| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.975 | 0.002 | 0.991 | Histone deacetylase 1 inhibitor | 0.991 0.002 CHEMBL734 | CHEMBL734 | |
| 0.973 | 0.002 | 0.994 | Histone deacetylase 6 inhibitor | 0.994 0.002 CHEMBL734 | CHEMBL734 | |
| 0.972 | 0.002 | 0.994 | Histone deacetylase class IIb inhibitor | 0.994 0.002 CHEMBL734 | CHEMBL734 | |
| 0.965 | 0.002 | 0.985 | Histone deacetylase class II inhibitor | 0.985 0.001 CHEMBL734 | CHEMBL734 | |
| 0.938 | 0.002 | 0.972 | Histone deacetylase 2 inhibitor | 0.972 0.002 CHEMBL734 | CHEMBL734 | |
| 0.803 | 0.002 | 0.923 | Histone deacetylase class IV inhibitor | 0.923 0.002 CHEMBL734 | CHEMBL734 | |
| 0.803 | 0.002 | 0.923 | Histone deacetylase 11 inhibitor | 0.923 0.002 CHEMBL734 | CHEMBL734 | |
| 0.799 | 0.003 | 0.955 | Histone deacetylase 3 inhibitor | 0.955 0.002 CHEMBL734 | CHEMBL734 | |
| 0.795 | 0.002 | 0.947 | Histone deacetylase class IIa inhibitor | 0.947 0.002 CHEMBL734 | CHEMBL734 | |
| 0.793 | 0.002 | 0.936 | Histone deacetylase 5 inhibitor | 0.936 0.001 CHEMBL734 | CHEMBL734 | |
| 0.791 | 0.001 | 0.791 | Aminopeptidase microsomal inhibitor | 0.577 0.002 CHEMBL734 | ||
| 0.783 | 0.001 | 0.783 | Aminopeptidase N inhibitor | 0.56 0.002 CHEMBL734 | ||
| 0.78 | 0.004 | 0.818 | Tumour necrosis factor alpha release inhibitor | 0.818 0.004 CHEMBL734 | CHEMBL734 | |
| 0.763 | 0.002 | 0.904 | Histone deacetylase 10 inhibitor | 0.904 0.002 CHEMBL734 | CHEMBL734 | |
| 0.744 | 0.002 | 0.744 | Peroxidase inhibitor | 0.622 0.004 CHEMBL734 | ||
| 0.728 | 0.003 | 0.728 | 5-Lipoxygenase inhibitor | 0.322 0.009 CHEMBL734 | ||
| 0.717 | 0.002 | 0.717 | Leukotriene A4 hydrolase inhibitor | 0.053 0.019 CHEMBL734 | ||
| 0.715 | 0.005 | 0.715 | Platelet antagonist | |||
| 0.56 | 0.002 | 0.56 | Chemokine receptor agonist | |||
| 0.543 | 0.014 | 0.543 | Lipoxygenase inhibitor | 0.374 0.044 CHEMBL734 | ||
| 0.529 | 0.002 | 0.529 | Glutamate decarboxylase inhibitor | 0.295 0.004 CHEMBL734 | ||
| 0.512 | 0.002 | 0.512 | CXC chemokine receptor agonist | |||
| 0.501 | 0.003 | 0.722 | Histone deacetylase 4 inhibitor | 0.722 0.002 CHEMBL734 | CHEMBL734 | |
| 0.494 | 0.003 | 0.494 | Leukotriene synthesis inhibitor | |||
| 0.435 | 0.001 | 0.435 | Retinoic acid alpha receptor agonist | |||
| 0.412 | 0.003 | 0.625 | Macrophage elastase inhibitor | 0.625 0.003 CHEMBL734 | CHEMBL734 | |
| 0.404 | 0.004 | 0.404 | Urease inhibitor | 0.304 0.005 CHEMBL734 | ||
| 0.401 | 0.003 | 0.484 | Triose-phosphate isomerase inhibitor | 0.484 0.003 CHEMBL734 | CHEMBL734 | |
| 0.401 | 0.004 | 0.401 | Alcohol oxidase inhibitor | 0.224 0.005 CHEMBL734 | ||
| 0.437 | 0.071 | 0.437 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.406 0.095 CHEMBL734 | ||
| 0.382 | 0.025 | 0.42 | Insulysin inhibitor | 0.42 0.019 CHEMBL734 | CHEMBL734 | |
| 0.347 | 0.007 | 0.347 | GABA C receptor agonist | 0.247 0.014 CHEMBL734 | ||
| 0.341 | 0.005 | 0.341 | Adenylate kinase inhibitor | 0.223 0.012 CHEMBL734 | ||
| 0.347 | 0.017 | 0.367 | Tyrosine 3 hydroxylase inhibitor | 0.367 0.013 CHEMBL734 | CHEMBL734 | |
| 0.362 | 0.034 | 0.362 | Superoxide dismutase inhibitor | 0.222 0.096 CHEMBL734 | ||
| 0.329 | 0.004 | 0.329 | GABA C receptor antagonist | 0.327 0.004 CHEMBL734 | ||
| 0.307 | 0.002 | 0.318 | ADAM10 endopeptidase inhibitor | 0.318 0.002 CHEMBL734 | CHEMBL734 | |
| 0.308 | 0.008 | 0.308 | Aminopeptidase B inhibitor | 0.283 0.01 CHEMBL734 | ||
| 0.371 | 0.075 | 0.441 | GABA C receptor rho-3 antagonist | 0.441 0.045 CHEMBL734 | CHEMBL734 | |
| 0.379 | 0.087 | 0.45 | Antibacterial | 0.45 0.057 CHEMBL734 | CHEMBL734 | |
| 0.411 | 0.133 | 0.411 | Antiinflammatory | |||
| 0.278 | 0.002 | 0.472 | Collagenase inhibitor | 0.472 0.002 CHEMBL734 | CHEMBL734 | |
| 0.278 | 0.004 | 0.546 | Phenylalanine 4-hydroxylase inhibitor | 0.546 0.002 CHEMBL734 | CHEMBL734 | |
| 0.292 | 0.02 | 0.372 | Tumour necrosis factor antagonist | 0.372 0.008 CHEMBL734 | CHEMBL734 | |
| 0.287 | 0.018 | 0.63 | Alpha-N-acetylglucosaminidase inhibitor | 0.63 0.004 CHEMBL734 | CHEMBL734 | |
| 0.246 | 0.024 | 0.246 | Interleukin 6 antagonist | 0.199 0.041 CHEMBL734 | ||
| 0.235 | 0.016 | 0.315 | Ferrochelatase inhibitor | 0.315 0.006 CHEMBL734 | CHEMBL734 | |
| 0.271 | 0.057 | 0.271 | Gastrin inhibitor | 0.232 0.101 CHEMBL734 | ||
| 0.211 | 0.002 | 0.211 | Nitric oxide donor | 0.064 0.041 CHEMBL734 | ||
| 0.214 | 0.007 | 0.214 | Carbamoyl phosphate synthetase inhibitor | 0.111 0.018 CHEMBL734 | ||
| 0.347 | 0.148 | 0.577 | Caspase 9 stimulant | 0.577 0.04 CHEMBL734 | CHEMBL734 | |
| 0.227 | 0.031 | 0.227 | Phospholipase C inhibitor | 0.166 0.079 CHEMBL734 | ||
| 0.263 | 0.069 | 0.267 | 5 Hydroxytryptamine uptake stimulant | 0.267 0.065 CHEMBL734 | CHEMBL734 | |
| 0.216 | 0.028 | 0.339 | M17 leucyl aminopeptidase inhibitor | 0.339 0.008 CHEMBL734 | CHEMBL734 | |
| 0.181 | 0.003 | 0.181 | Retinoic acid receptor agonist | |||
| 0.188 | 0.012 | 0.241 | Sphingomyelinase inhibitor | 0.241 0.005 CHEMBL734 | CHEMBL734 | |
| 0.19 | 0.019 | 0.305 | UDP-glucose 4-epimerase inhibitor | 0.305 0.01 CHEMBL734 | CHEMBL734 | |
| 0.189 | 0.019 | 0.189 | Adenylate cyclase stimulant | 0.187 0.021 CHEMBL734 | ||
| 0.206 | 0.044 | 0.241 | Succinate dehydrogenase inhibitor | 0.241 0.026 CHEMBL734 | CHEMBL734 | |
| 0.175 | 0.014 | 0.175 | Phosphofructokinase-1 inhibitor | 0.148 0.018 CHEMBL734 | ||
| 0.226 | 0.066 | 0.226 | MAP kinase kinase 2 inhibitor | 0.184 0.093 CHEMBL734 | ||
| 0.17 | 0.013 | 0.17 | Glutamate dehydrogenase inhibitor | 0.135 0.019 CHEMBL734 | ||
| 0.189 | 0.035 | 0.202 | Cell wall synthesis inhibitor | 0.202 0.029 CHEMBL734 | CHEMBL734 | |
| 0.233 | 0.08 | 0.233 | DNA synthesis inhibitor | 0.201 0.122 CHEMBL734 | ||
| 0.167 | 0.017 | 0.167 | Histidine decarboxylase inhibitor | 0.064 0.057 CHEMBL734 | ||
| 0.155 | 0.008 | 0.282 | Histone deacetylase inhibitor | 0.282 0.004 CHEMBL734 | CHEMBL734 | |
| 0.155 | 0.01 | 0.155 | Ribonucleoside-diphosphate reductase inhibitor | 0.086 0.023 CHEMBL734 | ||
| 0.15 | 0.007 | 0.273 | Phosphodiesterase 4C inhibitor | 0.273 0.004 CHEMBL734 | CHEMBL734 | |
| 0.174 | 0.032 | 0.227 | Adenylate cyclase inhibitor | 0.227 0.022 CHEMBL734 | CHEMBL734 | |
| 0.211 | 0.069 | 0.211 | Anesthetic general | 0.165 0.099 CHEMBL734 | ||
| 0.152 | 0.012 | 0.152 | Ribonucleotide reductase inhibitor | 0.086 0.024 CHEMBL734 | ||
| 0.153 | 0.014 | 0.153 | Keratolytic | 0.093 0.036 CHEMBL734 | ||
| 0.147 | 0.008 | 0.147 | NMDA receptor agonist | 0.115 0.015 CHEMBL734 | ||
| 0.141 | 0.004 | 0.141 | Aconitate hydratase inhibitor | 0.063 0.023 CHEMBL734 | ||
| 0.175 | 0.039 | 0.175 | Monophenol monooxygenase inhibitor | 0.136 0.053 CHEMBL734 | ||
| 0.128 | 0.004 | 0.128 | Glutamate (mGluR4) antagonist | 0.098 0.005 CHEMBL734 | ||
| 0.127 | 0.007 | 0.127 | NMDA receptor glycine site agonist | 0.115 0.01 CHEMBL734 | ||
| 0.123 | 0.003 | 0.143 | Glucose-6-phosphate isomerase inhibitor | 0.143 0.003 CHEMBL734 | CHEMBL734 | |
| 0.122 | 0.005 | 0.122 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.11 0.009 CHEMBL734 | ||
| 0.177 | 0.061 | 0.19 | ATPase inhibitor | 0.19 0.047 CHEMBL734 | CHEMBL734 | |
| 0.195 | 0.082 | 0.27 | DNA methylase inhibitor | 0.27 0.038 CHEMBL734 | CHEMBL734 | |
| 0.131 | 0.023 | 0.131 | NADH dehydrogenase inhibitor | 0.129 0.024 CHEMBL734 | ||
| 0.15 | 0.043 | 0.158 | Ca2+-transporting ATPase inhibitor | 0.158 0.026 CHEMBL734 | CHEMBL734 | |
| 0.12 | 0.014 | 0.124 | Biliverdin reductase inhibitor | 0.124 0.013 CHEMBL734 | CHEMBL734 | |
| 0.189 | 0.083 | 0.208 | 5 Hydroxytryptamine 3E antagonist | 0.208 0.051 CHEMBL734 | CHEMBL734 | |
| 0.104 | 0.003 | 0.119 | Peptide deformylase inhibitor | 0.119 0.003 CHEMBL734 | CHEMBL734 | |
| 0.209 | 0.108 | 0.209 | DNA damaging | 0.17 0.145 CHEMBL734 | ||
| 0.2 | 0.1 | 0.2 | RNA-directed DNA polymerase inhibitor | 0.186 0.122 CHEMBL734 | ||
| 0.103 | 0.004 | 0.145 | Immunoglobulin Fc receptor antagonist | 0.145 0.003 CHEMBL734 | CHEMBL734 | |
| 0.132 | 0.033 | 0.189 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.189 0.018 CHEMBL734 | CHEMBL734 | |
| 0.113 | 0.014 | 0.113 | Antimetabolite | 0.041 0.039 CHEMBL734 | ||
| 0.143 | 0.045 | 0.173 | Interleukin 1b antagonist | 0.173 0.027 CHEMBL734 | CHEMBL734 | |
| 0.127 | 0.031 | 0.127 | Catalase inhibitor | 0.097 0.039 CHEMBL734 | ||
| 0.129 | 0.033 | 0.13 | GABA C receptor rho-1 antagonist | 0.13 0.033 CHEMBL734 | CHEMBL734 | |
| 0.099 | 0.005 | 0.099 | Glutamate (mGluR group III) antagonist | 0.072 0.009 CHEMBL734 | ||
| 0.118 | 0.025 | 0.175 | Metalloproteinase-9 inhibitor | 0.175 0.011 CHEMBL734 | CHEMBL734 | |
| 0.107 | 0.015 | 0.107 | Ornithine carbamoyltransferase inhibitor | 0.066 0.028 CHEMBL734 | ||
| 0.096 | 0.005 | 0.226 | Aggrecanase 1 inhibitor | 0.226 0.003 CHEMBL734 | CHEMBL734 | |
| 0.111 | 0.019 | 0.111 | Amidase inhibitor | |||
| 0.174 | 0.083 | 0.289 | DNA methyltransferase I inhibitor | 0.289 0.03 CHEMBL734 | CHEMBL734 | |
| 0.134 | 0.045 | 0.134 | 5 Hydroxytryptamine 3A agonist | |||
| 0.121 | 0.035 | 0.121 | Electrolyte absorption antagonist | 0.105 0.051 CHEMBL734 | ||
| 0.191 | 0.105 | 0.212 | Nitric-oxide synthase stimulant | 0.212 0.071 CHEMBL734 | CHEMBL734 | |
| 0.12 | 0.035 | 0.12 | MAP kinase kinase 1 inhibitor | 0.119 0.036 CHEMBL734 | ||
| 0.116 | 0.031 | 0.175 | Metalloproteinase-2 inhibitor | 0.175 0.013 CHEMBL734 | CHEMBL734 | |
| 0.089 | 0.005 | 0.105 | Adenylate cyclase 1 inhibitor | 0.105 0.004 CHEMBL734 | CHEMBL734 | |
| 0.102 | 0.019 | 0.102 | Argininosuccinate synthase inhibitor | 0.081 0.025 CHEMBL734 | ||
| 0.104 | 0.021 | 0.145 | Neutrophil collagenase inhibitor | 0.145 0.013 CHEMBL734 | CHEMBL734 | |
| 0.091 | 0.009 | 0.091 | Kinesin-like protein 1 inhibitor | |||
| 0.091 | 0.009 | 0.091 | Kinesin antagonist | |||
| 0.087 | 0.006 | 0.087 | Ryanodine receptor antagonist | 0.083 0.007 CHEMBL734 | ||
| 0.092 | 0.011 | 0.11 | Potassium channel intermediate-conductance Ca-activated blocker | 0.11 0.007 CHEMBL734 | CHEMBL734 | |
| 0.201 | 0.121 | 0.201 | 5 Hydroxytryptamine release stimulant | 0.201 0.12 CHEMBL734 | ||
| 0.089 | 0.009 | 0.19 | Histone deacetylase class I inhibitor | 0.19 0.005 CHEMBL734 | CHEMBL734 | |
| 0.109 | 0.032 | 0.162 | Porphobilinogen synthase inhibitor | 0.162 0.018 CHEMBL734 | CHEMBL734 | |
| 0.176 | 0.099 | 0.224 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.224 0.056 CHEMBL734 | CHEMBL734 | |
| 0.157 | 0.082 | 0.157 | Growth hormone agonist | 0.144 0.092 CHEMBL734 | ||
| 0.092 | 0.018 | 0.129 | Acyl-CoA dehydrogenase inhibitor | 0.129 0.011 CHEMBL734 | CHEMBL734 | |
| 0.079 | 0.006 | 0.079 | Arginase inhibitor | 0.054 0.013 CHEMBL734 | ||
| 0.1 | 0.027 | 0.1 | Carbonic anhydrase V inhibitor | 0.075 0.039 CHEMBL734 | ||
| 0.185 | 0.113 | 0.207 | Aldehyde oxidase inhibitor | 0.207 0.101 CHEMBL734 | CHEMBL734 | |
| 0.119 | 0.046 | 0.119 | DOPA decarboxylase inhibitor | 0.115 0.051 CHEMBL734 | ||
| 0.146 | 0.074 | 0.146 | Hemostatic | |||
| 0.084 | 0.015 | 0.128 | Botulinum neurotoxin type A inhibitor | 0.128 0.005 CHEMBL734 | CHEMBL734 | |
| 0.098 | 0.029 | 0.098 | GABA aminotransferase inhibitor | 0.078 0.05 CHEMBL734 | ||
| 0.08 | 0.011 | 0.104 | Dihydroorotate oxidase inhibitor | 0.104 0.005 CHEMBL734 | CHEMBL734 | |
| 0.115 | 0.048 | 0.225 | Carbonic anhydrase III inhibitor | 0.225 0.012 CHEMBL734 | CHEMBL734 | |
| 0.084 | 0.02 | 0.084 | Glutamate (mGluR6) antagonist | 0.077 0.027 CHEMBL734 | ||
| 0.233 | 0.168 | 0.271 | Calcium channel activator | 0.271 0.122 CHEMBL734 | CHEMBL734 | |
| 0.085 | 0.021 | 0.166 | Collagenase 3 inhibitor | 0.166 0.007 CHEMBL734 | CHEMBL734 | |
| 0.111 | 0.048 | 0.132 | Creatine kinase inhibitor | 0.132 0.033 CHEMBL734 | CHEMBL734 | |
| 0.097 | 0.034 | 0.097 | Na+ K+ transporting ATPase inhibitor | 0.086 0.045 CHEMBL734 | ||
| 0.075 | 0.013 | 0.079 | Carbonic anhydrase IV inhibitor | 0.079 0.011 CHEMBL734 | CHEMBL734 | |
| 0.091 | 0.029 | 0.091 | Carbonic anhydrase VA inhibitor | 0.075 0.041 CHEMBL734 | ||
| 0.125 | 0.063 | 0.125 | Alkylator | 0.098 0.091 CHEMBL734 | ||
| 0.131 | 0.071 | 0.131 | Sphingosine 1-phosphate receptor 2 antagonist | 0.121 0.095 CHEMBL734 | ||
| 0.092 | 0.033 | 0.106 | Aminopeptidase I inhibitor | 0.106 0.025 CHEMBL734 | CHEMBL734 | |
| 0.102 | 0.042 | 0.115 | Phosphodiesterase I inhibitor | 0.115 0.03 CHEMBL734 | CHEMBL734 | |
| 0.164 | 0.105 | 0.197 | Psychostimulant | 0.197 0.082 CHEMBL734 | CHEMBL734 | |
| 0.097 | 0.039 | 0.121 | Myeloperoxidase inhibitor | 0.121 0.019 CHEMBL734 | CHEMBL734 | |
| 0.136 | 0.078 | 0.166 | Mannose-6-phosphate isomerase inhibitor | 0.166 0.052 CHEMBL734 | CHEMBL734 | |
| 0.089 | 0.032 | 0.152 | Matrix metalloproteinase inhibitor | 0.152 0.013 CHEMBL734 | CHEMBL734 | |
| 0.065 | 0.008 | 0.085 | Membrane dipeptidase inhibitor | 0.085 0.005 CHEMBL734 | CHEMBL734 | |
| 0.064 | 0.008 | 0.065 | Vascular adhesion protein 1 inhibitor | 0.065 0.007 CHEMBL734 | CHEMBL734 | |
| 0.077 | 0.022 | 0.144 | Phosphodiesterase 1C inhibitor | 0.144 0.005 CHEMBL734 | CHEMBL734 | |
| 0.077 | 0.022 | 0.077 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.076 0.022 CHEMBL734 | ||
| 0.086 | 0.032 | 0.09 | Glycine receptor agonist | 0.09 0.028 CHEMBL734 | CHEMBL734 | |
| 0.059 | 0.007 | 0.059 | Kainate receptor agonist | 0.052 0.012 CHEMBL734 | ||
| 0.065 | 0.014 | 0.065 | Thymidylate synthase inhibitor | |||
| 0.054 | 0.003 | 0.063 | Purinergic P2Y15 antagonist | 0.063 0.002 CHEMBL734 | CHEMBL734 | |
| 0.143 | 0.096 | 0.168 | Arachidonic acid antagonist | 0.168 0.067 CHEMBL734 | CHEMBL734 | |
| 0.089 | 0.042 | 0.089 | Somatostatin 1 agonist | |||
| 0.062 | 0.015 | 0.183 | Histone deacetylase 8 inhibitor | 0.183 0.005 CHEMBL734 | CHEMBL734 | |
| 0.123 | 0.077 | 0.153 | Antibacterial (Helicobacter pylori) | 0.153 0.044 CHEMBL734 | CHEMBL734 | |
| 0.082 | 0.038 | 0.093 | GABA B receptor agonist | 0.093 0.022 CHEMBL734 | CHEMBL734 | |
| 0.11 | 0.067 | 0.11 | Cystathionine beta-synthase inhibitor | 0.093 0.085 CHEMBL734 | ||
| 0.069 | 0.026 | 0.113 | Matrix metalloproteinase 1 inhibitor | 0.113 0.01 CHEMBL734 | CHEMBL734 | |
| 0.059 | 0.017 | 0.059 | Kainate receptor antagonist | |||
| 0.258 | 0.217 | 0.35 | 5 Hydroxytryptamine release inhibitor | 0.35 0.115 CHEMBL734 | CHEMBL734 | |
| 0.063 | 0.022 | 0.094 | Metalloproteinase-3 inhibitor | 0.094 0.012 CHEMBL734 | CHEMBL734 | |
| 0.088 | 0.048 | 0.088 | D-Ala-D-Ala ligase inhibitor | 0.082 0.062 CHEMBL734 | ||
| 0.044 | 0.005 | 0.123 | Aggrecanase 2 inhibitor | 0.123 0.003 CHEMBL734 | CHEMBL734 | |
| 0.052 | 0.013 | 0.052 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.051 0.014 CHEMBL734 | ||
| 0.135 | 0.097 | 0.168 | GABA C receptor rho-2 antagonist | 0.168 0.052 CHEMBL734 | CHEMBL734 | |
| 0.057 | 0.019 | 0.057 | Dopamine beta hydroxylase inhibitor | 0.053 0.024 CHEMBL734 | ||
| 0.085 | 0.049 | 0.118 | Glycine receptor antagonist | 0.118 0.019 CHEMBL734 | CHEMBL734 | |
| 0.137 | 0.102 | 0.158 | Melanin inhibitor | 0.158 0.072 CHEMBL734 | CHEMBL734 | |
| 0.048 | 0.013 | 0.048 | Glutamate (mGluR8) agonist | 0.045 0.016 CHEMBL734 | ||
| 0.052 | 0.02 | 0.052 | Histamine H2 receptor agonist | 0.04 0.034 CHEMBL734 | ||
| 0.047 | 0.015 | 0.051 | Fumarate hydratase inhibitor | 0.051 0.013 CHEMBL734 | CHEMBL734 | |
| 0.067 | 0.035 | 0.067 | Purinergic P2X1 antagonist | 0.055 0.053 CHEMBL734 | ||
| 0.049 | 0.019 | 0.176 | Histone deacetylase 7 inhibitor | 0.176 0.004 CHEMBL734 | CHEMBL734 | |
| 0.053 | 0.023 | 0.054 | Cytokine production stimulant | 0.054 0.021 CHEMBL734 | CHEMBL734 | |
| 0.039 | 0.01 | 0.039 | Glutamate (mGluR3) agonist | 0.035 0.016 CHEMBL734 | ||
| 0.047 | 0.018 | 0.17 | Histone deacetylase 9 inhibitor | 0.17 0.004 CHEMBL734 | CHEMBL734 | |
| 0.06 | 0.032 | 0.109 | Matrix metalloproteinase (membrane-type) inhibitor | 0.109 0.012 CHEMBL734 | CHEMBL734 | |
| 0.091 | 0.065 | 0.091 | Prolactin inhibitor | 0.084 0.075 CHEMBL734 | ||
| 0.034 | 0.009 | 0.034 | Thymidine phosphorylase inhibitor | |||
| 0.052 | 0.028 | 0.052 | Adenosine deaminase inhibitor | 0.051 0.029 CHEMBL734 | ||
| 0.066 | 0.042 | 0.066 | Carbonic anhydrase inhibitor | 0.063 0.044 CHEMBL734 | ||
| 0.094 | 0.072 | 0.11 | Anabolic | 0.11 0.05 CHEMBL734 | CHEMBL734 | |
| 0.089 | 0.067 | 0.089 | HIV-1 integrase (Overall Integration) inhibitor | |||
| 0.085 | 0.063 | 0.096 | Granulocyte macrophage colony stimulating factor agonist | 0.096 0.041 CHEMBL734 | CHEMBL734 | |
| 0.073 | 0.052 | 0.187 | Phosphodiesterase 4D inhibitor | 0.187 0.012 CHEMBL734 | CHEMBL734 | |
| 0.025 | 0.003 | 0.122 | 1-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor | 0.122 0.001 CHEMBL734 | CHEMBL734 | |
| 0.099 | 0.078 | 0.112 | Mucolytic | 0.112 0.063 CHEMBL734 | CHEMBL734 | |
| 0.163 | 0.144 | 0.193 | Immunostimulant | 0.193 0.124 CHEMBL734 | CHEMBL734 | |
| 0.107 | 0.087 | 0.107 | MAP kinase kinase inhibitor | 0.104 0.091 CHEMBL734 | ||
| 0.057 | 0.038 | 0.057 | Carbonic anhydrase II inhibitor | 0.057 0.038 CHEMBL734 | ||
| 0.054 | 0.035 | 0.061 | Alpha-mannosidase inhibitor | 0.061 0.026 CHEMBL734 | CHEMBL734 | |
| 0.036 | 0.018 | 0.036 | Carboxypeptidase B inhibitor | |||
| 0.028 | 0.01 | 0.028 | Complement factor 1s inhibitor | |||
| 0.102 | 0.084 | 0.179 | CDK3/cyclin E inhibitor | 0.179 0.012 CHEMBL734 | CHEMBL734 | |
| 0.098 | 0.08 | 0.098 | Nav1.4 sodium channel blocker | |||
| 0.025 | 0.008 | 0.034 | Aminopeptidase A inhibitor | 0.034 0.005 CHEMBL734 | CHEMBL734 | |
| 0.128 | 0.112 | 0.128 | MAP kinase 3 inhibitor | 0.126 0.118 CHEMBL734 | ||
| 0.041 | 0.026 | 0.041 | Dopamine D5 agonist | 0.036 0.033 CHEMBL734 | ||
| 0.059 | 0.044 | 0.121 | Phosphodiesterase 1B inhibitor | 0.121 0.01 CHEMBL734 | CHEMBL734 | |
| 0.026 | 0.011 | 0.026 | Glutamate (mGluR1a) agonist | 0.022 0.016 CHEMBL734 | ||
| 0.034 | 0.02 | 0.039 | Dipeptidyl peptidase II inhibitor | 0.039 0.015 CHEMBL734 | CHEMBL734 | |
| 0.036 | 0.023 | 0.036 | Gonadotropin-releasing hormone receptor antagonist | |||
| 0.101 | 0.089 | 0.101 | Microtubule formation inhibitor | 0.099 0.093 CHEMBL734 | ||
| 0.053 | 0.041 | 0.053 | Thromboxane synthase inhibitor | |||
| 0.026 | 0.015 | 0.026 | Glutamate (mGluR1) agonist | 0.025 0.016 CHEMBL734 | ||
| 0.041 | 0.03 | 0.041 | Oxytocin agonist | |||
| 0.047 | 0.038 | 0.047 | Bombesin 2 receptor antagonist | |||
| 0.055 | 0.047 | 0.055 | Carbonic anhydrase stimulant | |||
| 0.14 | 0.132 | 0.213 | Death-associated protein kinase 2 inhibitor | 0.213 0.026 CHEMBL734 | CHEMBL734 | |
| 0.03 | 0.025 | 0.041 | Methionyl aminopeptidase 1 inhibitor | 0.041 0.011 CHEMBL734 | CHEMBL734 | |
| 0.017 | 0.012 | 0.029 | Carbonic anhydrase X inhibitor | 0.029 0.004 CHEMBL734 | CHEMBL734 | |
| 0.017 | 0.012 | 0.029 | Carbonic anhydrase VIII inhibitor | 0.029 0.004 CHEMBL734 | CHEMBL734 | |
| 0.063 | 0.058 | 0.063 | Glutamate (mGluR7) antagonist | |||
| 0.025 | 0.021 | 0.025 | Lysine carboxypeptidase inhibitor | |||
| 0.064 | 0.06 | 0.068 | Exportin-1 inhibitor | 0.068 0.047 CHEMBL734 | CHEMBL734 | |
| 0.109 | 0.105 | 0.109 | Protein kinase stimulant | |||
| 0.041 | 0.037 | 0.041 | Fructose-1,6-bisphosphatase inhibitor | |||
| 0.041 | 0.038 | 0.045 | Mannosidase inhibitor | 0.045 0.032 CHEMBL734 | CHEMBL734 | |
| 0.016 | 0.013 | 0.016 | Telomerase stimulant | 0.016 0.014 CHEMBL734 | ||
| 0.032 | 0.031 | 0.047 | Inosine monophosphate dehydrogenase inhibitor | 0.047 0.017 CHEMBL734 | CHEMBL734 | |
| 0.074 | 0.073 | 0.097 | Glutathione S-transferase inhibitor | 0.097 0.04 CHEMBL734 | CHEMBL734 | |
| 0.102 | 0.103 | 0.127 | Cathepsin H inhibitor | 0.127 0.067 CHEMBL734 | CHEMBL734 | |
| 0.016 | 0.019 | 0.022 | Inosine monophosphate dehydrogenase 1 inhibitor | 0.022 0.012 CHEMBL734 | CHEMBL734 | |
| 0.032 | 0.035 | 0.043 | Diamine oxidase inhibitor | 0.043 0.02 CHEMBL734 | CHEMBL734 | |
| 0.016 | 0.02 | 0.019 | Methylmalonyl-CoA mutase inhibitor | 0.019 0.01 CHEMBL734 | CHEMBL734 | |
| 0.004 | 0.008 | 0.006 | Bone morphogenic protein 1 inhibitor | 0.006 0.004 CHEMBL734 | CHEMBL734 | |
| 0.047 | 0.052 | 0.054 | Lysine-specific demethylase 1A inhibitor | 0.054 0.037 CHEMBL734 | CHEMBL734 | |
| 0.101 | 0.106 | 0.121 | Transcription factor STAT6 inhibitor | 0.121 0.059 CHEMBL734 | CHEMBL734 | |
| 0.015 | 0.02 | 0.025 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.025 0.01 CHEMBL734 | CHEMBL734 | |
| 0.02 | 0.025 | 0.021 | Isoleucine-tRNA ligase inhibitor | 0.021 0.019 CHEMBL734 | CHEMBL734 | |
| 0.023 | 0.031 | 0.032 | CDK4/cyclin D3 inhibitor | 0.032 0.016 CHEMBL734 | CHEMBL734 | |
| 0.042 | 0.053 | 0.057 | Carbonic anhydrase VB inhibitor | 0.057 0.038 CHEMBL734 | CHEMBL734 | |
| 0.017 | 0.031 | 0.024 | Neuraminidase (Influenza B) inhibitor | 0.024 0.009 CHEMBL734 | CHEMBL734 | |
| 0.008 | 0.023 | 0.012 | Lysophosphatidic acid receptor 3 agonist | 0.012 0.011 CHEMBL734 | CHEMBL734 | |
| 0.065 | 0.082 | 0.076 | Carbonic anhydrase VI inhibitor | 0.076 0.063 CHEMBL734 | CHEMBL734 | |
| 0.167 | 0.185 | 0.201 | Transcription factor STAT3 inhibitor | 0.201 0.132 CHEMBL734 | CHEMBL734 | |
| 0.092 | 0.113 | 0.103 | Aldehyde dehydrogenase inhibitor | 0.103 0.093 CHEMBL734 | CHEMBL734 | |
| 0.037 | 0.058 | 0.057 | Carbonic anhydrase I inhibitor | 0.057 0.038 CHEMBL734 | CHEMBL734 | |
| 0.188 | 0.209 | 0.4 | Immunosuppressant | 0.4 0.063 CHEMBL734 | CHEMBL734 | |
| 0.007 | 0.029 | 0.012 | Carbonic anhydrase XI inhibitor | 0.012 0.01 CHEMBL734 | CHEMBL734 | |
| 0.018 | 0.042 | 0.026 | Lysophosphatidic acid receptor 1 agonist | 0.026 0.016 CHEMBL734 | CHEMBL734 | |
| 0.011 | 0.037 | 0.015 | Vitamin D receptor agonist | 0.015 0.014 CHEMBL734 | CHEMBL734 | |
| 0.072 | 0.1 | 0.089 | Estrogen-related receptor beta agonist | 0.089 0.042 CHEMBL734 | CHEMBL734 | |
| 0.007 | 0.038 | 0.012 | Human herpes virus 5 capsid protein P40 inhibitor | 0.012 0.011 CHEMBL734 | CHEMBL734 | |
| 0.115 | 0.148 | 0.136 | Interferon gamma antagonist | 0.136 0.099 CHEMBL734 | CHEMBL734 | |
| 0.128 | 0.166 | 0.143 | Neurotensin receptor agonist | 0.143 0.12 CHEMBL734 | CHEMBL734 | |
| 0.102 | 0.14 | 0.115 | Vanilloid 1 agonist | 0.115 0.102 CHEMBL734 | CHEMBL734 | |
| 0.124 | 0.163 | 0.207 | Non-steroidal antiinflammatory agent | 0.207 0.065 CHEMBL734 | CHEMBL734 | |
| 0.024 | 0.064 | 0.032 | Retinoid X alpha receptor antagonist | 0.032 0.029 CHEMBL734 | CHEMBL734 | |
| 0.085 | 0.125 | 0.114 | Photosensitizer | 0.114 0.065 CHEMBL734 | CHEMBL734 | |
| 0.088 | 0.129 | 0.109 | Toll-Like receptor 2 antagonist | 0.109 0.091 CHEMBL734 | CHEMBL734 | |
| 0.076 | 0.117 | 0.096 | Carbonic anhydrase XV inhibitor | 0.096 0.073 CHEMBL734 | CHEMBL734 | |
| 0.045 | 0.086 | 0.067 | Phosphodiesterase 4B inhibitor | 0.067 0.047 CHEMBL734 | CHEMBL734 | |
| 0.048 | 0.089 | 0.06 | Protease 3C (Human rhinovirus) inhibitor | 0.06 0.052 CHEMBL734 | CHEMBL734 | |
| 0.134 | 0.175 | 0.173 | Histone acetyltransferase inhibitor | 0.173 0.11 CHEMBL734 | CHEMBL734 | |
| 0.026 | 0.072 | 0.035 | Retinoid X receptor antagonist | 0.035 0.033 CHEMBL734 | CHEMBL734 | |
| 0.161 | 0.21 | 0.186 | Transcription factor STAT inhibitor | 0.186 0.159 CHEMBL734 | CHEMBL734 | |
| 0.021 | 0.079 | 0.056 | Endothelin-converting enzyme inhibitor | 0.056 0.027 CHEMBL734 | CHEMBL734 | |
| 0.127 | 0.188 | 0.27 | Interleukin agonist | 0.27 0.065 CHEMBL734 | CHEMBL734 | |
| 0.006 | 0.068 | 0.015 | Melatonin 2 antagonist | 0.015 0.005 CHEMBL734 | CHEMBL734 | |
| 0.147 | 0.212 | 0.222 | 12-Lipoxygenase inhibitor | 0.222 0.129 CHEMBL734 | CHEMBL734 | |
| 0.028 | 0.099 | 0.05 | Lysophosphatidic acid 3 receptor antagonist | 0.05 0.036 CHEMBL734 | CHEMBL734 | |
| 0.098 | 0.177 | 0.153 | Heat shock protein 90 alpha antagonist | 0.153 0.083 CHEMBL734 | CHEMBL734 | |
| 0.071 | 0.154 | 0.094 | Glutamate (mGluR7) agonist | 0.094 0.074 CHEMBL734 | CHEMBL734 | |
| 0.054 | 0.138 | 0.08 | Vanilloid 4 agonist | 0.08 0.041 CHEMBL734 | CHEMBL734 | |
| 0.123 | 0.21 | 0.162 | Cyclic AMP phosphodiesterase inhibitor | 0.162 0.133 CHEMBL734 | CHEMBL734 | |
| 0.107 | 0.205 | 0.139 | Lipocortins synthesis antagonist | 0.139 0.123 CHEMBL734 | CHEMBL734 | |
| 0.158 | 0.268 | 0.24 | Histamine release inhibitor | 0.24 0.163 CHEMBL734 | CHEMBL734 | |
| 0.058 | 0.178 | 0.097 | Proteasome inhibitor | 0.097 0.091 CHEMBL734 | CHEMBL734 | |
| 0.108 | 0.243 | 0.174 | Calpain inhibitor | 0.174 0.142 CHEMBL734 | CHEMBL734 | |
| 0.053 | 0.189 | 0.08 | Bromodomain-containing protein 2 inhibitor | 0.08 0.078 CHEMBL734 | CHEMBL734 | |
| 0.077 | 0.224 | 0.119 | Heat shock protein 90 antagonist | 0.119 0.116 CHEMBL734 | CHEMBL734 | |
| 0.061 | 0.215 | 0.121 | Cyclooxygenase 3 inhibitor | 0.121 0.076 CHEMBL734 | CHEMBL734 | |
| 0.039 | 0.203 | 0.092 | Falcipain 3 inhibitor | 0.092 0.079 CHEMBL734 | CHEMBL734 | |
| 0.079 | 0.244 | 0.135 | Interleukin antagonist | 0.135 0.13 CHEMBL734 | CHEMBL734 | |
| 0.015 | 0.195 | 0.111 | Neuraminidase inhibitor | 0.111 0.012 CHEMBL734 | CHEMBL734 | |
| 0.084 | 0.272 | 0.134 | 3C-like protease (Human coronavirus) inhibitor | 0.134 0.133 CHEMBL734 | CHEMBL734 | |
| 0.042 | 0.235 | 0.145 | Chelator | 0.145 0.037 CHEMBL734 | CHEMBL734 | |
| 0.012 | 0.236 | 0.063 | Phosphodiesterase 4A inhibitor | 0.063 0.028 CHEMBL734 | CHEMBL734 | |
| 0.112 | 0.347 | 0.215 | Peptidyltransferase inhibitor | 0.215 0.082 CHEMBL734 | CHEMBL734 | |
| 0.018 | 0.272 | 0.077 | Phosphodiesterase 5A inhibitor | 0.077 0.042 CHEMBL734 | CHEMBL734 | |
| 0.015 | 0.306 | 0.072 | Phosphodiesterase V inhibitor | 0.072 0.05 CHEMBL734 | CHEMBL734 | |
| 0.014 | 0.347 | 0.08 | Neuraminidase (influenza) inhibitor | 0.08 0.025 CHEMBL734 | CHEMBL734 | |
| 0.011 | 0.368 | 0.044 | Neuraminidase (Influenza A) inhibitor | 0.044 0.034 CHEMBL734 | CHEMBL734 | |
| 0.004 | 0.472 | 0.945 | Melatonin 1 antagonist | 0.945 0.001 CHEMBL734 | CHEMBL734 | |
| 0.004 | 0.487 | 0.948 | Melatonin antagonist | 0.948 0.001 CHEMBL734 | CHEMBL734 | |
| 0.06 | 0.74 | 0.233 | Interleukin 2 agonist | 0.233 0.139 CHEMBL734 | CHEMBL734 | |
| 0.026 | 0.764 | 0.364 | Apoptosis agonist | 0.364 0.131 CHEMBL734 | CHEMBL734 | |
| 0.003 | 0.832 | 0.643 | Melatonin agonist | 0.643 0.002 CHEMBL734 | CHEMBL734 | |
| 0.033 | 0.934 | 0.113 | Papain-like protease (SARS coronavirus) inhibitor | 0.113 0.103 CHEMBL734 | CHEMBL734 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |