| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.894 | 0.003 | 0.894 | ErbB-2 antagonist | 0.859 0.003 CHEMBL3526326 0.627 0.004 CHEMBL3526763 0.731 0.003 CHEMBL3526479 0.686 0.004 CHEMBL3527095 0.706 0.004 CHEMBL3526380 0.662 0.004 CHEMBL3542267 0.59 0.004 CHEMBL3706535 0.6 0.004 CHEMBL3526480 0.749 0.003 CHEMBL3526764 0.669 0.004 CHEMBL3542268 | ||
| 0.787 | 0.003 | 0.81 | ErbB-1 antagonist | 0.81 0.003 CHEMBL3526326 0.666 0.004 CHEMBL3526763 0.696 0.004 CHEMBL3526479 0.651 0.004 CHEMBL3527095 0.728 0.003 CHEMBL3526380 0.73 0.003 CHEMBL3542267 0.65 0.004 CHEMBL3706535 0.61 0.004 CHEMBL3526480 0.688 0.004 CHEMBL3526764 0.658 0.004 CHEMBL3542268 | CHEMBL3526326 | |
| 0.68 | 0.002 | 0.68 | EphB4 antagonist | 0.52 0.002 CHEMBL3526326 0.493 0.003 CHEMBL3526763 0.335 0.004 CHEMBL3526479 0.601 0.002 CHEMBL3527095 0.292 0.004 CHEMBL3526380 0.195 0.007 CHEMBL3542267 0.391 0.003 CHEMBL3706535 0.293 0.004 CHEMBL3526480 0.272 0.004 CHEMBL3526764 0.579 0.002 CHEMBL3542268 | ||
| 0.65 | 0.004 | 0.665 | Epidermal growth factor antagonist | 0.665 0.004 CHEMBL3526326 0.545 0.004 CHEMBL3526763 0.487 0.005 CHEMBL3526479 0.543 0.004 CHEMBL3527095 0.483 0.005 CHEMBL3526380 0.506 0.004 CHEMBL3542267 0.495 0.005 CHEMBL3706535 0.464 0.005 CHEMBL3526480 0.502 0.004 CHEMBL3526764 0.59 0.004 CHEMBL3542268 | CHEMBL3526326 | |
| 0.634 | 0.004 | 0.652 | Epidermal growth factor receptor kinase inhibitor | 0.652 0.004 CHEMBL3526326 0.577 0.004 CHEMBL3526763 0.487 0.005 CHEMBL3526479 0.57 0.004 CHEMBL3527095 0.495 0.004 CHEMBL3526380 0.493 0.004 CHEMBL3542267 0.536 0.004 CHEMBL3706535 0.53 0.004 CHEMBL3526480 0.511 0.004 CHEMBL3526764 0.635 0.004 CHEMBL3542268 | CHEMBL3526326 | |
| 0.455 | 0.014 | 0.458 | Growth factor antagonist | 0.442 0.014 CHEMBL3526326 0.424 0.016 CHEMBL3526763 0.277 0.031 CHEMBL3526479 0.443 0.014 CHEMBL3527095 0.223 0.04 CHEMBL3526380 0.248 0.035 CHEMBL3542267 0.404 0.017 CHEMBL3706535 0.342 0.023 CHEMBL3526480 0.293 0.028 CHEMBL3526764 0.458 0.014 CHEMBL3542268 | CHEMBL3542268 | |
| 0.43 | 0.005 | 0.483 | Ephrin antagonist | 0.456 0.005 CHEMBL3526326 0.423 0.005 CHEMBL3526763 0.322 0.008 CHEMBL3526479 0.483 0.004 CHEMBL3527095 0.306 0.009 CHEMBL3526380 0.332 0.007 CHEMBL3542267 0.38 0.005 CHEMBL3706535 0.338 0.007 CHEMBL3526480 0.316 0.008 CHEMBL3526764 0.463 0.005 CHEMBL3542268 | CHEMBL3527095 | |
| 0.281 | 0.004 | 0.287 | ErbB-3 antagonist | 0.287 0.004 CHEMBL3526326 0.223 0.007 CHEMBL3526763 0.226 0.006 CHEMBL3526479 0.214 0.008 CHEMBL3527095 0.225 0.007 CHEMBL3526380 0.239 0.005 CHEMBL3542267 0.209 0.008 CHEMBL3706535 0.188 0.011 CHEMBL3526480 0.225 0.007 CHEMBL3526764 0.222 0.007 CHEMBL3542268 | CHEMBL3526326 | |
| 0.247 | 0.008 | 0.276 | ErbB-4 antagonist | 0.225 0.01 CHEMBL3526326 0.272 0.006 CHEMBL3526763 0.187 0.014 CHEMBL3526479 0.262 0.007 CHEMBL3527095 0.125 0.029 CHEMBL3526380 0.169 0.017 CHEMBL3542267 0.256 0.008 CHEMBL3706535 0.233 0.009 CHEMBL3526480 0.199 0.013 CHEMBL3526764 0.276 0.006 CHEMBL3542268 | CHEMBL3542268 | |
| 0.213 | 0.011 | 0.282 | EphA2 antagonist | 0.212 0.011 CHEMBL3526326 0.269 0.005 CHEMBL3526763 0.19 0.016 CHEMBL3526479 0.269 0.005 CHEMBL3527095 0.107 0.068 CHEMBL3526380 0.196 0.015 CHEMBL3542267 0.262 0.005 CHEMBL3706535 0.252 0.006 CHEMBL3526480 0.2 0.014 CHEMBL3526764 0.282 0.004 CHEMBL3542268 | CHEMBL3542268 | |
| 0.22 | 0.046 | 0.298 | Src kinase inhibitor | 0.285 0.028 CHEMBL3526326 0.25 0.036 CHEMBL3526763 0.155 0.08 CHEMBL3526479 0.298 0.026 CHEMBL3527095 0.148 0.084 CHEMBL3526380 0.257 0.034 CHEMBL3542267 0.21 0.05 CHEMBL3706535 0.22 0.045 CHEMBL3526480 0.192 0.058 CHEMBL3526764 0.255 0.035 CHEMBL3542268 | CHEMBL3527095 | |
| 0.197 | 0.069 | 0.383 | CDC-like kinase 4 inhibitor | 0.252 0.045 CHEMBL3526326 0.358 0.02 CHEMBL3526763 0.152 0.1 CHEMBL3526479 0.325 0.026 CHEMBL3527095 0.179 0.079 CHEMBL3526380 0.145 0.105 CHEMBL3542267 0.315 0.028 CHEMBL3706535 0.298 0.032 CHEMBL3526480 0.129 0.118 CHEMBL3526764 0.383 0.016 CHEMBL3542268 | CHEMBL3542268 | |
| 0.243 | 0.128 | 0.322 | Angiogenesis inhibitor | 0.246 0.126 CHEMBL3526326 0.252 0.121 CHEMBL3526763 0.296 0.095 CHEMBL3527095 0.208 0.16 CHEMBL3526480 0.322 0.082 CHEMBL3542268 | CHEMBL3542268 | |
| 0.156 | 0.052 | 0.262 | c-Src kinase inhibitor | 0.223 0.03 CHEMBL3526326 0.239 0.027 CHEMBL3526763 0.113 0.08 CHEMBL3526479 0.239 0.027 CHEMBL3527095 0.161 0.05 CHEMBL3542267 0.195 0.037 CHEMBL3706535 0.22 0.03 CHEMBL3526480 0.154 0.053 CHEMBL3526764 0.262 0.023 CHEMBL3542268 | CHEMBL3542268 | |
| 0.162 | 0.063 | 0.162 | Insulin secretagoues | 0.125 0.104 CHEMBL3526326 0.124 0.106 CHEMBL3526479 0.121 0.109 CHEMBL3526764 | ||
| 0.183 | 0.091 | 0.238 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.18 0.094 CHEMBL3526326 0.232 0.051 CHEMBL3526763 0.156 0.125 CHEMBL3526479 0.238 0.048 CHEMBL3527095 0.152 0.13 CHEMBL3542267 0.198 0.075 CHEMBL3706535 0.204 0.069 CHEMBL3526480 0.174 0.101 CHEMBL3526764 0.23 0.052 CHEMBL3542268 | CHEMBL3527095 | |
| 0.177 | 0.093 | 0.372 | Clk dual-specificity kinase inhibitor | 0.239 0.059 CHEMBL3526326 0.355 0.027 CHEMBL3526763 0.134 0.13 CHEMBL3526479 0.308 0.037 CHEMBL3527095 0.151 0.113 CHEMBL3526380 0.135 0.129 CHEMBL3542267 0.296 0.039 CHEMBL3706535 0.282 0.043 CHEMBL3526480 0.372 0.024 CHEMBL3542268 | CHEMBL3542268 | |
| 0.14 | 0.058 | 0.473 | Vascular endothelial growth factor antagonist | 0.178 0.045 CHEMBL3526326 0.143 0.057 CHEMBL3526763 0.164 0.049 CHEMBL3527095 0.473 0.009 CHEMBL3526380 0.132 0.062 CHEMBL3542267 0.107 0.077 CHEMBL3706535 0.123 0.067 CHEMBL3526480 0.093 0.089 CHEMBL3526764 0.144 0.057 CHEMBL3542268 | CHEMBL3526380 | |
| 0.127 | 0.057 | 0.477 | Vascular endothelial growth factor 2 antagonist | 0.165 0.044 CHEMBL3526326 0.126 0.058 CHEMBL3526763 0.147 0.05 CHEMBL3527095 0.477 0.009 CHEMBL3526380 0.121 0.06 CHEMBL3542267 0.093 0.077 CHEMBL3706535 0.109 0.066 CHEMBL3526480 0.127 0.057 CHEMBL3542268 | CHEMBL3526380 | |
| 0.14 | 0.078 | 0.239 | CDC-like kinase 1 inhibitor | 0.19 0.041 CHEMBL3526326 0.214 0.029 CHEMBL3526763 0.203 0.034 CHEMBL3527095 0.138 0.079 CHEMBL3526380 0.119 0.096 CHEMBL3542267 0.192 0.04 CHEMBL3706535 0.2 0.036 CHEMBL3526480 0.239 0.021 CHEMBL3542268 | CHEMBL3542268 | |
| 0.06 | 0.019 | 0.073 | Sodium/calcium exchanger inhibitor | 0.073 0.011 CHEMBL3526763 0.067 0.014 CHEMBL3527095 0.069 0.013 CHEMBL3706535 0.051 0.033 CHEMBL3526480 0.059 0.02 CHEMBL3542268 | CHEMBL3526763 | |
| 0.135 | 0.098 | 0.176 | Tyrosine kinase inhibitor | 0.166 0.082 CHEMBL3526326 0.174 0.078 CHEMBL3526763 0.176 0.077 CHEMBL3527095 0.119 0.109 CHEMBL3706535 0.157 0.086 CHEMBL3542268 | CHEMBL3527095 | |
| 0.074 | 0.04 | 0.086 | MAP kinase kinase 8 inhibitor | 0.086 0.03 CHEMBL3526326 0.063 0.056 CHEMBL3526479 0.068 0.048 CHEMBL3526380 | CHEMBL3526326 | |
| 0.083 | 0.052 | 0.088 | Ca(v)3.1 blocker | 0.082 0.054 CHEMBL3526326 0.088 0.04 CHEMBL3526380 | CHEMBL3526380 | |
| 0.127 | 0.098 | 0.265 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.192 0.046 CHEMBL3526326 0.22 0.034 CHEMBL3526763 0.201 0.042 CHEMBL3527095 0.12 0.107 CHEMBL3526380 0.12 0.107 CHEMBL3542267 0.182 0.052 CHEMBL3706535 0.208 0.039 CHEMBL3526480 0.265 0.022 CHEMBL3542268 | CHEMBL3542268 | |
| 0.109 | 0.085 | 0.14 | MAP kinase kinase inhibitor | 0.121 0.073 CHEMBL3526326 0.129 0.066 CHEMBL3526763 0.14 0.057 CHEMBL3542268 | CHEMBL3542268 | |
| 0.155 | 0.133 | 0.197 | MAP kinase kinase 5 inhibitor | 0.158 0.121 CHEMBL3526326 0.197 0.036 CHEMBL3526763 0.178 0.066 CHEMBL3527095 0.183 0.058 CHEMBL3706535 0.167 0.093 CHEMBL3526480 0.185 0.054 CHEMBL3542268 | CHEMBL3526763 | |
| 0.07 | 0.048 | 0.08 | ZAP-70 protein tyrosine kinase inhibitor | 0.08 0.036 CHEMBL3526326 0.066 0.053 CHEMBL3542267 | CHEMBL3526326 | |
| 0.112 | 0.091 | 0.149 | Lck kinase inhibitor | 0.149 0.066 CHEMBL3526326 0.136 0.074 CHEMBL3526763 0.125 0.081 CHEMBL3527095 0.102 0.1 CHEMBL3526480 0.141 0.071 CHEMBL3542268 | CHEMBL3526326 | |
| 0.106 | 0.089 | 0.111 | MAP kinase 12 inhibitor | 0.111 0.082 CHEMBL3526763 0.104 0.092 CHEMBL3527095 | CHEMBL3526763 | |
| 0.105 | 0.092 | 0.154 | RET inhibitor | 0.154 0.059 CHEMBL3526326 0.141 0.066 CHEMBL3526763 0.127 0.074 CHEMBL3527095 0.113 0.085 CHEMBL3526380 0.112 0.085 CHEMBL3706535 0.126 0.074 CHEMBL3526480 0.148 0.062 CHEMBL3542268 | CHEMBL3526326 | |
| 0.054 | 0.047 | 0.059 | CDK9/cyclin T1 inhibitor | 0.059 0.041 CHEMBL3526326 0.054 0.046 CHEMBL3526763 0.052 0.049 CHEMBL3527095 0.054 0.047 CHEMBL3526480 0.054 0.047 CHEMBL3542268 | CHEMBL3526326 | |
| 0.116 | 0.115 | 0.128 | Aurora-C kinase inhibitor | 0.128 0.087 CHEMBL3526326 0.118 0.111 CHEMBL3542267 | CHEMBL3526326 | |
| 0.075 | 0.083 | 0.095 | Transforming growth factor beta 3 antagonist | 0.095 0.03 CHEMBL3526763 0.091 0.036 CHEMBL3527095 0.089 0.039 CHEMBL3706535 0.083 0.055 CHEMBL3526480 0.091 0.037 CHEMBL3542268 | CHEMBL3526763 | |
| 0.024 | 0.034 | 0.09 | Prostacyclin antagonist | 0.034 0.022 CHEMBL3526763 0.037 0.02 CHEMBL3527095 0.032 0.024 CHEMBL3706535 0.09 0.005 CHEMBL3542268 | CHEMBL3542268 | |
| 0.071 | 0.081 | 0.108 | Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor | 0.108 0.047 CHEMBL3526326 0.094 0.059 CHEMBL3526763 0.087 0.065 CHEMBL3527095 0.082 0.07 CHEMBL3526480 0.096 0.056 CHEMBL3542268 | CHEMBL3526326 | |
| 0.091 | 0.102 | 0.134 | CDC-like kinase 3 inhibitor | 0.111 0.057 CHEMBL3526326 0.121 0.041 CHEMBL3526763 0.116 0.049 CHEMBL3527095 0.096 0.088 CHEMBL3526380 0.113 0.054 CHEMBL3706535 0.134 0.029 CHEMBL3526480 0.109 0.061 CHEMBL3542268 | CHEMBL3526480 | |
| 0.057 | 0.068 | 0.088 | Raf kinase inhibitor | 0.088 0.04 CHEMBL3526326 0.071 0.053 CHEMBL3526763 0.068 0.056 CHEMBL3527095 0.063 0.062 CHEMBL3526480 0.077 0.048 CHEMBL3542268 | CHEMBL3526326 | |
| 0.103 | 0.115 | 0.167 | Vascular endothelial growth factor 3 antagonist | 0.167 0.056 CHEMBL3526763 0.16 0.06 CHEMBL3527095 0.133 0.082 CHEMBL3706535 0.133 0.082 CHEMBL3526480 0.153 0.064 CHEMBL3542268 | CHEMBL3526763 | |
| 0.087 | 0.103 | 0.143 | Multidrug resistance-associated protein 1 inhibitor | 0.134 0.035 CHEMBL3526763 0.13 0.039 CHEMBL3527095 0.143 0.029 CHEMBL3706535 0.119 0.049 CHEMBL3526480 0.137 0.033 CHEMBL3542268 | CHEMBL3706535 | |
| 0.146 | 0.164 | 0.213 | Tumour necrosis factor alpha release inhibitor | 0.213 0.098 CHEMBL3526479 0.156 0.151 CHEMBL3526764 | CHEMBL3526479 | |
| 0.073 | 0.094 | 0.143 | Vascular endothelial growth factor 1 antagonist | 0.143 0.044 CHEMBL3526763 0.117 0.056 CHEMBL3527095 0.11 0.06 CHEMBL3706535 0.088 0.075 CHEMBL3526480 0.127 0.05 CHEMBL3542268 | CHEMBL3526763 | |
| 0.042 | 0.064 | 0.068 | Raf kinase B inhibitor | 0.068 0.035 CHEMBL3526326 0.055 0.045 CHEMBL3542268 | CHEMBL3526326 | |
| 0.139 | 0.162 | 0.184 | Histone acetyltransferase inhibitor | 0.184 0.094 CHEMBL3542268 | CHEMBL3542268 | |
| 0.078 | 0.104 | 0.119 | Toll-Like receptor 3 antagonist | 0.119 0.03 CHEMBL3526763 0.105 0.044 CHEMBL3527095 0.1 0.051 CHEMBL3706535 0.095 0.059 CHEMBL3526480 0.103 0.046 CHEMBL3542268 | CHEMBL3526763 | |
| 0.082 | 0.113 | 0.094 | MAP kinase 13 inhibitor | 0.094 0.091 CHEMBL3526763 | CHEMBL3526763 | |
| 0.119 | 0.155 | 0.332 | DNA methylase inhibitor | 0.266 0.04 CHEMBL3526326 0.195 0.083 CHEMBL3526763 0.332 0.02 CHEMBL3527095 0.144 0.123 CHEMBL3706535 0.219 0.067 CHEMBL3526480 0.33 0.02 CHEMBL3542268 | CHEMBL3527095 | |
| 0.071 | 0.108 | 0.087 | Phosphodiesterase 7B inhibitor | 0.084 0.08 CHEMBL3526326 0.087 0.075 CHEMBL3526763 0.086 0.077 CHEMBL3706535 0.087 0.075 CHEMBL3542268 | CHEMBL3542268 | |
| 0.099 | 0.137 | 0.269 | CDC-like kinase 2 inhibitor | 0.152 0.092 CHEMBL3526326 0.232 0.052 CHEMBL3526763 0.203 0.065 CHEMBL3527095 0.173 0.081 CHEMBL3706535 0.204 0.064 CHEMBL3526480 0.269 0.039 CHEMBL3542268 | CHEMBL3542268 | |
| 0.055 | 0.101 | 0.095 | Proto-oncogene tyrosine-protein kinase c-hck inhibitor | 0.086 0.045 CHEMBL3526326 0.08 0.052 CHEMBL3526763 0.095 0.038 CHEMBL3527095 0.08 0.052 CHEMBL3526380 0.073 0.062 CHEMBL3542267 0.08 0.052 CHEMBL3542268 | CHEMBL3527095 | |
| 0.071 | 0.118 | 0.091 | Glycogen synthase kinase-3 beta inhibitor | 0.091 0.09 CHEMBL3526763 | CHEMBL3526763 | |
| 0.018 | 0.066 | 0.042 | G protein-coupled receptor agonist | 0.042 0.023 CHEMBL3526764 | CHEMBL3526764 | |
| 0.033 | 0.082 | 0.089 | Raf kinase C inhibitor | 0.077 0.033 CHEMBL3526763 0.087 0.029 CHEMBL3527095 0.058 0.043 CHEMBL3706535 0.054 0.047 CHEMBL3526480 0.089 0.029 CHEMBL3542268 | CHEMBL3542268 | |
| 0.064 | 0.116 | 0.083 | Aminoacyl-tRNA synthetase inhibitor | 0.083 0.071 CHEMBL3526763 | CHEMBL3526763 | |
| 0.032 | 0.086 | 0.054 | Fibroblast growth factor 4 antagonist | 0.054 0.045 CHEMBL3527095 | CHEMBL3527095 | |
| 0.08 | 0.137 | 0.176 | Cyclooxygenase 2 inhibitor | 0.176 0.039 CHEMBL3526479 0.166 0.044 CHEMBL3526764 | CHEMBL3526479 | |
| 0.17 | 0.232 | 0.272 | Sodium/bile acid cotransporter inhibitor | 0.272 0.105 CHEMBL3526326 0.24 0.139 CHEMBL3526380 0.254 0.124 CHEMBL3542267 | CHEMBL3526326 | |
| 0.051 | 0.113 | 0.099 | Platelet activating factor beta antagonist | 0.099 0.063 CHEMBL3526763 0.087 0.073 CHEMBL3527095 0.087 0.073 CHEMBL3542268 | CHEMBL3526763 | |
| 0.025 | 0.09 | 0.052 | Fructose-1,6-bisphosphatase inhibitor | 0.043 0.034 CHEMBL3526326 0.051 0.024 CHEMBL3526763 0.052 0.023 CHEMBL3542268 | CHEMBL3542268 | |
| 0.038 | 0.106 | 0.07 | Vanilloid 1 antagonist | 0.07 0.043 CHEMBL3542268 | CHEMBL3542268 | |
| 0.115 | 0.186 | 0.303 | Dyrk kinase inhibitor | 0.217 0.089 CHEMBL3526326 0.238 0.078 CHEMBL3526763 0.232 0.08 CHEMBL3527095 0.189 0.104 CHEMBL3706535 0.303 0.052 CHEMBL3526480 0.29 0.056 CHEMBL3542268 | CHEMBL3526480 | |
| 0.019 | 0.091 | 0.033 | Purinergic P2X3 antagonist | 0.033 0.025 CHEMBL3527095 | CHEMBL3527095 | |
| 0.096 | 0.17 | 0.186 | MAP3K9 inhibitor | 0.133 0.089 CHEMBL3526763 0.125 0.105 CHEMBL3527095 0.12 0.114 CHEMBL3706535 0.127 0.101 CHEMBL3526480 0.186 0.022 CHEMBL3542268 | CHEMBL3542268 | |
| 0.077 | 0.156 | 0.112 | Sodium channel (voltage-gated) blocker | 0.112 0.094 CHEMBL3526763 | CHEMBL3526763 | |
| 0.033 | 0.125 | 0.077 | Vanilloid antagonist | 0.077 0.049 CHEMBL3542268 | CHEMBL3542268 | |
| 0.075 | 0.168 | 0.19 | Cyclooxygenase inhibitor | 0.19 0.046 CHEMBL3526479 0.161 0.061 CHEMBL3526764 | CHEMBL3526479 | |
| 0.058 | 0.155 | 0.133 | Cyclin-dependent kinase 9 inhibitor | 0.109 0.054 CHEMBL3526763 0.092 0.073 CHEMBL3527095 0.085 0.083 CHEMBL3706535 0.133 0.039 CHEMBL3526480 0.099 0.064 CHEMBL3542268 | CHEMBL3526480 | |
| 0.088 | 0.192 | 0.217 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.163 0.107 CHEMBL3526763 0.185 0.089 CHEMBL3527095 0.217 0.064 CHEMBL3526480 0.163 0.108 CHEMBL3542268 | CHEMBL3526480 | |
| 0.11 | 0.213 | 0.29 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.268 0.052 CHEMBL3526763 0.29 0.043 CHEMBL3527095 0.184 0.104 CHEMBL3706535 0.155 0.138 CHEMBL3526480 0.215 0.08 CHEMBL3542268 | CHEMBL3527095 | |
| 0.049 | 0.156 | 0.084 | Pim-1 kinase inhibitor | 0.082 0.078 CHEMBL3526763 0.084 0.075 CHEMBL3527095 | CHEMBL3527095 | |
| 0.052 | 0.159 | 0.145 | Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor | 0.121 0.068 CHEMBL3526763 0.109 0.079 CHEMBL3527095 0.094 0.09 CHEMBL3526480 0.145 0.05 CHEMBL3542268 | CHEMBL3542268 | |
| 0.051 | 0.159 | 0.145 | Abl kinase inhibitor | 0.121 0.068 CHEMBL3526763 0.108 0.078 CHEMBL3527095 0.094 0.09 CHEMBL3526480 0.145 0.05 CHEMBL3542268 | CHEMBL3542268 | |
| 0.056 | 0.164 | 0.143 | Protein-tyrosine kinase Lyn inhibitor | 0.143 0.069 CHEMBL3526763 0.139 0.072 CHEMBL3527095 0.129 0.078 CHEMBL3542267 0.105 0.098 CHEMBL3706535 0.127 0.079 CHEMBL3526480 0.131 0.077 CHEMBL3542268 | CHEMBL3526763 | |
| 0.052 | 0.162 | 0.111 | Breast cancer-resistant protein inhibitor | 0.088 0.068 CHEMBL3526763 0.098 0.057 CHEMBL3527095 0.088 0.069 CHEMBL3706535 0.111 0.046 CHEMBL3542268 | CHEMBL3542268 | |
| 0.193 | 0.303 | 0.317 | MAP kinase 1 inhibitor | 0.317 0.162 CHEMBL3526326 0.306 0.173 CHEMBL3526380 0.297 0.183 CHEMBL3542268 | CHEMBL3526326 | |
| 0.095 | 0.207 | 0.306 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.191 0.098 CHEMBL3526326 0.224 0.079 CHEMBL3526763 0.227 0.078 CHEMBL3527095 0.184 0.103 CHEMBL3706535 0.306 0.048 CHEMBL3526480 0.268 0.06 CHEMBL3542268 | CHEMBL3526480 | |
| 0.045 | 0.169 | 0.103 | Granulocyte macrophage colony stimulating factor antagonist | 0.103 0.067 CHEMBL3527095 | CHEMBL3527095 | |
| 0.08 | 0.206 | 0.167 | Dual specificity phosphatase 3 inhibitor | 0.15 0.096 CHEMBL3527095 0.124 0.123 CHEMBL3526480 0.167 0.082 CHEMBL3542268 | CHEMBL3542268 | |
| 0.086 | 0.213 | 0.127 | Sphingosine 1-phosphate receptor 2 antagonist | 0.127 0.08 CHEMBL3526763 0.123 0.09 CHEMBL3542268 | CHEMBL3526763 | |
| 0.121 | 0.249 | 0.215 | MAP-kinase-activated kinase 5 inhibitor | 0.215 0.087 CHEMBL3526763 0.19 0.116 CHEMBL3527095 0.187 0.12 CHEMBL3542268 | CHEMBL3526763 | |
| 0.053 | 0.189 | 0.102 | Proto-oncogene tyrosine-protein kinase Yes inhibitor | 0.102 0.099 CHEMBL3542268 | CHEMBL3542268 | |
| 0.082 | 0.223 | 0.274 | DNA methyltransferase I inhibitor | 0.214 0.062 CHEMBL3526326 0.274 0.037 CHEMBL3527095 0.14 0.116 CHEMBL3526480 0.266 0.04 CHEMBL3542268 | CHEMBL3527095 | |
| 0.111 | 0.254 | 0.174 | Growth factor agonist | 0.159 0.121 CHEMBL3526763 0.174 0.095 CHEMBL3527095 0.151 0.139 CHEMBL3706535 0.17 0.102 CHEMBL3542268 | CHEMBL3527095 | |
| 0.036 | 0.185 | 0.082 | Protein kinase B gamma inhibitor | 0.082 0.045 CHEMBL3526763 | CHEMBL3526763 | |
| 0.05 | 0.205 | 0.251 | Phosphodiesterase 11A inhibitor | 0.251 0.004 CHEMBL3526763 | CHEMBL3526763 | |
| 0.05 | 0.205 | 0.251 | Phosphodiesterase XI inhibitor | 0.251 0.004 CHEMBL3526763 | CHEMBL3526763 | |
| 0.024 | 0.181 | 0.101 | Phosphodiesterase V inhibitor | 0.064 0.059 CHEMBL3526763 0.101 0.027 CHEMBL3542268 | CHEMBL3542268 | |
| 0.071 | 0.234 | 0.153 | EphB2 antagonist | 0.147 0.132 CHEMBL3526763 0.147 0.132 CHEMBL3527095 0.153 0.126 CHEMBL3542268 | CHEMBL3542268 | |
| 0.024 | 0.188 | 0.097 | Phosphodiesterase 5A inhibitor | 0.097 0.028 CHEMBL3542268 | CHEMBL3542268 | |
| 0.034 | 0.202 | 0.179 | MAP kinase kinase kinase inhibitor | 0.133 0.044 CHEMBL3526763 0.179 0.024 CHEMBL3542268 | CHEMBL3542268 | |
| 0.106 | 0.281 | 0.255 | Thioredoxin glutathione reductase inhibitor | 0.255 0.13 CHEMBL3526380 | CHEMBL3526380 | |
| 0.066 | 0.266 | 0.163 | Amyloid beta precursor protein antagonist | 0.163 0.087 CHEMBL3542268 | CHEMBL3542268 | |
| 0.064 | 0.266 | 0.157 | Protein kinase (CK1) gamma 3 inhibitor | 0.157 0.082 CHEMBL3526763 0.13 0.113 CHEMBL3527095 0.13 0.114 CHEMBL3542268 | CHEMBL3526763 | |
| 0.086 | 0.293 | 0.146 | Death-associated protein kinase 1 inhibitor | 0.127 0.091 CHEMBL3526763 0.126 0.093 CHEMBL3527095 0.134 0.07 CHEMBL3706535 0.146 0.046 CHEMBL3526480 0.129 0.084 CHEMBL3542268 | CHEMBL3526480 | |
| 0.056 | 0.265 | 0.133 | Protein kinase (CK1) gamma 1 inhibitor | 0.133 0.084 CHEMBL3526763 | CHEMBL3526763 | |
| 0.035 | 0.244 | 0.1 | Sphingosine 1-phosphate receptor antagonist | 0.1 0.022 CHEMBL3706535 0.076 0.054 CHEMBL3542268 | CHEMBL3706535 | |
| 0.028 | 0.238 | 0.118 | Check point kinase 2 inhibitor | 0.118 0.051 CHEMBL3526763 | CHEMBL3526763 | |
| 0.046 | 0.26 | 0.097 | Protein kinase (CK1) gamma 2 inhibitor | 0.097 0.087 CHEMBL3526763 | CHEMBL3526763 | |
| 0.062 | 0.279 | 0.135 | Dual specificity phosphatase inhibitor | 0.135 0.113 CHEMBL3542268 | CHEMBL3542268 | |
| 0.041 | 0.268 | 0.097 | MAP kinase kinase 1 inhibitor | 0.097 0.061 CHEMBL3542268 | CHEMBL3542268 | |
| 0.043 | 0.271 | 0.117 | Protein kinase (CK1) gamma inhibitor | 0.117 0.093 CHEMBL3526763 | CHEMBL3526763 | |
| 0.018 | 0.261 | 0.126 | Leukotriene synthesis inhibitor | 0.126 0.015 CHEMBL3526479 | CHEMBL3526479 | |
| 0.094 | 0.338 | 0.394 | Hypoxia-inducible factor 1 alpha inhibitor | 0.192 0.162 CHEMBL3526326 0.19 0.165 CHEMBL3526763 0.197 0.155 CHEMBL3527095 0.197 0.155 CHEMBL3526480 0.394 0.032 CHEMBL3542268 | CHEMBL3542268 | |
| 0.062 | 0.316 | 0.14 | Death-associated protein kinase 3 inhibitor | 0.14 0.138 CHEMBL3527095 | CHEMBL3527095 | |
| 0.022 | 0.28 | 0.048 | Factor IXa inhibitor | 0.048 0.041 CHEMBL3526763 | CHEMBL3526763 | |
| 0.06 | 0.33 | 0.208 | Antiamyloidogenic | 0.157 0.138 CHEMBL3526480 0.208 0.094 CHEMBL3526764 | CHEMBL3526764 | |
| 0.109 | 0.403 | 0.189 | Caspase 3 stimulant | 0.189 0.187 CHEMBL3526480 | CHEMBL3526480 | |
| 0.037 | 0.335 | 0.127 | Beta amyloid protein antagonist | 0.127 0.06 CHEMBL3526480 | CHEMBL3526480 | |
| 0.043 | 0.356 | 0.856 | Interleukin 1 antagonist | 0.171 0.046 CHEMBL3526480 0.856 0.003 CHEMBL3526764 | CHEMBL3526764 | |
| 0.015 | 0.329 | 0.104 | Protein kinase (CK2) alpha inhibitor | 0.104 0.073 CHEMBL3526326 0.097 0.079 CHEMBL3542268 | CHEMBL3526326 | |
| 0.037 | 0.353 | 0.863 | Interleukin 1b antagonist | 0.137 0.05 CHEMBL3526480 0.863 0.002 CHEMBL3526764 | CHEMBL3526764 | |
| 0.051 | 0.379 | 0.307 | Prostaglandin dehydrogenase inhibitor | 0.307 0.098 CHEMBL3526480 | CHEMBL3526480 | |
| 0.005 | 0.334 | 0.066 | Potassium channel small-conductance Ca-activated activator | 0.028 0.026 CHEMBL3526763 0.066 0.007 CHEMBL3526480 | CHEMBL3526480 | |
| 0.03 | 0.365 | 0.122 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.122 0.114 CHEMBL3526763 | CHEMBL3526763 | |
| 0.017 | 0.353 | 0.044 | Guanylate cyclase stimulant | 0.04 0.038 CHEMBL3527095 0.044 0.03 CHEMBL3542268 | CHEMBL3542268 | |
| 0.031 | 0.378 | 0.056 | Lipocortins synthesis agonist | 0.056 0.045 CHEMBL3526380 | CHEMBL3526380 | |
| 0.049 | 0.4 | 0.142 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.142 0.139 CHEMBL3526763 | CHEMBL3526763 | |
| 0.057 | 0.409 | 0.156 | MAP kinase 3 inhibitor | 0.128 0.112 CHEMBL3526763 0.142 0.08 CHEMBL3526480 0.156 0.059 CHEMBL3542268 | CHEMBL3542268 | |
| 0.02 | 0.38 | 0.079 | Macrophage migration inhibitory factor inhibitor | 0.078 0.054 CHEMBL3527095 0.079 0.053 CHEMBL3542268 | CHEMBL3542268 | |
| 0.015 | 0.379 | 0.095 | Bcr-Abl kinase inhibitor | 0.095 0.046 CHEMBL3542268 | CHEMBL3542268 | |
| 0.02 | 0.386 | 0.187 | Potassium channel (Ca-activated) activator | 0.122 0.04 CHEMBL3526763 0.091 0.064 CHEMBL3527095 0.112 0.046 CHEMBL3706535 0.153 0.027 CHEMBL3526480 0.187 0.017 CHEMBL3542268 | CHEMBL3542268 | |
| 0.065 | 0.432 | 0.128 | Sphingosine 1-phosphate receptor 5 antagonist | 0.128 0.105 CHEMBL3526763 0.126 0.109 CHEMBL3542268 | CHEMBL3526763 | |
| 0.021 | 0.394 | 0.096 | Myeloperoxidase inhibitor | 0.08 0.067 CHEMBL3526763 0.096 0.04 CHEMBL3542268 | CHEMBL3542268 | |
| 0.047 | 0.424 | 0.407 | Streptokinase A inhibitor | 0.176 0.149 CHEMBL3526480 0.407 0.045 CHEMBL3526764 | CHEMBL3526764 | |
| 0.015 | 0.397 | 0.498 | 5-Lipoxygenase inhibitor | 0.498 0.004 CHEMBL3526479 0.087 0.074 CHEMBL3526480 0.088 0.073 CHEMBL3526764 | CHEMBL3526479 | |
| 0.005 | 0.408 | 0.052 | 5 Hydroxytryptamine 2C agonist | 0.052 0.026 CHEMBL3526763 | CHEMBL3526763 | |
| 0.027 | 0.438 | 0.088 | Thioredoxin inhibitor | 0.088 0.065 CHEMBL3542268 | CHEMBL3542268 | |
| 0.039 | 0.499 | 0.105 | Transcription factor STAT6 inhibitor | 0.105 0.093 CHEMBL3526763 0.103 0.099 CHEMBL3527095 | CHEMBL3526763 | |
| 0.012 | 0.474 | 0.158 | Glycogen synthase kinase-3 alpha inhibitor | 0.122 0.083 CHEMBL3526763 0.111 0.092 CHEMBL3527095 0.158 0.061 CHEMBL3526480 0.106 0.098 CHEMBL3542268 | CHEMBL3526480 | |
| 0.047 | 0.511 | 0.293 | 15-Lipoxygenase inhibitor | 0.293 0.136 CHEMBL3526380 | CHEMBL3526380 | |
| 0.04 | 0.537 | 0.135 | Tumour necrosis factor antagonist | 0.135 0.12 CHEMBL3542268 | CHEMBL3542268 | |
| 0.014 | 0.512 | 0.038 | Calcium-independent phospholipase A2 inhibitor | 0.038 0.013 CHEMBL3527095 | CHEMBL3527095 | |
| 0.011 | 0.543 | 0.138 | LIM domain kinase 1 inhibitor | 0.138 0.11 CHEMBL3526763 0.136 0.114 CHEMBL3527095 | CHEMBL3526763 | |
| 0.014 | 0.579 | 0.14 | MAP kinase kinase 2 inhibitor | 0.14 0.13 CHEMBL3526763 | CHEMBL3526763 | |
| 0.018 | 0.62 | 0.203 | Lipoxygenase inhibitor | 0.203 0.137 CHEMBL3526480 | CHEMBL3526480 | |
| 0.018 | 0.624 | 0.677 | Interleukin antagonist | 0.677 0.005 CHEMBL3526764 | CHEMBL3526764 | |
| 0.013 | 0.631 | 0.143 | I kappa B kinase epsilon inhibitor | 0.143 0.128 CHEMBL3526763 0.142 0.128 CHEMBL3542268 | CHEMBL3526763 | |
| 0.023 | 0.644 | 0.158 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.158 0.131 CHEMBL3542268 | CHEMBL3542268 | |
| 0.012 | 0.671 | 0.702 | Free radical scavenger | 0.702 0.005 CHEMBL3526764 | CHEMBL3526764 | |
| 0.007 | 0.689 | 0.218 | Aryl hydrocarbon receptor agonist | 0.218 0.093 CHEMBL3527095 | CHEMBL3527095 | |
| 0.045 | 0.736 | 0.347 | Caspase 9 stimulant | 0.347 0.148 CHEMBL3527095 0.287 0.209 CHEMBL3526480 0.305 0.188 CHEMBL3542268 | CHEMBL3527095 | |
| 0.011 | 0.744 | 0.09 | Xanthine oxidase inhibitor | 0.09 0.071 CHEMBL3542268 | CHEMBL3542268 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |