 3 adrenoreceptor antagonist

0.064 0.046 CHEMBL3526874

CHEMBL3526874
0.0440.1480.074Adrenaline agonist

0.074 0.065 CHEMBL3526874

CHEMBL3526874
0.0280.1310.049Myc inhibitor

0.049 0.047 CHEMBL845

CHEMBL845
0.0890.1950.144Insulin secretagoues

0.126 0.102 CHEMBL845

0.128 0.099 CHEMBL3526422

0.139 0.087 CHEMBL3526420

0.132 0.095 CHEMBL3526421

0.144 0.081 CHEMBL3526423

CHEMBL3526423
0.0290.1370.08Macrophage colony-stimulating factor 1 receptor antagonist

0.08 0.041 CHEMBL1688

CHEMBL1688
0.060.1740.1Beta amyloid protein antagonist

0.1 0.09 CHEMBL4525772

CHEMBL4525772
0.0050.1220.03Cholecystokinin B antagonist

0.03 0.022 CHEMBL3526421

CHEMBL3526421
0.190.3080.263MAP kinase 1 inhibitor

0.263 0.218 CHEMBL4525772

0.25 0.233 CHEMBL3526632

CHEMBL4525772
0.050.170.12Topoisomerase II inhibitor

0.097 0.089 CHEMBL4525772

0.12 0.067 CHEMBL3526715

0.111 0.076 CHEMBL3526874

0.113 0.074 CHEMBL3526631

CHEMBL3526715
0.0970.2190.147CF transmembrane conductance regulator agonist

0.145 0.086 CHEMBL3526874

0.147 0.081 CHEMBL3526631

CHEMBL3526631
0.0320.1570.063Alpha 1b adrenoreceptor agonist

0.063 0.016 CHEMBL4525778

0.048 0.04 CHEMBL845

CHEMBL4525778
0.1630.2890.323Analgesic

0.323 0.124 CHEMBL1688

CHEMBL1688
0.0870.2180.457Interleukin antagonist

0.161 0.11 CHEMBL3526874

0.429 0.027 CHEMBL3526422

0.411 0.029 CHEMBL3526420

0.415 0.029 CHEMBL3526421

0.457 0.024 CHEMBL3526423

0.284 0.051 CHEMBL3526631

CHEMBL3526423
0.0290.1630.06Bombesin 1 receptor agonist

0.06 0.041 CHEMBL3526874

0.053 0.051 CHEMBL3526423

CHEMBL3526874
0.1460.2810.288Antiobesity

0.288 0.124 CHEMBL845

0.238 0.168 CHEMBL3526421

CHEMBL845
0.0170.1540.041Cholecystokinin B agonist

0.036 0.028 CHEMBL3526422

0.036 0.028 CHEMBL3526420

0.037 0.026 CHEMBL3526421

0.041 0.023 CHEMBL3526423

CHEMBL3526423
0.0780.220.193Heat shock protein 90 antagonist

0.193 0.042 CHEMBL3526632

0.177 0.051 CHEMBL3526715

CHEMBL3526632
0.0860.2280.152DNA methylase inhibitor

0.152 0.116 CHEMBL4525772

CHEMBL4525772
0.130.2790.701Immunomodulator

0.223 0.139 CHEMBL3526422

0.237 0.126 CHEMBL3526420

0.701 0.005 CHEMBL3526421

0.282 0.092 CHEMBL3526423

0.381 0.05 CHEMBL4525779

0.234 0.128 CHEMBL3526631

CHEMBL3526421
0.0180.1690.049Dihydrofolate reductase inhibitor

0.049 0.02 CHEMBL3526631

CHEMBL3526631
0.0470.20.079GABA B receptor agonist

0.079 0.044 CHEMBL3526631

CHEMBL3526631
0.0780.2360.135DNA methyltransferase I inhibitor

0.135 0.123 CHEMBL4525772

CHEMBL4525772
0.0350.1970.073Macrophage migration inhibitory factor inhibitor

0.073 0.061 CHEMBL4525772

CHEMBL4525772
0.0090.1730.035TRPM8 blocker

0.035 0.031 CHEMBL3526631

CHEMBL3526631
0.0940.2610.32Streptokinase A inhibitor

0.32 0.071 CHEMBL3526715

CHEMBL3526715
0.0560.2250.116Hematopoietic

0.107 0.03 CHEMBL3526422

0.102 0.033 CHEMBL3526420

0.108 0.029 CHEMBL3526421

0.116 0.024 CHEMBL3526423

CHEMBL3526423
0.0260.2050.08Parathyroid hormone antagonist

0.061 0.01 CHEMBL3526874

0.08 0.005 CHEMBL3526631

CHEMBL3526631
0.0340.220.16Inducible nitric-oxide synthase inhibitor

0.152 0.015 CHEMBL3526874

0.16 0.014 CHEMBL3526631

CHEMBL3526631
0.010.1990.051Urokinase inhibitor

0.051 0.032 CHEMBL3526631

CHEMBL3526631
0.0240.2160.091Botulinum neurotoxin type A inhibitor

0.063 0.033 CHEMBL3526874

0.091 0.012 CHEMBL3526631

CHEMBL3526631
0.0410.2360.206Glutathione S-transferase inhibitor

0.173 0.008 CHEMBL3526422

0.177 0.008 CHEMBL3526420

0.206 0.005 CHEMBL3526421

0.162 0.01 CHEMBL3526423

CHEMBL3526421
0.0090.2070.027Toll-Like receptor 8 agonist

0.027 0.005 CHEMBL3526631

CHEMBL3526631
0.0680.2670.149Heat shock protein 90 alpha antagonist

0.149 0.088 CHEMBL3526632

0.148 0.088 CHEMBL3526715

CHEMBL3526632
0.1320.3320.199Caspase 3 stimulant

0.199 0.171 CHEMBL3526874

CHEMBL3526874
0.0580.2610.13Peroxidase inhibitor

0.13 0.091 CHEMBL3526632

0.123 0.097 CHEMBL3526631

CHEMBL3526632
0.0470.2510.14Interleukin 5 antagonist

0.121 0.023 CHEMBL3526874

0.14 0.014 CHEMBL3526631

CHEMBL3526631
0.0520.2620.161Toll-Like receptor 3 antagonist

0.161 0.012 CHEMBL3526874

0.09 0.069 CHEMBL3526631

CHEMBL3526874
0.120.3330.167Nitric-oxide synthase stimulant

0.167 0.162 CHEMBL3526631

CHEMBL3526631
0.0580.2730.189Histone deacetylase SIRT1 inhibitor

0.168 0.047 CHEMBL3526422

0.165 0.049 CHEMBL3526420

0.172 0.044 CHEMBL3526421

0.189 0.035 CHEMBL3526423

0.135 0.076 CHEMBL3526631

CHEMBL3526423
0.0640.2820.127Thiol protease inhibitor

0.127 0.101 CHEMBL3526423

CHEMBL3526423
0.0230.2440.051CXC chemokine 1 receptor antagonist

0.051 0.035 CHEMBL3526715

CHEMBL3526715
0.0430.2650.104Acetylcholinesterase inhibitor

0.104 0.098 CHEMBL3526874

CHEMBL3526874
0.0240.2460.099Potassium channel (ATP-sensitive) blocker

0.099 0.016 CHEMBL3526874

0.082 0.026 CHEMBL3526631

CHEMBL3526874
0.0370.2610.301Aminoacyl-tRNA synthetase inhibitor

0.171 0.014 CHEMBL4525777

0.166 0.015 CHEMBL3526874

0.081 0.075 CHEMBL3526422

0.084 0.069 CHEMBL3526420

0.083 0.071 CHEMBL3526421

0.087 0.063 CHEMBL3526423

0.301 0.006 CHEMBL3526631

CHEMBL3526631
0.0260.2550.067S-adenosyl-L-methionine decarboxylase inhibitor

0.067 0.066 CHEMBL3526631

CHEMBL3526631
0.0420.2840.099Carbonic anhydrase III inhibitor

0.099 0.063 CHEMBL3526631

CHEMBL3526631
0.0070.250.029Alpha 1a adrenoreceptor agonist

0.029 0.011 CHEMBL4525778

CHEMBL4525778
0.0150.2580.08Glucagon-like peptide 1 agonist

0.08 0.035 CHEMBL3526422

0.08 0.034 CHEMBL3526420

0.077 0.037 CHEMBL3526421

0.078 0.036 CHEMBL3526423

CHEMBL3526420
0.0340.280.087GABA C receptor agonist

0.087 0.083 CHEMBL3526631

CHEMBL3526631
0.0360.2850.07Cell adhesion molecule inhibitor

0.07 0.069 CHEMBL3526422

CHEMBL3526422
0.0310.2960.166Nitric-oxide synthase inhibitor

0.157 0.02 CHEMBL3526874

0.166 0.017 CHEMBL3526631

CHEMBL3526631
0.0150.2920.039Neurokinin 2 agonist

0.037 0.036 CHEMBL3526422

0.038 0.035 CHEMBL3526420

0.038 0.033 CHEMBL3526421

0.039 0.031 CHEMBL3526423

CHEMBL3526423
0.0580.3410.173Antiamyloidogenic

0.173 0.12 CHEMBL3526874

CHEMBL3526874
0.0030.290.018Prokineticin receptor 1 antagonist

0.018 0.01 CHEMBL3526874

0.017 0.012 CHEMBL3526631

CHEMBL3526874
0.0040.2980.017Dipeptidyl peptidase IX inhibitor

0.017 0.01 CHEMBL4525779

0.016 0.011 CHEMBL4525780

CHEMBL4525779
0.0280.3260.073Carbonic anhydrase VI inhibitor

0.073 0.068 CHEMBL3526631

CHEMBL3526631
0.0970.3960.376Insulysin inhibitor

0.317 0.049 CHEMBL3526422

0.262 0.086 CHEMBL3526420

0.296 0.061 CHEMBL3526421

0.376 0.027 CHEMBL3526423

CHEMBL3526423
0.0420.3410.324Amyloid beta aggregation inhibitor

0.324 0.04 CHEMBL3526715

0.149 0.109 CHEMBL3526874

0.149 0.109 CHEMBL3526631

CHEMBL3526715
0.0040.3050.015Dipeptidyl peptidase VIII inhibitor

0.015 0.012 CHEMBL4525779

0.014 0.012 CHEMBL4525780

CHEMBL4525779
0.1030.4150.35Apoptosis antagonist

0.314 0.076 CHEMBL3526422

0.307 0.081 CHEMBL3526420

0.309 0.08 CHEMBL3526421

0.35 0.056 CHEMBL3526423

CHEMBL3526423
0.1140.4360.327Apoptosis agonist

0.237 0.229 CHEMBL3526874

0.325 0.155 CHEMBL3526422

0.293 0.177 CHEMBL3526420

0.24 0.226 CHEMBL3526421

0.327 0.154 CHEMBL3526423

CHEMBL3526423
0.0650.3910.17Phospholipase C inhibitor

0.14 0.129 CHEMBL3526422

0.15 0.106 CHEMBL3526420

0.163 0.083 CHEMBL3526421

0.17 0.072 CHEMBL3526423

CHEMBL3526423
0.0210.3520.073HIV-1 integrase inhibitor

0.073 0.044 CHEMBL3526715

CHEMBL3526715
0.010.3420.14Phosphodiesterase 4D inhibitor

0.14 0.022 CHEMBL3526715

CHEMBL3526715
0.0140.3470.083Glutamate decarboxylase inhibitor

0.083 0.041 CHEMBL3526423

CHEMBL3526423
0.0670.4040.269Transcription factor NF kappa B inhibitor

0.269 0.114 CHEMBL3526874

0.252 0.126 CHEMBL3526631

CHEMBL3526874
0.0050.3550.03Protocollagen prolyl hydroxylase inhibitor

0.027 0.019 CHEMBL3526422

0.025 0.024 CHEMBL3526420

0.026 0.021 CHEMBL3526421

0.03 0.016 CHEMBL3526423

CHEMBL3526423
0.110.4620.248Ca(v)3.3 blocker

0.248 0.104 CHEMBL4525780

CHEMBL4525780
0.0360.4080.116Cell adhesion inhibitor

0.116 0.068 CHEMBL3526422

CHEMBL3526422
0.0070.3820.055Toll-Like receptor 2 agonist

0.055 0.022 CHEMBL3526423

CHEMBL3526423
0.0330.410.2Anticoagulant

0.175 0.064 CHEMBL3526422

0.163 0.07 CHEMBL3526420

0.184 0.06 CHEMBL3526421

0.2 0.053 CHEMBL3526423

CHEMBL3526423
0.0370.4150.356Immunostimulant

0.266 0.09 CHEMBL3526422

0.356 0.063 CHEMBL3526420

0.28 0.085 CHEMBL3526421

0.34 0.067 CHEMBL3526423

CHEMBL3526420
0.0230.4350.205Chelator

0.205 0.024 CHEMBL3526715

0.1 0.077 CHEMBL3526423

CHEMBL3526715
0.0540.4970.238Antithrombotic

0.238 0.136 CHEMBL3526423

CHEMBL3526423
0.0210.4680.136Histone deacetylase class III inhibitor

0.136 0.056 CHEMBL3526422

0.104 0.086 CHEMBL3526420

0.11 0.08 CHEMBL3526421

0.128 0.063 CHEMBL3526423

CHEMBL3526422
0.0170.4670.044Integrin alpha1beta1 antagonist

0.044 0.013 CHEMBL3526422

CHEMBL3526422
0.0190.4970.073Somatostatin 1 agonist

0.073 0.06 CHEMBL3526423

0.073 0.061 CHEMBL3526631

CHEMBL3526631
0.0260.5050.14Nav1.4 sodium channel blocker

0.131 0.044 CHEMBL3526422

0.139 0.039 CHEMBL3526420

0.134 0.041 CHEMBL3526421

0.14 0.038 CHEMBL3526423

CHEMBL3526423
0.0350.5170.182Interleukin 4 antagonist

0.164 0.039 CHEMBL3526874

0.182 0.029 CHEMBL3526631

CHEMBL3526631
0.0210.5080.113Bone formation stimulant

0.113 0.093 CHEMBL3526423

CHEMBL3526423
0.0180.5130.094Aminopeptidase B inhibitor

0.094 0.069 CHEMBL3526423

CHEMBL3526423
0.0160.520.104Estrogen receptor beta antagonist

0.104 0.057 CHEMBL3526632

CHEMBL3526632
0.0230.5460.292Platelet antagonist

0.242 0.076 CHEMBL3526422

0.254 0.071 CHEMBL3526420

0.23 0.082 CHEMBL3526421

0.292 0.055 CHEMBL3526423

CHEMBL3526423
0.0770.6130.354Interleukin 2 agonist

0.334 0.053 CHEMBL3526422

0.339 0.051 CHEMBL3526420

0.344 0.048 CHEMBL3526421

0.354 0.044 CHEMBL3526423

CHEMBL3526423
0.0160.5770.269Thrombolytic

0.23 0.039 CHEMBL3526422

0.236 0.037 CHEMBL3526420

0.238 0.037 CHEMBL3526421

0.269 0.029 CHEMBL3526423

CHEMBL3526423
0.0030.5670.042GP IIb/IIIa receptor antagonist

0.042 0.039 CHEMBL3526423

CHEMBL3526423
0.0110.5790.131Bronchodilator

0.131 0.039 CHEMBL1688

CHEMBL1688
0.0150.5870.092Factor XII inhibitor

0.086 0.054 CHEMBL3526422

0.087 0.053 CHEMBL3526420

0.09 0.049 CHEMBL3526421

0.092 0.046 CHEMBL3526423

CHEMBL3526423
0.0170.6120.106Estrogen antagonist

0.106 0.084 CHEMBL3526632

CHEMBL3526632
0.0040.6010.033Catechol O-methyltransferase inhibitor

0.033 0.022 CHEMBL3526715

CHEMBL3526715
0.0360.6440.111Folate antagonist

0.099 0.067 CHEMBL3526422

0.1 0.064 CHEMBL3526420

0.103 0.059 CHEMBL3526421

0.111 0.048 CHEMBL3526423

CHEMBL3526423
0.0440.6630.263Cyclophilin D inhibitor

0.263 0.198 CHEMBL4525779

CHEMBL4525779
0.0050.6350.056Selectin antagonist

0.056 0.053 CHEMBL3526423

CHEMBL3526423
0.0390.670.128Factor V inhibitor

0.126 0.034 CHEMBL3526422

0.127 0.033 CHEMBL3526420

0.126 0.034 CHEMBL3526421

0.128 0.032 CHEMBL3526423

CHEMBL3526423
0.0030.6430.034Leukotriene A4 hydrolase inhibitor

0.034 0.029 CHEMBL3526423

CHEMBL3526423
0.0660.7530.236Peptidyltransferase inhibitor

0.22 0.076 CHEMBL3526422

0.22 0.076 CHEMBL3526420

0.228 0.068 CHEMBL3526421

0.236 0.061 CHEMBL3526423

CHEMBL3526423
0.0130.7250.343Angiogenesis stimulant

0.304 0.048 CHEMBL3526422

0.307 0.047 CHEMBL3526420

0.312 0.045 CHEMBL3526421

0.343 0.034 CHEMBL3526423

CHEMBL3526423
0.0320.8050.246Growth hormone agonist

0.204 0.057 CHEMBL3526422

0.204 0.057 CHEMBL3526420

0.215 0.053 CHEMBL3526421

0.246 0.044 CHEMBL3526423

CHEMBL3526423
0.0040.7880.053Angiotensin-converting enzyme inhibitor

0.05 0.047 CHEMBL3526422

0.05 0.046 CHEMBL3526421

0.053 0.042 CHEMBL3526423

CHEMBL3526423
0.0040.920.086Protease inhibitor

0.086 0.078 CHEMBL3526423

CHEMBL3526423
0.020.9390.348Sodium/bile acid cotransporter inhibitor

0.321 0.061 CHEMBL3526422

0.321 0.061 CHEMBL3526420

0.326 0.057 CHEMBL3526421

0.348 0.041 CHEMBL3526423

CHEMBL3526423
Ext Pa Pi Pmax Activity Other Results ID Pa_max