| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.991 | 0.002 | 0.992 | Vasodilator, coronary | 0.876 0.003 CHEMBL3526986 0.86 0.003 CHEMBL3527418 0.992 0.001 CHEMBL3526948 0.989 0.002 CHEMBL1600 0.988 0.002 CHEMBL3527235 0.958 0.002 CHEMBL447626 0.957 0.002 CHEMBL3527417 0.985 0.002 CHEMBL3527058 | CHEMBL3526948 | |
| 0.894 | 0.004 | 0.894 | Cardiotonic | 0.839 0.004 CHEMBL3526986 0.852 0.004 CHEMBL3527418 0.87 0.004 CHEMBL3526948 0.864 0.004 CHEMBL1600 0.858 0.004 CHEMBL3527235 0.836 0.004 CHEMBL447626 0.831 0.004 CHEMBL3527417 0.825 0.004 CHEMBL3527058 | ||
| 0.88 | 0.003 | 0.894 | Spasmolytic | 0.66 0.008 CHEMBL3526986 0.696 0.006 CHEMBL3527418 0.883 0.003 CHEMBL3526948 0.774 0.004 CHEMBL1600 0.894 0.003 CHEMBL3527235 0.693 0.006 CHEMBL447626 0.837 0.004 CHEMBL3527417 0.797 0.004 CHEMBL3527058 | CHEMBL3527235 | |
| 0.803 | 0.005 | 0.865 | Thyroid hormone antagonist | 0.865 0.004 CHEMBL3526986 0.772 0.006 CHEMBL3527418 0.736 0.008 CHEMBL3526948 0.748 0.007 CHEMBL1600 0.775 0.006 CHEMBL3527235 0.754 0.007 CHEMBL447626 0.78 0.005 CHEMBL3527417 0.712 0.009 CHEMBL3527058 | CHEMBL3526986 | |
| 0.712 | 0.009 | 0.789 | Thyroid hormone beta antagonist | 0.789 0.005 CHEMBL3526986 0.675 0.012 CHEMBL3527418 0.623 0.016 CHEMBL3526948 0.664 0.013 CHEMBL1600 0.652 0.013 CHEMBL3527235 0.661 0.013 CHEMBL447626 0.649 0.014 CHEMBL3527417 0.6 0.018 CHEMBL3527058 | CHEMBL3526986 | |
| 0.566 | 0.008 | 0.566 | Vasodilator | 0.564 0.008 CHEMBL3526986 0.522 0.01 CHEMBL3527418 0.539 0.009 CHEMBL3526948 0.55 0.009 CHEMBL1600 0.55 0.009 CHEMBL3527235 0.497 0.012 CHEMBL447626 0.503 0.012 CHEMBL3527417 0.535 0.009 CHEMBL3527058 | ||
| 0.473 | 0.037 | 0.608 | Aldehyde oxidase inhibitor | 0.409 0.046 CHEMBL3526986 0.608 0.018 CHEMBL3527418 0.5 0.033 CHEMBL3526948 0.468 0.037 CHEMBL3527235 0.485 0.035 CHEMBL3527417 | CHEMBL3527418 | |
| 0.435 | 0.004 | 0.435 | Alpha 2b adrenoreceptor antagonist | 0.189 0.026 CHEMBL3526986 0.181 0.029 CHEMBL3527418 0.241 0.016 CHEMBL3526948 0.415 0.005 CHEMBL1600 0.165 0.033 CHEMBL3527235 0.299 0.009 CHEMBL447626 0.112 0.064 CHEMBL3527417 0.154 0.037 CHEMBL3527058 | ||
| 0.417 | 0.004 | 0.671 | Uric acid excretion stimulant | 0.671 0.003 CHEMBL3526986 0.515 0.003 CHEMBL3527418 0.417 0.004 CHEMBL3526948 0.392 0.004 CHEMBL1600 0.428 0.004 CHEMBL3527235 0.41 0.004 CHEMBL447626 0.446 0.004 CHEMBL3527417 0.403 0.004 CHEMBL3527058 | CHEMBL3526986 | |
| 0.404 | 0.016 | 0.433 | Sodium/bile acid cotransporter inhibitor | 0.433 0.01 CHEMBL3526986 0.416 0.013 CHEMBL3527418 0.397 0.018 CHEMBL3526948 0.413 0.014 CHEMBL1600 0.424 0.011 CHEMBL3527235 0.41 0.014 CHEMBL447626 0.421 0.012 CHEMBL3527417 0.43 0.01 CHEMBL3527058 | CHEMBL3526986 | |
| 0.379 | 0.002 | 0.397 | Thyroid hormone alpha antagonist | 0.367 0.002 CHEMBL3526986 0.397 0.002 CHEMBL3527418 0.324 0.002 CHEMBL3526948 0.293 0.002 CHEMBL1600 0.357 0.002 CHEMBL3527235 0.182 0.003 CHEMBL447626 0.253 0.003 CHEMBL3527417 0.274 0.002 CHEMBL3527058 | CHEMBL3527418 | |
| 0.413 | 0.061 | 0.468 | Transcription factor NF kappa B inhibitor | 0.457 0.052 CHEMBL3526986 0.464 0.05 CHEMBL3527418 0.428 0.057 CHEMBL3526948 0.341 0.08 CHEMBL1600 0.457 0.051 CHEMBL3527235 0.352 0.076 CHEMBL447626 0.468 0.049 CHEMBL3527417 0.387 0.066 CHEMBL3527058 | CHEMBL3527417 | |
| 0.362 | 0.011 | 0.509 | Protein-tyrosine phosphatase inhibitor | 0.509 0.005 CHEMBL3526986 0.434 0.007 CHEMBL3527418 0.345 0.013 CHEMBL3526948 0.34 0.013 CHEMBL1600 0.396 0.009 CHEMBL3527235 0.31 0.017 CHEMBL447626 0.36 0.011 CHEMBL3527417 0.371 0.01 CHEMBL3527058 | CHEMBL3526986 | |
| 0.374 | 0.032 | 0.374 | HERG channel blocker | 0.173 0.107 CHEMBL3527418 0.283 0.054 CHEMBL3526948 0.23 0.074 CHEMBL1600 0.168 0.111 CHEMBL3527235 | ||
| 0.324 | 0.004 | 0.324 | CYP2A6 inhibitor | 0.234 0.005 CHEMBL3526986 0.173 0.011 CHEMBL3527418 0.187 0.009 CHEMBL3526948 0.286 0.004 CHEMBL1600 0.2 0.008 CHEMBL3527235 0.203 0.007 CHEMBL447626 0.138 0.02 CHEMBL3527417 0.178 0.01 CHEMBL3527058 | ||
| 0.328 | 0.009 | 0.473 | Protein-tyrosine phosphatase 1B inhibitor | 0.473 0.005 CHEMBL3526986 0.39 0.005 CHEMBL3527418 0.305 0.01 CHEMBL3526948 0.299 0.011 CHEMBL1600 0.352 0.008 CHEMBL3527235 0.265 0.014 CHEMBL447626 0.318 0.009 CHEMBL3527417 0.328 0.009 CHEMBL3527058 | CHEMBL3526986 | |
| 0.341 | 0.035 | 0.341 | Potassium channel blocker | 0.187 0.101 CHEMBL3527418 0.264 0.06 CHEMBL3526948 0.218 0.082 CHEMBL1600 | ||
| 0.331 | 0.041 | 0.331 | Potassium channel (Voltage-sensitive) blocker | 0.151 0.136 CHEMBL3527418 0.255 0.064 CHEMBL3526948 0.215 0.085 CHEMBL1600 | ||
| 0.28 | 0.004 | 0.28 | Acetylcholine M4 receptor antagonist | 0.103 0.026 CHEMBL3526986 0.131 0.014 CHEMBL3527418 0.186 0.007 CHEMBL3526948 0.137 0.013 CHEMBL1600 0.106 0.024 CHEMBL3527235 0.1 0.028 CHEMBL447626 0.078 0.048 CHEMBL3527417 | ||
| 0.302 | 0.029 | 0.302 | P-glycoprotein inhibitor | 0.231 0.048 CHEMBL3526986 0.298 0.029 CHEMBL3527418 0.298 0.029 CHEMBL3526948 0.257 0.039 CHEMBL1600 0.28 0.033 CHEMBL3527235 0.218 0.054 CHEMBL447626 0.239 0.045 CHEMBL3527417 0.243 0.043 CHEMBL3527058 | ||
| 0.334 | 0.061 | 0.334 | Calcium channel activator | 0.266 0.128 CHEMBL3526986 0.325 0.068 CHEMBL3526948 0.293 0.099 CHEMBL1600 0.316 0.076 CHEMBL3527235 0.295 0.097 CHEMBL447626 0.318 0.075 CHEMBL3527417 0.273 0.12 CHEMBL3527058 | ||
| 0.303 | 0.032 | 0.421 | Tyrosine 3 hydroxylase inhibitor | 0.421 0.006 CHEMBL3526986 0.258 0.061 CHEMBL3527418 0.281 0.044 CHEMBL3526948 0.243 0.075 CHEMBL1600 0.383 0.01 CHEMBL3527235 0.246 0.072 CHEMBL447626 0.386 0.01 CHEMBL3527417 0.309 0.029 CHEMBL3527058 | CHEMBL3526986 | |
| 0.279 | 0.049 | 0.335 | Amyloid beta aggregation inhibitor | 0.294 0.046 CHEMBL3526986 0.231 0.064 CHEMBL3527418 0.335 0.038 CHEMBL3526948 0.236 0.062 CHEMBL1600 0.27 0.052 CHEMBL3527235 0.246 0.059 CHEMBL447626 0.278 0.05 CHEMBL3527417 0.233 0.063 CHEMBL3527058 | CHEMBL3526948 | |
| 0.241 | 0.02 | 0.241 | 5 Hydroxytryptamine 2B antagonist | 0.119 0.062 CHEMBL3526986 0.117 0.063 CHEMBL3527418 0.142 0.044 CHEMBL3526948 0.147 0.042 CHEMBL1600 0.096 0.089 CHEMBL3527235 0.154 0.039 CHEMBL447626 0.101 0.083 CHEMBL3527417 | ||
| 0.24 | 0.022 | 0.24 | Anesthetic local | 0.199 0.033 CHEMBL3526948 0.162 0.044 CHEMBL1600 0.111 0.074 CHEMBL3527235 0.171 0.041 CHEMBL447626 0.117 0.069 CHEMBL3527417 | ||
| 0.297 | 0.093 | 0.571 | Cholesterol antagonist | 0.571 0.022 CHEMBL3526986 0.404 0.048 CHEMBL3527418 0.308 0.086 CHEMBL3526948 0.309 0.086 CHEMBL1600 0.444 0.041 CHEMBL3527235 0.316 0.081 CHEMBL447626 0.458 0.039 CHEMBL3527417 0.467 0.038 CHEMBL3527058 | CHEMBL3526986 | |
| 0.266 | 0.062 | 0.361 | Free radical scavenger | 0.361 0.036 CHEMBL3526986 0.277 0.058 CHEMBL3527418 0.277 0.058 CHEMBL3526948 0.25 0.069 CHEMBL1600 0.304 0.051 CHEMBL3527235 0.224 0.081 CHEMBL447626 0.274 0.059 CHEMBL3527417 0.285 0.056 CHEMBL3527058 | CHEMBL3526986 | |
| 0.336 | 0.148 | 0.47 | Apoptosis agonist | 0.47 0.084 CHEMBL3526986 0.402 0.113 CHEMBL3527418 0.328 0.153 CHEMBL3526948 0.326 0.155 CHEMBL1600 0.338 0.146 CHEMBL3527235 0.258 0.205 CHEMBL447626 0.277 0.189 CHEMBL3527417 0.329 0.152 CHEMBL3527058 | CHEMBL3526986 | |
| 0.222 | 0.034 | 0.222 | Acetylcholine M1 receptor antagonist | 0.124 0.102 CHEMBL3527418 0.203 0.041 CHEMBL3526948 0.163 0.064 CHEMBL1600 0.155 0.07 CHEMBL3527235 0.123 0.105 CHEMBL447626 0.116 0.114 CHEMBL3527417 | ||
| 0.267 | 0.086 | 0.519 | Hypoxia-inducible factor 1 alpha inhibitor | 0.519 0.013 CHEMBL3526986 0.247 0.104 CHEMBL3527418 0.235 0.114 CHEMBL3526948 0.194 0.159 CHEMBL1600 0.303 0.064 CHEMBL3527235 0.2 0.152 CHEMBL447626 0.31 0.061 CHEMBL3527417 0.224 0.125 CHEMBL3527058 | CHEMBL3526986 | |
| 0.202 | 0.036 | 0.263 | Tubulin antagonist | 0.263 0.024 CHEMBL3526986 0.263 0.024 CHEMBL3527418 0.182 0.043 CHEMBL3526948 0.2 0.037 CHEMBL1600 0.169 0.049 CHEMBL3527235 0.174 0.047 CHEMBL447626 0.143 0.062 CHEMBL3527417 0.169 0.049 CHEMBL3527058 | CHEMBL3527418 | |
| 0.273 | 0.108 | 0.418 | Antithrombotic | 0.293 0.093 CHEMBL3526986 0.309 0.083 CHEMBL3527418 0.275 0.107 CHEMBL3526948 0.195 0.184 CHEMBL1600 0.418 0.045 CHEMBL3527235 0.192 0.188 CHEMBL447626 0.413 0.046 CHEMBL3527417 0.312 0.08 CHEMBL3527058 | CHEMBL3527235 | |
| 0.167 | 0.005 | 0.24 | Beta adrenoreceptor antagonist | 0.147 0.006 CHEMBL3526986 0.179 0.004 CHEMBL3527418 0.186 0.004 CHEMBL3526948 0.227 0.004 CHEMBL1600 0.159 0.005 CHEMBL3527235 0.24 0.003 CHEMBL447626 0.167 0.005 CHEMBL3527417 0.214 0.004 CHEMBL3527058 | CHEMBL447626 | |
| 0.202 | 0.051 | 0.294 | Thrombolytic | 0.262 0.031 CHEMBL3526986 0.264 0.03 CHEMBL3527418 0.211 0.047 CHEMBL3526948 0.219 0.043 CHEMBL1600 0.267 0.03 CHEMBL3527235 0.245 0.035 CHEMBL447626 0.294 0.025 CHEMBL3527417 0.284 0.027 CHEMBL3527058 | CHEMBL3527417 | |
| 0.164 | 0.013 | 0.164 | Dopamine D1 antagonist | 0.142 0.016 CHEMBL3526986 0.092 0.028 CHEMBL3527418 0.16 0.014 CHEMBL3526948 0.092 0.028 CHEMBL1600 0.07 0.04 CHEMBL3527235 0.064 0.045 CHEMBL447626 | ||
| 0.154 | 0.01 | 0.253 | Purinergic P2X2 antagonist | 0.195 0.005 CHEMBL3526986 0.188 0.005 CHEMBL3527418 0.157 0.01 CHEMBL3526948 0.151 0.011 CHEMBL1600 0.139 0.014 CHEMBL3527235 0.253 0.003 CHEMBL447626 0.24 0.003 CHEMBL3527417 0.137 0.015 CHEMBL3527058 | CHEMBL447626 | |
| 0.183 | 0.04 | 0.244 | Hemostatic | 0.128 0.099 CHEMBL3526986 0.176 0.044 CHEMBL3527418 0.192 0.036 CHEMBL3526948 0.123 0.108 CHEMBL1600 0.244 0.023 CHEMBL3527235 0.16 0.057 CHEMBL3527417 0.157 0.06 CHEMBL3527058 | CHEMBL3527235 | |
| 0.301 | 0.164 | 0.416 | 5 Hydroxytryptamine release inhibitor | 0.362 0.105 CHEMBL3526986 0.416 0.068 CHEMBL3527418 0.294 0.172 CHEMBL3526948 0.252 0.225 CHEMBL3527235 0.255 0.221 CHEMBL3527417 | CHEMBL3527418 | |
| 0.154 | 0.018 | 0.204 | Electron transport complex I inhibitor | 0.204 0.008 CHEMBL3526986 0.169 0.013 CHEMBL3527418 0.139 0.028 CHEMBL3526948 0.148 0.022 CHEMBL1600 0.117 0.051 CHEMBL3527235 0.149 0.021 CHEMBL447626 0.119 0.049 CHEMBL3527417 0.113 0.057 CHEMBL3527058 | CHEMBL3526986 | |
| 0.144 | 0.008 | 0.144 | Acetylcholine M5 receptor antagonist | 0.074 0.027 CHEMBL3526986 0.088 0.021 CHEMBL3527418 0.125 0.012 CHEMBL3526948 0.123 0.012 CHEMBL1600 0.062 0.039 CHEMBL3527235 0.083 0.023 CHEMBL447626 0.054 0.052 CHEMBL3527058 | ||
| 0.195 | 0.06 | 0.25 | Lipocortins synthesis antagonist | 0.198 0.058 CHEMBL3526948 0.25 0.033 CHEMBL3527235 0.238 0.038 CHEMBL3527417 | CHEMBL3527235 | |
| 0.139 | 0.005 | 0.243 | Plasminogen activator inhibitor antagonist | 0.243 0.004 CHEMBL3526986 0.192 0.004 CHEMBL3527418 0.136 0.005 CHEMBL3526948 0.135 0.005 CHEMBL1600 0.189 0.004 CHEMBL3527235 0.168 0.005 CHEMBL447626 0.224 0.004 CHEMBL3527417 0.183 0.004 CHEMBL3527058 | CHEMBL3526986 | |
| 0.155 | 0.023 | 0.155 | Multidrug resistance-associated protein 1 inhibitor | 0.138 0.032 CHEMBL3526986 0.152 0.024 CHEMBL3527418 0.144 0.028 CHEMBL3526948 0.13 0.038 CHEMBL1600 0.141 0.03 CHEMBL3527235 0.13 0.038 CHEMBL447626 0.14 0.031 CHEMBL3527417 0.121 0.047 CHEMBL3527058 | ||
| 0.138 | 0.014 | 0.182 | Adenosine A3 receptor antagonist | 0.149 0.013 CHEMBL3526986 0.129 0.015 CHEMBL3527418 0.086 0.036 CHEMBL3526948 0.182 0.01 CHEMBL1600 0.087 0.035 CHEMBL3527235 0.128 0.016 CHEMBL447626 0.067 0.063 CHEMBL3527417 0.107 0.023 CHEMBL3527058 | CHEMBL1600 | |
| 0.148 | 0.027 | 0.148 | 5 Hydroxytryptamine 2C antagonist | 0.093 0.051 CHEMBL3526948 0.112 0.039 CHEMBL1600 0.121 0.035 CHEMBL447626 | ||
| 0.288 | 0.168 | 0.435 | Calcium channel L-type activator | 0.435 0.059 CHEMBL3526986 0.38 0.095 CHEMBL3527418 0.324 0.137 CHEMBL3526948 0.332 0.131 CHEMBL1600 0.328 0.134 CHEMBL3527235 0.345 0.121 CHEMBL447626 0.339 0.126 CHEMBL3527417 0.361 0.109 CHEMBL3527058 | CHEMBL3526986 | |
| 0.132 | 0.013 | 0.132 | Calcium channel L-type blocker | 0.078 0.042 CHEMBL3527418 0.1 0.025 CHEMBL3526948 0.099 0.025 CHEMBL1600 0.089 0.031 CHEMBL3527235 0.076 0.044 CHEMBL447626 0.068 0.055 CHEMBL3527417 0.067 0.057 CHEMBL3527058 | ||
| 0.16 | 0.042 | 0.283 | Aldehyde dehydrogenase inhibitor | 0.181 0.033 CHEMBL3526986 0.283 0.013 CHEMBL3527418 0.238 0.02 CHEMBL3526948 0.223 0.023 CHEMBL3527235 0.228 0.022 CHEMBL3527417 0.114 0.077 CHEMBL3527058 | CHEMBL3527418 | |
| 0.195 | 0.078 | 0.195 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.159 0.12 CHEMBL3527418 0.188 0.085 CHEMBL3526948 0.171 0.105 CHEMBL1600 0.17 0.107 CHEMBL3527235 0.148 0.136 CHEMBL3527058 | ||
| 0.139 | 0.025 | 0.139 | Alpha 2a adrenoreceptor antagonist | 0.12 0.029 CHEMBL1600 0.074 0.054 CHEMBL447626 | ||
| 0.215 | 0.104 | 0.295 | Antioxidant | 0.295 0.064 CHEMBL3526986 0.243 0.088 CHEMBL3527418 0.242 0.088 CHEMBL3526948 0.195 0.117 CHEMBL1600 0.259 0.079 CHEMBL3527235 0.182 0.13 CHEMBL447626 0.244 0.087 CHEMBL3527417 0.242 0.088 CHEMBL3527058 | CHEMBL3526986 | |
| 0.129 | 0.018 | 0.129 | Dopamine D3 antagonist | 0.075 0.035 CHEMBL3526948 0.114 0.021 CHEMBL1600 0.078 0.034 CHEMBL447626 | ||
| 0.125 | 0.015 | 0.125 | Acetylcholine M2 receptor antagonist | 0.093 0.023 CHEMBL3526948 0.078 0.03 CHEMBL1600 0.054 0.05 CHEMBL447626 | ||
| 0.119 | 0.01 | 0.14 | Beta 3 adrenoreceptor antagonist | 0.073 0.03 CHEMBL3526986 0.089 0.018 CHEMBL3527418 0.127 0.009 CHEMBL3526948 0.14 0.007 CHEMBL1600 0.092 0.017 CHEMBL3527235 0.12 0.01 CHEMBL447626 0.076 0.027 CHEMBL3527417 0.115 0.011 CHEMBL3527058 | CHEMBL1600 | |
| 0.126 | 0.018 | 0.136 | Histamine H2 receptor antagonist | 0.093 0.043 CHEMBL3526948 0.132 0.015 CHEMBL1600 0.136 0.014 CHEMBL447626 0.077 0.073 CHEMBL3527058 | CHEMBL447626 | |
| 0.148 | 0.045 | 0.148 | 5 Hydroxytryptamine 2 antagonist | 0.103 0.069 CHEMBL3526948 0.113 0.064 CHEMBL1600 0.132 0.052 CHEMBL447626 | ||
| 0.188 | 0.091 | 0.228 | Antimitotic | 0.15 0.121 CHEMBL3526986 0.228 0.069 CHEMBL3527418 0.18 0.096 CHEMBL3526948 0.171 0.102 CHEMBL1600 0.154 0.117 CHEMBL3527235 0.143 0.129 CHEMBL3527058 | CHEMBL3527418 | |
| 0.134 | 0.043 | 0.293 | Photosensitizer | 0.254 0.005 CHEMBL3526986 0.293 0.004 CHEMBL3527418 0.144 0.035 CHEMBL3526948 0.147 0.033 CHEMBL1600 0.18 0.018 CHEMBL3527235 0.133 0.043 CHEMBL447626 0.162 0.025 CHEMBL3527417 0.198 0.013 CHEMBL3527058 | CHEMBL3527418 | |
| 0.15 | 0.059 | 0.15 | Calcium channel blocker | 0.132 0.075 CHEMBL1600 | ||
| 0.129 | 0.039 | 0.152 | Estrogen antagonist | 0.152 0.022 CHEMBL3526986 0.122 0.051 CHEMBL3527418 0.132 0.036 CHEMBL3526948 0.115 0.064 CHEMBL1600 0.127 0.043 CHEMBL3527235 0.118 0.058 CHEMBL447626 0.129 0.04 CHEMBL3527417 0.114 0.066 CHEMBL3527058 | CHEMBL3526986 | |
| 0.202 | 0.112 | 0.253 | Calpain inhibitor | 0.22 0.095 CHEMBL3526986 0.253 0.062 CHEMBL1600 0.253 0.062 CHEMBL447626 0.185 0.128 CHEMBL3527058 | CHEMBL447626 | |
| 0.114 | 0.024 | 0.129 | ATPase (Vacuolar H+) inhibitor | 0.129 0.014 CHEMBL3526986 0.119 0.02 CHEMBL3527418 0.113 0.025 CHEMBL3526948 0.107 0.031 CHEMBL1600 0.113 0.025 CHEMBL3527235 0.106 0.032 CHEMBL447626 0.112 0.026 CHEMBL3527417 0.107 0.031 CHEMBL3527058 | CHEMBL3526986 | |
| 0.128 | 0.042 | 0.22 | Antiadrenergic | 0.116 0.047 CHEMBL3526948 0.22 0.021 CHEMBL1600 0.079 0.072 CHEMBL3527235 0.208 0.023 CHEMBL447626 0.076 0.075 CHEMBL3527417 0.148 0.036 CHEMBL3527058 | CHEMBL1600 | |
| 0.178 | 0.094 | 0.308 | Psychostimulant | 0.182 0.091 CHEMBL3526948 0.164 0.104 CHEMBL1600 0.219 0.07 CHEMBL3527235 0.237 0.063 CHEMBL447626 0.308 0.041 CHEMBL3527417 0.201 0.079 CHEMBL3527058 | CHEMBL3527417 | |
| 0.163 | 0.08 | 0.231 | ATPase inhibitor | 0.231 0.019 CHEMBL3526986 0.135 0.131 CHEMBL3527418 0.169 0.072 CHEMBL3526948 0.148 0.104 CHEMBL3527235 0.144 0.113 CHEMBL3527417 | CHEMBL3526986 | |
| 0.198 | 0.117 | 0.302 | DNA damaging | 0.185 0.129 CHEMBL3526986 0.209 0.108 CHEMBL3527418 0.214 0.105 CHEMBL3526948 0.212 0.106 CHEMBL1600 0.23 0.093 CHEMBL3527235 0.281 0.065 CHEMBL447626 0.302 0.056 CHEMBL3527417 0.244 0.084 CHEMBL3527058 | CHEMBL3527417 | |
| 0.181 | 0.104 | 0.22 | 5 Hydroxytryptamine 3E antagonist | 0.22 0.037 CHEMBL1600 0.219 0.037 CHEMBL447626 | CHEMBL1600 | |
| 0.115 | 0.038 | 0.115 | Alpha 2 adrenoreceptor antagonist | 0.107 0.043 CHEMBL1600 | ||
| 0.181 | 0.11 | 0.181 | Cyclic AMP phosphodiesterase inhibitor | 0.162 0.133 CHEMBL3526948 | ||
| 0.089 | 0.022 | 0.089 | Dopamine uptake inhibitor | 0.059 0.039 CHEMBL3526986 0.062 0.037 CHEMBL3526948 0.07 0.03 CHEMBL1600 0.075 0.027 CHEMBL447626 | ||
| 0.135 | 0.072 | 0.179 | Bone formation stimulant | 0.139 0.068 CHEMBL3526986 0.145 0.063 CHEMBL3527418 0.179 0.042 CHEMBL3526948 0.125 0.081 CHEMBL1600 0.174 0.044 CHEMBL3527235 0.125 0.081 CHEMBL447626 0.171 0.045 CHEMBL3527417 0.163 0.05 CHEMBL3527058 | CHEMBL3526948 | |
| 0.07 | 0.008 | 0.07 | Sigma 1 receptor antagonist | 0.033 0.016 CHEMBL3526986 0.037 0.014 CHEMBL3526948 0.031 0.017 CHEMBL1600 0.061 0.009 CHEMBL447626 0.043 0.012 CHEMBL3527417 | ||
| 0.094 | 0.034 | 0.105 | Interferon agonist | 0.105 0.025 CHEMBL3526948 0.091 0.038 CHEMBL3527235 0.084 0.046 CHEMBL3527417 | CHEMBL3526948 | |
| 0.108 | 0.049 | 0.204 | Adrenaline antagonist | 0.1 0.054 CHEMBL3526948 0.204 0.023 CHEMBL1600 0.192 0.025 CHEMBL447626 0.133 0.04 CHEMBL3527058 | CHEMBL1600 | |
| 0.116 | 0.058 | 0.157 | Chelator | 0.107 0.067 CHEMBL3526986 0.099 0.079 CHEMBL3527418 0.15 0.035 CHEMBL3526948 0.096 0.084 CHEMBL1600 0.157 0.033 CHEMBL3527235 0.097 0.082 CHEMBL447626 0.155 0.034 CHEMBL3527417 0.128 0.047 CHEMBL3527058 | CHEMBL3527235 | |
| 0.085 | 0.027 | 0.129 | Peroxisome proliferator-activated receptor gamma antagonist | 0.098 0.017 CHEMBL3526986 0.112 0.011 CHEMBL3527418 0.082 0.031 CHEMBL3526948 0.083 0.03 CHEMBL1600 0.119 0.01 CHEMBL3527235 0.087 0.025 CHEMBL447626 0.129 0.008 CHEMBL3527417 0.113 0.011 CHEMBL3527058 | CHEMBL3527417 | |
| 0.092 | 0.04 | 0.13 | Somatostatin 1 agonist | 0.13 0.019 CHEMBL3526986 0.103 0.032 CHEMBL3527418 0.09 0.041 CHEMBL3526948 0.095 0.037 CHEMBL1600 0.087 0.044 CHEMBL3527235 0.095 0.037 CHEMBL447626 0.087 0.044 CHEMBL3527417 0.09 0.041 CHEMBL3527058 | CHEMBL3526986 | |
| 0.151 | 0.1 | 0.248 | Amyloid beta precursor protein antagonist | 0.239 0.037 CHEMBL3526986 0.248 0.034 CHEMBL3527418 0.172 0.079 CHEMBL3526948 0.151 0.1 CHEMBL1600 0.156 0.095 CHEMBL3527235 0.153 0.098 CHEMBL447626 0.157 0.093 CHEMBL3527417 0.156 0.095 CHEMBL3527058 | CHEMBL3527418 | |
| 0.131 | 0.08 | 0.283 | Farnesoid X receptor antagonist | 0.283 0.007 CHEMBL3526986 0.164 0.039 CHEMBL3527418 0.168 0.036 CHEMBL3526948 0.128 0.085 CHEMBL1600 0.15 0.052 CHEMBL3527235 0.13 0.082 CHEMBL447626 0.151 0.051 CHEMBL3527417 0.147 0.056 CHEMBL3527058 | CHEMBL3526986 | |
| 0.073 | 0.023 | 0.117 | Beta 1 adrenoreceptor antagonist | 0.059 0.037 CHEMBL3526986 0.092 0.012 CHEMBL3527418 0.075 0.021 CHEMBL3526948 0.11 0.008 CHEMBL1600 0.062 0.033 CHEMBL3527235 0.117 0.007 CHEMBL447626 0.067 0.029 CHEMBL3527417 0.094 0.011 CHEMBL3527058 | CHEMBL447626 | |
| 0.071 | 0.023 | 0.071 | Sigma receptor antagonist | 0.052 0.033 CHEMBL3526986 0.052 0.033 CHEMBL3526948 0.041 0.04 CHEMBL1600 0.064 0.026 CHEMBL447626 0.047 0.036 CHEMBL3527417 | ||
| 0.086 | 0.04 | 0.099 | Estrogen receptor alpha antagonist | 0.099 0.027 CHEMBL3526986 0.083 0.044 CHEMBL3527418 0.086 0.04 CHEMBL3526948 0.079 0.051 CHEMBL3527235 0.072 0.064 CHEMBL447626 0.083 0.045 CHEMBL3527417 | CHEMBL3526986 | |
| 0.098 | 0.053 | 0.125 | ABCA1 expression enhancer | 0.125 0.028 CHEMBL3526986 0.117 0.033 CHEMBL3527418 0.105 0.044 CHEMBL3526948 0.089 0.067 CHEMBL1600 0.112 0.037 CHEMBL3527235 0.09 0.065 CHEMBL447626 0.112 0.037 CHEMBL3527417 0.103 0.046 CHEMBL3527058 | CHEMBL3526986 | |
| 0.094 | 0.05 | 0.094 | 5 Hydroxytryptamine 2A antagonist | 0.073 0.064 CHEMBL447626 | ||
| 0.095 | 0.051 | 0.142 | Aminoacyl-tRNA synthetase inhibitor | 0.122 0.029 CHEMBL3526986 0.142 0.021 CHEMBL3527418 0.114 0.034 CHEMBL3526948 0.101 0.044 CHEMBL1600 0.106 0.039 CHEMBL3527235 0.097 0.049 CHEMBL447626 0.102 0.043 CHEMBL3527417 0.111 0.035 CHEMBL3527058 | CHEMBL3527418 | |
| 0.094 | 0.051 | 0.094 | Histamine N-methyltransferase inhibitor | 0.082 0.064 CHEMBL3526948 | ||
| 0.082 | 0.039 | 0.082 | Dopamine D2 antagonist | 0.075 0.041 CHEMBL1600 | ||
| 0.114 | 0.073 | 0.114 | Acetylcholine muscarinic antagonist | 0.112 0.076 CHEMBL3526948 | ||
| 0.102 | 0.061 | 0.132 | Estrogen receptor beta antagonist | 0.132 0.022 CHEMBL3526986 0.098 0.069 CHEMBL3527418 0.103 0.059 CHEMBL3526948 0.099 0.066 CHEMBL3527235 0.102 0.061 CHEMBL3527417 | CHEMBL3526986 | |
| 0.083 | 0.046 | 0.083 | Dopamine antagonist | 0.074 0.051 CHEMBL1600 | ||
| 0.079 | 0.042 | 0.133 | Peroxisome proliferator-activated receptor gamma agonist | 0.127 0.018 CHEMBL3526986 0.122 0.019 CHEMBL3527418 0.075 0.044 CHEMBL3526948 0.075 0.045 CHEMBL1600 0.119 0.02 CHEMBL3527235 0.088 0.035 CHEMBL447626 0.133 0.017 CHEMBL3527417 0.112 0.022 CHEMBL3527058 | CHEMBL3527417 | |
| 0.049 | 0.012 | 0.055 | 2,3-Oxidosqualene-lanosterol cyclase inhibitor | 0.055 0.009 CHEMBL3526948 | CHEMBL3526948 | |
| 0.062 | 0.027 | 0.115 | Thromboxane A2 antagonist | 0.087 0.012 CHEMBL3526986 0.102 0.007 CHEMBL3527418 0.076 0.017 CHEMBL3526948 0.064 0.025 CHEMBL1600 0.111 0.005 CHEMBL3527235 0.043 0.042 CHEMBL447626 0.092 0.01 CHEMBL3527417 0.115 0.005 CHEMBL3527058 | CHEMBL3527058 | |
| 0.035 | 0.004 | 0.291 | Thyroid hormone alpha agonist | 0.291 0.001 CHEMBL3526986 0.046 0.003 CHEMBL3527418 0.032 0.004 CHEMBL3526948 0.033 0.004 CHEMBL1600 0.042 0.003 CHEMBL3527235 0.032 0.004 CHEMBL447626 0.04 0.003 CHEMBL3527417 0.039 0.003 CHEMBL3527058 | CHEMBL3526986 | |
| 0.131 | 0.101 | 0.131 | Sigma receptor agonist | |||
| 0.094 | 0.066 | 0.215 | Xanthine oxidase inhibitor | 0.215 0.017 CHEMBL3526986 0.185 0.023 CHEMBL3527418 0.094 0.066 CHEMBL3526948 0.12 0.047 CHEMBL3527235 0.094 0.066 CHEMBL447626 0.171 0.027 CHEMBL3527417 0.085 0.08 CHEMBL3527058 | CHEMBL3526986 | |
| 0.089 | 0.065 | 0.089 | Antihistaminic | 0.086 0.07 CHEMBL447626 | ||
| 0.109 | 0.085 | 0.109 | Cholinergic antagonist | 0.105 0.089 CHEMBL3526948 | ||
| 0.058 | 0.034 | 0.128 | Thromboxane antagonist | 0.09 0.015 CHEMBL3526986 0.107 0.009 CHEMBL3527418 0.077 0.022 CHEMBL3526948 0.066 0.028 CHEMBL1600 0.117 0.007 CHEMBL3527235 0.097 0.012 CHEMBL3527417 0.128 0.006 CHEMBL3527058 | CHEMBL3527058 | |
| 0.054 | 0.031 | 0.1 | Beta 2 adrenoreceptor antagonist | 0.07 0.017 CHEMBL3526986 0.076 0.013 CHEMBL3527418 0.054 0.03 CHEMBL3526948 0.092 0.009 CHEMBL1600 0.048 0.039 CHEMBL3527235 0.1 0.008 CHEMBL447626 0.052 0.034 CHEMBL3527417 0.083 0.011 CHEMBL3527058 | CHEMBL447626 | |
| 0.196 | 0.174 | 0.208 | Angiogenesis inhibitor | 0.203 0.166 CHEMBL3527418 0.208 0.16 CHEMBL3526948 0.196 0.174 CHEMBL1600 0.193 0.178 CHEMBL3527235 0.193 0.178 CHEMBL3527058 | CHEMBL3526948 | |
| 0.043 | 0.021 | 0.1 | Retinoid X receptor agonist | 0.1 0.005 CHEMBL3526986 0.072 0.01 CHEMBL3527418 0.042 0.021 CHEMBL3526948 0.085 0.007 CHEMBL3527235 0.083 0.007 CHEMBL3527417 0.064 0.012 CHEMBL3527058 | CHEMBL3526986 | |
| 0.036 | 0.017 | 0.039 | Calcium-independent phospholipase A2 inhibitor | 0.039 0.012 CHEMBL3526986 0.039 0.011 CHEMBL3527418 0.034 0.023 CHEMBL3526948 0.036 0.017 CHEMBL1600 0.035 0.02 CHEMBL3527235 0.037 0.017 CHEMBL447626 0.035 0.02 CHEMBL3527417 0.035 0.02 CHEMBL3527058 | CHEMBL3527418 | |
| 0.09 | 0.072 | 0.09 | Sphingomyelinase inhibitor | |||
| 0.104 | 0.087 | 0.104 | Acetylcholine antagonist | 0.101 0.092 CHEMBL3526948 | ||
| 0.104 | 0.087 | 0.119 | MAO inhibitor | 0.1 0.09 CHEMBL3526948 0.119 0.075 CHEMBL447626 | CHEMBL447626 | |
| 0.058 | 0.043 | 0.059 | Acetylcholine M3 receptor antagonist | 0.059 0.043 CHEMBL3526948 | CHEMBL3526948 | |
| 0.038 | 0.025 | 0.038 | Delayed rectifier potassium channel blocker | |||
| 0.062 | 0.049 | 0.068 | Interferon inducer | 0.068 0.037 CHEMBL3526948 | CHEMBL3526948 | |
| 0.028 | 0.015 | 0.077 | Thyroid hormone agonist | 0.073 0.003 CHEMBL3526986 0.034 0.009 CHEMBL3527418 0.03 0.012 CHEMBL3526948 0.024 0.022 CHEMBL1600 0.056 0.004 CHEMBL3527235 0.032 0.011 CHEMBL447626 0.077 0.003 CHEMBL3527417 0.047 0.005 CHEMBL3527058 | CHEMBL3527417 | |
| 0.078 | 0.066 | 0.078 | Histamine antagonist | 0.075 0.07 CHEMBL447626 | ||
| 0.033 | 0.025 | 0.053 | Melatonin receptor 1A agonist | 0.031 0.03 CHEMBL3526986 0.034 0.021 CHEMBL3527418 0.05 0.008 CHEMBL1600 0.053 0.007 CHEMBL447626 | CHEMBL447626 | |
| 0.026 | 0.018 | 0.03 | Complement factor 1r inhibitor | 0.03 0.011 CHEMBL3526986 0.026 0.018 CHEMBL3527418 0.026 0.018 CHEMBL1600 0.026 0.018 CHEMBL447626 | CHEMBL3526986 | |
| 0.094 | 0.088 | 0.231 | DOPA decarboxylase inhibitor | 0.231 0.004 CHEMBL3526986 0.164 0.015 CHEMBL3527418 0.11 0.059 CHEMBL3526948 0.121 0.044 CHEMBL3527235 0.124 0.041 CHEMBL3527417 0.116 0.05 CHEMBL3527058 | CHEMBL3526986 | |
| 0.047 | 0.041 | 0.049 | Squalene epoxidase inhibitor | 0.049 0.037 CHEMBL3526948 | CHEMBL3526948 | |
| 0.025 | 0.024 | 0.037 | Melatonin antagonist | 0.027 0.021 CHEMBL3526986 0.037 0.011 CHEMBL1600 0.036 0.012 CHEMBL447626 | CHEMBL1600 | |
| 0.016 | 0.017 | 0.025 | Melatonin 1 antagonist | 0.018 0.014 CHEMBL3526986 0.025 0.008 CHEMBL1600 0.025 0.008 CHEMBL447626 | CHEMBL447626 | |
| 0.075 | 0.076 | 0.09 | Alpha adrenoreceptor antagonist | 0.09 0.063 CHEMBL1600 | CHEMBL1600 | |
| 0.012 | 0.013 | 0.039 | Melatonin receptor 1A antagonist | 0.034 0.004 CHEMBL1600 0.039 0.004 CHEMBL447626 | CHEMBL447626 | |
| 0.084 | 0.087 | 0.096 | Electrolyte absorption antagonist | 0.096 0.064 CHEMBL3527235 0.09 0.075 CHEMBL3527417 | CHEMBL3527235 | |
| 0.013 | 0.017 | 0.018 | 4-Hydroxyphenylpyruvate dioxygenase inhibitor | 0.018 0.005 CHEMBL3526986 0.015 0.01 CHEMBL3527418 | CHEMBL3526986 | |
| 0.027 | 0.031 | 0.031 | Elastase 3B inhibitor | 0.031 0.021 CHEMBL3526986 0.029 0.027 CHEMBL3527417 | CHEMBL3526986 | |
| 0.027 | 0.031 | 0.031 | Elastase 2B inhibitor | 0.031 0.021 CHEMBL3526986 0.029 0.027 CHEMBL3527417 | CHEMBL3526986 | |
| 0.027 | 0.031 | 0.031 | Elastase 3A inhibitor | 0.031 0.021 CHEMBL3526986 0.029 0.027 CHEMBL3527417 | CHEMBL3526986 | |
| 0.051 | 0.055 | 0.054 | Acetyl-CoA transferase 2 inhibitor | 0.054 0.045 CHEMBL3526986 | CHEMBL3526986 | |
| 0.035 | 0.039 | 0.05 | Growth hormone release inhibitor | 0.05 0.022 CHEMBL3526986 0.041 0.03 CHEMBL3527418 0.037 0.036 CHEMBL1600 | CHEMBL3526986 | |
| 0.048 | 0.054 | 0.093 | Thromboxane synthase inhibitor | 0.056 0.035 CHEMBL3526986 0.073 0.015 CHEMBL3527418 0.059 0.029 CHEMBL3526948 0.051 0.045 CHEMBL1600 0.086 0.009 CHEMBL3527235 0.069 0.018 CHEMBL3527417 0.093 0.008 CHEMBL3527058 | CHEMBL3527058 | |
| 0.161 | 0.169 | 0.183 | Superoxide dismutase inhibitor | 0.177 0.145 CHEMBL3526986 0.183 0.137 CHEMBL3526948 | CHEMBL3526948 | |
| 0.063 | 0.071 | 0.143 | Glycine receptor agonist | 0.143 0.008 CHEMBL3526986 0.1 0.021 CHEMBL3527418 0.068 0.059 CHEMBL3526948 0.083 0.035 CHEMBL3527235 0.073 0.05 CHEMBL3527417 0.068 0.058 CHEMBL3527058 | CHEMBL3526986 | |
| 0.046 | 0.055 | 0.073 | Leukotriene B4 antagonist | 0.059 0.029 CHEMBL3526986 0.063 0.025 CHEMBL3527418 0.052 0.04 CHEMBL3526948 0.068 0.021 CHEMBL3527235 0.073 0.018 CHEMBL3527417 0.052 0.04 CHEMBL3527058 | CHEMBL3527417 | |
| 0.045 | 0.054 | 0.055 | Dopamine D4 antagonist | 0.055 0.045 CHEMBL1600 | CHEMBL1600 | |
| 0.032 | 0.042 | 0.041 | Histamine H3 receptor antagonist | 0.041 0.033 CHEMBL447626 | CHEMBL447626 | |
| 0.056 | 0.071 | 0.061 | Potassium channel (ATP-sensitive) blocker | 0.061 0.059 CHEMBL3527418 | CHEMBL3527418 | |
| 0.075 | 0.09 | 0.117 | Breast cancer-resistant protein inhibitor | 0.117 0.041 CHEMBL3526986 0.114 0.044 CHEMBL3527418 | CHEMBL3526986 | |
| 0.056 | 0.071 | 0.063 | Beta 2 adrenoreceptor agonist | 0.059 0.054 CHEMBL3527418 0.061 0.045 CHEMBL3526948 0.063 0.037 CHEMBL1600 0.059 0.054 CHEMBL447626 0.058 0.057 CHEMBL3527058 | CHEMBL1600 | |
| 0.024 | 0.04 | 0.038 | Melatonin 2 agonist | 0.038 0.018 CHEMBL1600 0.038 0.017 CHEMBL447626 | CHEMBL447626 | |
| 0.136 | 0.153 | 0.247 | Hypolipemic | 0.197 0.096 CHEMBL3526986 0.212 0.086 CHEMBL3527418 0.153 0.134 CHEMBL3526948 0.198 0.096 CHEMBL3527235 0.184 0.107 CHEMBL447626 0.247 0.069 CHEMBL3527417 0.192 0.1 CHEMBL3527058 | CHEMBL3527417 | |
| 0.028 | 0.046 | 0.2 | Urate transporter 1 inhibitor | 0.2 0.003 CHEMBL3526986 0.075 0.009 CHEMBL3527418 0.066 0.012 CHEMBL3527235 0.062 0.013 CHEMBL3527417 0.05 0.019 CHEMBL3527058 | CHEMBL3526986 | |
| 0.02 | 0.039 | 0.027 | Acid ceramidase inhibitor | 0.024 0.022 CHEMBL3526986 0.027 0.014 CHEMBL1600 0.026 0.017 CHEMBL447626 | CHEMBL1600 | |
| 0.222 | 0.245 | 0.438 | Cyclophilin D inhibitor | 0.269 0.192 CHEMBL3526986 0.388 0.098 CHEMBL3527418 0.29 0.171 CHEMBL3526948 0.288 0.174 CHEMBL1600 0.394 0.094 CHEMBL3527235 0.253 0.21 CHEMBL447626 0.361 0.115 CHEMBL3527417 0.438 0.072 CHEMBL3527058 | CHEMBL3527058 | |
| 0.04 | 0.062 | 0.048 | Beta adrenoreceptor agonist | 0.048 0.022 CHEMBL1600 0.044 0.035 CHEMBL447626 0.047 0.026 CHEMBL3527058 | CHEMBL1600 | |
| 0.017 | 0.04 | 0.028 | Squalene synthetase inhibitor | 0.028 0.025 CHEMBL3527058 | CHEMBL3527058 | |
| 0.022 | 0.049 | 0.039 | Catechol O-methyltransferase inhibitor | 0.039 0.015 CHEMBL3526986 | CHEMBL3526986 | |
| 0.071 | 0.099 | 0.131 | Alcohol dehydrogenase inhibitor | 0.119 0.035 CHEMBL3526986 0.131 0.028 CHEMBL3527418 0.098 0.054 CHEMBL3526948 0.114 0.039 CHEMBL3527235 0.113 0.04 CHEMBL3527417 | CHEMBL3527418 | |
| 0.004 | 0.032 | 0.025 | Thyroid hormone beta agonist | 0.025 0.003 CHEMBL3526986 0.008 0.007 CHEMBL3527235 0.009 0.006 CHEMBL3527417 0.01 0.005 CHEMBL3527058 | CHEMBL3526986 | |
| 0.136 | 0.165 | 0.155 | Antiamyloidogenic | 0.155 0.14 CHEMBL3526986 0.152 0.145 CHEMBL3526948 0.15 0.147 CHEMBL3527417 | CHEMBL3526986 | |
| 0.114 | 0.147 | 0.335 | Angiogenesis stimulant | 0.335 0.037 CHEMBL3526986 0.268 0.062 CHEMBL3527418 0.205 0.092 CHEMBL3526948 0.15 0.122 CHEMBL1600 0.226 0.081 CHEMBL3527235 0.145 0.126 CHEMBL447626 0.22 0.084 CHEMBL3527417 0.246 0.072 CHEMBL3527058 | CHEMBL3526986 | |
| 0.041 | 0.077 | 0.053 | Vanilloid 2 antagonist | 0.053 0.035 CHEMBL3526986 0.049 0.043 CHEMBL1600 0.05 0.04 CHEMBL447626 | CHEMBL3526986 | |
| 0.059 | 0.096 | 0.113 | Adrenaline agonist | 0.113 0.029 CHEMBL1600 0.086 0.05 CHEMBL447626 0.1 0.037 CHEMBL3527058 | CHEMBL1600 | |
| 0.02 | 0.057 | 0.053 | Retinoid X alpha receptor agonist | 0.053 0.013 CHEMBL3526986 0.032 0.028 CHEMBL3527418 0.041 0.019 CHEMBL3527235 0.039 0.02 CHEMBL3527417 | CHEMBL3526986 | |
| 0.02 | 0.057 | 0.034 | Melatonin agonist | 0.033 0.022 CHEMBL1600 0.034 0.022 CHEMBL447626 | CHEMBL447626 | |
| 0.079 | 0.119 | 0.117 | Adenylate kinase inhibitor | 0.099 0.069 CHEMBL3526986 0.117 0.046 CHEMBL3527235 0.102 0.064 CHEMBL3527417 | CHEMBL3527235 | |
| 0.023 | 0.063 | 0.034 | Peroxisome proliferator-activated receptor delta antagonist | 0.031 0.028 CHEMBL3527418 0.033 0.023 CHEMBL3527235 0.034 0.022 CHEMBL3527417 0.032 0.025 CHEMBL3527058 | CHEMBL3527417 | |
| 0.044 | 0.084 | 0.058 | Nitric oxide donor | 0.056 0.055 CHEMBL3527235 0.058 0.053 CHEMBL3527058 | CHEMBL3527058 | |
| 0.105 | 0.151 | 0.208 | Dual specificity phosphatase 3 inhibitor | 0.208 0.056 CHEMBL3526986 0.138 0.108 CHEMBL3527418 | CHEMBL3526986 | |
| 0.025 | 0.071 | 0.057 | NMDA 2A receptor antagonist | 0.057 0.032 CHEMBL3527058 | CHEMBL3527058 | |
| 0.022 | 0.068 | 0.055 | Purinergic P2X3 antagonist | 0.055 0.009 CHEMBL3527418 0.051 0.01 CHEMBL447626 0.054 0.01 CHEMBL3527417 | CHEMBL3527418 | |
| 0.012 | 0.06 | 0.024 | Beta 1 adrenoreceptor agonist | 0.024 0.014 CHEMBL1600 0.022 0.016 CHEMBL3527058 | CHEMBL1600 | |
| 0.059 | 0.109 | 0.106 | MAO A inhibitor | 0.106 0.06 CHEMBL447626 | CHEMBL447626 | |
| 0.041 | 0.093 | 0.147 | Leukotriene synthesis inhibitor | 0.147 0.01 CHEMBL3526986 0.072 0.043 CHEMBL3527418 0.063 0.052 CHEMBL3527235 0.065 0.049 CHEMBL3527417 0.063 0.052 CHEMBL3527058 | CHEMBL3526986 | |
| 0.023 | 0.076 | 0.064 | Peroxisome proliferator-activated receptor alpha agonist | 0.043 0.038 CHEMBL3527418 0.053 0.03 CHEMBL3527235 0.064 0.025 CHEMBL3527417 | CHEMBL3527417 | |
| 0.176 | 0.235 | 0.278 | Interleukin 2 agonist | 0.268 0.1 CHEMBL3526986 0.248 0.12 CHEMBL3527418 0.227 0.147 CHEMBL3526948 0.273 0.095 CHEMBL3527235 0.268 0.1 CHEMBL3527417 0.278 0.091 CHEMBL3527058 | CHEMBL3527058 | |
| 0.012 | 0.072 | 0.048 | Prostacyclin antagonist | 0.03 0.025 CHEMBL3527418 0.04 0.018 CHEMBL3527235 0.041 0.017 CHEMBL3527417 0.048 0.014 CHEMBL3527058 | CHEMBL3527058 | |
| 0.084 | 0.145 | 0.148 | NADPH oxidase inhibitor | 0.148 0.056 CHEMBL3526986 0.106 0.103 CHEMBL3527418 | CHEMBL3526986 | |
| 0.022 | 0.085 | 0.065 | Oleamide hydrolase inhibitor | 0.051 0.026 CHEMBL3526986 0.051 0.026 CHEMBL3527418 0.065 0.018 CHEMBL447626 | CHEMBL447626 | |
| 0.009 | 0.076 | 0.013 | Integrin beta6 antagonist | 0.013 0.012 CHEMBL3527058 | CHEMBL3527058 | |
| 0.107 | 0.178 | 0.216 | DNA methylase inhibitor | 0.216 0.069 CHEMBL3527235 0.209 0.074 CHEMBL3527417 | CHEMBL3527235 | |
| 0.03 | 0.101 | 0.062 | 5 Hydroxytryptamine 1A antagonist | 0.062 0.052 CHEMBL447626 | CHEMBL447626 | |
| 0.065 | 0.139 | 0.085 | Estrogen-related receptor beta agonist | 0.085 0.051 CHEMBL3526948 | CHEMBL3526948 | |
| 0.092 | 0.166 | 0.109 | DNA repair enzyme inhibitor | 0.108 0.102 CHEMBL3526986 0.109 0.099 CHEMBL3527058 | CHEMBL3527058 | |
| 0.047 | 0.122 | 0.096 | Ornithine decarboxylase inhibitor | 0.094 0.051 CHEMBL3526986 0.096 0.048 CHEMBL3527058 | CHEMBL3527058 | |
| 0.039 | 0.114 | 0.078 | Prostaglandin F2 alpha antagonist | 0.058 0.049 CHEMBL3526986 0.057 0.052 CHEMBL3527418 0.078 0.024 CHEMBL3527235 0.077 0.025 CHEMBL3527417 0.077 0.025 CHEMBL3527058 | CHEMBL3527235 | |
| 0.01 | 0.088 | 0.041 | Leukotriene A4 hydrolase inhibitor | 0.035 0.028 CHEMBL3527235 0.041 0.025 CHEMBL3527417 0.032 0.031 CHEMBL3527058 | CHEMBL3527417 | |
| 0.155 | 0.234 | 0.225 | Vasodilator, peripheral | 0.225 0.149 CHEMBL3527235 0.219 0.155 CHEMBL3527417 | CHEMBL3527235 | |
| 0.016 | 0.096 | 0.064 | NMDA receptor subunit 3A antagonist | 0.064 0.016 CHEMBL3526986 | CHEMBL3526986 | |
| 0.168 | 0.248 | 0.383 | Histamine release inhibitor | 0.248 0.157 CHEMBL3526986 0.383 0.084 CHEMBL3527418 0.237 0.165 CHEMBL3527235 0.236 0.166 CHEMBL3527417 | CHEMBL3527418 | |
| 0.017 | 0.101 | 0.027 | Estrogen-related receptor gamma antagonist | 0.027 0.023 CHEMBL3526948 | CHEMBL3526948 | |
| 0.021 | 0.106 | 0.041 | Retinoic acid alpha receptor agonist | 0.041 0.024 CHEMBL3527418 | CHEMBL3527418 | |
| 0.01 | 0.096 | 0.018 | Retinoic acid beta receptor agonist | 0.018 0.017 CHEMBL3527418 | CHEMBL3527418 | |
| 0.066 | 0.153 | 0.123 | Carbonic anhydrase XV inhibitor | 0.123 0.044 CHEMBL3526986 0.094 0.077 CHEMBL3527418 | CHEMBL3526986 | |
| 0.019 | 0.107 | 0.043 | Estrogen-related receptor beta antagonist | 0.043 0.009 CHEMBL3526948 | CHEMBL3526948 | |
| 0.051 | 0.141 | 0.083 | Chymotrypsin inhibitor | 0.083 0.051 CHEMBL3526986 0.072 0.067 CHEMBL3527417 | CHEMBL3526986 | |
| 0.086 | 0.178 | 0.141 | Phospholipase A2 inhibitor | 0.14 0.086 CHEMBL3527418 0.135 0.093 CHEMBL3527235 0.141 0.084 CHEMBL3527417 0.121 0.116 CHEMBL3527058 | CHEMBL3527417 | |
| 0.131 | 0.223 | 0.251 | 5 Hydroxytryptamine release stimulant | 0.214 0.11 CHEMBL3526986 0.251 0.088 CHEMBL1600 0.239 0.094 CHEMBL447626 | CHEMBL1600 | |
| 0.037 | 0.13 | 0.066 | Elastase 1 inhibitor | 0.066 0.053 CHEMBL3526986 | CHEMBL3526986 | |
| 0.096 | 0.194 | 0.173 | Dual specificity phosphatase inhibitor | 0.173 0.072 CHEMBL3526986 | CHEMBL3526986 | |
| 0.146 | 0.247 | 0.269 | Calpain 2 inhibitor | 0.262 0.141 CHEMBL1600 0.269 0.136 CHEMBL447626 | CHEMBL447626 | |
| 0.061 | 0.164 | 0.078 | Vanilloid agonist | 0.078 0.076 CHEMBL3526986 0.078 0.075 CHEMBL3527418 | CHEMBL3527418 | |
| 0.103 | 0.213 | 0.165 | Immunostimulant | 0.165 0.143 CHEMBL3527235 0.16 0.147 CHEMBL3527058 | CHEMBL3527235 | |
| 0.026 | 0.139 | 0.078 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.078 0.017 CHEMBL3526986 0.077 0.017 CHEMBL3527418 | CHEMBL3526986 | |
| 0.019 | 0.137 | 0.056 | NMDA receptor subunit 3B antagonist | 0.056 0.021 CHEMBL3526986 | CHEMBL3526986 | |
| 0.039 | 0.158 | 0.053 | Leukotriene C antagonist | 0.053 0.052 CHEMBL3527418 | CHEMBL3527418 | |
| 0.086 | 0.211 | 0.129 | Vanilloid 1 agonist | 0.128 0.071 CHEMBL3526986 0.129 0.068 CHEMBL3527418 0.115 0.099 CHEMBL3527058 | CHEMBL3527418 | |
| 0.081 | 0.205 | 0.172 | Arachidonic acid antagonist | 0.172 0.062 CHEMBL3526986 0.158 0.079 CHEMBL3527418 | CHEMBL3526986 | |
| 0.143 | 0.269 | 0.234 | Insulysin inhibitor | 0.2 0.156 CHEMBL3526986 0.234 0.113 CHEMBL3527235 0.232 0.115 CHEMBL3527417 0.221 0.128 CHEMBL3527058 | CHEMBL3527235 | |
| 0.054 | 0.188 | 0.12 | DNA polymerase I inhibitor | 0.12 0.068 CHEMBL3526986 | CHEMBL3526986 | |
| 0.111 | 0.255 | 0.228 | Hypoglycemic | 0.204 0.108 CHEMBL3527418 0.201 0.111 CHEMBL3527235 0.208 0.105 CHEMBL3527417 0.228 0.09 CHEMBL3527058 | CHEMBL3527058 | |
| 0.028 | 0.179 | 0.065 | Sphingosine kinase inhibitor | 0.065 0.031 CHEMBL3526986 0.056 0.047 CHEMBL3527418 | CHEMBL3526986 | |
| 0.049 | 0.203 | 0.119 | Bile acid receptor antagonist | 0.119 0.021 CHEMBL3526986 0.087 0.081 CHEMBL3527418 0.088 0.079 CHEMBL3527235 0.09 0.075 CHEMBL3527417 | CHEMBL3526986 | |
| 0.045 | 0.208 | 0.212 | Cystathionine beta-synthase inhibitor | 0.212 0.022 CHEMBL3526986 0.101 0.075 CHEMBL3527418 | CHEMBL3526986 | |
| 0.11 | 0.281 | 0.29 | 12-Lipoxygenase inhibitor | 0.29 0.085 CHEMBL3526986 | CHEMBL3526986 | |
| 0.104 | 0.277 | 0.4 | Lipoxygenase inhibitor | 0.4 0.037 CHEMBL3526986 0.194 0.147 CHEMBL3527418 | CHEMBL3526986 | |
| 0.074 | 0.251 | 0.143 | DNA methyltransferase I inhibitor | 0.143 0.112 CHEMBL3527235 0.138 0.119 CHEMBL3527417 | CHEMBL3527235 | |
| 0.027 | 0.211 | 0.077 | Androgen antagonist | 0.077 0.069 CHEMBL3526986 | CHEMBL3526986 | |
| 0.094 | 0.279 | 0.134 | MAP kinase kinase 4 inhibitor | 0.134 0.102 CHEMBL3526986 | CHEMBL3526986 | |
| 0.124 | 0.311 | 0.316 | 15-Lipoxygenase inhibitor | 0.316 0.121 CHEMBL3526986 | CHEMBL3526986 | |
| 0.029 | 0.223 | 0.067 | CDC25A inhibitor | 0.067 0.063 CHEMBL3526986 | CHEMBL3526986 | |
| 0.061 | 0.258 | 0.151 | Protein kinase stimulant | 0.134 0.08 CHEMBL3526986 0.151 0.068 CHEMBL3527418 | CHEMBL3527418 | |
| 0.036 | 0.245 | 0.105 | Creatine kinase inhibitor | 0.105 0.054 CHEMBL3526986 | CHEMBL3526986 | |
| 0.114 | 0.339 | 0.154 | MAP kinase kinase 5 inhibitor | 0.154 0.137 CHEMBL3527418 | CHEMBL3527418 | |
| 0.038 | 0.266 | 0.088 | Interleukin 1 beta converting enzyme inhibitor | 0.088 0.076 CHEMBL3527058 | CHEMBL3527058 | |
| 0.009 | 0.239 | 0.032 | ATP citrate lysase inhibitor | 0.032 0.021 CHEMBL3526986 | CHEMBL3526986 | |
| 0.121 | 0.353 | 0.398 | Antibacterial | 0.398 0.078 CHEMBL3526986 0.242 0.184 CHEMBL447626 | CHEMBL3526986 | |
| 0.078 | 0.313 | 0.177 | Succinate dehydrogenase inhibitor | 0.177 0.071 CHEMBL3526986 0.165 0.088 CHEMBL3527418 | CHEMBL3526986 | |
| 0.074 | 0.309 | 0.137 | 3C-like protease (Human coronavirus) inhibitor | 0.137 0.126 CHEMBL3526986 | CHEMBL3526986 | |
| 0.027 | 0.264 | 0.072 | Glutamate (mGluR7) antagonist | 0.072 0.039 CHEMBL3526986 | CHEMBL3526986 | |
| 0.009 | 0.248 | 0.037 | Dopamine D5 agonist | 0.037 0.032 CHEMBL3526986 | CHEMBL3526986 | |
| 0.032 | 0.274 | 0.072 | Carbonic anhydrase VI inhibitor | 0.072 0.069 CHEMBL3526986 | CHEMBL3526986 | |
| 0.06 | 0.306 | 0.157 | Interleukin antagonist | 0.14 0.126 CHEMBL3527235 0.142 0.124 CHEMBL3527417 0.157 0.113 CHEMBL3527058 | CHEMBL3527058 | |
| 0.052 | 0.298 | 0.087 | Interleukin 12 antagonist | 0.087 0.08 CHEMBL3527418 | CHEMBL3527418 | |
| 0.005 | 0.253 | 0.065 | Estradiol 17 beta-dehydrogenase inhibitor | 0.065 0.018 CHEMBL3526986 | CHEMBL3526986 | |
| 0.026 | 0.277 | 0.141 | 5-Lipoxygenase inhibitor | 0.141 0.041 CHEMBL3526986 | CHEMBL3526986 | |
| 0.059 | 0.313 | 0.145 | Sphingosine 1-phosphate receptor 4 antagonist | 0.109 0.097 CHEMBL3526986 0.145 0.038 CHEMBL3527418 | CHEMBL3527418 | |
| 0.004 | 0.266 | 0.019 | Estradiol 17 beta-dehydrogenase 1 inhibitor | 0.019 0.018 CHEMBL3526986 | CHEMBL3526986 | |
| 0.037 | 0.301 | 0.1 | MAP kinase kinase 1 inhibitor | 0.1 0.056 CHEMBL3527418 | CHEMBL3527418 | |
| 0.021 | 0.288 | 0.066 | NMDA receptor agonist | 0.066 0.04 CHEMBL3527058 | CHEMBL3527058 | |
| 0.049 | 0.337 | 0.126 | Interleukin 4 antagonist | 0.126 0.076 CHEMBL3526986 0.107 0.105 CHEMBL3527418 | CHEMBL3526986 | |
| 0.023 | 0.311 | 0.061 | Enoyl-[acyl-carrier-protein] reductase inhibitor | 0.061 0.042 CHEMBL3526986 | CHEMBL3526986 | |
| 0.038 | 0.337 | 0.136 | Cyclooxygenase inhibitor | 0.136 0.082 CHEMBL3526986 | CHEMBL3526986 | |
| 0.065 | 0.369 | 0.128 | Interferon gamma antagonist | 0.128 0.116 CHEMBL3526986 | CHEMBL3526986 | |
| 0.119 | 0.433 | 0.198 | 5 Hydroxytryptamine uptake stimulant | 0.198 0.156 CHEMBL3526986 | CHEMBL3526986 | |
| 0.056 | 0.374 | 0.186 | Streptokinase A inhibitor | 0.186 0.142 CHEMBL3526986 | CHEMBL3526986 | |
| 0.094 | 0.416 | 0.133 | Ca2+-transporting ATPase inhibitor | 0.133 0.105 CHEMBL3526986 | CHEMBL3526986 | |
| 0.098 | 0.425 | 0.233 | GABA C receptor rho-3 antagonist | 0.233 0.17 CHEMBL3526986 | CHEMBL3526986 | |
| 0.061 | 0.416 | 0.182 | Neurotrophic factor enhancer | 0.182 0.096 CHEMBL3526986 | CHEMBL3526986 | |
| 0.037 | 0.408 | 0.158 | Insulin sensitizer | 0.158 0.122 CHEMBL3527058 | CHEMBL3527058 | |
| 0.091 | 0.502 | 0.168 | Peptidyltransferase inhibitor | 0.168 0.151 CHEMBL3527058 | CHEMBL3527058 | |
| 0.017 | 0.429 | 0.062 | CXC chemokine 1 receptor antagonist | 0.062 0.019 CHEMBL3526986 | CHEMBL3526986 | |
| 0.07 | 0.557 | 0.221 | Apoptosis antagonist | 0.221 0.156 CHEMBL3527058 | CHEMBL3527058 | |
| 0.047 | 0.559 | 0.13 | Growth hormone agonist | 0.122 0.118 CHEMBL3527417 0.13 0.107 CHEMBL3527058 | CHEMBL3527058 | |
| 0.024 | 0.538 | 0.179 | Platelet antagonist | 0.178 0.119 CHEMBL3527235 0.174 0.122 CHEMBL3527417 0.179 0.118 CHEMBL3527058 | CHEMBL3527058 | |
| 0.018 | 0.537 | 0.137 | Pyruvate kinase inhibitor | 0.137 0.128 CHEMBL3526986 | CHEMBL3526986 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |