| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.843 | 0.003 | 0.885 | Platelet growth factor antagonist | 0.724 0.003 CHEMBL3542323 0.801 0.003 CHEMBL3542333 0.607 0.003 CHEMBL3542273 0.885 0.002 CHEMBL3542196 0.842 0.003 CHEMBL3542344 0.728 0.003 CHEMBL3542232 0.229 0.006 CHEMBL3542401 0.832 0.003 CHEMBL3542399 | CHEMBL3542196 | |
| 0.829 | 0.004 | 0.836 | Vascular endothelial growth factor antagonist | 0.708 0.005 CHEMBL3542323 0.829 0.004 CHEMBL3542333 0.54 0.007 CHEMBL3542273 0.621 0.005 CHEMBL3542196 0.836 0.004 CHEMBL3542344 0.689 0.005 CHEMBL3542232 0.116 0.071 CHEMBL3542401 0.768 0.004 CHEMBL3542399 | CHEMBL3542344 | |
| 0.811 | 0.005 | 0.834 | Angiogenesis inhibitor | 0.746 0.007 CHEMBL3542323 0.834 0.005 CHEMBL3542333 0.629 0.014 CHEMBL3542273 0.618 0.015 CHEMBL3542196 0.834 0.005 CHEMBL3542344 0.761 0.006 CHEMBL3542232 0.282 0.102 CHEMBL3542401 0.801 0.005 CHEMBL3542399 | CHEMBL3542344 | |
| 0.805 | 0.003 | 0.805 | Platelet activating factor beta antagonist | 0.704 0.004 CHEMBL3542323 0.782 0.003 CHEMBL3542333 0.594 0.004 CHEMBL3542273 0.79 0.003 CHEMBL3542196 0.795 0.003 CHEMBL3542344 0.702 0.004 CHEMBL3542232 0.199 0.025 CHEMBL3542401 0.777 0.003 CHEMBL3542399 | ||
| 0.801 | 0.004 | 0.801 | Platelet aggregation inhibitor | 0.737 0.004 CHEMBL3542323 0.792 0.004 CHEMBL3542333 0.577 0.005 CHEMBL3542273 0.749 0.004 CHEMBL3542196 0.796 0.004 CHEMBL3542344 0.795 0.004 CHEMBL3542232 0.381 0.021 CHEMBL3542401 0.799 0.004 CHEMBL3542399 | ||
| 0.782 | 0.004 | 0.788 | Vascular endothelial growth factor 2 antagonist | 0.659 0.005 CHEMBL3542323 0.776 0.004 CHEMBL3542333 0.482 0.009 CHEMBL3542273 0.556 0.006 CHEMBL3542196 0.788 0.004 CHEMBL3542344 0.623 0.005 CHEMBL3542232 0.088 0.08 CHEMBL3542401 0.715 0.005 CHEMBL3542399 | CHEMBL3542344 | |
| 0.743 | 0.004 | 0.743 | Platelet activating factor antagonist | 0.615 0.004 CHEMBL3542323 0.694 0.004 CHEMBL3542333 0.467 0.005 CHEMBL3542273 0.687 0.004 CHEMBL3542196 0.728 0.004 CHEMBL3542344 0.599 0.004 CHEMBL3542232 0.206 0.025 CHEMBL3542401 0.718 0.004 CHEMBL3542399 | ||
| 0.644 | 0.003 | 0.662 | MAP kinase kinase 2 inhibitor | 0.662 0.002 CHEMBL3542323 0.646 0.003 CHEMBL3542333 0.414 0.01 CHEMBL3542273 0.441 0.008 CHEMBL3542196 0.616 0.003 CHEMBL3542344 0.474 0.005 CHEMBL3542232 0.276 0.043 CHEMBL3542401 0.599 0.003 CHEMBL3542399 | CHEMBL3542323 | |
| 0.585 | 0.005 | 0.818 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.429 0.009 CHEMBL3542323 0.539 0.005 CHEMBL3542333 0.2 0.037 CHEMBL3542273 0.818 0.004 CHEMBL3542196 0.533 0.005 CHEMBL3542344 0.277 0.022 CHEMBL3542232 0.463 0.007 CHEMBL3542399 | CHEMBL3542196 | |
| 0.561 | 0.004 | 0.565 | Fibroblast growth factor 1 antagonist | 0.456 0.004 CHEMBL3542323 0.565 0.004 CHEMBL3542333 0.347 0.005 CHEMBL3542273 0.559 0.004 CHEMBL3542196 0.559 0.004 CHEMBL3542344 0.386 0.005 CHEMBL3542232 0.117 0.045 CHEMBL3542401 0.535 0.004 CHEMBL3542399 | CHEMBL3542333 | |
| 0.55 | 0.004 | 0.55 | Proto-oncogene tyrosine-protein kinase Kit inhibitor | 0.434 0.005 CHEMBL3542323 0.513 0.005 CHEMBL3542333 0.294 0.012 CHEMBL3542273 0.414 0.006 CHEMBL3542196 0.531 0.004 CHEMBL3542344 0.404 0.006 CHEMBL3542232 0.132 0.039 CHEMBL3542401 0.497 0.005 CHEMBL3542399 | ||
| 0.553 | 0.012 | 0.587 | Calcium channel L-type activator | 0.536 0.016 CHEMBL3542323 0.572 0.009 CHEMBL3542333 0.54 0.015 CHEMBL3542273 0.545 0.014 CHEMBL3542196 0.565 0.01 CHEMBL3542344 0.574 0.009 CHEMBL3542232 0.554 0.012 CHEMBL3542401 0.587 0.007 CHEMBL3542399 | CHEMBL3542399 | |
| 0.534 | 0.003 | 0.554 | Death-associated protein kinase 2 inhibitor | 0.475 0.003 CHEMBL3542323 0.554 0.002 CHEMBL3542333 0.451 0.003 CHEMBL3542273 0.492 0.003 CHEMBL3542196 0.519 0.003 CHEMBL3542344 0.476 0.003 CHEMBL3542232 0.383 0.004 CHEMBL3542401 0.529 0.003 CHEMBL3542399 | CHEMBL3542333 | |
| 0.535 | 0.004 | 0.582 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.486 0.005 CHEMBL3542323 0.582 0.004 CHEMBL3542333 0.438 0.008 CHEMBL3542273 0.457 0.006 CHEMBL3542196 0.512 0.004 CHEMBL3542344 0.46 0.006 CHEMBL3542232 0.34 0.028 CHEMBL3542401 0.512 0.004 CHEMBL3542399 | CHEMBL3542333 | |
| 0.525 | 0.005 | 0.532 | Vascular endothelial growth factor 3 antagonist | 0.419 0.009 CHEMBL3542323 0.532 0.005 CHEMBL3542333 0.3 0.018 CHEMBL3542273 0.359 0.013 CHEMBL3542196 0.518 0.005 CHEMBL3542344 0.392 0.01 CHEMBL3542232 0.123 0.092 CHEMBL3542401 0.468 0.006 CHEMBL3542399 | CHEMBL3542333 | |
| 0.524 | 0.004 | 0.524 | Platelet activating factor alpha antagonist | 0.462 0.004 CHEMBL3542323 0.503 0.004 CHEMBL3542333 0.339 0.005 CHEMBL3542273 0.415 0.005 CHEMBL3542196 0.514 0.004 CHEMBL3542344 0.398 0.005 CHEMBL3542232 0.196 0.017 CHEMBL3542401 0.517 0.004 CHEMBL3542399 | ||
| 0.523 | 0.005 | 0.548 | TRKC antagonist | 0.396 0.011 CHEMBL3542323 0.548 0.005 CHEMBL3542333 0.316 0.022 CHEMBL3542273 0.361 0.015 CHEMBL3542196 0.511 0.005 CHEMBL3542344 0.431 0.009 CHEMBL3542232 0.146 0.105 CHEMBL3542401 0.373 0.013 CHEMBL3542399 | CHEMBL3542333 | |
| 0.522 | 0.005 | 0.533 | RET inhibitor | 0.392 0.01 CHEMBL3542323 0.533 0.005 CHEMBL3542333 0.295 0.023 CHEMBL3542273 0.34 0.016 CHEMBL3542196 0.516 0.005 CHEMBL3542344 0.354 0.014 CHEMBL3542232 0.487 0.006 CHEMBL3542399 | CHEMBL3542333 | |
| 0.495 | 0.008 | 0.512 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.465 0.011 CHEMBL3542323 0.512 0.006 CHEMBL3542333 0.386 0.025 CHEMBL3542273 0.389 0.024 CHEMBL3542196 0.478 0.009 CHEMBL3542344 0.405 0.02 CHEMBL3542232 0.303 0.062 CHEMBL3542401 0.495 0.008 CHEMBL3542399 | CHEMBL3542333 | |
| 0.477 | 0.003 | 0.477 | Focal adhesion kinase 2 inhibitor | 0.38 0.005 CHEMBL3542323 0.417 0.004 CHEMBL3542333 0.241 0.042 CHEMBL3542273 0.309 0.013 CHEMBL3542196 0.393 0.004 CHEMBL3542344 0.323 0.01 CHEMBL3542232 0.175 0.094 CHEMBL3542401 0.441 0.004 CHEMBL3542399 | ||
| 0.477 | 0.007 | 0.508 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.444 0.01 CHEMBL3542323 0.508 0.005 CHEMBL3542333 0.355 0.025 CHEMBL3542273 0.377 0.021 CHEMBL3542196 0.461 0.009 CHEMBL3542344 0.401 0.017 CHEMBL3542232 0.137 0.098 CHEMBL3542401 0.467 0.008 CHEMBL3542399 | CHEMBL3542333 | |
| 0.472 | 0.009 | 0.508 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.435 0.012 CHEMBL3542323 0.508 0.006 CHEMBL3542333 0.331 0.028 CHEMBL3542273 0.35 0.023 CHEMBL3542196 0.463 0.009 CHEMBL3542344 0.37 0.019 CHEMBL3542232 0.18 0.094 CHEMBL3542401 0.459 0.01 CHEMBL3542399 | CHEMBL3542333 | |
| 0.454 | 0.01 | 0.523 | Death-associated protein kinase 3 inhibitor | 0.358 0.024 CHEMBL3542323 0.523 0.005 CHEMBL3542333 0.319 0.033 CHEMBL3542273 0.362 0.023 CHEMBL3542196 0.456 0.01 CHEMBL3542344 0.379 0.02 CHEMBL3542232 0.442 0.011 CHEMBL3542399 | CHEMBL3542333 | |
| 0.435 | 0.008 | 0.442 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.41 0.011 CHEMBL3542323 0.442 0.007 CHEMBL3542333 0.273 0.036 CHEMBL3542273 0.304 0.029 CHEMBL3542196 0.431 0.009 CHEMBL3542344 0.356 0.019 CHEMBL3542232 0.422 0.01 CHEMBL3542399 | CHEMBL3542333 | |
| 0.404 | 0.005 | 0.411 | Vascular endothelial growth factor 1 antagonist | 0.294 0.012 CHEMBL3542323 0.411 0.005 CHEMBL3542333 0.209 0.024 CHEMBL3542273 0.277 0.013 CHEMBL3542196 0.41 0.005 CHEMBL3542344 0.315 0.01 CHEMBL3542232 0.35 0.007 CHEMBL3542399 | CHEMBL3542333 | |
| 0.394 | 0.007 | 0.418 | Ca2+/calmodulin-dependent kinase II delta inhibitor | 0.34 0.012 CHEMBL3542323 0.418 0.005 CHEMBL3542333 0.167 0.057 CHEMBL3542273 0.237 0.035 CHEMBL3542196 0.341 0.011 CHEMBL3542344 0.218 0.041 CHEMBL3542232 0.135 0.074 CHEMBL3542401 0.381 0.008 CHEMBL3542399 | CHEMBL3542333 | |
| 0.372 | 0.023 | 0.451 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.322 0.037 CHEMBL3542323 0.451 0.012 CHEMBL3542333 0.161 0.103 CHEMBL3542196 0.316 0.038 CHEMBL3542344 0.168 0.097 CHEMBL3542232 0.373 0.022 CHEMBL3542399 | CHEMBL3542333 | |
| 0.356 | 0.01 | 0.375 | Proto-oncogene tyrosine-protein kinase Yes inhibitor | 0.309 0.016 CHEMBL3542323 0.362 0.01 CHEMBL3542333 0.226 0.035 CHEMBL3542273 0.319 0.014 CHEMBL3542196 0.364 0.01 CHEMBL3542344 0.306 0.016 CHEMBL3542232 0.375 0.009 CHEMBL3542399 | CHEMBL3542399 | |
| 0.352 | 0.01 | 0.38 | Protein kinase (CK1) gamma 3 inhibitor | 0.283 0.02 CHEMBL3542323 0.38 0.007 CHEMBL3542333 0.22 0.037 CHEMBL3542273 0.259 0.025 CHEMBL3542196 0.332 0.012 CHEMBL3542344 0.278 0.021 CHEMBL3542232 0.163 0.076 CHEMBL3542401 0.307 0.016 CHEMBL3542399 | CHEMBL3542333 | |
| 0.312 | 0.018 | 0.385 | LIM domain kinase 1 inhibitor | 0.288 0.024 CHEMBL3542323 0.385 0.008 CHEMBL3542333 0.129 0.122 CHEMBL3542273 0.161 0.088 CHEMBL3542196 0.3 0.021 CHEMBL3542344 0.179 0.074 CHEMBL3542232 0.28 0.026 CHEMBL3542399 | CHEMBL3542333 | |
| 0.301 | 0.015 | 0.301 | Growth factor agonist | 0.293 0.017 CHEMBL3542323 0.291 0.017 CHEMBL3542333 0.188 0.076 CHEMBL3542273 0.216 0.05 CHEMBL3542196 0.294 0.016 CHEMBL3542344 0.279 0.021 CHEMBL3542232 0.292 0.017 CHEMBL3542399 | ||
| 0.289 | 0.005 | 0.29 | Aurora-C kinase inhibitor | 0.278 0.006 CHEMBL3542323 0.29 0.005 CHEMBL3542333 0.233 0.012 CHEMBL3542273 0.254 0.009 CHEMBL3542196 0.289 0.005 CHEMBL3542344 0.257 0.009 CHEMBL3542232 0.158 0.042 CHEMBL3542401 0.273 0.007 CHEMBL3542399 | CHEMBL3542333 | |
| 0.281 | 0.014 | 0.33 | TRKA antagonist | 0.237 0.021 CHEMBL3542323 0.33 0.009 CHEMBL3542333 0.11 0.077 CHEMBL3542196 0.256 0.018 CHEMBL3542344 0.152 0.049 CHEMBL3542232 0.102 0.087 CHEMBL3542399 | CHEMBL3542333 | |
| 0.272 | 0.006 | 0.293 | Polo-like kinase-4 inhibitor | 0.223 0.011 CHEMBL3542323 0.293 0.005 CHEMBL3542333 0.185 0.019 CHEMBL3542273 0.217 0.012 CHEMBL3542196 0.265 0.006 CHEMBL3542344 0.234 0.01 CHEMBL3542232 0.269 0.006 CHEMBL3542399 | CHEMBL3542333 | |
| 0.279 | 0.014 | 0.3 | Protein kinase (CK1) gamma 2 inhibitor | 0.219 0.027 CHEMBL3542323 0.3 0.011 CHEMBL3542333 0.136 0.055 CHEMBL3542273 0.187 0.036 CHEMBL3542196 0.26 0.018 CHEMBL3542344 0.205 0.03 CHEMBL3542232 0.098 0.087 CHEMBL3542401 0.227 0.025 CHEMBL3542399 | CHEMBL3542333 | |
| 0.284 | 0.021 | 0.349 | Protein kinase (CK1) gamma inhibitor | 0.215 0.039 CHEMBL3542323 0.349 0.011 CHEMBL3542333 0.134 0.077 CHEMBL3542273 0.181 0.052 CHEMBL3542196 0.263 0.026 CHEMBL3542344 0.204 0.043 CHEMBL3542232 0.22 0.038 CHEMBL3542399 | CHEMBL3542333 | |
| 0.242 | 0.007 | 0.247 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.215 0.013 CHEMBL3542323 0.243 0.007 CHEMBL3542333 0.191 0.024 CHEMBL3542273 0.203 0.017 CHEMBL3542196 0.229 0.009 CHEMBL3542344 0.215 0.012 CHEMBL3542232 0.167 0.047 CHEMBL3542401 0.247 0.006 CHEMBL3542399 | CHEMBL3542399 | |
| 0.255 | 0.026 | 0.295 | Tyrosine-protein kinase receptor antagonist | 0.203 0.039 CHEMBL3542323 0.295 0.018 CHEMBL3542333 0.234 0.03 CHEMBL3542344 0.135 0.074 CHEMBL3542232 | CHEMBL3542333 | |
| 0.264 | 0.044 | 0.343 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.231 0.055 CHEMBL3542323 0.343 0.02 CHEMBL3542333 0.153 0.093 CHEMBL3542196 0.24 0.052 CHEMBL3542344 0.177 0.077 CHEMBL3542232 0.241 0.051 CHEMBL3542399 | CHEMBL3542333 | |
| 0.238 | 0.031 | 0.309 | Protein kinase (CK1) gamma 1 inhibitor | 0.167 0.057 CHEMBL3542323 0.309 0.018 CHEMBL3542333 0.139 0.079 CHEMBL3542196 0.193 0.045 CHEMBL3542344 0.14 0.078 CHEMBL3542232 0.186 0.048 CHEMBL3542399 | CHEMBL3542333 | |
| 0.242 | 0.036 | 0.242 | Growth factor antagonist | 0.186 0.051 CHEMBL3542323 0.22 0.041 CHEMBL3542333 0.228 0.039 CHEMBL3542196 0.228 0.039 CHEMBL3542344 0.132 0.082 CHEMBL3542232 0.183 0.052 CHEMBL3542399 | ||
| 0.218 | 0.021 | 0.218 | TRKB antagonist | 0.149 0.048 CHEMBL3542323 0.216 0.022 CHEMBL3542333 0.103 0.096 CHEMBL3542273 0.122 0.071 CHEMBL3542196 0.193 0.027 CHEMBL3542344 0.149 0.048 CHEMBL3542232 0.118 0.075 CHEMBL3542399 | ||
| 0.22 | 0.026 | 0.238 | Aurora-B kinase inhibitor | 0.189 0.034 CHEMBL3542323 0.238 0.023 CHEMBL3542333 0.189 0.034 CHEMBL3542344 0.158 0.043 CHEMBL3542399 | CHEMBL3542333 | |
| 0.217 | 0.031 | 0.27 | c-Src kinase inhibitor | 0.195 0.036 CHEMBL3542323 0.193 0.037 CHEMBL3542333 0.231 0.028 CHEMBL3542196 0.199 0.035 CHEMBL3542344 0.144 0.058 CHEMBL3542232 0.27 0.022 CHEMBL3542399 | CHEMBL3542399 | |
| 0.236 | 0.059 | 0.239 | ErbB-1 antagonist | 0.228 0.065 CHEMBL3542323 0.18 0.115 CHEMBL3542333 0.161 0.153 CHEMBL3542196 0.197 0.093 CHEMBL3542344 0.17 0.133 CHEMBL3542232 0.239 0.058 CHEMBL3542399 | CHEMBL3542399 | |
| 0.181 | 0.013 | 0.181 | Stem cell growth factor agonist | 0.138 0.023 CHEMBL3542323 0.156 0.018 CHEMBL3542333 0.114 0.035 CHEMBL3542196 0.157 0.017 CHEMBL3542344 0.106 0.04 CHEMBL3542232 0.134 0.024 CHEMBL3542399 | ||
| 0.219 | 0.062 | 0.225 | Tyrosine kinase inhibitor | 0.154 0.087 CHEMBL3542323 0.225 0.06 CHEMBL3542333 0.214 0.064 CHEMBL3542196 0.198 0.069 CHEMBL3542344 0.164 0.083 CHEMBL3542399 | CHEMBL3542333 | |
| 0.219 | 0.063 | 0.303 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.223 0.06 CHEMBL3542323 0.303 0.026 CHEMBL3542333 0.215 0.066 CHEMBL3542344 0.165 0.106 CHEMBL3542232 0.226 0.059 CHEMBL3542399 | CHEMBL3542333 | |
| 0.207 | 0.051 | 0.232 | Src kinase inhibitor | 0.193 0.058 CHEMBL3542323 0.197 0.055 CHEMBL3542333 0.187 0.061 CHEMBL3542196 0.19 0.059 CHEMBL3542344 0.131 0.098 CHEMBL3542232 0.232 0.041 CHEMBL3542399 | CHEMBL3542399 | |
| 0.161 | 0.011 | 0.163 | Fibroblast growth factor 3 antagonist | 0.154 0.013 CHEMBL3542323 0.163 0.011 CHEMBL3542333 0.158 0.012 CHEMBL3542344 0.124 0.022 CHEMBL3542399 | CHEMBL3542333 | |
| 0.19 | 0.051 | 0.344 | Protein kinase C nu inhibitor | 0.158 0.065 CHEMBL3542323 0.344 0.017 CHEMBL3542333 0.188 0.052 CHEMBL3542344 0.124 0.088 CHEMBL3542232 0.165 0.062 CHEMBL3542399 | CHEMBL3542333 | |
| 0.209 | 0.075 | 0.246 | Nitric-oxide synthase stimulant | 0.173 0.146 CHEMBL3542323 0.245 0.036 CHEMBL3542333 0.201 0.088 CHEMBL3542196 0.234 0.045 CHEMBL3542344 0.246 0.035 CHEMBL3542232 0.178 0.132 CHEMBL3542401 0.207 0.077 CHEMBL3542399 | CHEMBL3542232 | |
| 0.197 | 0.068 | 0.285 | CDC-like kinase 2 inhibitor | 0.176 0.079 CHEMBL3542323 0.285 0.035 CHEMBL3542333 0.193 0.07 CHEMBL3542344 0.122 0.116 CHEMBL3542232 0.153 0.091 CHEMBL3542399 | CHEMBL3542333 | |
| 0.144 | 0.021 | 0.144 | Interleukin 2 antagonist | 0.116 0.051 CHEMBL3542323 0.113 0.058 CHEMBL3542333 0.122 0.042 CHEMBL3542344 0.128 0.034 CHEMBL3542399 | ||
| 0.128 | 0.007 | 0.13 | Polo-like kinase-2 inhibitor | 0.118 0.011 CHEMBL3542323 0.126 0.008 CHEMBL3542333 0.104 0.022 CHEMBL3542273 0.109 0.018 CHEMBL3542196 0.13 0.006 CHEMBL3542344 0.115 0.013 CHEMBL3542232 0.115 0.013 CHEMBL3542399 | CHEMBL3542344 | |
| 0.216 | 0.105 | 0.362 | Cardiotonic | 0.263 0.074 CHEMBL3542323 0.362 0.036 CHEMBL3542401 0.23 0.096 CHEMBL3542399 | CHEMBL3542401 | |
| 0.156 | 0.055 | 0.218 | Cyclin-dependent kinase 7 inhibitor | 0.109 0.093 CHEMBL3542323 0.218 0.028 CHEMBL3542333 0.14 0.067 CHEMBL3542344 0.136 0.071 CHEMBL3542399 | CHEMBL3542333 | |
| 0.165 | 0.067 | 0.168 | Cyclin-dependent kinase 3 inhibitor | 0.155 0.085 CHEMBL3542323 0.146 0.107 CHEMBL3542333 0.137 0.132 CHEMBL3542196 0.16 0.075 CHEMBL3542344 0.147 0.103 CHEMBL3542232 0.145 0.108 CHEMBL3542401 0.168 0.063 CHEMBL3542399 | CHEMBL3542399 | |
| 0.142 | 0.052 | 0.149 | Death-associated protein kinase 1 inhibitor | 0.12 0.112 CHEMBL3542323 0.149 0.04 CHEMBL3542333 0.124 0.1 CHEMBL3542273 0.137 0.064 CHEMBL3542196 0.148 0.042 CHEMBL3542344 0.141 0.056 CHEMBL3542232 0.127 0.09 CHEMBL3542399 | CHEMBL3542333 | |
| 0.117 | 0.038 | 0.148 | MAP kinase kinase 1 inhibitor | 0.148 0.017 CHEMBL3542323 0.145 0.019 CHEMBL3542333 0.125 0.031 CHEMBL3542344 0.088 0.074 CHEMBL3542399 | CHEMBL3542323 | |
| 0.164 | 0.087 | 0.207 | Lipocortins synthesis antagonist | 0.207 0.052 CHEMBL3542323 0.16 0.092 CHEMBL3542401 0.173 0.078 CHEMBL3542399 | CHEMBL3542323 | |
| 0.18 | 0.102 | 0.223 | EphB2 antagonist | 0.223 0.073 CHEMBL3542333 0.202 0.086 CHEMBL3542344 0.204 0.085 CHEMBL3542232 0.173 0.109 CHEMBL3542399 | CHEMBL3542333 | |
| 0.135 | 0.059 | 0.153 | Epidermal growth factor receptor kinase inhibitor | 0.127 0.066 CHEMBL3542323 0.113 0.08 CHEMBL3542333 0.153 0.046 CHEMBL3542196 0.117 0.076 CHEMBL3542344 0.126 0.067 CHEMBL3542399 | CHEMBL3542196 | |
| 0.128 | 0.053 | 0.574 | DNA intercalator | 0.137 0.049 CHEMBL3542323 0.095 0.079 CHEMBL3542333 0.574 0.004 CHEMBL3542196 0.165 0.037 CHEMBL3542399 | CHEMBL3542196 | |
| 0.107 | 0.032 | 0.117 | MAP kinase 11 inhibitor | 0.109 0.03 CHEMBL3542333 0.117 0.027 CHEMBL3542344 | CHEMBL3542344 | |
| 0.135 | 0.062 | 0.183 | Protein kinase (CK1) delta inhibitor | 0.098 0.094 CHEMBL3542323 0.183 0.035 CHEMBL3542333 0.128 0.067 CHEMBL3542344 | CHEMBL3542333 | |
| 0.092 | 0.02 | 0.099 | Phospholipase D inhibitor | 0.099 0.015 CHEMBL3542323 0.07 0.054 CHEMBL3542333 0.073 0.046 CHEMBL3542344 0.09 0.022 CHEMBL3542232 0.092 0.02 CHEMBL3542401 | CHEMBL3542323 | |
| 0.168 | 0.099 | 0.238 | Clk dual-specificity kinase inhibitor | 0.134 0.13 CHEMBL3542323 0.238 0.06 CHEMBL3542333 0.158 0.107 CHEMBL3542344 0.158 0.107 CHEMBL3542399 | CHEMBL3542333 | |
| 0.114 | 0.047 | 0.125 | Insulin receptor antagonist | 0.098 0.064 CHEMBL3542323 0.125 0.039 CHEMBL3542333 0.093 0.072 CHEMBL3542344 | CHEMBL3542333 | |
| 0.147 | 0.087 | 0.279 | Sigma receptor agonist | 0.143 0.09 CHEMBL3542323 0.14 0.093 CHEMBL3542401 0.279 0.043 CHEMBL3542399 | CHEMBL3542399 | |
| 0.137 | 0.08 | 0.177 | CDC-like kinase 1 inhibitor | 0.111 0.105 CHEMBL3542323 0.177 0.05 CHEMBL3542333 0.143 0.076 CHEMBL3542344 0.109 0.108 CHEMBL3542232 0.161 0.062 CHEMBL3542399 | CHEMBL3542333 | |
| 0.135 | 0.079 | 0.208 | Protein kinase (CK1) inhibitor | 0.208 0.037 CHEMBL3542333 0.137 0.077 CHEMBL3542344 | CHEMBL3542333 | |
| 0.164 | 0.109 | 0.212 | Antimitotic | 0.147 0.124 CHEMBL3542323 0.212 0.077 CHEMBL3542333 0.204 0.081 CHEMBL3542196 0.153 0.118 CHEMBL3542344 0.183 0.094 CHEMBL3542399 | CHEMBL3542333 | |
| 0.133 | 0.078 | 0.142 | Ribosomal protein S6 kinase inhibitor | 0.11 0.102 CHEMBL3542323 0.142 0.071 CHEMBL3542333 0.112 0.1 CHEMBL3542344 0.125 0.085 CHEMBL3542399 | CHEMBL3542333 | |
| 0.095 | 0.045 | 0.095 | ALK inhibitor | 0.081 0.058 CHEMBL3542323 0.093 0.046 CHEMBL3542333 0.086 0.052 CHEMBL3542344 0.08 0.059 CHEMBL3542399 | ||
| 0.126 | 0.08 | 0.135 | Protein-tyrosine kinase Lyn inhibitor | 0.135 0.074 CHEMBL3542333 0.111 0.092 CHEMBL3542344 0.109 0.094 CHEMBL3542399 | CHEMBL3542333 | |
| 0.065 | 0.023 | 0.065 | Proto-oncogene tyrosine-protein kinase Met inhibitor | 0.044 0.037 CHEMBL3542323 0.061 0.025 CHEMBL3542333 0.056 0.028 CHEMBL3542344 | ||
| 0.089 | 0.05 | 0.089 | Leucine-rich repeat kinase 2 inhibitor | 0.075 0.062 CHEMBL3542333 0.077 0.061 CHEMBL3542344 | ||
| 0.078 | 0.039 | 0.118 | Check point kinase 1 inhibitor | 0.069 0.047 CHEMBL3542323 0.118 0.021 CHEMBL3542333 0.064 0.053 CHEMBL3542196 0.07 0.045 CHEMBL3542344 0.11 0.024 CHEMBL3542399 | CHEMBL3542333 | |
| 0.086 | 0.048 | 0.113 | Glycine receptor antagonist | 0.113 0.022 CHEMBL3542232 0.093 0.04 CHEMBL3542401 0.077 0.062 CHEMBL3542399 | CHEMBL3542232 | |
| 0.057 | 0.024 | 0.073 | Topoisomerase II beta inhibitor | 0.05 0.032 CHEMBL3542323 0.073 0.015 CHEMBL3542399 | CHEMBL3542399 | |
| 0.119 | 0.086 | 0.131 | Lck kinase inhibitor | 0.109 0.094 CHEMBL3542323 0.127 0.08 CHEMBL3542333 0.105 0.098 CHEMBL3542344 0.131 0.077 CHEMBL3542399 | CHEMBL3542399 | |
| 0.188 | 0.159 | 0.333 | Tyrosine 3 hydroxylase inhibitor | 0.191 0.153 CHEMBL3542401 0.333 0.02 CHEMBL3542399 | CHEMBL3542399 | |
| 0.09 | 0.063 | 0.094 | Hepatocyte growth factor antagonist | 0.094 0.059 CHEMBL3542333 0.093 0.059 CHEMBL3542344 | CHEMBL3542333 | |
| 0.077 | 0.053 | 0.125 | Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor | 0.069 0.061 CHEMBL3542323 0.125 0.025 CHEMBL3542333 0.07 0.06 CHEMBL3542344 0.103 0.034 CHEMBL3542399 | CHEMBL3542333 | |
| 0.087 | 0.064 | 0.103 | Pim-3 kinase inhibitor | 0.103 0.042 CHEMBL3542333 | CHEMBL3542333 | |
| 0.042 | 0.019 | 0.042 | Glucose-6-phosphate dehydrogenase inhibitor | 0.04 0.022 CHEMBL3542323 0.038 0.025 CHEMBL3542344 0.038 0.025 CHEMBL3542401 0.042 0.019 CHEMBL3542399 | ||
| 0.026 | 0.005 | 0.027 | Histone-lysine N-methyltransferase EZH2 inhibitor | 0.023 0.007 CHEMBL3542323 0.025 0.005 CHEMBL3542333 0.023 0.008 CHEMBL3542273 0.025 0.005 CHEMBL3542196 0.027 0.004 CHEMBL3542344 0.022 0.009 CHEMBL3542232 0.02 0.016 CHEMBL3542401 0.025 0.005 CHEMBL3542399 | CHEMBL3542344 | |
| 0.133 | 0.115 | 0.187 | CDC-like kinase 4 inhibitor | 0.187 0.074 CHEMBL3542333 | CHEMBL3542333 | |
| 0.167 | 0.152 | 0.231 | Peptidyltransferase inhibitor | 0.211 0.085 CHEMBL3542323 0.184 0.122 CHEMBL3542273 0.2 0.099 CHEMBL3542232 0.231 0.066 CHEMBL3542399 | CHEMBL3542399 | |
| 0.09 | 0.075 | 0.148 | Check point kinase 2 inhibitor | 0.148 0.032 CHEMBL3542333 0.084 0.079 CHEMBL3542344 0.092 0.073 CHEMBL3542399 | CHEMBL3542333 | |
| 0.098 | 0.084 | 0.122 | CDC-like kinase 3 inhibitor | 0.096 0.088 CHEMBL3542323 0.122 0.041 CHEMBL3542333 0.103 0.073 CHEMBL3542344 0.104 0.069 CHEMBL3542399 | CHEMBL3542333 | |
| 0.05 | 0.037 | 0.065 | Antiviral (Hepatitis D) | 0.053 0.032 CHEMBL3542323 0.049 0.038 CHEMBL3542344 0.049 0.04 CHEMBL3542232 0.065 0.017 CHEMBL3542401 | CHEMBL3542401 | |
| 0.269 | 0.257 | 0.303 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.303 0.208 CHEMBL3542333 0.292 0.224 CHEMBL3542344 | CHEMBL3542333 | |
| 0.041 | 0.046 | 0.057 | Mineralocorticoid receptor antagonist | 0.049 0.032 CHEMBL3542333 0.044 0.039 CHEMBL3542344 0.048 0.033 CHEMBL3542232 0.057 0.022 CHEMBL3542401 | CHEMBL3542401 | |
| 0.084 | 0.093 | 0.089 | Alpha 2b adrenoreceptor antagonist | 0.089 0.087 CHEMBL3542401 | CHEMBL3542401 | |
| 0.033 | 0.042 | 0.052 | Glutamate (mGluR1a) antagonist | 0.052 0.019 CHEMBL3542333 0.043 0.026 CHEMBL3542344 | CHEMBL3542333 | |
| 0.108 | 0.119 | 0.123 | Papain-like protease (SARS coronavirus) inhibitor | 0.113 0.102 CHEMBL3542333 0.111 0.109 CHEMBL3542344 0.123 0.075 CHEMBL3542399 | CHEMBL3542399 | |
| 0.075 | 0.089 | 0.106 | Pim-1 kinase inhibitor | 0.106 0.052 CHEMBL3542333 | CHEMBL3542333 | |
| 0.091 | 0.106 | 0.156 | MAP kinase kinase inhibitor | 0.141 0.056 CHEMBL3542323 0.156 0.048 CHEMBL3542333 0.118 0.076 CHEMBL3542344 | CHEMBL3542333 | |
| 0.222 | 0.247 | 0.365 | Apoptosis agonist | 0.365 0.131 CHEMBL3542399 | CHEMBL3542399 | |
| 0.126 | 0.151 | 0.14 | I kappa B kinase epsilon inhibitor | 0.14 0.131 CHEMBL3542399 | CHEMBL3542399 | |
| 0.023 | 0.054 | 0.087 | Kinesin-like protein 1 inhibitor | 0.061 0.014 CHEMBL3542333 0.087 0.009 CHEMBL3542196 | CHEMBL3542196 | |
| 0.023 | 0.054 | 0.087 | Kinesin antagonist | 0.061 0.014 CHEMBL3542333 0.087 0.009 CHEMBL3542196 | CHEMBL3542196 | |
| 0.013 | 0.044 | 0.022 | Progesterone receptor B antagonist | 0.022 0.01 CHEMBL3542401 | CHEMBL3542401 | |
| 0.079 | 0.111 | 0.149 | Chelator | 0.098 0.08 CHEMBL3542323 0.149 0.036 CHEMBL3542399 | CHEMBL3542399 | |
| 0.046 | 0.08 | 0.112 | DNA gyrase inhibitor | 0.064 0.043 CHEMBL3542273 0.112 0.015 CHEMBL3542344 | CHEMBL3542344 | |
| 0.05 | 0.085 | 0.067 | CDK2/cyclin E2 inhibitor | 0.067 0.053 CHEMBL3542333 | CHEMBL3542333 | |
| 0.095 | 0.13 | 0.163 | Histone deacetylase SIRT1 inhibitor | 0.163 0.051 CHEMBL3542333 0.121 0.089 CHEMBL3542344 0.121 0.09 CHEMBL3542232 0.119 0.093 CHEMBL3542399 | CHEMBL3542333 | |
| 0.127 | 0.164 | 0.311 | Dyrk kinase inhibitor | 0.214 0.09 CHEMBL3542333 0.311 0.049 CHEMBL3542273 0.203 0.097 CHEMBL3542399 | CHEMBL3542273 | |
| 0.064 | 0.101 | 0.108 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.108 0.032 CHEMBL3542333 0.08 0.065 CHEMBL3542232 0.097 0.042 CHEMBL3542399 | CHEMBL3542333 | |
| 0.143 | 0.181 | 0.158 | MAP kinase kinase 5 inhibitor | 0.158 0.121 CHEMBL3542323 0.155 0.134 CHEMBL3542333 | CHEMBL3542323 | |
| 0.071 | 0.114 | 0.095 | Granulocyte macrophage colony stimulating factor antagonist | 0.095 0.078 CHEMBL3542333 | CHEMBL3542333 | |
| 0.049 | 0.099 | 0.075 | Protein kinase B beta inhibitor | 0.075 0.048 CHEMBL3542333 | CHEMBL3542333 | |
| 0.062 | 0.111 | 0.084 | CDK2/cyclin A inhibitor | 0.084 0.074 CHEMBL3542273 | CHEMBL3542273 | |
| 0.022 | 0.074 | 0.03 | DNA topoisomerase IV inhibitor | 0.03 0.019 CHEMBL3542344 | CHEMBL3542344 | |
| 0.131 | 0.191 | 0.3 | Cyclic AMP phosphodiesterase inhibitor | 0.166 0.127 CHEMBL3542323 0.3 0.042 CHEMBL3542399 | CHEMBL3542399 | |
| 0.084 | 0.145 | 0.117 | NADPH oxidase inhibitor | 0.117 0.087 CHEMBL3542399 | CHEMBL3542399 | |
| 0.066 | 0.134 | 0.09 | Cyclin-dependent kinase 2 inhibitor | 0.09 0.082 CHEMBL3542333 | CHEMBL3542333 | |
| 0.137 | 0.21 | 0.17 | MAP-kinase-activated kinase 5 inhibitor | 0.17 0.147 CHEMBL3542399 | CHEMBL3542399 | |
| 0.063 | 0.137 | 0.103 | Topoisomerase II inhibitor | 0.103 0.083 CHEMBL3542399 | CHEMBL3542399 | |
| 0.076 | 0.153 | 0.126 | TRPA1 agonist | 0.126 0.052 CHEMBL3542399 | CHEMBL3542399 | |
| 0.008 | 0.09 | 0.034 | NMDA receptor glycine site antagonist | 0.034 0.01 CHEMBL3542232 | CHEMBL3542232 | |
| 0.042 | 0.126 | 0.143 | Gonadotropin-releasing hormone receptor agonist | 0.143 0.005 CHEMBL3542196 | CHEMBL3542196 | |
| 0.047 | 0.132 | 0.079 | Myeloperoxidase inhibitor | 0.079 0.069 CHEMBL3542333 | CHEMBL3542333 | |
| 0.053 | 0.152 | 0.083 | Glutathione S-transferase inhibitor | 0.083 0.057 CHEMBL3542232 | CHEMBL3542232 | |
| 0.104 | 0.211 | 0.212 | Immunostimulant | 0.168 0.14 CHEMBL3542323 0.174 0.136 CHEMBL3542232 0.212 0.113 CHEMBL3542399 | CHEMBL3542399 | |
| 0.039 | 0.168 | 0.084 | I kappa B kinase 1 inhibitor | 0.084 0.033 CHEMBL3542333 | CHEMBL3542333 | |
| 0.031 | 0.163 | 0.067 | Beta adrenoreceptor antagonist | 0.067 0.042 CHEMBL3542399 | CHEMBL3542399 | |
| 0.016 | 0.159 | 0.048 | Thymidylate synthase inhibitor | 0.048 0.031 CHEMBL3542232 | CHEMBL3542232 | |
| 0.101 | 0.245 | 0.184 | Vasodilator | 0.163 0.139 CHEMBL3542323 0.184 0.118 CHEMBL3542399 | CHEMBL3542399 | |
| 0.015 | 0.163 | 0.037 | Somatostatin 5 agonist | 0.037 0.021 CHEMBL3542333 | CHEMBL3542333 | |
| 0.021 | 0.17 | 0.06 | Biliverdin reductase inhibitor | 0.06 0.041 CHEMBL3542232 | CHEMBL3542232 | |
| 0.054 | 0.204 | 0.175 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.175 0.062 CHEMBL3542333 | CHEMBL3542333 | |
| 0.104 | 0.272 | 0.158 | Neurotensin receptor agonist | 0.147 0.109 CHEMBL3542333 0.138 0.135 CHEMBL3542344 0.158 0.083 CHEMBL3542232 0.153 0.094 CHEMBL3542399 | CHEMBL3542232 | |
| 0.178 | 0.348 | 0.316 | 5 Hydroxytryptamine release inhibitor | 0.316 0.147 CHEMBL3542399 | CHEMBL3542399 | |
| 0.045 | 0.217 | 0.106 | 5 Hydroxytryptamine 3A agonist | 0.106 0.069 CHEMBL3542333 | CHEMBL3542333 | |
| 0.07 | 0.246 | 0.258 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.258 0.064 CHEMBL3542273 | CHEMBL3542273 | |
| 0.136 | 0.318 | 0.303 | GABA C receptor rho-3 antagonist | 0.303 0.114 CHEMBL3542399 | CHEMBL3542399 | |
| 0.008 | 0.204 | 0.049 | Secretase gamma inhibitor | 0.049 0.026 CHEMBL3542273 | CHEMBL3542273 | |
| 0.028 | 0.234 | 0.075 | Protein kinase B alpha inhibitor | 0.075 0.044 CHEMBL3542401 | CHEMBL3542401 | |
| 0.038 | 0.246 | 0.1 | Ferrochelatase inhibitor | 0.1 0.071 CHEMBL3542232 | CHEMBL3542232 | |
| 0.007 | 0.22 | 0.113 | Protocollagen prolyl hydroxylase inhibitor | 0.113 0.004 CHEMBL3542232 | CHEMBL3542232 | |
| 0.033 | 0.252 | 0.082 | Protein kinase C delta inhibitor | 0.082 0.073 CHEMBL3542333 | CHEMBL3542333 | |
| 0.103 | 0.348 | 0.199 | Vasodilator, peripheral | 0.199 0.177 CHEMBL3542399 | CHEMBL3542399 | |
| 0.039 | 0.295 | 0.147 | Lipid peroxidase inhibitor | 0.147 0.07 CHEMBL3542399 | CHEMBL3542399 | |
| 0.107 | 0.366 | 0.193 | Insulysin inhibitor | 0.193 0.167 CHEMBL3542399 | CHEMBL3542399 | |
| 0.021 | 0.292 | 0.105 | Cyclin-dependent kinase 5 inhibitor | 0.105 0.071 CHEMBL3542273 | CHEMBL3542273 | |
| 0.027 | 0.305 | 0.075 | Somatostatin 1 agonist | 0.075 0.057 CHEMBL3542333 | CHEMBL3542333 | |
| 0.045 | 0.359 | 0.081 | Estrogen-related receptor beta agonist | 0.081 0.065 CHEMBL3542399 | CHEMBL3542399 | |
| 0.022 | 0.383 | 0.064 | Ca(v)3.2 blocker | 0.064 0.03 CHEMBL3542401 | CHEMBL3542401 | |
| 0.044 | 0.407 | 0.193 | Free radical scavenger | 0.193 0.104 CHEMBL3542399 | CHEMBL3542399 | |
| 0.026 | 0.408 | 0.129 | Thrombolytic | 0.129 0.1 CHEMBL3542232 | CHEMBL3542232 | |
| 0.041 | 0.432 | 0.259 | Aldehyde oxidase inhibitor | 0.259 0.079 CHEMBL3542399 | CHEMBL3542399 | |
| 0.042 | 0.456 | 0.177 | Antioxidant | 0.177 0.135 CHEMBL3542399 | CHEMBL3542399 | |
| 0.006 | 0.481 | 0.511 | Opioid mu receptor antagonist | 0.511 0.004 CHEMBL3542273 | CHEMBL3542273 | |
| 0.017 | 0.494 | 0.47 | Opioid antagonist | 0.47 0.004 CHEMBL3542273 | CHEMBL3542273 | |
| 0.034 | 0.54 | 0.085 | 3C-Like protease (SARS coronavirus) inhibitor | 0.085 0.056 CHEMBL3542401 | CHEMBL3542401 | |
| 0.024 | 0.905 | 0.347 | Sodium/bile acid cotransporter inhibitor | 0.347 0.042 CHEMBL3542232 | CHEMBL3542232 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |