| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.859 | 0.002 | 0.859 | Heat shock protein 90 antagonist | 0.574 0.003 CHEMBL226396 0.227 0.028 CHEMBL4525761 0.14 0.085 CHEMBL3526318 0.851 0.002 CHEMBL375462 0.833 0.002 CHEMBL3527205 0.704 0.002 CHEMBL3527204 0.627 0.003 CHEMBL3527203 0.12 0.113 CHEMBL3527549 0.786 0.002 CHEMBL3526210 0.487 0.004 CHEMBL3526912 0.209 0.034 CHEMBL3527548 | ||
| 0.813 | 0.002 | 0.817 | Heat shock protein 90 alpha antagonist | 0.397 0.005 CHEMBL226396 0.25 0.027 CHEMBL4525761 0.817 0.002 CHEMBL375462 0.621 0.003 CHEMBL3527205 0.646 0.003 CHEMBL3527204 0.6 0.003 CHEMBL3527203 0.593 0.003 CHEMBL3526210 0.368 0.007 CHEMBL3526912 | CHEMBL375462 | |
| 0.368 | 0.003 | 0.399 | H+/K+-transporting ATPase inhibitor | 0.399 0.003 CHEMBL4525761 0.08 0.013 CHEMBL3526318 0.312 0.004 CHEMBL375462 0.311 0.004 CHEMBL3527205 0.116 0.007 CHEMBL3527204 0.335 0.004 CHEMBL3527203 0.066 0.02 CHEMBL3527549 0.282 0.004 CHEMBL3526210 0.05 0.038 CHEMBL3526912 0.048 0.04 CHEMBL3527548 | CHEMBL4525761 | |
| 0.384 | 0.02 | 0.533 | RNA-directed DNA polymerase inhibitor | 0.458 0.013 CHEMBL226396 0.296 0.032 CHEMBL4525761 0.391 0.019 CHEMBL375462 0.252 0.048 CHEMBL3527205 0.433 0.015 CHEMBL3527204 0.533 0.009 CHEMBL3527203 0.237 0.058 CHEMBL3526210 0.318 0.028 CHEMBL3526912 0.48 0.012 CHEMBL3527548 | CHEMBL3527203 | |
| 0.379 | 0.02 | 0.729 | Death-associated protein kinase 3 inhibitor | 0.729 0.003 CHEMBL226396 0.402 0.017 CHEMBL375462 0.345 0.027 CHEMBL3527205 0.311 0.035 CHEMBL3527204 0.387 0.019 CHEMBL3526210 | CHEMBL226396 | |
| 0.302 | 0.002 | 0.334 | Heat shock protein 90 beta antagonist | 0.215 0.003 CHEMBL226396 0.072 0.027 CHEMBL4525761 0.334 0.002 CHEMBL375462 0.226 0.003 CHEMBL3527205 0.198 0.004 CHEMBL3527204 0.22 0.003 CHEMBL3527203 0.218 0.003 CHEMBL3526210 | CHEMBL375462 | |
| 0.343 | 0.056 | 0.343 | Nootropic | 0.197 0.162 CHEMBL226396 0.276 0.087 CHEMBL375462 0.207 0.149 CHEMBL3527204 | ||
| 0.245 | 0.02 | 0.322 | Interleukin 1 antagonist | 0.227 0.024 CHEMBL375462 0.201 0.032 CHEMBL3527205 0.215 0.027 CHEMBL3527204 0.322 0.009 CHEMBL3527203 0.191 0.037 CHEMBL3526210 0.146 0.06 CHEMBL3526912 0.214 0.027 CHEMBL3527548 | CHEMBL3527203 | |
| 0.26 | 0.042 | 0.737 | CDC-like kinase 2 inhibitor | 0.737 0.004 CHEMBL226396 0.255 0.044 CHEMBL375462 0.157 0.088 CHEMBL3527205 0.191 0.071 CHEMBL3527204 0.175 0.08 CHEMBL3526210 | CHEMBL226396 | |
| 0.272 | 0.054 | 0.524 | DNA synthesis inhibitor | 0.524 0.012 CHEMBL226396 0.273 0.054 CHEMBL4525761 0.329 0.035 CHEMBL375462 0.266 0.057 CHEMBL3527205 0.362 0.028 CHEMBL3527204 0.265 0.058 CHEMBL3527203 0.181 0.153 CHEMBL3527549 0.289 0.047 CHEMBL3526210 0.449 0.017 CHEMBL3526912 0.404 0.021 CHEMBL3527548 | CHEMBL226396 | |
| 0.266 | 0.061 | 0.753 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.753 0.004 CHEMBL226396 0.303 0.05 CHEMBL375462 0.219 0.082 CHEMBL3527204 0.168 0.116 CHEMBL3527203 0.149 0.132 CHEMBL3526210 | CHEMBL226396 | |
| 0.256 | 0.053 | 0.717 | Clk dual-specificity kinase inhibitor | 0.717 0.004 CHEMBL226396 0.233 0.062 CHEMBL375462 0.176 0.094 CHEMBL3527204 | CHEMBL226396 | |
| 0.264 | 0.066 | 0.765 | Dyrk kinase inhibitor | 0.765 0.004 CHEMBL226396 0.297 0.054 CHEMBL375462 0.217 0.089 CHEMBL3527204 0.154 0.132 CHEMBL3527203 0.146 0.14 CHEMBL3526210 | CHEMBL226396 | |
| 0.276 | 0.083 | 0.516 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.516 0.005 CHEMBL226396 0.304 0.061 CHEMBL375462 0.227 0.128 CHEMBL3527205 0.254 0.103 CHEMBL3527204 0.263 0.095 CHEMBL3526210 | CHEMBL226396 | |
| 0.198 | 0.034 | 0.5 | Cyclin-dependent kinase 7 inhibitor | 0.5 0.004 CHEMBL226396 0.211 0.03 CHEMBL375462 0.158 0.054 CHEMBL3527205 0.159 0.054 CHEMBL3527204 0.185 0.04 CHEMBL3526210 | CHEMBL226396 | |
| 0.217 | 0.059 | 0.638 | CDC-like kinase 4 inhibitor | 0.638 0.004 CHEMBL226396 0.196 0.069 CHEMBL375462 0.15 0.101 CHEMBL3527204 | CHEMBL226396 | |
| 0.203 | 0.051 | 0.235 | Tumour necrosis factor antagonist | 0.197 0.055 CHEMBL226396 0.235 0.035 CHEMBL4525761 0.227 0.039 CHEMBL3527205 0.166 0.081 CHEMBL3527204 0.149 0.102 CHEMBL3526210 | CHEMBL4525761 | |
| 0.19 | 0.055 | 0.477 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.477 0.005 CHEMBL226396 0.2 0.05 CHEMBL375462 0.203 0.05 CHEMBL3527205 0.124 0.098 CHEMBL3527204 0.232 0.041 CHEMBL3526210 | CHEMBL226396 | |
| 0.181 | 0.061 | 0.191 | MAP kinase kinase 5 inhibitor | 0.185 0.053 CHEMBL226396 0.172 0.081 CHEMBL375462 0.167 0.095 CHEMBL3527204 0.191 0.044 CHEMBL3527203 | CHEMBL3527203 | |
| 0.162 | 0.043 | 0.36 | DNA polymerase I inhibitor | 0.36 0.008 CHEMBL226396 0.116 0.071 CHEMBL3526318 0.193 0.03 CHEMBL375462 0.127 0.063 CHEMBL3527205 0.177 0.036 CHEMBL3527204 0.2 0.028 CHEMBL3527203 0.131 0.06 CHEMBL3527549 0.144 0.053 CHEMBL3526210 0.203 0.027 CHEMBL3526912 0.221 0.022 CHEMBL3527548 | CHEMBL226396 | |
| 0.156 | 0.043 | 0.225 | TRKB antagonist | 0.225 0.02 CHEMBL226396 0.135 0.058 CHEMBL375462 0.122 0.07 CHEMBL3527204 | CHEMBL226396 | |
| 0.126 | 0.015 | 0.184 | mTOR complex 2 inhibitor | 0.184 0.005 CHEMBL226396 0.087 0.052 CHEMBL4525761 0.123 0.016 CHEMBL375462 0.101 0.032 CHEMBL3527205 0.129 0.014 CHEMBL3527204 0.103 0.029 CHEMBL3527203 0.1 0.033 CHEMBL3526210 | CHEMBL226396 | |
| 0.147 | 0.044 | 0.242 | Death-associated protein kinase 1 inhibitor | 0.136 0.065 CHEMBL4525761 0.145 0.047 CHEMBL375462 0.133 0.073 CHEMBL3527204 0.242 0.004 CHEMBL3527203 0.157 0.03 CHEMBL3527548 | CHEMBL3527203 | |
| 0.125 | 0.023 | 0.271 | mTOR complex 1 inhibitor | 0.271 0.004 CHEMBL226396 0.124 0.024 CHEMBL375462 0.117 0.032 CHEMBL3527205 0.119 0.03 CHEMBL3527204 0.12 0.029 CHEMBL3526210 | CHEMBL226396 | |
| 0.141 | 0.045 | 0.575 | Cyclin-dependent kinase 1 inhibitor | 0.575 0.004 CHEMBL226396 0.161 0.037 CHEMBL375462 0.111 0.059 CHEMBL3527204 0.127 0.051 CHEMBL3527203 | CHEMBL226396 | |
| 0.094 | 0.004 | 0.127 | Protocollagen prolyl hydroxylase inhibitor | 0.039 0.008 CHEMBL4525761 0.104 0.004 CHEMBL3526318 0.127 0.004 CHEMBL375462 0.062 0.005 CHEMBL3527205 0.073 0.005 CHEMBL3527204 0.126 0.004 CHEMBL3527203 0.122 0.004 CHEMBL3527549 0.101 0.004 CHEMBL3526210 0.033 0.012 CHEMBL3526912 0.04 0.007 CHEMBL3527548 | CHEMBL375462 | |
| 0.113 | 0.024 | 0.132 | Purinergic P2X2 antagonist | 0.132 0.016 CHEMBL226396 0.074 0.043 CHEMBL4525761 0.109 0.025 CHEMBL375462 0.087 0.037 CHEMBL3527205 0.098 0.031 CHEMBL3527204 0.118 0.021 CHEMBL3527203 0.078 0.041 CHEMBL3526210 | CHEMBL226396 | |
| 0.224 | 0.137 | 0.683 | Immunomodulator | 0.445 0.033 CHEMBL226396 0.377 0.051 CHEMBL3526318 0.233 0.129 CHEMBL375462 0.659 0.007 CHEMBL3527205 0.218 0.144 CHEMBL3527204 0.29 0.088 CHEMBL3527203 0.384 0.049 CHEMBL3527549 0.683 0.006 CHEMBL3526210 0.433 0.035 CHEMBL3526912 0.479 0.026 CHEMBL3527548 | CHEMBL3526210 | |
| 0.115 | 0.03 | 0.184 | Phosphodiesterase I inhibitor | 0.167 0.014 CHEMBL226396 0.109 0.034 CHEMBL375462 0.088 0.062 CHEMBL3527205 0.116 0.03 CHEMBL3527204 0.184 0.012 CHEMBL3527203 0.088 0.062 CHEMBL3526210 | CHEMBL3527203 | |
| 0.108 | 0.023 | 0.28 | Adenosine A2a receptor antagonist | 0.28 0.006 CHEMBL226396 0.111 0.022 CHEMBL375462 0.106 0.024 CHEMBL3527204 0.127 0.019 CHEMBL3527203 | CHEMBL226396 | |
| 0.102 | 0.019 | 0.45 | Phosphatidylinositol 3-kinase delta inhibitor | 0.45 0.004 CHEMBL226396 0.104 0.019 CHEMBL375462 0.057 0.04 CHEMBL3527204 0.068 0.031 CHEMBL3527203 | CHEMBL226396 | |
| 0.083 | 0.003 | 0.09 | Egl nine homolog 2 inhibitor | 0.03 0.004 CHEMBL3526318 0.09 0.003 CHEMBL375462 0.073 0.003 CHEMBL3527205 0.07 0.003 CHEMBL3527204 0.08 0.003 CHEMBL3527203 0.038 0.004 CHEMBL3527549 0.085 0.003 CHEMBL3526210 0.019 0.005 CHEMBL3526912 0.019 0.005 CHEMBL3527548 | CHEMBL375462 | |
| 0.146 | 0.072 | 0.487 | Protein kinase (CK1) gamma 1 inhibitor | 0.487 0.005 CHEMBL226396 0.155 0.065 CHEMBL375462 0.126 0.091 CHEMBL3527205 0.147 0.071 CHEMBL3526210 | CHEMBL226396 | |
| 0.096 | 0.028 | 0.28 | Adenosine A2 receptor antagonist | 0.28 0.006 CHEMBL226396 0.098 0.028 CHEMBL375462 0.082 0.033 CHEMBL3527204 0.131 0.02 CHEMBL3527203 | CHEMBL226396 | |
| 0.084 | 0.021 | 0.193 | Interferon inducer | 0.085 0.02 CHEMBL226396 0.062 0.049 CHEMBL4525761 0.106 0.01 CHEMBL375462 0.132 0.006 CHEMBL3527205 0.113 0.009 CHEMBL3527204 0.138 0.005 CHEMBL3527203 0.151 0.005 CHEMBL3526210 0.128 0.006 CHEMBL3526912 0.193 0.004 CHEMBL3527548 | CHEMBL3527548 | |
| 0.095 | 0.033 | 0.261 | Interferon agonist | 0.098 0.03 CHEMBL226396 0.073 0.064 CHEMBL4525761 0.117 0.018 CHEMBL375462 0.16 0.009 CHEMBL3527205 0.13 0.014 CHEMBL3527204 0.175 0.008 CHEMBL3527203 0.188 0.007 CHEMBL3526210 0.157 0.009 CHEMBL3526912 0.261 0.004 CHEMBL3527548 | CHEMBL3527548 | |
| 0.118 | 0.059 | 0.415 | Cyclin-dependent kinase 5 inhibitor | 0.415 0.005 CHEMBL226396 0.136 0.048 CHEMBL375462 0.094 0.08 CHEMBL3527204 | CHEMBL226396 | |
| 0.138 | 0.079 | 0.329 | CDC-like kinase 1 inhibitor | 0.329 0.007 CHEMBL226396 0.118 0.097 CHEMBL375462 0.138 0.079 CHEMBL3527203 | CHEMBL226396 | |
| 0.109 | 0.05 | 0.219 | Folate antagonist | 0.219 0.008 CHEMBL226396 0.152 0.021 CHEMBL3526318 0.108 0.052 CHEMBL375462 0.107 0.054 CHEMBL3527205 0.101 0.063 CHEMBL3527204 0.129 0.032 CHEMBL3527203 0.151 0.022 CHEMBL3527549 0.105 0.056 CHEMBL3526210 0.098 0.068 CHEMBL3526912 0.11 0.049 CHEMBL3527548 | CHEMBL226396 | |
| 0.065 | 0.012 | 0.171 | Thymidine kinase inhibitor | 0.171 0.003 CHEMBL226396 0.086 0.008 CHEMBL375462 0.039 0.032 CHEMBL3527205 0.075 0.009 CHEMBL3527204 0.08 0.009 CHEMBL3527203 0.049 0.019 CHEMBL3526210 0.048 0.02 CHEMBL3526912 0.055 0.016 CHEMBL3527548 | CHEMBL226396 | |
| 0.13 | 0.077 | 0.499 | Ca2+/calmodulin-dependent kinase II delta inhibitor | 0.499 0.005 CHEMBL226396 0.142 0.069 CHEMBL375462 | CHEMBL226396 | |
| 0.131 | 0.082 | 0.555 | Protein kinase C nu inhibitor | 0.555 0.005 CHEMBL226396 0.136 0.078 CHEMBL375462 0.113 0.101 CHEMBL3527205 0.123 0.089 CHEMBL3526210 | CHEMBL226396 | |
| 0.136 | 0.088 | 0.47 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.47 0.005 CHEMBL226396 0.135 0.089 CHEMBL375462 | CHEMBL226396 | |
| 0.088 | 0.042 | 0.128 | Phosphodiesterase 4D inhibitor | 0.088 0.043 CHEMBL3527204 0.128 0.025 CHEMBL3527203 | CHEMBL3527203 | |
| 0.108 | 0.063 | 0.139 | Granulocyte macrophage colony stimulating factor antagonist | 0.139 0.041 CHEMBL226396 | CHEMBL226396 | |
| 0.141 | 0.1 | 0.361 | Protein kinase (CK1) gamma 3 inhibitor | 0.361 0.009 CHEMBL226396 0.148 0.092 CHEMBL375462 0.142 0.099 CHEMBL3527205 0.158 0.081 CHEMBL3526210 | CHEMBL226396 | |
| 0.061 | 0.021 | 0.062 | Alpha 1L adrenoreceptor antagonist | 0.061 0.021 CHEMBL4525761 0.052 0.036 CHEMBL3527205 0.051 0.04 CHEMBL3527204 0.062 0.019 CHEMBL3527203 | CHEMBL3527203 | |
| 0.112 | 0.072 | 0.376 | Protein kinase (CK1) gamma 2 inhibitor | 0.376 0.005 CHEMBL226396 0.115 0.069 CHEMBL375462 0.103 0.081 CHEMBL3527205 0.117 0.067 CHEMBL3526210 | CHEMBL226396 | |
| 0.098 | 0.065 | 0.295 | Cyclin-dependent kinase 9 inhibitor | 0.295 0.01 CHEMBL226396 0.091 0.073 CHEMBL375462 | CHEMBL226396 | |
| 0.122 | 0.09 | 0.476 | Protein kinase (CK1) inhibitor | 0.476 0.005 CHEMBL226396 0.123 0.089 CHEMBL375462 | CHEMBL226396 | |
| 0.151 | 0.119 | 0.422 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.422 0.009 CHEMBL226396 0.18 0.093 CHEMBL375462 | CHEMBL226396 | |
| 0.056 | 0.025 | 0.118 | Adenosine deaminase inhibitor | 0.118 0.004 CHEMBL226396 0.043 0.037 CHEMBL3526318 0.071 0.013 CHEMBL375462 0.073 0.012 CHEMBL3527204 0.076 0.011 CHEMBL3527203 0.058 0.023 CHEMBL3527549 0.06 0.021 CHEMBL3526912 0.072 0.012 CHEMBL3527548 | CHEMBL226396 | |
| 0.064 | 0.038 | 0.353 | Phosphatidylinositol kinase inhibitor | 0.353 0.005 CHEMBL226396 0.065 0.037 CHEMBL375462 0.064 0.038 CHEMBL3527204 | CHEMBL226396 | |
| 0.116 | 0.094 | 0.413 | Protein kinase (CK1) gamma inhibitor | 0.413 0.006 CHEMBL226396 0.116 0.094 CHEMBL375462 0.117 0.094 CHEMBL3526210 | CHEMBL226396 | |
| 0.089 | 0.071 | 0.119 | Phosphodiesterase 7B inhibitor | 0.097 0.06 CHEMBL226396 0.119 0.038 CHEMBL3527203 | CHEMBL3527203 | |
| 0.023 | 0.005 | 0.154 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.154 0.001 CHEMBL226396 0.023 0.004 CHEMBL375462 0.017 0.01 CHEMBL3527205 0.022 0.005 CHEMBL3527204 0.034 0.003 CHEMBL3527203 0.019 0.009 CHEMBL3526210 0.025 0.004 CHEMBL3526912 0.033 0.003 CHEMBL3527548 | CHEMBL226396 | |
| 0.098 | 0.081 | 0.119 | Platelet activating factor antagonist | 0.119 0.064 CHEMBL226396 | CHEMBL226396 | |
| 0.099 | 0.082 | 0.138 | Interleukin 1b antagonist | 0.138 0.049 CHEMBL3527203 0.099 0.082 CHEMBL3527548 | CHEMBL3527203 | |
| 0.139 | 0.123 | 0.582 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.582 0.005 CHEMBL226396 0.172 0.094 CHEMBL375462 | CHEMBL226396 | |
| 0.05 | 0.034 | 0.132 | Phosphatidylinositol 3-kinase beta inhibitor | 0.132 0.009 CHEMBL226396 0.049 0.034 CHEMBL375462 0.047 0.037 CHEMBL3526210 | CHEMBL226396 | |
| 0.11 | 0.1 | 0.262 | Cytokine production inhibitor | 0.262 0.021 CHEMBL3527205 0.158 0.057 CHEMBL3526210 | CHEMBL3527205 | |
| 0.109 | 0.099 | 0.443 | DNA repair enzyme inhibitor | 0.215 0.007 CHEMBL226396 0.116 0.08 CHEMBL4525761 0.109 0.097 CHEMBL375462 0.114 0.085 CHEMBL3527204 0.194 0.01 CHEMBL3527203 0.201 0.009 CHEMBL3526912 0.443 0.003 CHEMBL3527548 | CHEMBL3527548 | |
| 0.031 | 0.022 | 0.074 | Potassium channel small-conductance Ca-activated activator | 0.074 0.006 CHEMBL226396 | CHEMBL226396 | |
| 0.053 | 0.046 | 0.266 | Adenosine A1 receptor antagonist | 0.266 0.008 CHEMBL226396 0.078 0.029 CHEMBL375462 0.052 0.047 CHEMBL3527204 0.076 0.03 CHEMBL3527203 0.056 0.042 CHEMBL3526210 | CHEMBL226396 | |
| 0.015 | 0.01 | 0.021 | S-adenosyl-L-homocysteine hydrolase inhibitor | 0.021 0.006 CHEMBL226396 0.017 0.008 CHEMBL375462 0.016 0.009 CHEMBL3527204 0.016 0.009 CHEMBL3526912 | CHEMBL226396 | |
| 0.025 | 0.022 | 0.124 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.124 0.002 CHEMBL226396 0.038 0.013 CHEMBL375462 0.025 0.022 CHEMBL3527204 0.049 0.009 CHEMBL3527203 0.031 0.017 CHEMBL3527548 | CHEMBL226396 | |
| 0.096 | 0.094 | 0.533 | Cyclin-dependent kinase inhibitor | 0.533 0.006 CHEMBL226396 0.106 0.085 CHEMBL375462 | CHEMBL226396 | |
| 0.073 | 0.074 | 0.076 | MAP kinase 7 inhibitor | 0.076 0.059 CHEMBL3527203 | CHEMBL3527203 | |
| 0.078 | 0.08 | 0.205 | Platelet activating factor beta antagonist | 0.205 0.023 CHEMBL226396 | CHEMBL226396 | |
| 0.01 | 0.013 | 0.03 | Purine nucleoside phosphorylase inhibitor | 0.03 0.002 CHEMBL226396 0.014 0.005 CHEMBL375462 0.011 0.01 CHEMBL3527204 0.026 0.003 CHEMBL3527203 0.011 0.01 CHEMBL3527548 | CHEMBL226396 | |
| 0.07 | 0.077 | 0.088 | ErbB-3 antagonist | 0.088 0.051 CHEMBL226396 | CHEMBL226396 | |
| 0.037 | 0.049 | 0.061 | Dihydrofolate reductase inhibitor | 0.051 0.017 CHEMBL226396 0.046 0.025 CHEMBL4525761 0.061 0.01 CHEMBL3527203 | CHEMBL3527203 | |
| 0.082 | 0.097 | 0.387 | Cyclin-dependent kinase 2 inhibitor | 0.387 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.037 | 0.053 | 0.151 | Phosphatidylinositol 3-kinase alpha inhibitor | 0.151 0.01 CHEMBL226396 0.048 0.039 CHEMBL3527204 | CHEMBL226396 | |
| 0.079 | 0.095 | 0.167 | Gastric antisecretory | 0.167 0.02 CHEMBL4525761 0.108 0.056 CHEMBL3527203 | CHEMBL4525761 | |
| 0.053 | 0.072 | 0.392 | CDK1/cyclin B1 inhibitor | 0.392 0.004 CHEMBL226396 0.129 0.02 CHEMBL3527203 0.062 0.057 CHEMBL3527548 | CHEMBL226396 | |
| 0.042 | 0.062 | 0.175 | Cyclin B inhibitor | 0.175 0.005 CHEMBL226396 0.071 0.021 CHEMBL3527203 | CHEMBL226396 | |
| 0.045 | 0.066 | 0.38 | CDK1/cyclin B inhibitor | 0.38 0.005 CHEMBL226396 0.055 0.051 CHEMBL375462 0.084 0.032 CHEMBL3527203 | CHEMBL226396 | |
| 0.016 | 0.037 | 0.1 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.1 0.002 CHEMBL226396 0.022 0.011 CHEMBL375462 | CHEMBL226396 | |
| 0.046 | 0.067 | 0.191 | Cyclin B1 inhibitor | 0.191 0.004 CHEMBL226396 0.073 0.028 CHEMBL3527203 | CHEMBL226396 | |
| 0.023 | 0.046 | 0.097 | Phosphoglycerate kinase inhibitor | 0.097 0.007 CHEMBL226396 0.033 0.026 CHEMBL3527204 | CHEMBL226396 | |
| 0.003 | 0.027 | 0.013 | DNA polymerase III subunit alpha inhibitor | 0.013 0.003 CHEMBL3527203 0.007 0.005 CHEMBL3527548 | CHEMBL3527203 | |
| 0.01 | 0.036 | 0.023 | Inosine monophosphate dehydrogenase 1 inhibitor | 0.023 0.012 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.039 | 0.081 | Corticotropin releasing factor 1 receptor antagonist | 0.081 0.004 CHEMBL4525761 | CHEMBL4525761 | |
| 0.022 | 0.049 | 0.039 | DNA polymerase III inhibitor | 0.033 0.009 CHEMBL226396 0.029 0.018 CHEMBL4525761 0.039 0.005 CHEMBL3527203 | CHEMBL3527203 | |
| 0.107 | 0.135 | 0.448 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.448 0.01 CHEMBL226396 | CHEMBL226396 | |
| 0.038 | 0.066 | 0.097 | Histamine agonist | 0.097 0.009 CHEMBL226396 | CHEMBL226396 | |
| 0.013 | 0.042 | 0.025 | Adenosine A1 receptor agonist | 0.025 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.058 | 0.088 | 0.256 | Adenosine A3 receptor antagonist | 0.256 0.007 CHEMBL226396 0.066 0.065 CHEMBL375462 0.07 0.058 CHEMBL3527205 0.085 0.037 CHEMBL3527203 0.078 0.047 CHEMBL3526210 | CHEMBL226396 | |
| 0.094 | 0.125 | 0.315 | Ribosomal protein S6 kinase inhibitor | 0.315 0.01 CHEMBL226396 | CHEMBL226396 | |
| 0.03 | 0.061 | 0.077 | Histamine H2 receptor agonist | 0.077 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.072 | 0.104 | 0.12 | DNA directed RNA polymerase inhibitor | 0.11 0.046 CHEMBL226396 0.12 0.037 CHEMBL3527204 0.087 0.073 CHEMBL3527203 0.095 0.063 CHEMBL3526912 0.109 0.047 CHEMBL3527548 | CHEMBL3527204 | |
| 0.087 | 0.12 | 0.322 | Lck kinase inhibitor | 0.322 0.014 CHEMBL226396 | CHEMBL226396 | |
| 0.013 | 0.046 | 0.021 | Tryptophan hydroxylase 1 inhibitor | 0.021 0.005 CHEMBL226396 | CHEMBL226396 | |
| 0.156 | 0.191 | 0.285 | Nitric-oxide synthase stimulant | 0.285 0.016 CHEMBL226396 0.278 0.018 CHEMBL4525761 0.169 0.155 CHEMBL375462 0.172 0.146 CHEMBL3527204 0.174 0.143 CHEMBL3527203 | CHEMBL226396 | |
| 0.052 | 0.088 | 0.127 | I kappa B kinase 1 inhibitor | 0.127 0.013 CHEMBL226396 | CHEMBL226396 | |
| 0.117 | 0.154 | 0.19 | CF transmembrane conductance regulator agonist | 0.19 0.028 CHEMBL226396 0.158 0.063 CHEMBL4525761 0.129 0.122 CHEMBL375462 0.129 0.119 CHEMBL3527204 | CHEMBL226396 | |
| 0.009 | 0.046 | 0.034 | Adenosine A2 receptor agonist | 0.034 0.005 CHEMBL226396 | CHEMBL226396 | |
| 0.062 | 0.1 | 0.119 | Fibroblast growth factor 1 antagonist | 0.119 0.044 CHEMBL226396 0.104 0.054 CHEMBL3527203 | CHEMBL226396 | |
| 0.029 | 0.07 | 0.049 | Phosphodiesterase 4A inhibitor | 0.049 0.035 CHEMBL3527203 | CHEMBL3527203 | |
| 0.135 | 0.179 | 0.375 | Tumour necrosis factor alpha release inhibitor | 0.375 0.032 CHEMBL3526912 0.34 0.041 CHEMBL3527548 | CHEMBL3526912 | |
| 0.034 | 0.081 | 0.107 | CDK9/cyclin T1 inhibitor | 0.107 0.017 CHEMBL226396 | CHEMBL226396 | |
| 0.047 | 0.094 | 0.091 | CDK2/cyclin E2 inhibitor | 0.091 0.032 CHEMBL226396 | CHEMBL226396 | |
| 0.005 | 0.055 | 0.037 | Adenosine A2a receptor agonist | 0.037 0.004 CHEMBL226396 | CHEMBL226396 | |
| 0.05 | 0.1 | 0.083 | Fibroblast growth factor 3 antagonist | 0.083 0.047 CHEMBL226396 | CHEMBL226396 | |
| 0.03 | 0.081 | 0.086 | mTOR inhibitor | 0.086 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.112 | 0.163 | 0.2 | MAP kinase 3 inhibitor | 0.2 0.024 CHEMBL226396 0.141 0.083 CHEMBL4525761 0.15 0.068 CHEMBL3527203 | CHEMBL226396 | |
| 0.005 | 0.056 | 0.015 | Egl nine homolog 3 inhibitor | 0.015 0.005 CHEMBL4525761 | CHEMBL4525761 | |
| 0.091 | 0.143 | 0.346 | Src kinase inhibitor | 0.346 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.092 | 0.145 | 0.151 | Antibacterial (Helicobacter pylori) | 0.151 0.045 CHEMBL4525761 0.127 0.071 CHEMBL3527203 | CHEMBL4525761 | |
| 0.144 | 0.198 | 0.21 | ErbB-1 antagonist | 0.21 0.079 CHEMBL226396 0.175 0.124 CHEMBL375462 | CHEMBL226396 | |
| 0.112 | 0.166 | 0.435 | Interleukin antagonist | 0.4 0.031 CHEMBL3526318 0.135 0.13 CHEMBL375462 0.401 0.031 CHEMBL3527205 0.219 0.075 CHEMBL3527203 0.42 0.028 CHEMBL3527549 0.435 0.026 CHEMBL3526210 0.134 0.132 CHEMBL3527548 | CHEMBL3526210 | |
| 0.083 | 0.137 | 0.177 | Phosphodiesterase inhibitor | 0.177 0.043 CHEMBL3527205 0.112 0.091 CHEMBL3527203 0.147 0.06 CHEMBL3526210 | CHEMBL3527205 | |
| 0.028 | 0.082 | 0.157 | Adenosine A2b receptor antagonist | 0.157 0.006 CHEMBL226396 | CHEMBL226396 | |
| 0.037 | 0.091 | 0.049 | Autotaxin inhibitor | 0.049 0.043 CHEMBL4525761 0.049 0.043 CHEMBL3527205 | CHEMBL3527205 | |
| 0.005 | 0.063 | 0.018 | Egl nine homolog 1 inhibitor | 0.018 0.007 CHEMBL4525761 0.013 0.012 CHEMBL375462 0.014 0.011 CHEMBL3527203 | CHEMBL4525761 | |
| 0.037 | 0.095 | 0.105 | Alpha 2 adrenoreceptor agonist | 0.105 0.013 CHEMBL226396 | CHEMBL226396 | |
| 0.044 | 0.105 | 0.101 | Phosphodiesterase 1A inhibitor | 0.101 0.01 CHEMBL226396 | CHEMBL226396 | |
| 0.058 | 0.121 | 0.401 | CDK2/cyclin A inhibitor | 0.401 0.005 CHEMBL226396 | CHEMBL226396 | |
| 0.003 | 0.067 | 0.007 | Phosphoribosylglycinamide formyltransferase inhibitor | 0.007 0.005 CHEMBL226396 0.007 0.006 CHEMBL3527203 | CHEMBL3527203 | |
| 0.07 | 0.135 | 0.37 | Protein-tyrosine kinase Lyn inhibitor | 0.37 0.009 CHEMBL226396 | CHEMBL226396 | |
| 0.022 | 0.088 | 0.196 | Antimetabolite | 0.195 0.01 CHEMBL226396 0.149 0.012 CHEMBL3526318 0.052 0.03 CHEMBL3527203 0.196 0.01 CHEMBL3527549 0.069 0.022 CHEMBL3527548 | CHEMBL3527549 | |
| 0.009 | 0.074 | 0.013 | DNA polymerase III polC-type inhibitor | 0.013 0.01 CHEMBL4525761 | CHEMBL4525761 | |
| 0.066 | 0.131 | 0.226 | Protein kinase (CK1) delta inhibitor | 0.226 0.022 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.077 | 0.082 | Factor VII inhibitor | 0.082 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.084 | 0.103 | Factor VIIa inhibitor | 0.103 0.011 CHEMBL226396 | CHEMBL226396 | |
| 0.05 | 0.118 | 0.343 | CDK/cyclin complex inhibitor | 0.343 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.03 | 0.1 | 0.058 | EphB4 antagonist | 0.058 0.041 CHEMBL226396 | CHEMBL226396 | |
| 0.11 | 0.181 | 0.317 | I kappa B kinase epsilon inhibitor | 0.317 0.009 CHEMBL226396 | CHEMBL226396 | |
| 0.085 | 0.156 | 0.245 | Activin receptor-like kinase 2 inhibitor | 0.245 0.022 CHEMBL226396 | CHEMBL226396 | |
| 0.04 | 0.112 | 0.145 | Cyclin B3 inhibitor | 0.145 0.014 CHEMBL226396 0.074 0.042 CHEMBL3527203 | CHEMBL226396 | |
| 0.156 | 0.23 | 0.251 | Angiogenesis inhibitor | 0.25 0.123 CHEMBL3527203 0.251 0.122 CHEMBL3527548 | CHEMBL3527548 | |
| 0.028 | 0.101 | 0.13 | Cyclin B2 inhibitor | 0.13 0.005 CHEMBL226396 0.071 0.021 CHEMBL3527203 | CHEMBL226396 | |
| 0.032 | 0.107 | 0.142 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.142 0.009 CHEMBL226396 0.079 0.021 CHEMBL4525761 0.052 0.045 CHEMBL375462 0.105 0.013 CHEMBL3527203 0.113 0.012 CHEMBL3527548 | CHEMBL226396 | |
| 0.045 | 0.121 | 0.162 | Platelet growth factor antagonist | 0.162 0.016 CHEMBL226396 | CHEMBL226396 | |
| 0.115 | 0.194 | 0.401 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.401 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.07 | 0.155 | 0.148 | Epidermal growth factor receptor kinase inhibitor | 0.148 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.116 | 0.046 | Nicotinic receptor alpha4 subunit antagonist | 0.046 0.042 CHEMBL226396 | CHEMBL226396 | |
| 0.019 | 0.108 | 0.103 | CDK5/p25 inhibitor | 0.103 0.006 CHEMBL226396 | CHEMBL226396 | |
| 0.091 | 0.18 | 0.37 | TRKC antagonist | 0.37 0.014 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.12 | 0.155 | Histamine H4 receptor antagonist | 0.155 0.004 CHEMBL226396 | CHEMBL226396 | |
| 0.04 | 0.132 | 0.1 | Potassium channel (ATP-sensitive) blocker | 0.1 0.015 CHEMBL4525761 | CHEMBL4525761 | |
| 0.031 | 0.129 | 0.255 | CDC7 inhibitor | 0.255 0.004 CHEMBL226396 | CHEMBL226396 | |
| 0.007 | 0.108 | 0.026 | CDK2/cyclin A3 inhibitor | 0.026 0.004 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.119 | 0.039 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.039 0.005 CHEMBL226396 0.032 0.009 CHEMBL3527203 | CHEMBL226396 | |
| 0.062 | 0.167 | 0.152 | Beta amyloid protein antagonist | 0.152 0.039 CHEMBL4525761 | CHEMBL4525761 | |
| 0.006 | 0.113 | 0.052 | Histamine H4 receptor agonist | 0.052 0.004 CHEMBL226396 | CHEMBL226396 | |
| 0.057 | 0.166 | 0.101 | Polo-like kinase-1 inhibitor | 0.101 0.045 CHEMBL226396 | CHEMBL226396 | |
| 0.051 | 0.16 | 0.122 | Ephrin antagonist | 0.122 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.126 | 0.052 | CDK2/cyclin E inhibitor | 0.052 0.051 CHEMBL226396 | CHEMBL226396 | |
| 0.053 | 0.164 | 0.257 | c-Src kinase inhibitor | 0.257 0.024 CHEMBL226396 | CHEMBL226396 | |
| 0.02 | 0.132 | 0.051 | Tryptophan 5 hydroxylase inhibitor | 0.051 0.005 CHEMBL226396 | CHEMBL226396 | |
| 0.083 | 0.197 | 0.352 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.352 0.018 CHEMBL226396 | CHEMBL226396 | |
| 0.014 | 0.131 | 0.035 | Thymidine phosphorylase inhibitor | 0.035 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.053 | 0.171 | 0.338 | RET inhibitor | 0.338 0.016 CHEMBL226396 | CHEMBL226396 | |
| 0.023 | 0.145 | 0.068 | Cyclin A1 inhibitor | 0.068 0.024 CHEMBL226396 | CHEMBL226396 | |
| 0.039 | 0.162 | 0.371 | Protein kinase A inhibitor | 0.371 0.005 CHEMBL226396 | CHEMBL226396 | |
| 0.042 | 0.165 | 0.076 | Epidermal growth factor antagonist | 0.076 0.072 CHEMBL226396 | CHEMBL226396 | |
| 0.071 | 0.194 | 0.851 | Interleukin 4 antagonist | 0.812 0.003 CHEMBL3527205 0.851 0.003 CHEMBL3526210 0.138 0.062 CHEMBL3526912 0.145 0.054 CHEMBL3527548 | CHEMBL3526210 | |
| 0.084 | 0.209 | 0.307 | LIM domain kinase 1 inhibitor | 0.307 0.02 CHEMBL226396 | CHEMBL226396 | |
| 0.151 | 0.275 | 0.695 | Toll-Like receptor agonist | 0.349 0.082 CHEMBL226396 0.64 0.013 CHEMBL3527205 0.695 0.009 CHEMBL3526210 | CHEMBL3526210 | |
| 0.004 | 0.129 | 0.025 | Cyclin T1 inhibitor | 0.025 0.007 CHEMBL226396 | CHEMBL226396 | |
| 0.009 | 0.134 | 0.024 | Alpha 2d adrenoreceptor agonist | 0.024 0.013 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.137 | 0.021 | Toll-Like receptor 8 agonist | 0.021 0.012 CHEMBL3526210 | CHEMBL3526210 | |
| 0.015 | 0.143 | 0.085 | Phosphodiesterase 2A inhibitor | 0.085 0.012 CHEMBL3527205 0.081 0.013 CHEMBL3526210 | CHEMBL3527205 | |
| 0.021 | 0.149 | 0.053 | Potassium channel (Inward rectifier) blocker | 0.053 0.03 CHEMBL4525761 | CHEMBL4525761 | |
| 0.019 | 0.149 | 0.036 | Nicotinic acid receptor 1 agonist | 0.036 0.034 CHEMBL226396 | CHEMBL226396 | |
| 0.009 | 0.139 | 0.109 | Histamine H3 receptor agonist | 0.109 0.006 CHEMBL226396 | CHEMBL226396 | |
| 0.023 | 0.154 | 0.088 | Phosphatidylinositol 3-kinase gamma inhibitor | 0.088 0.018 CHEMBL226396 | CHEMBL226396 | |
| 0.024 | 0.155 | 0.131 | Cyclin A2 inhibitor | 0.131 0.016 CHEMBL226396 | CHEMBL226396 | |
| 0.066 | 0.198 | 0.11 | CDC-like kinase 3 inhibitor | 0.11 0.058 CHEMBL226396 | CHEMBL226396 | |
| 0.059 | 0.191 | 0.13 | Tyrosine-protein kinase receptor antagonist | 0.13 0.077 CHEMBL226396 | CHEMBL226396 | |
| 0.031 | 0.164 | 0.111 | Leucine-rich repeat kinase 2 inhibitor | 0.111 0.036 CHEMBL226396 | CHEMBL226396 | |
| 0.014 | 0.148 | 0.094 | Phosphodiesterase II inhibitor | 0.094 0.013 CHEMBL3527205 0.09 0.014 CHEMBL3526210 | CHEMBL3527205 | |
| 0.055 | 0.19 | 0.127 | ABCA1 expression enhancer | 0.127 0.026 CHEMBL4525761 | CHEMBL4525761 | |
| 0.056 | 0.193 | 0.128 | Cyclooxygenase 1 inhibitor | 0.128 0.073 CHEMBL375462 0.125 0.075 CHEMBL3526210 | CHEMBL375462 | |
| 0.053 | 0.19 | 0.15 | MAP kinase 13 inhibitor | 0.15 0.036 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.166 | 0.057 | Fibroblast growth factor 2 antagonist | 0.057 0.056 CHEMBL226396 | CHEMBL226396 | |
| 0.098 | 0.24 | 0.233 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.233 0.069 CHEMBL226396 | CHEMBL226396 | |
| 0.022 | 0.165 | 0.111 | Cyclin A inhibitor | 0.111 0.02 CHEMBL226396 | CHEMBL226396 | |
| 0.099 | 0.246 | 0.159 | MAP kinase kinase 4 inhibitor | 0.159 0.046 CHEMBL226396 0.141 0.081 CHEMBL3527203 | CHEMBL226396 | |
| 0.053 | 0.201 | 0.212 | MAP kinase 12 inhibitor | 0.212 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.03 | 0.179 | 0.09 | Proto-oncogene tyrosine-protein kinase c-hck inhibitor | 0.09 0.042 CHEMBL226396 | CHEMBL226396 | |
| 0.142 | 0.292 | 0.69 | Toll-Like receptor 7 agonist | 0.323 0.096 CHEMBL226396 0.634 0.014 CHEMBL3527205 0.69 0.009 CHEMBL3526210 | CHEMBL3526210 | |
| 0.04 | 0.19 | 0.098 | Phosphodiesterase VI inhibitor | 0.084 0.035 CHEMBL4525761 0.094 0.025 CHEMBL3527203 0.098 0.022 CHEMBL3527548 | CHEMBL3527548 | |
| 0.021 | 0.172 | 0.09 | Glucagon-like peptide 1 agonist | 0.088 0.029 CHEMBL3526318 0.09 0.028 CHEMBL3527549 | CHEMBL3527549 | |
| 0.033 | 0.185 | 0.146 | Protein kinase B beta inhibitor | 0.146 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.044 | 0.196 | 0.144 | Aurora-B kinase inhibitor | 0.144 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.024 | 0.177 | 0.053 | Cytokine production stimulant | 0.047 0.036 CHEMBL3526912 0.053 0.023 CHEMBL3527548 | CHEMBL3527548 | |
| 0.034 | 0.189 | 0.276 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.276 0.022 CHEMBL226396 | CHEMBL226396 | |
| 0.104 | 0.259 | 0.308 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.308 0.028 CHEMBL226396 | CHEMBL226396 | |
| 0.062 | 0.218 | 0.506 | Electron transport complex I inhibitor | 0.506 0.003 CHEMBL4525761 | CHEMBL4525761 | |
| 0.049 | 0.208 | 0.107 | TRKA antagonist | 0.107 0.08 CHEMBL226396 | CHEMBL226396 | |
| 0.015 | 0.176 | 0.039 | Protein kinase (CK1) epsilon inhibitor | 0.039 0.027 CHEMBL226396 | CHEMBL226396 | |
| 0.01 | 0.172 | 0.045 | Geranyltranstransferase inhibitor | 0.045 0.029 CHEMBL226396 | CHEMBL226396 | |
| 0.045 | 0.208 | 0.106 | EphA2 antagonist | 0.106 0.069 CHEMBL226396 | CHEMBL226396 | |
| 0.004 | 0.168 | 0.022 | Adenosine kinase inhibitor | 0.022 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.197 | 0.131 | TIE antagonist | 0.131 0.027 CHEMBL226396 | CHEMBL226396 | |
| 0.058 | 0.228 | 0.082 | T cell inhibitor | 0.082 0.057 CHEMBL3527203 | CHEMBL3527203 | |
| 0.034 | 0.203 | 0.088 | MAP kinase kinase kinase inhibitor | 0.088 0.078 CHEMBL226396 | CHEMBL226396 | |
| 0.033 | 0.203 | 0.088 | Vascular endothelial growth factor 2 antagonist | 0.088 0.081 CHEMBL226396 | CHEMBL226396 | |
| 0.142 | 0.313 | 0.616 | Antibacterial | 0.315 0.124 CHEMBL3526318 0.265 0.163 CHEMBL375462 0.235 0.192 CHEMBL3527203 0.419 0.069 CHEMBL3527549 0.592 0.02 CHEMBL3526912 0.616 0.017 CHEMBL3527548 | CHEMBL3527548 | |
| 0.041 | 0.214 | 0.098 | Vascular endothelial growth factor antagonist | 0.098 0.083 CHEMBL226396 | CHEMBL226396 | |
| 0.026 | 0.199 | 0.092 | Rho-associated kinase I inhibitor | 0.092 0.037 CHEMBL226396 | CHEMBL226396 | |
| 0.047 | 0.222 | 0.258 | NADH dehydrogenase inhibitor | 0.258 0.008 CHEMBL226396 0.104 0.04 CHEMBL4525761 0.129 0.024 CHEMBL3526912 0.168 0.014 CHEMBL3527548 | CHEMBL226396 | |
| 0.033 | 0.209 | 0.097 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.097 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.04 | 0.223 | 0.083 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.083 0.058 CHEMBL226396 | CHEMBL226396 | |
| 0.076 | 0.26 | 0.441 | MAP kinase kinase 2 inhibitor | 0.441 0.008 CHEMBL226396 | CHEMBL226396 | |
| 0.027 | 0.212 | 0.114 | TIE-2 antagonist | 0.114 0.032 CHEMBL226396 | CHEMBL226396 | |
| 0.032 | 0.217 | 0.141 | Protein kinase B gamma inhibitor | 0.141 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.013 | 0.199 | 0.025 | Complement factor 1s inhibitor | 0.025 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.012 | 0.198 | 0.047 | Factor XIa inhibitor | 0.047 0.021 CHEMBL226396 | CHEMBL226396 | |
| 0.027 | 0.215 | 0.227 | Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor | 0.227 0.014 CHEMBL226396 | CHEMBL226396 | |
| 0.047 | 0.235 | 0.116 | MAP kinase kinase 7 inhibitor | 0.116 0.005 CHEMBL226396 0.073 0.071 CHEMBL3527203 | CHEMBL226396 | |
| 0.035 | 0.225 | 0.063 | Phosphodiesterase 1C inhibitor | 0.06 0.047 CHEMBL4525761 0.063 0.041 CHEMBL3527203 | CHEMBL3527203 | |
| 0.018 | 0.209 | 0.171 | Carbamoyl phosphate synthetase inhibitor | 0.171 0.009 CHEMBL226396 | CHEMBL226396 | |
| 0.054 | 0.245 | 0.134 | Alpha 2d adrenoreceptor antagonist | 0.134 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.21 | 0.099 | AICAR transformylase inhibitor | 0.099 0.005 CHEMBL226396 0.056 0.017 CHEMBL3527203 | CHEMBL226396 | |
| 0.019 | 0.218 | 0.114 | HIV-1 reverse transcriptase inhibitor | 0.114 0.024 CHEMBL4525761 | CHEMBL4525761 | |
| 0.039 | 0.245 | 0.103 | Aminoacyl-tRNA synthetase inhibitor | 0.103 0.042 CHEMBL3526318 0.096 0.05 CHEMBL3527549 | CHEMBL3526318 | |
| 0.062 | 0.27 | 0.246 | Cell wall synthesis inhibitor | 0.12 0.1 CHEMBL3527549 0.195 0.032 CHEMBL3526912 0.246 0.017 CHEMBL3527548 | CHEMBL3527548 | |
| 0.016 | 0.226 | 0.054 | CDK4/cyclin D1 inhibitor | 0.054 0.045 CHEMBL226396 | CHEMBL226396 | |
| 0.015 | 0.227 | 0.057 | CDK4/cyclin D inhibitor | 0.057 0.043 CHEMBL226396 | CHEMBL226396 | |
| 0.103 | 0.316 | 0.282 | Hypoxia-inducible factor 1 alpha inhibitor | 0.2 0.151 CHEMBL226396 0.211 0.14 CHEMBL4525761 0.282 0.075 CHEMBL3527203 0.248 0.102 CHEMBL3527548 | CHEMBL3527203 | |
| 0.071 | 0.284 | 0.159 | Polo-like kinase-3 inhibitor | 0.159 0.075 CHEMBL226396 | CHEMBL226396 | |
| 0.005 | 0.219 | 0.015 | Purinergic P2Y1 agonist | 0.015 0.011 CHEMBL226396 | CHEMBL226396 | |
| 0.02 | 0.234 | 0.077 | Alpha adrenoreceptor agonist | 0.077 0.04 CHEMBL226396 | CHEMBL226396 | |
| 0.015 | 0.231 | 0.144 | Raf kinase inhibitor | 0.144 0.02 CHEMBL226396 | CHEMBL226396 | |
| 0.032 | 0.25 | 0.112 | Vascular endothelial growth factor 1 antagonist | 0.112 0.059 CHEMBL226396 | CHEMBL226396 | |
| 0.045 | 0.265 | 0.27 | Tyrosine kinase inhibitor | 0.27 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.042 | 0.262 | 0.234 | MAP kinase kinase inhibitor | 0.234 0.018 CHEMBL226396 | CHEMBL226396 | |
| 0.016 | 0.236 | 0.034 | ATR kinase inhibitor | 0.034 0.02 CHEMBL226396 | CHEMBL226396 | |
| 0.031 | 0.253 | 0.125 | AXL receptor tyrosine kinase inhibitor | 0.125 0.025 CHEMBL226396 | CHEMBL226396 | |
| 0.014 | 0.236 | 0.148 | Janus tyrosine kinase 3 inhibitor | 0.148 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.085 | 0.31 | 0.219 | ATPase inhibitor | 0.219 0.025 CHEMBL4525761 | CHEMBL4525761 | |
| 0.004 | 0.23 | 0.027 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.027 0.009 CHEMBL4525761 | CHEMBL4525761 | |
| 0.031 | 0.258 | 0.264 | Glycogen synthase kinase-3 inhibitor | 0.264 0.02 CHEMBL226396 0.094 0.085 CHEMBL3526210 | CHEMBL226396 | |
| 0.123 | 0.35 | 0.462 | GABA C receptor rho-3 antagonist | 0.462 0.037 CHEMBL226396 0.429 0.049 CHEMBL4525761 0.219 0.185 CHEMBL375462 | CHEMBL226396 | |
| 0.086 | 0.317 | 0.238 | Cyclic AMP phosphodiesterase inhibitor | 0.16 0.135 CHEMBL226396 0.238 0.07 CHEMBL4525761 0.164 0.13 CHEMBL3527203 0.178 0.113 CHEMBL3527548 | CHEMBL4525761 | |
| 0.066 | 0.298 | 0.44 | Immunostimulant | 0.256 0.094 CHEMBL226396 0.4 0.049 CHEMBL3526318 0.214 0.112 CHEMBL3527205 0.44 0.039 CHEMBL3527549 0.265 0.09 CHEMBL3526210 0.423 0.043 CHEMBL3526912 0.414 0.046 CHEMBL3527548 | CHEMBL3527549 | |
| 0.01 | 0.247 | 0.113 | Raf kinase B inhibitor | 0.113 0.02 CHEMBL226396 | CHEMBL226396 | |
| 0.066 | 0.303 | 0.151 | DNA methylase inhibitor | 0.151 0.116 CHEMBL3527548 | CHEMBL3527548 | |
| 0.024 | 0.262 | 0.05 | Bombesin 2 receptor antagonist | 0.05 0.033 CHEMBL226396 | CHEMBL226396 | |
| 0.038 | 0.277 | 0.087 | Factor XII inhibitor | 0.087 0.054 CHEMBL3526318 0.085 0.057 CHEMBL3527549 | CHEMBL3526318 | |
| 0.053 | 0.293 | 0.113 | Glutamate release inhibitor | 0.113 0.028 CHEMBL226396 | CHEMBL226396 | |
| 0.042 | 0.282 | 0.146 | Electrolyte absorption antagonist | 0.146 0.021 CHEMBL226396 | CHEMBL226396 | |
| 0.028 | 0.269 | 0.233 | Glycogen synthase kinase-3 beta inhibitor | 0.233 0.022 CHEMBL226396 0.091 0.09 CHEMBL3527205 0.1 0.078 CHEMBL3526210 | CHEMBL226396 | |
| 0.033 | 0.273 | 0.14 | Vascular endothelial growth factor 3 antagonist | 0.14 0.075 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.271 | 0.095 | Myeloperoxidase inhibitor | 0.095 0.041 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.261 | 0.087 | Syk tyrosine kinase inhibitor | 0.087 0.036 CHEMBL226396 | CHEMBL226396 | |
| 0.035 | 0.281 | 0.099 | Insulin receptor antagonist | 0.099 0.063 CHEMBL226396 | CHEMBL226396 | |
| 0.039 | 0.286 | 0.166 | MAP kinase kinase 1 inhibitor | 0.166 0.011 CHEMBL226396 0.107 0.048 CHEMBL4525761 | CHEMBL226396 | |
| 0.02 | 0.268 | 0.083 | Rho-associated kinase inhibitor | 0.083 0.044 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.26 | 0.072 | Xanthine dehydrogenase inhibitor | 0.072 0.03 CHEMBL226396 0.071 0.03 CHEMBL4525761 0.052 0.044 CHEMBL3527203 | CHEMBL226396 | |
| 0.058 | 0.31 | 0.183 | Cyclin-dependent kinase 8 inhibitor | 0.183 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.095 | 0.348 | 0.227 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.227 0.054 CHEMBL4525761 0.208 0.066 CHEMBL3527203 | CHEMBL4525761 | |
| 0.024 | 0.285 | 0.068 | Protein kinase B alpha inhibitor | 0.068 0.05 CHEMBL226396 | CHEMBL226396 | |
| 0.026 | 0.288 | 0.116 | Histamine N-methyltransferase inhibitor | 0.116 0.033 CHEMBL226396 | CHEMBL226396 | |
| 0.024 | 0.286 | 0.069 | Purinergic P2X1 antagonist | 0.069 0.033 CHEMBL226396 0.064 0.037 CHEMBL4525761 | CHEMBL226396 | |
| 0.029 | 0.292 | 0.152 | MAP kinase 9 inhibitor | 0.152 0.037 CHEMBL226396 | CHEMBL226396 | |
| 0.008 | 0.273 | 0.033 | Purinergic P2Y15 antagonist | 0.033 0.012 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.283 | 0.078 | Janus tyrosine kinase 2 inhibitor | 0.078 0.049 CHEMBL226396 | CHEMBL226396 | |
| 0.025 | 0.292 | 0.162 | I kappa B kinase inhibitor | 0.162 0.013 CHEMBL226396 | CHEMBL226396 | |
| 0.041 | 0.31 | 0.1 | Nav1.4 sodium channel blocker | 0.096 0.082 CHEMBL3526318 0.1 0.076 CHEMBL3527549 | CHEMBL3527549 | |
| 0.028 | 0.299 | 0.116 | Glutamate dehydrogenase inhibitor | 0.116 0.024 CHEMBL226396 0.082 0.043 CHEMBL3527549 | CHEMBL226396 | |
| 0.019 | 0.291 | 0.077 | CYP2A6 inhibitor | 0.077 0.051 CHEMBL4525761 | CHEMBL4525761 | |
| 0.035 | 0.308 | 0.132 | Proto-oncogene tyrosine-protein kinase Yes inhibitor | 0.132 0.073 CHEMBL226396 | CHEMBL226396 | |
| 0.006 | 0.285 | 0.054 | Dihydropteroate synthase inhibitor | 0.054 0.014 CHEMBL226396 | CHEMBL226396 | |
| 0.04 | 0.321 | 0.21 | Adenylate cyclase inhibitor | 0.21 0.024 CHEMBL226396 | CHEMBL226396 | |
| 0.017 | 0.298 | 0.041 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.038 0.037 CHEMBL226396 0.041 0.03 CHEMBL4525761 | CHEMBL4525761 | |
| 0.093 | 0.38 | 0.202 | Vasodilator, peripheral | 0.202 0.173 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.306 | 0.181 | Protein kinase (CK2) alpha inhibitor | 0.181 0.029 CHEMBL226396 | CHEMBL226396 | |
| 0.018 | 0.31 | 0.062 | Epithelial sodium channel blocker | 0.062 0.026 CHEMBL226396 | CHEMBL226396 | |
| 0.007 | 0.3 | 0.071 | Ornithine carbamoyltransferase inhibitor | 0.071 0.025 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.305 | 0.12 | Argininosuccinate synthase inhibitor | 0.12 0.015 CHEMBL226396 | CHEMBL226396 | |
| 0.007 | 0.303 | 0.042 | Inosine monophosphate dehydrogenase inhibitor | 0.042 0.02 CHEMBL4525761 | CHEMBL4525761 | |
| 0.005 | 0.303 | 0.032 | Fumarate hydratase inhibitor | 0.032 0.026 CHEMBL226396 | CHEMBL226396 | |
| 0.039 | 0.338 | 0.304 | EphB2 antagonist | 0.304 0.034 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.31 | 0.088 | Phosphofructokinase-1 inhibitor | 0.088 0.037 CHEMBL226396 0.063 0.054 CHEMBL4525761 0.059 0.058 CHEMBL3527548 | CHEMBL226396 | |
| 0.04 | 0.339 | 0.333 | Interleukin 5 antagonist | 0.291 0.004 CHEMBL3527205 0.333 0.004 CHEMBL3526210 | CHEMBL3526210 | |
| 0.119 | 0.422 | 0.396 | Apoptosis agonist | 0.396 0.115 CHEMBL3526912 0.283 0.185 CHEMBL3527548 | CHEMBL3526912 | |
| 0.077 | 0.385 | 0.482 | Immunosuppressant | 0.297 0.117 CHEMBL3526318 0.303 0.113 CHEMBL3527203 0.27 0.134 CHEMBL3527549 0.398 0.064 CHEMBL3526912 0.482 0.038 CHEMBL3527548 | CHEMBL3527548 | |
| 0.006 | 0.315 | 0.045 | Guanylate cyclase inhibitor | 0.045 0.026 CHEMBL4525761 | CHEMBL4525761 | |
| 0.082 | 0.393 | 0.248 | MAP-kinase-activated kinase 5 inhibitor | 0.248 0.061 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.327 | 0.089 | Interleukin-1 receptor-associated protein kinase 4 inhibitor | 0.089 0.058 CHEMBL226396 | CHEMBL226396 | |
| 0.056 | 0.372 | 0.203 | GABA C receptor rho-2 antagonist | 0.152 0.071 CHEMBL226396 0.203 0.027 CHEMBL4525761 | CHEMBL4525761 | |
| 0.024 | 0.347 | 0.09 | MAP kinase 8 inhibitor | 0.09 0.073 CHEMBL226396 | CHEMBL226396 | |
| 0.019 | 0.348 | 0.093 | Phosphodiesterase 3A inhibitor | 0.093 0.038 CHEMBL4525761 0.086 0.047 CHEMBL3527203 | CHEMBL4525761 | |
| 0.01 | 0.349 | 0.049 | Histamine H1 receptor agonist | 0.049 0.021 CHEMBL226396 | CHEMBL226396 | |
| 0.015 | 0.356 | 0.117 | Aurora-A kinase inhibitor | 0.117 0.056 CHEMBL226396 | CHEMBL226396 | |
| 0.024 | 0.366 | 0.112 | Tubulin antagonist | 0.112 0.088 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.355 | 0.061 | Biliverdin reductase inhibitor | 0.061 0.04 CHEMBL226396 0.056 0.045 CHEMBL4525761 | CHEMBL226396 | |
| 0.021 | 0.367 | 0.199 | Glycogen synthase kinase-3 alpha inhibitor | 0.199 0.042 CHEMBL226396 | CHEMBL226396 | |
| 0.007 | 0.357 | 0.057 | Thymidylate synthase inhibitor | 0.057 0.019 CHEMBL226396 0.051 0.026 CHEMBL3527549 | CHEMBL226396 | |
| 0.012 | 0.364 | 0.212 | Protein kinase (CK2) inhibitor | 0.212 0.017 CHEMBL226396 | CHEMBL226396 | |
| 0.066 | 0.422 | 0.229 | Superoxide dismutase inhibitor | 0.19 0.129 CHEMBL226396 0.229 0.09 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.369 | 0.072 | Phosphodiesterase 5A inhibitor | 0.072 0.048 CHEMBL3527203 | CHEMBL3527203 | |
| 0.012 | 0.376 | 0.071 | Phosphodiesterase V inhibitor | 0.071 0.051 CHEMBL3527203 | CHEMBL3527203 | |
| 0.02 | 0.391 | 0.047 | Carbonic anhydrase II stimulant | 0.047 0.046 CHEMBL3527549 | CHEMBL3527549 | |
| 0.033 | 0.404 | 0.107 | Granulocyte macrophage colony stimulating factor agonist | 0.107 0.027 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.385 | 0.069 | Check point kinase 1 inhibitor | 0.069 0.047 CHEMBL226396 | CHEMBL226396 | |
| 0.051 | 0.428 | 0.172 | NOS3 expression enhancer | 0.172 0.055 CHEMBL3526912 0.154 0.069 CHEMBL3527548 | CHEMBL3526912 | |
| 0.039 | 0.417 | 0.288 | Peroxidase inhibitor | 0.165 0.071 CHEMBL226396 0.287 0.04 CHEMBL4525761 0.288 0.04 CHEMBL3527549 | CHEMBL3527549 | |
| 0.143 | 0.522 | 0.39 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.317 0.19 CHEMBL226396 0.39 0.11 CHEMBL4525761 | CHEMBL4525761 | |
| 0.08 | 0.459 | 0.32 | Vasodilator, coronary | 0.228 0.156 CHEMBL4525761 0.261 0.123 CHEMBL3526912 0.32 0.072 CHEMBL3527548 | CHEMBL3527548 | |
| 0.026 | 0.41 | 0.181 | Aryl hydrocarbon receptor agonist | 0.181 0.113 CHEMBL4525761 | CHEMBL4525761 | |
| 0.125 | 0.511 | 0.202 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.202 0.161 CHEMBL226396 0.202 0.161 CHEMBL3527203 | CHEMBL3527203 | |
| 0.016 | 0.403 | 0.087 | Alcohol dehydrogenase inhibitor | 0.087 0.068 CHEMBL226396 0.082 0.077 CHEMBL3527549 | CHEMBL226396 | |
| 0.017 | 0.408 | 0.077 | Pregnane X receptor antagonist | 0.077 0.008 CHEMBL4525761 | CHEMBL4525761 | |
| 0.11 | 0.502 | 0.374 | 5 Hydroxytryptamine release inhibitor | 0.292 0.174 CHEMBL226396 0.374 0.096 CHEMBL4525761 | CHEMBL4525761 | |
| 0.041 | 0.434 | 0.123 | Adenylate kinase inhibitor | 0.123 0.041 CHEMBL226396 0.097 0.072 CHEMBL4525761 | CHEMBL226396 | |
| 0.013 | 0.412 | 0.171 | Pim-1 kinase inhibitor | 0.171 0.021 CHEMBL226396 | CHEMBL226396 | |
| 0.016 | 0.416 | 0.06 | Orexin receptor antagonist | 0.06 0.058 CHEMBL4525761 | CHEMBL4525761 | |
| 0.011 | 0.414 | 0.083 | Histidine decarboxylase inhibitor | 0.063 0.058 CHEMBL226396 0.081 0.042 CHEMBL4525761 0.083 0.04 CHEMBL3527549 | CHEMBL3527549 | |
| 0.033 | 0.448 | 0.061 | Calcium channel P-type blocker | 0.061 0.054 CHEMBL4525761 | CHEMBL4525761 | |
| 0.024 | 0.445 | 0.123 | Nav1.6 sodium channel blocker | 0.123 0.092 CHEMBL4525761 | CHEMBL4525761 | |
| 0.024 | 0.447 | 0.133 | GABA C receptor rho-1 antagonist | 0.133 0.03 CHEMBL226396 0.113 0.047 CHEMBL4525761 | CHEMBL226396 | |
| 0.067 | 0.491 | 0.348 | Histamine release inhibitor | 0.348 0.101 CHEMBL4525761 0.216 0.184 CHEMBL3527548 | CHEMBL4525761 | |
| 0.017 | 0.444 | 0.121 | Mucolytic | 0.121 0.054 CHEMBL4525761 | CHEMBL4525761 | |
| 0.007 | 0.434 | 0.059 | Acyl-CoA dehydrogenase inhibitor | 0.059 0.034 CHEMBL226396 | CHEMBL226396 | |
| 0.012 | 0.444 | 0.091 | Protein kinase C zeta inhibitor | 0.091 0.063 CHEMBL226396 | CHEMBL226396 | |
| 0.013 | 0.445 | 0.095 | Expectorant | 0.095 0.074 CHEMBL4525761 | CHEMBL4525761 | |
| 0.016 | 0.45 | 0.069 | Potassium channel (Tandem pore domain) blocker | 0.069 0.068 CHEMBL4525761 | CHEMBL4525761 | |
| 0.009 | 0.446 | 0.076 | Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor | 0.076 0.053 CHEMBL226396 | CHEMBL226396 | |
| 0.057 | 0.496 | 0.23 | Cholesterol antagonist | 0.23 0.14 CHEMBL4525761 0.22 0.148 CHEMBL3526912 | CHEMBL4525761 | |
| 0.033 | 0.472 | 0.146 | MAP3K9 inhibitor | 0.146 0.067 CHEMBL226396 | CHEMBL226396 | |
| 0.029 | 0.469 | 0.119 | Interleukin 8 antagonist | 0.119 0.063 CHEMBL226396 | CHEMBL226396 | |
| 0.008 | 0.45 | 0.078 | Na+ K+ transporting ATPase inhibitor | 0.078 0.053 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.456 | 0.117 | Phenylalanine 4-hydroxylase inhibitor | 0.117 0.019 CHEMBL226396 | CHEMBL226396 | |
| 0.1 | 0.547 | 0.243 | MAP kinase kinase 6 inhibitor | 0.243 0.199 CHEMBL3527203 | CHEMBL3527203 | |
| 0.034 | 0.484 | 0.087 | D-Ala-D-Ala ligase inhibitor | 0.087 0.051 CHEMBL4525761 | CHEMBL4525761 | |
| 0.036 | 0.487 | 0.148 | Aurora-C kinase inhibitor | 0.148 0.053 CHEMBL226396 | CHEMBL226396 | |
| 0.006 | 0.458 | 0.031 | Phosphodiesterase 6B inhibitor | 0.031 0.021 CHEMBL3527203 | CHEMBL3527203 | |
| 0.024 | 0.477 | 0.152 | Xanthine oxidase inhibitor | 0.104 0.056 CHEMBL226396 0.091 0.07 CHEMBL4525761 0.152 0.034 CHEMBL3527548 | CHEMBL3527548 | |
| 0.079 | 0.537 | 0.159 | Ca2+-transporting ATPase inhibitor | 0.159 0.025 CHEMBL4525761 | CHEMBL4525761 | |
| 0.009 | 0.468 | 0.139 | Porphobilinogen synthase inhibitor | 0.139 0.023 CHEMBL4525761 | CHEMBL4525761 | |
| 0.011 | 0.472 | 0.055 | Carbonic anhydrase stimulant | 0.055 0.047 CHEMBL226396 | CHEMBL226396 | |
| 0.033 | 0.496 | 0.127 | Sphingosine 1-phosphate receptor 2 antagonist | 0.127 0.08 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.482 | 0.235 | GABA C receptor agonist | 0.235 0.015 CHEMBL226396 0.169 0.028 CHEMBL4525761 | CHEMBL226396 | |
| 0.009 | 0.474 | 0.095 | Pim-3 kinase inhibitor | 0.095 0.051 CHEMBL226396 | CHEMBL226396 | |
| 0.025 | 0.493 | 0.427 | Angiogenesis stimulant | 0.292 0.052 CHEMBL3526318 0.304 0.048 CHEMBL3527549 0.414 0.019 CHEMBL3526912 0.427 0.018 CHEMBL3527548 | CHEMBL3527548 | |
| 0.035 | 0.502 | 0.226 | Nitric oxide antagonist | 0.226 0.059 CHEMBL3526912 0.214 0.063 CHEMBL3527548 | CHEMBL3526912 | |
| 0.027 | 0.496 | 0.07 | Transcription factor RelA inhibitor | 0.07 0.03 CHEMBL4525761 | CHEMBL4525761 | |
| 0.005 | 0.484 | 0.304 | Phosphodiesterase 3B inhibitor | 0.282 0.004 CHEMBL3527205 0.304 0.004 CHEMBL3526210 | CHEMBL3526210 | |
| 0.042 | 0.525 | 0.149 | Interferon gamma antagonist | 0.149 0.079 CHEMBL4525761 | CHEMBL4525761 | |
| 0.012 | 0.506 | 0.057 | Vanilloid 3 antagonist | 0.057 0.005 CHEMBL4525761 | CHEMBL4525761 | |
| 0.038 | 0.535 | 0.152 | Focal adhesion kinase 2 inhibitor | 0.152 0.128 CHEMBL226396 | CHEMBL226396 | |
| 0.024 | 0.526 | 0.103 | Bromodomain-containing protein 2 inhibitor | 0.103 0.037 CHEMBL4525761 | CHEMBL4525761 | |
| 0.035 | 0.539 | 0.137 | Adenylate cyclase stimulant | 0.137 0.086 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.515 | 0.031 | Hedgehog signaling activator | 0.031 0.011 CHEMBL4525761 | CHEMBL4525761 | |
| 0.03 | 0.536 | 0.334 | Antioxidant | 0.334 0.051 CHEMBL3526912 0.334 0.051 CHEMBL3527548 | CHEMBL3527548 | |
| 0.018 | 0.525 | 0.147 | AMP-activated protein kinase stimulant | 0.147 0.03 CHEMBL4525761 | CHEMBL4525761 | |
| 0.012 | 0.519 | 0.097 | Glutamate (mGluR7) antagonist | 0.097 0.012 CHEMBL4525761 | CHEMBL4525761 | |
| 0.015 | 0.526 | 0.115 | Protein kinase C gamma inhibitor | 0.115 0.056 CHEMBL226396 | CHEMBL226396 | |
| 0.007 | 0.523 | 0.053 | Lysophosphatidic acid 3 receptor antagonist | 0.053 0.031 CHEMBL4525761 | CHEMBL4525761 | |
| 0.047 | 0.569 | 0.246 | Gastrin inhibitor | 0.246 0.084 CHEMBL4525761 | CHEMBL4525761 | |
| 0.06 | 0.589 | 0.205 | 5 Hydroxytryptamine release stimulant | 0.205 0.117 CHEMBL4525761 | CHEMBL4525761 | |
| 0.016 | 0.548 | 0.16 | Lipid peroxidase inhibitor | 0.136 0.079 CHEMBL3526912 0.16 0.062 CHEMBL3527548 | CHEMBL3527548 | |
| 0.09 | 0.625 | 0.176 | 5 Hydroxytryptamine 3E antagonist | 0.176 0.116 CHEMBL226396 | CHEMBL226396 | |
| 0.019 | 0.557 | 0.069 | Glutamate (mGluR6) antagonist | 0.069 0.042 CHEMBL4525761 | CHEMBL4525761 | |
| 0.004 | 0.549 | 0.073 | Antineoplastic antibiotic | 0.069 0.066 CHEMBL3526912 0.073 0.062 CHEMBL3527548 | CHEMBL3527548 | |
| 0.039 | 0.585 | 0.129 | Sphingosine 1-phosphate receptor 5 antagonist | 0.129 0.101 CHEMBL4525761 | CHEMBL4525761 | |
| 0.069 | 0.62 | 0.219 | Tyrosine 3 hydroxylase inhibitor | 0.213 0.113 CHEMBL226396 0.219 0.105 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.57 | 0.173 | Mannose-6-phosphate isomerase inhibitor | 0.173 0.047 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.562 | 0.22 | Phosphodiesterase III inhibitor | 0.218 0.005 CHEMBL3527205 0.22 0.005 CHEMBL3526210 | CHEMBL3526210 | |
| 0.017 | 0.571 | 0.231 | Thrombolytic | 0.211 0.047 CHEMBL3526318 0.231 0.039 CHEMBL3527549 0.167 0.07 CHEMBL3526912 0.167 0.07 CHEMBL3527548 | CHEMBL3527549 | |
| 0.018 | 0.572 | 0.152 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.152 0.139 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.568 | 0.14 | GABA C receptor antagonist | 0.14 0.036 CHEMBL226396 0.14 0.036 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.574 | 0.11 | Bone formation stimulant | 0.11 0.095 CHEMBL3527549 | CHEMBL3527549 | |
| 0.005 | 0.565 | 0.069 | Alcohol oxidase inhibitor | 0.069 0.03 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.573 | 0.139 | Diuretic | 0.139 0.086 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.576 | 0.144 | Cytidine deaminase inhibitor | 0.144 0.08 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.584 | 0.162 | Insulin sensitizer | 0.162 0.116 CHEMBL4525761 | CHEMBL4525761 | |
| 0.031 | 0.602 | 0.19 | Interleukin agonist | 0.19 0.13 CHEMBL3527548 | CHEMBL3527548 | |
| 0.011 | 0.582 | 0.05 | Antibiotic Aminoglycoside-like | 0.049 0.014 CHEMBL3526912 0.05 0.013 CHEMBL3527548 | CHEMBL3527548 | |
| 0.034 | 0.612 | 0.174 | Neurotrophic factor enhancer | 0.174 0.105 CHEMBL4525761 | CHEMBL4525761 | |
| 0.004 | 0.585 | 0.065 | Dopamine D1 agonist | 0.065 0.004 CHEMBL4525761 | CHEMBL4525761 | |
| 0.055 | 0.644 | 0.3 | Calcium channel activator | 0.3 0.091 CHEMBL4525761 | CHEMBL4525761 | |
| 0.023 | 0.612 | 0.302 | Aldehyde oxidase inhibitor | 0.302 0.066 CHEMBL4525761 | CHEMBL4525761 | |
| 0.024 | 0.615 | 0.097 | Phosphodiesterase 6D inhibitor | 0.097 0.059 CHEMBL4525761 0.091 0.072 CHEMBL3527548 | CHEMBL4525761 | |
| 0.019 | 0.614 | 0.103 | Acetylcholine release stimulant | 0.103 0.08 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.615 | 0.056 | Fatty acid synthase inhibitor | 0.056 0.041 CHEMBL4525761 | CHEMBL4525761 | |
| 0.046 | 0.656 | 0.162 | Death-associated protein kinase 2 inhibitor | 0.162 0.081 CHEMBL4525761 | CHEMBL4525761 | |
| 0.018 | 0.628 | 0.101 | Cell adhesion inhibitor | 0.101 0.088 CHEMBL3527548 | CHEMBL3527548 | |
| 0.015 | 0.626 | 0.113 | Glycine receptor agonist | 0.113 0.015 CHEMBL4525761 | CHEMBL4525761 | |
| 0.005 | 0.626 | 0.085 | Check point kinase 2 inhibitor | 0.085 0.079 CHEMBL226396 | CHEMBL226396 | |
| 0.011 | 0.633 | 0.098 | Ferrochelatase inhibitor | 0.098 0.073 CHEMBL226396 0.098 0.073 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.636 | 0.101 | Beta glucuronidase inhibitor | 0.101 0.069 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.637 | 0.15 | Cystathionine beta-synthase inhibitor | 0.15 0.041 CHEMBL4525761 | CHEMBL4525761 | |
| 0.017 | 0.645 | 0.111 | DOPA decarboxylase inhibitor | 0.111 0.056 CHEMBL4525761 | CHEMBL4525761 | |
| 0.012 | 0.643 | 0.115 | UDP-glucose 4-epimerase inhibitor | 0.115 0.047 CHEMBL4525761 | CHEMBL4525761 | |
| 0.001 | 0.633 | 0.06 | Uridine phosphorylase inhibitor | 0.06 0.005 CHEMBL4525761 | CHEMBL4525761 | |
| 0.011 | 0.643 | 0.085 | Creatine kinase inhibitor | 0.085 0.079 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.652 | 0.113 | Keratolytic | 0.113 0.024 CHEMBL4525761 | CHEMBL4525761 | |
| 0.017 | 0.662 | 0.26 | Succinate dehydrogenase inhibitor | 0.26 0.019 CHEMBL4525761 | CHEMBL4525761 | |
| 0.009 | 0.66 | 0.06 | Ryanodine receptor antagonist | 0.06 0.037 CHEMBL4525761 | CHEMBL4525761 | |
| 0.013 | 0.666 | 0.049 | Phosphodiesterase 6C inhibitor | 0.049 0.024 CHEMBL3527203 | CHEMBL3527203 | |
| 0.01 | 0.666 | 0.084 | Uric acid excretion stimulant | 0.084 0.075 CHEMBL3527548 | CHEMBL3527548 | |
| 0.008 | 0.672 | 0.071 | Protein 50S ribosomal subunit inhibitor | 0.064 0.028 CHEMBL3526912 0.071 0.024 CHEMBL3527548 | CHEMBL3527548 | |
| 0.016 | 0.682 | 0.165 | Vasodilator | 0.165 0.137 CHEMBL3527548 | CHEMBL3527548 | |
| 0.049 | 0.718 | 0.435 | Caspase 9 stimulant | 0.435 0.091 CHEMBL4525761 | CHEMBL4525761 | |
| 0.016 | 0.693 | 0.256 | Transcription factor NF kappa B inhibitor | 0.256 0.123 CHEMBL4525761 0.195 0.174 CHEMBL3526912 0.24 0.135 CHEMBL3527548 | CHEMBL4525761 | |
| 0.025 | 0.704 | 0.087 | Estrogen-related receptor beta agonist | 0.087 0.047 CHEMBL4525761 | CHEMBL4525761 | |
| 0.009 | 0.69 | 0.106 | Microtubule formation inhibitor | 0.106 0.08 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.689 | 0.046 | Glucose-6-phosphate isomerase inhibitor | 0.046 0.037 CHEMBL4525761 | CHEMBL4525761 | |
| 0.017 | 0.7 | 0.066 | Adenine nucleotide translocase inhibitor | 0.066 0.019 CHEMBL3527549 0.056 0.036 CHEMBL3526912 0.057 0.035 CHEMBL3527548 | CHEMBL3527549 | |
| 0.024 | 0.719 | 0.172 | Hexokinase inhibitor | 0.172 0.056 CHEMBL4525761 | CHEMBL4525761 | |
| 0.037 | 0.734 | 0.456 | Antiinflammatory | 0.448 0.111 CHEMBL3526912 0.456 0.107 CHEMBL3527548 | CHEMBL3527548 | |
| 0.022 | 0.72 | 0.133 | Vanilloid 1 agonist | 0.133 0.061 CHEMBL4525761 | CHEMBL4525761 | |
| 0.012 | 0.712 | 0.087 | Anabolic | 0.087 0.084 CHEMBL4525761 | CHEMBL4525761 | |
| 0.064 | 0.773 | 0.272 | Peptidyltransferase inhibitor | 0.201 0.098 CHEMBL3526318 0.217 0.079 CHEMBL3527549 0.267 0.04 CHEMBL3526912 0.272 0.037 CHEMBL3527548 | CHEMBL3527548 | |
| 0.015 | 0.725 | 0.079 | Vanilloid agonist | 0.079 0.074 CHEMBL4525761 | CHEMBL4525761 | |
| 0.009 | 0.733 | 0.2 | 12-Lipoxygenase inhibitor | 0.2 0.151 CHEMBL4525761 | CHEMBL4525761 | |
| 0.015 | 0.742 | 0.146 | Melanin inhibitor | 0.146 0.087 CHEMBL4525761 | CHEMBL4525761 | |
| 0.006 | 0.74 | 0.043 | Kainate receptor agonist | 0.043 0.025 CHEMBL4525761 | CHEMBL4525761 | |
| 0.071 | 0.81 | 0.275 | Calcium channel L-type activator | 0.275 0.18 CHEMBL4525761 | CHEMBL4525761 | |
| 0.007 | 0.746 | 0.117 | Cholesterol synthesis inhibitor | 0.117 0.068 CHEMBL4525761 | CHEMBL4525761 | |
| 0.006 | 0.745 | 0.164 | Anesthetic general | 0.164 0.1 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.753 | 0.163 | Arachidonic acid antagonist | 0.163 0.073 CHEMBL4525761 | CHEMBL4525761 | |
| 0.011 | 0.761 | 0.098 | Aminopeptidase B inhibitor | 0.098 0.066 CHEMBL3527549 | CHEMBL3527549 | |
| 0.018 | 0.777 | 0.159 | 3C-like protease (Human coronavirus) inhibitor | 0.159 0.088 CHEMBL4525761 | CHEMBL4525761 | |
| 0.016 | 0.78 | 0.106 | Photosensitizer | 0.106 0.077 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.776 | 0.168 | Alpha-N-acetylglucosaminidase inhibitor | 0.168 0.046 CHEMBL4525761 | CHEMBL4525761 | |
| 0.011 | 0.78 | 0.082 | Triose-phosphate isomerase inhibitor | 0.082 0.072 CHEMBL4525761 | CHEMBL4525761 | |
| 0.051 | 0.822 | 0.275 | 5 Hydroxytryptamine uptake stimulant | 0.275 0.06 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.778 | 0.262 | Free radical scavenger | 0.247 0.069 CHEMBL3526912 0.262 0.064 CHEMBL3527548 | CHEMBL3527548 | |
| 0.011 | 0.787 | 0.118 | Sphingosine 1-phosphate receptor 4 antagonist | 0.118 0.076 CHEMBL4525761 | CHEMBL4525761 | |
| 0.012 | 0.789 | 0.084 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.084 0.074 CHEMBL4525761 | CHEMBL4525761 | |
| 0.005 | 0.785 | 0.258 | Lipoxygenase inhibitor | 0.258 0.095 CHEMBL4525761 | CHEMBL4525761 | |
| 0.019 | 0.8 | 0.199 | Insulysin inhibitor | 0.199 0.158 CHEMBL4525761 | CHEMBL4525761 | |
| 0.008 | 0.789 | 0.105 | Toll-Like receptor 2 antagonist | 0.105 0.097 CHEMBL4525761 | CHEMBL4525761 | |
| 0.004 | 0.789 | 0.057 | Dopamine agonist | 0.057 0.054 CHEMBL4525761 | CHEMBL4525761 | |
| 0.01 | 0.803 | 0.218 | 15-Lipoxygenase inhibitor | 0.218 0.193 CHEMBL4525761 | CHEMBL4525761 | |
| 0.021 | 0.822 | 0.08 | Transcription factor NF kappa B stimulant | 0.077 0.076 CHEMBL3526912 0.08 0.07 CHEMBL3527548 | CHEMBL3527548 | |
| 0.03 | 0.834 | 0.114 | Factor V inhibitor | 0.113 0.047 CHEMBL3526318 0.114 0.046 CHEMBL3527549 | CHEMBL3527549 | |
| 0.01 | 0.816 | 0.087 | Bile acid receptor antagonist | 0.087 0.083 CHEMBL4525761 | CHEMBL4525761 | |
| 0.019 | 0.835 | 0.104 | Hematopoietic | 0.095 0.042 CHEMBL3526318 0.104 0.032 CHEMBL3527549 | CHEMBL3527549 | |
| 0.008 | 0.832 | 0.209 | Antithrombotic | 0.209 0.167 CHEMBL3527548 | CHEMBL3527548 | |
| 0.006 | 0.845 | 0.107 | Chelator | 0.107 0.068 CHEMBL3527549 | CHEMBL3527549 | |
| 0.008 | 0.857 | 0.137 | Neurotensin receptor agonist | 0.137 0.136 CHEMBL4525761 | CHEMBL4525761 | |
| 0.019 | 0.9 | 0.301 | Apoptosis antagonist | 0.252 0.125 CHEMBL3526912 0.301 0.085 CHEMBL3527548 | CHEMBL3527548 | |
| 0.024 | 0.919 | 0.166 | Growth hormone agonist | 0.149 0.088 CHEMBL3526318 0.166 0.075 CHEMBL3527549 | CHEMBL3527549 | |
| 0.014 | 0.913 | 0.266 | Hepatoprotectant | 0.135 0.127 CHEMBL3527549 0.231 0.049 CHEMBL3526912 0.266 0.039 CHEMBL3527548 | CHEMBL3527548 | |
| 0.008 | 0.922 | 0.297 | Hypoglycemic | 0.283 0.059 CHEMBL3526912 0.297 0.054 CHEMBL3527548 | CHEMBL3527548 | |
| 0.015 | 0.929 | 0.062 | Heme oxygenase stimulant | 0.059 0.049 CHEMBL3527205 0.062 0.039 CHEMBL3526210 | CHEMBL3526210 | |
| 0.011 | 0.928 | 0.11 | Toll-Like receptor 4 antagonist | 0.107 0.058 CHEMBL3526912 0.11 0.055 CHEMBL3527548 | CHEMBL3527548 | |
| 0.02 | 0.944 | 0.347 | Sodium/bile acid cotransporter inhibitor | 0.337 0.049 CHEMBL3526318 0.347 0.042 CHEMBL3527549 | CHEMBL3527549 | |
| 0.031 | 0.957 | 0.381 | Interleukin 2 agonist | 0.221 0.155 CHEMBL3526318 0.247 0.121 CHEMBL3527549 0.371 0.037 CHEMBL3526912 0.381 0.034 CHEMBL3527548 | CHEMBL3527548 | |
| 0.008 | 0.938 | 0.132 | Histone deacetylase SIRT1 inhibitor | 0.132 0.078 CHEMBL3527549 | CHEMBL3527549 | |
| 0.005 | 0.937 | 0.434 | Cyclophilin D inhibitor | 0.434 0.074 CHEMBL3526912 0.419 0.08 CHEMBL3527548 | CHEMBL3526912 | |
| 0.004 | 0.952 | 0.202 | M17 leucyl aminopeptidase inhibitor | 0.202 0.032 CHEMBL4525761 | CHEMBL4525761 | |
| 0.003 | 0.957 | 0.183 | Selectin antagonist | 0.176 0.014 CHEMBL3526912 0.183 0.013 CHEMBL3527548 | CHEMBL3527548 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |