| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.922 | 0.002 | 0.922 | Vasodilator, peripheral | 0.763 0.004 CHEMBL3544675 0.901 0.003 CHEMBL1343 0.909 0.003 CHEMBL1514176 | ||
| 0.904 | 0.002 | 0.922 | Cyclic AMP phosphodiesterase inhibitor | 0.908 0.001 CHEMBL3544675 0.804 0.002 CHEMBL1343 0.922 0.001 CHEMBL1514176 | CHEMBL1514176 | |
| 0.645 | 0.009 | 0.751 | Spasmolytic | 0.447 0.031 CHEMBL3544675 0.633 0.01 CHEMBL1343 0.751 0.005 CHEMBL1514176 | CHEMBL1514176 | |
| 0.597 | 0.005 | 0.7 | Diuretic | 0.554 0.005 CHEMBL3544675 0.7 0.004 CHEMBL1343 0.542 0.006 CHEMBL1514176 | CHEMBL1343 | |
| 0.59 | 0.006 | 0.59 | Vasodilator | 0.496 0.012 CHEMBL3544675 0.55 0.009 CHEMBL1343 0.582 0.007 CHEMBL1514176 | ||
| 0.576 | 0.007 | 0.755 | Psychostimulant | 0.482 0.013 CHEMBL3544675 0.755 0.004 CHEMBL1343 0.569 0.007 CHEMBL1514176 | CHEMBL1343 | |
| 0.562 | 0.004 | 0.562 | Bronchodilator | 0.551 0.004 CHEMBL3544675 0.492 0.005 CHEMBL1343 0.513 0.004 CHEMBL1514176 | ||
| 0.549 | 0.003 | 0.549 | TRPA1 antagonist | 0.231 0.005 CHEMBL3544675 0.262 0.004 CHEMBL1343 0.337 0.004 CHEMBL1514176 | ||
| 0.521 | 0.02 | 0.636 | Immunomodulator | 0.304 0.08 CHEMBL3544675 0.55 0.017 CHEMBL1343 0.636 0.009 CHEMBL1514176 | CHEMBL1514176 | |
| 0.53 | 0.074 | 0.53 | DNA directed DNA polymerase inhibitor | 0.456 0.095 CHEMBL3544675 0.421 0.107 CHEMBL1343 0.396 0.117 CHEMBL1514176 | ||
| 0.446 | 0.004 | 0.517 | Adenosine A1 receptor antagonist | 0.517 0.003 CHEMBL3544675 0.418 0.004 CHEMBL1343 0.455 0.004 CHEMBL1514176 | CHEMBL3544675 | |
| 0.473 | 0.033 | 0.582 | Antithrombotic | 0.282 0.101 CHEMBL3544675 0.568 0.02 CHEMBL1343 0.582 0.018 CHEMBL1514176 | CHEMBL1514176 | |
| 0.471 | 0.041 | 0.471 | Immunosuppressant | 0.395 0.065 CHEMBL3544675 0.347 0.088 CHEMBL1343 0.398 0.064 CHEMBL1514176 | ||
| 0.427 | 0.003 | 0.498 | Adenosine A2b receptor antagonist | 0.498 0.002 CHEMBL3544675 0.33 0.003 CHEMBL1343 0.279 0.004 CHEMBL1514176 | CHEMBL3544675 | |
| 0.447 | 0.024 | 0.671 | Vasodilator, coronary | 0.333 0.064 CHEMBL3544675 0.586 0.008 CHEMBL1343 0.671 0.005 CHEMBL1514176 | CHEMBL1514176 | |
| 0.419 | 0.003 | 0.419 | Phosphodiesterase I inhibitor | 0.404 0.003 CHEMBL3544675 0.325 0.004 CHEMBL1343 0.289 0.005 CHEMBL1514176 | ||
| 0.408 | 0.004 | 0.436 | Adenosine A2 receptor antagonist | 0.436 0.004 CHEMBL3544675 0.351 0.004 CHEMBL1343 0.373 0.004 CHEMBL1514176 | CHEMBL3544675 | |
| 0.346 | 0.005 | 0.346 | Mediator release inhibitor | 0.159 0.025 CHEMBL3544675 0.268 0.009 CHEMBL1343 0.171 0.021 CHEMBL1514176 | ||
| 0.339 | 0.004 | 0.356 | Adenosine A2a receptor antagonist | 0.356 0.004 CHEMBL3544675 0.323 0.005 CHEMBL1343 0.325 0.005 CHEMBL1514176 | CHEMBL3544675 | |
| 0.371 | 0.038 | 0.409 | Hypoxia-inducible factor 1 alpha inhibitor | 0.363 0.041 CHEMBL3544675 0.409 0.028 CHEMBL1343 0.29 0.07 CHEMBL1514176 | CHEMBL1343 | |
| 0.328 | 0.01 | 0.328 | Acetylcholine M1 receptor antagonist | 0.262 0.022 CHEMBL3544675 0.23 0.031 CHEMBL1343 0.251 0.025 CHEMBL1514176 | ||
| 0.308 | 0.001 | 0.308 | Adenosine uptake inhibitor | 0.167 0.002 CHEMBL3544675 0.071 0.003 CHEMBL1343 0.064 0.003 CHEMBL1514176 | ||
| 0.287 | 0.02 | 0.287 | Tumour necrosis factor antagonist | 0.205 0.051 CHEMBL3544675 0.273 0.024 CHEMBL1343 0.211 0.047 CHEMBL1514176 | ||
| 0.238 | 0.007 | 0.247 | Interleukin 8 antagonist | 0.165 0.026 CHEMBL3544675 0.247 0.006 CHEMBL1343 0.138 0.042 CHEMBL1514176 | CHEMBL1343 | |
| 0.232 | 0.008 | 0.407 | Adenosine A3 receptor antagonist | 0.407 0.004 CHEMBL3544675 0.23 0.008 CHEMBL1343 0.228 0.008 CHEMBL1514176 | CHEMBL3544675 | |
| 0.228 | 0.006 | 0.355 | DNA repair enzyme inhibitor | 0.178 0.014 CHEMBL3544675 0.355 0.004 CHEMBL1343 0.202 0.008 CHEMBL1514176 | CHEMBL1343 | |
| 0.216 | 0.006 | 0.488 | Electrolyte absorption antagonist | 0.122 0.035 CHEMBL3544675 0.488 0.002 CHEMBL1343 0.314 0.004 CHEMBL1514176 | CHEMBL1343 | |
| 0.23 | 0.036 | 0.23 | Histone acetyltransferase inhibitor | 0.188 0.087 CHEMBL3544675 0.201 0.068 CHEMBL1343 0.177 0.104 CHEMBL1514176 | ||
| 0.263 | 0.074 | 0.432 | Cardiotonic | 0.275 0.067 CHEMBL3544675 0.321 0.048 CHEMBL1343 0.432 0.023 CHEMBL1514176 | CHEMBL1514176 | |
| 0.266 | 0.09 | 0.405 | Immunostimulant | 0.167 0.141 CHEMBL3544675 0.354 0.063 CHEMBL1343 0.405 0.048 CHEMBL1514176 | CHEMBL1514176 | |
| 0.227 | 0.054 | 0.316 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.162 0.123 CHEMBL3544675 0.316 0.019 CHEMBL1343 0.227 0.054 CHEMBL1514176 | CHEMBL1343 | |
| 0.192 | 0.026 | 0.192 | Acetylcholine muscarinic antagonist | 0.139 0.051 CHEMBL3544675 0.111 0.077 CHEMBL1343 0.115 0.072 CHEMBL1514176 | ||
| 0.289 | 0.124 | 0.328 | GABA C receptor rho-3 antagonist | 0.305 0.112 CHEMBL3544675 0.328 0.098 CHEMBL1343 | CHEMBL1343 | |
| 0.161 | 0.009 | 0.179 | Phosphodiesterase 5A inhibitor | 0.168 0.009 CHEMBL3544675 0.179 0.007 CHEMBL1343 0.132 0.015 CHEMBL1514176 | CHEMBL1343 | |
| 0.174 | 0.031 | 0.174 | Antibacterial (Helicobacter pylori) | 0.14 0.056 CHEMBL3544675 0.116 0.087 CHEMBL1343 0.133 0.064 CHEMBL1514176 | ||
| 0.153 | 0.01 | 0.17 | Phosphodiesterase V inhibitor | 0.162 0.009 CHEMBL3544675 0.17 0.008 CHEMBL1343 0.127 0.016 CHEMBL1514176 | CHEMBL1343 | |
| 0.15 | 0.007 | 0.163 | Phosphodiesterase 4C inhibitor | 0.163 0.006 CHEMBL3544675 0.138 0.009 CHEMBL1343 0.135 0.009 CHEMBL1514176 | CHEMBL3544675 | |
| 0.153 | 0.012 | 0.153 | Phosphodiesterase 4B inhibitor | 0.141 0.014 CHEMBL3544675 0.083 0.034 CHEMBL1343 | ||
| 0.146 | 0.007 | 0.213 | Phosphodiesterase VI inhibitor | 0.17 0.005 CHEMBL3544675 0.137 0.008 CHEMBL1343 0.213 0.004 CHEMBL1514176 | CHEMBL1514176 | |
| 0.146 | 0.011 | 0.223 | Phosphodiesterase 6D inhibitor | 0.149 0.01 CHEMBL3544675 0.154 0.009 CHEMBL1343 0.223 0.004 CHEMBL1514176 | CHEMBL1514176 | |
| 0.141 | 0.008 | 0.141 | Phosphodiesterase 1B inhibitor | 0.128 0.009 CHEMBL3544675 0.141 0.008 CHEMBL1343 0.097 0.015 CHEMBL1514176 | ||
| 0.151 | 0.019 | 0.151 | Phosphodiesterase 4D inhibitor | 0.148 0.02 CHEMBL3544675 0.151 0.019 CHEMBL1343 0.133 0.023 CHEMBL1514176 | ||
| 0.221 | 0.092 | 0.31 | Tumour necrosis factor alpha release inhibitor | 0.31 0.05 CHEMBL1514176 | CHEMBL1514176 | |
| 0.132 | 0.005 | 0.132 | Phosphodiesterase 1A inhibitor | 0.125 0.006 CHEMBL3544675 0.113 0.008 CHEMBL1343 0.082 0.015 CHEMBL1514176 | ||
| 0.17 | 0.047 | 0.199 | Interleukin 1 antagonist | 0.154 0.055 CHEMBL1343 0.199 0.033 CHEMBL1514176 | CHEMBL1514176 | |
| 0.169 | 0.047 | 0.171 | Phosphodiesterase inhibitor | 0.171 0.046 CHEMBL3544675 0.136 0.068 CHEMBL1343 0.133 0.07 CHEMBL1514176 | CHEMBL3544675 | |
| 0.131 | 0.011 | 0.133 | Phosphodiesterase 4A inhibitor | 0.133 0.011 CHEMBL3544675 0.064 0.028 CHEMBL1343 0.073 0.023 CHEMBL1514176 | CHEMBL3544675 | |
| 0.142 | 0.023 | 0.142 | Anabolic | 0.093 0.073 CHEMBL3544675 0.125 0.035 CHEMBL1343 0.116 0.043 CHEMBL1514176 | ||
| 0.154 | 0.037 | 0.216 | Heat shock protein 70 antagonist | 0.141 0.07 CHEMBL3544675 0.216 0.005 CHEMBL1343 0.161 0.026 CHEMBL1514176 | CHEMBL1343 | |
| 0.259 | 0.143 | 0.259 | Calpain 2 inhibitor | |||
| 0.257 | 0.142 | 0.587 | Toll-Like receptor agonist | 0.305 0.108 CHEMBL3544675 0.587 0.019 CHEMBL1343 0.479 0.036 CHEMBL1514176 | CHEMBL1343 | |
| 0.159 | 0.048 | 0.159 | Cholinergic antagonist | 0.133 0.063 CHEMBL3544675 | ||
| 0.194 | 0.083 | 0.268 | DNA methylase inhibitor | 0.149 0.118 CHEMBL3544675 0.268 0.039 CHEMBL1343 0.188 0.087 CHEMBL1514176 | CHEMBL1343 | |
| 0.151 | 0.044 | 0.301 | Adenylate cyclase inhibitor | 0.264 0.018 CHEMBL3544675 0.293 0.014 CHEMBL1343 0.301 0.013 CHEMBL1514176 | CHEMBL1514176 | |
| 0.115 | 0.008 | 0.115 | Phosphodiesterase II inhibitor | 0.07 0.023 CHEMBL3544675 0.097 0.012 CHEMBL1343 0.112 0.009 CHEMBL1514176 | ||
| 0.151 | 0.048 | 0.289 | DNA polymerase I inhibitor | 0.289 0.012 CHEMBL3544675 0.141 0.054 CHEMBL1343 0.105 0.081 CHEMBL1514176 | CHEMBL3544675 | |
| 0.236 | 0.135 | 0.51 | Cholesterol antagonist | 0.51 0.031 CHEMBL1343 0.492 0.034 CHEMBL1514176 | CHEMBL1343 | |
| 0.117 | 0.016 | 0.168 | Phosphodiesterase III inhibitor | 0.168 0.008 CHEMBL3544675 0.099 0.023 CHEMBL1343 0.099 0.023 CHEMBL1514176 | CHEMBL3544675 | |
| 0.15 | 0.05 | 0.15 | Acetylcholine antagonist | 0.126 0.065 CHEMBL3544675 | ||
| 0.157 | 0.059 | 0.277 | Cell wall synthesis inhibitor | 0.277 0.012 CHEMBL1343 0.218 0.024 CHEMBL1514176 | CHEMBL1343 | |
| 0.106 | 0.008 | 0.106 | Phosphodiesterase 2A inhibitor | 0.057 0.026 CHEMBL3544675 0.088 0.011 CHEMBL1343 0.103 0.009 CHEMBL1514176 | ||
| 0.247 | 0.15 | 0.583 | Toll-Like receptor 7 agonist | 0.294 0.114 CHEMBL3544675 0.583 0.019 CHEMBL1343 0.46 0.04 CHEMBL1514176 | CHEMBL1343 | |
| 0.174 | 0.083 | 0.261 | DNA methyltransferase I inhibitor | 0.149 0.105 CHEMBL3544675 0.261 0.042 CHEMBL1343 0.149 0.105 CHEMBL1514176 | CHEMBL1343 | |
| 0.089 | 0.007 | 0.121 | Thymidine kinase inhibitor | 0.102 0.006 CHEMBL3544675 0.121 0.005 CHEMBL1343 0.113 0.005 CHEMBL1514176 | CHEMBL1343 | |
| 0.18 | 0.099 | 0.197 | Anticonvulsant | 0.163 0.114 CHEMBL3544675 0.197 0.085 CHEMBL1343 | CHEMBL1343 | |
| 0.087 | 0.008 | 0.225 | Adenosine deaminase inhibitor | 0.079 0.009 CHEMBL3544675 0.117 0.004 CHEMBL1343 0.225 0.002 CHEMBL1514176 | CHEMBL1514176 | |
| 0.138 | 0.059 | 0.17 | Sphingosine 1-phosphate receptor 2 antagonist | 0.136 0.063 CHEMBL3544675 0.17 0.021 CHEMBL1343 0.143 0.051 CHEMBL1514176 | CHEMBL1343 | |
| 0.102 | 0.026 | 0.114 | Caspase 7 inhibitor | 0.082 0.056 CHEMBL3544675 0.114 0.017 CHEMBL1343 | CHEMBL1343 | |
| 0.219 | 0.145 | 0.267 | Thyroid hormone antagonist | 0.267 0.113 CHEMBL1343 | CHEMBL1343 | |
| 0.197 | 0.127 | 0.314 | DNA synthesis inhibitor | 0.216 0.1 CHEMBL3544675 0.314 0.039 CHEMBL1343 0.248 0.068 CHEMBL1514176 | CHEMBL1343 | |
| 0.119 | 0.049 | 0.119 | Electron transport complex I inhibitor | 0.11 0.062 CHEMBL3544675 0.108 0.067 CHEMBL1514176 | ||
| 0.083 | 0.018 | 0.09 | Phosphodiesterase 1C inhibitor | 0.074 0.025 CHEMBL3544675 0.09 0.013 CHEMBL1343 0.067 0.033 CHEMBL1514176 | CHEMBL1343 | |
| 0.067 | 0.003 | 0.067 | DNA polymerase III inhibitor | 0.059 0.003 CHEMBL3544675 0.061 0.003 CHEMBL1343 0.065 0.003 CHEMBL1514176 | ||
| 0.067 | 0.005 | 0.073 | Phosphodiesterase 6C inhibitor | 0.073 0.004 CHEMBL3544675 0.068 0.005 CHEMBL1343 0.062 0.007 CHEMBL1514176 | CHEMBL3544675 | |
| 0.208 | 0.147 | 0.235 | Thyroid hormone beta antagonist | 0.235 0.128 CHEMBL1343 | CHEMBL1343 | |
| 0.069 | 0.009 | 0.098 | Nicotinic acid receptor agonist | 0.098 0.005 CHEMBL3544675 0.048 0.015 CHEMBL1343 0.036 0.025 CHEMBL1514176 | CHEMBL3544675 | |
| 0.214 | 0.156 | 0.214 | Transcription factor NF kappa B inhibitor | |||
| 0.068 | 0.014 | 0.145 | Nicotinic acid receptor 1 agonist | 0.145 0.005 CHEMBL3544675 0.084 0.01 CHEMBL1343 0.066 0.014 CHEMBL1514176 | CHEMBL3544675 | |
| 0.138 | 0.084 | 0.138 | Cytidine deaminase inhibitor | 0.138 0.084 CHEMBL3544675 0.114 0.108 CHEMBL1514176 | ||
| 0.057 | 0.005 | 0.079 | Phosphodiesterase 6B inhibitor | 0.079 0.004 CHEMBL3544675 0.06 0.005 CHEMBL1343 0.049 0.007 CHEMBL1514176 | CHEMBL3544675 | |
| 0.107 | 0.058 | 0.167 | Adenylate kinase inhibitor | 0.1 0.067 CHEMBL3544675 0.167 0.021 CHEMBL1343 0.113 0.05 CHEMBL1514176 | CHEMBL1343 | |
| 0.076 | 0.03 | 0.196 | Carbamoyl phosphate synthetase inhibitor | 0.083 0.027 CHEMBL3544675 0.196 0.008 CHEMBL1343 0.092 0.023 CHEMBL1514176 | CHEMBL1343 | |
| 0.094 | 0.05 | 0.098 | Phosphodiesterase IV inhibitor | 0.098 0.047 CHEMBL3544675 | CHEMBL3544675 | |
| 0.207 | 0.17 | 0.207 | Apoptosis antagonist | 0.196 0.185 CHEMBL1343 | ||
| 0.153 | 0.116 | 0.313 | Interleukin antagonist | 0.24 0.065 CHEMBL1343 0.313 0.045 CHEMBL1514176 | CHEMBL1514176 | |
| 0.176 | 0.14 | 0.234 | RNA-directed DNA polymerase inhibitor | 0.178 0.137 CHEMBL3544675 0.234 0.061 CHEMBL1343 0.23 0.064 CHEMBL1514176 | CHEMBL1343 | |
| 0.043 | 0.007 | 0.043 | Calcium-independent phospholipase A2 inhibitor | 0.041 0.009 CHEMBL3544675 | ||
| 0.052 | 0.019 | 0.066 | Dipeptidyl peptidase IV inhibitor | 0.066 0.011 CHEMBL1343 0.046 0.028 CHEMBL1514176 | CHEMBL1343 | |
| 0.054 | 0.021 | 0.054 | Cytokine production stimulant | 0.05 0.03 CHEMBL1514176 | ||
| 0.068 | 0.038 | 0.068 | Acetylcholine M2 receptor antagonist | |||
| 0.138 | 0.109 | 0.235 | Antipruritic | 0.235 0.03 CHEMBL1343 0.189 0.057 CHEMBL1514176 | CHEMBL1343 | |
| 0.033 | 0.005 | 0.038 | Phosphodiesterase 6G inhibitor | 0.038 0.004 CHEMBL3544675 0.034 0.005 CHEMBL1343 0.03 0.008 CHEMBL1514176 | CHEMBL3544675 | |
| 0.033 | 0.005 | 0.038 | Phosphodiesterase 6H inhibitor | 0.038 0.004 CHEMBL3544675 0.034 0.005 CHEMBL1343 0.03 0.008 CHEMBL1514176 | CHEMBL3544675 | |
| 0.03 | 0.003 | 0.03 | DNA polymerase III polC-type inhibitor | 0.027 0.003 CHEMBL3544675 0.024 0.003 CHEMBL1343 0.027 0.003 CHEMBL1514176 | ||
| 0.056 | 0.031 | 0.065 | Dipeptidyl peptidase inhibitor | 0.065 0.021 CHEMBL1343 | CHEMBL1343 | |
| 0.03 | 0.007 | 0.042 | Phosphodiesterase 6A inhibitor | 0.042 0.004 CHEMBL3544675 0.031 0.006 CHEMBL1343 0.029 0.008 CHEMBL1514176 | CHEMBL3544675 | |
| 0.1 | 0.078 | 0.203 | Mucolytic | 0.203 0.013 CHEMBL1343 0.167 0.024 CHEMBL1514176 | CHEMBL1343 | |
| 0.078 | 0.056 | 0.157 | Interferon agonist | 0.117 0.018 CHEMBL1343 0.157 0.009 CHEMBL1514176 | CHEMBL1514176 | |
| 0.073 | 0.053 | 0.073 | Acetylcholine M4 receptor antagonist | |||
| 0.123 | 0.104 | 0.123 | Death-associated protein kinase 1 inhibitor | |||
| 0.078 | 0.06 | 0.13 | Histamine H1 receptor antagonist | 0.13 0.029 CHEMBL1343 | CHEMBL1343 | |
| 0.032 | 0.016 | 0.035 | Purinergic P2X agonist | 0.033 0.016 CHEMBL1343 0.035 0.015 CHEMBL1514176 | CHEMBL1514176 | |
| 0.07 | 0.056 | 0.129 | Glutamate dehydrogenase inhibitor | 0.076 0.049 CHEMBL3544675 0.129 0.02 CHEMBL1343 0.066 0.062 CHEMBL1514176 | CHEMBL1343 | |
| 0.053 | 0.039 | 0.089 | Acyl-CoA dehydrogenase inhibitor | 0.061 0.033 CHEMBL1343 0.089 0.019 CHEMBL1514176 | CHEMBL1514176 | |
| 0.089 | 0.075 | 0.149 | Interleukin 12 antagonist | 0.146 0.014 CHEMBL1343 0.149 0.013 CHEMBL1514176 | CHEMBL1514176 | |
| 0.042 | 0.029 | 0.058 | Angiotensin AT1 receptor antagonist | 0.058 0.008 CHEMBL1343 0.051 0.016 CHEMBL1514176 | CHEMBL1343 | |
| 0.017 | 0.005 | 0.017 | Calcium-dependent phospholipase A2 inhibitor | 0.015 0.005 CHEMBL3544675 | ||
| 0.013 | 0.003 | 0.021 | DNA polymerase III subunit alpha inhibitor | 0.008 0.004 CHEMBL3544675 0.016 0.002 CHEMBL1343 0.021 0.002 CHEMBL1514176 | CHEMBL1514176 | |
| 0.086 | 0.078 | 0.146 | Interleukin 1 beta converting enzyme inhibitor | 0.146 0.019 CHEMBL1343 | CHEMBL1343 | |
| 0.086 | 0.08 | 0.086 | Lanosterol 14 alpha demethylase inhibitor | |||
| 0.034 | 0.03 | 0.036 | ATM kinase inhibitor | 0.036 0.025 CHEMBL1343 | CHEMBL1343 | |
| 0.024 | 0.024 | 0.027 | Thymidine phosphorylase inhibitor | 0.026 0.017 CHEMBL3544675 0.027 0.016 CHEMBL1343 0.027 0.016 CHEMBL1514176 | CHEMBL1514176 | |
| 0.022 | 0.025 | 0.051 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.044 0.011 CHEMBL3544675 0.051 0.009 CHEMBL1343 0.039 0.013 CHEMBL1514176 | CHEMBL1343 | |
| 0.057 | 0.06 | 0.114 | Interferon inducer | 0.084 0.021 CHEMBL1343 0.114 0.008 CHEMBL1514176 | CHEMBL1514176 | |
| 0.077 | 0.081 | 0.143 | NADH dehydrogenase inhibitor | 0.088 0.06 CHEMBL3544675 0.143 0.019 CHEMBL1343 0.119 0.029 CHEMBL1514176 | CHEMBL1343 | |
| 0.018 | 0.022 | 0.024 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.024 0.008 CHEMBL3544675 0.024 0.008 CHEMBL1343 0.022 0.012 CHEMBL1514176 | CHEMBL1343 | |
| 0.024 | 0.028 | 0.03 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.029 0.012 CHEMBL3544675 0.029 0.013 CHEMBL1343 0.03 0.012 CHEMBL1514176 | CHEMBL1514176 | |
| 0.03 | 0.034 | 0.046 | Angiotensin II receptor antagonist | 0.046 0.009 CHEMBL1343 0.038 0.017 CHEMBL1514176 | CHEMBL1343 | |
| 0.037 | 0.042 | 0.04 | Phosphodiesterase 3B inhibitor | 0.04 0.036 CHEMBL3544675 | CHEMBL3544675 | |
| 0.044 | 0.051 | 0.058 | 5 Hydroxytryptamine 4 antagonist | 0.058 0.026 CHEMBL3544675 | CHEMBL3544675 | |
| 0.073 | 0.089 | 0.12 | Antihistaminic | 0.12 0.043 CHEMBL3544675 | CHEMBL3544675 | |
| 0.024 | 0.041 | 0.055 | Fumarate hydratase inhibitor | 0.055 0.012 CHEMBL1343 | CHEMBL1343 | |
| 0.007 | 0.024 | 0.019 | Angiotensin AT1B receptor antagonist | 0.019 0.006 CHEMBL1343 | CHEMBL1343 | |
| 0.04 | 0.061 | 0.049 | GABA receptor antagonist | 0.049 0.046 CHEMBL1343 | CHEMBL1343 | |
| 0.126 | 0.148 | 0.187 | Lipocortins synthesis antagonist | 0.187 0.066 CHEMBL1343 | CHEMBL1343 | |
| 0.077 | 0.101 | 0.233 | Expectorant | 0.198 0.021 CHEMBL1343 0.233 0.015 CHEMBL1514176 | CHEMBL1514176 | |
| 0.062 | 0.089 | 0.105 | Histamine antagonist | 0.105 0.045 CHEMBL3544675 | CHEMBL3544675 | |
| 0.05 | 0.078 | 0.087 | Alpha 1 adrenoreceptor antagonist | 0.087 0.049 CHEMBL3544675 0.074 0.057 CHEMBL1514176 | CHEMBL3544675 | |
| 0.045 | 0.077 | 0.068 | Alpha 1b adrenoreceptor antagonist | 0.064 0.058 CHEMBL3544675 0.068 0.054 CHEMBL1514176 | CHEMBL1514176 | |
| 0.007 | 0.038 | 0.011 | Purine nucleoside phosphorylase inhibitor | 0.011 0.01 CHEMBL1343 | CHEMBL1343 | |
| 0.011 | 0.043 | 0.023 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.023 0.005 CHEMBL3544675 | CHEMBL3544675 | |
| 0.023 | 0.059 | 0.038 | Purinergic P2X3 antagonist | 0.034 0.024 CHEMBL1343 0.038 0.019 CHEMBL1514176 | CHEMBL1514176 | |
| 0.125 | 0.167 | 0.33 | Aldehyde oxidase inhibitor | 0.266 0.076 CHEMBL3544675 0.237 0.087 CHEMBL1343 0.33 0.059 CHEMBL1514176 | CHEMBL1514176 | |
| 0.069 | 0.116 | 0.139 | Phosphodiesterase 7B inhibitor | 0.139 0.026 CHEMBL3544675 | CHEMBL3544675 | |
| 0.055 | 0.106 | 0.093 | Alpha adrenoreceptor antagonist | 0.093 0.061 CHEMBL3544675 0.078 0.073 CHEMBL1514176 | CHEMBL3544675 | |
| 0.033 | 0.083 | 0.062 | Argininosuccinate synthase inhibitor | 0.062 0.035 CHEMBL1343 | CHEMBL1343 | |
| 0.035 | 0.088 | 0.152 | Biliverdin reductase inhibitor | 0.152 0.009 CHEMBL1343 0.077 0.028 CHEMBL1514176 | CHEMBL1343 | |
| 0.025 | 0.078 | 0.07 | Antimetabolite | 0.041 0.039 CHEMBL3544675 0.07 0.022 CHEMBL1343 | CHEMBL1343 | |
| 0.121 | 0.175 | 0.14 | Ca2+-transporting ATPase inhibitor | 0.14 0.073 CHEMBL1343 | CHEMBL1343 | |
| 0.035 | 0.101 | 0.114 | Phosphofructokinase-1 inhibitor | 0.114 0.027 CHEMBL1343 | CHEMBL1343 | |
| 0.116 | 0.183 | 0.181 | ATPase inhibitor | 0.155 0.094 CHEMBL1343 0.181 0.057 CHEMBL1514176 | CHEMBL1514176 | |
| 0.109 | 0.178 | 0.144 | CF transmembrane conductance regulator agonist | 0.144 0.088 CHEMBL1343 | CHEMBL1343 | |
| 0.151 | 0.222 | 0.252 | Gastrin inhibitor | 0.252 0.076 CHEMBL1343 | CHEMBL1343 | |
| 0.051 | 0.125 | 0.126 | Antiadrenergic | 0.083 0.068 CHEMBL3544675 0.126 0.043 CHEMBL1514176 | CHEMBL1514176 | |
| 0.011 | 0.087 | 0.018 | Methylmalonyl-CoA mutase inhibitor | 0.018 0.012 CHEMBL1343 | CHEMBL1343 | |
| 0.111 | 0.188 | 0.15 | Non-steroidal antiinflammatory agent | 0.15 0.115 CHEMBL1343 0.146 0.12 CHEMBL1514176 | CHEMBL1343 | |
| 0.104 | 0.181 | 0.125 | Sphingosine 1-phosphate receptor 5 antagonist | 0.125 0.111 CHEMBL1343 | CHEMBL1343 | |
| 0.048 | 0.127 | 0.12 | Adrenaline antagonist | 0.08 0.068 CHEMBL3544675 0.12 0.043 CHEMBL1514176 | CHEMBL1514176 | |
| 0.033 | 0.123 | 0.084 | Thromboxane synthase inhibitor | 0.084 0.01 CHEMBL1343 | CHEMBL1343 | |
| 0.028 | 0.125 | 0.085 | Cyclin B inhibitor | 0.085 0.014 CHEMBL3544675 | CHEMBL3544675 | |
| 0.017 | 0.124 | 0.048 | Ornithine carbamoyltransferase inhibitor | 0.048 0.041 CHEMBL1343 | CHEMBL1343 | |
| 0.01 | 0.123 | 0.028 | Protocollagen prolyl hydroxylase inhibitor | 0.028 0.018 CHEMBL1343 | CHEMBL1343 | |
| 0.045 | 0.163 | 0.094 | ErbB-3 antagonist | 0.094 0.045 CHEMBL1343 | CHEMBL1343 | |
| 0.049 | 0.179 | 0.064 | MDM2 inhibitor | 0.064 0.06 CHEMBL1343 | CHEMBL1343 | |
| 0.05 | 0.183 | 0.201 | Ferrochelatase inhibitor | 0.201 0.022 CHEMBL1343 | CHEMBL1343 | |
| 0.023 | 0.19 | 0.042 | Glucagon-like peptide 1 receptor antagonist | 0.042 0.023 CHEMBL1343 | CHEMBL1343 | |
| 0.016 | 0.188 | 0.037 | AMPA 4 receptor antagonist | 0.037 0.032 CHEMBL1343 | CHEMBL1343 | |
| 0.035 | 0.208 | 0.085 | Alcohol dehydrogenase inhibitor | 0.085 0.072 CHEMBL1343 | CHEMBL1343 | |
| 0.122 | 0.295 | 0.204 | Peptidyltransferase inhibitor | 0.198 0.102 CHEMBL1343 0.204 0.094 CHEMBL1514176 | CHEMBL1514176 | |
| 0.018 | 0.193 | 0.053 | AICAR transformylase inhibitor | 0.053 0.019 CHEMBL1343 | CHEMBL1343 | |
| 0.043 | 0.222 | 0.093 | Cystathionine beta-synthase inhibitor | 0.093 0.086 CHEMBL1343 | CHEMBL1343 | |
| 0.082 | 0.264 | 0.169 | Platelet aggregation inhibitor | 0.169 0.107 CHEMBL1343 | CHEMBL1343 | |
| 0.02 | 0.203 | 0.086 | Cyclin B1 inhibitor | 0.086 0.017 CHEMBL3544675 | CHEMBL3544675 | |
| 0.015 | 0.202 | 0.077 | Cyclin B2 inhibitor | 0.077 0.017 CHEMBL3544675 | CHEMBL3544675 | |
| 0.007 | 0.204 | 0.036 | Histamine H3 receptor agonist | 0.036 0.015 CHEMBL3544675 | CHEMBL3544675 | |
| 0.058 | 0.26 | 0.162 | EphB2 antagonist | 0.162 0.118 CHEMBL3544675 | CHEMBL3544675 | |
| 0.032 | 0.236 | 0.084 | Myeloperoxidase inhibitor | 0.084 0.06 CHEMBL3544675 | CHEMBL3544675 | |
| 0.075 | 0.281 | 0.135 | Adenylate cyclase stimulant | 0.135 0.092 CHEMBL1343 | CHEMBL1343 | |
| 0.003 | 0.212 | 0.014 | Egl nine homolog 1 inhibitor | 0.014 0.011 CHEMBL1343 | CHEMBL1343 | |
| 0.052 | 0.262 | 0.11 | Alpha 2d adrenoreceptor antagonist | 0.11 0.033 CHEMBL3544675 | CHEMBL3544675 | |
| 0.15 | 0.36 | 0.441 | Cyclophilin D inhibitor | 0.441 0.071 CHEMBL1343 0.394 0.094 CHEMBL1514176 | CHEMBL1343 | |
| 0.067 | 0.317 | 0.326 | Insulin secretagoues | 0.208 0.032 CHEMBL1343 0.326 0.01 CHEMBL1514176 | CHEMBL1514176 | |
| 0.06 | 0.327 | 0.304 | Platelet antagonist | 0.304 0.051 CHEMBL1343 | CHEMBL1343 | |
| 0.034 | 0.301 | 0.122 | Cell adhesion molecule inhibitor | 0.122 0.023 CHEMBL1343 | CHEMBL1343 | |
| 0.032 | 0.3 | 0.191 | GABA C receptor agonist | 0.191 0.022 CHEMBL1343 | CHEMBL1343 | |
| 0.115 | 0.384 | 0.206 | Tyrosine 3 hydroxylase inhibitor | 0.206 0.125 CHEMBL1343 | CHEMBL1343 | |
| 0.048 | 0.325 | 0.087 | Hematopoietic | 0.087 0.055 CHEMBL1343 | CHEMBL1343 | |
| 0.043 | 0.325 | 0.091 | Nav1.1 sodium channel blocker | 0.091 0.079 CHEMBL1514176 | CHEMBL1514176 | |
| 0.106 | 0.392 | 0.323 | Histamine release inhibitor | 0.323 0.112 CHEMBL1343 0.235 0.167 CHEMBL1514176 | CHEMBL1343 | |
| 0.063 | 0.358 | 0.184 | Growth hormone agonist | 0.184 0.066 CHEMBL1343 | CHEMBL1343 | |
| 0.051 | 0.372 | 0.209 | Interleukin agonist | 0.207 0.114 CHEMBL1343 0.209 0.113 CHEMBL1514176 | CHEMBL1514176 | |
| 0.073 | 0.405 | 0.181 | Transcription factor STAT inhibitor | 0.181 0.166 CHEMBL1514176 | CHEMBL1514176 | |
| 0.083 | 0.445 | 0.19 | Insulysin inhibitor | 0.19 0.172 CHEMBL1343 | CHEMBL1343 | |
| 0.031 | 0.471 | 0.132 | Cell adhesion inhibitor | 0.132 0.058 CHEMBL1343 | CHEMBL1343 | |
| 0.065 | 0.702 | 0.214 | Interleukin 2 agonist | 0.214 0.166 CHEMBL1343 0.208 0.176 CHEMBL1514176 | CHEMBL1343 | |
| 0.048 | 0.688 | 0.17 | Catenin beta inhibitor | 0.17 0.066 CHEMBL1343 | CHEMBL1343 | |
| 0.028 | 0.801 | 0.093 | Folate antagonist | 0.093 0.078 CHEMBL1343 | CHEMBL1343 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |