| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.819 | 0.005 | 0.831 | Antiobesity | 0.758 0.007 CHEMBL3526894 0.505 0.036 CHEMBL3526895 0.412 0.061 CHEMBL724 0.765 0.007 CHEMBL3526729 0.79 0.005 CHEMBL3527573 0.451 0.049 CHEMBL3526569 0.806 0.005 CHEMBL3526733 0.529 0.032 CHEMBL3527515 0.377 0.075 CHEMBL3527516 0.528 0.032 CHEMBL3527229 0.338 0.093 CHEMBL3527230 0.472 0.044 CHEMBL3526734 0.724 0.009 CHEMBL3526644 0.831 0.005 CHEMBL3527572 | CHEMBL3527572 | |
| 0.727 | 0.012 | 0.867 | Cyclophilin D inhibitor | 0.736 0.011 CHEMBL3526894 0.382 0.101 CHEMBL3526895 0.707 0.013 CHEMBL3526729 0.769 0.009 CHEMBL3527573 0.538 0.04 CHEMBL3526569 0.777 0.008 CHEMBL3526733 0.56 0.035 CHEMBL3527515 0.673 0.017 CHEMBL3527516 0.555 0.036 CHEMBL3527229 0.659 0.019 CHEMBL3527230 0.575 0.032 CHEMBL3526734 0.867 0.005 CHEMBL3526644 0.736 0.011 CHEMBL3527572 | CHEMBL3526644 | |
| 0.691 | 0.001 | 0.691 | Dipeptidyl peptidase IV inhibitor | 0.493 0.002 CHEMBL3526894 0.124 0.004 CHEMBL3526895 0.073 0.009 CHEMBL724 0.404 0.002 CHEMBL3526729 0.205 0.003 CHEMBL3526569 0.231 0.003 CHEMBL3527515 0.401 0.002 CHEMBL3527229 0.299 0.002 CHEMBL3526734 0.072 0.009 CHEMBL3526644 0.205 0.003 CHEMBL3527572 | ||
| 0.68 | 0.001 | 0.68 | Dipeptidyl peptidase inhibitor | 0.509 0.002 CHEMBL3526894 0.126 0.005 CHEMBL3526895 0.081 0.013 CHEMBL724 0.387 0.002 CHEMBL3526729 0.196 0.004 CHEMBL3526569 0.212 0.003 CHEMBL3527515 0.365 0.002 CHEMBL3527229 0.291 0.003 CHEMBL3526734 0.078 0.014 CHEMBL3526644 0.222 0.003 CHEMBL3527572 | ||
| 0.602 | 0.01 | 0.602 | Nootropic | 0.299 0.075 CHEMBL3526894 0.368 0.048 CHEMBL3526895 0.36 0.051 CHEMBL724 0.507 0.019 CHEMBL3526729 0.232 0.124 CHEMBL3527573 0.322 0.064 CHEMBL3526569 0.283 0.083 CHEMBL3526733 0.411 0.036 CHEMBL3527515 0.442 0.029 CHEMBL3527229 0.191 0.171 CHEMBL3526734 0.338 0.058 CHEMBL3526644 0.49 0.021 CHEMBL3527572 | ||
| 0.582 | 0.03 | 0.707 | Analgesic | 0.573 0.032 CHEMBL3526894 0.5 0.049 CHEMBL3526895 0.491 0.052 CHEMBL3526729 0.362 0.102 CHEMBL3527573 0.639 0.02 CHEMBL3526569 0.408 0.081 CHEMBL3526733 0.481 0.055 CHEMBL3527515 0.227 0.206 CHEMBL3527516 0.707 0.013 CHEMBL3527229 0.549 0.037 CHEMBL3526734 0.327 0.122 CHEMBL3526644 0.375 0.096 CHEMBL3527572 | CHEMBL3527229 | |
| 0.556 | 0.004 | 0.556 | Histamine antagonist | 0.456 0.005 CHEMBL3526894 0.16 0.027 CHEMBL724 0.231 0.015 CHEMBL3526729 0.183 0.022 CHEMBL3526569 0.239 0.014 CHEMBL3527515 0.477 0.005 CHEMBL3527229 0.458 0.005 CHEMBL3526734 0.075 0.069 CHEMBL3527572 | ||
| 0.55 | 0.004 | 0.55 | Antihistaminic | 0.447 0.005 CHEMBL3526894 0.08 0.077 CHEMBL3526895 0.166 0.028 CHEMBL724 0.238 0.015 CHEMBL3526729 0.19 0.022 CHEMBL3526569 0.244 0.015 CHEMBL3527515 0.471 0.005 CHEMBL3527229 0.446 0.005 CHEMBL3526734 0.088 0.066 CHEMBL3527572 | ||
| 0.44 | 0.004 | 0.44 | Histamine H3 receptor antagonist | 0.306 0.004 CHEMBL3526894 0.056 0.023 CHEMBL724 0.143 0.008 CHEMBL3526729 0.101 0.012 CHEMBL3526569 0.041 0.034 CHEMBL3527515 0.339 0.004 CHEMBL3527229 0.094 0.013 CHEMBL3526734 | ||
| 0.435 | 0.022 | 0.435 | HERG channel blocker | 0.174 0.107 CHEMBL3526894 0.312 0.046 CHEMBL724 0.279 0.055 CHEMBL3526729 0.272 0.058 CHEMBL3526569 0.204 0.088 CHEMBL3527515 0.414 0.025 CHEMBL3527229 | ||
| 0.411 | 0.055 | 0.489 | Toll-Like receptor 7 agonist | 0.339 0.088 CHEMBL3526894 0.477 0.037 CHEMBL3526729 0.3 0.11 CHEMBL3527573 0.489 0.034 CHEMBL3526569 0.243 0.154 CHEMBL3526733 0.393 0.063 CHEMBL3527515 0.23 0.167 CHEMBL3527516 0.431 0.049 CHEMBL3527229 0.29 0.117 CHEMBL3527230 0.235 0.161 CHEMBL3526734 0.386 0.066 CHEMBL3526644 | CHEMBL3526569 | |
| 0.41 | 0.056 | 0.485 | Toll-Like receptor agonist | 0.336 0.089 CHEMBL3526894 0.473 0.037 CHEMBL3526729 0.312 0.103 CHEMBL3527573 0.485 0.035 CHEMBL3526569 0.254 0.144 CHEMBL3526733 0.385 0.067 CHEMBL3527515 0.239 0.158 CHEMBL3527516 0.428 0.05 CHEMBL3527229 0.3 0.111 CHEMBL3527230 0.228 0.17 CHEMBL3526734 0.399 0.061 CHEMBL3526644 | CHEMBL3526569 | |
| 0.443 | 0.114 | 0.731 | Antiinflammatory | 0.288 0.226 CHEMBL3526894 0.409 0.134 CHEMBL3526729 0.648 0.041 CHEMBL3527573 0.548 0.069 CHEMBL3526569 0.674 0.036 CHEMBL3526733 0.321 0.196 CHEMBL3527515 0.397 0.141 CHEMBL3527516 0.583 0.058 CHEMBL3527229 0.348 0.174 CHEMBL3527230 0.731 0.025 CHEMBL3526644 0.537 0.073 CHEMBL3527572 | CHEMBL3526644 | |
| 0.36 | 0.034 | 0.36 | Potassium channel (Voltage-sensitive) blocker | 0.256 0.064 CHEMBL724 0.215 0.086 CHEMBL3526729 0.196 0.098 CHEMBL3526569 0.321 0.043 CHEMBL3527229 | ||
| 0.315 | 0.008 | 0.59 | 5 Hydroxytryptamine agonist | 0.19 0.015 CHEMBL3526894 0.265 0.01 CHEMBL3526895 0.59 0.004 CHEMBL724 0.163 0.019 CHEMBL3526729 0.074 0.045 CHEMBL3527229 0.062 0.054 CHEMBL3527572 | CHEMBL724 | |
| 0.341 | 0.035 | 0.408 | Potassium channel blocker | 0.408 0.021 CHEMBL724 0.178 0.108 CHEMBL3526729 0.156 0.129 CHEMBL3526569 0.298 0.047 CHEMBL3527229 | CHEMBL724 | |
| 0.336 | 0.052 | 0.441 | Interleukin 2 agonist | 0.41 0.025 CHEMBL3526894 0.282 0.087 CHEMBL3526895 0.353 0.044 CHEMBL3526729 0.396 0.029 CHEMBL3527573 0.395 0.029 CHEMBL3526733 0.338 0.051 CHEMBL3527516 0.339 0.05 CHEMBL3527230 0.229 0.144 CHEMBL3526734 0.441 0.017 CHEMBL3526644 0.274 0.094 CHEMBL3527572 | CHEMBL3526644 | |
| 0.284 | 0.004 | 0.474 | Neurokinin antagonist | 0.293 0.004 CHEMBL3526894 0.211 0.004 CHEMBL3526895 0.206 0.005 CHEMBL3526729 0.1 0.011 CHEMBL3527573 0.262 0.004 CHEMBL3526569 0.112 0.009 CHEMBL3526733 0.394 0.004 CHEMBL3527515 0.067 0.021 CHEMBL3527516 0.335 0.004 CHEMBL3527229 0.056 0.028 CHEMBL3527230 0.474 0.003 CHEMBL3526734 0.071 0.019 CHEMBL3526644 0.113 0.009 CHEMBL3527572 | CHEMBL3526734 | |
| 0.269 | 0.003 | 0.316 | Neurokinin 3 antagonist | 0.26 0.003 CHEMBL3526894 0.191 0.004 CHEMBL3526895 0.208 0.003 CHEMBL3526729 0.11 0.005 CHEMBL3527573 0.204 0.003 CHEMBL3526569 0.116 0.005 CHEMBL3526733 0.282 0.003 CHEMBL3527515 0.094 0.006 CHEMBL3527516 0.257 0.003 CHEMBL3527229 0.085 0.008 CHEMBL3527230 0.316 0.003 CHEMBL3526734 0.084 0.008 CHEMBL3526644 0.148 0.004 CHEMBL3527572 | CHEMBL3526734 | |
| 0.258 | 0.002 | 0.258 | Dipeptidyl peptidase VIII inhibitor | 0.244 0.002 CHEMBL3526894 0.021 0.007 CHEMBL3526895 0.149 0.002 CHEMBL3526729 0.016 0.009 CHEMBL3527573 0.055 0.004 CHEMBL3526569 0.018 0.008 CHEMBL3526733 0.052 0.004 CHEMBL3527515 0.02 0.007 CHEMBL3527516 0.081 0.003 CHEMBL3527229 0.017 0.009 CHEMBL3527230 0.068 0.004 CHEMBL3526734 0.045 0.004 CHEMBL3526644 0.098 0.003 CHEMBL3527572 | ||
| 0.258 | 0.004 | 0.407 | Neurokinin 2 antagonist | 0.267 0.003 CHEMBL3526894 0.219 0.004 CHEMBL3526895 0.218 0.004 CHEMBL3526729 0.141 0.006 CHEMBL3527573 0.229 0.004 CHEMBL3526569 0.15 0.005 CHEMBL3526733 0.36 0.003 CHEMBL3527515 0.109 0.009 CHEMBL3527516 0.265 0.003 CHEMBL3527229 0.092 0.011 CHEMBL3527230 0.407 0.002 CHEMBL3526734 0.096 0.011 CHEMBL3526644 0.161 0.005 CHEMBL3527572 | CHEMBL3526734 | |
| 0.256 | 0.004 | 0.425 | Neurokinin 1 antagonist | 0.252 0.004 CHEMBL3526894 0.2 0.004 CHEMBL3526895 0.187 0.004 CHEMBL3526729 0.094 0.007 CHEMBL3527573 0.245 0.004 CHEMBL3526569 0.104 0.006 CHEMBL3526733 0.366 0.003 CHEMBL3527515 0.066 0.013 CHEMBL3527516 0.312 0.004 CHEMBL3527229 0.054 0.017 CHEMBL3527230 0.425 0.003 CHEMBL3526734 0.066 0.013 CHEMBL3526644 0.098 0.006 CHEMBL3527572 | CHEMBL3526734 | |
| 0.244 | 0.002 | 0.244 | Dipeptidyl peptidase II inhibitor | 0.197 0.002 CHEMBL3526894 0.039 0.015 CHEMBL3526895 0.113 0.003 CHEMBL3526729 0.042 0.013 CHEMBL3526569 0.034 0.02 CHEMBL3527515 0.09 0.004 CHEMBL3527229 0.057 0.007 CHEMBL3526734 0.085 0.004 CHEMBL3527572 | ||
| 0.197 | 0.004 | 0.25 | 5 Hydroxytryptamine 2C agonist | 0.165 0.005 CHEMBL3526894 0.154 0.005 CHEMBL3526895 0.25 0.004 CHEMBL724 0.151 0.005 CHEMBL3526729 0.05 0.028 CHEMBL3526644 0.094 0.008 CHEMBL3527572 | CHEMBL724 | |
| 0.258 | 0.073 | 0.446 | Interleukin agonist | 0.17 0.149 CHEMBL3526894 0.379 0.022 CHEMBL3526895 0.431 0.015 CHEMBL724 0.189 0.131 CHEMBL3526729 0.178 0.141 CHEMBL3527573 0.263 0.07 CHEMBL3526733 0.446 0.013 CHEMBL3527516 0.352 0.029 CHEMBL3527230 0.324 0.037 CHEMBL3526644 | CHEMBL3527516 | |
| 0.188 | 0.004 | 0.188 | Orexin receptor antagonist | 0.11 0.009 CHEMBL724 0.098 0.013 CHEMBL3526729 0.089 0.019 CHEMBL3526569 0.12 0.007 CHEMBL3527515 0.171 0.004 CHEMBL3527229 | ||
| 0.168 | 0.004 | 0.168 | Toll-Like receptor 8 antagonist | 0.066 0.026 CHEMBL3526894 0.07 0.023 CHEMBL3526895 0.111 0.006 CHEMBL724 0.126 0.005 CHEMBL3526729 0.055 0.035 CHEMBL3527229 | ||
| 0.166 | 0.004 | 0.166 | Orexin receptor 1 antagonist | 0.114 0.007 CHEMBL724 0.096 0.016 CHEMBL3526729 0.072 0.049 CHEMBL3526569 0.094 0.017 CHEMBL3527515 0.116 0.007 CHEMBL3527229 | ||
| 0.186 | 0.036 | 0.195 | Toll-Like receptor antagonist | 0.195 0.032 CHEMBL724 0.154 0.053 CHEMBL3526729 | CHEMBL724 | |
| 0.16 | 0.028 | 0.16 | Chemokine receptor antagonist | 0.15 0.032 CHEMBL3526894 0.105 0.059 CHEMBL3526729 0.1 0.063 CHEMBL3526569 0.15 0.032 CHEMBL3527229 0.093 0.07 CHEMBL3526734 | ||
| 0.134 | 0.005 | 0.134 | Glutamate (mGluR group I) agonist | 0.062 0.021 CHEMBL3526895 0.096 0.009 CHEMBL724 0.064 0.019 CHEMBL3526729 0.077 0.013 CHEMBL3527229 0.097 0.009 CHEMBL3527572 | ||
| 0.137 | 0.012 | 0.186 | Janus tyrosine kinase 1 inhibitor | 0.186 0.005 CHEMBL724 0.053 0.044 CHEMBL3526729 0.09 0.025 CHEMBL3526569 0.061 0.038 CHEMBL3527515 0.164 0.008 CHEMBL3527229 | CHEMBL724 | |
| 0.131 | 0.009 | 0.162 | Toll-Like receptor 7 antagonist | 0.06 0.055 CHEMBL3526894 0.098 0.022 CHEMBL3526895 0.162 0.005 CHEMBL724 0.096 0.024 CHEMBL3526729 0.059 0.056 CHEMBL3527229 | CHEMBL724 | |
| 0.116 | 0.004 | 0.116 | Orexin receptor 2 antagonist | 0.068 0.008 CHEMBL724 0.041 0.02 CHEMBL3526729 0.033 0.028 CHEMBL3526569 0.067 0.008 CHEMBL3527515 0.102 0.005 CHEMBL3527229 | ||
| 0.116 | 0.005 | 0.116 | Glutamate (mGluR5) agonist | 0.047 0.03 CHEMBL3526895 0.094 0.008 CHEMBL724 0.055 0.021 CHEMBL3526729 0.073 0.013 CHEMBL3527229 0.092 0.008 CHEMBL3527572 | ||
| 0.112 | 0.002 | 0.112 | Dipeptidyl peptidase IX inhibitor | 0.107 0.003 CHEMBL3526894 0.019 0.009 CHEMBL3526895 0.087 0.003 CHEMBL3526729 0.039 0.004 CHEMBL3526569 0.015 0.012 CHEMBL3526733 0.035 0.005 CHEMBL3527515 0.017 0.01 CHEMBL3527516 0.048 0.004 CHEMBL3527229 0.015 0.012 CHEMBL3527230 0.04 0.004 CHEMBL3526734 0.036 0.005 CHEMBL3526644 0.06 0.003 CHEMBL3527572 | ||
| 0.157 | 0.05 | 0.193 | Sodium channel (voltage-gated) blocker | 0.135 0.067 CHEMBL3526894 0.193 0.032 CHEMBL724 0.141 0.062 CHEMBL3527229 | CHEMBL724 | |
| 0.133 | 0.032 | 0.133 | Acetylcholine agonist | 0.101 0.046 CHEMBL3526895 0.121 0.036 CHEMBL724 0.08 0.066 CHEMBL3526729 | ||
| 0.173 | 0.071 | 0.173 | Antipruritic | 0.147 0.098 CHEMBL724 0.132 0.119 CHEMBL3526729 0.132 0.12 CHEMBL3526569 0.172 0.072 CHEMBL3527229 | ||
| 0.156 | 0.054 | 0.191 | Sodium channel blocker | 0.131 0.073 CHEMBL3526894 0.191 0.036 CHEMBL724 0.185 0.038 CHEMBL3527229 | CHEMBL724 | |
| 0.12 | 0.026 | 0.151 | Acetylcholine nicotinic agonist | 0.11 0.031 CHEMBL3526895 0.151 0.017 CHEMBL724 0.089 0.047 CHEMBL3526729 | CHEMBL724 | |
| 0.112 | 0.023 | 0.263 | Tyk2 inhibitor | 0.263 0.005 CHEMBL724 0.084 0.035 CHEMBL3526569 0.062 0.047 CHEMBL3527515 0.145 0.014 CHEMBL3527229 | CHEMBL724 | |
| 0.095 | 0.01 | 0.149 | Histamine agonist | 0.08 0.014 CHEMBL3526894 0.149 0.005 CHEMBL724 0.065 0.023 CHEMBL3527229 | CHEMBL724 | |
| 0.113 | 0.028 | 0.113 | CC chemokine receptor antagonist | 0.091 0.042 CHEMBL3526894 0.079 0.053 CHEMBL3526729 0.081 0.051 CHEMBL3526569 0.112 0.029 CHEMBL3527229 | ||
| 0.092 | 0.008 | 0.092 | Prolyl endopeptidase inhibitor | 0.068 0.017 CHEMBL3526894 0.069 0.016 CHEMBL3526729 0.068 0.017 CHEMBL3527573 0.068 0.017 CHEMBL3526569 0.081 0.01 CHEMBL3526733 0.053 0.032 CHEMBL3527515 0.09 0.008 CHEMBL3527229 0.05 0.036 CHEMBL3526734 | ||
| 0.092 | 0.01 | 0.092 | Purinergic P2X antagonist | 0.059 0.024 CHEMBL724 0.063 0.022 CHEMBL3526729 0.053 0.029 CHEMBL3527229 0.043 0.041 CHEMBL3527572 | ||
| 0.115 | 0.034 | 0.115 | Histamine H1 receptor antagonist | 0.078 0.059 CHEMBL3526895 0.115 0.034 CHEMBL724 0.075 0.063 CHEMBL3527515 0.077 0.061 CHEMBL3526734 | ||
| 0.086 | 0.015 | 0.086 | Antidiuretic hormone antagonist | 0.044 0.025 CHEMBL3526894 0.047 0.024 CHEMBL3526729 0.036 0.03 CHEMBL3526569 0.062 0.019 CHEMBL3527229 | ||
| 0.127 | 0.055 | 0.127 | Calcium channel N-type blocker | 0.125 0.057 CHEMBL724 | ||
| 0.104 | 0.034 | 0.3 | Janus tyrosine kinase 2 inhibitor | 0.3 0.005 CHEMBL724 0.104 0.034 CHEMBL3527229 | CHEMBL724 | |
| 0.074 | 0.005 | 0.074 | Glucose-dependent insulinotropic receptor agonist | 0.047 0.013 CHEMBL724 0.063 0.007 CHEMBL3526729 0.036 0.022 CHEMBL3527515 0.034 0.025 CHEMBL3527229 | ||
| 0.071 | 0.005 | 0.072 | ADAM10 endopeptidase inhibitor | 0.072 0.005 CHEMBL3526894 0.057 0.008 CHEMBL3526729 0.053 0.009 CHEMBL3527573 0.042 0.014 CHEMBL3526569 0.057 0.008 CHEMBL3526733 0.045 0.012 CHEMBL3527515 0.036 0.019 CHEMBL3527516 0.048 0.011 CHEMBL3527229 0.033 0.024 CHEMBL3527230 0.052 0.009 CHEMBL3526734 0.037 0.018 CHEMBL3526644 0.048 0.011 CHEMBL3527572 | CHEMBL3526894 | |
| 0.084 | 0.019 | 0.093 | Nicotinic neuronal receptor agonist | 0.093 0.015 CHEMBL724 0.05 0.045 CHEMBL3526729 | CHEMBL724 | |
| 0.08 | 0.015 | 0.08 | Ca(v)3.2 blocker | 0.071 0.022 CHEMBL724 0.07 0.023 CHEMBL3526729 0.061 0.036 CHEMBL3526569 0.058 0.043 CHEMBL3527515 0.068 0.024 CHEMBL3527229 | ||
| 0.094 | 0.031 | 0.15 | Polo-like kinase-2 inhibitor | 0.095 0.031 CHEMBL3526895 0.15 0.004 CHEMBL724 0.083 0.041 CHEMBL3526729 | CHEMBL724 | |
| 0.09 | 0.027 | 0.265 | CXC chemokine 4 receptor antagonist | 0.165 0.014 CHEMBL3526894 0.147 0.016 CHEMBL3526895 0.265 0.006 CHEMBL724 | CHEMBL724 | |
| 0.121 | 0.059 | 0.207 | 5 Hydroxytryptamine 2B antagonist | 0.207 0.025 CHEMBL724 | CHEMBL724 | |
| 0.102 | 0.044 | 0.146 | Interleukin-1 receptor-associated protein kinase 4 inhibitor | 0.146 0.024 CHEMBL724 0.093 0.053 CHEMBL3526729 | CHEMBL724 | |
| 0.086 | 0.029 | 0.086 | Purinergic P2 antagonist | 0.056 0.052 CHEMBL724 0.057 0.051 CHEMBL3526729 0.057 0.051 CHEMBL3527572 | ||
| 0.067 | 0.011 | 0.074 | CC chemokine 4 receptor antagonist | 0.061 0.015 CHEMBL3526895 0.074 0.009 CHEMBL724 0.046 0.035 CHEMBL3526729 | CHEMBL724 | |
| 0.064 | 0.009 | 0.064 | Purinergic P2X7 antagonist | 0.045 0.017 CHEMBL3526894 0.037 0.023 CHEMBL3526729 0.042 0.019 CHEMBL3527229 | ||
| 0.132 | 0.079 | 0.183 | Aurora-C kinase inhibitor | 0.183 0.025 CHEMBL724 | CHEMBL724 | |
| 0.066 | 0.013 | 0.066 | Acetyl-CoA carboxylase inhibitor | 0.039 0.032 CHEMBL3526894 0.056 0.017 CHEMBL3526729 0.046 0.024 CHEMBL3526569 0.038 0.034 CHEMBL3527515 0.052 0.019 CHEMBL3527229 | ||
| 0.096 | 0.045 | 0.104 | Leucine-rich repeat kinase 2 inhibitor | 0.104 0.04 CHEMBL724 | CHEMBL724 | |
| 0.058 | 0.01 | 0.188 | Vascular adhesion protein 1 inhibitor | 0.049 0.016 CHEMBL3526895 0.188 0.003 CHEMBL724 0.036 0.031 CHEMBL3526569 0.064 0.008 CHEMBL3527229 | CHEMBL724 | |
| 0.093 | 0.045 | 0.095 | Hematopoietic | 0.095 0.042 CHEMBL3526894 0.093 0.045 CHEMBL3526729 | CHEMBL3526894 | |
| 0.06 | 0.013 | 0.062 | G protein-coupled receptor agonist | 0.046 0.02 CHEMBL724 0.062 0.012 CHEMBL3526729 | CHEMBL3526729 | |
| 0.068 | 0.026 | 0.118 | CC chemokine 2 receptor antagonist | 0.049 0.048 CHEMBL3526729 0.08 0.019 CHEMBL3526569 0.118 0.01 CHEMBL3527229 | CHEMBL3527229 | |
| 0.076 | 0.037 | 0.116 | Nav1.7 sodium channel blocker | 0.116 0.018 CHEMBL724 | CHEMBL724 | |
| 0.057 | 0.021 | 0.066 | CC chemokine receptor 2B antagonist | 0.057 0.021 CHEMBL3526894 0.051 0.03 CHEMBL3526729 0.059 0.02 CHEMBL3526569 0.066 0.014 CHEMBL3527229 | CHEMBL3527229 | |
| 0.124 | 0.089 | 0.156 | Neurotrophic factor | 0.156 0.054 CHEMBL3526895 0.115 0.104 CHEMBL3526729 0.117 0.1 CHEMBL3526644 | CHEMBL3526895 | |
| 0.059 | 0.025 | 0.604 | 5 Hydroxytryptamine 1A agonist | 0.05 0.029 CHEMBL3526895 0.604 0.004 CHEMBL724 | CHEMBL724 | |
| 0.058 | 0.024 | 0.087 | Nicotinic receptor alpha4 subunit antagonist | 0.046 0.042 CHEMBL3526894 0.057 0.024 CHEMBL3526895 0.087 0.011 CHEMBL724 0.069 0.017 CHEMBL3526729 0.049 0.035 CHEMBL3527572 | CHEMBL724 | |
| 0.041 | 0.007 | 0.05 | Antidiuretic hormone agonist | 0.044 0.006 CHEMBL3526894 0.035 0.01 CHEMBL3526729 0.04 0.007 CHEMBL3526569 0.027 0.018 CHEMBL3527515 0.05 0.005 CHEMBL3527229 0.032 0.012 CHEMBL3526734 0.028 0.017 CHEMBL3527572 | CHEMBL3527229 | |
| 0.041 | 0.009 | 0.041 | Acetyl-CoA carboxylase 2 inhibitor | 0.029 0.012 CHEMBL3526729 0.019 0.018 CHEMBL3526569 0.026 0.014 CHEMBL3527229 | ||
| 0.044 | 0.013 | 0.044 | Histamine H3 receptor agonist | 0.041 0.013 CHEMBL3526894 0.024 0.022 CHEMBL3526729 0.025 0.021 CHEMBL3527229 | ||
| 0.081 | 0.052 | 0.129 | Glutamate receptor agonist | 0.129 0.023 CHEMBL3526895 0.087 0.047 CHEMBL724 | CHEMBL3526895 | |
| 0.057 | 0.03 | 0.116 | 5 Hydroxytryptamine 2 agonist | 0.116 0.007 CHEMBL724 | CHEMBL724 | |
| 0.037 | 0.01 | 0.05 | Nicotinic alpha4beta2 receptor agonist | 0.034 0.013 CHEMBL3526895 0.05 0.004 CHEMBL724 0.029 0.019 CHEMBL3526729 | CHEMBL724 | |
| 0.06 | 0.036 | 0.107 | 5 Hydroxytryptamine 6 antagonist | 0.107 0.013 CHEMBL724 | CHEMBL724 | |
| 0.048 | 0.026 | 0.061 | Poly(ADP-ribose) polymerase inhibitor | 0.061 0.016 CHEMBL724 | CHEMBL724 | |
| 0.027 | 0.005 | 0.055 | Nicotinic alpha4 receptor agonist | 0.017 0.011 CHEMBL3526895 0.055 0.004 CHEMBL724 0.019 0.008 CHEMBL3526729 | CHEMBL724 | |
| 0.043 | 0.021 | 0.046 | Poly(ADP-ribose) polymerase 1 inhibitor | 0.046 0.019 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.018 | 0.038 | Vasopressin 1 antagonist | 0.037 0.019 CHEMBL3527229 | ||
| 0.029 | 0.01 | 0.029 | Phosphodiesterase 9A inhibitor | 0.023 0.02 CHEMBL3526729 0.023 0.019 CHEMBL3527229 | ||
| 0.033 | 0.013 | 0.033 | Potassium channel (Inward rectifier) 1 blocker | 0.031 0.019 CHEMBL3526895 0.032 0.016 CHEMBL724 0.03 0.02 CHEMBL3526729 0.029 0.025 CHEMBL3526569 0.03 0.022 CHEMBL3527515 0.031 0.017 CHEMBL3527229 | ||
| 0.05 | 0.034 | 0.09 | Potassium channel (Inward rectifier) blocker | 0.049 0.035 CHEMBL3526895 0.09 0.009 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.018 | 0.052 | Nicotinic alpha3beta4 receptor agonist | 0.03 0.021 CHEMBL3526895 0.052 0.005 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.012 | 0.026 | Phosphodiesterase IX inhibitor | |||
| 0.048 | 0.034 | 0.118 | Histamine H4 receptor antagonist | 0.091 0.006 CHEMBL3526894 0.118 0.004 CHEMBL724 0.044 0.042 CHEMBL3527229 0.05 0.031 CHEMBL3526734 | CHEMBL724 | |
| 0.02 | 0.009 | 0.022 | Vasopressin 2 agonist | 0.022 0.007 CHEMBL3526894 0.016 0.012 CHEMBL3526729 0.018 0.01 CHEMBL3526569 0.021 0.008 CHEMBL3527229 | CHEMBL3526894 | |
| 0.02 | 0.009 | 0.052 | Complement factor D inhibitor | 0.025 0.005 CHEMBL724 0.032 0.004 CHEMBL3526569 0.052 0.003 CHEMBL3527229 | CHEMBL3527229 | |
| 0.028 | 0.02 | 0.028 | Vasopressin 1A antagonist | 0.028 0.021 CHEMBL3527229 | ||
| 0.088 | 0.082 | 0.236 | 5 Hydroxytryptamine 2 antagonist | 0.236 0.023 CHEMBL724 | CHEMBL724 | |
| 0.075 | 0.072 | 0.098 | Phosphodiesterase 11A inhibitor | 0.082 0.056 CHEMBL3526569 0.08 0.06 CHEMBL3527515 0.098 0.034 CHEMBL3527229 | CHEMBL3527229 | |
| 0.075 | 0.072 | 0.098 | Phosphodiesterase XI inhibitor | 0.082 0.056 CHEMBL3526569 0.08 0.06 CHEMBL3527515 0.098 0.034 CHEMBL3527229 | CHEMBL3527229 | |
| 0.026 | 0.024 | 0.026 | HCV NS5A inhibitor | |||
| 0.184 | 0.183 | 0.414 | Immunomodulator | 0.284 0.091 CHEMBL3526895 0.374 0.052 CHEMBL3527573 0.412 0.041 CHEMBL3526733 0.336 0.065 CHEMBL3527516 0.296 0.084 CHEMBL3527230 0.414 0.04 CHEMBL3526644 | CHEMBL3526644 | |
| 0.045 | 0.044 | 0.054 | CC chemokine 5 receptor antagonist | 0.046 0.042 CHEMBL3527515 0.054 0.031 CHEMBL3526734 | CHEMBL3526734 | |
| 0.119 | 0.119 | 0.165 | Cyclin-dependent kinase 8 inhibitor | 0.165 0.065 CHEMBL724 0.143 0.087 CHEMBL3526569 0.16 0.07 CHEMBL3527229 | CHEMBL724 | |
| 0.036 | 0.036 | 0.135 | Protein kinase (CK1) epsilon inhibitor | 0.135 0.004 CHEMBL724 | CHEMBL724 | |
| 0.051 | 0.053 | 0.139 | Cyclin-dependent kinase 6 inhibitor | 0.077 0.024 CHEMBL3526895 0.139 0.005 CHEMBL724 | CHEMBL724 | |
| 0.041 | 0.044 | 0.45 | 5 Hydroxytryptamine 1 agonist | 0.45 0.005 CHEMBL724 | CHEMBL724 | |
| 0.115 | 0.124 | 0.168 | Heat shock protein 90 antagonist | 0.168 0.057 CHEMBL3527515 | CHEMBL3527515 | |
| 0.093 | 0.102 | 0.501 | Acetylcholine antagonist | 0.268 0.017 CHEMBL3526894 0.097 0.096 CHEMBL3526729 0.203 0.03 CHEMBL3527515 0.501 0.005 CHEMBL3526734 | CHEMBL3526734 | |
| 0.057 | 0.066 | 0.222 | Janus tyrosine kinase 3 inhibitor | 0.222 0.009 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.027 | 0.022 | Baculoviral IAP repeat-containing protein 3 inhibitor | 0.022 0.01 CHEMBL3526895 | CHEMBL3526895 | |
| 0.041 | 0.052 | 0.046 | Baculoviral IAP repeat-containing protein inhibitor | 0.046 0.033 CHEMBL3526895 | CHEMBL3526895 | |
| 0.044 | 0.056 | 0.276 | NMDA 2B receptor antagonist | 0.05 0.043 CHEMBL3526729 0.276 0.004 CHEMBL3527572 | CHEMBL3527572 | |
| 0.093 | 0.105 | 0.489 | Cholinergic antagonist | 0.262 0.019 CHEMBL3526894 0.203 0.031 CHEMBL3527515 0.489 0.005 CHEMBL3526734 | CHEMBL3526734 | |
| 0.046 | 0.06 | 0.113 | Glucosylceramidase inhibitor | 0.055 0.037 CHEMBL3526895 0.113 0.006 CHEMBL724 0.102 0.008 CHEMBL3527516 0.074 0.019 CHEMBL3527230 | CHEMBL724 | |
| 0.042 | 0.058 | 0.061 | Nicotinic alpha7 receptor agonist | 0.061 0.031 CHEMBL724 | CHEMBL724 | |
| 0.051 | 0.069 | 0.127 | Neuronal nicotinic receptor antagonist | 0.127 0.016 CHEMBL3526895 0.103 0.023 CHEMBL724 | CHEMBL3526895 | |
| 0.06 | 0.078 | 0.138 | Nicotinic alpha4beta2 receptor antagonist | 0.114 0.021 CHEMBL3526895 0.138 0.01 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.038 | 0.043 | Poly(ADP-ribose) polymerase 2 inhibitor | 0.043 0.01 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.035 | 0.029 | Melanocortin 4 agonist | 0.029 0.016 CHEMBL3526894 | CHEMBL3526894 | |
| 0.078 | 0.102 | 0.263 | 5 Hydroxytryptamine antagonist | 0.263 0.023 CHEMBL724 | CHEMBL724 | |
| 0.062 | 0.087 | 0.081 | Potassium channel (Tandem pore domain) blocker | 0.081 0.032 CHEMBL724 | CHEMBL724 | |
| 0.146 | 0.171 | 0.236 | MAP kinase kinase 5 inhibitor | 0.167 0.094 CHEMBL3526895 0.236 0.01 CHEMBL724 | CHEMBL724 | |
| 0.057 | 0.083 | 0.161 | Protein kinase B beta inhibitor | 0.161 0.006 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.054 | 0.042 | Vanilloid 4 antagonist | 0.042 0.01 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.041 | 0.03 | Aminopeptidase P inhibitor | 0.026 0.013 CHEMBL3526569 0.024 0.015 CHEMBL3527515 0.028 0.012 CHEMBL3527229 0.03 0.01 CHEMBL3526734 | CHEMBL3526734 | |
| 0.01 | 0.041 | 0.026 | Melanocortin agonist | 0.026 0.018 CHEMBL3526894 | CHEMBL3526894 | |
| 0.004 | 0.039 | 0.013 | Melatonin 5 antagonist | 0.013 0.007 CHEMBL724 | CHEMBL724 | |
| 0.051 | 0.087 | 0.126 | Protein kinase C beta inhibitor | 0.081 0.028 CHEMBL3526894 0.111 0.009 CHEMBL3526895 0.126 0.006 CHEMBL724 | CHEMBL724 | |
| 0.04 | 0.077 | 0.072 | Nicotinic receptor alpha7 subunit antagonist | 0.072 0.02 CHEMBL3526895 0.071 0.021 CHEMBL724 | CHEMBL3526895 | |
| 0.029 | 0.068 | 0.038 | Phenylethanolamine N methyltransferase inhibitor | 0.038 0.034 CHEMBL3526895 | CHEMBL3526895 | |
| 0.061 | 0.104 | 0.082 | Viral attachment inhibitor | 0.078 0.054 CHEMBL724 0.082 0.046 CHEMBL3527515 | CHEMBL3527515 | |
| 0.025 | 0.068 | 0.122 | Factor XIa inhibitor | 0.122 0.004 CHEMBL3526894 0.092 0.006 CHEMBL3526734 0.044 0.025 CHEMBL3527572 | CHEMBL3526894 | |
| 0.028 | 0.073 | 0.1 | 5 Hydroxytryptamine 2B agonist | 0.1 0.004 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.07 | 0.547 | Cholecystokinin B agonist | 0.547 0.002 CHEMBL3527572 | CHEMBL3527572 | |
| 0.054 | 0.102 | 0.14 | Acetylcholine nicotinic antagonist | 0.14 0.023 CHEMBL3526895 0.107 0.035 CHEMBL724 | CHEMBL3526895 | |
| 0.067 | 0.116 | 0.128 | mTOR complex 2 inhibitor | 0.105 0.028 CHEMBL3526895 0.128 0.014 CHEMBL724 | CHEMBL724 | |
| 0.068 | 0.119 | 0.121 | Polo-like kinase-1 inhibitor | 0.121 0.029 CHEMBL724 0.088 0.066 CHEMBL3527515 | CHEMBL724 | |
| 0.023 | 0.076 | 0.046 | Substance P antagonist | 0.041 0.025 CHEMBL3527515 0.046 0.02 CHEMBL3526734 | CHEMBL3526734 | |
| 0.018 | 0.075 | 0.069 | Dopamine D5 antagonist | 0.069 0.015 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.084 | 0.047 | Melanocortin antagonist | 0.047 0.032 CHEMBL3526894 | CHEMBL3526894 | |
| 0.045 | 0.105 | 0.115 | CXC chemokine receptor antagonist | 0.115 0.019 CHEMBL724 | CHEMBL724 | |
| 0.036 | 0.096 | 0.1 | Acetylcholine M5 receptor antagonist | 0.1 0.017 CHEMBL3526894 0.08 0.024 CHEMBL3526734 | CHEMBL3526894 | |
| 0.039 | 0.101 | 0.061 | Fibroblast growth factor 2 antagonist | 0.061 0.05 CHEMBL724 | CHEMBL724 | |
| 0.064 | 0.129 | 0.077 | MAP kinase 7 inhibitor | 0.077 0.057 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.078 | 0.037 | Bradykinin B2 receptor agonist | 0.027 0.021 CHEMBL3526569 0.026 0.023 CHEMBL3527515 0.029 0.019 CHEMBL3527229 0.037 0.013 CHEMBL3526734 | CHEMBL3526734 | |
| 0.082 | 0.149 | 0.234 | Toll-Like receptor 9 antagonist | 0.234 0.024 CHEMBL724 | CHEMBL724 | |
| 0.049 | 0.119 | 0.209 | ALK inhibitor | 0.209 0.01 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.109 | 0.085 | Alpha 1L adrenoreceptor antagonist | 0.085 0.006 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.096 | 0.062 | Nerve growth factor antagonist | 0.056 0.013 CHEMBL3526895 0.062 0.008 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.09 | 0.036 | 5 Hydroxytryptamine 6 agonist | 0.036 0.01 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.097 | 0.095 | Phosphatidylinositol 3-kinase alpha inhibitor | 0.095 0.018 CHEMBL724 | CHEMBL724 | |
| 0.03 | 0.105 | 0.073 | Pim-2 kinase inhibitor | 0.073 0.023 CHEMBL724 | CHEMBL724 | |
| 0.042 | 0.118 | 0.126 | Protein kinase B alpha inhibitor | 0.126 0.016 CHEMBL724 | CHEMBL724 | |
| 0.078 | 0.157 | 0.333 | Tyrosine kinase inhibitor | 0.333 0.037 CHEMBL724 | CHEMBL724 | |
| 0.03 | 0.11 | 0.112 | 5 Hydroxytryptamine 2A agonist | 0.112 0.011 CHEMBL724 | CHEMBL724 | |
| 0.066 | 0.149 | 0.477 | Acetylcholine muscarinic antagonist | 0.216 0.021 CHEMBL3526894 0.154 0.042 CHEMBL3527515 0.477 0.004 CHEMBL3526734 | CHEMBL3526734 | |
| 0.023 | 0.106 | 0.106 | Dopamine D4 antagonist | 0.106 0.024 CHEMBL724 | CHEMBL724 | |
| 0.055 | 0.139 | 0.161 | Pim-3 kinase inhibitor | 0.161 0.015 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.122 | 0.262 | 5 Hydroxytryptamine 3 agonist | 0.079 0.028 CHEMBL3526894 0.072 0.033 CHEMBL3526895 0.262 0.003 CHEMBL724 | CHEMBL724 | |
| 0.039 | 0.126 | 0.084 | Fibroblast growth factor 3 antagonist | 0.084 0.045 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.115 | 0.097 | Potassium channel small-conductance Ca-activated blocker | 0.097 0.007 CHEMBL724 | CHEMBL724 | |
| 0.095 | 0.185 | 0.125 | Heat shock protein 90 alpha antagonist | 0.125 0.119 CHEMBL3527515 | CHEMBL3527515 | |
| 0.033 | 0.127 | 0.044 | Phosphodiesterase 6C inhibitor | 0.044 0.041 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.121 | 0.359 | Alpha 1 adrenoreceptor agonist | 0.359 0.004 CHEMBL724 | CHEMBL724 | |
| 0.033 | 0.128 | 0.439 | Alpha adrenoreceptor agonist | 0.439 0.004 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.117 | 0.058 | Protein kinase (CK2) beta inhibitor | 0.058 0.005 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.118 | 0.062 | Antibiotic Aminoglycoside-like | 0.057 0.01 CHEMBL3527573 0.056 0.01 CHEMBL3526733 0.05 0.013 CHEMBL3527516 0.051 0.013 CHEMBL3527230 0.062 0.008 CHEMBL3526644 | CHEMBL3526644 | |
| 0.067 | 0.164 | 0.096 | Calcium channel (voltage-sensitive) blocker | 0.096 0.091 CHEMBL3527229 | CHEMBL3527229 | |
| 0.007 | 0.104 | 0.06 | Arginase inhibitor | 0.06 0.01 CHEMBL3526895 0.037 0.024 CHEMBL3526644 | CHEMBL3526895 | |
| 0.01 | 0.11 | 0.034 | Glutaminyl-peptide cyclotransferase inhibitor | 0.034 0.005 CHEMBL724 | CHEMBL724 | |
| 0.042 | 0.143 | 0.279 | Alpha adrenoreceptor antagonist | 0.279 0.017 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.125 | 0.092 | mTOR inhibitor | 0.092 0.014 CHEMBL724 | CHEMBL724 | |
| 0.045 | 0.147 | 0.116 | Insulin like growth factor 1 antagonist | 0.116 0.031 CHEMBL724 | CHEMBL724 | |
| 0.029 | 0.132 | 0.097 | Phosphatidylinositol kinase inhibitor | 0.097 0.022 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.114 | 0.035 | Endothelial nitric-oxide synthase inhibitor | 0.035 0.017 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.112 | 0.016 | Kainate receptor 3 antagonist | 0.016 0.014 CHEMBL3526895 | CHEMBL3526895 | |
| 0.025 | 0.13 | 0.086 | Protein kinase C theta inhibitor | 0.086 0.012 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.126 | 0.051 | Acetylcholine muscarinic agonist | 0.051 0.042 CHEMBL724 | CHEMBL724 | |
| 0.054 | 0.16 | 0.113 | Aurora-B kinase inhibitor | 0.113 0.07 CHEMBL724 | CHEMBL724 | |
| 0.028 | 0.136 | 0.235 | Alpha 1 adrenoreceptor antagonist | 0.235 0.016 CHEMBL724 | CHEMBL724 | |
| 0.031 | 0.14 | 0.19 | 5 Hydroxytryptamine 2A antagonist | 0.19 0.021 CHEMBL724 | CHEMBL724 | |
| 0.041 | 0.152 | 0.256 | Alpha 2 adrenoreceptor antagonist | 0.081 0.065 CHEMBL3526895 0.256 0.011 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.129 | 0.053 | Membrane dipeptidase inhibitor | 0.053 0.014 CHEMBL3526894 | CHEMBL3526894 | |
| 0.062 | 0.174 | 0.078 | CC chemokine 5 receptor agonist | 0.078 0.074 CHEMBL724 | CHEMBL724 | |
| 0.042 | 0.155 | 0.123 | Insulin growth factor antagonist | 0.123 0.032 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.126 | 0.123 | Bradykinin antagonist | 0.044 0.018 CHEMBL3526894 0.123 0.005 CHEMBL3526734 | CHEMBL3526734 | |
| 0.056 | 0.174 | 0.162 | Nitric-oxide synthase inhibitor | 0.114 0.042 CHEMBL3526894 0.143 0.025 CHEMBL3526895 0.162 0.018 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.139 | 0.21 | Alpha 1a adrenoreceptor antagonist | 0.21 0.015 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.132 | 0.031 | Cholesterol ester transfer protein antagonist | 0.031 0.023 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.147 | 0.112 | Dopamine antagonist | 0.112 0.034 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.13 | 0.365 | Cholecystokinin agonist | 0.365 0.002 CHEMBL3527572 | CHEMBL3527572 | |
| 0.074 | 0.201 | 0.21 | Acetylcholine M1 receptor antagonist | 0.21 0.038 CHEMBL3526894 0.195 0.045 CHEMBL3526734 | CHEMBL3526894 | |
| 0.046 | 0.174 | 0.232 | Polo-like kinase-4 inhibitor | 0.091 0.087 CHEMBL3526895 0.232 0.01 CHEMBL724 | CHEMBL724 | |
| 0.029 | 0.16 | 0.093 | Acetylcholine M4 receptor antagonist | 0.093 0.034 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.142 | 0.02 | Factor XIII inhibitor | 0.02 0.017 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.176 | 0.375 | Antiadrenergic | 0.078 0.073 CHEMBL3526895 0.375 0.009 CHEMBL724 | CHEMBL724 | |
| 0.027 | 0.167 | 0.07 | Syk tyrosine kinase inhibitor | 0.07 0.049 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.159 | 0.034 | Protein kinase C beta I inhibitor | 0.034 0.02 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.162 | 0.071 | Kallikrein inhibitor | 0.071 0.018 CHEMBL3526894 0.046 0.034 CHEMBL3526734 | CHEMBL3526894 | |
| 0.01 | 0.155 | 0.052 | DNA gyrase subunit B inhibitor | 0.039 0.025 CHEMBL3526895 0.052 0.012 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.161 | 0.208 | 5 Hydroxytryptamine 1A antagonist | 0.208 0.014 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.158 | 0.043 | CDK6/cyclin D3 inhibitor | 0.043 0.01 CHEMBL724 | CHEMBL724 | |
| 0.035 | 0.181 | 0.374 | Adrenaline antagonist | 0.374 0.009 CHEMBL724 | CHEMBL724 | |
| 0.034 | 0.181 | 0.097 | Fibroblast growth factor 1 antagonist | 0.097 0.06 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.156 | 0.055 | Potassium channel small-conductance Ca-activated activator | 0.055 0.01 CHEMBL724 | CHEMBL724 | |
| 0.036 | 0.185 | 0.091 | Secretase beta inhibitor | 0.091 0.024 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.159 | 0.03 | Tryptophan hydroxylase 1 inhibitor | 0.03 0.004 CHEMBL3526895 | CHEMBL3526895 | |
| 0.016 | 0.165 | 0.096 | Dopamine D2 antagonist | 0.096 0.034 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.168 | 0.051 | Sphingosine kinase 1 inhibitor | 0.05 0.017 CHEMBL3526894 0.051 0.016 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.165 | 0.031 | Protein kinase C beta II inhibitor | 0.031 0.026 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.168 | 0.215 | Adenosine A2a receptor antagonist | 0.058 0.046 CHEMBL724 0.196 0.01 CHEMBL3527516 0.215 0.009 CHEMBL3527230 | CHEMBL3527230 | |
| 0.031 | 0.184 | 0.239 | Alpha 2a adrenoreceptor antagonist | 0.239 0.01 CHEMBL724 | CHEMBL724 | |
| 0.131 | 0.285 | 0.463 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.463 0.011 CHEMBL724 0.322 0.049 CHEMBL3527515 0.227 0.128 CHEMBL3526734 | CHEMBL724 | |
| 0.056 | 0.211 | 0.15 | Phosphodiesterase inhibitor | 0.15 0.058 CHEMBL724 0.125 0.077 CHEMBL3527515 | CHEMBL724 | |
| 0.044 | 0.2 | 0.171 | Caspase 7 inhibitor | 0.171 0.005 CHEMBL724 | CHEMBL724 | |
| 0.039 | 0.197 | 0.159 | Inducible nitric-oxide synthase inhibitor | 0.08 0.062 CHEMBL3526895 0.159 0.014 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.178 | 0.083 | Phosphatidylinositol 3-kinase gamma inhibitor | 0.083 0.019 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.176 | 0.199 | NMDA 2 receptor antagonist | 0.199 0.009 CHEMBL3526894 0.08 0.044 CHEMBL3526895 0.093 0.036 CHEMBL3527572 | CHEMBL3526894 | |
| 0.054 | 0.213 | 0.133 | Tyrosine-protein kinase receptor antagonist | 0.133 0.075 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.165 | 0.03 | Acetylcholine M4 receptor agonist | 0.03 0.022 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.18 | 0.209 | 5 Hydroxytryptamine 1 antagonist | 0.209 0.016 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.171 | 0.047 | Plasma kallikrein inhibitor | 0.047 0.013 CHEMBL3526894 0.041 0.018 CHEMBL3526734 | CHEMBL3526894 | |
| 0.008 | 0.172 | 0.44 | Trypsin I inhibitor | 0.44 0.004 CHEMBL3526894 0.298 0.004 CHEMBL3526734 | CHEMBL3526894 | |
| 0.017 | 0.182 | 0.036 | ATR kinase inhibitor | 0.036 0.017 CHEMBL724 | CHEMBL724 | |
| 0.029 | 0.194 | 0.136 | 5 Hydroxytryptamine 2C antagonist | 0.136 0.03 CHEMBL724 | CHEMBL724 | |
| 0.057 | 0.224 | 0.096 | mTOR complex 1 inhibitor | 0.096 0.071 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.182 | 0.066 | 5 Hydroxytryptamine uptake inhibitor | 0.066 0.042 CHEMBL724 | CHEMBL724 | |
| 0.066 | 0.237 | 0.269 | Protein kinase stimulant | 0.196 0.043 CHEMBL3527573 0.16 0.062 CHEMBL3526733 0.227 0.033 CHEMBL3527516 0.269 0.022 CHEMBL3527230 0.243 0.028 CHEMBL3526644 | CHEMBL3527230 | |
| 0.025 | 0.197 | 0.076 | Sphingosine kinase inhibitor | 0.073 0.021 CHEMBL3526894 0.076 0.019 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.194 | 0.048 | Purinergic P2X4 antagonist | 0.048 0.028 CHEMBL724 | CHEMBL724 | |
| 0.047 | 0.221 | 0.115 | TRKA antagonist | 0.115 0.072 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.185 | 0.06 | Guanylate cyclase inhibitor | 0.06 0.012 CHEMBL3526895 0.049 0.022 CHEMBL724 0.055 0.016 CHEMBL3527516 0.049 0.022 CHEMBL3527230 | CHEMBL3526895 | |
| 0.01 | 0.185 | 0.05 | NMDA 2D receptor antagonist | 0.043 0.009 CHEMBL3526895 0.05 0.007 CHEMBL3527572 | CHEMBL3527572 | |
| 0.026 | 0.202 | 0.089 | Rho-associated kinase inhibitor | 0.089 0.04 CHEMBL724 | CHEMBL724 | |
| 0.167 | 0.346 | 0.331 | MAP kinase 1 inhibitor | 0.331 0.15 CHEMBL724 0.26 0.221 CHEMBL3527229 | CHEMBL724 | |
| 0.017 | 0.2 | 0.075 | Cyclin A1 inhibitor | 0.075 0.017 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.192 | 0.097 | Diamine oxidase inhibitor | 0.097 0.004 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.2 | 0.115 | Acetylcholine M2 receptor antagonist | 0.115 0.018 CHEMBL3526734 | CHEMBL3526734 | |
| 0.014 | 0.201 | 0.21 | Alpha 1b adrenoreceptor antagonist | 0.21 0.014 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.196 | 0.026 | LFA antagonist | 0.026 0.023 CHEMBL724 | CHEMBL724 | |
| 0.037 | 0.226 | 0.188 | Protein kinase C delta inhibitor | 0.084 0.071 CHEMBL3526895 0.188 0.01 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.193 | 0.018 | CXC chemokine 4 receptor agonist | 0.018 0.007 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.198 | 0.023 | Cyclin D2 inhibitor | 0.023 0.003 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.212 | 0.168 | 5 Hydroxytryptamine 3A antagonist | 0.168 0.004 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.211 | 0.286 | Alpha 2 adrenoreceptor agonist | 0.286 0.004 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.208 | 0.022 | Granulocyte colony stimulating factor receptor agonist | 0.022 0.006 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.216 | 0.137 | CDC7 inhibitor | 0.137 0.012 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.231 | 0.12 | Pim-1 kinase inhibitor | 0.12 0.042 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.212 | 0.087 | Dopamine D4 agonist | 0.087 0.018 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.204 | 0.014 | Egl nine homolog 1 inhibitor | 0.014 0.01 CHEMBL3526895 | CHEMBL3526895 | |
| 0.004 | 0.206 | 0.042 | Dopamine autoreceptor agonist | 0.042 0.009 CHEMBL724 | CHEMBL724 | |
| 0.033 | 0.236 | 0.077 | AXL receptor tyrosine kinase inhibitor | 0.077 0.065 CHEMBL724 | CHEMBL724 | |
| 0.104 | 0.307 | 0.47 | 5 Hydroxytryptamine release stimulant | 0.204 0.118 CHEMBL3526895 0.47 0.032 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.215 | 0.19 | Alpha 1d adrenoreceptor antagonist | 0.19 0.01 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.225 | 0.131 | Phosphodiesterase V inhibitor | 0.072 0.049 CHEMBL3526895 0.131 0.015 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.222 | 0.035 | DNA topoisomerase IV inhibitor | 0.035 0.013 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.232 | 0.422 | Thrombin inhibitor | 0.422 0.004 CHEMBL3526894 0.339 0.004 CHEMBL3526734 0.074 0.05 CHEMBL3527572 | CHEMBL3526894 | |
| 0.006 | 0.213 | 0.052 | Factor XI inhibitor | 0.052 0.009 CHEMBL3526894 | CHEMBL3526894 | |
| 0.105 | 0.313 | 0.399 | DNA synthesis inhibitor | 0.271 0.055 CHEMBL3526895 0.258 0.061 CHEMBL724 0.399 0.022 CHEMBL3527516 0.399 0.022 CHEMBL3527230 0.281 0.051 CHEMBL3526644 | CHEMBL3527230 | |
| 0.016 | 0.224 | 0.139 | 5 Hydroxytryptamine 3 antagonist | 0.139 0.01 CHEMBL724 | CHEMBL724 | |
| 0.106 | 0.315 | 0.188 | Heat shock protein 70 antagonist | 0.184 0.01 CHEMBL3526895 0.188 0.009 CHEMBL724 0.143 0.064 CHEMBL3527516 | CHEMBL724 | |
| 0.075 | 0.285 | 0.198 | Adenylate cyclase stimulant | 0.154 0.056 CHEMBL3526895 0.198 0.014 CHEMBL724 | CHEMBL724 | |
| 0.041 | 0.251 | 0.086 | Phosphodiesterase I inhibitor | 0.086 0.065 CHEMBL724 | CHEMBL724 | |
| 0.133 | 0.344 | 0.505 | Calcium channel activator | 0.33 0.064 CHEMBL3526895 0.505 0.005 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.231 | 0.057 | Myc inhibitor | 0.057 0.034 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.237 | 0.149 | NMDA receptor antagonist | 0.133 0.03 CHEMBL3526894 0.149 0.025 CHEMBL3526895 | CHEMBL3526895 | |
| 0.054 | 0.27 | 0.121 | Hedgehog signaling inhibitor | 0.121 0.039 CHEMBL724 | CHEMBL724 | |
| 0.034 | 0.252 | 0.396 | Trypsin inhibitor | 0.396 0.004 CHEMBL3526894 0.325 0.004 CHEMBL3526734 | CHEMBL3526894 | |
| 0.037 | 0.257 | 0.341 | GABA C receptor agonist | 0.228 0.016 CHEMBL3526895 0.341 0.007 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.235 | 0.122 | Cyclin A inhibitor | 0.122 0.017 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.225 | 0.075 | Histamine H4 receptor agonist | 0.075 0.004 CHEMBL724 | CHEMBL724 | |
| 0.037 | 0.26 | 0.12 | TRKB antagonist | 0.12 0.072 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.235 | 0.146 | Adenosine A2 receptor antagonist | 0.058 0.051 CHEMBL724 0.136 0.019 CHEMBL3527516 0.146 0.017 CHEMBL3527230 | CHEMBL3527230 | |
| 0.049 | 0.273 | 0.298 | Activin receptor-like kinase 2 inhibitor | 0.298 0.013 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.246 | 0.082 | DNA gyrase inhibitor | 0.066 0.041 CHEMBL3526895 0.077 0.029 CHEMBL724 0.082 0.026 CHEMBL3526644 | CHEMBL3526644 | |
| 0.014 | 0.239 | 0.065 | Tryptophan 5 hydroxylase inhibitor | 0.065 0.004 CHEMBL3526895 0.037 0.02 CHEMBL724 | CHEMBL3526895 | |
| 0.153 | 0.379 | 0.388 | MAP kinase kinase 6 inhibitor | 0.388 0.066 CHEMBL724 | CHEMBL724 | |
| 0.044 | 0.273 | 0.113 | Growth factor antagonist | 0.113 0.099 CHEMBL724 | CHEMBL724 | |
| 0.061 | 0.291 | 0.175 | Anticonvulsant | 0.175 0.103 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.253 | 0.091 | Phospholipase D inhibitor | 0.091 0.021 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.234 | 0.017 | Cyclin T1 inhibitor | 0.017 0.014 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.257 | 0.067 | Aminopeptidase I inhibitor | 0.067 0.058 CHEMBL724 | CHEMBL724 | |
| 0.052 | 0.287 | 0.14 | Acetylcholine release stimulant | 0.14 0.024 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.255 | 0.129 | Phosphodiesterase 5A inhibitor | 0.066 0.054 CHEMBL3526895 0.129 0.016 CHEMBL724 | CHEMBL724 | |
| 0.104 | 0.343 | 0.629 | Vasodilator, peripheral | 0.414 0.051 CHEMBL3526895 0.629 0.013 CHEMBL724 0.417 0.05 CHEMBL3527516 0.312 0.091 CHEMBL3527230 | CHEMBL724 | |
| 0.041 | 0.279 | 0.208 | Cyclin-dependent kinase 7 inhibitor | 0.208 0.031 CHEMBL724 | CHEMBL724 | |
| 0.036 | 0.276 | 0.213 | Cyclin-dependent kinase inhibitor | 0.213 0.034 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.254 | 0.105 | CDK4/cyclin D1 inhibitor | 0.105 0.013 CHEMBL724 | CHEMBL724 | |
| 0.04 | 0.281 | 0.169 | Nav1.3 sodium channel blocker | 0.169 0.037 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.262 | 0.134 | Protein kinase C alpha inhibitor | 0.134 0.013 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.25 | 0.035 | Alpha 1a adrenoreceptor agonist | 0.035 0.008 CHEMBL724 | CHEMBL724 | |
| 0.037 | 0.28 | 0.221 | Alpha 2c adrenoreceptor antagonist | 0.221 0.014 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.261 | 0.098 | Protein kinase C eta inhibitor | 0.049 0.045 CHEMBL3526895 0.098 0.018 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.267 | 0.082 | 5 Hydroxytryptamine 1B agonist | 0.082 0.011 CHEMBL724 | CHEMBL724 | |
| 0.047 | 0.296 | 0.131 | Nav1.5 sodium channel blocker | 0.131 0.042 CHEMBL724 | CHEMBL724 | |
| 0.031 | 0.281 | 0.341 | Glutamate receptor antagonist | 0.341 0.007 CHEMBL3526895 | CHEMBL3526895 | |
| 0.019 | 0.27 | 0.142 | Cyclin-dependent kinase 4 inhibitor | 0.142 0.013 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.272 | 0.09 | Protein kinase C iota inhibitor | 0.09 0.022 CHEMBL724 | CHEMBL724 | |
| 0.041 | 0.295 | 0.226 | Alpha-N-acetylglucosaminidase inhibitor | 0.226 0.027 CHEMBL3526895 0.192 0.037 CHEMBL724 | CHEMBL3526895 | |
| 0.027 | 0.281 | 0.313 | Protein kinase (CK1) inhibitor | 0.313 0.016 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.27 | 0.027 | Thymidine phosphorylase inhibitor | 0.027 0.016 CHEMBL724 | CHEMBL724 | |
| 0.048 | 0.309 | 0.662 | Anticoagulant | 0.662 0.005 CHEMBL3526894 0.135 0.095 CHEMBL3527573 0.145 0.085 CHEMBL3526733 0.593 0.006 CHEMBL3526734 0.178 0.062 CHEMBL3526644 0.34 0.023 CHEMBL3527572 | CHEMBL3526894 | |
| 0.018 | 0.285 | 0.092 | Sphingosine kinase 2 inhibitor | 0.051 0.045 CHEMBL3526894 0.092 0.01 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.291 | 0.051 | Nicotinic alpha3beta2 receptor antagonist | 0.051 0.041 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.273 | 0.055 | Bradykinin B2 receptor antagonist | 0.03 0.023 CHEMBL3526894 0.055 0.005 CHEMBL3526734 | CHEMBL3526734 | |
| 0.06 | 0.331 | 0.389 | Platelet adhesion inhibitor | 0.389 0.013 CHEMBL3526894 0.263 0.045 CHEMBL3527573 0.256 0.047 CHEMBL3526733 0.148 0.107 CHEMBL3527516 0.153 0.102 CHEMBL3527230 0.269 0.043 CHEMBL3526734 0.31 0.031 CHEMBL3526644 0.258 0.047 CHEMBL3527572 | CHEMBL3526894 | |
| 0.012 | 0.284 | 0.072 | Acetylcholine M5 receptor agonist | 0.072 0.042 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.292 | 0.284 | Protein kinase (CK1) delta inhibitor | 0.284 0.013 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.308 | 0.247 | 5 Hydroxytryptamine 3A agonist | 0.247 0.005 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.303 | 0.212 | Glycogen synthase kinase-3 beta inhibitor | 0.212 0.026 CHEMBL724 | CHEMBL724 | |
| 0.055 | 0.334 | 0.138 | Thiol protease inhibitor | 0.138 0.082 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.284 | 0.033 | 5 Hydroxytryptamine 1D agonist | 0.033 0.017 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.288 | 0.035 | Kainate receptor antagonist | 0.035 0.034 CHEMBL3526895 | CHEMBL3526895 | |
| 0.012 | 0.3 | 0.094 | CDK4/cyclin D inhibitor | 0.094 0.016 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.321 | 0.193 | Antineoplastic alkaloid | 0.193 0.016 CHEMBL3527515 0.159 0.025 CHEMBL3526734 | CHEMBL3527515 | |
| 0.042 | 0.331 | 0.283 | Activin receptor-like kinase 4 inhibitor | 0.283 0.005 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.295 | 0.016 | S-adenosyl-L-homocysteine hydrolase inhibitor | 0.016 0.009 CHEMBL3527516 0.016 0.009 CHEMBL3527230 | CHEMBL3527230 | |
| 0.004 | 0.295 | 0.05 | Antimetabolite | 0.05 0.031 CHEMBL3527516 0.042 0.038 CHEMBL3527230 | CHEMBL3527516 | |
| 0.012 | 0.303 | 0.067 | Dopamine agonist | 0.067 0.046 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.305 | 0.345 | Plasmin inhibitor | 0.345 0.004 CHEMBL3526894 0.286 0.004 CHEMBL3526734 | CHEMBL3526894 | |
| 0.002 | 0.295 | 0.029 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.029 0.019 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.317 | 0.082 | Heat shock protein 90 beta antagonist | 0.082 0.019 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.308 | 0.072 | Dopamine D3 antagonist | 0.072 0.037 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.322 | 0.118 | Protein kinase C zeta inhibitor | 0.084 0.077 CHEMBL3526894 0.118 0.033 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.308 | 0.133 | 5 Hydroxytryptamine 7 antagonist | 0.133 0.02 CHEMBL724 | CHEMBL724 | |
| 0.109 | 0.409 | 0.234 | Tyrosine 3 hydroxylase inhibitor | 0.206 0.125 CHEMBL3526895 0.234 0.085 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.327 | 0.113 | Hepatocyte growth factor antagonist | 0.113 0.04 CHEMBL724 | CHEMBL724 | |
| 0.002 | 0.305 | 0.014 | Egl nine homolog 3 inhibitor | 0.014 0.006 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.311 | 0.037 | CDK4/cyclin D3 inhibitor | 0.037 0.012 CHEMBL724 | CHEMBL724 | |
| 0.033 | 0.336 | 0.239 | Thrombolytic | 0.128 0.102 CHEMBL3527573 0.127 0.102 CHEMBL3526733 0.239 0.036 CHEMBL3526644 0.136 0.093 CHEMBL3527572 | CHEMBL3526644 | |
| 0.011 | 0.316 | 0.063 | Histamine H1 receptor agonist | 0.063 0.007 CHEMBL724 | CHEMBL724 | |
| 0.059 | 0.365 | 0.209 | Hemostatic | 0.127 0.1 CHEMBL3526894 0.137 0.086 CHEMBL3526895 0.209 0.029 CHEMBL724 0.194 0.035 CHEMBL3526644 0.201 0.032 CHEMBL3527572 | CHEMBL724 | |
| 0.017 | 0.329 | 0.117 | Aurora-A kinase inhibitor | 0.117 0.056 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.326 | 0.138 | Cyclin A2 inhibitor | 0.138 0.015 CHEMBL724 | CHEMBL724 | |
| 0.036 | 0.35 | 0.159 | Beta amyloid protein antagonist | 0.159 0.035 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.325 | 0.174 | Tryptase inhibitor | 0.174 0.004 CHEMBL3526894 0.098 0.005 CHEMBL3526734 | CHEMBL3526894 | |
| 0.022 | 0.341 | 0.208 | Glycogen synthase kinase-3 inhibitor | 0.208 0.03 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.334 | 0.088 | Vanilloid antagonist | 0.088 0.042 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.33 | 0.054 | Stearoyl-CoA desaturase inhibitor | 0.054 0.02 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.333 | 0.06 | Phosphodiesterase 4B inhibitor | 0.06 0.056 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.334 | 0.046 | Mannosidase inhibitor | 0.046 0.03 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.339 | 0.049 | Alpha-mannosidase inhibitor | 0.049 0.045 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.344 | 0.042 | Kainate receptor agonist | 0.042 0.026 CHEMBL3526895 | CHEMBL3526895 | |
| 0.008 | 0.338 | 0.115 | Adenosine A1 receptor antagonist | 0.115 0.02 CHEMBL3527516 0.083 0.027 CHEMBL3527230 | CHEMBL3527516 | |
| 0.114 | 0.446 | 0.24 | 5 Hydroxytryptamine 3E antagonist | 0.24 0.021 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.355 | 0.152 | Cyclin-dependent kinase 9 inhibitor | 0.152 0.033 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.356 | 0.09 | Glutamate (mGluR7) antagonist | 0.09 0.017 CHEMBL3526895 0.088 0.019 CHEMBL724 | CHEMBL3526895 | |
| 0.008 | 0.345 | 0.057 | Glutamate (mGluR3) antagonist | 0.057 0.009 CHEMBL3526895 | CHEMBL3526895 | |
| 0.013 | 0.351 | 0.12 | Protein kinase (CK2) inhibitor | 0.12 0.048 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.354 | 0.055 | 5 Hydroxytryptamine 7 agonist | 0.055 0.041 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.365 | 0.068 | Exportin-1 inhibitor | 0.068 0.048 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.344 | 0.066 | Geranyltranstransferase inhibitor | 0.066 0.009 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.357 | 0.112 | Rho-associated kinase I inhibitor | 0.112 0.024 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.361 | 0.05 | Angiotensin-converting enzyme inhibitor | 0.05 0.047 CHEMBL3526895 | CHEMBL3526895 | |
| 0.007 | 0.355 | 0.055 | NMDA 2C receptor antagonist | 0.055 0.053 CHEMBL3526895 | CHEMBL3526895 | |
| 0.01 | 0.359 | 0.074 | 5 Hydroxytryptamine 1D antagonist | 0.074 0.035 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.382 | 0.124 | MAP kinase 13 inhibitor | 0.124 0.053 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.359 | 0.06 | Histamine H2 receptor agonist | 0.06 0.014 CHEMBL724 | CHEMBL724 | |
| 0.15 | 0.502 | 0.502 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.294 0.221 CHEMBL3526895 0.502 0.033 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.362 | 0.077 | 5 Hydroxytryptamine 1B antagonist | 0.077 0.036 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.361 | 0.076 | Cyclin D3 inhibitor | 0.076 0.011 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.383 | 0.167 | Ribosomal protein S6 kinase inhibitor | 0.167 0.054 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.376 | 0.062 | Potassium channel (Ca-activated) blocker | 0.062 0.037 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.367 | 0.233 | Cholecystokinin A agonist | 0.233 0.002 CHEMBL3527572 | CHEMBL3527572 | |
| 0.056 | 0.424 | 0.172 | MAP kinase 3 inhibitor | 0.172 0.041 CHEMBL724 | CHEMBL724 | |
| 0.031 | 0.4 | 0.238 | Anesthetic general | 0.238 0.056 CHEMBL724 | CHEMBL724 | |
| 0.095 | 0.466 | 0.251 | Nitric-oxide synthase stimulant | 0.251 0.032 CHEMBL724 | CHEMBL724 | |
| 0.044 | 0.418 | 0.09 | Transforming growth factor beta 3 antagonist | 0.09 0.038 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.391 | 0.133 | Adrenaline agonist | 0.133 0.02 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.379 | 0.064 | 5 Hydroxytryptamine 3B antagonist | 0.064 0.01 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.397 | 0.11 | GABA A receptor agonist | 0.11 0.03 CHEMBL724 | CHEMBL724 | |
| 0.034 | 0.413 | 0.105 | Alpha 2d adrenoreceptor antagonist | 0.105 0.04 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.405 | 0.327 | Psychostimulant | 0.295 0.044 CHEMBL3526895 0.327 0.036 CHEMBL724 | CHEMBL724 | |
| 0.048 | 0.431 | 0.216 | Polo-like kinase-3 inhibitor | 0.216 0.037 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.407 | 0.162 | UDP-glucose 4-epimerase inhibitor | 0.107 0.053 CHEMBL724 0.157 0.026 CHEMBL3527516 0.162 0.025 CHEMBL3527230 | CHEMBL3527230 | |
| 0.02 | 0.41 | 0.066 | Corticotropin releasing factor 2 receptor antagonist | 0.066 0.034 CHEMBL724 | CHEMBL724 | |
| 0.084 | 0.477 | 0.127 | CC chemokine 6 receptor antagonist | 0.12 0.116 CHEMBL3527573 0.121 0.112 CHEMBL3526733 0.127 0.081 CHEMBL3526644 | CHEMBL3526644 | |
| 0.048 | 0.441 | 0.24 | 5 Hydroxytryptamine 1E antagonist | 0.24 0.085 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.398 | 0.279 | Factor X inhibitor | 0.279 0.005 CHEMBL3526894 0.196 0.005 CHEMBL3526734 | CHEMBL3526894 | |
| 0.006 | 0.401 | 0.046 | Dopamine D5 agonist | 0.046 0.021 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.416 | 0.11 | Lck kinase inhibitor | 0.11 0.093 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.406 | 0.162 | 5 Hydroxytryptamine 1F antagonist | 0.162 0.014 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.41 | 0.081 | Protein kinase C epsilon inhibitor | 0.081 0.019 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.435 | 0.195 | Cell wall synthesis inhibitor | 0.195 0.032 CHEMBL3526895 0.17 0.047 CHEMBL3526644 0.157 0.059 CHEMBL3527572 | CHEMBL3526895 | |
| 0.02 | 0.425 | 0.15 | MAP-kinase-activated kinase inhibitor | 0.15 0.015 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.417 | 0.091 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.091 0.017 CHEMBL724 0.061 0.033 CHEMBL3527516 | CHEMBL724 | |
| 0.074 | 0.482 | 0.245 | Insulysin inhibitor | 0.245 0.101 CHEMBL3526895 0.218 0.132 CHEMBL724 | CHEMBL3526895 | |
| 0.014 | 0.428 | 0.132 | MAP-kinase-activated kinase 2 inhibitor | 0.132 0.016 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.437 | 0.083 | Prolactin inhibitor | 0.083 0.076 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.433 | 0.068 | Lysine-specific demethylase 1A inhibitor | 0.068 0.019 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.445 | 0.15 | Interleukin 1 beta converting enzyme inhibitor | 0.094 0.065 CHEMBL3526895 0.15 0.017 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.428 | 0.06 | GP IIb/IIIa receptor antagonist | 0.06 0.028 CHEMBL3526894 | CHEMBL3526894 | |
| 0.019 | 0.445 | 0.071 | Histone deacetylase SIRT3 inhibitor | 0.071 0.027 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.442 | 0.098 | Focal adhesion kinase 1 inhibitor | 0.098 0.031 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.441 | 0.228 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.228 0.03 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.454 | 0.096 | Histamine H2 receptor antagonist | 0.096 0.039 CHEMBL724 | CHEMBL724 | |
| 0.042 | 0.478 | 0.152 | Glutamate release inhibitor | 0.089 0.064 CHEMBL3526895 0.152 0.009 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.445 | 0.073 | Amidase inhibitor | 0.073 0.045 CHEMBL724 | CHEMBL724 | |
| 0.023 | 0.461 | 0.294 | Alpha 2b adrenoreceptor antagonist | 0.294 0.009 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.448 | 0.099 | Phenylalanine 4-hydroxylase inhibitor | 0.099 0.026 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.478 | 0.323 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.323 0.036 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.456 | 0.136 | CDK/cyclin complex inhibitor | 0.136 0.034 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.455 | 0.085 | Carbonic anhydrase stimulant | 0.085 0.024 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.457 | 0.174 | RET inhibitor | 0.174 0.05 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.466 | 0.178 | Protein kinase C gamma inhibitor | 0.104 0.071 CHEMBL3526895 0.178 0.019 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.456 | 0.041 | NMDA receptor subunit 3B antagonist | 0.041 0.034 CHEMBL3526895 | CHEMBL3526895 | |
| 0.011 | 0.464 | 0.161 | CDK2/cyclin E2 inhibitor | 0.161 0.015 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.476 | 0.082 | Alpha 1b adrenoreceptor agonist | 0.082 0.008 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.487 | 0.098 | MAP kinase kinase 7 inhibitor | 0.098 0.015 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.478 | 0.169 | Ca2+/calmodulin-dependent kinase II delta inhibitor | 0.169 0.056 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.481 | 0.129 | Src kinase inhibitor | 0.129 0.1 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.471 | 0.065 | Carbamoyl phosphate synthetase inhibitor | 0.065 0.038 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.478 | 0.073 | Cyclin H inhibitor | 0.073 0.025 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.475 | 0.05 | Aconitate hydratase inhibitor | 0.05 0.039 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.472 | 0.112 | Protein kinase (CK2) alpha inhibitor | 0.112 0.067 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.495 | 0.072 | Vanilloid 4 agonist | 0.072 0.058 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.494 | 0.124 | MAP kinase 12 inhibitor | 0.124 0.066 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.476 | 0.04 | NMDA receptor subunit 3A antagonist | 0.04 0.025 CHEMBL3526895 | CHEMBL3526895 | |
| 0.011 | 0.486 | 0.086 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.086 0.028 CHEMBL724 | CHEMBL724 | |
| 0.027 | 0.508 | 0.376 | Platelet antagonist | 0.376 0.032 CHEMBL3526894 0.156 0.138 CHEMBL3526733 0.375 0.032 CHEMBL3526734 0.174 0.122 CHEMBL3526644 | CHEMBL3526894 | |
| 0.005 | 0.487 | 0.024 | Protein 30S ribosomal subunit inhibitor | 0.022 0.02 CHEMBL3527573 0.024 0.017 CHEMBL3526644 | CHEMBL3526644 | |
| 0.007 | 0.491 | 0.04 | Glutamate (mGluR1a) antagonist | 0.04 0.03 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.49 | 0.049 | Argininosuccinate synthase inhibitor | 0.049 0.048 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.492 | 0.061 | Check point kinase 1 inhibitor | 0.061 0.057 CHEMBL724 | CHEMBL724 | |
| 0.049 | 0.534 | 0.127 | Sphingosine 1-phosphate receptor 5 antagonist | 0.127 0.108 CHEMBL3526895 | CHEMBL3526895 | |
| 0.011 | 0.497 | 0.068 | Dopamine beta hydroxylase inhibitor | 0.068 0.009 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.503 | 0.07 | Alpha 1L adrenoreceptor agonist | 0.07 0.005 CHEMBL724 | CHEMBL724 | |
| 0.03 | 0.518 | 0.127 | Neuropeptide Y1 antagonist | 0.127 0.106 CHEMBL724 | CHEMBL724 | |
| 0.029 | 0.517 | 0.126 | Nav1.1 sodium channel blocker | 0.126 0.044 CHEMBL3526894 | CHEMBL3526894 | |
| 0.01 | 0.499 | 0.059 | Epithelial sodium channel blocker | 0.059 0.03 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.492 | 0.024 | Methionyl aminopeptidase 2 inhibitor | 0.024 0.019 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.509 | 0.154 | Nav1.6 sodium channel blocker | 0.154 0.049 CHEMBL724 | CHEMBL724 | |
| 0.027 | 0.517 | 0.139 | TRPA1 agonist | 0.139 0.04 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.51 | 0.085 | Somatostatin 1 agonist | 0.085 0.046 CHEMBL3526895 | CHEMBL3526895 | |
| 0.017 | 0.51 | 0.148 | GABA receptor agonist | 0.148 0.037 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.51 | 0.186 | Ferrochelatase inhibitor | 0.186 0.026 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.511 | 0.056 | Neurotensin receptor antagonist | 0.056 0.025 CHEMBL3526894 0.044 0.032 CHEMBL3526734 | CHEMBL3526894 | |
| 0.003 | 0.503 | 0.038 | Kainate receptor 2 antagonist | 0.038 0.023 CHEMBL3526895 | CHEMBL3526895 | |
| 0.046 | 0.547 | 0.414 | Superoxide dismutase inhibitor | 0.201 0.117 CHEMBL3526895 0.414 0.024 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.507 | 0.03 | 1,3-Beta-glucan synthase inhibitor | 0.03 0.014 CHEMBL3527572 | CHEMBL3527572 | |
| 0.024 | 0.527 | 0.08 | Bromodomain-containing protein 2 inhibitor | 0.08 0.077 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.51 | 0.037 | Delayed rectifier potassium channel blocker | 0.037 0.027 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.518 | 0.064 | Glutamate (mGluR4) antagonist | 0.064 0.012 CHEMBL3526895 | CHEMBL3526895 | |
| 0.003 | 0.507 | 0.016 | CDK2/cyclin A3 inhibitor | 0.016 0.012 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.524 | 0.229 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.229 0.055 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.523 | 0.13 | Histamine N-methyltransferase inhibitor | 0.13 0.023 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.513 | 0.041 | Oleamide hydrolase inhibitor | 0.041 0.037 CHEMBL724 | CHEMBL724 | |
| 0.073 | 0.584 | 0.139 | Ca2+-transporting ATPase inhibitor | 0.139 0.079 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.519 | 0.028 | Estrogen-related receptor gamma antagonist | 0.028 0.021 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.518 | 0.063 | Alcohol oxidase inhibitor | 0.063 0.033 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.518 | 0.059 | CDK1/cyclin B inhibitor | 0.059 0.048 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.519 | 0.026 | Acid ceramidase inhibitor | 0.026 0.016 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.534 | 0.168 | GABA C receptor rho-1 antagonist | 0.168 0.015 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.525 | 0.047 | CDK7/cyclin H inhibitor | 0.047 0.029 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.532 | 0.061 | Phosphodiesterase 1A inhibitor | 0.061 0.038 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.527 | 0.062 | Histidine decarboxylase inhibitor | 0.062 0.059 CHEMBL724 | CHEMBL724 | |
| 0.052 | 0.573 | 0.259 | Vasodilator, coronary | 0.233 0.151 CHEMBL3526895 0.252 0.132 CHEMBL724 0.254 0.13 CHEMBL3527516 0.259 0.125 CHEMBL3527230 | CHEMBL3527230 | |
| 0.012 | 0.534 | 0.061 | 5 Hydroxytryptamine 5A antagonist | 0.061 0.043 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.548 | 0.089 | Granulocyte macrophage colony stimulating factor agonist | 0.089 0.054 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.532 | 0.114 | Porphobilinogen synthase inhibitor | 0.114 0.03 CHEMBL724 | CHEMBL724 | |
| 0.057 | 0.585 | 0.125 | Death-associated protein kinase 1 inhibitor | 0.125 0.097 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.547 | 0.086 | Phosphodiesterase VI inhibitor | 0.086 0.033 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.541 | 0.071 | Glutamate (mGluR group III) antagonist | 0.071 0.009 CHEMBL3526895 | CHEMBL3526895 | |
| 0.021 | 0.554 | 0.175 | Interleukin 8 antagonist | 0.175 0.021 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.536 | 0.03 | Myristoyl transferase inhibitor | 0.03 0.013 CHEMBL724 | CHEMBL724 | |
| 0.038 | 0.573 | 0.14 | DNA repair enzyme inhibitor | 0.14 0.042 CHEMBL724 0.11 0.095 CHEMBL3527516 0.111 0.094 CHEMBL3527230 | CHEMBL724 | |
| 0.011 | 0.547 | 0.08 | Glycine receptor antagonist | 0.08 0.057 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.555 | 0.073 | Phosphodiesterase VIII inhibitor | 0.073 0.047 CHEMBL3527515 0.066 0.064 CHEMBL3526734 | CHEMBL3527515 | |
| 0.037 | 0.578 | 0.282 | Hepatoprotectant | 0.27 0.038 CHEMBL3527573 0.272 0.038 CHEMBL3526733 0.168 0.091 CHEMBL3527516 0.166 0.093 CHEMBL3527230 0.282 0.035 CHEMBL3526644 | CHEMBL3526644 | |
| 0.016 | 0.558 | 0.091 | Aminopeptidase B inhibitor | 0.091 0.071 CHEMBL3526895 | CHEMBL3526895 | |
| 0.01 | 0.551 | 0.056 | 5 Hydroxytryptamine 5 antagonist | 0.056 0.043 CHEMBL724 | CHEMBL724 | |
| 0.002 | 0.546 | 0.036 | Imidazoline I1 receptor antagonist | 0.036 0.005 CHEMBL724 | CHEMBL724 | |
| 0.084 | 0.631 | 0.282 | 5 Hydroxytryptamine uptake stimulant | 0.282 0.055 CHEMBL724 | CHEMBL724 | |
| 0.037 | 0.585 | 0.147 | CF transmembrane conductance regulator agonist | 0.147 0.082 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.555 | 0.09 | Phosphodiesterase IV inhibitor | 0.09 0.053 CHEMBL724 | CHEMBL724 | |
| 0.049 | 0.599 | 0.154 | Neurotensin receptor agonist | 0.154 0.091 CHEMBL724 | CHEMBL724 | |
| 0.051 | 0.602 | 0.279 | MAP-kinase-activated kinase 5 inhibitor | 0.279 0.042 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.554 | 0.054 | Glutamate (mGluR1) antagonist | 0.054 0.044 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.555 | 0.078 | Alpha 1d adrenoreceptor agonist | 0.078 0.005 CHEMBL724 | CHEMBL724 | |
| 0.001 | 0.553 | 0.013 | Imidazoline I2 receptor antagonist | 0.013 0.006 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.558 | 0.06 | Biliverdin reductase inhibitor | 0.06 0.04 CHEMBL724 | CHEMBL724 | |
| 0.059 | 0.614 | 0.311 | Apoptosis antagonist | 0.311 0.079 CHEMBL3527573 0.303 0.083 CHEMBL3526733 0.247 0.13 CHEMBL3527516 0.256 0.122 CHEMBL3527230 0.306 0.081 CHEMBL3526644 | CHEMBL3527573 | |
| 0.057 | 0.611 | 0.491 | GABA C receptor rho-3 antagonist | 0.491 0.028 CHEMBL724 | CHEMBL724 | |
| 0.07 | 0.636 | 0.664 | Caspase 9 stimulant | 0.664 0.028 CHEMBL724 | CHEMBL724 | |
| 0.032 | 0.599 | 0.141 | Transcription factor STAT6 inhibitor | 0.141 0.03 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.581 | 0.06 | Glutamate (mGluR8) antagonist | 0.06 0.005 CHEMBL3526895 | CHEMBL3526895 | |
| 0.04 | 0.614 | 0.415 | Hypoglycemic | 0.348 0.038 CHEMBL3527573 0.346 0.039 CHEMBL3526733 0.189 0.124 CHEMBL3527516 0.191 0.121 CHEMBL3527230 0.415 0.025 CHEMBL3526644 | CHEMBL3526644 | |
| 0.003 | 0.577 | 0.024 | Alpha 2b adrenoreceptor agonist | 0.024 0.006 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.582 | 0.044 | Transforming growth factor beta 1 antagonist | 0.044 0.041 CHEMBL724 | CHEMBL724 | |
| 0.048 | 0.625 | 0.15 | MAP kinase kinase 4 inhibitor | 0.15 0.061 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.59 | 0.098 | Cell adhesion molecule inhibitor | 0.098 0.036 CHEMBL3527573 0.096 0.037 CHEMBL3526733 | CHEMBL3527573 | |
| 0.005 | 0.585 | 0.036 | AMPA 4 receptor antagonist | 0.036 0.034 CHEMBL3526895 | CHEMBL3526895 | |
| 0.032 | 0.611 | 0.142 | Interferon gamma antagonist | 0.142 0.09 CHEMBL3526895 0.138 0.095 CHEMBL724 | CHEMBL3526895 | |
| 0.004 | 0.586 | 0.022 | Alpha 2d adrenoreceptor agonist | 0.022 0.014 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.604 | 0.068 | Glutamate (mGluR6) antagonist | 0.068 0.045 CHEMBL3526895 | CHEMBL3526895 | |
| 0.096 | 0.685 | 0.233 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.233 0.091 CHEMBL724 | CHEMBL724 | |
| 0.027 | 0.617 | 0.196 | GABA C receptor rho-2 antagonist | 0.196 0.031 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.616 | 0.31 | Peroxidase inhibitor | 0.31 0.035 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.608 | 0.239 | Immunostimulant | 0.155 0.15 CHEMBL3527573 0.186 0.129 CHEMBL3527516 0.194 0.124 CHEMBL3527230 0.239 0.101 CHEMBL3526644 | CHEMBL3526644 | |
| 0.001 | 0.595 | 0.028 | Alpha 2a adrenoreceptor agonist | 0.028 0.005 CHEMBL724 | CHEMBL724 | |
| 0.015 | 0.61 | 0.186 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.186 0.056 CHEMBL724 | CHEMBL724 | |
| 0.085 | 0.68 | 0.19 | MAP kinase kinase 3 inhibitor | 0.19 0.153 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.605 | 0.059 | I kappa B kinase 2 inhibitor | 0.059 0.048 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.605 | 0.093 | Expectorant | 0.093 0.077 CHEMBL3526895 | CHEMBL3526895 | |
| 0.021 | 0.618 | 0.241 | DNA methylase inhibitor | 0.234 0.058 CHEMBL3526895 0.241 0.053 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.602 | 0.026 | Kainate receptor 4 antagonist | 0.026 0.016 CHEMBL3526895 | CHEMBL3526895 | |
| 0.028 | 0.63 | 0.455 | Hypoxia-inducible factor 1 alpha inhibitor | 0.455 0.019 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.614 | 0.17 | GABA C receptor antagonist | 0.17 0.021 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.614 | 0.179 | Protein kinase C mu inhibitor | 0.179 0.016 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.624 | 0.199 | Cell adhesion inhibitor | 0.112 0.072 CHEMBL3526895 0.199 0.025 CHEMBL3527573 0.196 0.026 CHEMBL3526733 0.125 0.062 CHEMBL3526644 | CHEMBL3527573 | |
| 0.004 | 0.61 | 0.067 | Cyclin E1 inhibitor | 0.067 0.029 CHEMBL724 | CHEMBL724 | |
| 0.02 | 0.627 | 0.098 | NADH dehydrogenase inhibitor | 0.098 0.046 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.619 | 0.057 | Ryanodine receptor antagonist | 0.057 0.047 CHEMBL724 | CHEMBL724 | |
| 0.035 | 0.644 | 0.191 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.191 0.082 CHEMBL724 | CHEMBL724 | |
| 0.028 | 0.638 | 0.125 | Interleukin 2 antagonist | 0.125 0.038 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.625 | 0.251 | MAP kinase kinase 2 inhibitor | 0.251 0.053 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.63 | 0.082 | ATPase (Vacuolar H+) inhibitor | 0.082 0.072 CHEMBL3526644 | CHEMBL3526644 | |
| 0.028 | 0.645 | 0.297 | Antithrombotic | 0.199 0.179 CHEMBL3526894 0.202 0.175 CHEMBL724 0.194 0.184 CHEMBL3526733 0.297 0.09 CHEMBL3526644 | CHEMBL3526644 | |
| 0.006 | 0.628 | 0.066 | Protein kinase B gamma inhibitor | 0.066 0.064 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.635 | 0.09 | Creatine kinase inhibitor | 0.09 0.071 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.636 | 0.087 | Cyclin D1 inhibitor | 0.087 0.013 CHEMBL724 | CHEMBL724 | |
| 0.002 | 0.631 | 0.029 | Cyclin E2 inhibitor | 0.029 0.02 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.635 | 0.053 | CDK2/cyclin E inhibitor | 0.053 0.05 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.64 | 0.101 | Mucolytic | 0.101 0.077 CHEMBL3526895 | CHEMBL3526895 | |
| 0.013 | 0.645 | 0.226 | I kappa B kinase epsilon inhibitor | 0.226 0.051 CHEMBL724 | CHEMBL724 | |
| 0.019 | 0.652 | 0.238 | Focal adhesion kinase 2 inhibitor | 0.238 0.044 CHEMBL724 | CHEMBL724 | |
| 0.046 | 0.68 | 0.121 | Sphingosine 1-phosphate receptor 2 agonist | 0.121 0.054 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.641 | 0.081 | Cyclin E inhibitor | 0.081 0.032 CHEMBL724 | CHEMBL724 | |
| 0.002 | 0.642 | 0.023 | Alpha 2c adrenoreceptor agonist | 0.023 0.008 CHEMBL724 | CHEMBL724 | |
| 0.022 | 0.664 | 0.104 | CDK3/cyclin E inhibitor | 0.104 0.079 CHEMBL724 | CHEMBL724 | |
| 0.033 | 0.676 | 0.206 | RNA-directed DNA polymerase inhibitor | 0.206 0.091 CHEMBL724 0.176 0.141 CHEMBL3527516 0.166 0.16 CHEMBL3527230 | CHEMBL724 | |
| 0.01 | 0.661 | 0.103 | Protein-tyrosine kinase Lyn inhibitor | 0.103 0.1 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.656 | 0.146 | Cyclin-dependent kinase 2 inhibitor | 0.146 0.04 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.66 | 0.08 | CDK1/cyclin B1 inhibitor | 0.08 0.039 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.658 | 0.124 | Cyclin-dependent kinase 1 inhibitor | 0.124 0.053 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.664 | 0.145 | Plasminogen activator inhibitor | 0.145 0.007 CHEMBL3526894 0.114 0.012 CHEMBL3526734 | CHEMBL3526894 | |
| 0.024 | 0.681 | 0.164 | Phospholipase C inhibitor | 0.137 0.135 CHEMBL3526895 0.164 0.082 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.666 | 0.149 | CDC-like kinase 2 inhibitor | 0.149 0.093 CHEMBL724 | CHEMBL724 | |
| 0.025 | 0.686 | 0.103 | Adenylate kinase inhibitor | 0.103 0.062 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.668 | 0.166 | Glycogen synthase kinase-3 alpha inhibitor | 0.166 0.056 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.667 | 0.045 | Factor Xa inhibitor | 0.045 0.033 CHEMBL3526734 | CHEMBL3526734 | |
| 0.01 | 0.675 | 0.079 | Myeloperoxidase inhibitor | 0.079 0.069 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.678 | 0.157 | Protein kinase (CK1) gamma 3 inhibitor | 0.157 0.082 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.672 | 0.111 | CDK2/cyclin A inhibitor | 0.111 0.049 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.673 | 0.249 | Phosphodiesterase 4D inhibitor | 0.249 0.007 CHEMBL3527515 0.151 0.019 CHEMBL3526734 | CHEMBL3527515 | |
| 0.007 | 0.681 | 0.097 | CYP2A6 inhibitor | 0.097 0.037 CHEMBL724 | CHEMBL724 | |
| 0.042 | 0.718 | 0.344 | 5 Hydroxytryptamine release inhibitor | 0.344 0.12 CHEMBL3526895 0.329 0.134 CHEMBL724 | CHEMBL3526895 | |
| 0.01 | 0.688 | 0.292 | Death-associated protein kinase 3 inhibitor | 0.292 0.04 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.689 | 0.074 | I kappa B kinase inhibitor | 0.074 0.07 CHEMBL724 | CHEMBL724 | |
| 0.024 | 0.709 | 0.225 | Tumour necrosis factor antagonist | 0.225 0.04 CHEMBL724 | CHEMBL724 | |
| 0.021 | 0.707 | 0.51 | Antibacterial | 0.306 0.131 CHEMBL3526895 0.51 0.038 CHEMBL3526644 | CHEMBL3526644 | |
| 0.004 | 0.69 | 0.088 | Cyclin-dependent kinase 5 inhibitor | 0.088 0.086 CHEMBL724 | CHEMBL724 | |
| 0.014 | 0.7 | 0.11 | Nav1.2 sodium channel blocker | 0.11 0.096 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.689 | 0.024 | Kainate receptor 5 antagonist | 0.024 0.012 CHEMBL3526895 | CHEMBL3526895 | |
| 0.008 | 0.696 | 0.1 | Protein kinase (CK1) gamma 2 inhibitor | 0.1 0.084 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.703 | 0.114 | MAP kinase kinase inhibitor | 0.114 0.08 CHEMBL724 | CHEMBL724 | |
| 0.013 | 0.714 | 0.141 | Antibacterial (Helicobacter pylori) | 0.141 0.055 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.719 | 0.143 | Cytokine production inhibitor | 0.143 0.068 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.707 | 0.261 | Selectin antagonist | 0.202 0.011 CHEMBL3527573 0.169 0.015 CHEMBL3526733 0.078 0.037 CHEMBL3527230 0.261 0.008 CHEMBL3526644 0.097 0.029 CHEMBL3527572 | CHEMBL3526644 | |
| 0.004 | 0.71 | 0.05 | Beta 1 adrenoreceptor antagonist | 0.05 0.047 CHEMBL724 | CHEMBL724 | |
| 0.018 | 0.725 | 0.076 | Kallikrein 1 inhibitor | 0.076 0.02 CHEMBL3526894 0.067 0.026 CHEMBL3526734 | CHEMBL3526894 | |
| 0.002 | 0.709 | 0.037 | Methionyl aminopeptidase 1 inhibitor | 0.037 0.015 CHEMBL724 | CHEMBL724 | |
| 0.016 | 0.727 | 0.306 | Cyclic AMP phosphodiesterase inhibitor | 0.306 0.039 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.729 | 0.096 | Lanosterol 14 alpha demethylase inhibitor | 0.096 0.062 CHEMBL724 | CHEMBL724 | |
| 0.026 | 0.739 | 0.089 | Interleukin 12 antagonist | 0.089 0.075 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.728 | 0.104 | MAP kinase kinase 1 inhibitor | 0.104 0.052 CHEMBL724 | CHEMBL724 | |
| 0.011 | 0.735 | 0.068 | Telomerase inhibitor | 0.068 0.054 CHEMBL724 | CHEMBL724 | |
| 0.004 | 0.729 | 0.073 | AMPA 2 receptor antagonist | 0.073 0.008 CHEMBL3526895 | CHEMBL3526895 | |
| 0.008 | 0.737 | 0.198 | Protein kinase C nu inhibitor | 0.198 0.048 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.75 | 0.142 | ATPase inhibitor | 0.142 0.116 CHEMBL724 | CHEMBL724 | |
| 0.007 | 0.741 | 0.126 | Lipid peroxidase inhibitor | 0.126 0.088 CHEMBL3526644 | CHEMBL3526644 | |
| 0.019 | 0.755 | 0.137 | 3C-like protease (Human coronavirus) inhibitor | 0.137 0.125 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.739 | 0.074 | Antineoplastic antibiotic | 0.071 0.064 CHEMBL3527573 0.074 0.062 CHEMBL3526644 | CHEMBL3526644 | |
| 0.008 | 0.744 | 0.072 | Cyclin B3 inhibitor | 0.072 0.044 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.748 | 0.115 | Multidrug resistance-associated protein 1 inhibitor | 0.115 0.055 CHEMBL3527572 | CHEMBL3527572 | |
| 0.004 | 0.747 | 0.135 | Cytidine deaminase inhibitor | 0.135 0.087 CHEMBL724 | CHEMBL724 | |
| 0.008 | 0.757 | 0.058 | Phosphodiesterase 1C inhibitor | 0.058 0.054 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.768 | 0.101 | Toll-Like receptor 4 antagonist | 0.101 0.068 CHEMBL3527573 0.1 0.07 CHEMBL3526733 0.1 0.069 CHEMBL3526644 | CHEMBL3527573 | |
| 0.005 | 0.758 | 0.078 | Protein kinase A inhibitor | 0.078 0.062 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.763 | 0.178 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.178 0.096 CHEMBL724 | CHEMBL724 | |
| 0.01 | 0.77 | 0.143 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.143 0.094 CHEMBL724 | CHEMBL724 | |
| 0.012 | 0.774 | 0.164 | Aldehyde oxidase inhibitor | 0.164 0.127 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.771 | 0.211 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.211 0.069 CHEMBL724 | CHEMBL724 | |
| 0.005 | 0.77 | 0.166 | CDC-like kinase 4 inhibitor | 0.166 0.089 CHEMBL724 | CHEMBL724 | |
| 0.059 | 0.825 | 0.301 | Peptidyltransferase inhibitor | 0.265 0.041 CHEMBL3527573 0.267 0.04 CHEMBL3526733 0.248 0.052 CHEMBL3527516 0.246 0.053 CHEMBL3527230 0.301 0.024 CHEMBL3526644 | CHEMBL3526644 | |
| 0.004 | 0.777 | 0.143 | Clk dual-specificity kinase inhibitor | 0.143 0.12 CHEMBL724 | CHEMBL724 | |
| 0.006 | 0.779 | 0.065 | Protein 50S ribosomal subunit inhibitor | 0.055 0.035 CHEMBL3527573 0.055 0.035 CHEMBL3526733 0.049 0.042 CHEMBL3527516 0.048 0.042 CHEMBL3527230 0.065 0.027 CHEMBL3526644 | CHEMBL3526644 | |
| 0.009 | 0.783 | 0.145 | Platelet aggregation inhibitor | 0.145 0.135 CHEMBL3526734 | CHEMBL3526734 | |
| 0.005 | 0.78 | 0.094 | Gastric antisecretory | 0.094 0.073 CHEMBL724 | CHEMBL724 | |
| 0.017 | 0.795 | 0.265 | Immunosuppressant | 0.218 0.178 CHEMBL3527573 0.252 0.146 CHEMBL3526733 0.265 0.137 CHEMBL3526644 | CHEMBL3526644 | |
| 0.002 | 0.78 | 0.03 | Purinergic P2X agonist | 0.029 0.018 CHEMBL3527516 0.03 0.017 CHEMBL3527230 | CHEMBL3527230 | |
| 0.012 | 0.793 | 0.18 | Cardiotonic | 0.18 0.14 CHEMBL3526734 | CHEMBL3526734 | |
| 0.005 | 0.799 | 0.117 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.117 0.111 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.8 | 0.098 | Cholecystokinin A antagonist | 0.098 0.009 CHEMBL3527572 | CHEMBL3527572 | |
| 0.007 | 0.805 | 0.092 | Beta glucuronidase inhibitor | 0.092 0.085 CHEMBL724 | CHEMBL724 | |
| 0.003 | 0.837 | 0.017 | Adenosine A2b receptor agonist | 0.017 0.008 CHEMBL3527516 0.017 0.008 CHEMBL3527230 | CHEMBL3527230 | |
| 0.025 | 0.862 | 0.132 | NOS3 expression enhancer | 0.132 0.094 CHEMBL3526644 | CHEMBL3526644 | |
| 0.003 | 0.841 | 0.061 | Cholecystokinin antagonist | 0.061 0.018 CHEMBL3527572 | CHEMBL3527572 | |
| 0.003 | 0.852 | 0.059 | Trypsin II inhibitor | 0.039 0.014 CHEMBL3526894 0.059 0.008 CHEMBL3526734 | CHEMBL3526734 | |
| 0.002 | 0.869 | 0.039 | Cholecystokinin B antagonist | 0.039 0.015 CHEMBL3527572 | CHEMBL3527572 | |
| 0.004 | 0.878 | 0.088 | Urokinase inhibitor | 0.088 0.019 CHEMBL3526894 0.063 0.027 CHEMBL3526734 | CHEMBL3526894 | |
| 0.004 | 0.878 | 0.096 | Factor VIIa inhibitor | 0.096 0.012 CHEMBL3526894 0.078 0.014 CHEMBL3526734 | CHEMBL3526894 | |
| 0.008 | 0.888 | 0.394 | Angiogenesis stimulant | 0.35 0.033 CHEMBL3527573 0.348 0.033 CHEMBL3526733 0.394 0.023 CHEMBL3526644 0.208 0.09 CHEMBL3527572 | CHEMBL3526644 | |
| 0.007 | 0.892 | 0.129 | Interleukin 1 antagonist | 0.129 0.076 CHEMBL724 | CHEMBL724 | |
| 0.009 | 0.895 | 0.263 | Apoptosis agonist | 0.253 0.211 CHEMBL3527573 0.263 0.201 CHEMBL3526733 0.252 0.212 CHEMBL3526644 | CHEMBL3526733 | |
| 0.005 | 0.894 | 0.194 | Chelator | 0.194 0.026 CHEMBL3526729 0.122 0.051 CHEMBL3527573 0.122 0.051 CHEMBL3526569 0.132 0.044 CHEMBL3527515 0.12 0.054 CHEMBL3527230 | CHEMBL3526729 | |
| 0.003 | 0.897 | 0.073 | Neuraminidase inhibitor | 0.073 0.031 CHEMBL3526895 | CHEMBL3526895 | |
| 0.003 | 0.911 | 0.02 | Adenosine A3 receptor agonist | 0.02 0.009 CHEMBL3527516 0.019 0.009 CHEMBL3527230 | CHEMBL3527516 | |
| 0.001 | 0.926 | 0.014 | Purinergic receptor agonist | 0.014 0.011 CHEMBL3527516 0.014 0.011 CHEMBL3527230 | CHEMBL3527230 | |
| 0.001 | 0.926 | 0.014 | Purinergic P2 agonist | 0.014 0.011 CHEMBL3527516 0.014 0.011 CHEMBL3527230 | CHEMBL3527230 | |
| 0.005 | 0.934 | 0.181 | Nitric oxide antagonist | 0.181 0.076 CHEMBL3527573 0.176 0.079 CHEMBL3526733 0.176 0.078 CHEMBL3526644 | CHEMBL3527573 | |
| 0.011 | 0.941 | 0.169 | DNA polymerase I inhibitor | 0.164 0.042 CHEMBL3527516 0.169 0.04 CHEMBL3527230 | CHEMBL3527230 | |
| 0.004 | 0.953 | 0.225 | Free radical scavenger | 0.194 0.103 CHEMBL3527573 0.184 0.111 CHEMBL3526733 0.225 0.08 CHEMBL3526644 | CHEMBL3526644 | |
| 0.004 | 0.955 | 0.107 | Topoisomerase I inhibitor | 0.105 0.066 CHEMBL3527516 0.107 0.065 CHEMBL3527230 | CHEMBL3527230 | |
| 0.004 | 0.976 | 0.33 | Antioxidant | 0.33 0.052 CHEMBL3527573 0.209 0.108 CHEMBL3526733 0.18 0.132 CHEMBL3527230 0.269 0.074 CHEMBL3526644 | CHEMBL3527573 | |
| 0.004 | 0.984 | 0.088 | Aminoacyl-tRNA synthetase inhibitor | 0.088 0.062 CHEMBL3527516 0.085 0.068 CHEMBL3527230 | CHEMBL3527516 | |
| 0.002 | 0.99 | 0.04 | Adenosine A1 receptor agonist | 0.04 0.008 CHEMBL3527516 0.039 0.008 CHEMBL3527230 | CHEMBL3527516 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |