| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.957 | 0.003 | 0.958 | Antioxidant | 0.946 0.003 CHEMBL4525790 0.958 0.003 CHEMBL527285 | CHEMBL527285 | |
| 0.898 | 0.001 | 0.904 | Lipid peroxidase inhibitor | 0.848 0.001 CHEMBL4525790 0.904 0.001 CHEMBL527285 | CHEMBL527285 | |
| 0.893 | 0.001 | 0.893 | Peroxidase inhibitor | 0.85 0.001 CHEMBL4525790 0.82 0.002 CHEMBL527285 | ||
| 0.847 | 0.01 | 0.874 | Antiinflammatory | 0.813 0.014 CHEMBL4525790 0.874 0.007 CHEMBL527285 | CHEMBL527285 | |
| 0.796 | 0.004 | 0.832 | Lipoxygenase inhibitor | 0.675 0.006 CHEMBL4525790 0.832 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.784 | 0.004 | 0.818 | Free radical scavenger | 0.752 0.004 CHEMBL4525790 0.818 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.781 | 0.004 | 0.781 | Cholesterol antagonist | 0.755 0.005 CHEMBL4525790 0.779 0.004 CHEMBL527285 | ||
| 0.752 | 0.023 | 0.752 | Apoptosis agonist | 0.748 0.023 CHEMBL4525790 0.709 0.029 CHEMBL527285 | ||
| 0.721 | 0.003 | 0.721 | NOS3 expression enhancer | 0.676 0.004 CHEMBL4525790 0.713 0.003 CHEMBL527285 | ||
| 0.723 | 0.018 | 0.723 | Transcription factor NF kappa B inhibitor | 0.706 0.02 CHEMBL4525790 0.697 0.021 CHEMBL527285 | ||
| 0.652 | 0.001 | 0.652 | Cholesterol synthesis inhibitor | 0.588 0.001 CHEMBL4525790 0.558 0.002 CHEMBL527285 | ||
| 0.635 | 0.001 | 0.665 | Maillard reaction inhibitor | 0.556 0.002 CHEMBL4525790 0.665 0.001 CHEMBL527285 | CHEMBL527285 | |
| 0.614 | 0.006 | 0.614 | Hypolipemic | 0.576 0.008 CHEMBL4525790 0.589 0.007 CHEMBL527285 | ||
| 0.592 | 0.029 | 0.795 | Cyclophilin D inhibitor | 0.651 0.019 CHEMBL4525790 0.795 0.007 CHEMBL527285 | CHEMBL527285 | |
| 0.549 | 0.002 | 0.549 | Vanilloid 1 agonist | 0.504 0.002 CHEMBL4525790 0.363 0.004 CHEMBL527285 | ||
| 0.551 | 0.011 | 0.695 | Hypoglycemic | 0.592 0.009 CHEMBL4525790 0.695 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.529 | 0.02 | 0.532 | Spasmolytic | 0.463 0.029 CHEMBL4525790 0.532 0.019 CHEMBL527285 | CHEMBL527285 | |
| 0.512 | 0.002 | 0.512 | Keratolytic | 0.502 0.002 CHEMBL4525790 0.499 0.002 CHEMBL527285 | ||
| 0.521 | 0.018 | 0.593 | Apoptosis antagonist | 0.431 0.031 CHEMBL4525790 0.593 0.01 CHEMBL527285 | CHEMBL527285 | |
| 0.519 | 0.028 | 0.536 | Immunosuppressant | 0.536 0.024 CHEMBL4525790 0.456 0.045 CHEMBL527285 | CHEMBL4525790 | |
| 0.503 | 0.016 | 0.555 | Antiamyloidogenic | 0.555 0.011 CHEMBL4525790 0.376 0.033 CHEMBL527285 | CHEMBL4525790 | |
| 0.482 | 0.016 | 0.623 | Platelet antagonist | 0.526 0.011 CHEMBL4525790 0.623 0.006 CHEMBL527285 | CHEMBL527285 | |
| 0.462 | 0.005 | 0.495 | 5-Lipoxygenase inhibitor | 0.358 0.007 CHEMBL4525790 0.495 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.489 | 0.036 | 0.489 | 5 Hydroxytryptamine release inhibitor | 0.441 0.056 CHEMBL4525790 0.405 0.075 CHEMBL527285 | ||
| 0.469 | 0.033 | 0.469 | Immunostimulant | 0.441 0.039 CHEMBL4525790 0.433 0.041 CHEMBL527285 | ||
| 0.424 | 0.014 | 0.424 | P-glycoprotein inhibitor | 0.349 0.021 CHEMBL4525790 0.373 0.019 CHEMBL527285 | ||
| 0.419 | 0.012 | 0.453 | Hepatoprotectant | 0.39 0.014 CHEMBL4525790 0.453 0.009 CHEMBL527285 | CHEMBL527285 | |
| 0.451 | 0.049 | 0.51 | Histamine release inhibitor | 0.409 0.071 CHEMBL4525790 0.51 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.349 | 0.003 | 0.349 | Interferon agonist | 0.338 0.003 CHEMBL4525790 0.267 0.004 CHEMBL527285 | ||
| 0.37 | 0.033 | 0.37 | Tumour necrosis factor alpha release inhibitor | 0.349 0.038 CHEMBL4525790 0.233 0.083 CHEMBL527285 | ||
| 0.351 | 0.016 | 0.351 | Melanin inhibitor | 0.3 0.022 CHEMBL4525790 0.268 0.026 CHEMBL527285 | ||
| 0.357 | 0.031 | 0.382 | Nitric oxide antagonist | 0.328 0.035 CHEMBL4525790 0.382 0.028 CHEMBL527285 | CHEMBL527285 | |
| 0.327 | 0.003 | 0.337 | Papain-like protease (SARS coronavirus) inhibitor | 0.284 0.004 CHEMBL4525790 0.337 0.003 CHEMBL527285 | CHEMBL527285 | |
| 0.305 | 0.003 | 0.332 | Glutathione S-transferase inhibitor | 0.274 0.003 CHEMBL4525790 0.332 0.003 CHEMBL527285 | CHEMBL527285 | |
| 0.306 | 0.005 | 0.306 | Electron transport complex I inhibitor | 0.231 0.006 CHEMBL4525790 0.171 0.013 CHEMBL527285 | ||
| 0.33 | 0.039 | 0.339 | Vasodilator | 0.28 0.055 CHEMBL4525790 0.339 0.036 CHEMBL527285 | CHEMBL527285 | |
| 0.292 | 0.002 | 0.292 | Interferon inducer | 0.278 0.002 CHEMBL4525790 0.185 0.004 CHEMBL527285 | ||
| 0.376 | 0.088 | 0.376 | Antibacterial | 0.316 0.123 CHEMBL4525790 0.26 0.168 CHEMBL527285 | ||
| 0.3 | 0.017 | 0.3 | Protein kinase stimulant | 0.252 0.026 CHEMBL4525790 0.278 0.02 CHEMBL527285 | ||
| 0.3 | 0.018 | 0.411 | Monophenol monooxygenase inhibitor | 0.251 0.024 CHEMBL4525790 0.411 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.297 | 0.023 | 0.558 | Diuretic | 0.335 0.018 CHEMBL4525790 0.558 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.268 | 0.01 | 0.268 | Neurotrophic factor | 0.229 0.017 CHEMBL4525790 0.185 0.035 CHEMBL527285 | ||
| 0.26 | 0.009 | 0.382 | Mediator release inhibitor | 0.213 0.013 CHEMBL4525790 0.382 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.273 | 0.023 | 0.35 | Insulin sensitizer | 0.255 0.032 CHEMBL4525790 0.35 0.009 CHEMBL527285 | CHEMBL527285 | |
| 0.311 | 0.073 | 0.325 | Caspase 3 stimulant | 0.242 0.119 CHEMBL4525790 0.325 0.068 CHEMBL527285 | CHEMBL527285 | |
| 0.242 | 0.009 | 0.249 | Beta amyloid protein antagonist | 0.165 0.031 CHEMBL4525790 0.249 0.009 CHEMBL527285 | CHEMBL527285 | |
| 0.305 | 0.072 | 0.343 | Nootropic | 0.343 0.056 CHEMBL4525790 | CHEMBL4525790 | |
| 0.253 | 0.037 | 0.263 | Neurotrophic factor enhancer | 0.237 0.046 CHEMBL4525790 0.263 0.032 CHEMBL527285 | CHEMBL527285 | |
| 0.237 | 0.027 | 0.299 | Phospholipase A2 inhibitor | 0.217 0.035 CHEMBL4525790 0.299 0.014 CHEMBL527285 | CHEMBL527285 | |
| 0.215 | 0.006 | 0.215 | Vanilloid agonist | 0.148 0.011 CHEMBL4525790 0.128 0.015 CHEMBL527285 | ||
| 0.188 | 0.009 | 0.188 | Inducible nitric-oxide synthase inhibitor | 0.113 0.028 CHEMBL4525790 0.171 0.012 CHEMBL527285 | ||
| 0.203 | 0.03 | 0.226 | Arachidonic acid antagonist | 0.203 0.03 CHEMBL4525790 0.226 0.014 CHEMBL527285 | CHEMBL527285 | |
| 0.301 | 0.131 | 0.301 | 15-Lipoxygenase inhibitor | 0.277 0.145 CHEMBL527285 | ||
| 0.224 | 0.055 | 0.368 | Non-steroidal antiinflammatory agent | 0.221 0.056 CHEMBL4525790 0.368 0.017 CHEMBL527285 | CHEMBL527285 | |
| 0.242 | 0.073 | 0.242 | Calpain inhibitor | |||
| 0.176 | 0.007 | 0.243 | Leukotriene antagonist | 0.164 0.009 CHEMBL4525790 0.243 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.173 | 0.015 | 0.173 | Nitric-oxide synthase inhibitor | 0.12 0.037 CHEMBL4525790 0.168 0.017 CHEMBL527285 | ||
| 0.16 | 0.007 | 0.16 | Androgen agonist | 0.124 0.009 CHEMBL4525790 0.15 0.007 CHEMBL527285 | ||
| 0.191 | 0.041 | 0.439 | Insulin secretagoues | 0.282 0.014 CHEMBL4525790 0.439 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.173 | 0.023 | 0.173 | Pregnane X receptor agonist | 0.155 0.045 CHEMBL4525790 0.166 0.03 CHEMBL527285 | ||
| 0.174 | 0.026 | 0.179 | Antineoplastic antibiotic | 0.179 0.025 CHEMBL4525790 0.118 0.039 CHEMBL527285 | CHEMBL4525790 | |
| 0.162 | 0.015 | 0.232 | ABCA1 expression enhancer | 0.232 0.007 CHEMBL4525790 0.166 0.014 CHEMBL527285 | CHEMBL4525790 | |
| 0.235 | 0.089 | 0.283 | DNA damaging | 0.178 0.136 CHEMBL4525790 0.283 0.064 CHEMBL527285 | CHEMBL527285 | |
| 0.203 | 0.058 | 0.225 | Growth hormone agonist | 0.17 0.073 CHEMBL4525790 0.225 0.05 CHEMBL527285 | CHEMBL527285 | |
| 0.183 | 0.042 | 0.237 | Cyclooxygenase 1 inhibitor | 0.131 0.07 CHEMBL4525790 0.237 0.024 CHEMBL527285 | CHEMBL527285 | |
| 0.164 | 0.025 | 0.249 | Mucolytic | 0.167 0.024 CHEMBL4525790 0.249 0.006 CHEMBL527285 | CHEMBL527285 | |
| 0.167 | 0.029 | 0.3 | Expectorant | 0.171 0.028 CHEMBL4525790 0.3 0.009 CHEMBL527285 | CHEMBL527285 | |
| 0.211 | 0.074 | 0.389 | Platelet aggregation inhibitor | 0.233 0.06 CHEMBL4525790 0.389 0.02 CHEMBL527285 | CHEMBL527285 | |
| 0.14 | 0.004 | 0.14 | Glucose-6-phosphate translocase inhibitor | 0.122 0.004 CHEMBL4525790 0.137 0.004 CHEMBL527285 | ||
| 0.17 | 0.035 | 0.17 | Farnesoid X receptor antagonist | 0.154 0.048 CHEMBL4525790 0.17 0.035 CHEMBL527285 | ||
| 0.254 | 0.123 | 0.302 | Antithrombotic | 0.296 0.091 CHEMBL4525790 0.302 0.086 CHEMBL527285 | CHEMBL527285 | |
| 0.142 | 0.014 | 0.142 | CDC25A inhibitor | 0.104 0.025 CHEMBL4525790 0.086 0.037 CHEMBL527285 | ||
| 0.137 | 0.015 | 0.205 | Prostaglandin-E synthase inhibitor | 0.073 0.045 CHEMBL4525790 0.205 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.126 | 0.004 | 0.31 | Thromboxane synthase inhibitor | 0.143 0.004 CHEMBL4525790 0.31 0.003 CHEMBL527285 | CHEMBL527285 | |
| 0.123 | 0.005 | 0.135 | Bcl-xL inhibitor | 0.096 0.007 CHEMBL4525790 0.135 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.248 | 0.129 | 0.248 | Vasodilator, peripheral | 0.208 0.167 CHEMBL4525790 | ||
| 0.175 | 0.059 | 0.175 | Interleukin 6 antagonist | 0.153 0.084 CHEMBL4525790 | ||
| 0.195 | 0.08 | 0.195 | Amyloid beta aggregation inhibitor | 0.163 0.099 CHEMBL4525790 0.14 0.116 CHEMBL527285 | ||
| 0.157 | 0.043 | 0.157 | Proteasome inhibitor | 0.131 0.058 CHEMBL4525790 | ||
| 0.128 | 0.023 | 0.128 | Lanosterol 14 alpha demethylase inhibitor | 0.086 0.079 CHEMBL4525790 0.085 0.081 CHEMBL527285 | ||
| 0.157 | 0.052 | 0.185 | Adenylate cyclase stimulant | 0.148 0.066 CHEMBL4525790 0.185 0.022 CHEMBL527285 | CHEMBL527285 | |
| 0.135 | 0.033 | 0.136 | Estrogen antagonist | 0.128 0.041 CHEMBL4525790 0.136 0.031 CHEMBL527285 | CHEMBL527285 | |
| 0.119 | 0.017 | 0.124 | Na+ K+ transporting ATPase inhibitor | 0.122 0.015 CHEMBL4525790 0.124 0.014 CHEMBL527285 | CHEMBL527285 | |
| 0.125 | 0.027 | 0.127 | Estrogen receptor beta antagonist | 0.114 0.04 CHEMBL4525790 0.127 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.115 | 0.017 | 0.115 | Ribonucleoside-diphosphate reductase inhibitor | 0.083 0.023 CHEMBL4525790 0.098 0.019 CHEMBL527285 | ||
| 0.134 | 0.038 | 0.169 | Bronchodilator | 0.107 0.055 CHEMBL4525790 0.169 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.101 | 0.004 | 0.101 | Adenine nucleotide translocase inhibitor | 0.089 0.006 CHEMBL4525790 0.077 0.01 CHEMBL527285 | ||
| 0.117 | 0.021 | 0.243 | Peroxisome proliferator-activated receptor gamma agonist | 0.104 0.025 CHEMBL4525790 0.243 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.166 | 0.07 | 0.216 | Thrombolytic | 0.167 0.07 CHEMBL4525790 0.216 0.045 CHEMBL527285 | CHEMBL527285 | |
| 0.206 | 0.113 | 0.221 | DNA synthesis inhibitor | 0.196 0.129 CHEMBL4525790 0.221 0.093 CHEMBL527285 | CHEMBL527285 | |
| 0.11 | 0.019 | 0.11 | Ribonucleotide reductase inhibitor | 0.082 0.026 CHEMBL4525790 0.096 0.022 CHEMBL527285 | ||
| 0.167 | 0.077 | 0.167 | Antipruritic | 0.133 0.117 CHEMBL4525790 0.144 0.101 CHEMBL527285 | ||
| 0.117 | 0.028 | 0.125 | Ornithine decarboxylase inhibitor | 0.102 0.043 CHEMBL4525790 0.125 0.022 CHEMBL527285 | CHEMBL527285 | |
| 0.177 | 0.089 | 0.196 | Anesthetic general | 0.148 0.116 CHEMBL4525790 0.196 0.076 CHEMBL527285 | CHEMBL527285 | |
| 0.228 | 0.14 | 0.246 | Angiogenesis inhibitor | 0.19 0.181 CHEMBL4525790 0.246 0.126 CHEMBL527285 | CHEMBL527285 | |
| 0.169 | 0.087 | 0.36 | DNA methyltransferase I inhibitor | 0.135 0.123 CHEMBL4525790 0.36 0.013 CHEMBL527285 | CHEMBL527285 | |
| 0.092 | 0.013 | 0.097 | Nitric oxide donor | 0.086 0.017 CHEMBL4525790 0.097 0.01 CHEMBL527285 | CHEMBL527285 | |
| 0.121 | 0.046 | 0.121 | Butyrylcholinesterase inhibitor | 0.089 0.072 CHEMBL527285 | ||
| 0.128 | 0.057 | 0.154 | Protein-tyrosine phosphatase 1B inhibitor | 0.143 0.049 CHEMBL4525790 0.154 0.044 CHEMBL527285 | CHEMBL527285 | |
| 0.141 | 0.071 | 0.153 | Ca2+-transporting ATPase inhibitor | 0.139 0.078 CHEMBL4525790 0.153 0.036 CHEMBL527285 | CHEMBL527285 | |
| 0.114 | 0.046 | 0.147 | Anabolic | 0.095 0.07 CHEMBL4525790 0.147 0.019 CHEMBL527285 | CHEMBL527285 | |
| 0.174 | 0.108 | 0.174 | Histone acetyltransferase inhibitor | 0.155 0.132 CHEMBL527285 | ||
| 0.102 | 0.038 | 0.102 | Topoisomerase II alpha inhibitor | 0.088 0.047 CHEMBL4525790 0.091 0.045 CHEMBL527285 | ||
| 0.072 | 0.007 | 0.13 | Leukotriene D4 antagonist | 0.05 0.01 CHEMBL4525790 0.13 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.073 | 0.011 | 0.1 | Pregnane X receptor antagonist | 0.066 0.019 CHEMBL4525790 0.1 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.078 | 0.018 | 0.181 | Peroxisome proliferator-activated receptor alpha agonist | 0.074 0.02 CHEMBL4525790 0.181 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.068 | 0.01 | 0.068 | Squalene synthetase inhibitor | 0.055 0.013 CHEMBL4525790 | ||
| 0.061 | 0.004 | 0.068 | Thiazolidinedione | 0.055 0.004 CHEMBL4525790 0.068 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.08 | 0.024 | 0.099 | Glutamate (mGluR6) antagonist | 0.075 0.03 CHEMBL4525790 0.099 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.117 | 0.061 | 0.139 | Photosensitizer | 0.103 0.084 CHEMBL4525790 0.139 0.039 CHEMBL527285 | CHEMBL527285 | |
| 0.12 | 0.065 | 0.252 | Cell adhesion inhibitor | 0.252 0.015 CHEMBL527285 | CHEMBL527285 | |
| 0.114 | 0.059 | 0.134 | Topoisomerase I inhibitor | 0.089 0.08 CHEMBL4525790 0.134 0.048 CHEMBL527285 | CHEMBL527285 | |
| 0.084 | 0.033 | 0.094 | Glycine receptor agonist | 0.084 0.034 CHEMBL4525790 0.094 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.066 | 0.017 | 0.066 | Vanilloid 2 antagonist | 0.062 0.021 CHEMBL4525790 0.062 0.02 CHEMBL527285 | ||
| 0.138 | 0.092 | 0.17 | Protein-tyrosine phosphatase inhibitor | 0.15 0.078 CHEMBL4525790 0.17 0.062 CHEMBL527285 | CHEMBL527285 | |
| 0.125 | 0.082 | 0.125 | Calcium channel blocker | |||
| 0.123 | 0.083 | 0.123 | Bone formation stimulant | 0.117 0.088 CHEMBL4525790 | ||
| 0.083 | 0.043 | 0.088 | Estrogen receptor alpha antagonist | 0.088 0.038 CHEMBL527285 | CHEMBL527285 | |
| 0.057 | 0.018 | 0.057 | Microtubule stabilization | 0.056 0.02 CHEMBL4525790 0.054 0.022 CHEMBL527285 | ||
| 0.077 | 0.039 | 0.165 | Peroxisome proliferator-activated receptor gamma antagonist | 0.072 0.048 CHEMBL4525790 0.165 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.068 | 0.033 | 0.093 | Transcription factor AP-1 inhibitor | 0.055 0.054 CHEMBL4525790 0.093 0.015 CHEMBL527285 | CHEMBL527285 | |
| 0.095 | 0.061 | 0.109 | Prolactin inhibitor | 0.109 0.047 CHEMBL527285 | CHEMBL527285 | |
| 0.063 | 0.028 | 0.063 | Acetyl-CoA transferase inhibitor | |||
| 0.044 | 0.01 | 0.053 | HMG CoA reductase inhibitor | 0.048 0.008 CHEMBL4525790 0.053 0.006 CHEMBL527285 | CHEMBL527285 | |
| 0.044 | 0.012 | 0.118 | Prostaglandin EP3 antagonist | 0.027 0.024 CHEMBL4525790 0.118 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.045 | 0.014 | 0.128 | Peroxisome proliferator-activated receptor delta agonist | 0.045 0.014 CHEMBL4525790 0.128 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.188 | 0.159 | 0.287 | Tyrosine 3 hydroxylase inhibitor | 0.287 0.04 CHEMBL527285 | CHEMBL527285 | |
| 0.044 | 0.016 | 0.044 | 2,3-Oxidosqualene-lanosterol cyclase inhibitor | 0.037 0.026 CHEMBL4525790 | ||
| 0.033 | 0.009 | 0.041 | Retinoic acid receptor agonist | 0.03 0.01 CHEMBL4525790 0.041 0.006 CHEMBL527285 | CHEMBL527285 | |
| 0.076 | 0.054 | 0.128 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.128 0.026 CHEMBL527285 | CHEMBL527285 | |
| 0.031 | 0.01 | 0.031 | Toll-Like receptor 4 agonist | 0.029 0.013 CHEMBL4525790 0.027 0.017 CHEMBL527285 | ||
| 0.055 | 0.035 | 0.074 | Leukotriene B4 antagonist | 0.056 0.034 CHEMBL4525790 0.074 0.018 CHEMBL527285 | CHEMBL527285 | |
| 0.026 | 0.006 | 0.026 | Toll-Like receptor 8 agonist | 0.024 0.007 CHEMBL4525790 | ||
| 0.031 | 0.012 | 0.031 | 1,3-Beta-glucan synthase inhibitor | 0.03 0.015 CHEMBL4525790 | ||
| 0.045 | 0.028 | 0.045 | HIV-1 protease inhibitor | 0.039 0.037 CHEMBL4525790 | ||
| 0.059 | 0.042 | 0.084 | HIV-1 integrase (Strand Transfer) inhibitor | 0.084 0.029 CHEMBL527285 | CHEMBL527285 | |
| 0.139 | 0.123 | 0.23 | Lipocortins synthesis antagonist | 0.138 0.125 CHEMBL4525790 0.23 0.041 CHEMBL527285 | CHEMBL527285 | |
| 0.117 | 0.103 | 0.178 | Cyclooxygenase inhibitor | 0.178 0.052 CHEMBL527285 | CHEMBL527285 | |
| 0.027 | 0.013 | 0.173 | Peroxisome proliferator-activated receptor alpha antagonist | 0.022 0.014 CHEMBL4525790 0.173 0.003 CHEMBL527285 | CHEMBL527285 | |
| 0.061 | 0.046 | 0.084 | HIV-1 integrase (3'-Processing) inhibitor | 0.084 0.032 CHEMBL527285 | CHEMBL527285 | |
| 0.042 | 0.029 | 0.058 | DNA gyrase subunit A inhibitor | 0.058 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.027 | 0.014 | 0.027 | Vanilloid 2 agonist | |||
| 0.089 | 0.076 | 0.112 | Bile acid receptor antagonist | 0.112 0.028 CHEMBL527285 | CHEMBL527285 | |
| 0.139 | 0.127 | 0.326 | DNA methylase inhibitor | 0.326 0.021 CHEMBL527285 | CHEMBL527285 | |
| 0.036 | 0.025 | 0.069 | Retinoid X receptor agonist | 0.069 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.079 | 0.07 | 0.094 | Estrogen-related receptor beta agonist | 0.094 0.033 CHEMBL4525790 | CHEMBL4525790 | |
| 0.047 | 0.04 | 0.047 | Collagenase inhibitor | |||
| 0.065 | 0.059 | 0.065 | Lipase inhibitor | |||
| 0.041 | 0.039 | 0.056 | Antimetabolite | 0.056 0.028 CHEMBL527285 | CHEMBL527285 | |
| 0.142 | 0.14 | 0.142 | Anticonvulsant | |||
| 0.03 | 0.029 | 0.037 | Glutamate (mGluR3) agonist | 0.037 0.013 CHEMBL527285 | CHEMBL527285 | |
| 0.016 | 0.016 | 0.026 | Retinoic acid receptor antagonist | 0.026 0.007 CHEMBL527285 | CHEMBL527285 | |
| 0.164 | 0.165 | 0.186 | RNA-directed DNA polymerase inhibitor | 0.186 0.121 CHEMBL527285 | CHEMBL527285 | |
| 0.015 | 0.021 | 0.018 | Inosine monophosphate dehydrogenase 1 inhibitor | 0.018 0.016 CHEMBL527285 | CHEMBL527285 | |
| 0.026 | 0.033 | 0.032 | ATP citrate lysase inhibitor | 0.032 0.021 CHEMBL527285 | CHEMBL527285 | |
| 0.187 | 0.194 | 0.248 | Vasodilator, coronary | 0.248 0.137 CHEMBL527285 | CHEMBL527285 | |
| 0.052 | 0.062 | 0.054 | Lipocortins synthesis agonist | 0.054 0.053 CHEMBL4525790 | CHEMBL4525790 | |
| 0.028 | 0.039 | 0.103 | Peroxisome proliferator-activated receptor delta antagonist | 0.103 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.1 | 0.112 | 0.177 | NADPH oxidase inhibitor | 0.177 0.042 CHEMBL527285 | CHEMBL527285 | |
| 0.172 | 0.188 | 0.286 | Thyroid hormone antagonist | 0.286 0.101 CHEMBL527285 | CHEMBL527285 | |
| 0.019 | 0.04 | 0.058 | Thyroid hormone agonist | 0.058 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.049 | 0.07 | 0.072 | Leukotriene C antagonist | 0.072 0.012 CHEMBL527285 | CHEMBL527285 | |
| 0.118 | 0.14 | 0.132 | Interferon gamma antagonist | 0.132 0.107 CHEMBL527285 | CHEMBL527285 | |
| 0.05 | 0.073 | 0.102 | Leukotriene synthesis inhibitor | 0.102 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.13 | 0.155 | 0.143 | Phospholipase C inhibitor | 0.143 0.121 CHEMBL527285 | CHEMBL527285 | |
| 0.015 | 0.042 | 0.041 | Leukotriene B4 receptor 1 antagonist | 0.041 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.186 | 0.215 | 0.23 | Interleukin 2 agonist | 0.213 0.168 CHEMBL4525790 0.23 0.143 CHEMBL527285 | CHEMBL527285 | |
| 0.036 | 0.066 | 0.061 | Glucose-6-phosphate isomerase inhibitor | 0.061 0.018 CHEMBL527285 | CHEMBL527285 | |
| 0.031 | 0.067 | 0.05 | Leukotriene C4 antagonist | 0.05 0.011 CHEMBL527285 | CHEMBL527285 | |
| 0.003 | 0.044 | 0.016 | Thyroid hormone beta agonist | 0.016 0.004 CHEMBL527285 | CHEMBL527285 | |
| 0.076 | 0.117 | 0.138 | Chelator | 0.138 0.04 CHEMBL527285 | CHEMBL527285 | |
| 0.053 | 0.096 | 0.092 | HIV-1 integrase inhibitor | 0.092 0.03 CHEMBL527285 | CHEMBL527285 | |
| 0.041 | 0.085 | 0.113 | Phosphofructokinase-1 inhibitor | 0.113 0.027 CHEMBL527285 | CHEMBL527285 | |
| 0.123 | 0.173 | 0.196 | Succinate dehydrogenase inhibitor | 0.196 0.052 CHEMBL527285 | CHEMBL527285 | |
| 0.152 | 0.203 | 0.26 | Thyroid hormone beta antagonist | 0.26 0.112 CHEMBL527285 | CHEMBL527285 | |
| 0.227 | 0.283 | 0.287 | Caspase 9 stimulant | 0.287 0.208 CHEMBL527285 | CHEMBL527285 | |
| 0.007 | 0.068 | 0.016 | Thyroid hormone alpha antagonist | 0.016 0.01 CHEMBL527285 | CHEMBL527285 | |
| 0.17 | 0.232 | 0.345 | Sodium/bile acid cotransporter inhibitor | 0.202 0.185 CHEMBL4525790 0.345 0.043 CHEMBL527285 | CHEMBL527285 | |
| 0.132 | 0.201 | 0.221 | Cardiotonic | 0.221 0.102 CHEMBL527285 | CHEMBL527285 | |
| 0.075 | 0.146 | 0.12 | Cyclooxygenase 2 inhibitor | 0.12 0.08 CHEMBL527285 | CHEMBL527285 | |
| 0.003 | 0.075 | 0.009 | Integrin alphaVbeta5 antagonist | 0.009 0.007 CHEMBL527285 | CHEMBL527285 | |
| 0.015 | 0.088 | 0.043 | Retinoid X alpha receptor agonist | 0.043 0.018 CHEMBL527285 | CHEMBL527285 | |
| 0.048 | 0.123 | 0.079 | GABA aminotransferase inhibitor | 0.079 0.048 CHEMBL527285 | CHEMBL527285 | |
| 0.029 | 0.109 | 0.049 | Aldosterone antagonist | 0.049 0.031 CHEMBL527285 | CHEMBL527285 | |
| 0.028 | 0.119 | 0.052 | Aconitate hydratase inhibitor | 0.052 0.035 CHEMBL527285 | CHEMBL527285 | |
| 0.064 | 0.156 | 0.113 | Amylase inhibitor | 0.101 0.096 CHEMBL4525790 0.113 0.086 CHEMBL527285 | CHEMBL527285 | |
| 0.025 | 0.121 | 0.061 | Argininosuccinate synthase inhibitor | 0.061 0.036 CHEMBL527285 | CHEMBL527285 | |
| 0.021 | 0.125 | 0.042 | Retinoid X receptor antagonist | 0.042 0.02 CHEMBL527285 | CHEMBL527285 | |
| 0.019 | 0.124 | 0.039 | Retinoic acid alpha receptor agonist | 0.039 0.027 CHEMBL527285 | CHEMBL527285 | |
| 0.081 | 0.19 | 0.151 | Psychostimulant | 0.151 0.115 CHEMBL527285 | CHEMBL527285 | |
| 0.018 | 0.127 | 0.034 | Retinoid X alpha receptor antagonist | 0.034 0.024 CHEMBL527285 | CHEMBL527285 | |
| 0.019 | 0.146 | 0.054 | Thromboxane antagonist | 0.054 0.037 CHEMBL527285 | CHEMBL527285 | |
| 0.039 | 0.166 | 0.083 | Glutamate dehydrogenase inhibitor | 0.083 0.042 CHEMBL527285 | CHEMBL527285 | |
| 0.003 | 0.137 | 0.016 | G-protein-coupled receptor 120 agonist | 0.016 0.013 CHEMBL527285 | CHEMBL527285 | |
| 0.036 | 0.183 | 0.063 | Potassium channel large-conductance Ca-activated activator | 0.063 0.053 CHEMBL527285 | CHEMBL527285 | |
| 0.004 | 0.157 | 0.05 | Free fatty acid receptor 1 agonist | 0.05 0.005 CHEMBL527285 | CHEMBL527285 | |
| 0.147 | 0.303 | 0.214 | 5 Hydroxytryptamine uptake stimulant | 0.214 0.126 CHEMBL527285 | CHEMBL527285 | |
| 0.059 | 0.221 | 0.102 | DOPA decarboxylase inhibitor | 0.102 0.071 CHEMBL527285 | CHEMBL527285 | |
| 0.009 | 0.172 | 0.031 | Fumarate hydratase inhibitor | 0.031 0.027 CHEMBL527285 | CHEMBL527285 | |
| 0.014 | 0.178 | 0.043 | Thromboxane A2 antagonist | 0.043 0.042 CHEMBL527285 | CHEMBL527285 | |
| 0.043 | 0.213 | 0.107 | Cell adhesion molecule inhibitor | 0.107 0.03 CHEMBL527285 | CHEMBL527285 | |
| 0.014 | 0.185 | 0.08 | Aldose reductase inhibitor | 0.08 0.023 CHEMBL527285 | CHEMBL527285 | |
| 0.129 | 0.317 | 0.361 | Toll-Like receptor agonist | 0.361 0.077 CHEMBL527285 | CHEMBL527285 | |
| 0.04 | 0.235 | 0.178 | GABA C receptor agonist | 0.178 0.025 CHEMBL527285 | CHEMBL527285 | |
| 0.042 | 0.246 | 0.107 | Triose-phosphate isomerase inhibitor | 0.107 0.042 CHEMBL527285 | CHEMBL527285 | |
| 0.017 | 0.228 | 0.078 | Carbamoyl phosphate synthetase inhibitor | 0.078 0.029 CHEMBL527285 | CHEMBL527285 | |
| 0.011 | 0.241 | 0.057 | Prostaglandin antagonist | 0.057 0.034 CHEMBL527285 | CHEMBL527285 | |
| 0.044 | 0.276 | 0.143 | Alpha-N-acetylglucosaminidase inhibitor | 0.143 0.059 CHEMBL527285 | CHEMBL527285 | |
| 0.027 | 0.269 | 0.102 | Alcohol dehydrogenase inhibitor | 0.102 0.05 CHEMBL527285 | CHEMBL527285 | |
| 0.018 | 0.265 | 0.165 | Porphobilinogen synthase inhibitor | 0.165 0.017 CHEMBL527285 | CHEMBL527285 | |
| 0.019 | 0.268 | 0.076 | Glutamate decarboxylase inhibitor | 0.076 0.048 CHEMBL527285 | CHEMBL527285 | |
| 0.037 | 0.297 | 0.07 | GABA B receptor agonist | 0.07 0.068 CHEMBL527285 | CHEMBL527285 | |
| 0.034 | 0.296 | 0.084 | Uric acid excretion stimulant | 0.084 0.076 CHEMBL527285 | CHEMBL527285 | |
| 0.106 | 0.373 | 0.337 | Toll-Like receptor 7 agonist | 0.337 0.089 CHEMBL527285 | CHEMBL527285 | |
| 0.086 | 0.364 | 0.188 | Hypoxia-inducible factor 1 alpha inhibitor | 0.188 0.168 CHEMBL527285 | CHEMBL527285 | |
| 0.011 | 0.331 | 0.071 | Biliverdin reductase inhibitor | 0.071 0.031 CHEMBL527285 | CHEMBL527285 | |
| 0.014 | 0.363 | 0.058 | Sphingosine 1-phosphate receptor 5 agonist | 0.058 0.028 CHEMBL527285 | CHEMBL527285 | |
| 0.025 | 0.379 | 0.165 | Ferrochelatase inhibitor | 0.165 0.032 CHEMBL527285 | CHEMBL527285 | |
| 0.122 | 0.499 | 0.231 | Calcium channel L-type activator | 0.231 0.228 CHEMBL527285 | CHEMBL527285 | |
| 0.011 | 0.412 | 0.07 | Phenylalanine 4-hydroxylase inhibitor | 0.07 0.047 CHEMBL527285 | CHEMBL527285 | |
| 0.04 | 0.447 | 0.188 | Platelet adhesion inhibitor | 0.188 0.077 CHEMBL4525790 | CHEMBL4525790 | |
| 0.027 | 0.533 | 0.13 | Amyloid beta precursor protein antagonist | 0.13 0.126 CHEMBL4525790 | CHEMBL4525790 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |