| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.832 | 0.004 | 0.878 | Antithrombotic | 0.82 0.004 CHEMBL107471 0.878 0.003 CHEMBL65267 | CHEMBL65267 | |
| 0.584 | 0.007 | 0.803 | Platelet antagonist | 0.627 0.005 CHEMBL107471 0.803 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.578 | 0.006 | 0.858 | Anticoagulant | 0.658 0.005 CHEMBL107471 0.858 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.448 | 0.041 | 0.448 | Vasodilator, peripheral | 0.31 0.092 CHEMBL65267 | ||
| 0.415 | 0.045 | 0.415 | Immunostimulant | 0.288 0.082 CHEMBL107471 0.378 0.056 CHEMBL65267 | ||
| 0.373 | 0.022 | 0.625 | Platelet aggregation inhibitor | 0.413 0.017 CHEMBL107471 0.625 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.238 | 0.005 | 0.627 | GP IIb/IIIa receptor antagonist | 0.34 0.004 CHEMBL107471 0.627 0.003 CHEMBL65267 | CHEMBL65267 | |
| 0.279 | 0.066 | 0.279 | Cardiotonic | 0.164 0.159 CHEMBL107471 0.198 0.121 CHEMBL65267 | ||
| 0.208 | 0.005 | 0.279 | Factor Xa inhibitor | 0.115 0.011 CHEMBL107471 0.279 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.288 | 0.097 | 0.288 | Vasodilator, coronary | 0.198 0.184 CHEMBL65267 | ||
| 0.254 | 0.067 | 0.254 | Vasodilator | 0.174 0.127 CHEMBL65267 | ||
| 0.224 | 0.041 | 0.383 | Thrombolytic | 0.279 0.028 CHEMBL107471 0.383 0.013 CHEMBL65267 | CHEMBL65267 | |
| 0.211 | 0.029 | 0.514 | Hemostatic | 0.31 0.015 CHEMBL107471 0.514 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.208 | 0.075 | 0.208 | Psychostimulant | 0.156 0.111 CHEMBL65267 | ||
| 0.132 | 0.009 | 0.258 | Factor VIIa inhibitor | 0.154 0.007 CHEMBL107471 0.258 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.135 | 0.014 | 0.331 | Thrombin inhibitor | 0.163 0.009 CHEMBL107471 0.331 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.169 | 0.057 | 0.169 | NOS3 expression enhancer | |||
| 0.135 | 0.027 | 0.135 | Acetylcholine M3 receptor agonist | 0.088 0.053 CHEMBL65267 | ||
| 0.11 | 0.014 | 0.39 | Trypsin inhibitor | 0.128 0.009 CHEMBL107471 0.39 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.212 | 0.116 | 0.212 | Tyrosine 3 hydroxylase inhibitor | 0.184 0.168 CHEMBL65267 | ||
| 0.215 | 0.126 | 0.247 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.21 0.14 CHEMBL107471 0.247 0.069 CHEMBL65267 | CHEMBL65267 | |
| 0.097 | 0.011 | 0.321 | Factor X inhibitor | 0.114 0.009 CHEMBL107471 0.321 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.09 | 0.014 | 0.09 | Nitric oxide donor | |||
| 0.236 | 0.16 | 0.236 | Immunosuppressant | 0.227 0.169 CHEMBL107471 | ||
| 0.164 | 0.092 | 0.369 | Platelet adhesion inhibitor | 0.187 0.078 CHEMBL107471 0.369 0.016 CHEMBL65267 | CHEMBL65267 | |
| 0.089 | 0.019 | 0.199 | Urokinase inhibitor | 0.115 0.013 CHEMBL107471 0.199 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.201 | 0.137 | 0.201 | Transcription factor STAT inhibitor | |||
| 0.067 | 0.006 | 0.121 | Trypsin II inhibitor | 0.071 0.006 CHEMBL107471 0.121 0.003 CHEMBL65267 | CHEMBL65267 | |
| 0.113 | 0.053 | 0.117 | Protease inhibitor | 0.091 0.074 CHEMBL107471 0.117 0.05 CHEMBL65267 | CHEMBL65267 | |
| 0.197 | 0.138 | 0.197 | Transcription factor STAT3 inhibitor | |||
| 0.144 | 0.092 | 0.255 | Growth hormone agonist | 0.224 0.051 CHEMBL107471 0.255 0.042 CHEMBL65267 | CHEMBL65267 | |
| 0.18 | 0.136 | 0.195 | Spasmolytic | 0.195 0.124 CHEMBL65267 | CHEMBL65267 | |
| 0.072 | 0.031 | 0.177 | Plasminogen activator inhibitor | 0.088 0.021 CHEMBL107471 0.177 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.064 | 0.025 | 0.07 | Angiotensin-converting enzyme inhibitor | 0.067 0.022 CHEMBL107471 0.07 0.02 CHEMBL65267 | CHEMBL65267 | |
| 0.052 | 0.015 | 0.075 | Acid-sensing ion channel blocker | 0.052 0.014 CHEMBL107471 0.075 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.109 | 0.076 | 0.155 | Adenylate cyclase inhibitor | 0.155 0.042 CHEMBL107471 0.153 0.043 CHEMBL65267 | CHEMBL107471 | |
| 0.044 | 0.014 | 0.317 | Trypsin I inhibitor | 0.057 0.01 CHEMBL107471 0.317 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.056 | 0.029 | 0.258 | Plasmin inhibitor | 0.101 0.018 CHEMBL107471 0.258 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.061 | 0.034 | 0.081 | Ribonucleoside-diphosphate reductase inhibitor | 0.081 0.024 CHEMBL107471 0.047 0.043 CHEMBL65267 | CHEMBL107471 | |
| 0.058 | 0.031 | 0.058 | Acetylcholine M2 receptor agonist | |||
| 0.055 | 0.028 | 0.073 | Antimetabolite | 0.073 0.021 CHEMBL65267 | CHEMBL65267 | |
| 0.057 | 0.032 | 0.057 | Lysine-specific demethylase 1A inhibitor | |||
| 0.061 | 0.036 | 0.081 | Ribonucleotide reductase inhibitor | 0.081 0.026 CHEMBL107471 0.047 0.044 CHEMBL65267 | CHEMBL107471 | |
| 0.244 | 0.219 | 0.404 | Cyclophilin D inhibitor | 0.316 0.149 CHEMBL107471 0.404 0.089 CHEMBL65267 | CHEMBL65267 | |
| 0.127 | 0.102 | 0.175 | Thiol protease inhibitor | 0.175 0.051 CHEMBL65267 | CHEMBL65267 | |
| 0.053 | 0.029 | 0.113 | Factor III inhibitor | 0.067 0.012 CHEMBL107471 0.113 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.078 | 0.057 | 0.099 | Chymotrypsin inhibitor | 0.094 0.04 CHEMBL107471 0.099 0.037 CHEMBL65267 | CHEMBL65267 | |
| 0.056 | 0.04 | 0.18 | Kallikrein 1 inhibitor | 0.058 0.036 CHEMBL107471 0.18 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.029 | 0.014 | 0.029 | Thyroid hormone agonist | |||
| 0.038 | 0.025 | 0.107 | Tryptase inhibitor | 0.036 0.027 CHEMBL107471 0.107 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.058 | 0.052 | 0.064 | Caspase 9 inhibitor | 0.064 0.039 CHEMBL65267 | CHEMBL65267 | |
| 0.022 | 0.018 | 0.022 | ICAM 1 antagonist | |||
| 0.048 | 0.046 | 0.057 | Elastase inhibitor | 0.057 0.033 CHEMBL65267 | CHEMBL65267 | |
| 0.154 | 0.153 | 0.291 | Tumour necrosis factor alpha release inhibitor | 0.291 0.057 CHEMBL107471 | CHEMBL107471 | |
| 0.036 | 0.035 | 0.042 | Integrin alpha1beta1 antagonist | 0.038 0.026 CHEMBL107471 0.042 0.017 CHEMBL65267 | CHEMBL65267 | |
| 0.092 | 0.092 | 0.115 | Factor V inhibitor | 0.098 0.073 CHEMBL107471 0.115 0.044 CHEMBL65267 | CHEMBL65267 | |
| 0.069 | 0.073 | 0.13 | Cell adhesion molecule inhibitor | 0.13 0.02 CHEMBL65267 | CHEMBL65267 | |
| 0.046 | 0.052 | 0.088 | Aminopeptidase microsomal inhibitor | 0.088 0.021 CHEMBL107471 | CHEMBL107471 | |
| 0.035 | 0.042 | 0.065 | Leukocyte elastase inhibitor | 0.065 0.016 CHEMBL65267 | CHEMBL65267 | |
| 0.017 | 0.024 | 0.02 | Purinergic P2Y12 antagonist | 0.02 0.019 CHEMBL65267 | CHEMBL65267 | |
| 0.094 | 0.103 | 0.183 | Cell adhesion inhibitor | 0.1 0.09 CHEMBL107471 0.183 0.03 CHEMBL65267 | CHEMBL65267 | |
| 0.013 | 0.024 | 0.18 | Integrin beta3 antagonist | 0.033 0.008 CHEMBL107471 0.18 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.02 | 0.034 | 0.15 | Factor VII inhibitor | 0.029 0.022 CHEMBL107471 0.15 0.004 CHEMBL65267 | CHEMBL65267 | |
| 0.086 | 0.101 | 0.127 | Folate antagonist | 0.112 0.046 CHEMBL107471 0.127 0.034 CHEMBL65267 | CHEMBL65267 | |
| 0.021 | 0.037 | 0.03 | Caspase 2 inhibitor | 0.03 0.023 CHEMBL65267 | CHEMBL65267 | |
| 0.024 | 0.04 | 0.044 | Histone deacetylase 2 inhibitor | 0.044 0.016 CHEMBL107471 | CHEMBL107471 | |
| 0.012 | 0.029 | 0.035 | Factor IX inhibitor | 0.035 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.04 | 0.058 | 0.043 | Baculoviral IAP repeat-containing protein inhibitor | 0.043 0.042 CHEMBL65267 | CHEMBL65267 | |
| 0.192 | 0.211 | 0.304 | Toll-Like receptor 7 agonist | 0.304 0.107 CHEMBL65267 | CHEMBL65267 | |
| 0.027 | 0.046 | 0.047 | ADAM10 endopeptidase inhibitor | 0.047 0.011 CHEMBL107471 | CHEMBL107471 | |
| 0.032 | 0.051 | 0.067 | Aminopeptidase N inhibitor | 0.067 0.021 CHEMBL107471 | CHEMBL107471 | |
| 0.022 | 0.043 | 0.039 | Calcitonin receptor agonist | 0.039 0.02 CHEMBL65267 | CHEMBL65267 | |
| 0.04 | 0.061 | 0.122 | Factor IXa inhibitor | 0.122 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.191 | 0.214 | 0.302 | Toll-Like receptor agonist | 0.302 0.11 CHEMBL65267 | CHEMBL65267 | |
| 0.025 | 0.056 | 0.037 | Ceramide glucosyltransferase inhibitor | 0.037 0.021 CHEMBL65267 | CHEMBL65267 | |
| 0.028 | 0.06 | 0.046 | Integrin alpha5beta1 antagonist | 0.037 0.035 CHEMBL107471 0.046 0.022 CHEMBL65267 | CHEMBL65267 | |
| 0.101 | 0.134 | 0.225 | Diuretic | 0.225 0.036 CHEMBL65267 | CHEMBL65267 | |
| 0.02 | 0.053 | 0.187 | Integrin antagonist | 0.076 0.02 CHEMBL107471 0.187 0.008 CHEMBL65267 | CHEMBL65267 | |
| 0.041 | 0.075 | 0.093 | Sphingosine kinase 2 inhibitor | 0.093 0.01 CHEMBL65267 | CHEMBL65267 | |
| 0.113 | 0.148 | 0.229 | Angiogenesis stimulant | 0.186 0.102 CHEMBL107471 0.229 0.08 CHEMBL65267 | CHEMBL65267 | |
| 0.042 | 0.077 | 0.11 | Epithelial sodium channel blocker | 0.11 0.005 CHEMBL65267 | CHEMBL65267 | |
| 0.04 | 0.076 | 0.058 | Selectin antagonist | 0.058 0.051 CHEMBL107471 | CHEMBL107471 | |
| 0.015 | 0.053 | 0.066 | Prostacyclin antagonist | 0.046 0.015 CHEMBL107471 0.066 0.008 CHEMBL65267 | CHEMBL65267 | |
| 0.029 | 0.067 | 0.041 | Neurotensin receptor antagonist | 0.041 0.036 CHEMBL65267 | CHEMBL65267 | |
| 0.007 | 0.046 | 0.014 | Prostacyclin agonist | 0.014 0.012 CHEMBL65267 | CHEMBL65267 | |
| 0.011 | 0.054 | 0.045 | Histone deacetylase 6 inhibitor | 0.045 0.011 CHEMBL107471 | CHEMBL107471 | |
| 0.012 | 0.054 | 0.046 | Histone deacetylase class IIb inhibitor | 0.046 0.011 CHEMBL107471 | CHEMBL107471 | |
| 0.011 | 0.054 | 0.019 | Complement factor 1 inhibitor | 0.019 0.01 CHEMBL65267 | CHEMBL65267 | |
| 0.013 | 0.064 | 0.056 | Histone deacetylase class II inhibitor | 0.056 0.011 CHEMBL107471 | CHEMBL107471 | |
| 0.027 | 0.081 | 0.122 | Kallikrein inhibitor | 0.122 0.008 CHEMBL65267 | CHEMBL65267 | |
| 0.063 | 0.118 | 0.103 | Factor XII inhibitor | 0.103 0.035 CHEMBL65267 | CHEMBL65267 | |
| 0.013 | 0.075 | 0.037 | Histone deacetylase 4 inhibitor | 0.037 0.019 CHEMBL107471 | CHEMBL107471 | |
| 0.154 | 0.218 | 0.206 | Gastrin inhibitor | 0.206 0.139 CHEMBL65267 | CHEMBL65267 | |
| 0.029 | 0.093 | 0.055 | Collagenase inhibitor | 0.055 0.023 CHEMBL107471 | CHEMBL107471 | |
| 0.009 | 0.075 | 0.02 | Integrin beta5 antagonist | 0.02 0.015 CHEMBL65267 | CHEMBL65267 | |
| 0.069 | 0.136 | 0.145 | DNA polymerase I inhibitor | 0.142 0.054 CHEMBL107471 0.145 0.052 CHEMBL65267 | CHEMBL65267 | |
| 0.167 | 0.236 | 0.196 | Apoptosis antagonist | 0.196 0.184 CHEMBL65267 | CHEMBL65267 | |
| 0.024 | 0.094 | 0.057 | Neuropeptide agonist | 0.057 0.039 CHEMBL65267 | CHEMBL65267 | |
| 0.012 | 0.081 | 0.065 | Plasma kallikrein inhibitor | 0.065 0.008 CHEMBL65267 | CHEMBL65267 | |
| 0.135 | 0.209 | 0.213 | Hypoglycemic | 0.213 0.101 CHEMBL65267 | CHEMBL65267 | |
| 0.024 | 0.105 | 0.057 | Sphingosine kinase 1 inhibitor | 0.057 0.01 CHEMBL65267 | CHEMBL65267 | |
| 0.14 | 0.225 | 0.217 | Peptidyltransferase inhibitor | 0.164 0.16 CHEMBL107471 0.217 0.079 CHEMBL65267 | CHEMBL65267 | |
| 0.012 | 0.097 | 0.042 | Complement C3a chemotactic receptor antagonist | 0.042 0.031 CHEMBL65267 | CHEMBL65267 | |
| 0.013 | 0.103 | 0.035 | Histone deacetylase 11 inhibitor | 0.035 0.019 CHEMBL107471 | CHEMBL107471 | |
| 0.013 | 0.103 | 0.035 | Histone deacetylase class IV inhibitor | 0.035 0.019 CHEMBL107471 | CHEMBL107471 | |
| 0.01 | 0.102 | 0.053 | Lysine carboxypeptidase inhibitor | 0.053 0.007 CHEMBL65267 | CHEMBL65267 | |
| 0.048 | 0.143 | 0.097 | Aminopeptidase B inhibitor | 0.097 0.067 CHEMBL107471 | CHEMBL107471 | |
| 0.039 | 0.135 | 0.083 | Aminopeptidase I inhibitor | 0.083 0.039 CHEMBL65267 | CHEMBL65267 | |
| 0.034 | 0.133 | 0.083 | Sphingosine kinase inhibitor | 0.083 0.014 CHEMBL65267 | CHEMBL65267 | |
| 0.022 | 0.125 | 0.047 | Neuraminidase (Influenza A) inhibitor | 0.047 0.028 CHEMBL65267 | CHEMBL65267 | |
| 0.009 | 0.115 | 0.042 | Histone deacetylase class IIa inhibitor | 0.042 0.016 CHEMBL107471 | CHEMBL107471 | |
| 0.034 | 0.14 | 0.065 | Neuraminidase (influenza) inhibitor | 0.065 0.043 CHEMBL65267 | CHEMBL65267 | |
| 0.114 | 0.222 | 0.16 | Neurotensin receptor agonist | 0.16 0.079 CHEMBL65267 | CHEMBL65267 | |
| 0.023 | 0.133 | 0.061 | Neuraminidase inhibitor | 0.061 0.043 CHEMBL65267 | CHEMBL65267 | |
| 0.064 | 0.184 | 0.165 | Alpha-N-acetylglucosaminidase inhibitor | 0.112 0.086 CHEMBL107471 0.165 0.047 CHEMBL65267 | CHEMBL65267 | |
| 0.008 | 0.14 | 0.028 | Histone deacetylase 10 inhibitor | 0.028 0.022 CHEMBL107471 | CHEMBL107471 | |
| 0.053 | 0.194 | 0.109 | Interleukin 1 beta converting enzyme inhibitor | 0.109 0.046 CHEMBL65267 | CHEMBL65267 | |
| 0.007 | 0.15 | 0.035 | Histone deacetylase 1 inhibitor | 0.035 0.014 CHEMBL107471 | CHEMBL107471 | |
| 0.085 | 0.231 | 0.185 | Insulin sensitizer | 0.185 0.09 CHEMBL65267 | CHEMBL65267 | |
| 0.008 | 0.155 | 0.048 | Histone deacetylase 5 inhibitor | 0.048 0.017 CHEMBL107471 | CHEMBL107471 | |
| 0.031 | 0.179 | 0.133 | Cathepsin G inhibitor | 0.133 0.024 CHEMBL65267 | CHEMBL65267 | |
| 0.043 | 0.197 | 0.098 | Expectorant | 0.098 0.071 CHEMBL65267 | CHEMBL65267 | |
| 0.052 | 0.214 | 0.103 | Mucolytic | 0.103 0.073 CHEMBL65267 | CHEMBL65267 | |
| 0.143 | 0.322 | 0.186 | 5 Hydroxytryptamine uptake stimulant | 0.186 0.183 CHEMBL65267 | CHEMBL65267 | |
| 0.012 | 0.197 | 0.042 | Factor XIa inhibitor | 0.042 0.027 CHEMBL65267 | CHEMBL65267 | |
| 0.054 | 0.254 | 0.103 | Glutamate (mGluR7) agonist | 0.103 0.053 CHEMBL65267 | CHEMBL65267 | |
| 0.121 | 0.33 | 0.244 | Sodium/bile acid cotransporter inhibitor | 0.206 0.18 CHEMBL107471 0.244 0.135 CHEMBL65267 | CHEMBL65267 | |
| 0.047 | 0.268 | 0.094 | Nav1.4 sodium channel blocker | 0.094 0.086 CHEMBL65267 | CHEMBL65267 | |
| 0.005 | 0.228 | 0.031 | Factor XI inhibitor | 0.031 0.028 CHEMBL65267 | CHEMBL65267 | |
| 0.129 | 0.362 | 0.275 | Interleukin 2 agonist | 0.214 0.166 CHEMBL107471 0.275 0.094 CHEMBL65267 | CHEMBL65267 | |
| 0.112 | 0.351 | 0.227 | Insulysin inhibitor | 0.227 0.12 CHEMBL107471 | CHEMBL107471 | |
| 0.094 | 0.341 | 0.226 | DNA synthesis inhibitor | 0.226 0.087 CHEMBL65267 | CHEMBL65267 | |
| 0.067 | 0.323 | 0.157 | Antipruritic | 0.157 0.087 CHEMBL65267 | CHEMBL65267 | |
| 0.059 | 0.321 | 0.214 | Interleukin agonist | 0.214 0.108 CHEMBL65267 | CHEMBL65267 | |
| 0.037 | 0.35 | 0.121 | Cathepsin H inhibitor | 0.121 0.074 CHEMBL65267 | CHEMBL65267 | |
| 0.118 | 0.481 | 0.267 | 5 Hydroxytryptamine release inhibitor | 0.267 0.205 CHEMBL65267 | CHEMBL65267 | |
| 0.07 | 0.455 | 0.242 | Antiobesity | 0.242 0.164 CHEMBL65267 | CHEMBL65267 | |
| 0.042 | 0.427 | 0.306 | Aldehyde oxidase inhibitor | 0.306 0.065 CHEMBL65267 | CHEMBL65267 | |
| 0.056 | 0.477 | 0.185 | Superoxide dismutase inhibitor | 0.185 0.135 CHEMBL65267 | CHEMBL65267 | |
| 0.017 | 0.459 | 0.113 | Nitric-oxide synthase inhibitor | 0.113 0.043 CHEMBL65267 | CHEMBL65267 | |
| 0.018 | 0.607 | 0.102 | HIV-1 integrase (Overall Integration) inhibitor | 0.102 0.052 CHEMBL65267 | CHEMBL65267 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |