| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.869 | 0.002 | 0.88 | Antibacterial | 0.845 0.003 CHEMBL451929 0.856 0.002 CHEMBL3544891 0.88 0.002 CHEMBL3544697 0.859 0.002 CHEMBL3544548 0.809 0.004 CHEMBL447570 0.857 0.002 CHEMBL3544713 | CHEMBL3544697 | |
| 0.76 | 0.002 | 0.76 | Pregnane X receptor agonist | 0.638 0.002 CHEMBL451929 0.469 0.003 CHEMBL3544891 0.53 0.002 CHEMBL3544697 0.469 0.003 CHEMBL3544548 0.402 0.003 CHEMBL447570 0.416 0.003 CHEMBL3544713 | ||
| 0.696 | 0.008 | 0.731 | Cholesterol antagonist | 0.627 0.015 CHEMBL451929 0.707 0.007 CHEMBL3544891 0.731 0.006 CHEMBL3544697 0.715 0.007 CHEMBL3544548 0.487 0.035 CHEMBL447570 0.664 0.011 CHEMBL3544713 | CHEMBL3544697 | |
| 0.664 | 0 | 0.664 | Antibiotic Rifamycin-like | 0.319 0 CHEMBL451929 0.389 0 CHEMBL3544891 0.459 0 CHEMBL3544697 0.536 0 CHEMBL3544548 0.12 0 CHEMBL447570 0.219 0 CHEMBL3544713 | ||
| 0.643 | 0.004 | 0.674 | RNA-directed DNA polymerase inhibitor | 0.61 0.005 CHEMBL451929 0.658 0.003 CHEMBL3544891 0.674 0.003 CHEMBL3544697 0.63 0.004 CHEMBL3544548 0.574 0.007 CHEMBL447570 0.635 0.004 CHEMBL3544713 | CHEMBL3544697 | |
| 0.531 | 0.004 | 0.535 | DNA directed RNA polymerase inhibitor | 0.535 0.004 CHEMBL451929 0.478 0.004 CHEMBL3544891 0.492 0.004 CHEMBL3544697 0.472 0.004 CHEMBL3544548 0.496 0.004 CHEMBL447570 0.494 0.004 CHEMBL3544713 | CHEMBL451929 | |
| 0.459 | 0.004 | 0.459 | Antibacterial (Helicobacter pylori) | 0.35 0.005 CHEMBL451929 0.394 0.004 CHEMBL3544891 0.431 0.004 CHEMBL3544697 0.36 0.005 CHEMBL3544548 0.156 0.042 CHEMBL447570 0.323 0.005 CHEMBL3544713 | ||
| 0.372 | 0.019 | 0.372 | P-glycoprotein inhibitor | 0.275 0.034 CHEMBL451929 0.314 0.026 CHEMBL3544891 0.324 0.025 CHEMBL3544697 0.328 0.024 CHEMBL3544548 0.206 0.06 CHEMBL447570 0.243 0.044 CHEMBL3544713 | ||
| 0.384 | 0.07 | 0.384 | Immunosuppressant | 0.341 0.092 CHEMBL451929 0.362 0.08 CHEMBL3544891 0.374 0.074 CHEMBL3544697 0.364 0.08 CHEMBL3544548 0.223 0.173 CHEMBL447570 0.332 0.096 CHEMBL3544713 | ||
| 0.214 | 0.004 | 0.214 | Protein 50S ribosomal subunit inhibitor | 0.195 0.005 CHEMBL451929 0.18 0.005 CHEMBL3544891 0.195 0.005 CHEMBL3544697 0.187 0.005 CHEMBL3544548 0.182 0.005 CHEMBL447570 0.177 0.005 CHEMBL3544713 | ||
| 0.282 | 0.075 | 0.282 | Hypoxia-inducible factor 1 alpha inhibitor | 0.26 0.091 CHEMBL451929 0.206 0.145 CHEMBL3544891 0.212 0.138 CHEMBL3544697 0.242 0.108 CHEMBL3544548 0.191 0.163 CHEMBL3544713 | ||
| 0.194 | 0.022 | 0.194 | Antineoplastic antibiotic | 0.186 0.024 CHEMBL451929 0.168 0.027 CHEMBL3544891 0.185 0.024 CHEMBL3544697 0.175 0.025 CHEMBL3544548 0.175 0.025 CHEMBL447570 0.176 0.025 CHEMBL3544713 | ||
| 0.232 | 0.079 | 0.264 | Angiogenesis stimulant | 0.229 0.08 CHEMBL451929 0.264 0.064 CHEMBL3544891 0.257 0.067 CHEMBL3544697 0.252 0.069 CHEMBL3544548 0.211 0.089 CHEMBL447570 0.256 0.067 CHEMBL3544713 | CHEMBL3544891 | |
| 0.158 | 0.006 | 0.158 | ATPase (Vacuolar H+) inhibitor | 0.153 0.007 CHEMBL451929 0.138 0.011 CHEMBL3544891 0.153 0.007 CHEMBL3544697 0.154 0.007 CHEMBL3544548 0.147 0.008 CHEMBL447570 0.147 0.008 CHEMBL3544713 | ||
| 0.277 | 0.145 | 0.295 | 15-Lipoxygenase inhibitor | 0.295 0.135 CHEMBL451929 | CHEMBL451929 | |
| 0.225 | 0.107 | 0.275 | Immunostimulant | 0.153 0.152 CHEMBL451929 0.263 0.091 CHEMBL3544891 0.275 0.087 CHEMBL3544697 0.27 0.088 CHEMBL3544548 0.197 0.122 CHEMBL3544713 | CHEMBL3544697 | |
| 0.13 | 0.024 | 0.13 | ABCA1 expression enhancer | 0.118 0.032 CHEMBL451929 0.117 0.033 CHEMBL3544891 0.119 0.031 CHEMBL3544697 0.121 0.03 CHEMBL3544548 0.105 0.044 CHEMBL447570 0.108 0.041 CHEMBL3544713 | ||
| 0.267 | 0.198 | 0.267 | Apoptosis agonist | 0.246 0.219 CHEMBL3544891 0.25 0.215 CHEMBL3544697 0.26 0.204 CHEMBL3544548 | ||
| 0.153 | 0.084 | 0.153 | Interleukin 6 antagonist | 0.142 0.102 CHEMBL3544891 0.136 0.114 CHEMBL3544697 0.142 0.102 CHEMBL3544548 | ||
| 0.145 | 0.099 | 0.154 | Nitric oxide antagonist | 0.126 0.125 CHEMBL451929 0.154 0.091 CHEMBL3544891 0.15 0.095 CHEMBL3544697 0.149 0.095 CHEMBL3544548 0.132 0.116 CHEMBL3544713 | CHEMBL3544891 | |
| 0.042 | 0.003 | 0.042 | Antibiotic Macrolide-like | 0.037 0.004 CHEMBL451929 0.032 0.004 CHEMBL3544891 0.039 0.004 CHEMBL3544697 0.034 0.004 CHEMBL3544548 0.034 0.004 CHEMBL447570 0.035 0.004 CHEMBL3544713 | ||
| 0.056 | 0.02 | 0.056 | Microtubule stabilization | 0.051 0.027 CHEMBL3544891 0.054 0.023 CHEMBL3544697 0.055 0.022 CHEMBL3544548 | ||
| 0.228 | 0.206 | 0.326 | DNA directed DNA polymerase inhibitor | 0.275 0.176 CHEMBL451929 0.275 0.176 CHEMBL3544697 0.326 0.149 CHEMBL3544713 | CHEMBL3544713 | |
| 0.036 | 0.02 | 0.036 | Tubulin agonist | 0.036 0.02 CHEMBL451929 0.035 0.023 CHEMBL3544891 0.034 0.024 CHEMBL3544697 0.035 0.023 CHEMBL3544548 0.035 0.023 CHEMBL447570 0.034 0.024 CHEMBL3544713 | ||
| 0.078 | 0.072 | 0.08 | T cell inhibitor | 0.078 0.075 CHEMBL451929 0.08 0.067 CHEMBL3544891 0.078 0.074 CHEMBL3544697 | CHEMBL3544891 | |
| 0.029 | 0.023 | 0.03 | DNA topoisomerase IV inhibitor | 0.03 0.022 CHEMBL451929 | CHEMBL451929 | |
| 0.095 | 0.091 | 0.096 | Topoisomerase II inhibitor | 0.096 0.09 CHEMBL3544548 | CHEMBL3544548 | |
| 0.123 | 0.17 | 0.15 | Hypolipemic | 0.15 0.136 CHEMBL3544548 | CHEMBL3544548 | |
| 0.023 | 0.648 | 0.171 | Tumour necrosis factor alpha release inhibitor | 0.171 0.133 CHEMBL447570 | CHEMBL447570 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |