| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.837 | 0.004 | 0.837 | Caspase 3 stimulant | 0.715 0.005 CHEMBL3527504 0.771 0.004 CHEMBL3526805 | ||
| 0.813 | 0.004 | 0.813 | 12-Lipoxygenase inhibitor | |||
| 0.819 | 0.014 | 0.85 | Apoptosis agonist | 0.85 0.011 CHEMBL3527504 0.823 0.014 CHEMBL3526805 | CHEMBL3527504 | |
| 0.787 | 0.007 | 0.787 | 15-Lipoxygenase inhibitor | |||
| 0.79 | 0.012 | 0.79 | Caspase 9 stimulant | 0.712 0.022 CHEMBL3527504 0.764 0.016 CHEMBL3526805 | ||
| 0.767 | 0.005 | 0.767 | Aldehyde oxidase inhibitor | |||
| 0.754 | 0.007 | 0.754 | Aryl hydrocarbon receptor agonist | 0.254 0.077 CHEMBL3527504 0.289 0.064 CHEMBL3526805 | ||
| 0.738 | 0.005 | 0.738 | Lipoxygenase inhibitor | 0.235 0.11 CHEMBL3526805 | ||
| 0.68 | 0.005 | 0.704 | Hypoxia-inducible factor 1 alpha inhibitor | 0.687 0.005 CHEMBL3527504 0.704 0.004 CHEMBL3526805 | CHEMBL3526805 | |
| 0.666 | 0.003 | 0.825 | Melanin inhibitor | 0.815 0.002 CHEMBL3527504 0.825 0.002 CHEMBL3526805 | CHEMBL3526805 | |
| 0.658 | 0.004 | 0.658 | Breast cancer-resistant protein inhibitor | 0.162 0.02 CHEMBL3527504 0.19 0.015 CHEMBL3526805 | ||
| 0.643 | 0.005 | 0.643 | Tubulin antagonist | 0.186 0.042 CHEMBL3527504 0.304 0.019 CHEMBL3526805 | ||
| 0.64 | 0.009 | 0.789 | Antioxidant | 0.789 0.004 CHEMBL3527504 0.751 0.005 CHEMBL3526805 | CHEMBL3527504 | |
| 0.625 | 0.008 | 0.731 | Histamine release inhibitor | 0.705 0.005 CHEMBL3527504 0.731 0.004 CHEMBL3526805 | CHEMBL3526805 | |
| 0.622 | 0.007 | 0.867 | Vasodilator, coronary | 0.833 0.003 CHEMBL3527504 0.867 0.003 CHEMBL3526805 | CHEMBL3526805 | |
| 0.608 | 0.004 | 0.708 | Hepatoprotectant | 0.706 0.004 CHEMBL3527504 0.708 0.004 CHEMBL3526805 | CHEMBL3526805 | |
| 0.59 | 0.005 | 0.623 | Topoisomerase II inhibitor | 0.623 0.004 CHEMBL3527504 0.569 0.005 CHEMBL3526805 | CHEMBL3527504 | |
| 0.581 | 0.002 | 0.581 | Histidine decarboxylase inhibitor | 0.173 0.016 CHEMBL3527504 0.19 0.014 CHEMBL3526805 | ||
| 0.571 | 0.004 | 0.828 | Amylase inhibitor | 0.828 0.001 CHEMBL3527504 0.801 0.002 CHEMBL3526805 | CHEMBL3527504 | |
| 0.612 | 0.051 | 0.822 | Alpha-glucosidase inhibitor | 0.819 0.016 CHEMBL3527504 0.822 0.016 CHEMBL3526805 | CHEMBL3526805 | |
| 0.587 | 0.033 | 0.841 | Transcription factor NF kappa B inhibitor | 0.841 0.01 CHEMBL3527504 0.841 0.01 CHEMBL3526805 | CHEMBL3526805 | |
| 0.552 | 0.005 | 0.552 | MAO A inhibitor | |||
| 0.55 | 0.006 | 0.55 | MAO inhibitor | |||
| 0.552 | 0.009 | 0.552 | Antimitotic | 0.289 0.047 CHEMBL3527504 0.394 0.024 CHEMBL3526805 | ||
| 0.54 | 0.006 | 0.54 | P-glycoprotein inhibitor | 0.417 0.014 CHEMBL3527504 0.432 0.013 CHEMBL3526805 | ||
| 0.536 | 0.006 | 0.536 | Pyruvate kinase inhibitor | 0.211 0.075 CHEMBL3527504 0.204 0.079 CHEMBL3526805 | ||
| 0.536 | 0.013 | 0.691 | Free radical scavenger | 0.691 0.005 CHEMBL3527504 0.652 0.006 CHEMBL3526805 | CHEMBL3527504 | |
| 0.533 | 0.019 | 0.637 | Spasmolytic | 0.575 0.015 CHEMBL3527504 0.637 0.01 CHEMBL3526805 | CHEMBL3526805 | |
| 0.501 | 0.02 | 0.599 | Apoptosis antagonist | 0.594 0.01 CHEMBL3527504 0.599 0.01 CHEMBL3526805 | CHEMBL3526805 | |
| 0.47 | 0.004 | 0.47 | NADPH oxidase inhibitor | 0.356 0.007 CHEMBL3527504 0.369 0.006 CHEMBL3526805 | ||
| 0.456 | 0.018 | 0.456 | Amyloid beta aggregation inhibitor | 0.408 0.024 CHEMBL3527504 0.321 0.041 CHEMBL3526805 | ||
| 0.44 | 0.006 | 0.44 | MAO B inhibitor | |||
| 0.476 | 0.047 | 0.476 | Prostaglandin dehydrogenase inhibitor | |||
| 0.432 | 0.01 | 0.736 | Monophenol monooxygenase inhibitor | 0.736 0.004 CHEMBL3527504 0.696 0.004 CHEMBL3526805 | CHEMBL3527504 | |
| 0.442 | 0.02 | 0.473 | DNA damaging | 0.463 0.018 CHEMBL3527504 0.473 0.017 CHEMBL3526805 | CHEMBL3526805 | |
| 0.418 | 0.007 | 0.528 | NOS3 expression enhancer | 0.528 0.005 CHEMBL3527504 0.472 0.005 CHEMBL3526805 | CHEMBL3527504 | |
| 0.431 | 0.022 | 0.606 | Nitric oxide antagonist | 0.606 0.009 CHEMBL3527504 0.558 0.012 CHEMBL3526805 | CHEMBL3527504 | |
| 0.396 | 0.005 | 0.427 | Aldehyde dehydrogenase inhibitor | 0.427 0.005 CHEMBL3527504 0.336 0.009 CHEMBL3526805 | CHEMBL3527504 | |
| 0.386 | 0.002 | 0.386 | Papain-like protease (SARS coronavirus) inhibitor | 0.253 0.005 CHEMBL3527504 0.24 0.005 CHEMBL3526805 | ||
| 0.383 | 0.002 | 0.383 | DOPA decarboxylase inhibitor | 0.2 0.007 CHEMBL3527504 0.163 0.016 CHEMBL3526805 | ||
| 0.402 | 0.023 | 0.485 | Vasodilator | 0.485 0.013 CHEMBL3527504 0.468 0.014 CHEMBL3526805 | CHEMBL3527504 | |
| 0.383 | 0.006 | 0.417 | Topoisomerase I inhibitor | 0.417 0.005 CHEMBL3527504 0.399 0.005 CHEMBL3526805 | CHEMBL3527504 | |
| 0.377 | 0.005 | 0.386 | Topoisomerase II alpha inhibitor | 0.386 0.005 CHEMBL3527504 0.36 0.005 CHEMBL3526805 | CHEMBL3527504 | |
| 0.372 | 0.008 | 0.372 | Acetylcholinesterase inhibitor | 0.128 0.071 CHEMBL3527504 0.162 0.048 CHEMBL3526805 | ||
| 0.39 | 0.027 | 0.39 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | |||
| 0.437 | 0.105 | 0.437 | DNA polymerase beta inhibitor | |||
| 0.343 | 0.013 | 0.343 | Bone formation stimulant | 0.271 0.021 CHEMBL3527504 0.252 0.024 CHEMBL3526805 | ||
| 0.343 | 0.014 | 0.418 | Lipid peroxidase inhibitor | 0.418 0.009 CHEMBL3527504 0.407 0.009 CHEMBL3526805 | CHEMBL3527504 | |
| 0.356 | 0.035 | 0.356 | Dyrk kinase inhibitor | |||
| 0.381 | 0.064 | 0.381 | Thioredoxin glutathione reductase inhibitor | |||
| 0.307 | 0.009 | 0.307 | Heat shock protein 90 antagonist | 0.125 0.105 CHEMBL3527504 0.118 0.117 CHEMBL3526805 | ||
| 0.301 | 0.004 | 0.301 | Macrophage migration inhibitory factor inhibitor | |||
| 0.304 | 0.018 | 0.304 | Cholinergic | |||
| 0.294 | 0.011 | 0.294 | CDC-like kinase 1 inhibitor | 0.115 0.1 CHEMBL3526805 | ||
| 0.289 | 0.016 | 0.289 | Heat shock protein 90 alpha antagonist | |||
| 0.358 | 0.098 | 0.7 | Antibacterial | 0.7 0.009 CHEMBL3527504 0.67 0.011 CHEMBL3526805 | CHEMBL3527504 | |
| 0.289 | 0.034 | 0.321 | RNA-directed DNA polymerase inhibitor | 0.321 0.028 CHEMBL3527504 0.236 0.059 CHEMBL3526805 | CHEMBL3527504 | |
| 0.378 | 0.125 | 0.378 | DNA directed DNA polymerase inhibitor | |||
| 0.359 | 0.108 | 0.436 | 5 Hydroxytryptamine release inhibitor | 0.436 0.058 CHEMBL3527504 0.418 0.068 CHEMBL3526805 | CHEMBL3527504 | |
| 0.313 | 0.066 | 0.313 | 5 Hydroxytryptamine release stimulant | 0.193 0.127 CHEMBL3527504 0.189 0.132 CHEMBL3526805 | ||
| 0.253 | 0.007 | 0.253 | Estrogen receptor beta antagonist | 0.118 0.034 CHEMBL3527504 | ||
| 0.278 | 0.045 | 0.278 | Clk dual-specificity kinase inhibitor | |||
| 0.238 | 0.008 | 0.238 | CF transmembrane conductance regulator agonist | 0.183 0.033 CHEMBL3527504 0.178 0.038 CHEMBL3526805 | ||
| 0.239 | 0.009 | 0.239 | Estrogen antagonist | 0.148 0.024 CHEMBL3527504 0.118 0.058 CHEMBL3526805 | ||
| 0.306 | 0.076 | 0.306 | Streptokinase A inhibitor | |||
| 0.356 | 0.127 | 0.356 | Transcription factor inhibitor | |||
| 0.233 | 0.005 | 0.233 | Interleukin 5 antagonist | 0.185 0.006 CHEMBL3527504 0.174 0.007 CHEMBL3526805 | ||
| 0.243 | 0.016 | 0.243 | Butyrylcholinesterase inhibitor | |||
| 0.283 | 0.06 | 0.544 | Tumour necrosis factor alpha release inhibitor | 0.544 0.01 CHEMBL3527504 0.465 0.018 CHEMBL3526805 | CHEMBL3527504 | |
| 0.227 | 0.005 | 0.227 | Alpha tubulin antagonist | 0.051 0.04 CHEMBL3526805 | ||
| 0.278 | 0.061 | 0.654 | Hypoglycemic | 0.654 0.006 CHEMBL3527504 0.625 0.007 CHEMBL3526805 | CHEMBL3527504 | |
| 0.209 | 0.009 | 0.209 | Multidrug resistance-associated protein 1 inhibitor | 0.165 0.019 CHEMBL3527504 0.198 0.011 CHEMBL3526805 | ||
| 0.208 | 0.007 | 0.208 | Beta tubulin antagonist | |||
| 0.21 | 0.011 | 0.21 | Antineoplastic alkaloid | 0.1 0.048 CHEMBL3526805 | ||
| 0.209 | 0.011 | 0.209 | MAP kinase kinase 4 inhibitor | 0.144 0.074 CHEMBL3527504 0.136 0.097 CHEMBL3526805 | ||
| 0.236 | 0.038 | 0.236 | Amyloid beta precursor protein antagonist | |||
| 0.242 | 0.043 | 0.28 | Neurotrophic factor enhancer | 0.28 0.024 CHEMBL3527504 0.245 0.041 CHEMBL3526805 | CHEMBL3527504 | |
| 0.201 | 0.007 | 0.201 | CDC-like kinase 3 inhibitor | 0.12 0.043 CHEMBL3527504 0.12 0.044 CHEMBL3526805 | ||
| 0.252 | 0.058 | 0.265 | Psychostimulant | 0.265 0.053 CHEMBL3527504 0.259 0.055 CHEMBL3526805 | CHEMBL3527504 | |
| 0.208 | 0.018 | 0.339 | Xanthine oxidase inhibitor | 0.339 0.006 CHEMBL3527504 0.299 0.008 CHEMBL3526805 | CHEMBL3527504 | |
| 0.238 | 0.048 | 0.238 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.17 0.108 CHEMBL3527504 0.166 0.114 CHEMBL3526805 | ||
| 0.225 | 0.038 | 0.255 | Protein-tyrosine phosphatase inhibitor | 0.255 0.029 CHEMBL3527504 0.204 0.045 CHEMBL3526805 | CHEMBL3527504 | |
| 0.193 | 0.008 | 0.193 | Estrogen agonist | 0.117 0.014 CHEMBL3527504 0.1 0.017 CHEMBL3526805 | ||
| 0.191 | 0.01 | 0.439 | DNA repair enzyme inhibitor | 0.437 0.003 CHEMBL3527504 0.439 0.003 CHEMBL3526805 | CHEMBL3526805 | |
| 0.184 | 0.004 | 0.184 | Potassium channel Kv1.3 blocker | |||
| 0.231 | 0.053 | 0.231 | CDC-like kinase 4 inhibitor | |||
| 0.195 | 0.027 | 0.232 | DNA intercalator | 0.232 0.019 CHEMBL3527504 0.222 0.02 CHEMBL3526805 | CHEMBL3527504 | |
| 0.191 | 0.027 | 0.191 | Cystathionine beta-synthase inhibitor | 0.165 0.035 CHEMBL3527504 0.148 0.042 CHEMBL3526805 | ||
| 0.171 | 0.01 | 0.171 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.119 0.025 CHEMBL3527504 0.117 0.026 CHEMBL3526805 | ||
| 0.337 | 0.182 | 0.776 | Antiinflammatory | 0.776 0.019 CHEMBL3527504 0.73 0.026 CHEMBL3526805 | CHEMBL3527504 | |
| 0.178 | 0.025 | 0.178 | Interleukin 1b antagonist | 0.126 0.058 CHEMBL3527504 0.148 0.042 CHEMBL3526805 | ||
| 0.231 | 0.08 | 0.415 | Antiamyloidogenic | 0.415 0.026 CHEMBL3527504 0.323 0.045 CHEMBL3526805 | CHEMBL3527504 | |
| 0.157 | 0.01 | 0.157 | Phosphodiesterase V inhibitor | |||
| 0.157 | 0.011 | 0.157 | Estrogen receptor alpha antagonist | |||
| 0.189 | 0.048 | 0.189 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | |||
| 0.173 | 0.037 | 0.205 | Protein-tyrosine phosphatase 1B inhibitor | 0.205 0.028 CHEMBL3527504 0.183 0.034 CHEMBL3526805 | CHEMBL3527504 | |
| 0.142 | 0.012 | 0.142 | Phosphodiesterase 5A inhibitor | |||
| 0.135 | 0.009 | 0.15 | Phosphodiesterase VI inhibitor | 0.132 0.009 CHEMBL3527504 0.15 0.007 CHEMBL3526805 | CHEMBL3526805 | |
| 0.142 | 0.019 | 0.142 | CYP2A6 inhibitor | |||
| 0.148 | 0.026 | 0.446 | Beta glucuronidase inhibitor | 0.446 0.004 CHEMBL3527504 0.411 0.004 CHEMBL3526805 | CHEMBL3527504 | |
| 0.194 | 0.073 | 0.194 | 5 Hydroxytryptamine 3E antagonist | |||
| 0.184 | 0.063 | 0.184 | Succinate dehydrogenase inhibitor | |||
| 0.158 | 0.04 | 0.158 | Antibacterial (Helicobacter pylori) | |||
| 0.153 | 0.036 | 0.206 | Microtubule formation inhibitor | 0.189 0.022 CHEMBL3527504 0.206 0.018 CHEMBL3526805 | CHEMBL3526805 | |
| 0.192 | 0.075 | 0.417 | Platelet adhesion inhibitor | 0.417 0.01 CHEMBL3527504 0.406 0.011 CHEMBL3526805 | CHEMBL3527504 | |
| 0.2 | 0.084 | 0.2 | Interleukin antagonist | |||
| 0.128 | 0.017 | 0.128 | Phosphodiesterase XI inhibitor | |||
| 0.128 | 0.017 | 0.128 | Phosphodiesterase 11A inhibitor | |||
| 0.178 | 0.068 | 0.178 | Mcl-1 antagonist | |||
| 0.131 | 0.025 | 0.131 | NAD(P)H dehydrogenase (quinone) inhibitor | |||
| 0.15 | 0.045 | 0.157 | Heat shock protein 70 antagonist | 0.157 0.032 CHEMBL3527504 0.154 0.037 CHEMBL3526805 | CHEMBL3527504 | |
| 0.211 | 0.107 | 0.441 | DNA synthesis inhibitor | 0.441 0.018 CHEMBL3527504 0.359 0.028 CHEMBL3526805 | CHEMBL3527504 | |
| 0.108 | 0.007 | 0.108 | Glutamate (mGluR7) antagonist | |||
| 0.107 | 0.008 | 0.107 | Estrogen receptor alpha agonist | |||
| 0.184 | 0.09 | 0.184 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | |||
| 0.108 | 0.016 | 0.125 | Aldose reductase inhibitor | 0.125 0.014 CHEMBL3527504 0.124 0.014 CHEMBL3526805 | CHEMBL3527504 | |
| 0.134 | 0.043 | 0.194 | Photosensitizer | 0.192 0.015 CHEMBL3527504 0.194 0.014 CHEMBL3526805 | CHEMBL3526805 | |
| 0.105 | 0.014 | 0.105 | Xanthine dehydrogenase inhibitor | 0.06 0.038 CHEMBL3527504 | ||
| 0.168 | 0.077 | 0.168 | Dual specificity phosphatase inhibitor | |||
| 0.15 | 0.06 | 0.152 | Alkaline phosphatase inhibitor | 0.148 0.061 CHEMBL3527504 0.152 0.059 CHEMBL3526805 | CHEMBL3526805 | |
| 0.166 | 0.078 | 0.169 | Phospholipase C inhibitor | 0.169 0.074 CHEMBL3527504 0.143 0.122 CHEMBL3526805 | CHEMBL3527504 | |
| 0.093 | 0.005 | 0.093 | Endothelin receptor antagonist | |||
| 0.209 | 0.121 | 0.209 | 5 Hydroxytryptamine 1E antagonist | |||
| 0.16 | 0.073 | 0.16 | Peroxidase inhibitor | |||
| 0.129 | 0.046 | 0.129 | 5-Lipoxygenase inhibitor | |||
| 0.148 | 0.067 | 0.174 | Mannose-6-phosphate isomerase inhibitor | 0.174 0.047 CHEMBL3527504 0.159 0.057 CHEMBL3526805 | CHEMBL3527504 | |
| 0.141 | 0.062 | 0.141 | Cyclooxygenase 1 inhibitor | 0.11 0.09 CHEMBL3527504 0.107 0.092 CHEMBL3526805 | ||
| 0.136 | 0.061 | 0.325 | Cyclooxygenase 3 inhibitor | 0.324 0.005 CHEMBL3527504 0.325 0.005 CHEMBL3526805 | CHEMBL3526805 | |
| 0.122 | 0.049 | 0.355 | Expectorant | 0.32 0.007 CHEMBL3527504 0.355 0.006 CHEMBL3526805 | CHEMBL3526805 | |
| 0.077 | 0.005 | 0.077 | Endothelin B receptor antagonist | |||
| 0.099 | 0.028 | 0.104 | GABA aminotransferase inhibitor | 0.104 0.024 CHEMBL3527504 0.089 0.037 CHEMBL3526805 | CHEMBL3527504 | |
| 0.111 | 0.042 | 0.276 | Antineoplastic antibiotic | 0.276 0.011 CHEMBL3527504 0.237 0.016 CHEMBL3526805 | CHEMBL3527504 | |
| 0.077 | 0.012 | 0.077 | Acetyl-CoA transferase 2 inhibitor | 0.059 0.033 CHEMBL3527504 0.059 0.033 CHEMBL3526805 | ||
| 0.12 | 0.055 | 0.12 | Sphingosine 1-phosphate receptor 2 agonist | |||
| 0.068 | 0.004 | 0.068 | Estrogen-related receptor beta antagonist | 0.032 0.024 CHEMBL3527504 | ||
| 0.085 | 0.024 | 0.085 | CDC25B inhibitor | |||
| 0.084 | 0.023 | 0.129 | Neuraminidase inhibitor | 0.129 0.008 CHEMBL3527504 0.114 0.011 CHEMBL3526805 | CHEMBL3527504 | |
| 0.069 | 0.011 | 0.072 | Factor III inhibitor | 0.072 0.01 CHEMBL3527504 0.071 0.01 CHEMBL3526805 | CHEMBL3527504 | |
| 0.13 | 0.072 | 0.137 | Interleukin 4 antagonist | 0.137 0.064 CHEMBL3527504 0.13 0.072 CHEMBL3526805 | CHEMBL3527504 | |
| 0.269 | 0.213 | 0.269 | MAP kinase 1 inhibitor | |||
| 0.095 | 0.041 | 0.095 | Myeloperoxidase inhibitor | |||
| 0.088 | 0.038 | 0.088 | Glutamate decarboxylase inhibitor | |||
| 0.055 | 0.005 | 0.055 | Endothelin A receptor antagonist | |||
| 0.099 | 0.051 | 0.099 | ABCA1 expression enhancer | |||
| 0.087 | 0.041 | 0.087 | Keratolytic | |||
| 0.13 | 0.083 | 0.251 | Protein kinase stimulant | 0.251 0.026 CHEMBL3527504 0.251 0.026 CHEMBL3526805 | CHEMBL3526805 | |
| 0.079 | 0.034 | 0.111 | HIV-1 integrase (3'-Processing) inhibitor | 0.111 0.022 CHEMBL3527504 0.058 0.049 CHEMBL3526805 | CHEMBL3527504 | |
| 0.148 | 0.104 | 0.148 | 3C-like protease (Human coronavirus) inhibitor | |||
| 0.066 | 0.024 | 0.066 | Ryanodine receptor antagonist | |||
| 0.124 | 0.083 | 0.124 | Interleukin 1 antagonist | |||
| 0.082 | 0.041 | 0.082 | Lipase inhibitor | 0.075 0.049 CHEMBL3527504 | ||
| 0.157 | 0.118 | 0.659 | Angiogenesis stimulant | 0.659 0.005 CHEMBL3527504 0.62 0.006 CHEMBL3526805 | CHEMBL3527504 | |
| 0.045 | 0.008 | 0.045 | Dopamine autoreceptor agonist | |||
| 0.101 | 0.066 | 0.101 | Urease inhibitor | |||
| 0.079 | 0.045 | 0.114 | Telomerase inhibitor | 0.114 0.028 CHEMBL3527504 | CHEMBL3527504 | |
| 0.218 | 0.187 | 0.218 | GABA C receptor rho-3 antagonist | |||
| 0.114 | 0.084 | 0.114 | Toll-Like receptor 2 antagonist | |||
| 0.067 | 0.037 | 0.102 | HIV-1 integrase (Strand Transfer) inhibitor | 0.102 0.022 CHEMBL3527504 0.051 0.049 CHEMBL3526805 | CHEMBL3527504 | |
| 0.088 | 0.06 | 0.125 | ATPase (Vacuolar H+) inhibitor | 0.123 0.018 CHEMBL3527504 0.125 0.016 CHEMBL3526805 | CHEMBL3526805 | |
| 0.044 | 0.019 | 0.044 | Estradiol 17 beta-dehydrogenase 2 inhibitor | |||
| 0.147 | 0.122 | 0.147 | I kappa B kinase epsilon inhibitor | |||
| 0.049 | 0.025 | 0.049 | Estradiol 17 beta-dehydrogenase inhibitor | |||
| 0.119 | 0.097 | 0.119 | Neurotrophic factor | 0.117 0.1 CHEMBL3527504 0.116 0.102 CHEMBL3526805 | ||
| 0.143 | 0.125 | 0.335 | Non-steroidal antiinflammatory agent | 0.238 0.048 CHEMBL3527504 0.335 0.022 CHEMBL3526805 | CHEMBL3526805 | |
| 0.048 | 0.03 | 0.048 | Carbonic anhydrase VII inhibitor | |||
| 0.074 | 0.057 | 0.074 | GABA B receptor agonist | |||
| 0.047 | 0.03 | 0.047 | Phosphodiesterase 6C inhibitor | |||
| 0.038 | 0.022 | 0.038 | Estrogen receptor beta agonist | |||
| 0.029 | 0.014 | 0.12 | Sodium/glucose cotransporter 2 inhibitor | 0.12 0.002 CHEMBL3527504 0.118 0.002 CHEMBL3526805 | CHEMBL3527504 | |
| 0.14 | 0.124 | 0.14 | Cyclin-dependent kinase 3 inhibitor | |||
| 0.103 | 0.091 | 0.103 | Interleukin 8 antagonist | |||
| 0.129 | 0.117 | 0.129 | Dual specificity phosphatase 3 inhibitor | |||
| 0.084 | 0.073 | 0.1 | Alcohol dehydrogenase inhibitor | 0.1 0.052 CHEMBL3527504 | CHEMBL3527504 | |
| 0.048 | 0.037 | 0.048 | Topoisomerase II beta inhibitor | |||
| 0.049 | 0.038 | 0.049 | CD45 antagonist | |||
| 0.074 | 0.065 | 0.074 | Carbonic anhydrase VI inhibitor | |||
| 0.077 | 0.07 | 0.077 | Thioredoxin reductase inhibitor | |||
| 0.053 | 0.046 | 0.053 | Aromatase inhibitor | |||
| 0.052 | 0.045 | 0.071 | DNA helicase inhibitor | 0.071 0.016 CHEMBL3527504 | CHEMBL3527504 | |
| 0.136 | 0.13 | 0.257 | DNA methylase inhibitor | 0.233 0.059 CHEMBL3527504 0.257 0.044 CHEMBL3526805 | CHEMBL3526805 | |
| 0.054 | 0.05 | 0.054 | Heat shock protein 90 beta antagonist | |||
| 0.152 | 0.148 | 0.278 | Cyclic AMP phosphodiesterase inhibitor | 0.264 0.057 CHEMBL3527504 0.278 0.051 CHEMBL3526805 | CHEMBL3526805 | |
| 0.059 | 0.056 | 0.115 | Neuraminidase (influenza) inhibitor | 0.115 0.013 CHEMBL3527504 0.096 0.018 CHEMBL3526805 | CHEMBL3527504 | |
| 0.12 | 0.118 | 0.253 | Hexokinase inhibitor | 0.253 0.017 CHEMBL3527504 0.236 0.02 CHEMBL3526805 | CHEMBL3527504 | |
| 0.093 | 0.097 | 0.267 | Alkylator | 0.267 0.015 CHEMBL3527504 0.198 0.027 CHEMBL3526805 | CHEMBL3527504 | |
| 0.022 | 0.029 | 0.094 | Sodium/glucose cotransporter inhibitor | 0.094 0.003 CHEMBL3527504 0.09 0.003 CHEMBL3526805 | CHEMBL3527504 | |
| 0.159 | 0.17 | 0.375 | Peptidyltransferase inhibitor | 0.375 0.009 CHEMBL3527504 0.359 0.011 CHEMBL3526805 | CHEMBL3527504 | |
| 0.017 | 0.031 | 0.066 | Protein 30S ribosomal subunit inhibitor | 0.066 0.005 CHEMBL3527504 0.057 0.007 CHEMBL3526805 | CHEMBL3527504 | |
| 0.083 | 0.098 | 0.133 | Phosphodiesterase 6D inhibitor | 0.133 0.016 CHEMBL3527504 0.12 0.025 CHEMBL3526805 | CHEMBL3527504 | |
| 0.172 | 0.193 | 0.433 | Cholesterol antagonist | 0.433 0.043 CHEMBL3527504 0.371 0.057 CHEMBL3526805 | CHEMBL3527504 | |
| 0.119 | 0.147 | 0.206 | DNA methyltransferase I inhibitor | 0.17 0.087 CHEMBL3527504 0.206 0.066 CHEMBL3526805 | CHEMBL3526805 | |
| 0.047 | 0.076 | 0.079 | Nitric oxide donor | 0.079 0.023 CHEMBL3527504 0.076 0.026 CHEMBL3526805 | CHEMBL3527504 | |
| 0.072 | 0.103 | 0.133 | Uric acid excretion stimulant | 0.133 0.031 CHEMBL3527504 0.113 0.042 CHEMBL3526805 | CHEMBL3527504 | |
| 0.012 | 0.052 | 0.02 | Antibiotic Anthracycline-like | 0.019 0.012 CHEMBL3527504 0.02 0.01 CHEMBL3526805 | CHEMBL3526805 | |
| 0.036 | 0.084 | 0.052 | Leukotriene B4 antagonist | 0.052 0.041 CHEMBL3527504 0.05 0.045 CHEMBL3526805 | CHEMBL3527504 | |
| 0.012 | 0.061 | 0.024 | Dopamine D1 agonist | 0.024 0.013 CHEMBL3527504 | CHEMBL3527504 | |
| 0.045 | 0.096 | 0.101 | Na+ K+ transporting ATPase inhibitor | 0.101 0.031 CHEMBL3527504 0.091 0.04 CHEMBL3526805 | CHEMBL3527504 | |
| 0.172 | 0.227 | 0.482 | Immunosuppressant | 0.482 0.038 CHEMBL3527504 0.457 0.045 CHEMBL3526805 | CHEMBL3527504 | |
| 0.115 | 0.186 | 0.225 | ATPase inhibitor | 0.22 0.024 CHEMBL3527504 0.225 0.021 CHEMBL3526805 | CHEMBL3526805 | |
| 0.031 | 0.104 | 0.076 | Alpha-mannosidase inhibitor | 0.076 0.013 CHEMBL3527504 0.074 0.014 CHEMBL3526805 | CHEMBL3527504 | |
| 0.113 | 0.198 | 0.448 | Immunostimulant | 0.448 0.037 CHEMBL3527504 0.418 0.045 CHEMBL3526805 | CHEMBL3527504 | |
| 0.028 | 0.118 | 0.051 | Glucose-6-phosphate isomerase inhibitor | 0.051 0.028 CHEMBL3527504 | CHEMBL3527504 | |
| 0.108 | 0.201 | 0.145 | CC chemokine 6 receptor antagonist | 0.145 0.029 CHEMBL3527504 0.139 0.041 CHEMBL3526805 | CHEMBL3527504 | |
| 0.062 | 0.167 | 0.218 | AMP-activated protein kinase stimulant | 0.218 0.009 CHEMBL3527504 0.189 0.013 CHEMBL3526805 | CHEMBL3527504 | |
| 0.018 | 0.131 | 0.066 | Mannosidase inhibitor | 0.066 0.013 CHEMBL3527504 0.061 0.016 CHEMBL3526805 | CHEMBL3527504 | |
| 0.028 | 0.153 | 0.072 | Glucose-6-phosphate translocase inhibitor | 0.069 0.016 CHEMBL3527504 0.072 0.015 CHEMBL3526805 | CHEMBL3526805 | |
| 0.055 | 0.186 | 0.124 | Transcription factor NF kappa B stimulant | 0.124 0.024 CHEMBL3527504 0.122 0.024 CHEMBL3526805 | CHEMBL3527504 | |
| 0.091 | 0.234 | 0.162 | Interferon gamma antagonist | 0.162 0.064 CHEMBL3527504 0.156 0.071 CHEMBL3526805 | CHEMBL3527504 | |
| 0.047 | 0.194 | 0.159 | UDP-glucose 4-epimerase inhibitor | 0.159 0.026 CHEMBL3527504 0.1 0.06 CHEMBL3526805 | CHEMBL3527504 | |
| 0.026 | 0.181 | 0.087 | Heparanase inhibitor | 0.082 0.006 CHEMBL3527504 0.087 0.005 CHEMBL3526805 | CHEMBL3526805 | |
| 0.081 | 0.238 | 0.231 | Insulin secretagoues | 0.231 0.024 CHEMBL3527504 0.216 0.029 CHEMBL3526805 | CHEMBL3527504 | |
| 0.048 | 0.217 | 0.098 | NADH dehydrogenase inhibitor | 0.098 0.046 CHEMBL3527504 0.08 0.075 CHEMBL3526805 | CHEMBL3527504 | |
| 0.053 | 0.226 | 0.145 | Alpha-N-acetylglucosaminidase inhibitor | 0.145 0.058 CHEMBL3527504 | CHEMBL3527504 | |
| 0.018 | 0.202 | 0.08 | Phosphofructokinase-1 inhibitor | 0.08 0.041 CHEMBL3527504 | CHEMBL3527504 | |
| 0.017 | 0.201 | 0.047 | Neuraminidase (Influenza A) inhibitor | 0.047 0.028 CHEMBL3527504 0.043 0.036 CHEMBL3526805 | CHEMBL3527504 | |
| 0.077 | 0.262 | 0.303 | Hemostatic | 0.228 0.025 CHEMBL3527504 0.303 0.015 CHEMBL3526805 | CHEMBL3526805 | |
| 0.074 | 0.274 | 0.233 | Hypolipemic | 0.227 0.079 CHEMBL3527504 0.233 0.076 CHEMBL3526805 | CHEMBL3526805 | |
| 0.042 | 0.245 | 0.102 | Triose-phosphate isomerase inhibitor | 0.102 0.046 CHEMBL3527504 | CHEMBL3527504 | |
| 0.074 | 0.283 | 0.175 | Interleukin 6 antagonist | 0.175 0.059 CHEMBL3527504 0.169 0.065 CHEMBL3526805 | CHEMBL3527504 | |
| 0.035 | 0.261 | 0.058 | Lipocortins synthesis agonist | 0.058 0.04 CHEMBL3527504 0.057 0.043 CHEMBL3526805 | CHEMBL3527504 | |
| 0.048 | 0.274 | 0.136 | Toll-Like receptor 4 antagonist | 0.135 0.03 CHEMBL3527504 0.136 0.03 CHEMBL3526805 | CHEMBL3526805 | |
| 0.101 | 0.331 | 0.226 | Angiogenesis inhibitor | 0.201 0.168 CHEMBL3527504 0.226 0.142 CHEMBL3526805 | CHEMBL3526805 | |
| 0.016 | 0.248 | 0.086 | Protein 50S ribosomal subunit inhibitor | 0.086 0.017 CHEMBL3527504 0.085 0.017 CHEMBL3526805 | CHEMBL3527504 | |
| 0.053 | 0.304 | 0.169 | Diuretic | 0.169 0.062 CHEMBL3527504 0.125 0.099 CHEMBL3526805 | CHEMBL3527504 | |
| 0.038 | 0.298 | 0.087 | Thioredoxin inhibitor | 0.087 0.066 CHEMBL3527504 0.086 0.07 CHEMBL3526805 | CHEMBL3527504 | |
| 0.03 | 0.361 | 0.257 | Thrombolytic | 0.257 0.032 CHEMBL3527504 0.232 0.039 CHEMBL3526805 | CHEMBL3527504 | |
| 0.047 | 0.381 | 0.229 | Platelet antagonist | 0.216 0.09 CHEMBL3527504 0.229 0.082 CHEMBL3526805 | CHEMBL3526805 | |
| 0.043 | 0.399 | 0.078 | T cell inhibitor | 0.078 0.073 CHEMBL3527504 0.078 0.073 CHEMBL3526805 | CHEMBL3526805 | |
| 0.014 | 0.371 | 0.064 | Antibiotic Aminoglycoside-like | 0.064 0.007 CHEMBL3527504 0.062 0.008 CHEMBL3526805 | CHEMBL3527504 | |
| 0.072 | 0.429 | 0.453 | Antithrombotic | 0.453 0.037 CHEMBL3527504 0.426 0.043 CHEMBL3526805 | CHEMBL3527504 | |
| 0.033 | 0.426 | 0.187 | Cell wall synthesis inhibitor | 0.187 0.036 CHEMBL3527504 0.148 0.068 CHEMBL3526805 | CHEMBL3527504 | |
| 0.034 | 0.428 | 0.179 | Cell adhesion inhibitor | 0.177 0.032 CHEMBL3527504 0.179 0.031 CHEMBL3526805 | CHEMBL3526805 | |
| 0.024 | 0.429 | 0.052 | Adenine nucleotide translocase inhibitor | 0.052 0.05 CHEMBL3527504 | CHEMBL3527504 | |
| 0.006 | 0.542 | 0.307 | Selectin antagonist | 0.307 0.005 CHEMBL3527504 0.289 0.006 CHEMBL3526805 | CHEMBL3527504 | |
| 0.051 | 0.634 | 0.685 | Cyclophilin D inhibitor | 0.685 0.015 CHEMBL3527504 0.629 0.023 CHEMBL3526805 | CHEMBL3527504 | |
| 0.009 | 0.669 | 0.025 | Toll-Like receptor 4 agonist | 0.025 0.023 CHEMBL3526805 | CHEMBL3526805 | |
| 0.051 | 0.814 | 0.335 | Interleukin 2 agonist | 0.335 0.053 CHEMBL3527504 0.309 0.068 CHEMBL3526805 | CHEMBL3527504 | |
| 0.009 | 0.917 | 0.225 | Immunomodulator | 0.225 0.137 CHEMBL3527504 | CHEMBL3527504 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |