| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.964 | 0.001 | 0.964 | Histone deacetylase class I inhibitor | 0.364 0.004 CHEMBL4525771 0.078 0.01 CHEMBL3527526 0.893 0.002 CHEMBL3527527 0.439 0.003 CHEMBL3527525 0.8 0.002 CHEMBL3526395 0.266 0.004 CHEMBL3526942 0.178 0.005 CHEMBL3526396 0.11 0.007 CHEMBL3526943 | ||
| 0.963 | 0.001 | 0.963 | Histone deacetylase inhibitor | 0.463 0.003 CHEMBL4525771 0.144 0.009 CHEMBL3527526 0.895 0.002 CHEMBL3527527 0.465 0.003 CHEMBL3527525 0.836 0.002 CHEMBL3526395 0.079 0.031 CHEMBL3526397 0.319 0.004 CHEMBL3526942 0.249 0.005 CHEMBL3526396 0.182 0.006 CHEMBL3526943 | ||
| 0.877 | 0.003 | 0.995 | Histone deacetylase 1 inhibitor | 0.657 0.003 CHEMBL4525771 0.024 0.017 CHEMBL3527526 0.745 0.003 CHEMBL3527527 0.083 0.009 CHEMBL3527525 0.995 0.001 CHEMBL3526395 0.935 0.002 CHEMBL3526397 0.052 0.011 CHEMBL3526942 0.966 0.002 CHEMBL3526396 0.943 0.002 CHEMBL3526943 | CHEMBL3526395 | |
| 0.814 | 0.001 | 0.814 | Histone deacetylase 7 inhibitor | 0.276 0.003 CHEMBL4525771 0.127 0.006 CHEMBL3527526 0.606 0.002 CHEMBL3527527 0.214 0.004 CHEMBL3527525 0.059 0.016 CHEMBL3526395 0.135 0.005 CHEMBL3526942 | ||
| 0.807 | 0.002 | 0.862 | Histone deacetylase 8 inhibitor | 0.251 0.004 CHEMBL4525771 0.049 0.023 CHEMBL3527526 0.675 0.002 CHEMBL3527527 0.191 0.004 CHEMBL3527525 0.862 0.002 CHEMBL3526395 0.068 0.013 CHEMBL3526397 0.14 0.006 CHEMBL3526942 0.269 0.004 CHEMBL3526396 0.203 0.004 CHEMBL3526943 | CHEMBL3526395 | |
| 0.791 | 0.001 | 0.791 | Histone deacetylase 9 inhibitor | 0.278 0.003 CHEMBL4525771 0.091 0.007 CHEMBL3527526 0.607 0.002 CHEMBL3527527 0.194 0.004 CHEMBL3527525 0.054 0.014 CHEMBL3526395 0.12 0.005 CHEMBL3526942 | ||
| 0.722 | 0.003 | 0.995 | Histone deacetylase 2 inhibitor | 0.551 0.004 CHEMBL4525771 0.034 0.023 CHEMBL3527526 0.606 0.003 CHEMBL3527527 0.071 0.012 CHEMBL3527525 0.995 0.001 CHEMBL3526395 0.979 0.002 CHEMBL3526397 0.051 0.014 CHEMBL3526942 0.983 0.001 CHEMBL3526396 0.978 0.002 CHEMBL3526943 | CHEMBL3526395 | |
| 0.693 | 0.003 | 0.987 | Histone deacetylase class II inhibitor | 0.487 0.003 CHEMBL4525771 0.496 0.003 CHEMBL3527527 0.04 0.013 CHEMBL3527525 0.987 0.001 CHEMBL3526395 0.796 0.003 CHEMBL3526397 0.033 0.016 CHEMBL3526942 0.866 0.002 CHEMBL3526396 0.8 0.003 CHEMBL3526943 | CHEMBL3526395 | |
| 0.688 | 0.003 | 0.688 | Histone deacetylase 5 inhibitor | 0.548 0.003 CHEMBL4525771 0.042 0.019 CHEMBL3527526 0.557 0.003 CHEMBL3527527 0.077 0.012 CHEMBL3527525 0.373 0.004 CHEMBL3526395 0.059 0.014 CHEMBL3526942 | ||
| 0.655 | 0.003 | 0.655 | Histone deacetylase class IV inhibitor | 0.406 0.003 CHEMBL4525771 0.037 0.019 CHEMBL3527526 0.453 0.003 CHEMBL3527527 0.05 0.013 CHEMBL3527525 0.185 0.004 CHEMBL3526395 0.041 0.017 CHEMBL3526942 | ||
| 0.655 | 0.003 | 0.655 | Histone deacetylase 11 inhibitor | 0.406 0.003 CHEMBL4525771 0.037 0.019 CHEMBL3527526 0.453 0.003 CHEMBL3527527 0.05 0.013 CHEMBL3527525 0.185 0.004 CHEMBL3526395 0.041 0.017 CHEMBL3526942 | ||
| 0.644 | 0.003 | 0.972 | Histone deacetylase class IIa inhibitor | 0.493 0.003 CHEMBL4525771 0.031 0.023 CHEMBL3527526 0.5 0.003 CHEMBL3527527 0.063 0.012 CHEMBL3527525 0.972 0.001 CHEMBL3526395 0.94 0.002 CHEMBL3526397 0.049 0.014 CHEMBL3526942 0.946 0.002 CHEMBL3526396 0.939 0.002 CHEMBL3526943 | CHEMBL3526395 | |
| 0.64 | 0.003 | 0.995 | Histone deacetylase 3 inhibitor | 0.414 0.004 CHEMBL4525771 0.49 0.004 CHEMBL3527527 0.035 0.013 CHEMBL3527525 0.995 0.001 CHEMBL3526395 0.98 0.001 CHEMBL3526397 0.024 0.017 CHEMBL3526942 0.984 0.001 CHEMBL3526396 0.978 0.001 CHEMBL3526943 | CHEMBL3526395 | |
| 0.542 | 0.003 | 0.995 | Histone deacetylase class IIb inhibitor | 0.353 0.004 CHEMBL4525771 0.372 0.004 CHEMBL3527527 0.029 0.016 CHEMBL3527525 0.995 0.001 CHEMBL3526395 0.926 0.002 CHEMBL3526397 0.024 0.02 CHEMBL3526942 0.95 0.002 CHEMBL3526396 0.919 0.002 CHEMBL3526943 | CHEMBL3526395 | |
| 0.539 | 0.003 | 0.995 | Histone deacetylase 6 inhibitor | 0.351 0.004 CHEMBL4525771 0.369 0.004 CHEMBL3527527 0.029 0.016 CHEMBL3527525 0.995 0.001 CHEMBL3526395 0.927 0.002 CHEMBL3526397 0.023 0.02 CHEMBL3526942 0.952 0.002 CHEMBL3526396 0.92 0.002 CHEMBL3526943 | CHEMBL3526395 | |
| 0.531 | 0.003 | 0.531 | Histone deacetylase 10 inhibitor | 0.298 0.003 CHEMBL4525771 0.026 0.023 CHEMBL3527526 0.322 0.003 CHEMBL3527527 0.044 0.014 CHEMBL3527525 0.155 0.004 CHEMBL3526395 0.036 0.018 CHEMBL3526942 | ||
| 0.472 | 0.04 | 0.544 | Calcium channel L-type activator | 0.529 0.018 CHEMBL3527526 0.507 0.025 CHEMBL3527527 0.517 0.022 CHEMBL3527525 0.266 0.188 CHEMBL3526397 0.544 0.014 CHEMBL3526942 0.248 0.207 CHEMBL3526396 0.355 0.113 CHEMBL3526943 | CHEMBL3526942 | |
| 0.488 | 0.078 | 0.523 | Apoptosis agonist | 0.334 0.149 CHEMBL4525771 0.398 0.114 CHEMBL3527526 0.523 0.068 CHEMBL3527527 0.26 0.204 CHEMBL3527525 0.249 0.216 CHEMBL3526395 0.344 0.142 CHEMBL3526942 | CHEMBL3527527 | |
| 0.382 | 0.003 | 0.99 | Histone deacetylase 4 inhibitor | 0.244 0.004 CHEMBL4525771 0.267 0.004 CHEMBL3527527 0.045 0.014 CHEMBL3527525 0.99 0.001 CHEMBL3526395 0.984 0.001 CHEMBL3526397 0.038 0.019 CHEMBL3526942 0.986 0.001 CHEMBL3526396 0.983 0.001 CHEMBL3526943 | CHEMBL3526395 | |
| 0.357 | 0.009 | 0.559 | 5 Hydroxytryptamine 1E antagonist | 0.367 0.007 CHEMBL3527526 0.335 0.014 CHEMBL3527527 0.559 0.003 CHEMBL3527525 0.461 0.004 CHEMBL3526942 | CHEMBL3527525 | |
| 0.375 | 0.027 | 0.375 | Insulysin inhibitor | 0.319 0.048 CHEMBL4525771 0.32 0.047 CHEMBL3527526 0.367 0.029 CHEMBL3527527 0.323 0.046 CHEMBL3527525 0.316 0.049 CHEMBL3526942 | ||
| 0.313 | 0.043 | 0.404 | Amyloid beta aggregation inhibitor | 0.147 0.11 CHEMBL4525771 0.37 0.03 CHEMBL3527526 0.37 0.03 CHEMBL3527527 0.351 0.034 CHEMBL3527525 0.404 0.024 CHEMBL3526942 0.162 0.1 CHEMBL3526943 | CHEMBL3526942 | |
| 0.313 | 0.048 | 0.313 | Tumour necrosis factor alpha release inhibitor | 0.304 0.052 CHEMBL3527527 | ||
| 0.287 | 0.032 | 0.347 | DNA methylase inhibitor | 0.142 0.125 CHEMBL3527526 0.347 0.017 CHEMBL3527527 0.197 0.081 CHEMBL3526942 | CHEMBL3527527 | |
| 0.277 | 0.035 | 0.334 | DNA methyltransferase I inhibitor | 0.334 0.017 CHEMBL3527527 0.16 0.094 CHEMBL3526942 | CHEMBL3527527 | |
| 0.225 | 0.004 | 0.243 | Myeloperoxidase inhibitor | 0.109 0.026 CHEMBL4525771 0.116 0.022 CHEMBL3527526 0.243 0.004 CHEMBL3527527 0.176 0.007 CHEMBL3527525 0.194 0.005 CHEMBL3526942 | CHEMBL3527527 | |
| 0.318 | 0.104 | 0.32 | Immunosuppressant | 0.318 0.104 CHEMBL4525771 0.237 0.16 CHEMBL3527526 0.32 0.103 CHEMBL3527527 | CHEMBL3527527 | |
| 0.214 | 0.006 | 0.445 | Prostaglandin EP2 antagonist | 0.445 0.004 CHEMBL3527526 0.194 0.007 CHEMBL3527527 0.207 0.006 CHEMBL3527525 0.085 0.024 CHEMBL3526397 0.186 0.007 CHEMBL3526942 | CHEMBL3527526 | |
| 0.19 | 0.004 | 0.19 | Botulinum neurotoxin type A inhibitor | 0.1 0.009 CHEMBL4525771 0.069 0.026 CHEMBL3527526 0.176 0.004 CHEMBL3527527 0.073 0.023 CHEMBL3527525 0.072 0.023 CHEMBL3526942 | ||
| 0.336 | 0.157 | 0.43 | Caspase 9 stimulant | 0.325 0.168 CHEMBL4525771 0.353 0.143 CHEMBL3527526 0.43 0.094 CHEMBL3527527 0.257 0.244 CHEMBL3526395 0.269 0.23 CHEMBL3526397 0.257 0.244 CHEMBL3526942 | CHEMBL3527527 | |
| 0.201 | 0.025 | 0.202 | Adenylate cyclase inhibitor | 0.165 0.036 CHEMBL3527526 0.202 0.025 CHEMBL3527527 0.141 0.051 CHEMBL3527525 0.148 0.046 CHEMBL3526942 | CHEMBL3527527 | |
| 0.158 | 0.017 | 0.158 | Metalloproteinase-2 inhibitor | 0.071 0.063 CHEMBL4525771 0.073 0.061 CHEMBL3527526 0.155 0.018 CHEMBL3527527 | ||
| 0.153 | 0.015 | 0.153 | Metalloproteinase-9 inhibitor | 0.071 0.054 CHEMBL4525771 0.151 0.015 CHEMBL3527527 | ||
| 0.232 | 0.113 | 0.305 | Lipoxygenase inhibitor | 0.237 0.109 CHEMBL3527526 0.305 0.069 CHEMBL3527527 0.174 0.172 CHEMBL3526942 | CHEMBL3527527 | |
| 0.13 | 0.011 | 0.13 | Aminopeptidase microsomal inhibitor | 0.112 0.014 CHEMBL4525771 0.114 0.014 CHEMBL3527527 0.072 0.029 CHEMBL3526395 | ||
| 0.257 | 0.139 | 0.392 | Calcium channel activator | 0.392 0.028 CHEMBL3527526 0.256 0.139 CHEMBL3527527 0.338 0.058 CHEMBL3527525 0.336 0.06 CHEMBL3526942 | CHEMBL3527526 | |
| 0.146 | 0.039 | 0.176 | 5-Lipoxygenase inhibitor | 0.094 0.069 CHEMBL3527526 0.176 0.03 CHEMBL3527527 | CHEMBL3527527 | |
| 0.117 | 0.012 | 0.233 | 5 Hydroxytryptamine 5A antagonist | 0.081 0.023 CHEMBL3527526 0.08 0.024 CHEMBL3527527 0.233 0.004 CHEMBL3527525 0.141 0.009 CHEMBL3526942 | CHEMBL3527525 | |
| 0.111 | 0.011 | 0.111 | Aminopeptidase N inhibitor | 0.095 0.014 CHEMBL4525771 0.095 0.014 CHEMBL3527527 0.051 0.03 CHEMBL3526395 | ||
| 0.108 | 0.014 | 0.221 | 5 Hydroxytryptamine 5 antagonist | 0.073 0.024 CHEMBL3527526 0.069 0.027 CHEMBL3527527 0.221 0.004 CHEMBL3527525 0.135 0.009 CHEMBL3526942 | CHEMBL3527525 | |
| 0.193 | 0.104 | 0.313 | Free radical scavenger | 0.313 0.048 CHEMBL3527526 0.284 0.056 CHEMBL3527527 0.175 0.119 CHEMBL3527525 0.18 0.114 CHEMBL3526397 0.28 0.057 CHEMBL3526942 0.152 0.143 CHEMBL3526943 | CHEMBL3527526 | |
| 0.209 | 0.122 | 0.418 | Transcription factor STAT3 inhibitor | 0.234 0.098 CHEMBL3527526 0.21 0.121 CHEMBL3527527 0.413 0.016 CHEMBL3527525 0.418 0.015 CHEMBL3526942 | CHEMBL3526942 | |
| 0.098 | 0.017 | 0.143 | NMDA receptor glycine site agonist | 0.138 0.005 CHEMBL3527526 0.071 0.035 CHEMBL3527527 0.143 0.005 CHEMBL3527525 0.122 0.008 CHEMBL3526942 | CHEMBL3527525 | |
| 0.124 | 0.05 | 0.16 | Chelator | 0.14 0.039 CHEMBL3527526 0.16 0.032 CHEMBL3527527 0.098 0.08 CHEMBL3527525 0.134 0.043 CHEMBL3526942 | CHEMBL3527527 | |
| 0.076 | 0.007 | 0.076 | Immunoglobulin Fc receptor antagonist | 0.055 0.038 CHEMBL4525771 0.067 0.014 CHEMBL3527527 0.057 0.031 CHEMBL3527525 0.052 0.051 CHEMBL3526942 | ||
| 0.075 | 0.01 | 0.075 | Adenylate cyclase 1 inhibitor | 0.045 0.033 CHEMBL4525771 0.045 0.033 CHEMBL3527526 0.061 0.017 CHEMBL3527527 | ||
| 0.092 | 0.03 | 0.092 | Matrix metalloproteinase inhibitor | 0.08 0.037 CHEMBL3527527 | ||
| 0.069 | 0.01 | 0.069 | Collagenase inhibitor | 0.064 0.012 CHEMBL4525771 0.063 0.014 CHEMBL3527527 0.054 0.025 CHEMBL3526395 | ||
| 0.084 | 0.026 | 0.202 | NMDA receptor agonist | 0.202 0.005 CHEMBL3527526 0.063 0.043 CHEMBL3527527 0.166 0.006 CHEMBL3527525 0.141 0.009 CHEMBL3526942 | CHEMBL3527526 | |
| 0.145 | 0.088 | 0.202 | Melanin inhibitor | 0.183 0.049 CHEMBL3527526 0.187 0.047 CHEMBL3527527 0.149 0.083 CHEMBL3527525 0.135 0.105 CHEMBL3526397 0.202 0.04 CHEMBL3526942 0.139 0.097 CHEMBL3526943 | CHEMBL3526942 | |
| 0.123 | 0.075 | 0.156 | Papain-like protease (SARS coronavirus) inhibitor | 0.124 0.073 CHEMBL4525771 0.136 0.051 CHEMBL3527526 0.137 0.049 CHEMBL3527527 0.144 0.04 CHEMBL3527525 0.156 0.028 CHEMBL3526942 0.119 0.083 CHEMBL3526943 | CHEMBL3526942 | |
| 0.151 | 0.104 | 0.206 | Death-associated protein kinase 2 inhibitor | 0.206 0.03 CHEMBL4525771 0.147 0.114 CHEMBL3527527 | CHEMBL4525771 | |
| 0.091 | 0.046 | 0.207 | Inducible nitric-oxide synthase inhibitor | 0.196 0.009 CHEMBL3527526 0.207 0.007 CHEMBL3527525 0.151 0.016 CHEMBL3526942 | CHEMBL3527525 | |
| 0.062 | 0.017 | 0.062 | Macrophage elastase inhibitor | 0.043 0.031 CHEMBL4525771 0.053 0.023 CHEMBL3527527 | ||
| 0.149 | 0.108 | 0.191 | Catenin beta inhibitor | 0.191 0.04 CHEMBL3527526 0.165 0.074 CHEMBL3527527 0.168 0.07 CHEMBL3527525 0.185 0.046 CHEMBL3526942 | CHEMBL3527526 | |
| 0.05 | 0.01 | 0.05 | ADAM10 endopeptidase inhibitor | 0.046 0.012 CHEMBL4525771 0.043 0.013 CHEMBL3527527 0.044 0.013 CHEMBL3526395 | ||
| 0.19 | 0.152 | 0.43 | Transcription factor STAT inhibitor | 0.212 0.122 CHEMBL3527526 0.187 0.157 CHEMBL3527527 0.43 0.014 CHEMBL3527525 0.43 0.014 CHEMBL3526942 | CHEMBL3526942 | |
| 0.065 | 0.028 | 0.065 | Matrix metalloproteinase 1 inhibitor | 0.062 0.03 CHEMBL3527527 | ||
| 0.076 | 0.041 | 0.099 | Phenylalanine 4-hydroxylase inhibitor | 0.073 0.044 CHEMBL3527526 0.099 0.026 CHEMBL3527527 | CHEMBL3527527 | |
| 0.107 | 0.073 | 0.107 | Interleukin 1b antagonist | 0.101 0.08 CHEMBL3527526 0.098 0.083 CHEMBL3527527 | ||
| 0.097 | 0.063 | 0.097 | Sphingomyelinase inhibitor | |||
| 0.042 | 0.014 | 0.062 | Melatonin 2 agonist | 0.053 0.009 CHEMBL3527526 0.041 0.015 CHEMBL3527527 0.062 0.007 CHEMBL3527525 0.056 0.009 CHEMBL3526942 | CHEMBL3527525 | |
| 0.17 | 0.143 | 0.304 | Antioxidant | 0.304 0.06 CHEMBL3527526 0.256 0.081 CHEMBL3527527 0.17 0.142 CHEMBL3527525 0.188 0.124 CHEMBL3526397 0.271 0.074 CHEMBL3526942 | CHEMBL3527526 | |
| 0.04 | 0.015 | 0.059 | Melatonin 1 agonist | 0.053 0.009 CHEMBL3527526 0.036 0.019 CHEMBL3527527 0.059 0.007 CHEMBL3527525 0.048 0.01 CHEMBL3526942 | CHEMBL3527525 | |
| 0.039 | 0.016 | 0.049 | Melatonin agonist | 0.043 0.013 CHEMBL3527526 0.035 0.02 CHEMBL3527527 0.049 0.01 CHEMBL3527525 0.04 0.015 CHEMBL3526942 | CHEMBL3527525 | |
| 0.059 | 0.037 | 0.114 | Potassium channel Kv1.5 blocker | 0.098 0.019 CHEMBL3527526 0.114 0.014 CHEMBL3527525 0.079 0.025 CHEMBL3526942 | CHEMBL3527525 | |
| 0.028 | 0.008 | 0.041 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.041 0.005 CHEMBL3527527 | CHEMBL3527527 | |
| 0.032 | 0.015 | 0.04 | Melatonin antagonist | 0.025 0.024 CHEMBL3527526 0.04 0.01 CHEMBL3527525 0.028 0.02 CHEMBL3526942 | CHEMBL3527525 | |
| 0.076 | 0.064 | 0.095 | Glycine receptor antagonist | 0.095 0.037 CHEMBL3527526 0.092 0.04 CHEMBL3527525 | CHEMBL3527526 | |
| 0.036 | 0.026 | 0.044 | Inosine monophosphate dehydrogenase inhibitor | 0.044 0.018 CHEMBL3527527 | CHEMBL3527527 | |
| 0.124 | 0.114 | 0.161 | Adenylate cyclase stimulant | 0.161 0.047 CHEMBL3527526 0.137 0.086 CHEMBL3527527 0.135 0.09 CHEMBL3527525 0.151 0.06 CHEMBL3526942 | CHEMBL3527526 | |
| 0.03 | 0.021 | 0.03 | Peptide deformylase inhibitor | |||
| 0.047 | 0.044 | 0.051 | Factor III inhibitor | 0.051 0.033 CHEMBL3527527 | CHEMBL3527527 | |
| 0.087 | 0.084 | 0.186 | Nitric-oxide synthase inhibitor | 0.152 0.022 CHEMBL3527526 0.186 0.012 CHEMBL3527525 0.129 0.033 CHEMBL3526942 | CHEMBL3527525 | |
| 0.016 | 0.017 | 0.02 | Melatonin 1 antagonist | 0.02 0.012 CHEMBL3527525 | CHEMBL3527525 | |
| 0.176 | 0.177 | 0.236 | 12-Lipoxygenase inhibitor | 0.236 0.117 CHEMBL3527527 0.198 0.153 CHEMBL3526942 | CHEMBL3527527 | |
| 0.02 | 0.022 | 0.047 | NMDA receptor glycine site antagonist | 0.047 0.006 CHEMBL3527526 0.041 0.008 CHEMBL3527525 0.038 0.009 CHEMBL3526942 | CHEMBL3527526 | |
| 0.108 | 0.12 | 0.164 | Vanilloid 1 agonist | 0.153 0.035 CHEMBL3527526 0.118 0.092 CHEMBL3527527 0.148 0.04 CHEMBL3527525 0.164 0.027 CHEMBL3526942 | CHEMBL3526942 | |
| 0.158 | 0.172 | 0.237 | Peptidyltransferase inhibitor | 0.199 0.1 CHEMBL3527526 0.18 0.128 CHEMBL3527527 0.215 0.081 CHEMBL3527525 0.163 0.162 CHEMBL3526397 0.237 0.06 CHEMBL3526942 0.194 0.108 CHEMBL3526396 0.198 0.101 CHEMBL3526943 | CHEMBL3526942 | |
| 0.087 | 0.101 | 0.094 | GABA C receptor antagonist | 0.094 0.088 CHEMBL3527526 | CHEMBL3527526 | |
| 0.079 | 0.094 | 0.148 | Carbonic anhydrase III inhibitor | 0.148 0.029 CHEMBL3527526 0.125 0.041 CHEMBL3527527 0.121 0.044 CHEMBL3526942 | CHEMBL3527526 | |
| 0.09 | 0.108 | 0.173 | TRPA1 agonist | 0.173 0.018 CHEMBL3527526 0.153 0.029 CHEMBL3527525 0.149 0.032 CHEMBL3526942 | CHEMBL3527526 | |
| 0.101 | 0.12 | 0.123 | Antibacterial (Helicobacter pylori) | 0.123 0.077 CHEMBL3527526 | CHEMBL3527526 | |
| 0.036 | 0.056 | 0.152 | Prostaglandin E2 antagonist | 0.152 0.009 CHEMBL3527526 0.047 0.039 CHEMBL3527525 | CHEMBL3527526 | |
| 0.204 | 0.225 | 0.278 | Antibacterial | 0.278 0.152 CHEMBL4525771 0.244 0.183 CHEMBL3527527 0.26 0.168 CHEMBL3526942 | CHEMBL4525771 | |
| 0.167 | 0.189 | 0.276 | Neuropeptide Y2 antagonist | 0.219 0.09 CHEMBL3527526 0.276 0.033 CHEMBL3527525 0.178 0.163 CHEMBL3526397 0.256 0.051 CHEMBL3526942 0.237 0.069 CHEMBL3526396 0.217 0.092 CHEMBL3526943 | CHEMBL3527525 | |
| 0.025 | 0.049 | 0.062 | Melanocortin 1 antagonist | 0.062 0.016 CHEMBL3527525 0.037 0.027 CHEMBL3526942 | CHEMBL3527525 | |
| 0.073 | 0.098 | 0.087 | Vanilloid agonist | 0.079 0.073 CHEMBL3527526 0.079 0.072 CHEMBL3527527 0.079 0.074 CHEMBL3527525 0.087 0.053 CHEMBL3526942 | CHEMBL3526942 | |
| 0.015 | 0.049 | 0.121 | Urotensin II agonist | 0.121 0.002 CHEMBL4525771 | CHEMBL4525771 | |
| 0.046 | 0.083 | 0.089 | 5 Hydroxytryptamine 1F antagonist | 0.089 0.037 CHEMBL3527525 | CHEMBL3527525 | |
| 0.061 | 0.1 | 0.373 | NMDA receptor antagonist | 0.218 0.012 CHEMBL3527526 0.085 0.059 CHEMBL3527527 0.249 0.009 CHEMBL3527525 0.373 0.005 CHEMBL3526942 | CHEMBL3526942 | |
| 0.175 | 0.214 | 0.223 | Caspase 3 stimulant | 0.223 0.139 CHEMBL3527527 | CHEMBL3527527 | |
| 0.055 | 0.096 | 0.103 | Somatostatin 1 agonist | 0.069 0.066 CHEMBL3527526 0.097 0.036 CHEMBL3527525 0.103 0.032 CHEMBL3526942 | CHEMBL3526942 | |
| 0.065 | 0.114 | 0.1 | Aminoacyl-tRNA synthetase inhibitor | 0.1 0.045 CHEMBL3527526 0.089 0.061 CHEMBL3527525 0.089 0.06 CHEMBL3526942 | CHEMBL3527526 | |
| 0.234 | 0.285 | 0.268 | Antiinflammatory | 0.259 0.257 CHEMBL3527526 0.268 0.248 CHEMBL3527527 | CHEMBL3527527 | |
| 0.069 | 0.121 | 0.087 | 3C-Like protease (SARS coronavirus) inhibitor | 0.087 0.052 CHEMBL3527525 0.08 0.068 CHEMBL3526942 | CHEMBL3527525 | |
| 0.051 | 0.104 | 0.096 | HIV-1 integrase inhibitor | 0.096 0.027 CHEMBL3527526 0.065 0.057 CHEMBL3527527 0.083 0.036 CHEMBL3526397 | CHEMBL3527526 | |
| 0.038 | 0.092 | 0.096 | Thromboxane synthase inhibitor | 0.096 0.007 CHEMBL3527526 | CHEMBL3527526 | |
| 0.064 | 0.122 | 0.162 | Gastric antisecretory | 0.162 0.022 CHEMBL3527526 | CHEMBL3527526 | |
| 0.034 | 0.096 | 0.045 | Bombesin 2 receptor antagonist | 0.045 0.041 CHEMBL3527525 | CHEMBL3527525 | |
| 0.065 | 0.131 | 0.079 | Ca(v)3.1 blocker | 0.076 0.074 CHEMBL3527526 0.079 0.065 CHEMBL3527525 | CHEMBL3527525 | |
| 0.087 | 0.156 | 0.132 | Transcription factor STAT6 inhibitor | 0.132 0.041 CHEMBL3527525 0.125 0.052 CHEMBL3526942 | CHEMBL3527525 | |
| 0.085 | 0.156 | 0.124 | Peroxidase inhibitor | 0.124 0.096 CHEMBL3527527 | CHEMBL3527527 | |
| 0.036 | 0.11 | 0.052 | Vanilloid 2 antagonist | 0.052 0.036 CHEMBL3526942 | CHEMBL3526942 | |
| 0.117 | 0.193 | 0.298 | Antiamyloidogenic | 0.266 0.064 CHEMBL3527526 0.157 0.138 CHEMBL3527527 0.227 0.082 CHEMBL3527525 0.298 0.052 CHEMBL3526942 | CHEMBL3526942 | |
| 0.176 | 0.252 | 0.265 | Transcription factor inhibitor | 0.265 0.176 CHEMBL3527525 | CHEMBL3527525 | |
| 0.012 | 0.089 | 0.034 | Kainate receptor 2 antagonist | 0.034 0.026 CHEMBL3527526 | CHEMBL3527526 | |
| 0.054 | 0.13 | 0.084 | Butyrylcholinesterase inhibitor | 0.084 0.077 CHEMBL3527525 | CHEMBL3527525 | |
| 0.037 | 0.116 | 0.118 | Carbonic anhydrase VA inhibitor | 0.118 0.019 CHEMBL3527526 | CHEMBL3527526 | |
| 0.148 | 0.23 | 0.205 | 5 Hydroxytryptamine 3E antagonist | 0.164 0.158 CHEMBL3527526 0.205 0.054 CHEMBL3527525 0.164 0.158 CHEMBL3526396 | CHEMBL3527525 | |
| 0.156 | 0.239 | 0.242 | Tyrosine 3 hydroxylase inhibitor | 0.242 0.077 CHEMBL3527526 0.186 0.162 CHEMBL3527525 0.242 0.077 CHEMBL3526397 0.216 0.108 CHEMBL3526942 0.196 0.143 CHEMBL3526396 0.207 0.123 CHEMBL3526943 | CHEMBL3526397 | |
| 0.008 | 0.093 | 0.049 | Prostaglandin EP3 antagonist | 0.049 0.01 CHEMBL3527526 0.038 0.015 CHEMBL3526397 | CHEMBL3527526 | |
| 0.044 | 0.129 | 0.069 | Beta 3 adrenoreceptor antagonist | 0.062 0.05 CHEMBL3527526 0.069 0.036 CHEMBL3526942 | CHEMBL3526942 | |
| 0.067 | 0.155 | 0.11 | Tubulin antagonist | 0.11 0.091 CHEMBL3527527 | CHEMBL3527527 | |
| 0.031 | 0.119 | 0.118 | Carbonic anhydrase V inhibitor | 0.118 0.022 CHEMBL3527526 | CHEMBL3527526 | |
| 0.097 | 0.185 | 0.152 | Nitric oxide antagonist | 0.136 0.11 CHEMBL3527526 0.129 0.121 CHEMBL3527527 0.152 0.093 CHEMBL3526397 0.131 0.118 CHEMBL3526943 | CHEMBL3526397 | |
| 0.02 | 0.111 | 0.044 | Melanocortin antagonist | 0.044 0.038 CHEMBL3527525 | CHEMBL3527525 | |
| 0.021 | 0.112 | 0.072 | NMDA receptor subunit 3B antagonist | 0.053 0.023 CHEMBL3527526 0.072 0.015 CHEMBL3526942 | CHEMBL3526942 | |
| 0.061 | 0.158 | 0.129 | DNA polymerase I inhibitor | 0.129 0.062 CHEMBL3527526 | CHEMBL3527526 | |
| 0.066 | 0.163 | 0.122 | Cyclooxygenase 1 inhibitor | 0.122 0.079 CHEMBL3527526 | CHEMBL3527526 | |
| 0.123 | 0.222 | 0.187 | DNA damaging | 0.187 0.127 CHEMBL3527526 | CHEMBL3527526 | |
| 0.015 | 0.115 | 0.033 | Thrombin receptor antagonist | 0.033 0.015 CHEMBL3527525 | CHEMBL3527525 | |
| 0.084 | 0.185 | 0.229 | Phospholipase A2 inhibitor | 0.229 0.03 CHEMBL3527526 0.196 0.045 CHEMBL3527525 0.22 0.033 CHEMBL3526942 | CHEMBL3527526 | |
| 0.084 | 0.186 | 0.166 | Psychostimulant | 0.166 0.103 CHEMBL3527526 0.159 0.108 CHEMBL3527525 0.151 0.115 CHEMBL3526942 | CHEMBL3527526 | |
| 0.014 | 0.117 | 0.043 | NMDA receptor subunit 3A antagonist | 0.041 0.024 CHEMBL3527526 0.043 0.023 CHEMBL3526942 | CHEMBL3526942 | |
| 0.029 | 0.136 | 0.065 | HIV-1 reverse transcriptase inhibitor | 0.065 0.054 CHEMBL3527526 | CHEMBL3527526 | |
| 0.092 | 0.204 | 0.23 | Interleukin antagonist | 0.197 0.086 CHEMBL3527526 0.18 0.096 CHEMBL3527525 0.23 0.07 CHEMBL3526942 | CHEMBL3526942 | |
| 0.099 | 0.212 | 0.138 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.138 0.097 CHEMBL4525771 | CHEMBL4525771 | |
| 0.011 | 0.125 | 0.022 | Retinoic acid gamma receptor agonist | 0.022 0.016 CHEMBL3527526 0.021 0.019 CHEMBL3526397 | CHEMBL3527526 | |
| 0.067 | 0.182 | 0.123 | Lipid peroxidase inhibitor | 0.119 0.094 CHEMBL3527526 0.123 0.09 CHEMBL3527527 0.117 0.097 CHEMBL3526942 | CHEMBL3527527 | |
| 0.051 | 0.167 | 0.084 | GABA B receptor agonist | 0.084 0.035 CHEMBL3527526 0.072 0.062 CHEMBL3527525 0.082 0.038 CHEMBL3526942 | CHEMBL3527526 | |
| 0.041 | 0.158 | 0.099 | Monophenol monooxygenase inhibitor | 0.099 0.077 CHEMBL3527527 0.088 0.085 CHEMBL3526942 | CHEMBL3527527 | |
| 0.14 | 0.259 | 0.571 | Vasodilator, peripheral | 0.571 0.019 CHEMBL3527526 0.253 0.125 CHEMBL3527525 0.207 0.167 CHEMBL3526397 0.243 0.133 CHEMBL3526942 | CHEMBL3527526 | |
| 0.017 | 0.14 | 0.149 | Prostaglandin antagonist | 0.149 0.01 CHEMBL3527526 | CHEMBL3527526 | |
| 0.018 | 0.146 | 0.047 | Histamine H2 receptor agonist | 0.047 0.024 CHEMBL3527525 | CHEMBL3527525 | |
| 0.064 | 0.195 | 0.115 | Adenylate kinase inhibitor | 0.115 0.048 CHEMBL3527526 | CHEMBL3527526 | |
| 0.014 | 0.148 | 0.079 | Carbonic anhydrase VB inhibitor | 0.079 0.023 CHEMBL3527526 | CHEMBL3527526 | |
| 0.084 | 0.221 | 0.191 | Growth hormone agonist | 0.136 0.1 CHEMBL3526395 0.166 0.075 CHEMBL3526397 0.128 0.11 CHEMBL3526942 0.191 0.062 CHEMBL3526396 0.185 0.065 CHEMBL3526943 | CHEMBL3526396 | |
| 0.042 | 0.179 | 0.15 | Carbonic anhydrase VI inhibitor | 0.15 0.021 CHEMBL3527526 0.08 0.057 CHEMBL3526942 | CHEMBL3527526 | |
| 0.144 | 0.287 | 0.304 | Apoptosis antagonist | 0.304 0.083 CHEMBL3527526 0.192 0.19 CHEMBL3527525 0.248 0.13 CHEMBL3526397 0.24 0.138 CHEMBL3526942 | CHEMBL3527526 | |
| 0.067 | 0.21 | 0.109 | Interleukin 1 antagonist | 0.109 0.107 CHEMBL3527526 | CHEMBL3527526 | |
| 0.085 | 0.229 | 0.294 | Insulin sensitizer | 0.294 0.017 CHEMBL3527526 0.187 0.087 CHEMBL3527525 0.166 0.112 CHEMBL3526397 0.208 0.065 CHEMBL3526942 | CHEMBL3527526 | |
| 0.105 | 0.25 | 0.236 | Calpain inhibitor | 0.168 0.151 CHEMBL3527526 0.236 0.079 CHEMBL3527525 0.194 0.119 CHEMBL3526942 | CHEMBL3527525 | |
| 0.019 | 0.165 | 0.073 | Acetylcholine M5 receptor antagonist | 0.073 0.028 CHEMBL3527525 0.056 0.048 CHEMBL3526942 | CHEMBL3527525 | |
| 0.013 | 0.162 | 0.054 | NMDA 2A receptor antagonist | 0.047 0.041 CHEMBL3527526 0.054 0.034 CHEMBL3526942 | CHEMBL3526942 | |
| 0.061 | 0.21 | 0.125 | Cyclooxygenase inhibitor | 0.125 0.093 CHEMBL3527526 | CHEMBL3527526 | |
| 0.08 | 0.232 | 0.172 | Neuropeptide Y1 antagonist | 0.151 0.064 CHEMBL3527526 0.172 0.037 CHEMBL3527525 0.165 0.045 CHEMBL3526942 | CHEMBL3527525 | |
| 0.032 | 0.183 | 0.137 | Calcium antagonist | 0.137 0.027 CHEMBL3527526 0.075 0.068 CHEMBL3527525 | CHEMBL3527526 | |
| 0.014 | 0.169 | 0.04 | Factor XIIIa inhibitor | 0.04 0.023 CHEMBL3527525 | CHEMBL3527525 | |
| 0.019 | 0.176 | 0.082 | 5 Hydroxytryptamine 1D antagonist | 0.082 0.03 CHEMBL3527525 | CHEMBL3527525 | |
| 0.049 | 0.208 | 0.106 | Cyclooxygenase 2 inhibitor | 0.106 0.097 CHEMBL3527526 | CHEMBL3527526 | |
| 0.023 | 0.183 | 0.058 | HIV-1 integrase (3'-Processing) inhibitor | 0.058 0.049 CHEMBL3527526 | CHEMBL3527526 | |
| 0.007 | 0.169 | 0.047 | Protease activated receptor 1 antagonist | 0.047 0.034 CHEMBL3527525 | CHEMBL3527525 | |
| 0.04 | 0.203 | 0.08 | Beta 2 adrenoreceptor agonist | 0.062 0.042 CHEMBL3527526 0.064 0.035 CHEMBL3527525 0.08 0.009 CHEMBL3526942 | CHEMBL3526942 | |
| 0.018 | 0.182 | 0.054 | Maillard reaction inhibitor | 0.054 0.039 CHEMBL3526942 | CHEMBL3526942 | |
| 0.013 | 0.182 | 0.051 | Glycine transporter 2 inhibitor | 0.051 0.03 CHEMBL3527526 0.047 0.032 CHEMBL3526942 | CHEMBL3527526 | |
| 0.11 | 0.28 | 0.171 | Heat shock protein 70 antagonist | 0.171 0.017 CHEMBL3527526 0.141 0.072 CHEMBL3527525 0.138 0.081 CHEMBL3526397 0.143 0.065 CHEMBL3526942 | CHEMBL3527526 | |
| 0.063 | 0.233 | 0.092 | Folate antagonist | 0.092 0.083 CHEMBL3527526 | CHEMBL3527526 | |
| 0.028 | 0.201 | 0.075 | Beta adrenoreceptor antagonist | 0.075 0.032 CHEMBL3527526 0.068 0.041 CHEMBL3526942 | CHEMBL3527526 | |
| 0.081 | 0.256 | 0.155 | Interleukin 6 antagonist | 0.155 0.082 CHEMBL3526395 0.14 0.106 CHEMBL3526397 0.136 0.113 CHEMBL3526396 0.143 0.101 CHEMBL3526943 | CHEMBL3526395 | |
| 0.019 | 0.194 | 0.066 | Beta 1 adrenoreceptor antagonist | 0.066 0.03 CHEMBL3527526 0.054 0.041 CHEMBL3526942 | CHEMBL3527526 | |
| 0.015 | 0.194 | 0.072 | Opioid delta receptor antagonist | 0.072 0.039 CHEMBL3526942 | CHEMBL3526942 | |
| 0.018 | 0.201 | 0.065 | 5 Hydroxytryptamine 1B antagonist | 0.065 0.046 CHEMBL3527525 | CHEMBL3527525 | |
| 0.019 | 0.204 | 0.05 | Beta 2 adrenoreceptor antagonist | 0.05 0.036 CHEMBL3527526 0.046 0.042 CHEMBL3526942 | CHEMBL3527526 | |
| 0.103 | 0.29 | 0.309 | Superoxide dismutase inhibitor | 0.309 0.047 CHEMBL3527526 0.288 0.055 CHEMBL3527525 0.308 0.048 CHEMBL3526942 | CHEMBL3527526 | |
| 0.015 | 0.206 | 0.07 | Opioid mu receptor antagonist | 0.07 0.046 CHEMBL3526942 0.058 0.056 CHEMBL3526943 | CHEMBL3526942 | |
| 0.071 | 0.263 | 0.124 | Sigma receptor agonist | 0.124 0.11 CHEMBL3526943 | CHEMBL3526943 | |
| 0.029 | 0.226 | 0.07 | Protease 3C (Human rhinovirus) inhibitor | 0.07 0.037 CHEMBL3527525 | CHEMBL3527525 | |
| 0.014 | 0.212 | 0.048 | Retinoic acid alpha receptor agonist | 0.048 0.016 CHEMBL3527526 0.047 0.017 CHEMBL3526397 | CHEMBL3527526 | |
| 0.011 | 0.212 | 0.097 | NMDA 2C receptor antagonist | 0.097 0.017 CHEMBL3527526 0.061 0.043 CHEMBL3527525 0.076 0.028 CHEMBL3526942 | CHEMBL3527526 | |
| 0.121 | 0.326 | 0.187 | Nitric-oxide synthase stimulant | 0.187 0.112 CHEMBL3527526 0.177 0.134 CHEMBL3527525 0.187 0.114 CHEMBL3526942 | CHEMBL3526942 | |
| 0.037 | 0.245 | 0.126 | Prolactin inhibitor | 0.126 0.034 CHEMBL3527526 0.088 0.069 CHEMBL3527525 0.095 0.06 CHEMBL3526942 | CHEMBL3527526 | |
| 0.037 | 0.246 | 0.079 | Opioid kappa receptor antagonist | 0.079 0.059 CHEMBL3526942 0.076 0.065 CHEMBL3526943 | CHEMBL3526942 | |
| 0.054 | 0.266 | 0.112 | Interleukin 12 antagonist | 0.088 0.078 CHEMBL3527525 0.112 0.037 CHEMBL3526942 | CHEMBL3526942 | |
| 0.007 | 0.222 | 0.042 | Prostaglandin EP4 antagonist | 0.042 0.01 CHEMBL3527526 | CHEMBL3527526 | |
| 0.006 | 0.225 | 0.028 | AMPA 3 receptor antagonist | 0.028 0.022 CHEMBL3527526 | CHEMBL3527526 | |
| 0.027 | 0.248 | 0.107 | M18 aspartyl aminopeptidase inhibitor | 0.107 0.083 CHEMBL3526942 | CHEMBL3526942 | |
| 0.039 | 0.261 | 0.092 | Alpha 2c adrenoreceptor antagonist | 0.092 0.074 CHEMBL3527525 | CHEMBL3527525 | |
| 0.038 | 0.262 | 0.112 | 5 Hydroxytryptamine 3A agonist | 0.112 0.063 CHEMBL3527525 | CHEMBL3527525 | |
| 0.048 | 0.274 | 0.102 | Carbonic anhydrase XV inhibitor | 0.102 0.064 CHEMBL3526942 | CHEMBL3526942 | |
| 0.05 | 0.276 | 0.158 | Mcl-1 antagonist | 0.142 0.097 CHEMBL3527526 0.133 0.109 CHEMBL3527525 0.158 0.082 CHEMBL3526942 | CHEMBL3526942 | |
| 0.023 | 0.249 | 0.091 | Carbonic anhydrase XIII inhibitor | 0.091 0.042 CHEMBL3527526 | CHEMBL3527526 | |
| 0.04 | 0.267 | 0.092 | Beta glucuronidase inhibitor | 0.092 0.084 CHEMBL3527526 | CHEMBL3527526 | |
| 0.051 | 0.279 | 0.147 | Angiogenesis stimulant | 0.147 0.124 CHEMBL3526942 | CHEMBL3526942 | |
| 0.008 | 0.238 | 0.032 | Retinoid X gamma receptor antagonist | 0.032 0.01 CHEMBL3527526 0.029 0.014 CHEMBL3526397 | CHEMBL3527526 | |
| 0.109 | 0.342 | 0.352 | Vasodilator, coronary | 0.352 0.054 CHEMBL3527526 0.258 0.126 CHEMBL3527525 0.263 0.122 CHEMBL3526942 | CHEMBL3527526 | |
| 0.133 | 0.37 | 0.2 | Ca(v)3.3 blocker | 0.2 0.192 CHEMBL3527525 | CHEMBL3527525 | |
| 0.035 | 0.272 | 0.126 | Ferrochelatase inhibitor | 0.126 0.05 CHEMBL3527526 0.107 0.064 CHEMBL3527525 | CHEMBL3527526 | |
| 0.004 | 0.244 | 0.02 | Retinoic acid alpha receptor antagonist | 0.02 0.014 CHEMBL3527526 | CHEMBL3527526 | |
| 0.03 | 0.275 | 0.089 | Opioid antagonist | 0.089 0.057 CHEMBL3526942 0.083 0.065 CHEMBL3526943 | CHEMBL3526942 | |
| 0.074 | 0.32 | 0.202 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.202 0.089 CHEMBL3527525 0.164 0.125 CHEMBL3526942 | CHEMBL3527525 | |
| 0.048 | 0.294 | 0.1 | Calcium channel N-type blocker | 0.1 0.096 CHEMBL3527525 | CHEMBL3527525 | |
| 0.008 | 0.258 | 0.046 | Phosphorylase inhibitor | 0.046 0.033 CHEMBL3527526 | CHEMBL3527526 | |
| 0.015 | 0.266 | 0.064 | 5 Hydroxytryptamine 2A agonist | 0.064 0.043 CHEMBL3527525 0.056 0.051 CHEMBL3526942 | CHEMBL3527525 | |
| 0.099 | 0.35 | 0.401 | Antithrombotic | 0.401 0.049 CHEMBL3527526 | CHEMBL3527526 | |
| 0.015 | 0.271 | 0.069 | Leukotriene antagonist | 0.069 0.041 CHEMBL3527526 | CHEMBL3527526 | |
| 0.064 | 0.32 | 0.207 | NOS3 expression enhancer | 0.207 0.038 CHEMBL3527526 0.204 0.039 CHEMBL3526397 | CHEMBL3527526 | |
| 0.02 | 0.284 | 0.049 | Beta adrenoreceptor agonist | 0.049 0.021 CHEMBL3526942 | CHEMBL3526942 | |
| 0.063 | 0.328 | 0.127 | GABA C receptor rho-2 antagonist | 0.127 0.111 CHEMBL3527526 | CHEMBL3527526 | |
| 0.027 | 0.291 | 0.052 | DNA helicase inhibitor | 0.052 0.043 CHEMBL3527526 | CHEMBL3527526 | |
| 0.109 | 0.373 | 0.167 | ErbB-1 antagonist | 0.167 0.139 CHEMBL3526942 | CHEMBL3526942 | |
| 0.011 | 0.278 | 0.06 | Thromboxane antagonist | 0.06 0.032 CHEMBL3527526 | CHEMBL3527526 | |
| 0.046 | 0.319 | 0.149 | Acetylcholine M1 receptor antagonist | 0.149 0.076 CHEMBL3527525 0.138 0.087 CHEMBL3526942 | CHEMBL3527525 | |
| 0.022 | 0.295 | 0.207 | MAO inhibitor | 0.1 0.091 CHEMBL3527526 0.153 0.059 CHEMBL3527525 0.207 0.039 CHEMBL3526942 | CHEMBL3526942 | |
| 0.008 | 0.292 | 0.055 | Thromboxane A2 antagonist | 0.055 0.032 CHEMBL3527526 | CHEMBL3527526 | |
| 0.004 | 0.288 | 0.023 | Prostaglandin D2 antagonist | 0.023 0.015 CHEMBL3527526 | CHEMBL3527526 | |
| 0.006 | 0.295 | 0.11 | NMDA 2 receptor antagonist | 0.073 0.049 CHEMBL3527526 0.11 0.027 CHEMBL3526942 | CHEMBL3526942 | |
| 0.107 | 0.396 | 0.226 | GABA C receptor rho-3 antagonist | 0.212 0.193 CHEMBL3527526 0.226 0.178 CHEMBL3526942 | CHEMBL3526942 | |
| 0.077 | 0.367 | 0.125 | Death-associated protein kinase 1 inhibitor | 0.125 0.098 CHEMBL4525771 | CHEMBL4525771 | |
| 0.089 | 0.378 | 0.243 | 15-Lipoxygenase inhibitor | 0.243 0.17 CHEMBL3527526 | CHEMBL3527526 | |
| 0.026 | 0.318 | 0.124 | Mediator release inhibitor | 0.124 0.044 CHEMBL3527526 0.104 0.065 CHEMBL3526942 | CHEMBL3527526 | |
| 0.075 | 0.371 | 0.34 | Transcription factor NF kappa B inhibitor | 0.34 0.08 CHEMBL3527526 0.282 0.105 CHEMBL3526942 | CHEMBL3527526 | |
| 0.023 | 0.323 | 0.068 | Calcium channel L-type blocker | 0.068 0.055 CHEMBL3527526 | CHEMBL3527526 | |
| 0.024 | 0.324 | 0.089 | Protein kinase C delta inhibitor | 0.089 0.064 CHEMBL3527525 0.08 0.076 CHEMBL3526942 | CHEMBL3527525 | |
| 0.104 | 0.404 | 0.178 | MAP kinase kinase 5 inhibitor | 0.178 0.066 CHEMBL4525771 | CHEMBL4525771 | |
| 0.029 | 0.33 | 0.16 | GABA C receptor agonist | 0.16 0.03 CHEMBL3527526 | CHEMBL3527526 | |
| 0.004 | 0.311 | 0.024 | Retinoid X beta receptor agonist | 0.024 0.011 CHEMBL3527526 | CHEMBL3527526 | |
| 0.019 | 0.328 | 0.076 | Analgesic, opioid | 0.076 0.053 CHEMBL3526943 | CHEMBL3526943 | |
| 0.085 | 0.398 | 0.184 | 5 Hydroxytryptamine release stimulant | 0.184 0.136 CHEMBL3527526 0.172 0.15 CHEMBL3527525 | CHEMBL3527526 | |
| 0.015 | 0.33 | 0.052 | Sphingosine 1-phosphate receptor 5 agonist | 0.052 0.042 CHEMBL3527526 | CHEMBL3527526 | |
| 0.032 | 0.348 | 0.123 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.123 0.113 CHEMBL3527525 | CHEMBL3527525 | |
| 0.039 | 0.356 | 0.119 | Calcium channel blocker | 0.119 0.088 CHEMBL3527526 0.109 0.1 CHEMBL3527525 | CHEMBL3527526 | |
| 0.051 | 0.37 | 0.199 | Interleukin agonist | 0.199 0.121 CHEMBL3527525 0.184 0.135 CHEMBL3526396 | CHEMBL3527525 | |
| 0.004 | 0.324 | 0.029 | Retinoid X gamma receptor agonist | 0.029 0.011 CHEMBL3527526 0.023 0.017 CHEMBL3526397 | CHEMBL3527526 | |
| 0.008 | 0.337 | 0.105 | MAO B inhibitor | 0.105 0.057 CHEMBL3526942 | CHEMBL3526942 | |
| 0.038 | 0.367 | 0.107 | Toll-Like receptor 2 antagonist | 0.103 0.1 CHEMBL3527526 0.107 0.094 CHEMBL3526942 | CHEMBL3526942 | |
| 0.039 | 0.369 | 0.119 | Estrogen antagonist | 0.101 0.096 CHEMBL3527526 0.109 0.077 CHEMBL3527527 0.113 0.069 CHEMBL3526397 0.116 0.063 CHEMBL3526942 0.119 0.058 CHEMBL3526943 | CHEMBL3526943 | |
| 0.014 | 0.344 | 0.096 | MAO A inhibitor | 0.096 0.067 CHEMBL3526942 | CHEMBL3526942 | |
| 0.061 | 0.392 | 0.326 | Cardiotonic | 0.208 0.111 CHEMBL3526395 0.315 0.05 CHEMBL3526397 0.326 0.046 CHEMBL3526396 0.292 0.06 CHEMBL3526943 | CHEMBL3526396 | |
| 0.062 | 0.394 | 0.186 | Thyroid hormone beta antagonist | 0.186 0.167 CHEMBL3527526 | CHEMBL3527526 | |
| 0.034 | 0.37 | 0.113 | Cathepsin H inhibitor | 0.113 0.085 CHEMBL3527525 | CHEMBL3527525 | |
| 0.052 | 0.389 | 0.119 | Sphingosine 1-phosphate receptor 2 antagonist | 0.119 0.099 CHEMBL3527526 | CHEMBL3527526 | |
| 0.123 | 0.471 | 0.247 | MAP kinase kinase 3 inhibitor | 0.247 0.034 CHEMBL4525771 0.185 0.171 CHEMBL3527525 0.188 0.163 CHEMBL3526396 | CHEMBL4525771 | |
| 0.051 | 0.403 | 0.226 | Vasodilator | 0.226 0.085 CHEMBL3527526 | CHEMBL3527526 | |
| 0.013 | 0.366 | 0.12 | Histidine decarboxylase inhibitor | 0.12 0.026 CHEMBL3527526 | CHEMBL3527526 | |
| 0.012 | 0.369 | 0.078 | Sphingosine 1-phosphate receptor 4 agonist | 0.078 0.038 CHEMBL3527526 | CHEMBL3527526 | |
| 0.059 | 0.417 | 0.149 | Phospholipase C inhibitor | 0.149 0.109 CHEMBL3527526 | CHEMBL3527526 | |
| 0.057 | 0.415 | 0.196 | Thyroid hormone antagonist | 0.196 0.165 CHEMBL3527526 | CHEMBL3527526 | |
| 0.027 | 0.399 | 0.141 | Thrombolytic | 0.141 0.089 CHEMBL3527526 | CHEMBL3527526 | |
| 0.037 | 0.412 | 0.134 | ABCA1 expression enhancer | 0.134 0.022 CHEMBL3527526 | CHEMBL3527526 | |
| 0.011 | 0.388 | 0.069 | Catalase inhibitor | 0.069 0.056 CHEMBL3527526 | CHEMBL3527526 | |
| 0.005 | 0.382 | 0.045 | Peroxisome proliferator-activated receptor alpha agonist | 0.045 0.036 CHEMBL3527526 | CHEMBL3527526 | |
| 0.016 | 0.394 | 0.081 | Protein kinase B gamma inhibitor | 0.081 0.045 CHEMBL3527525 | CHEMBL3527525 | |
| 0.05 | 0.428 | 0.227 | Thioredoxin glutathione reductase inhibitor | 0.227 0.15 CHEMBL3527525 0.209 0.165 CHEMBL3526942 | CHEMBL3527525 | |
| 0.082 | 0.462 | 0.291 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.291 0.071 CHEMBL4525771 | CHEMBL4525771 | |
| 0.006 | 0.386 | 0.322 | Antineoplastic antibiotic | 0.322 0.008 CHEMBL4525771 | CHEMBL4525771 | |
| 0.016 | 0.403 | 0.097 | Adrenaline agonist | 0.097 0.039 CHEMBL3526942 | CHEMBL3526942 | |
| 0.007 | 0.4 | 0.071 | Peroxisome proliferator-activated receptor gamma agonist | 0.071 0.048 CHEMBL3527526 | CHEMBL3527526 | |
| 0.067 | 0.462 | 0.23 | Gastrin inhibitor | 0.23 0.105 CHEMBL3527526 0.182 0.177 CHEMBL3526397 | CHEMBL3527526 | |
| 0.032 | 0.436 | 0.114 | Toll-Like receptor 4 antagonist | 0.114 0.05 CHEMBL3526397 | CHEMBL3526397 | |
| 0.018 | 0.426 | 0.078 | Peroxisome proliferator-activated receptor gamma antagonist | 0.078 0.037 CHEMBL3527526 | CHEMBL3527526 | |
| 0.048 | 0.463 | 0.134 | Hepatoprotectant | 0.134 0.128 CHEMBL3527526 | CHEMBL3527526 | |
| 0.019 | 0.434 | 0.086 | Ornithine decarboxylase inhibitor | 0.086 0.061 CHEMBL3527526 | CHEMBL3527526 | |
| 0.076 | 0.492 | 0.15 | Cyclin-dependent kinase 3 inhibitor | 0.15 0.095 CHEMBL4525771 | CHEMBL4525771 | |
| 0.041 | 0.464 | 0.148 | Succinate dehydrogenase inhibitor | 0.148 0.116 CHEMBL3527526 | CHEMBL3527526 | |
| 0.036 | 0.461 | 0.17 | Platelet aggregation inhibitor | 0.17 0.107 CHEMBL3527526 | CHEMBL3527526 | |
| 0.021 | 0.45 | 0.103 | Estrogen receptor beta antagonist | 0.09 0.083 CHEMBL3527527 0.098 0.068 CHEMBL3526942 0.103 0.059 CHEMBL3526943 | CHEMBL3526943 | |
| 0.03 | 0.462 | 0.221 | Spasmolytic | 0.215 0.108 CHEMBL3527526 0.198 0.121 CHEMBL3527525 0.221 0.105 CHEMBL3526942 | CHEMBL3526942 | |
| 0.012 | 0.447 | 0.269 | MAP3K7 inhibitor | 0.269 0.004 CHEMBL3527525 0.238 0.005 CHEMBL3526942 0.239 0.005 CHEMBL3526396 0.222 0.005 CHEMBL3526943 | CHEMBL3527525 | |
| 0.034 | 0.499 | 0.222 | Alpha-glucosidase inhibitor | 0.222 0.204 CHEMBL3526942 | CHEMBL3526942 | |
| 0.035 | 0.501 | 0.111 | Histone deacetylase SIRT1 inhibitor | 0.111 0.103 CHEMBL3527525 0.11 0.104 CHEMBL3526942 | CHEMBL3527525 | |
| 0.028 | 0.5 | 0.251 | Platelet antagonist | 0.251 0.072 CHEMBL3527526 | CHEMBL3527526 | |
| 0.005 | 0.482 | 0.053 | NMDA 2B receptor antagonist | 0.053 0.039 CHEMBL3526943 | CHEMBL3526943 | |
| 0.112 | 0.589 | 0.261 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.261 0.053 CHEMBL4525771 | CHEMBL4525771 | |
| 0.051 | 0.531 | 0.204 | Hypoglycemic | 0.204 0.108 CHEMBL3527526 | CHEMBL3527526 | |
| 0.008 | 0.496 | 0.091 | Protein-tyrosine phosphatase 1B inhibitor | 0.091 0.088 CHEMBL3527526 | CHEMBL3527526 | |
| 0.019 | 0.508 | 0.097 | Telomerase inhibitor | 0.097 0.035 CHEMBL3526397 0.096 0.035 CHEMBL3526396 0.082 0.043 CHEMBL3526943 | CHEMBL3526397 | |
| 0.057 | 0.552 | 0.153 | Neurotensin receptor agonist | 0.139 0.13 CHEMBL3527526 0.153 0.094 CHEMBL3526942 | CHEMBL3526942 | |
| 0.028 | 0.527 | 0.147 | Nav1.1 sodium channel blocker | 0.128 0.043 CHEMBL3526397 0.147 0.034 CHEMBL3526396 0.138 0.038 CHEMBL3526943 | CHEMBL3526396 | |
| 0.008 | 0.511 | 0.077 | Protein kinase C eta inhibitor | 0.077 0.025 CHEMBL4525771 | CHEMBL4525771 | |
| 0.024 | 0.537 | 0.122 | Amylase inhibitor | 0.122 0.08 CHEMBL3526397 | CHEMBL3526397 | |
| 0.011 | 0.561 | 0.1 | Cholesterol synthesis inhibitor | 0.1 0.088 CHEMBL3527526 | CHEMBL3527526 | |
| 0.028 | 0.596 | 0.243 | Platelet adhesion inhibitor | 0.243 0.052 CHEMBL3527526 0.147 0.11 CHEMBL3526397 | CHEMBL3527526 | |
| 0.051 | 0.631 | 0.196 | Sodium/bile acid cotransporter inhibitor | 0.196 0.193 CHEMBL3527526 | CHEMBL3527526 | |
| 0.014 | 0.603 | 0.089 | AMP-activated protein kinase stimulant | 0.089 0.088 CHEMBL3527526 | CHEMBL3527526 | |
| 0.018 | 0.612 | 0.092 | Thioredoxin inhibitor | 0.092 0.059 CHEMBL3526397 | CHEMBL3526397 | |
| 0.01 | 0.667 | 0.119 | Protein kinase C nu inhibitor | 0.119 0.094 CHEMBL4525771 | CHEMBL4525771 | |
| 0.027 | 0.687 | 0.21 | Cholesterol antagonist | 0.21 0.156 CHEMBL3527526 | CHEMBL3527526 | |
| 0.009 | 0.672 | 0.412 | Anticonvulsant | 0.154 0.125 CHEMBL3527525 0.19 0.091 CHEMBL3526397 0.412 0.02 CHEMBL3526396 0.215 0.073 CHEMBL3526943 | CHEMBL3526396 | |
| 0.007 | 0.68 | 0.135 | Protein-tyrosine phosphatase inhibitor | 0.135 0.095 CHEMBL3527526 | CHEMBL3527526 | |
| 0.005 | 0.696 | 0.096 | Anesthetic local | 0.096 0.086 CHEMBL3526397 | CHEMBL3526397 | |
| 0.01 | 0.71 | 0.254 | Hypolipemic | 0.254 0.065 CHEMBL3526397 | CHEMBL3526397 | |
| 0.013 | 0.72 | 0.183 | DNA synthesis inhibitor | 0.183 0.149 CHEMBL3527526 | CHEMBL3527526 | |
| 0.006 | 0.765 | 0.018 | Granulocyte colony stimulating factor receptor agonist | 0.018 0.016 CHEMBL3526397 | CHEMBL3526397 | |
| 0.008 | 0.776 | 0.158 | Protein kinase C mu inhibitor | 0.158 0.023 CHEMBL4525771 | CHEMBL4525771 | |
| 0.017 | 0.798 | 0.172 | MAP3K9 inhibitor | 0.172 0.033 CHEMBL4525771 | CHEMBL4525771 | |
| 0.009 | 0.798 | 0.144 | Sphingosine 1-phosphate receptor 5 antagonist | 0.144 0.072 CHEMBL3526397 0.127 0.108 CHEMBL3526396 | CHEMBL3526397 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |