Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7740.0040.869Anticonvulsant

0.664 0.005 CHEMBL3526444

0.629 0.006 CHEMBL3526726

0.632 0.005 CHEMBL3526727

0.66 0.005 CHEMBL3526549

0.772 0.004 CHEMBL3527118

0.367 0.026 CHEMBL3526443

0.627 0.006 CHEMBL3526583

0.869 0.004 CHEMBL4525793

0.661 0.005 CHEMBL4525794

CHEMBL4525793
0.3660.0020.366Benzodiazepine antagonist

0.165 0.003 CHEMBL3526444

0.11 0.004 CHEMBL3526726

0.132 0.003 CHEMBL3526727

0.078 0.005 CHEMBL3526549

0.142 0.003 CHEMBL3527118

0.135 0.003 CHEMBL3526443

0.127 0.003 CHEMBL3526583

0.149 0.003 CHEMBL4525793

0.133 0.003 CHEMBL4525794

0.3220.0620.405Spasmolytic

0.405 0.039 CHEMBL3526726

0.353 0.052 CHEMBL3526727

0.203 0.117 CHEMBL3526549

0.395 0.041 CHEMBL3527118

0.224 0.103 CHEMBL3526443

0.324 0.061 CHEMBL3526583

0.348 0.053 CHEMBL4525793

0.256 0.089 CHEMBL4525794

CHEMBL3526726
0.2560.0210.271Phosphodiesterase inhibitor

0.254 0.021 CHEMBL3526444

0.162 0.051 CHEMBL3526726

0.261 0.02 CHEMBL3526727

0.269 0.019 CHEMBL3526549

0.271 0.019 CHEMBL3527118

0.139 0.066 CHEMBL3526443

0.227 0.027 CHEMBL3526583

0.161 0.051 CHEMBL4525793

0.112 0.09 CHEMBL4525794

CHEMBL3527118
0.1950.0050.195Phosphodiesterase X inhibitor

0.171 0.005 CHEMBL3526444

0.088 0.012 CHEMBL3526726

0.134 0.007 CHEMBL3526727

0.161 0.005 CHEMBL3526549

0.181 0.005 CHEMBL3527118

0.091 0.011 CHEMBL3526443

0.114 0.009 CHEMBL3526583

0.099 0.01 CHEMBL4525793

0.063 0.019 CHEMBL4525794

0.1950.0050.195Phosphodiesterase 10A inhibitor

0.171 0.005 CHEMBL3526444

0.088 0.012 CHEMBL3526726

0.134 0.007 CHEMBL3526727

0.161 0.005 CHEMBL3526549

0.181 0.005 CHEMBL3527118

0.091 0.011 CHEMBL3526443

0.114 0.009 CHEMBL3526583

0.099 0.01 CHEMBL4525793

0.063 0.019 CHEMBL4525794

0.1760.0030.176Benzodiazepine receptor peripheral-type antagonist

0.067 0.004 CHEMBL3526444

0.153 0.003 CHEMBL3526726

0.143 0.003 CHEMBL3526727

0.053 0.006 CHEMBL3526549

0.137 0.003 CHEMBL3527118

0.144 0.003 CHEMBL3526443

0.133 0.003 CHEMBL3526583

0.134 0.003 CHEMBL4525793

0.13 0.003 CHEMBL4525794

0.2240.0770.224HERG channel blocker

0.167 0.113 CHEMBL3526444

0.143 0.138 CHEMBL3527118

0.1940.10.194Potassium channel (Voltage-sensitive) blocker

0.166 0.125 CHEMBL3526444

0.1110.0250.216Phosphodiesterase 3A inhibitor

0.102 0.03 CHEMBL3526444

0.216 0.007 CHEMBL3526727

0.131 0.019 CHEMBL3526549

0.146 0.016 CHEMBL3527118

0.09 0.041 CHEMBL3526443

0.192 0.009 CHEMBL3526583

0.083 0.051 CHEMBL4525793

0.079 0.057 CHEMBL4525794

CHEMBL3526727
0.1310.0480.146GABA receptor agonist

0.146 0.038 CHEMBL3526726

0.127 0.051 CHEMBL3526727

0.123 0.054 CHEMBL3527118

0.091 0.088 CHEMBL3526443

0.097 0.08 CHEMBL3526583

0.111 0.065 CHEMBL4525793

CHEMBL3526726
0.1390.0570.175Sphingosine 1-phosphate receptor 2 antagonist

0.175 0.017 CHEMBL3526444

0.154 0.036 CHEMBL3526549

0.117 0.104 CHEMBL3527118

0.125 0.085 CHEMBL4525793

0.114 0.113 CHEMBL4525794

CHEMBL3526444
0.1030.0350.103GABA A receptor agonist

0.092 0.046 CHEMBL3526726

0.097 0.04 CHEMBL3526727

0.096 0.042 CHEMBL3527118

0.081 0.061 CHEMBL3526443

0.081 0.062 CHEMBL3526583

0.083 0.059 CHEMBL4525793

0.0880.020.088Orexin receptor antagonist
0.0980.0320.0985 Hydroxytryptamine 1F antagonist

0.071 0.049 CHEMBL3526726

0.064 0.055 CHEMBL3526727

0.073 0.048 CHEMBL3526443

0.062 0.057 CHEMBL3526583

0.0850.0280.085Orexin receptor 1 antagonist
0.080.0240.085 Hydroxytryptamine 5A antagonist

0.06 0.045 CHEMBL3526444

0.0760.0260.081Caspase 9 inhibitor

0.081 0.022 CHEMBL3526444

0.078 0.025 CHEMBL3526727

0.078 0.024 CHEMBL3526549

0.074 0.028 CHEMBL3527118

0.073 0.028 CHEMBL3526443

0.074 0.028 CHEMBL3526583

0.073 0.029 CHEMBL4525793

0.073 0.029 CHEMBL4525794

CHEMBL3526444
0.1080.0660.262Electron transport complex I inhibitor

0.116 0.052 CHEMBL3526444

0.099 0.084 CHEMBL3526727

0.108 0.066 CHEMBL3526549

0.1 0.082 CHEMBL3527118

0.262 0.005 CHEMBL3526443

0.1 0.082 CHEMBL3526583

0.099 0.085 CHEMBL4525793

0.099 0.085 CHEMBL4525794

CHEMBL3526443
0.1120.0710.127Estrogen antagonist

0.107 0.081 CHEMBL3526444

0.127 0.042 CHEMBL3526726

0.107 0.081 CHEMBL3526727

0.105 0.087 CHEMBL3526549

0.109 0.077 CHEMBL3527118

0.121 0.053 CHEMBL3526443

0.105 0.086 CHEMBL3526583

0.108 0.08 CHEMBL4525793

0.106 0.083 CHEMBL4525794

CHEMBL3526726
0.180.140.22Cardiotonic

0.22 0.102 CHEMBL3526726

0.165 0.158 CHEMBL3526549

0.191 0.127 CHEMBL3527118

0.172 0.149 CHEMBL3526583

0.175 0.146 CHEMBL4525793

CHEMBL3526726
0.0670.0280.0675 Hydroxytryptamine 5 antagonist

0.053 0.049 CHEMBL3526444

0.0450.0060.045Corticotropin releasing factor 1 receptor antagonist

0.039 0.008 CHEMBL3526444

0.027 0.012 CHEMBL3526726

0.02 0.019 CHEMBL3526549

0.022 0.016 CHEMBL3527118

0.022 0.016 CHEMBL3526583

0.0420.0090.083Kainate receptor 4 antagonist

0.083 0.004 CHEMBL3526726

0.041 0.009 CHEMBL3526727

0.036 0.011 CHEMBL3527118

0.042 0.009 CHEMBL3526443

0.036 0.011 CHEMBL3526583

0.054 0.006 CHEMBL4525793

0.054 0.006 CHEMBL4525794

CHEMBL3526726
0.0780.0510.085Estrogen receptor alpha antagonist

0.07 0.068 CHEMBL3526444

0.085 0.041 CHEMBL3526726

0.076 0.056 CHEMBL3526443

CHEMBL3526726
0.0820.0570.092Caspase 7 inhibitor

0.092 0.038 CHEMBL3526444

CHEMBL3526444
0.0920.0690.117Interleukin 1 beta converting enzyme inhibitor

0.117 0.038 CHEMBL3526444

0.096 0.062 CHEMBL3526549

0.091 0.07 CHEMBL4525793

0.089 0.073 CHEMBL4525794

CHEMBL3526444
0.0350.0130.035Caspase 6 inhibitor

0.035 0.012 CHEMBL3526444

0.035 0.013 CHEMBL3526727

0.034 0.014 CHEMBL3526549

0.033 0.015 CHEMBL3527118

0.034 0.014 CHEMBL3526443

0.033 0.015 CHEMBL3526583

0.034 0.013 CHEMBL4525793

0.034 0.013 CHEMBL4525794

0.0410.020.041Orexin receptor 2 antagonist
0.0570.0370.068Phosphodiesterase II inhibitor

0.061 0.031 CHEMBL3526444

0.054 0.04 CHEMBL3526727

0.068 0.024 CHEMBL3526549

0.064 0.028 CHEMBL3527118

0.064 0.028 CHEMBL3526583

CHEMBL3526549
0.0450.0290.067Phosphodiesterase 3B inhibitor

0.043 0.032 CHEMBL3526444

0.067 0.017 CHEMBL3526727

0.059 0.02 CHEMBL3526549

0.064 0.018 CHEMBL3527118

0.045 0.03 CHEMBL3526443

0.05 0.025 CHEMBL3526583

CHEMBL3526727
0.150.1350.15Potassium channel blocker
0.1970.1830.367Apoptosis antagonist

0.228 0.149 CHEMBL3526444

0.249 0.129 CHEMBL3526727

0.264 0.114 CHEMBL3526549

0.243 0.135 CHEMBL3527118

0.367 0.049 CHEMBL3526443

0.254 0.124 CHEMBL3526583

0.239 0.138 CHEMBL4525793

0.223 0.154 CHEMBL4525794

CHEMBL3526443
0.0490.0350.061Phosphodiesterase 2A inhibitor

0.053 0.03 CHEMBL3526444

0.047 0.038 CHEMBL3526727

0.061 0.023 CHEMBL3526549

0.056 0.027 CHEMBL3527118

0.056 0.027 CHEMBL3526583

CHEMBL3526549
0.0620.0490.0625 Hydroxytryptamine 1B antagonist
0.0680.0590.072Phosphodiesterase VIII inhibitor

0.072 0.05 CHEMBL3526444

CHEMBL3526444
0.130.1210.139TRKC antagonist

0.139 0.111 CHEMBL3526444

CHEMBL3526444
0.0570.0480.091Adenosine A2a receptor antagonist

0.091 0.027 CHEMBL3526444

0.068 0.038 CHEMBL3526726

0.09 0.028 CHEMBL3526549

0.056 0.048 CHEMBL3527118

CHEMBL3526444
0.0650.0580.075Benzodiazepine agonist

0.068 0.053 CHEMBL3526726

0.075 0.045 CHEMBL3527118

CHEMBL3527118
0.020.0150.055Kainate receptor 5 antagonist

0.055 0.005 CHEMBL3526726

0.021 0.014 CHEMBL3526727

0.021 0.014 CHEMBL3526443

0.035 0.008 CHEMBL4525793

0.035 0.008 CHEMBL4525794

CHEMBL3526726
0.0160.0130.033Kainate receptor 3 antagonist

0.033 0.005 CHEMBL3526726

0.016 0.013 CHEMBL3526727

0.016 0.013 CHEMBL3526443

0.021 0.008 CHEMBL4525793

0.021 0.008 CHEMBL4525794

CHEMBL3526726
0.0570.0550.109Phosphodiesterase III inhibitor

0.06 0.052 CHEMBL3526444

0.109 0.019 CHEMBL3526727

0.079 0.036 CHEMBL3526549

0.077 0.038 CHEMBL3527118

0.097 0.024 CHEMBL3526583

CHEMBL3526727
0.020.0190.028Leukotriene B4 receptor 2 antagonist

0.028 0.01 CHEMBL3526726

0.022 0.016 CHEMBL3526727

0.02 0.019 CHEMBL3527118

0.022 0.016 CHEMBL3526443

0.02 0.019 CHEMBL3526583

0.024 0.013 CHEMBL4525793

0.024 0.013 CHEMBL4525794

CHEMBL3526726
0.1270.1280.16Amyloid beta aggregation inhibitor

0.16 0.101 CHEMBL3526443

CHEMBL3526443
0.0250.0290.027Glucosylceramidase stimulant

0.026 0.023 CHEMBL3526444

0.027 0.018 CHEMBL3526726

CHEMBL3526726
0.0350.0470.051Angiotensin AT1 receptor antagonist

0.05 0.018 CHEMBL3526726

0.038 0.037 CHEMBL3527118

0.038 0.037 CHEMBL3526583

0.051 0.017 CHEMBL4525793

0.045 0.025 CHEMBL4525794

CHEMBL4525793
0.020.0330.066AMPA 2 receptor antagonist

0.066 0.008 CHEMBL3526726

0.031 0.02 CHEMBL3526727

0.028 0.023 CHEMBL3527118

0.041 0.014 CHEMBL4525793

0.037 0.016 CHEMBL4525794

CHEMBL3526726
0.0470.0660.083Adenosine A2 receptor antagonist

0.083 0.033 CHEMBL3526444

0.058 0.05 CHEMBL3526726

0.077 0.036 CHEMBL3526549

CHEMBL3526444
0.0770.0960.087ABCA1 expression enhancer

0.087 0.071 CHEMBL4525793

0.087 0.071 CHEMBL4525794

CHEMBL4525794
0.0350.0550.04Guanylate cyclase stimulant

0.04 0.037 CHEMBL4525793

CHEMBL4525793
0.050.0750.098Phosphodiesterase 4B inhibitor

0.061 0.055 CHEMBL3526444

0.098 0.026 CHEMBL3526727

0.082 0.034 CHEMBL3526549

0.066 0.048 CHEMBL3527118

0.067 0.047 CHEMBL3526583

CHEMBL3526727
0.2180.2450.536Calcium channel L-type activator

0.262 0.193 CHEMBL3526444

0.408 0.076 CHEMBL3526726

0.508 0.025 CHEMBL3526727

0.536 0.016 CHEMBL3526549

0.53 0.018 CHEMBL3527118

0.271 0.184 CHEMBL3526443

0.53 0.018 CHEMBL3526583

0.305 0.153 CHEMBL4525793

0.305 0.153 CHEMBL4525794

CHEMBL3526549
0.1490.1810.286Calpain inhibitor

0.286 0.037 CHEMBL3526444

0.247 0.068 CHEMBL3526549

CHEMBL3526444
0.0070.0470.012Glucose-dependent insulinotropic receptor antagonist

0.012 0.008 CHEMBL3526443

CHEMBL3526443
0.0220.0630.037Angiotensin II receptor antagonist

0.037 0.019 CHEMBL3526726

0.035 0.022 CHEMBL4525793

CHEMBL3526726
0.0060.0570.057Prostaglandin EP1 antagonist

0.057 0.005 CHEMBL4525793

0.023 0.012 CHEMBL4525794

CHEMBL4525793
0.0740.1310.203M18 aspartyl aminopeptidase inhibitor

0.203 0.033 CHEMBL3526726

CHEMBL3526726
0.0460.1250.059Heme oxygenase stimulant

0.059 0.049 CHEMBL3526726

CHEMBL3526726
0.0420.1240.092Phosphodiesterase IV inhibitor

0.092 0.052 CHEMBL3526727

CHEMBL3526727
0.0620.1460.122Estrogen receptor beta antagonist

0.122 0.03 CHEMBL3526726

CHEMBL3526726
0.020.1060.041Melatonin receptor 1A agonist

0.041 0.013 CHEMBL3526444

0.032 0.027 CHEMBL3526549

CHEMBL3526444
0.0540.1420.092Histamine H2 receptor antagonist

0.092 0.044 CHEMBL3526444

CHEMBL3526444
0.0480.150.072Opioid kappa receptor antagonist

0.072 0.071 CHEMBL3526726

CHEMBL3526726
0.1170.2270.298Cyclic AMP phosphodiesterase inhibitor

0.298 0.043 CHEMBL3526726

0.161 0.134 CHEMBL3527118

CHEMBL3526726
0.1610.2840.255Ca(v)3.3 blocker

0.255 0.094 CHEMBL3526444

0.206 0.179 CHEMBL3526549

CHEMBL3526444
0.0640.1980.196Cyclooxygenase inhibitor

0.196 0.043 CHEMBL3526443

CHEMBL3526443
0.1280.2680.373Calpain 2 inhibitor

0.373 0.075 CHEMBL3526444

0.222 0.169 CHEMBL3526549

CHEMBL3526444
0.1460.2970.416GABA C receptor rho-3 antagonist

0.416 0.055 CHEMBL3526726

CHEMBL3526726
0.0550.2120.082Ca(v)3.1 blocker

0.082 0.055 CHEMBL3526444

CHEMBL3526444
0.0960.2540.235Vasodilator

0.235 0.078 CHEMBL3526726

0.16 0.143 CHEMBL3526549

CHEMBL3526726
0.010.1730.034Nicotinic acid receptor 2 agonist

0.034 0.027 CHEMBL4525793

0.034 0.027 CHEMBL4525794

CHEMBL4525794
0.0140.1820.052Prostaglandin antagonist

0.052 0.038 CHEMBL4525793

CHEMBL4525793
0.0320.2020.144Potassium channel (Ca-activated) activator

0.144 0.03 CHEMBL3526726

CHEMBL3526726
0.0280.2020.071Antiviral (Hepatitis D)

0.071 0.013 CHEMBL3526727

0.069 0.014 CHEMBL3526583

CHEMBL3526727
0.0130.1920.075Prostaglandin E2 antagonist

0.075 0.021 CHEMBL4525793

CHEMBL4525793
0.0610.2840.121Farnesoid X receptor antagonist

0.121 0.101 CHEMBL3526726

CHEMBL3526726
0.020.2450.145Porphobilinogen synthase inhibitor

0.145 0.022 CHEMBL3526726

CHEMBL3526726
0.060.2930.28Amyloid beta precursor protein antagonist

0.28 0.023 CHEMBL4525794

CHEMBL4525794
0.1570.4020.548Antiinflammatory

0.292 0.223 CHEMBL3526549

0.548 0.069 CHEMBL3526443

CHEMBL3526443
0.0060.2510.026AMPA 3 receptor antagonist

0.026 0.024 CHEMBL3526726

CHEMBL3526726
0.060.3470.141GABA C receptor rho-2 antagonist

0.141 0.087 CHEMBL3526726

CHEMBL3526726
0.070.3670.206Thyroid hormone beta antagonist

0.206 0.149 CHEMBL3526726

CHEMBL3526726
0.0670.3810.216Thyroid hormone antagonist

0.216 0.148 CHEMBL3526726

CHEMBL3526726
0.0550.3790.172Streptokinase A inhibitor

0.172 0.153 CHEMBL3526726

CHEMBL3526726
0.0760.4050.147Death-associated protein kinase 2 inhibitor

0.147 0.114 CHEMBL3526726

CHEMBL3526726
0.0130.3660.062Phenylalanine 4-hydroxylase inhibitor

0.062 0.055 CHEMBL3526726

CHEMBL3526726
0.0450.4010.192Prostaglandin dehydrogenase inhibitor

0.192 0.162 CHEMBL3526726

CHEMBL3526726
0.1180.4820.2535 Hydroxytryptamine release inhibitor

0.253 0.224 CHEMBL3526726

CHEMBL3526726
0.0250.3980.086Uric acid excretion stimulant

0.086 0.072 CHEMBL4525793

CHEMBL4525793
0.0220.4050.106Creatine kinase inhibitor

0.106 0.053 CHEMBL3526726

CHEMBL3526726
0.0890.5060.229Tyrosine 3 hydroxylase inhibitor

0.229 0.091 CHEMBL3526726

CHEMBL3526726
0.0450.4640.262DNA polymerase beta inhibitor

0.262 0.186 CHEMBL3526726

CHEMBL3526726
0.060.4860.234Transcription factor inhibitor

0.234 0.199 CHEMBL3526726

CHEMBL3526726
0.0490.4810.136CF transmembrane conductance regulator agonist

0.136 0.104 CHEMBL3526726

CHEMBL3526726
0.0370.4850.292Alpha-glucosidase inhibitor

0.292 0.164 CHEMBL3526726

CHEMBL3526726
0.0560.5160.152Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.152 0.144 CHEMBL3526726

CHEMBL3526726
0.0410.5410.3515-Lipoxygenase inhibitor

0.35 0.099 CHEMBL3526726

CHEMBL3526726
0.0510.5910.142Neurotensin receptor agonist

0.142 0.123 CHEMBL3526726

CHEMBL3526726
0.0110.6720.103Chelator

0.103 0.073 CHEMBL3526443

CHEMBL3526443
Ext Pa Pi Pmax Activity Other Results ID Pa_max