| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.467 | 0.033 | 0.821 | 5 Hydroxytryptamine release stimulant | 0.821 0.003 CHEMBL3542244 0.4 0.046 CHEMBL3542389 0.175 0.146 CHEMBL3542208 0.4 0.046 CHEMBL3542339 0.25 0.089 CHEMBL3542187 0.8 0.004 CHEMBL3542256 0.743 0.005 CHEMBL3542258 0.465 0.033 CHEMBL3542257 0.656 0.01 CHEMBL4525788 0.656 0.01 CHEMBL3542390 0.373 0.051 CHEMBL3542269 0.17 0.153 CHEMBL3542243 | CHEMBL3542244 | |
| 0.44 | 0.056 | 0.535 | Calcium channel L-type activator | 0.479 0.036 CHEMBL3542244 0.444 0.054 CHEMBL3542389 0.433 0.06 CHEMBL3542208 0.444 0.054 CHEMBL3542339 0.467 0.042 CHEMBL3542187 0.48 0.036 CHEMBL3542256 0.535 0.017 CHEMBL3542258 0.436 0.058 CHEMBL3542257 0.444 0.054 CHEMBL4525788 0.444 0.054 CHEMBL3542390 0.458 0.047 CHEMBL3542269 0.367 0.105 CHEMBL3542243 0.438 0.057 CHEMBL4525787 0.438 0.057 CHEMBL3542266 | CHEMBL3542258 | |
| 0.371 | 0.002 | 0.371 | Orexin receptor antagonist | 0.1 0.012 CHEMBL3542244 0.223 0.003 CHEMBL3542389 0.14 0.005 CHEMBL3542208 0.223 0.003 CHEMBL3542339 0.114 0.008 CHEMBL3542187 0.099 0.012 CHEMBL3542257 0.203 0.003 CHEMBL3542269 0.115 0.008 CHEMBL3542243 0.083 0.024 CHEMBL4525787 0.083 0.024 CHEMBL3542266 | ||
| 0.42 | 0.058 | 0.586 | Antiobesity | 0.567 0.025 CHEMBL3542244 0.365 0.08 CHEMBL3542389 0.365 0.08 CHEMBL3542339 0.387 0.071 CHEMBL3542187 0.484 0.041 CHEMBL3542256 0.586 0.022 CHEMBL3542258 0.205 0.202 CHEMBL3542257 0.319 0.104 CHEMBL4525788 0.319 0.104 CHEMBL3542390 0.471 0.044 CHEMBL3542269 | CHEMBL3542258 | |
| 0.329 | 0.012 | 0.329 | Nav1.2 sodium channel blocker | 0.13 0.073 CHEMBL3542244 0.229 0.026 CHEMBL3542389 0.182 0.041 CHEMBL3542208 0.229 0.026 CHEMBL3542339 0.14 0.064 CHEMBL3542187 0.27 0.019 CHEMBL3542269 0.134 0.068 CHEMBL3542243 0.121 0.082 CHEMBL4525787 0.121 0.082 CHEMBL3542266 | ||
| 0.397 | 0.086 | 0.532 | Analgesic | 0.519 0.044 CHEMBL3542244 0.344 0.111 CHEMBL3542389 0.344 0.111 CHEMBL3542339 0.338 0.115 CHEMBL3542187 0.444 0.067 CHEMBL3542256 0.532 0.04 CHEMBL3542258 0.258 0.176 CHEMBL3542257 0.505 0.048 CHEMBL4525788 0.505 0.048 CHEMBL3542390 0.456 0.063 CHEMBL3542269 | CHEMBL3542258 | |
| 0.311 | 0.049 | 0.365 | Tumour necrosis factor alpha release inhibitor | 0.208 0.102 CHEMBL3542244 0.317 0.047 CHEMBL3542389 0.364 0.034 CHEMBL3542208 0.317 0.047 CHEMBL3542339 0.226 0.088 CHEMBL3542256 0.322 0.046 CHEMBL3542257 0.261 0.07 CHEMBL3542269 0.287 0.059 CHEMBL3542243 0.365 0.034 CHEMBL4525787 0.365 0.034 CHEMBL3542266 | CHEMBL3542266 | |
| 0.248 | 0.003 | 0.248 | Orexin receptor 1 antagonist | 0.089 0.022 CHEMBL3542244 0.166 0.004 CHEMBL3542389 0.095 0.017 CHEMBL3542208 0.166 0.004 CHEMBL3542339 0.088 0.024 CHEMBL3542257 0.156 0.004 CHEMBL3542269 | ||
| 0.26 | 0.017 | 0.26 | Sodium channel blocker | 0.201 0.032 CHEMBL3542244 0.154 0.055 CHEMBL3542389 0.223 0.025 CHEMBL3542208 0.154 0.055 CHEMBL3542339 0.116 0.089 CHEMBL3542187 0.11 0.097 CHEMBL3542256 0.122 0.082 CHEMBL3542258 0.208 0.029 CHEMBL3542257 0.166 0.047 CHEMBL3542269 0.16 0.051 CHEMBL3542243 0.124 0.08 CHEMBL4525787 0.124 0.08 CHEMBL3542266 | ||
| 0.254 | 0.014 | 0.308 | Nav1.3 sodium channel blocker | 0.131 0.063 CHEMBL3542244 0.171 0.036 CHEMBL3542389 0.308 0.008 CHEMBL3542208 0.171 0.036 CHEMBL3542339 0.148 0.049 CHEMBL3542257 0.198 0.025 CHEMBL3542269 0.189 0.028 CHEMBL3542243 0.205 0.023 CHEMBL4525787 0.205 0.023 CHEMBL3542266 | CHEMBL3542208 | |
| 0.209 | 0.002 | 0.209 | Orexin receptor 2 antagonist | 0.043 0.018 CHEMBL3542244 0.124 0.004 CHEMBL3542389 0.068 0.008 CHEMBL3542208 0.124 0.004 CHEMBL3542339 0.045 0.016 CHEMBL3542257 0.11 0.004 CHEMBL3542269 | ||
| 0.216 | 0.01 | 0.216 | Nav1.5 sodium channel blocker | 0.158 0.023 CHEMBL3542244 0.158 0.023 CHEMBL3542389 0.175 0.018 CHEMBL3542208 0.158 0.023 CHEMBL3542339 0.13 0.043 CHEMBL3542187 0.122 0.052 CHEMBL3542256 0.12 0.054 CHEMBL3542258 0.15 0.027 CHEMBL3542257 0.188 0.015 CHEMBL3542269 0.142 0.032 CHEMBL3542243 0.132 0.041 CHEMBL4525787 0.132 0.041 CHEMBL3542266 | ||
| 0.238 | 0.045 | 0.261 | P-glycoprotein inhibitor | 0.213 0.056 CHEMBL3542244 0.235 0.046 CHEMBL3542389 0.235 0.046 CHEMBL3542339 0.261 0.038 CHEMBL3542187 0.212 0.057 CHEMBL3542256 0.18 0.08 CHEMBL3542258 0.167 0.094 CHEMBL4525788 0.167 0.094 CHEMBL3542390 0.2 0.064 CHEMBL3542269 0.167 0.093 CHEMBL3542243 | CHEMBL3542187 | |
| 0.263 | 0.097 | 0.263 | Nootropic | 0.2 0.158 CHEMBL3542244 0.212 0.143 CHEMBL3542389 0.212 0.143 CHEMBL3542339 0.208 0.147 CHEMBL3542257 0.247 0.111 CHEMBL3542269 | ||
| 0.245 | 0.086 | 0.26 | Cardiotonic | 0.227 0.098 CHEMBL3542389 0.26 0.075 CHEMBL3542208 0.227 0.098 CHEMBL3542339 0.164 0.158 CHEMBL3542187 0.26 0.076 CHEMBL3542257 0.23 0.096 CHEMBL3542269 0.17 0.152 CHEMBL3542243 0.244 0.087 CHEMBL4525787 0.244 0.087 CHEMBL3542266 | CHEMBL3542257 | |
| 0.232 | 0.075 | 0.3 | Potassium channel blocker | 0.217 0.082 CHEMBL3542244 0.3 0.046 CHEMBL3542208 0.199 0.093 CHEMBL3542187 0.257 0.063 CHEMBL3542258 0.183 0.104 CHEMBL3542257 0.164 0.121 CHEMBL3542269 0.236 0.073 CHEMBL3542243 0.178 0.108 CHEMBL4525787 0.178 0.108 CHEMBL3542266 | CHEMBL3542208 | |
| 0.202 | 0.052 | 0.203 | Tumour necrosis factor antagonist | 0.203 0.052 CHEMBL3542244 0.178 0.069 CHEMBL3542389 0.146 0.106 CHEMBL3542208 0.178 0.069 CHEMBL3542339 0.179 0.068 CHEMBL3542256 0.165 0.082 CHEMBL3542257 0.188 0.061 CHEMBL3542243 | CHEMBL3542244 | |
| 0.182 | 0.037 | 0.184 | Sodium channel (voltage-gated) blocker | 0.165 0.045 CHEMBL3542244 0.184 0.036 CHEMBL3542208 0.109 0.098 CHEMBL3542187 0.13 0.074 CHEMBL3542258 0.183 0.036 CHEMBL3542257 0.108 0.1 CHEMBL3542269 0.142 0.06 CHEMBL3542243 | CHEMBL3542208 | |
| 0.148 | 0.013 | 0.148 | Glutamate (mGluR7) agonist | 0.12 0.03 CHEMBL3542244 0.111 0.041 CHEMBL3542389 0.111 0.041 CHEMBL3542339 0.146 0.013 CHEMBL3542187 0.09 0.085 CHEMBL3542256 0.127 0.024 CHEMBL3542258 0.097 0.066 CHEMBL4525788 0.097 0.066 CHEMBL3542390 0.098 0.064 CHEMBL3542269 | ||
| 0.141 | 0.017 | 0.285 | 5 Hydroxytryptamine uptake inhibitor | 0.186 0.012 CHEMBL3542244 0.094 0.028 CHEMBL3542389 0.094 0.028 CHEMBL3542339 0.158 0.015 CHEMBL3542187 0.107 0.024 CHEMBL3542256 0.285 0.007 CHEMBL3542258 0.105 0.025 CHEMBL4525788 0.105 0.025 CHEMBL3542390 0.116 0.021 CHEMBL3542269 | CHEMBL3542258 | |
| 0.117 | 0.008 | 0.117 | Neurokinin antagonist | 0.08 0.017 CHEMBL3542244 0.085 0.015 CHEMBL3542389 0.063 0.023 CHEMBL3542208 0.085 0.015 CHEMBL3542339 0.106 0.01 CHEMBL3542187 0.048 0.036 CHEMBL3542256 0.064 0.023 CHEMBL3542258 0.104 0.01 CHEMBL3542269 0.067 0.021 CHEMBL3542243 0.045 0.041 CHEMBL4525787 0.045 0.041 CHEMBL3542266 | ||
| 0.114 | 0.007 | 0.38 | Potassium channel (Ca-activated) blocker | 0.127 0.006 CHEMBL3542244 0.088 0.014 CHEMBL3542389 0.363 0.004 CHEMBL3542208 0.088 0.014 CHEMBL3542339 0.07 0.027 CHEMBL3542187 0.087 0.014 CHEMBL3542256 0.064 0.035 CHEMBL3542258 0.135 0.005 CHEMBL3542257 0.086 0.014 CHEMBL3542269 0.38 0.004 CHEMBL3542243 0.285 0.004 CHEMBL4525787 0.285 0.004 CHEMBL3542266 | CHEMBL3542243 | |
| 0.211 | 0.111 | 0.349 | Spasmolytic | 0.25 0.091 CHEMBL3542244 0.268 0.084 CHEMBL3542389 0.268 0.084 CHEMBL3542339 0.202 0.118 CHEMBL3542187 0.307 0.067 CHEMBL3542256 0.295 0.072 CHEMBL3542258 0.349 0.053 CHEMBL4525788 0.349 0.053 CHEMBL3542390 0.25 0.091 CHEMBL3542269 | CHEMBL3542390 | |
| 0.175 | 0.09 | 0.219 | Anesthetic general | 0.194 0.078 CHEMBL3542244 0.199 0.075 CHEMBL3542389 0.199 0.075 CHEMBL3542339 0.208 0.07 CHEMBL3542187 0.219 0.064 CHEMBL3542256 0.168 0.096 CHEMBL3542258 0.166 0.098 CHEMBL4525788 0.166 0.098 CHEMBL3542390 0.208 0.07 CHEMBL3542269 | CHEMBL3542256 | |
| 0.088 | 0.008 | 0.193 | Potassium channel small-conductance Ca-activated blocker | 0.193 0.004 CHEMBL3542244 0.044 0.032 CHEMBL3542389 0.104 0.006 CHEMBL3542208 0.044 0.032 CHEMBL3542339 0.092 0.008 CHEMBL3542256 0.045 0.03 CHEMBL3542258 0.134 0.005 CHEMBL3542257 0.04 0.039 CHEMBL3542269 0.062 0.016 CHEMBL3542243 0.05 0.024 CHEMBL4525787 0.05 0.024 CHEMBL3542266 | CHEMBL3542244 | |
| 0.074 | 0.004 | 0.074 | Microsomal triglyceride transfer protein inhibitor | 0.037 0.004 CHEMBL3542389 0.053 0.004 CHEMBL3542208 0.037 0.004 CHEMBL3542339 0.062 0.004 CHEMBL3542269 0.03 0.005 CHEMBL4525787 0.03 0.005 CHEMBL3542266 | ||
| 0.075 | 0.005 | 0.075 | Melatonin antagonist | 0.041 0.009 CHEMBL3542244 0.042 0.009 CHEMBL3542389 0.042 0.009 CHEMBL3542339 0.027 0.021 CHEMBL3542256 0.037 0.011 CHEMBL3542269 | ||
| 0.174 | 0.106 | 0.294 | Neurotrophic factor enhancer | 0.243 0.042 CHEMBL3542244 0.223 0.056 CHEMBL3542389 0.223 0.056 CHEMBL3542339 0.154 0.133 CHEMBL3542187 0.294 0.02 CHEMBL3542256 0.227 0.053 CHEMBL3542258 0.274 0.027 CHEMBL3542257 0.203 0.074 CHEMBL4525788 0.203 0.074 CHEMBL3542390 0.238 0.046 CHEMBL3542269 0.167 0.114 CHEMBL4525787 0.167 0.114 CHEMBL3542266 | CHEMBL3542256 | |
| 0.22 | 0.152 | 0.287 | Ca(v)3.3 blocker | 0.209 0.172 CHEMBL3542244 0.215 0.16 CHEMBL3542208 0.287 0.054 CHEMBL3542257 0.205 0.182 CHEMBL3542243 | CHEMBL3542257 | |
| 0.093 | 0.03 | 0.096 | Viral attachment inhibitor | 0.084 0.041 CHEMBL3542389 0.084 0.041 CHEMBL3542339 0.08 0.049 CHEMBL3542187 0.096 0.027 CHEMBL3542269 | CHEMBL3542269 | |
| 0.127 | 0.066 | 0.14 | Papain-like protease (SARS coronavirus) inhibitor | 0.137 0.048 CHEMBL3542389 0.127 0.066 CHEMBL3542208 0.137 0.048 CHEMBL3542339 0.112 0.106 CHEMBL3542187 0.14 0.045 CHEMBL3542269 0.116 0.093 CHEMBL3542243 0.138 0.047 CHEMBL4525787 0.138 0.047 CHEMBL3542266 | CHEMBL3542269 | |
| 0.071 | 0.012 | 0.071 | Neurokinin 1 antagonist | 0.071 0.012 CHEMBL3542244 0.048 0.021 CHEMBL3542389 0.057 0.016 CHEMBL3542208 0.048 0.021 CHEMBL3542339 0.067 0.013 CHEMBL3542187 0.043 0.025 CHEMBL3542256 0.063 0.014 CHEMBL3542258 0.037 0.035 CHEMBL3542257 0.057 0.016 CHEMBL3542269 0.059 0.015 CHEMBL3542243 0.041 0.028 CHEMBL4525787 0.041 0.028 CHEMBL3542266 | ||
| 0.06 | 0.005 | 0.06 | Urotensin II antagonist | 0.034 0.009 CHEMBL3542389 0.021 0.017 CHEMBL3542208 0.034 0.009 CHEMBL3542339 0.02 0.019 CHEMBL3542187 0.028 0.011 CHEMBL3542269 | ||
| 0.064 | 0.01 | 0.064 | Substance P antagonist | 0.063 0.01 CHEMBL3542244 0.047 0.019 CHEMBL3542389 0.059 0.012 CHEMBL3542208 0.047 0.019 CHEMBL3542339 0.048 0.018 CHEMBL3542187 0.042 0.024 CHEMBL3542256 0.051 0.016 CHEMBL3542258 0.035 0.033 CHEMBL3542257 0.051 0.016 CHEMBL3542269 0.052 0.015 CHEMBL3542243 0.043 0.023 CHEMBL4525787 0.043 0.023 CHEMBL3542266 | ||
| 0.056 | 0.005 | 0.056 | Melatonin 1 antagonist | 0.022 0.01 CHEMBL3542244 0.029 0.007 CHEMBL3542389 0.029 0.007 CHEMBL3542339 0.025 0.008 CHEMBL3542269 | ||
| 0.273 | 0.225 | 0.551 | Caspase 9 stimulant | 0.483 0.067 CHEMBL3542244 0.326 0.167 CHEMBL3542389 0.326 0.167 CHEMBL3542339 0.551 0.044 CHEMBL3542256 0.387 0.119 CHEMBL3542258 0.537 0.048 CHEMBL3542257 0.456 0.08 CHEMBL4525788 0.456 0.08 CHEMBL3542390 0.255 0.247 CHEMBL3542269 0.252 0.251 CHEMBL4525787 0.252 0.251 CHEMBL3542266 | CHEMBL3542256 | |
| 0.09 | 0.042 | 0.091 | CC chemokine receptor antagonist | 0.068 0.066 CHEMBL3542389 0.068 0.066 CHEMBL3542339 0.078 0.054 CHEMBL3542187 0.091 0.041 CHEMBL3542269 | CHEMBL3542269 | |
| 0.066 | 0.021 | 0.071 | CC chemokine 5 receptor antagonist | 0.054 0.032 CHEMBL3542389 0.054 0.032 CHEMBL3542339 0.071 0.017 CHEMBL3542269 | CHEMBL3542269 | |
| 0.051 | 0.01 | 0.051 | 5 Hydroxytryptamine 1D agonist | 0.041 0.014 CHEMBL3542269 | ||
| 0.084 | 0.043 | 0.109 | Analgesic, opioid | 0.071 0.06 CHEMBL3542244 0.087 0.04 CHEMBL3542389 0.087 0.04 CHEMBL3542339 0.076 0.052 CHEMBL3542256 0.109 0.027 CHEMBL3542269 | CHEMBL3542269 | |
| 0.055 | 0.016 | 0.055 | Oxytocin antagonist | 0.042 0.022 CHEMBL3542389 0.039 0.025 CHEMBL3542208 0.042 0.022 CHEMBL3542339 0.046 0.019 CHEMBL3542269 | ||
| 0.078 | 0.042 | 0.14 | Calcium channel L-type blocker | 0.14 0.012 CHEMBL3542244 0.102 0.024 CHEMBL3542256 0.072 0.05 CHEMBL3542258 0.077 0.042 CHEMBL4525788 0.077 0.042 CHEMBL3542390 | CHEMBL3542244 | |
| 0.066 | 0.031 | 0.072 | Potassium channel intermediate-conductance Ca-activated blocker | 0.06 0.042 CHEMBL3542244 0.061 0.04 CHEMBL3542187 0.072 0.025 CHEMBL3542257 0.055 0.054 CHEMBL3542243 | CHEMBL3542257 | |
| 0.033 | 0.005 | 0.033 | Apolipoprotein B-100 inhibitor | 0.022 0.009 CHEMBL3542269 | ||
| 0.076 | 0.05 | 0.157 | Phosphodiesterase 4D inhibitor | 0.066 0.059 CHEMBL3542244 0.157 0.018 CHEMBL3542257 | CHEMBL3542257 | |
| 0.069 | 0.045 | 0.075 | Matrix metalloproteinase inhibitor | 0.067 0.046 CHEMBL3542389 0.067 0.046 CHEMBL3542339 0.075 0.04 CHEMBL3542269 | CHEMBL3542269 | |
| 0.044 | 0.02 | 0.077 | Growth hormone secretagogue receptor antagonist | 0.03 0.029 CHEMBL3542208 0.077 0.01 CHEMBL3542257 0.033 0.027 CHEMBL3542269 0.03 0.029 CHEMBL3542243 | CHEMBL3542257 | |
| 0.08 | 0.057 | 0.1 | Opioid kappa receptor antagonist | 0.087 0.049 CHEMBL3542389 0.087 0.049 CHEMBL3542339 0.1 0.035 CHEMBL3542269 | CHEMBL3542269 | |
| 0.066 | 0.044 | 0.083 | Glucagon-like peptide 1 agonist | 0.059 0.049 CHEMBL3542389 0.059 0.049 CHEMBL3542339 0.083 0.033 CHEMBL3542187 0.071 0.041 CHEMBL3542269 | CHEMBL3542187 | |
| 0.154 | 0.133 | 0.246 | Potassium channel (Voltage-sensitive) blocker | 0.246 0.069 CHEMBL3542244 0.182 0.11 CHEMBL3542208 0.246 0.069 CHEMBL3542258 0.205 0.093 CHEMBL3542257 0.16 0.129 CHEMBL3542243 | CHEMBL3542258 | |
| 0.026 | 0.01 | 0.053 | Bombesin agonist | 0.044 0.005 CHEMBL3542244 0.022 0.016 CHEMBL3542389 0.022 0.016 CHEMBL3542339 0.028 0.009 CHEMBL3542256 0.053 0.005 CHEMBL3542257 0.021 0.019 CHEMBL4525788 0.021 0.019 CHEMBL3542390 0.028 0.009 CHEMBL3542269 | CHEMBL3542257 | |
| 0.07 | 0.055 | 0.08 | Metalloproteinase-9 inhibitor | 0.074 0.049 CHEMBL3542389 0.074 0.049 CHEMBL3542339 0.08 0.044 CHEMBL3542269 | CHEMBL3542269 | |
| 0.089 | 0.075 | 0.098 | Chemokine receptor antagonist | 0.098 0.065 CHEMBL3542269 | CHEMBL3542269 | |
| 0.111 | 0.098 | 0.198 | Calcium channel blocker | 0.198 0.031 CHEMBL3542244 0.128 0.078 CHEMBL3542256 0.132 0.075 CHEMBL3542258 0.165 0.048 CHEMBL4525788 0.165 0.048 CHEMBL3542390 | CHEMBL3542244 | |
| 0.019 | 0.006 | 0.019 | Melatonin receptor 1A antagonist | 0.015 0.008 CHEMBL3542244 | ||
| 0.041 | 0.029 | 0.041 | Neurokinin 2 antagonist | 0.037 0.035 CHEMBL3542244 0.039 0.031 CHEMBL3542269 | ||
| 0.022 | 0.01 | 0.047 | Bombesin 3 receptor agonist | 0.04 0.005 CHEMBL3542244 0.018 0.014 CHEMBL3542389 0.018 0.014 CHEMBL3542339 0.023 0.009 CHEMBL3542256 0.047 0.005 CHEMBL3542257 0.023 0.009 CHEMBL3542269 | CHEMBL3542257 | |
| 0.052 | 0.04 | 0.323 | NMDA 2B receptor antagonist | 0.101 0.015 CHEMBL3542244 0.056 0.035 CHEMBL3542389 0.056 0.035 CHEMBL3542339 0.249 0.005 CHEMBL3542187 0.104 0.014 CHEMBL3542256 0.323 0.004 CHEMBL3542258 0.218 0.005 CHEMBL4525788 0.218 0.005 CHEMBL3542390 0.084 0.02 CHEMBL3542269 | CHEMBL3542258 | |
| 0.047 | 0.037 | 0.047 | CC chemokine receptor 2B antagonist | 0.047 0.037 CHEMBL3542243 | ||
| 0.024 | 0.014 | 0.037 | CYP24 inhibitor | 0.023 0.016 CHEMBL3542389 0.035 0.008 CHEMBL3542208 0.023 0.016 CHEMBL3542339 0.021 0.019 CHEMBL3542257 0.022 0.016 CHEMBL3542269 0.037 0.008 CHEMBL3542243 0.032 0.009 CHEMBL4525787 0.032 0.009 CHEMBL3542266 | CHEMBL3542243 | |
| 0.039 | 0.03 | 0.043 | Glucagon-like peptide 1 receptor antagonist | 0.043 0.021 CHEMBL3542187 | CHEMBL3542187 | |
| 0.105 | 0.097 | 0.146 | Acetylcholinesterase inhibitor | 0.146 0.058 CHEMBL3542244 0.104 0.098 CHEMBL3542389 0.104 0.098 CHEMBL3542339 0.139 0.063 CHEMBL3542256 0.108 0.092 CHEMBL4525788 0.108 0.092 CHEMBL3542390 | CHEMBL3542244 | |
| 0.095 | 0.091 | 0.129 | Calcium channel (voltage-sensitive) blocker | 0.129 0.047 CHEMBL3542244 0.102 0.08 CHEMBL4525788 0.102 0.08 CHEMBL3542390 | CHEMBL3542244 | |
| 0.054 | 0.051 | 0.054 | Adrenaline uptake inhibitor | |||
| 0.044 | 0.042 | 0.052 | Matrix metalloproteinase 1 inhibitor | 0.047 0.04 CHEMBL3542389 0.047 0.04 CHEMBL3542339 0.052 0.037 CHEMBL3542269 | CHEMBL3542269 | |
| 0.056 | 0.058 | 0.064 | Heme oxygenase stimulant | 0.058 0.052 CHEMBL3542244 0.059 0.048 CHEMBL3542389 0.059 0.048 CHEMBL3542339 0.062 0.041 CHEMBL3542256 0.06 0.047 CHEMBL3542257 0.058 0.054 CHEMBL4525788 0.058 0.054 CHEMBL3542390 0.064 0.037 CHEMBL3542269 | CHEMBL3542269 | |
| 0.058 | 0.061 | 0.077 | Nav1.7 sodium channel blocker | 0.062 0.055 CHEMBL3542244 0.066 0.049 CHEMBL3542208 0.077 0.036 CHEMBL3542257 | CHEMBL3542257 | |
| 0.028 | 0.031 | 0.04 | Melatonin 2 agonist | 0.04 0.015 CHEMBL3542208 0.035 0.02 CHEMBL4525787 0.035 0.02 CHEMBL3542266 | CHEMBL3542208 | |
| 0.084 | 0.088 | 0.125 | Interleukin 12 antagonist | 0.095 0.062 CHEMBL3542244 0.089 0.074 CHEMBL3542389 0.094 0.064 CHEMBL3542208 0.089 0.074 CHEMBL3542339 0.101 0.053 CHEMBL3542256 0.125 0.025 CHEMBL3542257 0.106 0.044 CHEMBL4525788 0.106 0.044 CHEMBL3542390 0.087 0.08 CHEMBL3542269 0.108 0.042 CHEMBL3542243 0.099 0.056 CHEMBL4525787 0.099 0.056 CHEMBL3542266 | CHEMBL3542257 | |
| 0.04 | 0.044 | 0.078 | Dopamine transporter inhibitor | 0.059 0.026 CHEMBL3542244 0.046 0.036 CHEMBL3542256 0.078 0.018 CHEMBL3542258 0.057 0.027 CHEMBL4525788 0.057 0.027 CHEMBL3542390 | CHEMBL3542258 | |
| 0.073 | 0.08 | 0.096 | Opioid antagonist | 0.081 0.068 CHEMBL3542389 0.081 0.068 CHEMBL3542339 0.077 0.073 CHEMBL3542187 0.096 0.051 CHEMBL3542269 | CHEMBL3542269 | |
| 0.035 | 0.044 | 0.043 | HIV-1 protease inhibitor | 0.043 0.03 CHEMBL3542269 | CHEMBL3542269 | |
| 0.094 | 0.104 | 0.286 | Cholinergic antagonist | 0.113 0.08 CHEMBL3542244 0.286 0.016 CHEMBL3542187 0.103 0.092 CHEMBL3542256 0.233 0.024 CHEMBL3542258 0.125 0.069 CHEMBL4525788 0.125 0.069 CHEMBL3542390 0.11 0.084 CHEMBL3542269 | CHEMBL3542187 | |
| 0.092 | 0.103 | 0.283 | Acetylcholine antagonist | 0.112 0.078 CHEMBL3542244 0.283 0.015 CHEMBL3542187 0.102 0.09 CHEMBL3542256 0.23 0.024 CHEMBL3542258 0.122 0.068 CHEMBL4525788 0.122 0.068 CHEMBL3542390 0.107 0.084 CHEMBL3542269 | CHEMBL3542187 | |
| 0.042 | 0.06 | 0.121 | Dopamine uptake inhibitor | 0.097 0.019 CHEMBL3542244 0.069 0.031 CHEMBL3542256 0.121 0.014 CHEMBL3542258 0.088 0.022 CHEMBL4525788 0.088 0.022 CHEMBL3542390 | CHEMBL3542258 | |
| 0.108 | 0.128 | 0.333 | Acetylcholine M1 receptor antagonist | 0.333 0.01 CHEMBL3542187 0.198 0.043 CHEMBL3542258 0.146 0.078 CHEMBL3542269 | CHEMBL3542187 | |
| 0.13 | 0.152 | 0.231 | HERG channel blocker | 0.231 0.074 CHEMBL3542244 0.218 0.08 CHEMBL3542258 0.177 0.105 CHEMBL3542257 | CHEMBL3542244 | |
| 0.034 | 0.056 | 0.097 | Phosphodiesterase 4A inhibitor | 0.097 0.016 CHEMBL3542257 | CHEMBL3542257 | |
| 0.029 | 0.055 | 0.039 | Opioid kappa receptor agonist | 0.039 0.035 CHEMBL3542256 | CHEMBL3542256 | |
| 0.045 | 0.072 | 0.079 | 5 Hydroxytryptamine 7 agonist | 0.079 0.013 CHEMBL3542244 0.061 0.03 CHEMBL3542256 0.051 0.049 CHEMBL3542257 | CHEMBL3542244 | |
| 0.015 | 0.043 | 0.079 | Growth hormone secretagogue receptor agonist | 0.079 0.011 CHEMBL3542244 0.03 0.027 CHEMBL3542256 | CHEMBL3542244 | |
| 0.031 | 0.059 | 0.089 | Phenylethanolamine N methyltransferase inhibitor | 0.089 0.004 CHEMBL3542244 0.081 0.004 CHEMBL3542256 0.08 0.004 CHEMBL3542258 0.06 0.008 CHEMBL4525788 0.06 0.008 CHEMBL3542390 | CHEMBL3542244 | |
| 0.048 | 0.077 | 0.269 | Dopamine antagonist | 0.265 0.014 CHEMBL3542244 0.269 0.013 CHEMBL3542256 0.121 0.032 CHEMBL3542258 | CHEMBL3542256 | |
| 0.07 | 0.104 | 0.146 | Sphingomyelinase inhibitor | 0.13 0.035 CHEMBL3542244 0.106 0.053 CHEMBL3542256 0.146 0.026 CHEMBL3542258 0.097 0.063 CHEMBL3542257 0.086 0.077 CHEMBL4525788 0.086 0.077 CHEMBL3542390 | CHEMBL3542258 | |
| 0.071 | 0.106 | 0.26 | 5 Hydroxytryptamine 2 antagonist | 0.26 0.02 CHEMBL3542244 0.153 0.043 CHEMBL3542256 0.138 0.049 CHEMBL3542258 | CHEMBL3542244 | |
| 0.041 | 0.079 | 0.067 | 5 Hydroxytryptamine 1D antagonist | 0.067 0.042 CHEMBL3542244 | CHEMBL3542244 | |
| 0.03 | 0.067 | 0.041 | GHS receptor agonist | 0.041 0.032 CHEMBL3542244 | CHEMBL3542244 | |
| 0.023 | 0.063 | 0.037 | Melanocortin 4 antagonist | 0.037 0.036 CHEMBL3542244 | CHEMBL3542244 | |
| 0.018 | 0.059 | 0.036 | Liver X receptor alpha antagonist | 0.027 0.024 CHEMBL3542244 0.03 0.019 CHEMBL3542256 0.036 0.011 CHEMBL3542257 | CHEMBL3542257 | |
| 0.028 | 0.071 | 0.038 | Aggrecanase 1 inhibitor | 0.038 0.03 CHEMBL3542257 | CHEMBL3542257 | |
| 0.098 | 0.142 | 0.164 | Cholinergic | 0.164 0.066 CHEMBL3542244 0.142 0.084 CHEMBL3542256 | CHEMBL3542244 | |
| 0.04 | 0.085 | 0.062 | Opioid mu receptor antagonist | 0.062 0.052 CHEMBL3542269 | CHEMBL3542269 | |
| 0.029 | 0.074 | 0.045 | Nerve growth factor antagonist | 0.04 0.035 CHEMBL3542244 0.04 0.036 CHEMBL3542256 0.04 0.035 CHEMBL3542257 0.045 0.026 CHEMBL3542269 | CHEMBL3542269 | |
| 0.031 | 0.076 | 0.048 | Mineralocorticoid receptor antagonist | 0.048 0.033 CHEMBL3542208 0.048 0.033 CHEMBL3542243 0.045 0.039 CHEMBL4525787 0.045 0.039 CHEMBL3542266 | CHEMBL3542243 | |
| 0.023 | 0.068 | 0.077 | Sigma receptor antagonist | 0.057 0.03 CHEMBL3542244 0.077 0.021 CHEMBL3542258 | CHEMBL3542258 | |
| 0.061 | 0.116 | 0.084 | Protease inhibitor | 0.084 0.081 CHEMBL4525788 0.084 0.081 CHEMBL3542390 | CHEMBL3542390 | |
| 0.031 | 0.087 | 0.173 | Dopamine D2 antagonist | 0.17 0.02 CHEMBL3542244 0.173 0.019 CHEMBL3542256 0.077 0.04 CHEMBL3542258 | CHEMBL3542256 | |
| 0.035 | 0.092 | 0.176 | 5 Hydroxytryptamine 2A agonist | 0.176 0.004 CHEMBL3542244 0.13 0.007 CHEMBL3542256 0.099 0.015 CHEMBL3542258 0.055 0.053 CHEMBL4525788 0.055 0.053 CHEMBL3542390 | CHEMBL3542244 | |
| 0.051 | 0.111 | 0.074 | Focal adhesion kinase 1 inhibitor | 0.068 0.065 CHEMBL3542244 0.074 0.056 CHEMBL3542257 | CHEMBL3542257 | |
| 0.011 | 0.073 | 0.04 | Dopamine D1 agonist | 0.025 0.013 CHEMBL3542244 0.04 0.005 CHEMBL3542256 0.021 0.019 CHEMBL3542269 | CHEMBL3542256 | |
| 0.03 | 0.092 | 0.073 | Acetylcholine M2 receptor antagonist | 0.073 0.034 CHEMBL3542187 | CHEMBL3542187 | |
| 0.046 | 0.11 | 0.151 | Nicotinic alpha4beta2 receptor antagonist | 0.151 0.008 CHEMBL3542244 0.119 0.018 CHEMBL3542256 0.145 0.009 CHEMBL3542258 0.103 0.029 CHEMBL3542257 0.088 0.042 CHEMBL4525788 0.088 0.042 CHEMBL3542390 | CHEMBL3542244 | |
| 0.016 | 0.08 | 0.056 | Cholesterol ester transfer protein antagonist | 0.036 0.016 CHEMBL3542258 0.056 0.005 CHEMBL3542257 | CHEMBL3542257 | |
| 0.071 | 0.138 | 0.225 | Acetylcholine muscarinic antagonist | 0.225 0.019 CHEMBL3542187 0.139 0.051 CHEMBL3542258 | CHEMBL3542187 | |
| 0.05 | 0.118 | 0.106 | Ca(v)2.2 blocker | 0.106 0.045 CHEMBL3542244 0.091 0.055 CHEMBL3542257 | CHEMBL3542244 | |
| 0.078 | 0.15 | 0.147 | Electron transport complex I inhibitor | 0.104 0.075 CHEMBL3542244 0.112 0.059 CHEMBL3542187 0.103 0.075 CHEMBL3542256 0.147 0.022 CHEMBL3542258 0.125 0.04 CHEMBL3542257 | CHEMBL3542258 | |
| 0.013 | 0.089 | 0.035 | Liver X receptor antagonist | 0.035 0.017 CHEMBL3542257 | CHEMBL3542257 | |
| 0.157 | 0.234 | 0.403 | Tyrosine 3 hydroxylase inhibitor | 0.335 0.02 CHEMBL3542244 0.195 0.144 CHEMBL3542389 0.195 0.144 CHEMBL3542339 0.403 0.008 CHEMBL3542256 0.264 0.056 CHEMBL3542258 0.205 0.126 CHEMBL4525788 0.205 0.126 CHEMBL3542390 0.233 0.086 CHEMBL3542269 | CHEMBL3542256 | |
| 0.094 | 0.172 | 0.139 | Vanilloid 1 agonist | 0.118 0.092 CHEMBL3542244 0.114 0.104 CHEMBL3542389 0.114 0.104 CHEMBL3542339 0.139 0.051 CHEMBL3542256 | CHEMBL3542256 | |
| 0.149 | 0.228 | 0.498 | Transcription factor NF kappa B inhibitor | 0.381 0.068 CHEMBL3542244 0.239 0.136 CHEMBL3542389 0.239 0.136 CHEMBL3542339 0.498 0.044 CHEMBL3542256 0.327 0.084 CHEMBL3542258 0.367 0.072 CHEMBL3542257 0.377 0.069 CHEMBL4525788 0.377 0.069 CHEMBL3542390 0.197 0.172 CHEMBL3542269 0.197 0.172 CHEMBL4525787 0.197 0.172 CHEMBL3542266 | CHEMBL3542256 | |
| 0.011 | 0.091 | 0.024 | Motilin receptor agonist | 0.024 0.015 CHEMBL3542244 | CHEMBL3542244 | |
| 0.045 | 0.125 | 0.183 | Acetylcholine nicotinic antagonist | 0.169 0.016 CHEMBL3542244 0.128 0.028 CHEMBL3542256 0.183 0.014 CHEMBL3542258 0.104 0.037 CHEMBL4525788 0.104 0.037 CHEMBL3542390 | CHEMBL3542258 | |
| 0.074 | 0.157 | 0.153 | Nav1.6 sodium channel blocker | 0.153 0.051 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.11 | 0.134 | 5 Hydroxytryptamine 2 agonist | 0.134 0.005 CHEMBL3542244 0.08 0.015 CHEMBL3542256 0.061 0.025 CHEMBL3542258 | CHEMBL3542244 | |
| 0.034 | 0.12 | 0.06 | Epithelial sodium channel blocker | 0.06 0.029 CHEMBL3542244 0.051 0.047 CHEMBL3542256 | CHEMBL3542244 | |
| 0.028 | 0.116 | 0.059 | Dopamine D3 antagonist | 0.059 0.045 CHEMBL3542244 | CHEMBL3542244 | |
| 0.056 | 0.145 | 0.099 | Breast cancer-resistant protein inhibitor | 0.085 0.073 CHEMBL3542244 0.087 0.07 CHEMBL3542187 0.09 0.066 CHEMBL3542256 0.099 0.056 CHEMBL3542243 | CHEMBL3542243 | |
| 0.014 | 0.105 | 0.03 | Estrogen-related receptor alpha antagonist | 0.03 0.026 CHEMBL4525788 0.03 0.026 CHEMBL3542390 | CHEMBL3542390 | |
| 0.028 | 0.119 | 0.067 | Acetylcholine M5 receptor antagonist | 0.067 0.033 CHEMBL3542187 | CHEMBL3542187 | |
| 0.146 | 0.239 | 0.181 | Neuropeptide Y2 antagonist | 0.181 0.158 CHEMBL3542187 | CHEMBL3542187 | |
| 0.045 | 0.141 | 0.356 | NMDA receptor antagonist | 0.137 0.028 CHEMBL3542244 0.157 0.022 CHEMBL3542187 0.178 0.018 CHEMBL3542256 0.356 0.005 CHEMBL3542258 0.125 0.033 CHEMBL4525788 0.125 0.033 CHEMBL3542390 0.125 0.033 CHEMBL3542269 | CHEMBL3542258 | |
| 0.03 | 0.128 | 0.119 | Potassium channel Kv1.5 blocker | 0.119 0.013 CHEMBL3542208 0.115 0.014 CHEMBL3542243 0.086 0.023 CHEMBL4525787 0.086 0.023 CHEMBL3542266 | CHEMBL3542208 | |
| 0.026 | 0.127 | 0.069 | 5 Hydroxytryptamine agonist | 0.069 0.048 CHEMBL3542244 | CHEMBL3542244 | |
| 0.03 | 0.132 | 0.126 | Neuronal nicotinic receptor antagonist | 0.126 0.016 CHEMBL3542244 0.092 0.028 CHEMBL3542256 0.115 0.019 CHEMBL3542258 0.064 0.05 CHEMBL4525788 0.064 0.05 CHEMBL3542390 | CHEMBL3542244 | |
| 0.033 | 0.135 | 0.209 | 5 Hydroxytryptamine 2A antagonist | 0.209 0.019 CHEMBL3542244 0.113 0.041 CHEMBL3542256 0.089 0.053 CHEMBL3542258 | CHEMBL3542244 | |
| 0.017 | 0.119 | 0.06 | Beta tubulin antagonist | 0.06 0.04 CHEMBL3542256 | CHEMBL3542256 | |
| 0.032 | 0.137 | 0.104 | Dopamine D1 antagonist | 0.063 0.046 CHEMBL3542244 0.104 0.024 CHEMBL3542256 | CHEMBL3542256 | |
| 0.04 | 0.147 | 0.128 | Alpha adrenoreceptor antagonist | 0.128 0.044 CHEMBL3542244 0.105 0.054 CHEMBL3542256 0.116 0.049 CHEMBL3542258 | CHEMBL3542244 | |
| 0.061 | 0.168 | 0.093 | Vanilloid agonist | 0.093 0.042 CHEMBL3542256 | CHEMBL3542256 | |
| 0.024 | 0.132 | 0.05 | CC chemokine 4 receptor antagonist | 0.05 0.027 CHEMBL3542244 | CHEMBL3542244 | |
| 0.087 | 0.204 | 0.166 | Insulin secretagoues | 0.154 0.07 CHEMBL3542244 0.166 0.059 CHEMBL3542256 0.146 0.078 CHEMBL4525788 0.146 0.078 CHEMBL3542390 | CHEMBL3542256 | |
| 0.12 | 0.237 | 0.209 | 5 Hydroxytryptamine 1E antagonist | 0.209 0.121 CHEMBL3542244 0.185 0.148 CHEMBL3542256 | CHEMBL3542244 | |
| 0.013 | 0.13 | 0.077 | Glycine transporter inhibitor | 0.077 0.018 CHEMBL3542244 0.075 0.019 CHEMBL3542258 | CHEMBL3542244 | |
| 0.01 | 0.129 | 0.029 | Estradiol 17 beta-dehydrogenase 3 inhibitor | 0.029 0.026 CHEMBL3542256 | CHEMBL3542256 | |
| 0.161 | 0.282 | 0.396 | Calcium channel activator | 0.365 0.041 CHEMBL3542244 0.326 0.068 CHEMBL3542256 0.365 0.04 CHEMBL3542258 0.396 0.026 CHEMBL3542257 0.319 0.074 CHEMBL4525788 0.319 0.074 CHEMBL3542390 | CHEMBL3542257 | |
| 0.022 | 0.145 | 0.381 | NMDA 2 receptor antagonist | 0.175 0.012 CHEMBL3542244 0.14 0.019 CHEMBL3542187 0.213 0.008 CHEMBL3542256 0.381 0.004 CHEMBL3542258 0.204 0.009 CHEMBL4525788 0.204 0.009 CHEMBL3542390 0.086 0.04 CHEMBL3542269 | CHEMBL3542258 | |
| 0.017 | 0.143 | 0.032 | Melatonin receptor 1A agonist | 0.032 0.027 CHEMBL3542257 | CHEMBL3542257 | |
| 0.04 | 0.168 | 0.194 | Antiadrenergic | 0.117 0.047 CHEMBL3542244 0.113 0.049 CHEMBL3542256 0.194 0.025 CHEMBL3542258 | CHEMBL3542258 | |
| 0.038 | 0.168 | 0.19 | Adrenaline antagonist | 0.113 0.046 CHEMBL3542244 0.109 0.048 CHEMBL3542256 0.19 0.025 CHEMBL3542258 | CHEMBL3542258 | |
| 0.028 | 0.16 | 0.087 | Sphingosine kinase 2 inhibitor | 0.07 0.022 CHEMBL3542244 0.083 0.014 CHEMBL3542256 0.087 0.012 CHEMBL4525788 0.087 0.012 CHEMBL3542390 0.05 0.048 CHEMBL3542269 | CHEMBL3542390 | |
| 0.046 | 0.18 | 0.069 | Calcium channel P-type blocker | 0.069 0.031 CHEMBL3542244 0.069 0.03 CHEMBL3542257 0.061 0.055 CHEMBL4525788 0.061 0.055 CHEMBL3542390 | CHEMBL3542257 | |
| 0.032 | 0.167 | 0.232 | Phosphodiesterase IV inhibitor | 0.232 0.009 CHEMBL3542257 | CHEMBL3542257 | |
| 0.052 | 0.19 | 0.192 | Tubulin antagonist | 0.152 0.057 CHEMBL3542244 0.192 0.039 CHEMBL3542256 0.102 0.1 CHEMBL3542258 0.144 0.061 CHEMBL3542257 0.141 0.063 CHEMBL4525788 0.141 0.063 CHEMBL3542390 0.112 0.088 CHEMBL4525787 0.112 0.088 CHEMBL3542266 | CHEMBL3542256 | |
| 0.033 | 0.172 | 0.222 | Alpha 2a adrenoreceptor antagonist | 0.207 0.013 CHEMBL3542244 0.222 0.011 CHEMBL3542256 0.182 0.016 CHEMBL3542258 | CHEMBL3542256 | |
| 0.066 | 0.206 | 0.107 | Acetylcholine release stimulant | 0.107 0.071 CHEMBL3542257 | CHEMBL3542257 | |
| 0.033 | 0.173 | 0.152 | 5 Hydroxytryptamine 2C antagonist | 0.152 0.026 CHEMBL3542244 0.087 0.055 CHEMBL3542256 0.116 0.038 CHEMBL3542257 | CHEMBL3542244 | |
| 0.037 | 0.179 | 0.209 | Alpha 2 adrenoreceptor antagonist | 0.209 0.016 CHEMBL3542244 0.206 0.017 CHEMBL3542256 0.163 0.024 CHEMBL3542258 | CHEMBL3542244 | |
| 0.023 | 0.166 | 0.087 | 5 Hydroxytryptamine 1 antagonist | 0.087 0.043 CHEMBL3542244 | CHEMBL3542244 | |
| 0.027 | 0.17 | 0.073 | Vanilloid 1 antagonist | 0.073 0.041 CHEMBL3542257 | CHEMBL3542257 | |
| 0.045 | 0.19 | 0.113 | Prolactin inhibitor | 0.09 0.067 CHEMBL3542244 0.113 0.043 CHEMBL3542256 0.084 0.075 CHEMBL3542269 | CHEMBL3542256 | |
| 0.086 | 0.233 | 0.142 | Anticonvulsant | 0.142 0.139 CHEMBL3542244 | CHEMBL3542244 | |
| 0.009 | 0.16 | 0.084 | 5 Hydroxytryptamine 2C agonist | 0.084 0.01 CHEMBL3542244 0.064 0.018 CHEMBL3542256 0.051 0.027 CHEMBL3542258 | CHEMBL3542244 | |
| 0.015 | 0.173 | 0.078 | Dopamine D4 antagonist | 0.078 0.033 CHEMBL3542244 0.058 0.043 CHEMBL3542256 | CHEMBL3542244 | |
| 0.009 | 0.171 | 0.076 | TRPM8 blocker | 0.076 0.009 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.188 | 0.084 | Nav1.8 sodium channel blocker | 0.073 0.052 CHEMBL3542244 0.084 0.038 CHEMBL3542257 | CHEMBL3542257 | |
| 0.019 | 0.186 | 0.106 | Nicotinic receptor alpha4 subunit antagonist | 0.06 0.021 CHEMBL3542244 0.046 0.042 CHEMBL3542187 0.049 0.034 CHEMBL3542256 0.106 0.007 CHEMBL3542258 0.05 0.032 CHEMBL4525788 0.05 0.032 CHEMBL3542390 | CHEMBL3542258 | |
| 0.032 | 0.198 | 0.058 | 5 Hydroxytryptamine 5A antagonist | 0.058 0.049 CHEMBL3542244 | CHEMBL3542244 | |
| 0.058 | 0.226 | 0.079 | CC chemokine 5 receptor agonist | 0.079 0.07 CHEMBL3542244 0.077 0.076 CHEMBL3542256 | CHEMBL3542244 | |
| 0.027 | 0.196 | 0.052 | Bombesin 3 receptor antagonist | 0.052 0.043 CHEMBL3542257 | CHEMBL3542257 | |
| 0.029 | 0.198 | 0.053 | 5 Hydroxytryptamine 5 antagonist | 0.053 0.049 CHEMBL3542244 | CHEMBL3542244 | |
| 0.018 | 0.19 | 0.08 | 5 Hydroxytryptamine 2B agonist | 0.08 0.005 CHEMBL3542244 0.046 0.016 CHEMBL3542256 0.051 0.013 CHEMBL3542258 | CHEMBL3542244 | |
| 0.062 | 0.236 | 0.148 | Neurotrophic factor | 0.134 0.075 CHEMBL3542244 0.148 0.061 CHEMBL3542256 0.137 0.073 CHEMBL3542258 | CHEMBL3542256 | |
| 0.017 | 0.193 | 0.078 | 5 Hydroxytryptamine 6 antagonist | 0.078 0.024 CHEMBL3542244 | CHEMBL3542244 | |
| 0.004 | 0.186 | 0.035 | Acetyl-CoA carboxylase 2 inhibitor | 0.035 0.01 CHEMBL4525788 0.035 0.01 CHEMBL3542390 | CHEMBL3542390 | |
| 0.081 | 0.264 | 0.331 | Antiamyloidogenic | 0.226 0.083 CHEMBL3542244 0.331 0.043 CHEMBL3542256 0.213 0.091 CHEMBL3542258 0.224 0.084 CHEMBL3542257 0.183 0.112 CHEMBL4525787 0.183 0.112 CHEMBL3542266 | CHEMBL3542256 | |
| 0.059 | 0.242 | 0.404 | Amyloid beta aggregation inhibitor | 0.281 0.049 CHEMBL3542244 0.133 0.122 CHEMBL3542389 0.133 0.122 CHEMBL3542339 0.404 0.024 CHEMBL3542256 0.24 0.061 CHEMBL3542258 0.178 0.09 CHEMBL4525788 0.178 0.09 CHEMBL3542390 0.134 0.122 CHEMBL4525787 0.134 0.122 CHEMBL3542266 | CHEMBL3542256 | |
| 0.009 | 0.197 | 0.148 | NMDA receptor subunit 3A antagonist | 0.04 0.025 CHEMBL3542256 0.148 0.005 CHEMBL3542258 | CHEMBL3542258 | |
| 0.037 | 0.226 | 0.15 | Expectorant | 0.093 0.078 CHEMBL3542244 0.126 0.046 CHEMBL3542256 0.15 0.035 CHEMBL3542258 0.097 0.073 CHEMBL4525788 0.097 0.073 CHEMBL3542390 | CHEMBL3542258 | |
| 0.026 | 0.218 | 0.068 | Nicotinic alpha3beta2 receptor antagonist | 0.068 0.019 CHEMBL3542244 0.052 0.039 CHEMBL3542256 | CHEMBL3542244 | |
| 0.039 | 0.237 | 0.141 | 5 Hydroxytryptamine 2B antagonist | 0.141 0.045 CHEMBL3542244 0.103 0.08 CHEMBL3542256 0.11 0.071 CHEMBL3542258 0.105 0.078 CHEMBL3542257 | CHEMBL3542244 | |
| 0.123 | 0.322 | 0.233 | Insulysin inhibitor | 0.207 0.147 CHEMBL3542244 0.233 0.114 CHEMBL3542256 | CHEMBL3542256 | |
| 0.014 | 0.213 | 0.065 | Acetyl-CoA carboxylase inhibitor | 0.065 0.013 CHEMBL4525788 0.065 0.013 CHEMBL3542390 | CHEMBL3542390 | |
| 0.015 | 0.215 | 0.079 | Phosphodiesterase 4C inhibitor | 0.079 0.022 CHEMBL3542257 | CHEMBL3542257 | |
| 0.037 | 0.243 | 0.264 | Bronchodilator | 0.182 0.022 CHEMBL3542187 0.264 0.012 CHEMBL3542258 0.088 0.076 CHEMBL3542257 | CHEMBL3542258 | |
| 0.01 | 0.216 | 0.047 | Phosphodiesterase 2A inhibitor | 0.047 0.04 CHEMBL3542257 | CHEMBL3542257 | |
| 0.018 | 0.225 | 0.094 | Dopamine agonist | 0.057 0.055 CHEMBL3542244 0.094 0.03 CHEMBL3542256 | CHEMBL3542256 | |
| 0.039 | 0.247 | 0.213 | Nitric-oxide synthase inhibitor | 0.213 0.008 CHEMBL3542244 0.186 0.012 CHEMBL3542256 0.119 0.038 CHEMBL3542258 0.093 0.072 CHEMBL3542257 0.128 0.033 CHEMBL4525788 0.128 0.033 CHEMBL3542390 | CHEMBL3542244 | |
| 0.038 | 0.247 | 0.09 | EphA2 antagonist | 0.09 0.087 CHEMBL3542257 | CHEMBL3542257 | |
| 0.031 | 0.241 | 0.119 | Beta 3 adrenoreceptor antagonist | 0.069 0.036 CHEMBL3542244 0.092 0.017 CHEMBL3542256 0.119 0.01 CHEMBL3542258 | CHEMBL3542258 | |
| 0.08 | 0.29 | 0.138 | Pregnane X receptor agonist | 0.138 0.079 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.224 | 0.152 | NMDA receptor subunit 3B antagonist | 0.041 0.033 CHEMBL3542244 0.055 0.022 CHEMBL3542256 0.152 0.006 CHEMBL3542258 | CHEMBL3542258 | |
| 0.007 | 0.219 | 0.04 | Liver X receptor beta antagonist | 0.04 0.013 CHEMBL3542257 | CHEMBL3542257 | |
| 0.029 | 0.241 | 0.335 | Ca(v)3.2 blocker | 0.335 0.003 CHEMBL4525788 0.335 0.003 CHEMBL3542390 | CHEMBL3542390 | |
| 0.009 | 0.222 | 0.054 | Phosphodiesterase II inhibitor | 0.054 0.041 CHEMBL3542257 | CHEMBL3542257 | |
| 0.01 | 0.223 | 0.057 | Nicotinic receptor beta4 subunit antagonist | 0.033 0.032 CHEMBL3542187 0.057 0.013 CHEMBL3542258 | CHEMBL3542258 | |
| 0.03 | 0.244 | 0.248 | Inducible nitric-oxide synthase inhibitor | 0.248 0.005 CHEMBL3542244 0.22 0.006 CHEMBL3542256 0.15 0.016 CHEMBL3542258 0.103 0.035 CHEMBL3542257 0.155 0.015 CHEMBL4525788 0.155 0.015 CHEMBL3542390 | CHEMBL3542244 | |
| 0.086 | 0.304 | 0.145 | ATPase inhibitor | 0.145 0.11 CHEMBL3542257 | CHEMBL3542257 | |
| 0.028 | 0.246 | 0.132 | 5 Hydroxytryptamine antagonist | 0.132 0.058 CHEMBL3542244 | CHEMBL3542244 | |
| 0.013 | 0.233 | 0.041 | Ceramide glucosyltransferase inhibitor | 0.041 0.016 CHEMBL3542258 0.038 0.02 CHEMBL4525788 0.038 0.02 CHEMBL3542390 | CHEMBL3542258 | |
| 0.114 | 0.336 | 0.164 | ErbB-1 antagonist | 0.164 0.145 CHEMBL3542244 | CHEMBL3542244 | |
| 0.012 | 0.236 | 0.055 | Alpha tubulin antagonist | 0.055 0.035 CHEMBL3542256 0.047 0.046 CHEMBL4525788 0.047 0.046 CHEMBL3542390 | CHEMBL3542256 | |
| 0.045 | 0.272 | 0.487 | Psychostimulant | 0.223 0.069 CHEMBL3542244 0.196 0.082 CHEMBL3542187 0.215 0.072 CHEMBL3542256 0.487 0.012 CHEMBL3542258 0.195 0.083 CHEMBL4525788 0.195 0.083 CHEMBL3542390 | CHEMBL3542258 | |
| 0.007 | 0.243 | 0.044 | Sphingosine 1-phosphate receptor 1 agonist | 0.044 0.026 CHEMBL3542244 0.043 0.027 CHEMBL3542258 0.043 0.029 CHEMBL3542257 | CHEMBL3542244 | |
| 0.009 | 0.25 | 0.061 | 5 Hydroxytryptamine 1A antagonist | 0.061 0.052 CHEMBL3542244 | CHEMBL3542244 | |
| 0.017 | 0.258 | 0.076 | Vanilloid antagonist | 0.076 0.05 CHEMBL3542257 | CHEMBL3542257 | |
| 0.019 | 0.261 | 0.107 | Sphingosine kinase inhibitor | 0.08 0.016 CHEMBL3542244 0.096 0.009 CHEMBL3542256 0.107 0.006 CHEMBL4525788 0.107 0.006 CHEMBL3542390 | CHEMBL3542390 | |
| 0.008 | 0.252 | 0.03 | 5 Hydroxytryptamine 6 agonist | 0.03 0.018 CHEMBL3542244 | CHEMBL3542244 | |
| 0.063 | 0.307 | 0.253 | Nitric oxide antagonist | 0.139 0.107 CHEMBL3542244 0.189 0.072 CHEMBL3542256 0.136 0.111 CHEMBL3542258 0.253 0.051 CHEMBL4525788 0.253 0.051 CHEMBL3542390 | CHEMBL3542390 | |
| 0.023 | 0.27 | 0.074 | Calcium antagonist | 0.074 0.07 CHEMBL3542244 | CHEMBL3542244 | |
| 0.007 | 0.255 | 0.029 | 1,3-Beta-glucan synthase inhibitor | 0.029 0.018 CHEMBL3542258 0.027 0.023 CHEMBL4525788 0.027 0.023 CHEMBL3542390 | CHEMBL3542258 | |
| 0.009 | 0.263 | 0.297 | NMDA 2C receptor antagonist | 0.084 0.022 CHEMBL3542244 0.083 0.023 CHEMBL3542187 0.086 0.022 CHEMBL3542256 0.297 0.004 CHEMBL3542258 | CHEMBL3542258 | |
| 0.009 | 0.266 | 0.089 | Dopamine D5 agonist | 0.056 0.014 CHEMBL3542244 0.089 0.005 CHEMBL3542256 | CHEMBL3542256 | |
| 0.005 | 0.264 | 0.038 | Peroxisome proliferator-activated receptor delta agonist | 0.038 0.019 CHEMBL3542257 | CHEMBL3542257 | |
| 0.064 | 0.324 | 0.149 | Platelet aggregation inhibitor | 0.149 0.13 CHEMBL3542257 | CHEMBL3542257 | |
| 0.059 | 0.32 | 0.215 | Antimitotic | 0.179 0.096 CHEMBL3542244 0.215 0.076 CHEMBL3542256 0.202 0.083 CHEMBL3542258 0.138 0.134 CHEMBL3542257 0.204 0.082 CHEMBL4525788 0.204 0.082 CHEMBL3542390 | CHEMBL3542256 | |
| 0.025 | 0.287 | 0.124 | Platelet activating factor antagonist | 0.124 0.061 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.288 | 0.09 | Glutamate (mGluR7) antagonist | 0.09 0.017 CHEMBL3542257 | CHEMBL3542257 | |
| 0.116 | 0.38 | 0.303 | Caspase 3 stimulant | 0.231 0.131 CHEMBL3542256 0.303 0.077 CHEMBL3542257 0.215 0.148 CHEMBL4525788 0.215 0.148 CHEMBL3542390 0.192 0.181 CHEMBL4525787 0.192 0.181 CHEMBL3542266 | CHEMBL3542257 | |
| 0.005 | 0.269 | 0.03 | Imidazoline I1 receptor antagonist | 0.03 0.007 CHEMBL3542244 | CHEMBL3542244 | |
| 0.058 | 0.324 | 0.179 | Interleukin agonist | 0.179 0.14 CHEMBL3542187 | CHEMBL3542187 | |
| 0.004 | 0.273 | 0.027 | Nicotinic alpha4beta2 receptor agonist | 0.027 0.022 CHEMBL3542244 | CHEMBL3542244 | |
| 0.005 | 0.278 | 0.041 | Vascular adhesion protein 1 inhibitor | 0.041 0.024 CHEMBL3542257 | CHEMBL3542257 | |
| 0.011 | 0.288 | 0.073 | Acetylcholine M5 receptor agonist | 0.073 0.041 CHEMBL3542257 | CHEMBL3542257 | |
| 0.001 | 0.277 | 0.007 | CC chemokine 6 receptor agonist | 0.007 0.004 CHEMBL3542257 | CHEMBL3542257 | |
| 0.054 | 0.332 | 0.205 | Hypolipemic | 0.205 0.09 CHEMBL3542258 0.144 0.143 CHEMBL3542257 | CHEMBL3542258 | |
| 0.143 | 0.421 | 0.461 | 5 Hydroxytryptamine release inhibitor | 0.371 0.098 CHEMBL3542244 0.341 0.123 CHEMBL3542256 0.334 0.13 CHEMBL3542258 0.461 0.046 CHEMBL3542257 0.283 0.185 CHEMBL4525788 0.283 0.185 CHEMBL3542390 | CHEMBL3542257 | |
| 0.015 | 0.297 | 0.087 | Beta 1 adrenoreceptor antagonist | 0.059 0.036 CHEMBL3542244 0.076 0.021 CHEMBL3542256 0.087 0.014 CHEMBL3542258 | CHEMBL3542258 | |
| 0.01 | 0.293 | 0.058 | Toll-Like receptor 8 antagonist | 0.058 0.033 CHEMBL3542244 0.054 0.037 CHEMBL3542257 | CHEMBL3542244 | |
| 0.016 | 0.3 | 0.046 | Histamine H4 receptor antagonist | 0.046 0.038 CHEMBL3542244 | CHEMBL3542244 | |
| 0.015 | 0.304 | 0.11 | Beta 2 adrenoreceptor antagonist | 0.071 0.016 CHEMBL3542244 0.094 0.009 CHEMBL3542256 0.11 0.007 CHEMBL3542258 0.061 0.023 CHEMBL4525788 0.061 0.023 CHEMBL3542390 | CHEMBL3542258 | |
| 0.063 | 0.352 | 0.177 | Adenylate cyclase stimulant | 0.148 0.067 CHEMBL3542244 0.173 0.032 CHEMBL3542256 0.177 0.029 CHEMBL3542258 0.139 0.083 CHEMBL4525788 0.139 0.083 CHEMBL3542390 | CHEMBL3542258 | |
| 0.026 | 0.321 | 0.073 | Beta 2 adrenoreceptor agonist | 0.058 0.057 CHEMBL3542244 0.068 0.024 CHEMBL3542256 0.073 0.015 CHEMBL3542258 0.059 0.053 CHEMBL4525788 0.059 0.053 CHEMBL3542390 | CHEMBL3542258 | |
| 0.011 | 0.306 | 0.051 | Liver X receptor alpha agonist | 0.051 0.018 CHEMBL3542257 | CHEMBL3542257 | |
| 0.004 | 0.299 | 0.034 | Nicotinic alpha3beta4 receptor agonist | 0.034 0.016 CHEMBL3542244 | CHEMBL3542244 | |
| 0.016 | 0.311 | 0.194 | Phosphodiesterase III inhibitor | 0.194 0.007 CHEMBL3542257 | CHEMBL3542257 | |
| 0.065 | 0.361 | 0.101 | Sphingosine 1-phosphate receptor 2 agonist | 0.101 0.099 CHEMBL3542244 | CHEMBL3542244 | |
| 0.001 | 0.301 | 0.006 | Insulin like growth factor 3 antagonist | 0.006 0.004 CHEMBL3542257 | CHEMBL3542257 | |
| 0.095 | 0.405 | 0.437 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.437 0.015 CHEMBL3542244 0.432 0.015 CHEMBL3542256 0.285 0.075 CHEMBL3542258 0.368 0.03 CHEMBL4525788 0.368 0.03 CHEMBL3542390 | CHEMBL3542244 | |
| 0.009 | 0.319 | 0.046 | Sphingosine 1-phosphate receptor agonist | 0.041 0.036 CHEMBL3542244 0.046 0.028 CHEMBL3542257 | CHEMBL3542257 | |
| 0.056 | 0.366 | 0.167 | Interleukin 6 antagonist | 0.138 0.109 CHEMBL3542244 0.159 0.077 CHEMBL3542256 0.158 0.078 CHEMBL3542257 0.167 0.068 CHEMBL4525788 0.167 0.068 CHEMBL3542390 | CHEMBL3542390 | |
| 0.016 | 0.326 | 0.075 | Lipase inhibitor | 0.075 0.048 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.325 | 0.068 | H+/K+-transporting ATPase inhibitor | 0.068 0.019 CHEMBL3542257 | CHEMBL3542257 | |
| 0.012 | 0.323 | 0.04 | Tryptophan 5 hydroxylase inhibitor | 0.034 0.03 CHEMBL3542244 0.04 0.015 CHEMBL3542258 | CHEMBL3542258 | |
| 0.025 | 0.339 | 0.323 | Vascular endothelial growth factor 3 antagonist | 0.323 0.016 CHEMBL3542257 | CHEMBL3542257 | |
| 0.067 | 0.381 | 0.174 | Focal adhesion kinase 2 inhibitor | 0.174 0.095 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.344 | 0.102 | TRKB antagonist | 0.102 0.098 CHEMBL3542257 | CHEMBL3542257 | |
| 0.073 | 0.392 | 0.402 | Superoxide dismutase inhibitor | 0.299 0.051 CHEMBL3542244 0.402 0.026 CHEMBL3542256 0.237 0.083 CHEMBL3542258 0.24 0.081 CHEMBL3542257 0.209 0.108 CHEMBL4525788 0.209 0.108 CHEMBL3542390 | CHEMBL3542256 | |
| 0.018 | 0.339 | 0.13 | Beta adrenoreceptor antagonist | 0.083 0.025 CHEMBL3542244 0.111 0.013 CHEMBL3542256 0.13 0.008 CHEMBL3542258 0.073 0.034 CHEMBL4525788 0.073 0.034 CHEMBL3542390 | CHEMBL3542258 | |
| 0.01 | 0.332 | 0.142 | TRPA1 antagonist | 0.142 0.01 CHEMBL3542257 | CHEMBL3542257 | |
| 0.158 | 0.481 | 0.335 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.335 0.168 CHEMBL3542257 | CHEMBL3542257 | |
| 0.01 | 0.337 | 0.056 | Sphingosine kinase 1 inhibitor | 0.041 0.029 CHEMBL3542244 0.047 0.019 CHEMBL3542256 0.056 0.012 CHEMBL4525788 0.056 0.012 CHEMBL3542390 | CHEMBL3542390 | |
| 0.1 | 0.427 | 0.217 | Apoptosis antagonist | 0.217 0.159 CHEMBL3542256 | CHEMBL3542256 | |
| 0.051 | 0.378 | 0.097 | Folate antagonist | 0.097 0.07 CHEMBL3542257 | CHEMBL3542257 | |
| 0.006 | 0.336 | 0.076 | Raf kinase C inhibitor | 0.076 0.034 CHEMBL3542257 | CHEMBL3542257 | |
| 0.02 | 0.35 | 0.075 | Pregnane X receptor antagonist | 0.053 0.052 CHEMBL3542256 0.075 0.01 CHEMBL3542257 | CHEMBL3542257 | |
| 0.009 | 0.344 | 0.051 | Nicotinic receptor alpha7 subunit antagonist | 0.051 0.042 CHEMBL3542244 0.049 0.046 CHEMBL3542258 | CHEMBL3542244 | |
| 0.004 | 0.34 | 0.054 | Diamine oxidase inhibitor | 0.054 0.013 CHEMBL3542257 | CHEMBL3542257 | |
| 0.082 | 0.423 | 0.384 | Vasodilator, peripheral | 0.243 0.133 CHEMBL3542244 0.272 0.112 CHEMBL3542256 0.384 0.06 CHEMBL3542258 0.24 0.135 CHEMBL3542257 | CHEMBL3542258 | |
| 0.114 | 0.458 | 0.297 | 5 Hydroxytryptamine uptake stimulant | 0.268 0.065 CHEMBL3542244 0.297 0.047 CHEMBL3542256 0.197 0.159 CHEMBL3542258 0.203 0.146 CHEMBL3542257 0.221 0.115 CHEMBL4525788 0.221 0.115 CHEMBL3542390 | CHEMBL3542256 | |
| 0.098 | 0.443 | 0.208 | Peptidyltransferase inhibitor | 0.204 0.094 CHEMBL3542187 0.208 0.089 CHEMBL3542258 | CHEMBL3542258 | |
| 0.004 | 0.349 | 0.025 | Beta 1 adrenoreceptor agonist | 0.021 0.019 CHEMBL3542256 0.025 0.012 CHEMBL3542258 | CHEMBL3542258 | |
| 0.015 | 0.361 | 0.12 | Platelet activating factor alpha antagonist | 0.12 0.045 CHEMBL3542257 | CHEMBL3542257 | |
| 0.015 | 0.37 | 0.069 | Vanilloid 3 antagonist | 0.069 0.004 CHEMBL3542257 | CHEMBL3542257 | |
| 0.01 | 0.369 | 0.046 | Lysophosphatidic acid 3 receptor antagonist | 0.046 0.042 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.387 | 0.086 | Exportin-1 inhibitor | 0.072 0.038 CHEMBL3542244 0.071 0.04 CHEMBL3542258 0.086 0.018 CHEMBL3542257 0.065 0.056 CHEMBL4525788 0.065 0.056 CHEMBL3542390 | CHEMBL3542257 | |
| 0.032 | 0.394 | 0.174 | Beta amyloid protein antagonist | 0.174 0.027 CHEMBL3542257 | CHEMBL3542257 | |
| 0.038 | 0.401 | 0.153 | Cyclooxygenase 3 inhibitor | 0.103 0.099 CHEMBL3542244 0.113 0.085 CHEMBL3542256 0.153 0.045 CHEMBL3542258 | CHEMBL3542258 | |
| 0.044 | 0.412 | 0.136 | Platelet adhesion inhibitor | 0.136 0.123 CHEMBL4525788 0.136 0.123 CHEMBL3542390 | CHEMBL3542390 | |
| 0.005 | 0.373 | 0.115 | Phosphodiesterase 3B inhibitor | 0.115 0.009 CHEMBL3542257 | CHEMBL3542257 | |
| 0.01 | 0.382 | 0.064 | Androgen agonist | 0.054 0.051 CHEMBL3542256 0.064 0.036 CHEMBL3542258 | CHEMBL3542258 | |
| 0.021 | 0.393 | 0.094 | Mucolytic | 0.094 0.086 CHEMBL3542258 | CHEMBL3542258 | |
| 0.033 | 0.405 | 0.118 | Anticoagulant | 0.118 0.115 CHEMBL3542244 | CHEMBL3542244 | |
| 0.034 | 0.406 | 0.149 | Toll-Like receptor 2 antagonist | 0.149 0.053 CHEMBL3542256 0.102 0.101 CHEMBL3542257 | CHEMBL3542256 | |
| 0.031 | 0.406 | 0.133 | Toll-Like receptor antagonist | 0.128 0.074 CHEMBL3542244 0.133 0.069 CHEMBL3542256 0.115 0.092 CHEMBL3542257 | CHEMBL3542256 | |
| 0.016 | 0.391 | 0.15 | Fibroblast growth factor 1 antagonist | 0.15 0.031 CHEMBL3542257 | CHEMBL3542257 | |
| 0.02 | 0.395 | 0.426 | Vascular endothelial growth factor 1 antagonist | 0.426 0.005 CHEMBL3542257 | CHEMBL3542257 | |
| 0.099 | 0.476 | 0.316 | Apoptosis agonist | 0.316 0.161 CHEMBL3542256 0.264 0.2 CHEMBL4525788 0.264 0.2 CHEMBL3542390 | CHEMBL3542256 | |
| 0.115 | 0.495 | 0.336 | MAP kinase kinase 6 inhibitor | 0.336 0.103 CHEMBL3542257 | CHEMBL3542257 | |
| 0.026 | 0.407 | 0.307 | Phosphodiesterase inhibitor | 0.307 0.014 CHEMBL3542257 | CHEMBL3542257 | |
| 0.016 | 0.397 | 0.194 | Phosphodiesterase 3A inhibitor | 0.194 0.009 CHEMBL3542257 | CHEMBL3542257 | |
| 0.035 | 0.422 | 0.297 | Cytokine production inhibitor | 0.297 0.015 CHEMBL3542257 | CHEMBL3542257 | |
| 0.087 | 0.477 | 0.136 | Ca2+-transporting ATPase inhibitor | 0.13 0.12 CHEMBL3542244 0.133 0.105 CHEMBL3542256 0.136 0.092 CHEMBL3542258 0.131 0.115 CHEMBL3542257 0.136 0.088 CHEMBL4525788 0.136 0.088 CHEMBL3542390 | CHEMBL3542390 | |
| 0.015 | 0.407 | 0.053 | Beta adrenoreceptor agonist | 0.047 0.025 CHEMBL3542256 0.053 0.014 CHEMBL3542258 | CHEMBL3542258 | |
| 0.064 | 0.457 | 0.191 | Antithrombotic | 0.191 0.189 CHEMBL3542258 | CHEMBL3542258 | |
| 0.011 | 0.406 | 0.065 | Fibroblast growth factor 2 antagonist | 0.065 0.045 CHEMBL3542257 | CHEMBL3542257 | |
| 0.017 | 0.416 | 0.203 | Glutamate receptor antagonist | 0.203 0.025 CHEMBL3542258 | CHEMBL3542258 | |
| 0.031 | 0.43 | 0.079 | mTOR complex 2 inhibitor | 0.079 0.071 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.431 | 0.123 | Thrombolytic | 0.123 0.107 CHEMBL3542256 | CHEMBL3542256 | |
| 0.025 | 0.432 | 0.129 | HIV-1 integrase (Overall Integration) inhibitor | 0.089 0.066 CHEMBL3542244 0.129 0.034 CHEMBL3542256 0.129 0.034 CHEMBL3542258 | CHEMBL3542258 | |
| 0.009 | 0.418 | 0.091 | Proto-oncogene tyrosine-protein kinase Kit inhibitor | 0.091 0.063 CHEMBL3542257 | CHEMBL3542257 | |
| 0.029 | 0.438 | 0.124 | Protein kinase stimulant | 0.116 0.097 CHEMBL3542256 0.124 0.088 CHEMBL3542258 | CHEMBL3542258 | |
| 0.019 | 0.432 | 0.076 | Myeloperoxidase inhibitor | 0.076 0.074 CHEMBL3542257 | CHEMBL3542257 | |
| 0.016 | 0.429 | 0.075 | Transcription factor AP-1 inhibitor | 0.075 0.025 CHEMBL3542257 | CHEMBL3542257 | |
| 0.008 | 0.423 | 0.088 | Phosphodiesterase 4B inhibitor | 0.088 0.031 CHEMBL3542257 | CHEMBL3542257 | |
| 0.022 | 0.441 | 0.105 | AMP-activated protein kinase stimulant | 0.091 0.085 CHEMBL3542256 0.105 0.065 CHEMBL3542257 | CHEMBL3542257 | |
| 0.028 | 0.45 | 0.08 | Transcription factor RelA inhibitor | 0.08 0.017 CHEMBL3542257 | CHEMBL3542257 | |
| 0.007 | 0.43 | 0.058 | Dihydrofolate reductase inhibitor | 0.058 0.012 CHEMBL3542257 | CHEMBL3542257 | |
| 0.014 | 0.439 | 0.091 | Platelet growth factor antagonist | 0.091 0.047 CHEMBL3542257 | CHEMBL3542257 | |
| 0.087 | 0.512 | 0.378 | Cyclophilin D inhibitor | 0.288 0.174 CHEMBL3542244 0.332 0.137 CHEMBL3542256 0.369 0.109 CHEMBL3542258 0.32 0.146 CHEMBL3542257 0.378 0.104 CHEMBL4525788 0.378 0.104 CHEMBL3542390 | CHEMBL3542390 | |
| 0.014 | 0.439 | 0.175 | Adrenaline agonist | 0.089 0.047 CHEMBL3542244 0.134 0.02 CHEMBL3542256 0.175 0.01 CHEMBL3542258 | CHEMBL3542258 | |
| 0.018 | 0.443 | 0.112 | TRKA antagonist | 0.112 0.075 CHEMBL3542257 | CHEMBL3542257 | |
| 0.03 | 0.46 | 0.182 | Insulin sensitizer | 0.182 0.093 CHEMBL3542258 0.163 0.115 CHEMBL3542257 | CHEMBL3542258 | |
| 0.03 | 0.462 | 0.096 | Phosphodiesterase 7B inhibitor | 0.096 0.061 CHEMBL3542257 | CHEMBL3542257 | |
| 0.016 | 0.449 | 0.066 | Peroxisome proliferator-activated receptor gamma antagonist | 0.066 0.065 CHEMBL3542257 | CHEMBL3542257 | |
| 0.033 | 0.468 | 0.134 | MAP3K9 inhibitor | 0.134 0.087 CHEMBL3542258 | CHEMBL3542258 | |
| 0.025 | 0.462 | 0.21 | I kappa B kinase epsilon inhibitor | 0.21 0.062 CHEMBL3542257 | CHEMBL3542257 | |
| 0.012 | 0.451 | 0.104 | Granulocyte macrophage colony stimulating factor antagonist | 0.104 0.067 CHEMBL3542257 | CHEMBL3542257 | |
| 0.068 | 0.516 | 0.17 | Catenin beta inhibitor | 0.17 0.067 CHEMBL4525788 0.17 0.067 CHEMBL3542390 | CHEMBL3542390 | |
| 0.017 | 0.47 | 0.122 | Tyrosine-protein kinase receptor antagonist | 0.122 0.084 CHEMBL3542257 | CHEMBL3542257 | |
| 0.031 | 0.486 | 0.09 | Carbonic anhydrase XV inhibitor | 0.09 0.083 CHEMBL3542257 | CHEMBL3542257 | |
| 0.088 | 0.544 | 0.202 | Interleukin 2 agonist | 0.202 0.186 CHEMBL3542258 | CHEMBL3542258 | |
| 0.003 | 0.459 | 0.042 | Free fatty acid receptor 1 antagonist | 0.042 0.014 CHEMBL3542257 | CHEMBL3542257 | |
| 0.028 | 0.484 | 0.088 | Granulocyte macrophage colony stimulating factor agonist | 0.088 0.056 CHEMBL3542257 | CHEMBL3542257 | |
| 0.008 | 0.468 | 0.06 | Alpha 2 adrenoreceptor agonist | 0.056 0.047 CHEMBL3542244 0.054 0.051 CHEMBL3542256 0.06 0.042 CHEMBL3542258 | CHEMBL3542258 | |
| 0.017 | 0.48 | 0.074 | Histone deacetylase SIRT1 stimulant | 0.074 0.05 CHEMBL3542257 | CHEMBL3542257 | |
| 0.017 | 0.48 | 0.074 | Histone deacetylase stimulant | 0.074 0.05 CHEMBL3542257 | CHEMBL3542257 | |
| 0.006 | 0.475 | 0.08 | Fibroblast growth factor 3 antagonist | 0.08 0.051 CHEMBL3542257 | CHEMBL3542257 | |
| 0.031 | 0.504 | 0.117 | Sphingosine 1-phosphate receptor 2 antagonist | 0.117 0.105 CHEMBL3542256 | CHEMBL3542256 | |
| 0.015 | 0.488 | 0.084 | Polo-like kinase-1 inhibitor | 0.084 0.074 CHEMBL3542244 | CHEMBL3542244 | |
| 0.011 | 0.485 | 0.071 | Aryl hydrocarbon receptor antagonist | 0.071 0.036 CHEMBL3542257 | CHEMBL3542257 | |
| 0.057 | 0.537 | 0.386 | Toll-Like receptor 7 agonist | 0.285 0.12 CHEMBL3542208 0.302 0.108 CHEMBL3542258 0.386 0.066 CHEMBL3542257 0.299 0.111 CHEMBL3542243 0.262 0.137 CHEMBL4525787 0.262 0.137 CHEMBL3542266 | CHEMBL3542257 | |
| 0.103 | 0.584 | 0.196 | MAP kinase kinase 3 inhibitor | 0.196 0.133 CHEMBL3542257 0.184 0.176 CHEMBL3542243 | CHEMBL3542257 | |
| 0.017 | 0.505 | 0.057 | Corticotropin releasing factor 2 receptor antagonist | 0.057 0.054 CHEMBL3542257 | CHEMBL3542257 | |
| 0.005 | 0.494 | 0.075 | Alpha adrenoreceptor agonist | 0.075 0.041 CHEMBL3542258 | CHEMBL3542258 | |
| 0.016 | 0.505 | 0.125 | Gastric antisecretory | 0.125 0.04 CHEMBL3542257 | CHEMBL3542257 | |
| 0.082 | 0.571 | 0.13 | Heat shock protein 70 antagonist | 0.13 0.12 CHEMBL3542257 | CHEMBL3542257 | |
| 0.026 | 0.515 | 0.112 | Cell wall synthesis inhibitor | 0.112 0.111 CHEMBL3542258 | CHEMBL3542258 | |
| 0.009 | 0.5 | 0.149 | Vascular endothelial growth factor 2 antagonist | 0.149 0.049 CHEMBL3542257 | CHEMBL3542257 | |
| 0.014 | 0.505 | 0.188 | Vascular endothelial growth factor antagonist | 0.188 0.042 CHEMBL3542257 | CHEMBL3542257 | |
| 0.08 | 0.571 | 0.2 | Nitric-oxide synthase stimulant | 0.182 0.123 CHEMBL3542256 0.189 0.108 CHEMBL3542258 0.2 0.089 CHEMBL3542257 0.198 0.093 CHEMBL4525788 0.198 0.093 CHEMBL3542390 | CHEMBL3542257 | |
| 0.027 | 0.522 | 0.131 | Interleukin 1b antagonist | 0.131 0.054 CHEMBL3542257 | CHEMBL3542257 | |
| 0.053 | 0.548 | 0.381 | Toll-Like receptor agonist | 0.28 0.124 CHEMBL3542208 0.3 0.111 CHEMBL3542258 0.381 0.068 CHEMBL3542257 0.297 0.113 CHEMBL3542243 0.257 0.142 CHEMBL4525787 0.257 0.142 CHEMBL3542266 | CHEMBL3542257 | |
| 0.052 | 0.548 | 0.296 | Histamine release inhibitor | 0.296 0.126 CHEMBL3542257 | CHEMBL3542257 | |
| 0.035 | 0.537 | 0.138 | Melanin inhibitor | 0.138 0.099 CHEMBL3542256 0.13 0.115 CHEMBL3542258 | CHEMBL3542256 | |
| 0.045 | 0.552 | 0.128 | Sphingosine 1-phosphate receptor 5 antagonist | 0.126 0.111 CHEMBL3542244 0.128 0.106 CHEMBL3542256 | CHEMBL3542256 | |
| 0.054 | 0.564 | 0.267 | Vasodilator, coronary | 0.212 0.171 CHEMBL3542244 0.232 0.152 CHEMBL3542256 0.267 0.118 CHEMBL3542258 | CHEMBL3542258 | |
| 0.016 | 0.532 | 0.112 | Growth factor antagonist | 0.112 0.101 CHEMBL3542257 | CHEMBL3542257 | |
| 0.033 | 0.55 | 0.113 | Interleukin 4 antagonist | 0.113 0.096 CHEMBL3542256 | CHEMBL3542256 | |
| 0.024 | 0.541 | 0.099 | DOPA decarboxylase inhibitor | 0.099 0.077 CHEMBL3542256 0.093 0.09 CHEMBL3542257 | CHEMBL3542256 | |
| 0.004 | 0.526 | 0.07 | Phosphodiesterase X inhibitor | 0.07 0.016 CHEMBL3542257 | CHEMBL3542257 | |
| 0.004 | 0.526 | 0.07 | Phosphodiesterase 10A inhibitor | 0.07 0.016 CHEMBL3542257 | CHEMBL3542257 | |
| 0.006 | 0.535 | 0.052 | Mannosidase inhibitor | 0.052 0.024 CHEMBL4525788 0.052 0.024 CHEMBL3542390 | CHEMBL3542390 | |
| 0.023 | 0.552 | 0.16 | EphB2 antagonist | 0.16 0.12 CHEMBL3542257 | CHEMBL3542257 | |
| 0.037 | 0.567 | 0.514 | Angiogenesis inhibitor | 0.514 0.027 CHEMBL3542257 | CHEMBL3542257 | |
| 0.022 | 0.561 | 0.132 | Activin receptor-like kinase 2 inhibitor | 0.132 0.083 CHEMBL3542257 | CHEMBL3542257 | |
| 0.007 | 0.557 | 0.057 | Alpha-mannosidase inhibitor | 0.051 0.041 CHEMBL3542258 0.057 0.031 CHEMBL4525788 0.057 0.031 CHEMBL3542390 | CHEMBL3542390 | |
| 0.002 | 0.553 | 0.059 | Glutamate (mGluR2) antagonist | 0.059 0.006 CHEMBL3542257 | CHEMBL3542257 | |
| 0.003 | 0.557 | 0.076 | Glutamate (mGluR group II) antagonist | 0.076 0.007 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.581 | 0.188 | Antioxidant | 0.188 0.124 CHEMBL3542256 | CHEMBL3542256 | |
| 0.021 | 0.581 | 0.181 | Interleukin antagonist | 0.181 0.095 CHEMBL3542257 | CHEMBL3542257 | |
| 0.034 | 0.608 | 0.214 | Immunosuppressant | 0.214 0.183 CHEMBL3542258 0.21 0.187 CHEMBL4525788 0.21 0.187 CHEMBL3542390 | CHEMBL3542258 | |
| 0.023 | 0.605 | 0.121 | Hemostatic | 0.121 0.111 CHEMBL3542256 | CHEMBL3542256 | |
| 0.021 | 0.606 | 0.184 | 12-Lipoxygenase inhibitor | 0.184 0.169 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.604 | 0.061 | Purinergic P2X1 antagonist | 0.061 0.042 CHEMBL3542257 | CHEMBL3542257 | |
| 0.007 | 0.623 | 0.072 | Secretase beta inhibitor | 0.072 0.046 CHEMBL3542257 | CHEMBL3542257 | |
| 0.025 | 0.641 | 0.198 | Cyclic AMP phosphodiesterase inhibitor | 0.198 0.095 CHEMBL3542257 | CHEMBL3542257 | |
| 0.008 | 0.634 | 0.09 | CYP2A6 inhibitor | 0.09 0.041 CHEMBL3542257 | CHEMBL3542257 | |
| 0.02 | 0.649 | 0.179 | Amylase inhibitor | 0.179 0.052 CHEMBL3542256 0.155 0.062 CHEMBL3542258 0.177 0.053 CHEMBL4525788 0.177 0.053 CHEMBL3542390 | CHEMBL3542256 | |
| 0.011 | 0.642 | 0.108 | Lipid peroxidase inhibitor | 0.108 0.107 CHEMBL3542256 | CHEMBL3542256 | |
| 0.03 | 0.663 | 0.217 | Cholesterol antagonist | 0.217 0.15 CHEMBL3542257 | CHEMBL3542257 | |
| 0.024 | 0.663 | 0.372 | Hypoxia-inducible factor 1 alpha inhibitor | 0.186 0.171 CHEMBL3542244 0.251 0.099 CHEMBL3542256 0.372 0.038 CHEMBL3542258 0.293 0.069 CHEMBL3542257 0.185 0.172 CHEMBL4525788 0.185 0.172 CHEMBL3542390 | CHEMBL3542258 | |
| 0.042 | 0.683 | 0.174 | Growth factor agonist | 0.174 0.096 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.656 | 0.204 | Free radical scavenger | 0.204 0.094 CHEMBL3542256 | CHEMBL3542256 | |
| 0.009 | 0.652 | 0.074 | Macrophage migration inhibitory factor inhibitor | 0.074 0.059 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.701 | 0.073 | Factor IXa inhibitor | 0.073 0.019 CHEMBL3542257 | CHEMBL3542257 | |
| 0.009 | 0.713 | 0.16 | Death-associated protein kinase 3 inhibitor | 0.16 0.108 CHEMBL3542257 | CHEMBL3542257 | |
| 0.021 | 0.728 | 0.188 | Histone acetyltransferase inhibitor | 0.188 0.088 CHEMBL3542257 | CHEMBL3542257 | |
| 0.013 | 0.724 | 0.234 | Non-steroidal antiinflammatory agent | 0.138 0.134 CHEMBL3542258 0.234 0.05 CHEMBL3542257 | CHEMBL3542257 | |
| 0.014 | 0.732 | 0.145 | Interleukin 1 antagonist | 0.145 0.061 CHEMBL3542257 | CHEMBL3542257 | |
| 0.006 | 0.726 | 0.147 | Aryl hydrocarbon receptor agonist | 0.147 0.138 CHEMBL3542257 | CHEMBL3542257 | |
| 0.005 | 0.745 | 0.054 | Glucosylceramidase inhibitor | 0.054 0.04 CHEMBL4525788 0.054 0.04 CHEMBL3542390 | CHEMBL3542390 | |
| 0.022 | 0.765 | 0.14 | CF transmembrane conductance regulator agonist | 0.14 0.095 CHEMBL3542257 | CHEMBL3542257 | |
| 0.004 | 0.781 | 0.113 | Alcohol dehydrogenase inhibitor | 0.113 0.04 CHEMBL3542257 | CHEMBL3542257 | |
| 0.015 | 0.862 | 0.414 | Antiinflammatory | 0.414 0.131 CHEMBL3542258 0.325 0.193 CHEMBL4525788 0.325 0.193 CHEMBL3542390 | CHEMBL3542258 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |