| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.774 | 0.004 | 0.869 | Anticonvulsant | 0.664 0.005 CHEMBL3526444 0.629 0.006 CHEMBL3526726 0.632 0.005 CHEMBL3526727 0.66 0.005 CHEMBL3526549 0.772 0.004 CHEMBL3527118 0.367 0.026 CHEMBL3526443 0.627 0.006 CHEMBL3526583 0.869 0.004 CHEMBL4525793 0.661 0.005 CHEMBL4525794 | CHEMBL4525793 | |
| 0.366 | 0.002 | 0.366 | Benzodiazepine antagonist | 0.165 0.003 CHEMBL3526444 0.11 0.004 CHEMBL3526726 0.132 0.003 CHEMBL3526727 0.078 0.005 CHEMBL3526549 0.142 0.003 CHEMBL3527118 0.135 0.003 CHEMBL3526443 0.127 0.003 CHEMBL3526583 0.149 0.003 CHEMBL4525793 0.133 0.003 CHEMBL4525794 | ||
| 0.322 | 0.062 | 0.405 | Spasmolytic | 0.405 0.039 CHEMBL3526726 0.353 0.052 CHEMBL3526727 0.203 0.117 CHEMBL3526549 0.395 0.041 CHEMBL3527118 0.224 0.103 CHEMBL3526443 0.324 0.061 CHEMBL3526583 0.348 0.053 CHEMBL4525793 0.256 0.089 CHEMBL4525794 | CHEMBL3526726 | |
| 0.256 | 0.021 | 0.271 | Phosphodiesterase inhibitor | 0.254 0.021 CHEMBL3526444 0.162 0.051 CHEMBL3526726 0.261 0.02 CHEMBL3526727 0.269 0.019 CHEMBL3526549 0.271 0.019 CHEMBL3527118 0.139 0.066 CHEMBL3526443 0.227 0.027 CHEMBL3526583 0.161 0.051 CHEMBL4525793 0.112 0.09 CHEMBL4525794 | CHEMBL3527118 | |
| 0.195 | 0.005 | 0.195 | Phosphodiesterase X inhibitor | 0.171 0.005 CHEMBL3526444 0.088 0.012 CHEMBL3526726 0.134 0.007 CHEMBL3526727 0.161 0.005 CHEMBL3526549 0.181 0.005 CHEMBL3527118 0.091 0.011 CHEMBL3526443 0.114 0.009 CHEMBL3526583 0.099 0.01 CHEMBL4525793 0.063 0.019 CHEMBL4525794 | ||
| 0.195 | 0.005 | 0.195 | Phosphodiesterase 10A inhibitor | 0.171 0.005 CHEMBL3526444 0.088 0.012 CHEMBL3526726 0.134 0.007 CHEMBL3526727 0.161 0.005 CHEMBL3526549 0.181 0.005 CHEMBL3527118 0.091 0.011 CHEMBL3526443 0.114 0.009 CHEMBL3526583 0.099 0.01 CHEMBL4525793 0.063 0.019 CHEMBL4525794 | ||
| 0.176 | 0.003 | 0.176 | Benzodiazepine receptor peripheral-type antagonist | 0.067 0.004 CHEMBL3526444 0.153 0.003 CHEMBL3526726 0.143 0.003 CHEMBL3526727 0.053 0.006 CHEMBL3526549 0.137 0.003 CHEMBL3527118 0.144 0.003 CHEMBL3526443 0.133 0.003 CHEMBL3526583 0.134 0.003 CHEMBL4525793 0.13 0.003 CHEMBL4525794 | ||
| 0.224 | 0.077 | 0.224 | HERG channel blocker | 0.167 0.113 CHEMBL3526444 0.143 0.138 CHEMBL3527118 | ||
| 0.194 | 0.1 | 0.194 | Potassium channel (Voltage-sensitive) blocker | 0.166 0.125 CHEMBL3526444 | ||
| 0.111 | 0.025 | 0.216 | Phosphodiesterase 3A inhibitor | 0.102 0.03 CHEMBL3526444 0.216 0.007 CHEMBL3526727 0.131 0.019 CHEMBL3526549 0.146 0.016 CHEMBL3527118 0.09 0.041 CHEMBL3526443 0.192 0.009 CHEMBL3526583 0.083 0.051 CHEMBL4525793 0.079 0.057 CHEMBL4525794 | CHEMBL3526727 | |
| 0.131 | 0.048 | 0.146 | GABA receptor agonist | 0.146 0.038 CHEMBL3526726 0.127 0.051 CHEMBL3526727 0.123 0.054 CHEMBL3527118 0.091 0.088 CHEMBL3526443 0.097 0.08 CHEMBL3526583 0.111 0.065 CHEMBL4525793 | CHEMBL3526726 | |
| 0.139 | 0.057 | 0.175 | Sphingosine 1-phosphate receptor 2 antagonist | 0.175 0.017 CHEMBL3526444 0.154 0.036 CHEMBL3526549 0.117 0.104 CHEMBL3527118 0.125 0.085 CHEMBL4525793 0.114 0.113 CHEMBL4525794 | CHEMBL3526444 | |
| 0.103 | 0.035 | 0.103 | GABA A receptor agonist | 0.092 0.046 CHEMBL3526726 0.097 0.04 CHEMBL3526727 0.096 0.042 CHEMBL3527118 0.081 0.061 CHEMBL3526443 0.081 0.062 CHEMBL3526583 0.083 0.059 CHEMBL4525793 | ||
| 0.088 | 0.02 | 0.088 | Orexin receptor antagonist | |||
| 0.098 | 0.032 | 0.098 | 5 Hydroxytryptamine 1F antagonist | 0.071 0.049 CHEMBL3526726 0.064 0.055 CHEMBL3526727 0.073 0.048 CHEMBL3526443 0.062 0.057 CHEMBL3526583 | ||
| 0.085 | 0.028 | 0.085 | Orexin receptor 1 antagonist | |||
| 0.08 | 0.024 | 0.08 | 5 Hydroxytryptamine 5A antagonist | 0.06 0.045 CHEMBL3526444 | ||
| 0.076 | 0.026 | 0.081 | Caspase 9 inhibitor | 0.081 0.022 CHEMBL3526444 0.078 0.025 CHEMBL3526727 0.078 0.024 CHEMBL3526549 0.074 0.028 CHEMBL3527118 0.073 0.028 CHEMBL3526443 0.074 0.028 CHEMBL3526583 0.073 0.029 CHEMBL4525793 0.073 0.029 CHEMBL4525794 | CHEMBL3526444 | |
| 0.108 | 0.066 | 0.262 | Electron transport complex I inhibitor | 0.116 0.052 CHEMBL3526444 0.099 0.084 CHEMBL3526727 0.108 0.066 CHEMBL3526549 0.1 0.082 CHEMBL3527118 0.262 0.005 CHEMBL3526443 0.1 0.082 CHEMBL3526583 0.099 0.085 CHEMBL4525793 0.099 0.085 CHEMBL4525794 | CHEMBL3526443 | |
| 0.112 | 0.071 | 0.127 | Estrogen antagonist | 0.107 0.081 CHEMBL3526444 0.127 0.042 CHEMBL3526726 0.107 0.081 CHEMBL3526727 0.105 0.087 CHEMBL3526549 0.109 0.077 CHEMBL3527118 0.121 0.053 CHEMBL3526443 0.105 0.086 CHEMBL3526583 0.108 0.08 CHEMBL4525793 0.106 0.083 CHEMBL4525794 | CHEMBL3526726 | |
| 0.18 | 0.14 | 0.22 | Cardiotonic | 0.22 0.102 CHEMBL3526726 0.165 0.158 CHEMBL3526549 0.191 0.127 CHEMBL3527118 0.172 0.149 CHEMBL3526583 0.175 0.146 CHEMBL4525793 | CHEMBL3526726 | |
| 0.067 | 0.028 | 0.067 | 5 Hydroxytryptamine 5 antagonist | 0.053 0.049 CHEMBL3526444 | ||
| 0.045 | 0.006 | 0.045 | Corticotropin releasing factor 1 receptor antagonist | 0.039 0.008 CHEMBL3526444 0.027 0.012 CHEMBL3526726 0.02 0.019 CHEMBL3526549 0.022 0.016 CHEMBL3527118 0.022 0.016 CHEMBL3526583 | ||
| 0.042 | 0.009 | 0.083 | Kainate receptor 4 antagonist | 0.083 0.004 CHEMBL3526726 0.041 0.009 CHEMBL3526727 0.036 0.011 CHEMBL3527118 0.042 0.009 CHEMBL3526443 0.036 0.011 CHEMBL3526583 0.054 0.006 CHEMBL4525793 0.054 0.006 CHEMBL4525794 | CHEMBL3526726 | |
| 0.078 | 0.051 | 0.085 | Estrogen receptor alpha antagonist | 0.07 0.068 CHEMBL3526444 0.085 0.041 CHEMBL3526726 0.076 0.056 CHEMBL3526443 | CHEMBL3526726 | |
| 0.082 | 0.057 | 0.092 | Caspase 7 inhibitor | 0.092 0.038 CHEMBL3526444 | CHEMBL3526444 | |
| 0.092 | 0.069 | 0.117 | Interleukin 1 beta converting enzyme inhibitor | 0.117 0.038 CHEMBL3526444 0.096 0.062 CHEMBL3526549 0.091 0.07 CHEMBL4525793 0.089 0.073 CHEMBL4525794 | CHEMBL3526444 | |
| 0.035 | 0.013 | 0.035 | Caspase 6 inhibitor | 0.035 0.012 CHEMBL3526444 0.035 0.013 CHEMBL3526727 0.034 0.014 CHEMBL3526549 0.033 0.015 CHEMBL3527118 0.034 0.014 CHEMBL3526443 0.033 0.015 CHEMBL3526583 0.034 0.013 CHEMBL4525793 0.034 0.013 CHEMBL4525794 | ||
| 0.041 | 0.02 | 0.041 | Orexin receptor 2 antagonist | |||
| 0.057 | 0.037 | 0.068 | Phosphodiesterase II inhibitor | 0.061 0.031 CHEMBL3526444 0.054 0.04 CHEMBL3526727 0.068 0.024 CHEMBL3526549 0.064 0.028 CHEMBL3527118 0.064 0.028 CHEMBL3526583 | CHEMBL3526549 | |
| 0.045 | 0.029 | 0.067 | Phosphodiesterase 3B inhibitor | 0.043 0.032 CHEMBL3526444 0.067 0.017 CHEMBL3526727 0.059 0.02 CHEMBL3526549 0.064 0.018 CHEMBL3527118 0.045 0.03 CHEMBL3526443 0.05 0.025 CHEMBL3526583 | CHEMBL3526727 | |
| 0.15 | 0.135 | 0.15 | Potassium channel blocker | |||
| 0.197 | 0.183 | 0.367 | Apoptosis antagonist | 0.228 0.149 CHEMBL3526444 0.249 0.129 CHEMBL3526727 0.264 0.114 CHEMBL3526549 0.243 0.135 CHEMBL3527118 0.367 0.049 CHEMBL3526443 0.254 0.124 CHEMBL3526583 0.239 0.138 CHEMBL4525793 0.223 0.154 CHEMBL4525794 | CHEMBL3526443 | |
| 0.049 | 0.035 | 0.061 | Phosphodiesterase 2A inhibitor | 0.053 0.03 CHEMBL3526444 0.047 0.038 CHEMBL3526727 0.061 0.023 CHEMBL3526549 0.056 0.027 CHEMBL3527118 0.056 0.027 CHEMBL3526583 | CHEMBL3526549 | |
| 0.062 | 0.049 | 0.062 | 5 Hydroxytryptamine 1B antagonist | |||
| 0.068 | 0.059 | 0.072 | Phosphodiesterase VIII inhibitor | 0.072 0.05 CHEMBL3526444 | CHEMBL3526444 | |
| 0.13 | 0.121 | 0.139 | TRKC antagonist | 0.139 0.111 CHEMBL3526444 | CHEMBL3526444 | |
| 0.057 | 0.048 | 0.091 | Adenosine A2a receptor antagonist | 0.091 0.027 CHEMBL3526444 0.068 0.038 CHEMBL3526726 0.09 0.028 CHEMBL3526549 0.056 0.048 CHEMBL3527118 | CHEMBL3526444 | |
| 0.065 | 0.058 | 0.075 | Benzodiazepine agonist | 0.068 0.053 CHEMBL3526726 0.075 0.045 CHEMBL3527118 | CHEMBL3527118 | |
| 0.02 | 0.015 | 0.055 | Kainate receptor 5 antagonist | 0.055 0.005 CHEMBL3526726 0.021 0.014 CHEMBL3526727 0.021 0.014 CHEMBL3526443 0.035 0.008 CHEMBL4525793 0.035 0.008 CHEMBL4525794 | CHEMBL3526726 | |
| 0.016 | 0.013 | 0.033 | Kainate receptor 3 antagonist | 0.033 0.005 CHEMBL3526726 0.016 0.013 CHEMBL3526727 0.016 0.013 CHEMBL3526443 0.021 0.008 CHEMBL4525793 0.021 0.008 CHEMBL4525794 | CHEMBL3526726 | |
| 0.057 | 0.055 | 0.109 | Phosphodiesterase III inhibitor | 0.06 0.052 CHEMBL3526444 0.109 0.019 CHEMBL3526727 0.079 0.036 CHEMBL3526549 0.077 0.038 CHEMBL3527118 0.097 0.024 CHEMBL3526583 | CHEMBL3526727 | |
| 0.02 | 0.019 | 0.028 | Leukotriene B4 receptor 2 antagonist | 0.028 0.01 CHEMBL3526726 0.022 0.016 CHEMBL3526727 0.02 0.019 CHEMBL3527118 0.022 0.016 CHEMBL3526443 0.02 0.019 CHEMBL3526583 0.024 0.013 CHEMBL4525793 0.024 0.013 CHEMBL4525794 | CHEMBL3526726 | |
| 0.127 | 0.128 | 0.16 | Amyloid beta aggregation inhibitor | 0.16 0.101 CHEMBL3526443 | CHEMBL3526443 | |
| 0.025 | 0.029 | 0.027 | Glucosylceramidase stimulant | 0.026 0.023 CHEMBL3526444 0.027 0.018 CHEMBL3526726 | CHEMBL3526726 | |
| 0.035 | 0.047 | 0.051 | Angiotensin AT1 receptor antagonist | 0.05 0.018 CHEMBL3526726 0.038 0.037 CHEMBL3527118 0.038 0.037 CHEMBL3526583 0.051 0.017 CHEMBL4525793 0.045 0.025 CHEMBL4525794 | CHEMBL4525793 | |
| 0.02 | 0.033 | 0.066 | AMPA 2 receptor antagonist | 0.066 0.008 CHEMBL3526726 0.031 0.02 CHEMBL3526727 0.028 0.023 CHEMBL3527118 0.041 0.014 CHEMBL4525793 0.037 0.016 CHEMBL4525794 | CHEMBL3526726 | |
| 0.047 | 0.066 | 0.083 | Adenosine A2 receptor antagonist | 0.083 0.033 CHEMBL3526444 0.058 0.05 CHEMBL3526726 0.077 0.036 CHEMBL3526549 | CHEMBL3526444 | |
| 0.077 | 0.096 | 0.087 | ABCA1 expression enhancer | 0.087 0.071 CHEMBL4525793 0.087 0.071 CHEMBL4525794 | CHEMBL4525794 | |
| 0.035 | 0.055 | 0.04 | Guanylate cyclase stimulant | 0.04 0.037 CHEMBL4525793 | CHEMBL4525793 | |
| 0.05 | 0.075 | 0.098 | Phosphodiesterase 4B inhibitor | 0.061 0.055 CHEMBL3526444 0.098 0.026 CHEMBL3526727 0.082 0.034 CHEMBL3526549 0.066 0.048 CHEMBL3527118 0.067 0.047 CHEMBL3526583 | CHEMBL3526727 | |
| 0.218 | 0.245 | 0.536 | Calcium channel L-type activator | 0.262 0.193 CHEMBL3526444 0.408 0.076 CHEMBL3526726 0.508 0.025 CHEMBL3526727 0.536 0.016 CHEMBL3526549 0.53 0.018 CHEMBL3527118 0.271 0.184 CHEMBL3526443 0.53 0.018 CHEMBL3526583 0.305 0.153 CHEMBL4525793 0.305 0.153 CHEMBL4525794 | CHEMBL3526549 | |
| 0.149 | 0.181 | 0.286 | Calpain inhibitor | 0.286 0.037 CHEMBL3526444 0.247 0.068 CHEMBL3526549 | CHEMBL3526444 | |
| 0.007 | 0.047 | 0.012 | Glucose-dependent insulinotropic receptor antagonist | 0.012 0.008 CHEMBL3526443 | CHEMBL3526443 | |
| 0.022 | 0.063 | 0.037 | Angiotensin II receptor antagonist | 0.037 0.019 CHEMBL3526726 0.035 0.022 CHEMBL4525793 | CHEMBL3526726 | |
| 0.006 | 0.057 | 0.057 | Prostaglandin EP1 antagonist | 0.057 0.005 CHEMBL4525793 0.023 0.012 CHEMBL4525794 | CHEMBL4525793 | |
| 0.074 | 0.131 | 0.203 | M18 aspartyl aminopeptidase inhibitor | 0.203 0.033 CHEMBL3526726 | CHEMBL3526726 | |
| 0.046 | 0.125 | 0.059 | Heme oxygenase stimulant | 0.059 0.049 CHEMBL3526726 | CHEMBL3526726 | |
| 0.042 | 0.124 | 0.092 | Phosphodiesterase IV inhibitor | 0.092 0.052 CHEMBL3526727 | CHEMBL3526727 | |
| 0.062 | 0.146 | 0.122 | Estrogen receptor beta antagonist | 0.122 0.03 CHEMBL3526726 | CHEMBL3526726 | |
| 0.02 | 0.106 | 0.041 | Melatonin receptor 1A agonist | 0.041 0.013 CHEMBL3526444 0.032 0.027 CHEMBL3526549 | CHEMBL3526444 | |
| 0.054 | 0.142 | 0.092 | Histamine H2 receptor antagonist | 0.092 0.044 CHEMBL3526444 | CHEMBL3526444 | |
| 0.048 | 0.15 | 0.072 | Opioid kappa receptor antagonist | 0.072 0.071 CHEMBL3526726 | CHEMBL3526726 | |
| 0.117 | 0.227 | 0.298 | Cyclic AMP phosphodiesterase inhibitor | 0.298 0.043 CHEMBL3526726 0.161 0.134 CHEMBL3527118 | CHEMBL3526726 | |
| 0.161 | 0.284 | 0.255 | Ca(v)3.3 blocker | 0.255 0.094 CHEMBL3526444 0.206 0.179 CHEMBL3526549 | CHEMBL3526444 | |
| 0.064 | 0.198 | 0.196 | Cyclooxygenase inhibitor | 0.196 0.043 CHEMBL3526443 | CHEMBL3526443 | |
| 0.128 | 0.268 | 0.373 | Calpain 2 inhibitor | 0.373 0.075 CHEMBL3526444 0.222 0.169 CHEMBL3526549 | CHEMBL3526444 | |
| 0.146 | 0.297 | 0.416 | GABA C receptor rho-3 antagonist | 0.416 0.055 CHEMBL3526726 | CHEMBL3526726 | |
| 0.055 | 0.212 | 0.082 | Ca(v)3.1 blocker | 0.082 0.055 CHEMBL3526444 | CHEMBL3526444 | |
| 0.096 | 0.254 | 0.235 | Vasodilator | 0.235 0.078 CHEMBL3526726 0.16 0.143 CHEMBL3526549 | CHEMBL3526726 | |
| 0.01 | 0.173 | 0.034 | Nicotinic acid receptor 2 agonist | 0.034 0.027 CHEMBL4525793 0.034 0.027 CHEMBL4525794 | CHEMBL4525794 | |
| 0.014 | 0.182 | 0.052 | Prostaglandin antagonist | 0.052 0.038 CHEMBL4525793 | CHEMBL4525793 | |
| 0.032 | 0.202 | 0.144 | Potassium channel (Ca-activated) activator | 0.144 0.03 CHEMBL3526726 | CHEMBL3526726 | |
| 0.028 | 0.202 | 0.071 | Antiviral (Hepatitis D) | 0.071 0.013 CHEMBL3526727 0.069 0.014 CHEMBL3526583 | CHEMBL3526727 | |
| 0.013 | 0.192 | 0.075 | Prostaglandin E2 antagonist | 0.075 0.021 CHEMBL4525793 | CHEMBL4525793 | |
| 0.061 | 0.284 | 0.121 | Farnesoid X receptor antagonist | 0.121 0.101 CHEMBL3526726 | CHEMBL3526726 | |
| 0.02 | 0.245 | 0.145 | Porphobilinogen synthase inhibitor | 0.145 0.022 CHEMBL3526726 | CHEMBL3526726 | |
| 0.06 | 0.293 | 0.28 | Amyloid beta precursor protein antagonist | 0.28 0.023 CHEMBL4525794 | CHEMBL4525794 | |
| 0.157 | 0.402 | 0.548 | Antiinflammatory | 0.292 0.223 CHEMBL3526549 0.548 0.069 CHEMBL3526443 | CHEMBL3526443 | |
| 0.006 | 0.251 | 0.026 | AMPA 3 receptor antagonist | 0.026 0.024 CHEMBL3526726 | CHEMBL3526726 | |
| 0.06 | 0.347 | 0.141 | GABA C receptor rho-2 antagonist | 0.141 0.087 CHEMBL3526726 | CHEMBL3526726 | |
| 0.07 | 0.367 | 0.206 | Thyroid hormone beta antagonist | 0.206 0.149 CHEMBL3526726 | CHEMBL3526726 | |
| 0.067 | 0.381 | 0.216 | Thyroid hormone antagonist | 0.216 0.148 CHEMBL3526726 | CHEMBL3526726 | |
| 0.055 | 0.379 | 0.172 | Streptokinase A inhibitor | 0.172 0.153 CHEMBL3526726 | CHEMBL3526726 | |
| 0.076 | 0.405 | 0.147 | Death-associated protein kinase 2 inhibitor | 0.147 0.114 CHEMBL3526726 | CHEMBL3526726 | |
| 0.013 | 0.366 | 0.062 | Phenylalanine 4-hydroxylase inhibitor | 0.062 0.055 CHEMBL3526726 | CHEMBL3526726 | |
| 0.045 | 0.401 | 0.192 | Prostaglandin dehydrogenase inhibitor | 0.192 0.162 CHEMBL3526726 | CHEMBL3526726 | |
| 0.118 | 0.482 | 0.253 | 5 Hydroxytryptamine release inhibitor | 0.253 0.224 CHEMBL3526726 | CHEMBL3526726 | |
| 0.025 | 0.398 | 0.086 | Uric acid excretion stimulant | 0.086 0.072 CHEMBL4525793 | CHEMBL4525793 | |
| 0.022 | 0.405 | 0.106 | Creatine kinase inhibitor | 0.106 0.053 CHEMBL3526726 | CHEMBL3526726 | |
| 0.089 | 0.506 | 0.229 | Tyrosine 3 hydroxylase inhibitor | 0.229 0.091 CHEMBL3526726 | CHEMBL3526726 | |
| 0.045 | 0.464 | 0.262 | DNA polymerase beta inhibitor | 0.262 0.186 CHEMBL3526726 | CHEMBL3526726 | |
| 0.06 | 0.486 | 0.234 | Transcription factor inhibitor | 0.234 0.199 CHEMBL3526726 | CHEMBL3526726 | |
| 0.049 | 0.481 | 0.136 | CF transmembrane conductance regulator agonist | 0.136 0.104 CHEMBL3526726 | CHEMBL3526726 | |
| 0.037 | 0.485 | 0.292 | Alpha-glucosidase inhibitor | 0.292 0.164 CHEMBL3526726 | CHEMBL3526726 | |
| 0.056 | 0.516 | 0.152 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.152 0.144 CHEMBL3526726 | CHEMBL3526726 | |
| 0.041 | 0.541 | 0.35 | 15-Lipoxygenase inhibitor | 0.35 0.099 CHEMBL3526726 | CHEMBL3526726 | |
| 0.051 | 0.591 | 0.142 | Neurotensin receptor agonist | 0.142 0.123 CHEMBL3526726 | CHEMBL3526726 | |
| 0.011 | 0.672 | 0.103 | Chelator | 0.103 0.073 CHEMBL3526443 | CHEMBL3526443 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |